TPD ID	TPD NAME	PubChem synonyms	SMILES	Fomula	Target Symbol	Target ID	Ligase	Source
TPD-O7725Z	SCHEMBL25026569	N-[4-cyano-3-(trifluoromethyl)phenyl]-2-[4-[2-[1-[[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]methyl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide; SCHEMBL31597200	Cn1c(=O)n(C2CCC(=O)NC2=O)c2ccc(CN3CC(C#Cc4cnn(C(C)(C)C(=O)Nc5ccc(C#N)c(C(F)(F)F)c5)c4)C3)cc21	C34H31F3N8O4	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-V33ART	SCHEMBL25024749	N-[4-cyano-3-(trifluoromethyl)phenyl]-2-[4-[2-[1-[[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-4-yl]methyl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(CN3CC(C#Cc4cnn(C(C)(C)C(=O)Nc5ccc(C#N)c(C(F)(F)F)c5)c4)C3)c21	C34H31F3N8O4	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-LIZKQI	SCHEMBL25026841	N-[4-cyano-3-(trifluoromethyl)phenyl]-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide	CC(C)(C(=O)Nc1ccc(C#N)c(C(F)(F)F)c1)n1cc(C#CC2CN(c3cc4c(cc3F)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C33H25F4N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-9A79FR	SCHEMBL25026248	N-[6-cyano-5-(trifluoromethyl)pyridin-3-yl]-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide; SCHEMBL30137302	CC(C)(C(=O)Nc1cnc(C#N)c(C(F)(F)F)c1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C32H25F3N8O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-6JNEMB	SCHEMBL25026842	N-[6-cyano-5-(trifluoromethyl)pyridin-3-yl]-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide	CC(C)(C(=O)Nc1cnc(C#N)c(C(F)(F)F)c1)n1cc(C#CC2CN(c3ccc4c(c3)CN(C3CCC(=O)NC3=O)C4=O)C2)cn1	C32H27F3N8O4	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-URYS5S	SCHEMBL25026586	N-[4-cyano-3-(trifluoromethyl)phenyl]-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide	CC(C)(C(=O)Nc1ccc(C#N)c(C(F)(F)F)c1)n1cc(C#CC2CN(c3ccc4c(c3)CN(C3CCC(=O)NC3=O)C4=O)C2)cn1	C33H28F3N7O4	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-NMQ9M9	SCHEMBL25026585	N-[4-cyano-3-(trifluoromethyl)phenyl]-2-[4-[2-[1-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide	Cn1c(=O)n(C2CCC(=O)NC2=O)c2ccc(N3CC(C#Cc4cnn(C(C)(C)C(=O)Nc5ccc(C#N)c(C(F)(F)F)c5)c4)C3)cc21	C33H29F3N8O4	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-LE82DT	SCHEMBL25026610	N-[4-cyano-3-(trifluoromethyl)phenyl]-2-[4-[2-[1-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-4-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(N3CC(C#Cc4cnn(C(C)(C)C(=O)Nc5ccc(C#N)c(C(F)(F)F)c5)c4)C3)c21	C33H29F3N8O4	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-C9KPAL	EP-4385985-A1_9	.	CC(C)(C(=O)Nc1ccc(C#N)c(C(F)(F)F)c1)n1cc(CCC2CN(c3ccc4c(c3)C(=O)N(C3CCC(O)NC3=O)C4=O)C2)cn1	C33H32F3N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-0BHQT1	SCHEMBL25026269	N-[6-cyano-5-(trifluoromethyl)pyridin-3-yl]-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethyl]pyrazol-1-yl]-2-methylpropanamide	CC(C)(C(=O)Nc1cnc(C#N)c(C(F)(F)F)c1)n1cc(CCC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C32H29F3N8O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-BNZ0OP	SCHEMBL25026297	N-[2-chloro-4-(trifluoromethyl)phenyl]-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide; SCHEMBL30137390	CC(C)(C(=O)Nc1ccc(C(F)(F)F)cc1Cl)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C32H26ClF3N6O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-E1GH4M	SCHEMBL25024839	N-(3-chloro-4-cyanophenyl)-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide; SCHEMBL30137360	CC(C)(C(=O)Nc1ccc(C#N)c(Cl)c1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C32H26ClN7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-5ZEAYS	EP-4385985-A1_13	.	Cc1cc(NC(=O)C(C)(C)n2cc(C#CC3CN(c4ccc5c(c4)S(=O)N(C4CCC(=O)NC4=O)C5=O)C3)cn2)ccc1C#N	C32H29N7O5S	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-CM8I7Z	SCHEMBL25026964	N-[2-chloro-4-(trifluoromethyl)phenyl]-1-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]cyclobutane-1-carboxamide; SCHEMBL30137296	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cnn(C6(C(=O)Nc7ccc(C(F)(F)F)cc7Cl)CCC6)c5)C4)cc3C2=O)C(=O)N1	C33H26ClF3N6O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-A69PYV	SCHEMBL25026682	N-[2-chloro-4-(trifluoromethyl)phenyl]-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide	CC(C)(C(=O)Nc1ccc(C(F)(F)F)cc1Cl)n1cc(C#CC2CN(c3cc4c(cc3F)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C32H25ClF4N6O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-RJ81II	SCHEMBL25027080	N-(4-chloro-3-methylphenyl)-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide; SCHEMBL30137309	Cc1cc(NC(=O)C(C)(C)n2cc(C#CC3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)cn2)ccc1Cl	C32H29ClN6O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-OOPNWA	SCHEMBL25027157	N-[3-chloro-4-(trifluoromethyl)phenyl]-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide; SCHEMBL30137370; SCHEMBL30137372	CC(C)(C(=O)Nc1ccc(C(F)(F)F)c(Cl)c1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C32H26ClF3N6O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-B0AMNH	SCHEMBL25026347	N-(3-chloro-4-methylphenyl)-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide; SCHEMBL30137363	Cc1ccc(NC(=O)C(C)(C)n2cc(C#CC3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)cn2)cc1Cl	C32H29ClN6O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-2EIMJ7	SCHEMBL25027027	N-(3-chloro-5-cyanophenyl)-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide; SCHEMBL30137241	CC(C)(C(=O)Nc1cc(Cl)cc(C#N)c1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C32H26ClN7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-4J55N7	SCHEMBL25026862	N-(2-chloro-4-cyanophenyl)-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide; SCHEMBL30137379	CC(C)(C(=O)Nc1ccc(C#N)cc1Cl)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C32H26ClN7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-AYWJ40	SCHEMBL25026698	N-(4-cyanonaphthalen-1-yl)-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide; SCHEMBL30137255	CC(C)(C(=O)Nc1ccc(C#N)c2ccccc12)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C36H29N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-H1QVBD	EP-4385985-A1_22	.	CC(C)(C(=O)Nc1cc(Cl)c(C(F)(F)F)c(Cl)c1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)OC3=O)C4=O)C2)cn1	C32H24Cl2F3N5O6	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-YGW0YJ	SCHEMBL25026822	N-(4-cyano-3-methoxyphenyl)-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide; SCHEMBL30137434	COc1cc(NC(=O)C(C)(C)n2cc(C#CC3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)cn2)ccc1C#N	C33H29N7O6	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-QDYIEQ	SCHEMBL25024783	N-(5-cyanothiophen-3-yl)-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide; SCHEMBL30137485	CC(C)(C(=O)Nc1csc(C#N)c1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C30H25N7O5S	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-ATBQ4R	SCHEMBL25024883	N-(3-chloro-4-nitrophenyl)-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide; SCHEMBL30137415	CC(C)(C(=O)Nc1ccc([N+](=O)[O-])c(Cl)c1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C31H26ClN7O7	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-ZXFXWJ	SCHEMBL25026363	2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methyl-N-[4-nitro-3-(trifluoromethyl)phenyl]propanamide	CC(C)(C(=O)Nc1ccc([N+](=O)[O-])c(C(F)(F)F)c1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C32H26F3N7O7	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-NW8152	SCHEMBL25026877	N-(4-cyano-2-fluorophenyl)-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide; SCHEMBL30137399	CC(C)(C(=O)Nc1ccc(C#N)cc1F)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C32H26FN7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-LU74UK	SCHEMBL25024851	N-[2-bromo-4-(trifluoromethyl)phenyl]-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide; SCHEMBL30137375	CC(C)(C(=O)Nc1ccc(C(F)(F)F)cc1Br)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C32H26BrF3N6O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-SWLEK9	SCHEMBL25024884	N-(4-cyano-3-cyclopropylphenyl)-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide; SCHEMBL30137264	CC(C)(C(=O)Nc1ccc(C#N)c(C2CC2)c1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C35H31N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-DDJEMO	SCHEMBL25026886	N-[2-cyclopropyl-4-(trifluoromethyl)phenyl]-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide; SCHEMBL30137347	CC(C)(C(=O)Nc1ccc(C(F)(F)F)cc1C1CC1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C35H31F3N6O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-P5AX4H	SCHEMBL25027153	2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-N-[2-fluoro-4-(trifluoromethyl)phenyl]-2-methylpropanamide; SCHEMBL30137307	CC(C)(C(=O)Nc1ccc(C(F)(F)F)cc1F)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C32H26F4N6O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-J6C11B	SCHEMBL25024872	N-(4-cyano-3-fluorophenyl)-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide; SCHEMBL30137382	CC(C)(C(=O)Nc1ccc(C#N)c(F)c1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C32H26FN7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-NGBE6N	SCHEMBL25027189	N-[2-chloro-4-(trifluoromethyl)phenyl]-1-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]cyclobutane-1-carboxamide	O=C1CCC(N2C(=O)c3cc(F)c(N4CC(C#Cc5cnn(C6(C(=O)Nc7ccc(C(F)(F)F)cc7Cl)CCC6)c5)C4)cc3C2=O)C(=O)N1	C33H25ClF4N6O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-3RV9XQ	SCHEMBL30137350	N-(4-cyanonaphthalen-1-yl)-1-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]cyclobutane-1-carboxamide	N#Cc1ccc(NC(=O)C2(n3cc(C#CC4CN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)cn3)CCC2)c2ccccc12	C37H29N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-BWC9JX	SCHEMBL25024891	N-[2-cyclopropyl-4-(trifluoromethyl)phenyl]-1-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]cyclobutane-1-carboxamide; SCHEMBL30137401	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cnn(C6(C(=O)Nc7ccc(C(F)(F)F)cc7C7CC7)CCC6)c5)C4)cc3C2=O)C(=O)N1	C36H31F3N6O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-LO1EFG	SCHEMBL25027168	N-(3-bromo-4-cyanophenyl)-1-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]cyclobutane-1-carboxamide; SCHEMBL30137494; SCHEMBL30137495	N#Cc1ccc(NC(=O)C2(n3cc(C#CC4CN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)cn3)CCC2)cc1Br	C33H26BrN7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-ZFLZBR	SCHEMBL25026899	N-(3-bromo-4-cyanophenyl)-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide; SCHEMBL30137286	CC(C)(C(=O)Nc1ccc(C#N)c(Br)c1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C32H26BrN7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-T271YC	SCHEMBL25024877	N-(4-cyano-3-pyrrolidin-1-ylphenyl)-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide; SCHEMBL30137333	CC(C)(C(=O)Nc1ccc(C#N)c(N2CCCC2)c1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C36H34N8O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-SYU9FG	SCHEMBL25024898	N-(4-cyano-2-cyclopropylphenyl)-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide; SCHEMBL30137326	CC(C)(C(=O)Nc1ccc(C#N)cc1C1CC1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C35H31N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-4F6LCN	SCHEMBL25024856	N-(4-cyano-3-cyclopropylphenyl)-1-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]cyclobutane-1-carboxamide; SCHEMBL30137268	N#Cc1ccc(NC(=O)C2(n3cc(C#CC4CN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)cn3)CCC2)cc1C1CC1	C36H31N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-Y34R9V	SCHEMBL25026689	N-[4-cyano-3-(trifluoromethyl)phenyl]-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-ethylbutanamide; SCHEMBL30137331	CCC(CC)(C(=O)Nc1ccc(C#N)c(C(F)(F)F)c1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C35H30F3N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-E9MFAP	SCHEMBL25024902	N-[2-cyano-4-(trifluoromethyl)phenyl]-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide; SCHEMBL30137254	CC(C)(C(=O)Nc1ccc(C(F)(F)F)cc1C#N)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C33H26F3N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-VKUL9N	SCHEMBL25026314	N-(8-cyanoquinolin-5-yl)-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide; SCHEMBL30137300	CC(C)(C(=O)Nc1ccc(C#N)c2ncccc12)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C35H28N8O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-6OV6C2	SCHEMBL25026684	N-[4-cyano-2-(trifluoromethyl)phenyl]-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide; SCHEMBL30137404	CC(C)(C(=O)Nc1ccc(C#N)cc1C(F)(F)F)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C33H26F3N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-JY6VYV	SCHEMBL25024907	N-(4-cyano-2-cyclopropylphenyl)-1-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]cyclobutane-1-carboxamide; SCHEMBL30137353	N#Cc1ccc(NC(=O)C2(n3cc(C#CC4CN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)cn3)CCC2)c(C2CC2)c1	C36H31N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-FV5R62	SCHEMBL25024887	N-[4-cyano-3-(trifluoromethyl)phenyl]-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylbutanamide; SCHEMBL30137418	CCC(C)(C(=O)Nc1ccc(C#N)c(C(F)(F)F)c1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C34H28F3N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-UBOA2B	EP-4385985-A1_47	.	N#CC1CC=C(NC(=O)Cn2cc(C#CC3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)cn2)C=C1C(F)(F)F	C31H24F3N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-TXHCLS	SCHEMBL25026901	N-[4-cyano-3-(trifluoromethyl)phenyl]-1-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]cyclopentane-1-carboxamide; SCHEMBL30137144	N#Cc1ccc(NC(=O)C2(n3cc(C#CC4CN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)cn3)CCCC2)cc1C(F)(F)F	C35H28F3N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-K6LLZ7	SCHEMBL25026376	N-[2-cyano-4-(trifluoromethyl)phenyl]-1-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]cyclopropane-1-carboxamide; SCHEMBL30137365	N#Cc1cc(C(F)(F)F)ccc1NC(=O)C1(n2cc(C#CC3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)cn2)CC1	C33H24F3N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-UO7IET	SCHEMBL25026739	N-(4-cyano-3-pyrrolidin-1-ylphenyl)-1-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]cyclobutane-1-carboxamide; SCHEMBL30137378	N#Cc1ccc(NC(=O)C2(n3cc(C#CC4CN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)cn3)CCC2)cc1N1CCCC1	C37H34N8O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-RMQDXR	SCHEMBL25026723	2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methyl-N-[2-pyrazol-1-yl-4-(trifluoromethyl)phenyl]propanamide	CC(C)(C(=O)Nc1ccc(C(F)(F)F)cc1-n1cccn1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C35H29F3N8O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-ZYWJ5K	SCHEMBL25026721	2-[[2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanoyl]amino]-N-methyl-5-(trifluoromethyl)benzamide; SCHEMBL30137297	CNC(=O)c1cc(C(F)(F)F)ccc1NC(=O)C(C)(C)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C34H30F3N7O6	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-0J397Z	SCHEMBL25027025	N-[2-chloro-4-(trifluoromethyl)phenyl]-1-[4-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]cyclobutane-1-carboxamide; SCHEMBL30137428	O=C1CCC(N2C(=O)c3ccc(N4CC(N5CC(C#Cc6cnn(C7(C(=O)Nc8ccc(C(F)(F)F)cc8Cl)CCC7)c6)C5)C4)cc3C2=O)C(=O)N1	C36H31ClF3N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-18I72L	SCHEMBL25024810	N-(4-cyanonaphthalen-1-yl)-2-[4-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide	CC(C)(C(=O)Nc1ccc(C#N)c2ccccc12)n1cc(C#CC2CN(C3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)C2)cn1	C39H34N8O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-L3YLP5	EP-4385985-A1_55	.	CC(C)(C(=O)Nc1ccc(N)c2ccccc12)n1cc(C2CCN(C3C[C@@H]4CN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C[C@@H]4C3)CC2)cn1	C42H46N8O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-LH7S4C	EP-4385985-A1_56	.	CC(C)(C(=O)Nc1ccc(C#N)c2c1CCCC2)N1C=C(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)CN1	C36H35N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-CBQOUY	SCHEMBL25026900	N-[2-chloro-4-(trifluoromethyl)phenyl]-1-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]pyrazol-1-yl]cyclobutane-1-carboxamide; SCHEMBL30137267	O=C1CCC(N2C(=O)c3ccc(-c4cnn(C5(C(=O)Nc6ccc(C(F)(F)F)cc6Cl)CCC5)c4)cc3C2=O)C(=O)N1	C28H21ClF3N5O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-T2QM8O	SCHEMBL25026368	N-[2-chloro-4-(trifluoromethyl)phenyl]-1-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]ethynyl]pyrazol-1-yl]cyclobutane-1-carboxamide; SCHEMBL30137361	O=C1CCC(N2C(=O)c3ccc(C#Cc4cnn(C5(C(=O)Nc6ccc(C(F)(F)F)cc6Cl)CCC5)c4)cc3C2=O)C(=O)N1	C30H21ClF3N5O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-D80N61	SCHEMBL25024917	2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methyl-N-[2-methyl-4-(trifluoromethyl)phenyl]propanamide; SCHEMBL30137487	Cc1cc(C(F)(F)F)ccc1NC(=O)C(C)(C)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C33H29F3N6O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-JX3RJ8	SCHEMBL25026196	N-(4-cyanonaphthalen-1-yl)-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide; SCHEMBL30137385	CC(C)(C(=O)Nc1ccc(C#N)c2ccccc12)n1cc(C#CC2CCN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)cn1	C38H33N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-MB3VEM	EP-4385985-A1_61	.	O=C1CCC(N2C(=O)c3ccc(N4CCC(C#Cc5cnn(C6(C(=O)Nc7ccc(C(F)(F)F)cc7Cl)CCC6)c5)CC4)cc3C2=O)C(=O)N1	C35H30ClF3N6O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-83OIJ3	SCHEMBL25026695	2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methyl-N-[2-(1-methylpyrazol-4-yl)-4-(trifluoromethyl)phenyl]propanamide	Cn1cc(-c2cc(C(F)(F)F)ccc2NC(=O)C(C)(C)n2cc(C#CC3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)cn2)cn1	C36H31F3N8O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-QXHCJ9	SCHEMBL25024926	5-[3-[2-[1-[1-[(4-cyanonaphthalen-1-yl)amino]-2-methyl-1-oxopropan-2-yl]pyrazol-4-yl]ethynyl]azetidin-1-yl]-N-(2,6-dioxopiperidin-3-yl)pyridine-2-carboxamide; SCHEMBL30137400	CC(C)(C(=O)Nc1ccc(C#N)c2ccccc12)n1cc(C#CC2CN(c3ccc(C(=O)NC4CCC(=O)NC4=O)nc3)C2)cn1	C34H30N8O4	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-99QIRU	EP-4385985-A1_64	.	O=C1CCC(NC(=O)c2ccc(N3CC(C#Cc4cnn(C5(C(=O)Nc6ccc(C(F)(F)F)cc6Cl)CCC5)c4)C3)cn2)C(=O)N1	C31H27ClF3N7O4	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-9A4F1Y	SCHEMBL25026199	N-(4-cyanonaphthalen-1-yl)-2-[4-[1-[7-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-7-azaspiro[3.5]nonan-2-yl]piperidin-4-yl]pyrazol-1-yl]-2-methylpropanamide; SCHEMBL30137282	CC(C)(C(=O)Nc1ccc(C#N)c2ccccc12)n1cc(C2CCN(C3CC4(CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C3)CC2)cn1	C44H46N8O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-HW1F0D	SCHEMBL25026195	N-(4-cyanonaphthalen-1-yl)-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-3-hydroxyazetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide; SCHEMBL30137262	CC(C)(C(=O)Nc1ccc(C#N)c2ccccc12)n1cc(C#CC2(O)CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C36H29N7O6	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-X1Q31S	SCHEMBL25026200	N-[2-chloro-4-(trifluoromethyl)phenyl]-1-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-3-hydroxyazetidin-3-yl]ethynyl]pyrazol-1-yl]cyclobutane-1-carboxamide	O=C1CCC(N2C(=O)c3ccc(N4CC(O)(C#Cc5cnn(C6(C(=O)Nc7ccc(C(F)(F)F)cc7Cl)CCC6)c5)C4)cc3C2=O)C(=O)N1	C33H26ClF3N6O6	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-P82MAT	SCHEMBL25026202	N-(4-cyanonaphthalen-1-yl)-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-3-fluoroazetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide; SCHEMBL30137499	CC(C)(C(=O)Nc1ccc(C#N)c2ccccc12)n1cc(C#CC2(F)CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C36H28FN7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-E2126F	SCHEMBL25024892	N-[2-chloro-4-(trifluoromethyl)phenyl]-1-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]cyclopentane-1-carboxamide; SCHEMBL30137273	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cnn(C6(C(=O)Nc7ccc(C(F)(F)F)cc7Cl)CCCC6)c5)C4)cc3C2=O)C(=O)N1	C34H28ClF3N6O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-DKYOIB	SCHEMBL25024925	N-[2-dimethylphosphoryl-4-(trifluoromethyl)phenyl]-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide; SCHEMBL30137383	CC(C)(C(=O)Nc1ccc(C(F)(F)F)cc1P(C)(C)=O)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C34H32F3N6O6P	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-4K7UZT	EP-4385985-A1_71	.	O=C1CCC(N2C(=O)c3ccc(N4CC(F)(C#Cc5cnn(C6(C(=O)Nc7ccc(C(F)(F)F)cc7Cl)CCC6)c5)C4)cc3C2=O)C(=O)N1	C33H25ClF4N6O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-5H03GO	SCHEMBL25026197	N-[2-chloro-4-(trifluoromethyl)phenyl]-1-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]cyclopropane-1-carboxamide; SCHEMBL30137287	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cnn(C6(C(=O)Nc7ccc(C(F)(F)F)cc7Cl)CC6)c5)C4)cc3C2=O)C(=O)N1	C32H24ClF3N6O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-HFQMLA	SCHEMBL25024937	N-(4-cyanonaphthalen-1-yl)-2-[4-[2-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]cyclohexyl]ethynyl]pyrazol-1-yl]-2-methylpropanamide; SCHEMBL30137403	CC(C)(C(=O)Nc1ccc(C#N)c2ccccc12)n1cc(C#CC2CCC(N3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)cn1	C43H42N8O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-UI9KO6	EP-4385985-A1_74	.	O=C1CCC(N2C(=O)c3ccc(N4CCN(C5CCC(C#Cc6cnn(C7(C(=O)Nc8ccc(C(F)(F)F)cc8Cl)CCC7)c6)CC5)CC4)cc3C2=O)C(=O)N1	C40H39ClF3N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-7VR4A7	SCHEMBL25026201	N-[3-cyclopropyl-4-(trifluoromethyl)phenyl]-1-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]cyclobutane-1-carboxamide; SCHEMBL30137458	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cnn(C6(C(=O)Nc7ccc(C(F)(F)F)c(C8CC8)c7)CCC6)c5)C4)cc3C2=O)C(=O)N1	C36H31F3N6O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-EZWK0Q	EP-4385985-A1_76	.	CC(C)(C(=O)Nc1ccc(C#N)c2c1C=CCC2)n1cc(C2CCN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)cn1	C36H35N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-RX9FKM	SCHEMBL25024922	N-[4-cyano-3-(trifluoromethyl)phenyl]-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]propanamide; SCHEMBL30137314; SCHEMBL30137318	CC(C(=O)Nc1ccc(C#N)c(C(F)(F)F)c1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C32H24F3N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-2VQFZK	SCHEMBL25026206	N-(4-cyanonaphthalen-1-yl)-2-[4-[1-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]methyl]piperidin-4-yl]pyrazol-1-yl]-2-methylpropanamide	CC(C)(C(=O)Nc1ccc(C#N)c2ccccc12)n1cc(C2CCN(Cc3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)cn1	C37H35N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-BX4NH0	SCHEMBL25024897	N-(4-cyanonaphthalen-1-yl)-2-[4-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperidin-4-yl]pyrazol-1-yl]-2-methylpropanamide; SCHEMBL30137258	CC(C)(C(=O)Nc1ccc(C#N)c2ccccc12)n1cc(C2CCN(C3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)CC2)cn1	C39H38N8O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-4RG32N	EP-4385985-A1_80	.	N#Cc1ccc(NC(=O)C2(n3cc(C#CC4CN(c5cc6c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)cn3)CCC2)c2ccccc12	C37H28FN7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-4WJ2EQ	SCHEMBL25026198	N-(4-cyanonaphthalen-1-yl)-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide	CC(C)(C(=O)Nc1ccc(C#N)c2ccccc12)n1cc(C#CC2CN(c3cc4c(cc3F)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C36H28FN7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-96JJDN	SCHEMBL25026204	N-(2-bromo-4-cyanophenyl)-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide; SCHEMBL30137364	CC(C)(C(=O)Nc1ccc(C#N)cc1Br)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C32H26BrN7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-RKUK3H	SCHEMBL25026209	N-[2-chloro-4-(trifluoromethyl)phenyl]-1-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]pyrazol-1-yl]cyclobutane-1-carboxamide; SCHEMBL30137425	O=C1CCC(N2C(=O)c3ccc(N4CCC(c5cnn(C6(C(=O)Nc7ccc(C(F)(F)F)cc7Cl)CCC6)c5)CC4)cc3C2=O)C(=O)N1	C33H30ClF3N6O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-FBXRN5	SCHEMBL25026218	N-[2-chloro-4-(trifluoromethyl)phenyl]-1-[4-[1-[7-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-7-azaspiro[3.5]nonan-2-yl]piperidin-4-yl]pyrazol-1-yl]cyclobutane-1-carboxamide; SCHEMBL30137423	O=C1CCC(N2C(=O)c3ccc(N4CCC5(CC4)CC(N4CCC(c6cnn(C7(C(=O)Nc8ccc(C(F)(F)F)cc8Cl)CCC7)c6)CC4)C5)cc3C2=O)C(=O)N1	C41H43ClF3N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-U2V71J	SCHEMBL25026213	N-[2-chloro-4-(trifluoromethyl)phenyl]-1-[4-[1-[[7-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-7-azaspiro[3.5]nonan-2-yl]methyl]piperidin-4-yl]pyrazol-1-yl]cyclobutane-1-carboxamide; SCHEMBL30137362	O=C1CCC(N2C(=O)c3ccc(N4CCC5(CC4)CC(CN4CCC(c6cnn(C7(C(=O)Nc8ccc(C(F)(F)F)cc8Cl)CCC7)c6)CC4)C5)cc3C2=O)C(=O)N1	C42H45ClF3N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-1LRBQR	SCHEMBL25024946	N-[2-chloro-4-(trifluoromethyl)phenyl]-1-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxophthalazin-6-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]cyclobutane-1-carboxamide; SCHEMBL30137263	O=C1CCC(n2ncc3cc(N4CC(C#Cc5cnn(C6(C(=O)Nc7ccc(C(F)(F)F)cc7Cl)CCC6)c5)C4)ccc3c2=O)C(=O)N1	C33H27ClF3N7O4	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-TTGR3P	SCHEMBL25024929	N-[2-chloro-4-(trifluoromethyl)phenyl]-1-[4-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperidin-4-yl]pyrazol-1-yl]cyclobutane-1-carboxamide; SCHEMBL30137298	O=C1CCC(N2C(=O)c3ccc(N4CCC(CN5CCC(c6cnn(C7(C(=O)Nc8ccc(C(F)(F)F)cc8Cl)CCC7)c6)CC5)CC4)cc3C2=O)C(=O)N1	C39H41ClF3N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-LKOU5H	SCHEMBL25024939	N-[2-chloro-4-(trifluoromethyl)phenyl]-1-[4-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]methyl]piperidin-4-yl]pyrazol-1-yl]cyclobutane-1-carboxamide; SCHEMBL30137343	O=C1CCC(N2C(=O)c3ccc(N4CC(CN5CCC(c6cnn(C7(C(=O)Nc8ccc(C(F)(F)F)cc8Cl)CCC7)c6)CC5)C4)cc3C2=O)C(=O)N1	C37H37ClF3N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-RG9SG6	SCHEMBL25026737	2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methyl-N-[2-methylsulfonyl-4-(trifluoromethyl)phenyl]propanamide	CC(C)(C(=O)Nc1ccc(C(F)(F)F)cc1S(C)(=O)=O)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C33H29F3N6O7S	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-74KXHC	SCHEMBL25026214	N-[2-chloro-4-(trifluoromethyl)phenyl]-1-[4-[1-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-3,3a,4,5,6,6a-hexahydro-1H-cyclopenta[c]pyrrol-5-yl]piperidin-4-yl]pyrazol-1-yl]cyclobutane-1-carboxamide; SCHEMBL30137479	O=C1CCC(N2C(=O)c3ccc(N4CC5CC(N6CCC(c7cnn(C8(C(=O)Nc9ccc(C(F)(F)F)cc9Cl)CCC8)c7)CC6)CC5C4)cc3C2=O)C(=O)N1	C40H41ClF3N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-7J76XA	SCHEMBL25026210	N-[2-chloro-4-(trifluoromethyl)phenyl]-1-[4-[1-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-3,3a,4,5,6,6a-hexahydro-1H-cyclopenta[c]pyrrol-5-yl]methyl]piperidin-4-yl]pyrazol-1-yl]cyclobutane-1-carboxamide; SCHEMBL30137366	O=C1CCC(N2C(=O)c3ccc(N4CC5CC(CN6CCC(c7cnn(C8(C(=O)Nc9ccc(C(F)(F)F)cc9Cl)CCC8)c7)CC6)CC5C4)cc3C2=O)C(=O)N1	C41H43ClF3N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-9I9W6L	SCHEMBL25026212	N-[2-chloro-4-(trifluoromethyl)phenyl]-1-[4-[1-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]azetidin-3-yl]piperidin-4-yl]pyrazol-1-yl]cyclobutane-1-carboxamide; SCHEMBL30137306	O=C1CCC(N2C(=O)c3ccc(N4CC(N5CC(N6CCC(c7cnn(C8(C(=O)Nc9ccc(C(F)(F)F)cc9Cl)CCC8)c7)CC6)C5)C4)cc3C2=O)C(=O)N1	C39H40ClF3N8O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-B8X099	SCHEMBL25026216	N-[2-chloro-4-(trifluoromethyl)phenyl]-1-[4-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-3-fluoroazetidin-3-yl]methyl]piperidin-4-yl]pyrazol-1-yl]cyclobutane-1-carboxamide; SCHEMBL30137338	O=C1CCC(N2C(=O)c3ccc(N4CC(F)(CN5CCC(c6cnn(C7(C(=O)Nc8ccc(C(F)(F)F)cc8Cl)CCC7)c6)CC5)C4)cc3C2=O)C(=O)N1	C37H36ClF4N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-XF7NFW	SCHEMBL25026217	N-[1-[1-[[2-chloro-4-(trifluoromethyl)phenyl]carbamoyl]cyclobutyl]pyrazol-4-yl]-N'-[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]heptanediamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCC(=O)Nc2cnn(C3(C(=O)Nc4ccc(C(F)(F)F)cc4Cl)CCC3)c2)C(C)(C)C)cc1	C45H54ClF3N8O6S	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-D54X7X	SCHEMBL25026211	N-(4-cyanonaphthalen-1-yl)-2-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]pyrazol-1-yl]-2-methylpropanamide; SCHEMBL30137447	CC(C)(C(=O)Nc1ccc(C#N)c2ccccc12)n1cc(CN2CCN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)cn1	C36H34N8O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-9YX45L	SCHEMBL25026220	N-[2-chloro-4-(trifluoromethyl)phenyl]-1-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]pyrazol-1-yl]cyclobutane-1-carboxamide; SCHEMBL30137308	O=C1CCC(N2C(=O)c3ccc(N4CCN(Cc5cnn(C6(C(=O)Nc7ccc(C(F)(F)F)cc7Cl)CCC6)c5)CC4)cc3C2=O)C(=O)N1	C33H31ClF3N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-RMIX87	SCHEMBL27242968	N-[2-chloro-4-(trifluoromethyl)phenyl]-1-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-2,7-diazaspiro[3.5]nonan-7-yl]pyrazol-1-yl]cyclobutane-1-carboxamide	O=C1CCC(N2C(=O)c3ccc(N4CC5(CCN(c6cnn(C7(C(=O)Nc8ccc(C(F)(F)F)cc8Cl)CCC7)c6)CC5)C4)cc3C2=O)C(=O)N1	C35H33ClF3N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-I6HEY8	SCHEMBL25026219	N-[2-chloro-4-(trifluoromethyl)phenyl]-1-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]pyrazol-1-yl]cyclobutane-1-carboxamide; SCHEMBL30137148	O=C1CCC(N2C(=O)c3ccc(N4CCN(CC5CCN(c6cnn(C7(C(=O)Nc8ccc(C(F)(F)F)cc8Cl)CCC7)c6)CC5)CC4)cc3C2=O)C(=O)N1	C38H40ClF3N8O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-KHNP3T	SCHEMBL25026215	N-[2-chloro-4-(trifluoromethyl)phenyl]-1-[4-[4-[[(1R,4R)-5-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-2,5-diazabicyclo[2.2.1]heptan-2-yl]methyl]piperidin-1-yl]pyrazol-1-yl]cyclobutane-1-carboxamide; SCHEMBL31597143	O=C1CCC(N2C(=O)c3ccc(N4C[C@H]5C[C@@H]4CN5CC4CCN(c5cnn(C6(C(=O)Nc7ccc(C(F)(F)F)cc7Cl)CCC6)c5)CC4)cc3C2=O)C(=O)N1	C39H40ClF3N8O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-SABLTA	SCHEMBL25026221	N-[2-chloro-4-(trifluoromethyl)phenyl]-1-[4-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-2,7-diazaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]pyrazol-1-yl]cyclobutane-1-carboxamide; SCHEMBL30990852	O=C1CCC(N2C(=O)c3ccc(N4CC5(CCN(CC6CCN(c7cnn(C8(C(=O)Nc9ccc(C(F)(F)F)cc9Cl)CCC8)c7)CC6)CC5)C4)cc3C2=O)C(=O)N1	C41H44ClF3N8O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-KCKZ7N	SCHEMBL25026222	N-[2-chloro-4-(trifluoromethyl)phenyl]-1-[4-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]pyrazol-1-yl]cyclobutane-1-carboxamide; SCHEMBL30990842	O=C1CCC(N2C(=O)c3ccc(N4CCN(CC5CCN(c6ccc(-c7cnn(C8(C(=O)Nc9ccc(C(F)(F)F)cc9Cl)CCC8)c7)cc6)CC5)CC4)cc3C2=O)C(=O)N1	C44H44ClF3N8O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-C5IH5J	SCHEMBL25024951	N-[2-chloro-4-(trifluoromethyl)phenyl]-1-[4-[4-[4-[(2,6-dioxopiperidin-3-yl)amino]-2-fluorophenyl]piperazine-1-carbonyl]pyrazol-1-yl]cyclobutane-1-carboxamide; SCHEMBL30137517	O=C1CCC(Nc2ccc(N3CCN(C(=O)c4cnn(C5(C(=O)Nc6ccc(C(F)(F)F)cc6Cl)CCC5)c4)CC3)c(F)c2)C(=O)N1	C31H30ClF4N7O4	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-PN9AJ2	EP-4385985-A1_103	.	O=C1CCC(N2Cc3cc(C#CC4CN(C(=O)c5cnn(C6(C(=O)NC7CC=C(C(F)(F)F)C=C7Cl)CCC6)c5)C4)ccc3C2=O)C(=O)N1	C34H30ClF3N6O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-LZDA8L	SCHEMBL30137463	N-[1-[1-[[2-chloro-4-(trifluoromethyl)phenyl]carbamoyl]cyclobutyl]pyrazol-4-yl]-1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidine-4-carboxamide	O=C1CCC(N2C(=O)c3ccc(N4CCC(C(=O)Nc5cnn(C6(C(=O)Nc7ccc(C(F)(F)F)cc7Cl)CCC6)c5)CC4)cc3C2=O)C(=O)N1	C34H31ClF3N7O6	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-94Z39S	SCHEMBL25024944	N-[2-chloro-4-(trifluoromethyl)phenyl]-1-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxopyrrolo[3,4-c]pyridin-6-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]cyclobutane-1-carboxamide; SCHEMBL30137293	O=C1CCC(N2C(=O)c3cnc(N4CC(C#Cc5cnn(C6(C(=O)Nc7ccc(C(F)(F)F)cc7Cl)CCC6)c5)C4)cc3C2=O)C(=O)N1	C32H25ClF3N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-VNWNGM	SCHEMBL25026180	N-(4-cyanonaphthalen-1-yl)-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxopyrrolo[3,4-c]pyridin-6-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide	CC(C)(C(=O)Nc1ccc(C#N)c2ccccc12)n1cc(C#CC2CN(c3cc4c(cn3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C35H28N8O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-B9ITNC	SCHEMBL25027248	N-[2-chloro-4-(trifluoromethyl)phenyl]-1-[4-[4-[[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]methyl]piperazine-1-carbonyl]pyrazol-1-yl]cyclobutane-1-carboxamide; SCHEMBL30137317	Cn1c(=O)n(C2CCC(=O)NC2=O)c2ccc(CN3CCN(C(=O)c4cnn(C5(C(=O)Nc6ccc(C(F)(F)F)cc6Cl)CCC5)c4)CC3)cc21	C34H34ClF3N8O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-OMRCZ0	SCHEMBL25024972	2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methyl-N-[2-(oxan-4-yl)-4-(trifluoromethyl)phenyl]propanamide; SCHEMBL30137468	CC(C)(C(=O)Nc1ccc(C(F)(F)F)cc1C1CCOCC1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C37H35F3N6O6	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-L25ARQ	SCHEMBL25026433	N-[2-(6-azaspiro[2.5]octan-6-yl)-4-(trifluoromethyl)phenyl]-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide; SCHEMBL30137276	CC(C)(C(=O)Nc1ccc(C(F)(F)F)cc1N1CCC2(CC1)CC2)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C39H38F3N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-HMOFNN	SCHEMBL25026741	N-[2-(3,3a,4,5,6,6a-hexahydro-1H-cyclopenta[c]pyrrol-2-yl)-4-(trifluoromethyl)phenyl]-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide; SCHEMBL31597128	CC(C)(C(=O)Nc1ccc(C(F)(F)F)cc1N1CC2CCCC2C1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C39H38F3N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-AKVYGT	SCHEMBL25026738	2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methyl-N-[2-(morpholin-4-ylmethyl)-4-(trifluoromethyl)phenyl]propanamide; SCHEMBL30137454	CC(C)(C(=O)Nc1ccc(C(F)(F)F)cc1CN1CCOCC1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C37H36F3N7O6	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-MS8UJ0	SCHEMBL25024978	2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methyl-N-[2-phenyl-4-(trifluoromethyl)phenyl]propanamide; SCHEMBL30137291	CC(C)(C(=O)Nc1ccc(C(F)(F)F)cc1-c1ccccc1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C38H31F3N6O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-6AHNKE	EP-4385985-A1_113	.	CC1(C)C(C)(C)C(C(=O)Nc2ccc(C(F)(F)F)cc2Cl)(n2cc(C#CC3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)cn2)C1(C)C	C39H38ClF3N6O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-09BUJO	SCHEMBL25024989	N-(3,4-dihydro-2H-chromen-5-yl)-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide; SCHEMBL31597146	CC(C)(C(=O)Nc1cccc2c1CCCO2)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C34H32N6O6	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-BO6DV1	SCHEMBL25026888	N-[2-chloro-4-(trifluoromethyl)phenyl]-1-[3-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]-2-oxopyridin-1-yl]cyclobutane-1-carboxamide	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cccn(C6(C(=O)Nc7ccc(C(F)(F)F)cc7Cl)CCC6)c5=O)C4)cc3C2=O)C(=O)N1	C35H27ClF3N5O6	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-QJELUV	SCHEMBL25024787	N-[2-(2-cyclopropylethynyl)-4-(trifluoromethyl)phenyl]-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide; SCHEMBL30137249	CC(C)(C(=O)Nc1ccc(C(F)(F)F)cc1C#CC1CC1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C37H31F3N6O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-C8QLAO	SCHEMBL25024984	2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methyl-N-[2-(1,2,4-triazol-1-yl)-4-(trifluoromethyl)phenyl]propanamide; SCHEMBL30137341	CC(C)(C(=O)Nc1ccc(C(F)(F)F)cc1-n1cncn1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C34H28F3N9O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-UZZRI4	SCHEMBL25024805	2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methyl-N-[2-prop-1-ynyl-4-(trifluoromethyl)phenyl]propanamide	CC#Cc1cc(C(F)(F)F)ccc1NC(=O)C(C)(C)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C35H29F3N6O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-FNCAV4	SCHEMBL30137394	N-(5-cyano-2-adamantyl)-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide	CC(C)(C(=O)NC1C2CC3CC1CC(C#N)(C3)C2)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C36H37N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-MQ7X03	SCHEMBL25024985	N-[2-chloro-4-(trifluoromethyl)phenyl]-1-[4-[2-[1-[3-(2,6-dioxopiperidin-3-yl)-4-oxo-1,2,3-benzotriazin-7-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]cyclobutane-1-carboxamide	O=C1CCC(n2nnc3cc(N4CC(C#Cc5cnn(C6(C(=O)Nc7ccc(C(F)(F)F)cc7Cl)CCC6)c5)C4)ccc3c2=O)C(=O)N1	C32H26ClF3N8O4	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-UM17QB	SCHEMBL25026181	N-(4-cyanonaphthalen-1-yl)-2-[4-[2-[1-[3-(2,6-dioxopiperidin-3-yl)-4-oxo-1,2,3-benzotriazin-7-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide; SCHEMBL30137368	CC(C)(C(=O)Nc1ccc(C#N)c2ccccc12)n1cc(C#CC2CN(c3ccc4c(=O)n(C5CCC(=O)NC5=O)nnc4c3)C2)cn1	C35H29N9O4	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-XKDGXV	SCHEMBL27242977	N-[2-chloro-4-(trifluoromethyl)phenyl]-1-[4-[[3-[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]ethynyl]azetidin-1-yl]methyl]pyrazol-1-yl]cyclobutane-1-carboxamide	O=C1CCC(N2Cc3cc(C#CC4CN(Cc5cnn(C6(C(=O)Nc7ccc(C(F)(F)F)cc7Cl)CCC6)c5)C4)ccc3C2=O)C(=O)N1	C34H30ClF3N6O4	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-TMCI26	SCHEMBL25027273	N-[2-chloro-4-(trifluoromethyl)phenyl]-1-[4-[[3-[2-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]ethynyl]azetidin-1-yl]methyl]pyrazol-1-yl]cyclobutane-1-carboxamide	Cn1c(=O)n(C2CCC(=O)NC2=O)c2ccc(C#CC3CN(Cc4cnn(C5(C(=O)Nc6ccc(C(F)(F)F)cc6Cl)CCC5)c4)C3)cc21	C34H31ClF3N7O4	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-Z7QPDS	SCHEMBL25024993	N-[2-[4-(azetidin-1-yl)piperidin-1-yl]-4-(trifluoromethyl)phenyl]-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide; SCHEMBL30137238	CC(C)(C(=O)Nc1ccc(C(F)(F)F)cc1N1CCC(N2CCC2)CC1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C40H41F3N8O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-8B97Q6	SCHEMBL30137540	N-(8-cyano-1,2,3,5,6,7-hexahydro-s-indacen-4-yl)-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide	CC(C)(C(=O)Nc1c2c(c(C#N)c3c1CCC3)CCC2)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C38H35N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-EDQJ90	SCHEMBL25024992	2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methyl-N-[2-(6-oxopyridazin-1-yl)-4-(trifluoromethyl)phenyl]propanamide; SCHEMBL30137374	CC(C)(C(=O)Nc1ccc(C(F)(F)F)cc1-n1ncccc1=O)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C36H29F3N8O6	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-YHVUCO	SCHEMBL25027292	N-[2-chloro-4-(trifluoromethyl)phenyl]-1-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-3-methylazetidin-3-yl]ethynyl]pyrazol-1-yl]cyclobutane-1-carboxamide; SCHEMBL30137265	CC1(C#Cc2cnn(C3(C(=O)Nc4ccc(C(F)(F)F)cc4Cl)CCC3)c2)CN(c2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)C1	C34H28ClF3N6O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-E2OI5F	EP-4385985-A1_128	.	CC1(C#Cc2cnn(C(C)(C)C(=O)Nc3ccc(N)c4ccccc34)c2)CN(c2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)C1	C36H33N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-ZUUF63	SCHEMBL25026188	N-[2-chloro-4-(trifluoromethyl)phenyl]-1-[4-[[3-[2-[3-(2,6-dioxopiperidin-3-yl)-1-methylindazol-7-yl]ethynyl]azetidin-1-yl]methyl]pyrazol-1-yl]cyclobutane-1-carboxamide	Cn1nc(C2CCC(=O)NC2=O)c2cccc(C#CC3CN(Cc4cnn(C5(C(=O)Nc6ccc(C(F)(F)F)cc6Cl)CCC5)c4)C3)c21	C34H31ClF3N7O3	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-BGLGS1	SCHEMBL25026182	N-[2-chloro-4-(trifluoromethyl)phenyl]-1-[4-[[3-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]ethynyl]azetidin-1-yl]methyl]pyrazol-1-yl]cyclobutane-1-carboxamide	O=C1CCC(N2C(=O)c3ccc(C#CC4CN(Cc5cnn(C6(C(=O)Nc7ccc(C(F)(F)F)cc7Cl)CCC6)c5)C4)cc3C2=O)C(=O)N1	C34H28ClF3N6O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-HCE5JC	SCHEMBL25027037	N-[2-(2,3-dihydroindol-1-yl)-5-(trifluoromethyl)phenyl]-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide; SCHEMBL30137346	CC(C)(C(=O)Nc1cc(C(F)(F)F)ccc1N1CCc2ccccc21)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C40H34F3N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-WKZB9W	SCHEMBL25027079	N-[2-chloro-4-(trifluoromethyl)phenyl]-1-[4-[2-[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]azetidin-3-yl]ethynyl]pyrazol-1-yl]cyclobutane-1-carboxamide	O=C1CCN(c2ccc(N3CC(C#Cc4cnn(C5(C(=O)Nc6ccc(C(F)(F)F)cc6Cl)CCC5)c4)C3)cc2)C(=O)N1	C30H26ClF3N6O3	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-AQWESD	SCHEMBL25026669	2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methyl-N-[2-pyrrol-1-yl-4-(trifluoromethyl)phenyl]propanamide; SCHEMBL30137419	CC(C)(C(=O)Nc1ccc(C(F)(F)F)cc1-n1cccc1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C36H30F3N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-N5SZDT	SCHEMBL25027184	N-(4-cyano-1-bicyclo[2.2.2]octanyl)-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide	CC(C)(C(=O)NC12CCC(C#N)(CC1)CC2)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C34H35N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-3HIEYK	SCHEMBL25027329	N-[2-chloro-4-(trifluoromethyl)phenyl]-1-[4-[2-[3-(2,4-dioxo-1,3-diazinan-1-yl)-1-methylindazol-6-yl]-2,7-diazaspiro[3.5]nonane-7-carbonyl]pyrazol-1-yl]cyclobutane-1-carboxamide; SCHEMBL30137233	Cn1nc(N2CCC(=O)NC2=O)c2ccc(N3CC4(CCN(C(=O)c5cnn(C6(C(=O)Nc7ccc(C(F)(F)F)cc7Cl)CCC6)c5)CC4)C3)cc21	C35H35ClF3N9O4	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-P9R2CG	SCHEMBL25025004	N-[2-(cyclopropylmethoxy)-4-(trifluoromethyl)phenyl]-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide; SCHEMBL30137528	CC(C)(C(=O)Nc1ccc(C(F)(F)F)cc1OCC1CC1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C36H33F3N6O6	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-CXLF2H	SCHEMBL25027051	N-[2-chloro-4-(trifluoromethyl)phenyl]-1-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazine-1-carbonyl]pyrazol-1-yl]cyclobutane-1-carboxamide	O=C1CCC(N2C(=O)c3ccc(N4CCN(C(=O)c5cnn(C6(C(=O)Nc7ccc(C(F)(F)F)cc7Cl)CCC6)c5)CC4)cc3C2=O)C(=O)N1	C33H29ClF3N7O6	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-VDWYSJ	EP-4385985-A1_138	.	CC(C)(C(=O)Nc1ccc(C(F)(F)F)cc1Cl)n1c(=O)[nH]c2ccc(C#CC3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)cc21	C36H28ClF3N6O6	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-5KYZ2H	SCHEMBL25027054	N-[2-chloro-4-(trifluoromethyl)phenyl]-1-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]imidazol-1-yl]cyclobutane-1-carboxamide; SCHEMBL30137290	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cn(C6(C(=O)Nc7ccc(C(F)(F)F)cc7Cl)CCC6)cn5)C4)cc3C2=O)C(=O)N1	C33H26ClF3N6O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-YRD99O	SCHEMBL25024969	N-[2-chloro-4-(trifluoromethyl)phenyl]-1-[4-[[3-[2-[1-(2,6-dioxopiperidin-3-yl)-2-oxobenzo[cd]indol-6-yl]ethynyl]azetidin-1-yl]methyl]pyrazol-1-yl]cyclobutane-1-carboxamide	O=C1CCC(N2C(=O)c3cccc4c(C#CC5CN(Cc6cnn(C7(C(=O)Nc8ccc(C(F)(F)F)cc8Cl)CCC7)c6)C5)ccc2c34)C(=O)N1	C37H30ClF3N6O4	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-R8TFTE	SCHEMBL25026651	N-(7-cyano-2,3-dihydro-1H-inden-4-yl)-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide; SCHEMBL30137329	CC(C)(C(=O)Nc1ccc(C#N)c2c1CCC2)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C35H31N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-ZK8NJQ	SCHEMBL25026460	N-[2-chloro-4-(trifluoromethyl)phenyl]-1-[4-[2-[1-[4-[(2,6-dioxopiperidin-3-yl)amino]-2-fluorophenyl]azetidin-3-yl]ethynyl]pyrazol-1-yl]cyclobutane-1-carboxamide	O=C1CCC(Nc2ccc(N3CC(C#Cc4cnn(C5(C(=O)Nc6ccc(C(F)(F)F)cc6Cl)CCC5)c4)C3)c(F)c2)C(=O)N1	C31H27ClF4N6O3	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-RC7M2D	EP-4385985-A1_143	.	O=C1CCC(N2C(=O)c3cc(N4CC(C#Cc5cnn(C6(C(=O)Nc7ccc(C(F)(F)F)cc7Cl)CCC6)c5)C4)c4c(c3C2O)OCO4)C(=O)N1	C34H28ClF3N6O7	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-SS631R	SCHEMBL25025013	N-(7-cyano-2,2-difluoro-1,3-benzodioxol-4-yl)-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide; SCHEMBL30137313	CC(C)(C(=O)Nc1ccc(C#N)c2c1OC(F)(F)O2)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C33H25F2N7O7	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-IXE6XW	SCHEMBL25026346	N-(4-chloro-3-cyanophenyl)-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide; SCHEMBL30137250	CC(C)(C(=O)Nc1ccc(Cl)c(C#N)c1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C32H26ClN7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-M0T7AQ	SCHEMBL25025005	2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methyl-N-[4-(trifluoromethyl)phenyl]propanamide	CC(C)(C(=O)Nc1ccc(C(F)(F)F)cc1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C32H27F3N6O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-R054SX	SCHEMBL25026318	N-[4-cyano-3-(trifluoromethyl)phenyl]-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-3-methylbutanamide; SCHEMBL30137336	CC(C)C(C(=O)Nc1ccc(C#N)c(C(F)(F)F)c1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C34H28F3N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-W3R9B2	EP-4385985-A1_148	.	COc1c(C)cc(NC(=O)C(C)(C)n2cc(C#CC3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)cn2)cc1C#N	C34H31N7O6	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-V96GNS	SCHEMBL25026466	2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-N-[2-(2-methoxyethoxy)-4-(trifluoromethyl)phenyl]-2-methylpropanamide	COCCOc1cc(C(F)(F)F)ccc1NC(=O)C(C)(C)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C35H33F3N6O7	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-XQG8LT	SCHEMBL25026189	N-[2-chloro-4-(trifluoromethyl)phenyl]-1-[4-[2-[1-[3-(2,6-dioxopiperidin-3-yl)-2-methyl-4-oxoquinazolin-7-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]cyclobutane-1-carboxamide	Cc1nc2cc(N3CC(C#Cc4cnn(C5(C(=O)Nc6ccc(C(F)(F)F)cc6Cl)CCC5)c4)C3)ccc2c(=O)n1C1CCC(=O)NC1=O	C34H29ClF3N7O4	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-6PDDKB	SCHEMBL25026320	1-[4-[(3aS,6aR)-2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-5-yl]pyrazol-1-yl]-N-[2-chloro-4-(trifluoromethyl)phenyl]cyclobutane-1-carboxamide; SCHEMBL31597113	O=C1CCC(N2C(=O)c3ccc(N4C[C@@H]5CN(c6cnn(C7(C(=O)Nc8ccc(C(F)(F)F)cc8Cl)CCC7)c6)C[C@@H]5C4)cc3C2=O)C(=O)N1	C34H31ClF3N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-CEMGYY	SCHEMBL25025033	N-(4-cyano-2,3-dimethylphenyl)-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide; SCHEMBL30137345	Cc1c(C#N)ccc(NC(=O)C(C)(C)n2cc(C#CC3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)cn2)c1C	C34H31N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-MJD0CU	SCHEMBL25026310	N-[2-chloro-4-(trifluoromethyl)phenyl]-1-[4-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperidin-1-yl]pyrazol-1-yl]cyclobutane-1-carboxamide; SCHEMBL30137412	O=C1CCC(N2C(=O)c3ccc(N4CCC(C5CCN(c6cnn(C7(C(=O)Nc8ccc(C(F)(F)F)cc8Cl)CCC7)c6)CC5)CC4)cc3C2=O)C(=O)N1	C38H39ClF3N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-WHQUK3	SCHEMBL25026326	2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-N-[2-hydroxy-4-(trifluoromethyl)phenyl]-2-methylpropanamide; SCHEMBL30137426	CC(C)(C(=O)Nc1ccc(C(F)(F)F)cc1O)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C32H27F3N6O6	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-J7V5IK	SCHEMBL25026474	2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methyl-N-[2-(1,3-thiazol-2-yl)-4-(trifluoromethyl)phenyl]propanamide; SCHEMBL30137299	CC(C)(C(=O)Nc1ccc(C(F)(F)F)cc1-c1nccs1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C35H28F3N7O5S	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-O20CC6	SCHEMBL25025010	2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-N-[2-imidazol-1-yl-4-(trifluoromethyl)phenyl]-2-methylpropanamide; SCHEMBL31597270	CC(C)(C(=O)Nc1ccc(C(F)(F)F)cc1-n1ccnc1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C35H29F3N8O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-J9VSBE	SCHEMBL25026655	N-[2-(4-cyclopropylpiperidin-1-yl)-4-(trifluoromethyl)phenyl]-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide; SCHEMBL30137246	CC(C)(C(=O)Nc1ccc(C(F)(F)F)cc1N1CCC(C2CC2)CC1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C40H40F3N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-C2CYRQ	SCHEMBL25026652	2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methyl-N-[6-prop-2-enylidene-4-(trifluoromethyl)cyclohexa-2,4-dien-1-ylidene]propanamide; SCHEMBL30137407	C=C=Cc1cc(C(F)(F)F)ccc1NC(=O)C(C)(C)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C35H29F3N6O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-ZUDCY6	SCHEMBL25024983	N-[2-chloro-4-(trifluoromethyl)phenyl]-1-[5-cyano-4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]cyclobutane-1-carboxamide; SCHEMBL30137397	N#Cc1c(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cnn1C1(C(=O)Nc2ccc(C(F)(F)F)cc2Cl)CCC1	C34H25ClF3N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-9VCS5F	SCHEMBL25026325	N-[2-chloro-4-(trifluoromethyl)phenyl]-1-[3-cyano-4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]cyclobutane-1-carboxamide; SCHEMBL30137320	N#Cc1nn(C2(C(=O)Nc3ccc(C(F)(F)F)cc3Cl)CCC2)cc1C#CC1CN(c2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)C1	C34H25ClF3N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-M779PR	SCHEMBL25025000	N-[2-chloro-4-(trifluoromethyl)phenyl]-2-[6-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]benzimidazol-1-yl]-2-methylpropanamide	CC(C)(C(=O)Nc1ccc(C(F)(F)F)cc1Cl)n1cnc2ccc(C#CC3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)cc21	C36H28ClF3N6O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-BBLL3A	SCHEMBL25024997	N-[2-chloro-4-(trifluoromethyl)phenyl]-2-[5-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]benzimidazol-1-yl]-2-methylpropanamide	CC(C)(C(=O)Nc1ccc(C(F)(F)F)cc1Cl)n1cnc2cc(C#CC3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)ccc21	C36H28ClF3N6O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-V57O8T	SCHEMBL25026324	N-[2-chloro-4-(trifluoromethyl)phenyl]-1-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]-5-methylpyrazol-1-yl]cyclobutane-1-carboxamide; SCHEMBL30137272	Cc1c(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cnn1C1(C(=O)Nc2ccc(C(F)(F)F)cc2Cl)CCC1	C34H28ClF3N6O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-ZNRZPO	SCHEMBL25026335	N-[2-chloro-4-(trifluoromethyl)phenyl]-1-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]-3-methylpyrazol-1-yl]cyclobutane-1-carboxamide; SCHEMBL30137371	Cc1nn(C2(C(=O)Nc3ccc(C(F)(F)F)cc3Cl)CCC2)cc1C#CC1CN(c2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)C1	C34H28ClF3N6O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-BN6R5R	SCHEMBL25025054	N-(6-cyano-3-tricyclo[6.2.1.02,7]undeca-2,4,6-trienyl)-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide; SCHEMBL30137260	CC(C)(C(=O)Nc1ccc(C#N)c2c1C1CCC2C1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C37H33N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-26J00A	SCHEMBL25026334	N-[2-chloro-4-(trifluoromethyl)phenyl]-1-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]-3,5-dimethylpyrazol-1-yl]cyclobutane-1-carboxamide; SCHEMBL30137355	Cc1nn(C2(C(=O)Nc3ccc(C(F)(F)F)cc3Cl)CCC2)c(C)c1C#CC1CN(c2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)C1	C35H30ClF3N6O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-2ZGTYW	SCHEMBL25025037	2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methyl-N-[2-(2-oxopyrrolidin-1-yl)-4-(trifluoromethyl)phenyl]propanamide	CC(C)(C(=O)Nc1ccc(C(F)(F)F)cc1N1CCCC1=O)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C36H32F3N7O6	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-JN1VDH	SCHEMBL25026490	N-[2-chloro-4-(trifluoromethyl)phenyl]-1-[4-[2-[1-[4-(2,6-dioxopiperidin-3-yl)phenyl]azetidin-3-yl]ethynyl]pyrazol-1-yl]cyclobutane-1-carboxamide; SCHEMBL30137327	O=C1CCC(c2ccc(N3CC(C#Cc4cnn(C5(C(=O)Nc6ccc(C(F)(F)F)cc6Cl)CCC5)c4)C3)cc2)C(=O)N1	C31H27ClF3N5O3	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-BPU86R	SCHEMBL25026485	2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methyl-N-[2-prop-2-enyl-4-(trifluoromethyl)phenyl]propanamide; SCHEMBL30137391	C=CCc1cc(C(F)(F)F)ccc1NC(=O)C(C)(C)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C35H31F3N6O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-BIEU8P	SCHEMBL30137369	N-[2-chloro-4-(1,1,1,2,3,3,3-heptafluoropropan-2-yl)phenyl]-1-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]cyclobutane-1-carboxamide	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cnn(C6(C(=O)Nc7ccc(C(F)(C(F)(F)F)C(F)(F)F)cc7Cl)CCC6)c5)C4)cc3C2=O)C(=O)N1	C35H26ClF7N6O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-DNL2DR	SCHEMBL30137432	N-[2-chloro-4-(trifluoromethyl)phenyl]-1-[4-[2-[1-[2-(2,5-dioxopyrrolidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]cyclobutane-1-carboxamide	O=C1CC(N2C(=O)c3ccc(N4CC(C#Cc5cnn(C6(C(=O)Nc7ccc(C(F)(F)F)cc7Cl)CCC6)c5)C4)cc3C2=O)C(=O)N1	C32H24ClF3N6O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-1138DY	SCHEMBL25025066	N-(4-cyano-2-pyrazol-1-ylphenyl)-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide; SCHEMBL30137431	CC(C)(C(=O)Nc1ccc(C#N)cc1-n1cccn1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C35H29N9O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-HDJAX4	SCHEMBL25026333	N-[2-cyclopentyl-4-(trifluoromethyl)phenyl]-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide; SCHEMBL30137410	CC(C)(C(=O)Nc1ccc(C(F)(F)F)cc1C1CCCC1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C37H35F3N6O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-GAYRL3	SCHEMBL30137442	N-[2-chloro-4-(trifluoromethyl)phenyl]-1-[4-[2-[1-[2-(2,7-dioxoazepan-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]cyclobutane-1-carboxamide	O=C1CCCC(N2C(=O)c3ccc(N4CC(C#Cc5cnn(C6(C(=O)Nc7ccc(C(F)(F)F)cc7Cl)CCC6)c5)C4)cc3C2=O)C(=O)N1	C34H28ClF3N6O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-LFR7SS	SCHEMBL25026332	N-[2-cyclohexyl-4-(trifluoromethyl)phenyl]-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide; SCHEMBL30137245	CC(C)(C(=O)Nc1ccc(C(F)(F)F)cc1C1CCCCC1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C38H37F3N6O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-ASXIKE	SCHEMBL25025071	N-[2-(cyclopropylmethyl)-4-(trifluoromethyl)phenyl]-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide; SCHEMBL30137349	CC(C)(C(=O)Nc1ccc(C(F)(F)F)cc1CC1CC1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C36H33F3N6O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-98105M	SCHEMBL25024833	2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methyl-N-[1-methyl-2-oxo-6-(trifluoromethyl)pyridin-3-yl]propanamide	Cn1c(C(F)(F)F)ccc(NC(=O)C(C)(C)n2cc(C#CC3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)cn2)c1=O	C32H28F3N7O6	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-ZOME9A	SCHEMBL25026508	N-(4-cyano-2-cyclopropylphenyl)-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]-3,5-dimethylpyrazol-1-yl]-2-methylpropanamide; SCHEMBL30137324	Cc1nn(C(C)(C)C(=O)Nc2ccc(C#N)cc2C2CC2)c(C)c1C#CC1CN(c2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)C1	C37H35N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-8PFMUL	SCHEMBL25024836	N-(2-chloro-4-prop-1-ynylphenyl)-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide; SCHEMBL30137417	CC#Cc1ccc(NC(=O)C(C)(C)n2cc(C#CC3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)cn2)c(Cl)c1	C34H29ClN6O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-UH9K4Y	SCHEMBL25024837	N-[2-chloro-4-(dimethylamino)phenyl]-1-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]cyclobutane-1-carboxamide; SCHEMBL30137356	CN(C)c1ccc(NC(=O)C2(n3cc(C#CC4CN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)cn3)CCC2)c(Cl)c1	C34H32ClN7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-3C30J6	SCHEMBL25024838	N-[2-(dimethylamino)-4-(trifluoromethyl)phenyl]-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide; SCHEMBL30137303	CN(C)c1cc(C(F)(F)F)ccc1NC(=O)C(C)(C)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C34H32F3N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-Y6292A	SCHEMBL25024835	N-(4-cyano-2-cyclopropylphenyl)-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide	CC(C)(C(=O)Nc1ccc(C#N)cc1C1CC1)n1cc(C#CC2CN(c3cc4c(cc3F)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C35H30FN7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-U6VYIJ	SCHEMBL25026835	N-(4-cyano-2-cyclopropylphenyl)-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]-3-methylpyrazol-1-yl]-2-methylpropanamide; SCHEMBL30137460	Cc1nn(C(C)(C)C(=O)Nc2ccc(C#N)cc2C2CC2)cc1C#CC1CN(c2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)C1	C36H33N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-ICOQL2	SCHEMBL25026838	N-(4-cyano-2-cyclopropylphenyl)-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]-5-methylpyrazol-1-yl]-2-methylpropanamide; SCHEMBL31597116	Cc1c(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cnn1C(C)(C)C(=O)Nc1ccc(C#N)cc1C1CC1	C36H33N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-IMMFYV	SCHEMBL25024793	2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-N-[2-ethynyl-4-(trifluoromethyl)phenyl]-2-methylpropanamide	C#Cc1cc(C(F)(F)F)ccc1NC(=O)C(C)(C)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C34H27F3N6O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-BRGWPG	SCHEMBL25026657	N-(4-cyano-2-ethynylphenyl)-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide; SCHEMBL30137352	C#Cc1cc(C#N)ccc1NC(=O)C(C)(C)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C34H27N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-5D7K4T	SCHEMBL25024808	N-[2-(2,2-difluoroethenyl)-4-(trifluoromethyl)phenyl]-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide; SCHEMBL30137439	CC(C)(C(=O)Nc1ccc(C(F)(F)F)cc1C=C(F)F)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C34H27F5N6O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-8OPWOV	SCHEMBL25026356	N-[2-chloro-4-(trifluoromethyl)phenyl]-1-[3-cyclopropyl-4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]cyclobutane-1-carboxamide; SCHEMBL30137357	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cn(C6(C(=O)Nc7ccc(C(F)(F)F)cc7Cl)CCC6)nc5C5CC5)C4)cc3C2=O)C(=O)N1	C36H30ClF3N6O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-952OT4	SCHEMBL25024829	2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]-3,5-dimethylpyrazol-1-yl]-2-methyl-N-[2-prop-1-ynyl-4-(trifluoromethyl)phenyl]propanamide	CC#Cc1cc(C(F)(F)F)ccc1NC(=O)C(C)(C)n1nc(C)c(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)c1C	C37H33F3N6O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-Q73DGE	SCHEMBL25026580	2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]-3-methylpyrazol-1-yl]-2-methyl-N-[2-prop-1-ynyl-4-(trifluoromethyl)phenyl]propanamide	CC#Cc1cc(C(F)(F)F)ccc1NC(=O)C(C)(C)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)c(C)n1	C36H31F3N6O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-VCEDSQ	SCHEMBL25024842	2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]-5-methylpyrazol-1-yl]-2-methyl-N-[2-prop-1-ynyl-4-(trifluoromethyl)phenyl]propanamide	CC#Cc1cc(C(F)(F)F)ccc1NC(=O)C(C)(C)n1ncc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)c1C	C36H31F3N6O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-OGR45F	SCHEMBL25024843	N-[2-chloro-4-(trifluoromethyl)phenyl]-1-[5-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]-4,6-dihydropyrrolo[3,4-c]pyrazol-2-yl]cyclobutane-1-carboxamide; SCHEMBL30137351	O=C1CCC(N2C(=O)c3ccc(N4CCC(N5Cc6cn(C7(C(=O)Nc8ccc(C(F)(F)F)cc8Cl)CCC7)nc6C5)CC4)cc3C2=O)C(=O)N1	C35H33ClF3N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-7LQ42Z	SCHEMBL30137247	N-[2-chloro-4-(trifluoromethyl)phenyl]-1-[5-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]-4,6-dihydropyrrolo[3,4-c]pyrazol-1-yl]cyclobutane-1-carboxamide	O=C1CCC(N2C(=O)c3ccc(N4CCC(N5Cc6cnn(C7(C(=O)Nc8ccc(C(F)(F)F)cc8Cl)CCC7)c6C5)CC4)cc3C2=O)C(=O)N1	C35H33ClF3N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-SFVBHH	SCHEMBL25025084	N-[2-chloro-4-(trifluoromethyl)phenyl]-1-[5-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]-4,6-dihydropyrrolo[3,4-c]pyrazol-2-yl]cyclobutane-1-carboxamide; SCHEMBL30137387	O=C1CCC(N2C(=O)c3ccc(N4CC(N5Cc6cn(C7(C(=O)Nc8ccc(C(F)(F)F)cc8Cl)CCC7)nc6C5)C4)cc3C2=O)C(=O)N1	C33H29ClF3N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-NAHKMI	SCHEMBL25026577	N-[2-chloro-4-(trifluoromethyl)phenyl]-1-[5-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]-4,6-dihydropyrrolo[3,4-c]pyrazol-1-yl]cyclobutane-1-carboxamide; SCHEMBL30137325	O=C1CCC(N2C(=O)c3ccc(N4CC(N5Cc6cnn(C7(C(=O)Nc8ccc(C(F)(F)F)cc8Cl)CCC7)c6C5)C4)cc3C2=O)C(=O)N1	C33H29ClF3N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-1B8LE2	SCHEMBL25026578	N-[2-chloro-4-(trifluoromethyl)phenyl]-1-[5-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]methyl]-4,6-dihydropyrrolo[3,4-c]pyrazol-2-yl]cyclobutane-1-carboxamide; SCHEMBL30137422	O=C1CCC(N2C(=O)c3ccc(N4CC(CN5Cc6cn(C7(C(=O)Nc8ccc(C(F)(F)F)cc8Cl)CCC7)nc6C5)C4)cc3C2=O)C(=O)N1	C34H31ClF3N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-J7IC1Q	SCHEMBL30137294	N-[2-chloro-4-(trifluoromethyl)phenyl]-1-[5-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]methyl]-4,6-dihydropyrrolo[3,4-c]pyrazol-1-yl]cyclobutane-1-carboxamide	O=C1CCC(N2C(=O)c3ccc(N4CC(CN5Cc6cnn(C7(C(=O)Nc8ccc(C(F)(F)F)cc8Cl)CCC7)c6C5)C4)cc3C2=O)C(=O)N1	C34H31ClF3N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-BHL331	SCHEMBL25025090	N-(4-cyano-2-cyclopropylphenyl)-2-[3-cyano-4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide; SCHEMBL30137448	CC(C)(C(=O)Nc1ccc(C#N)cc1C1CC1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)c(C#N)n1	C36H30N8O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-H3YPXF	SCHEMBL25025087	2-[3-cyano-4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methyl-N-[2-prop-1-ynyl-4-(trifluoromethyl)phenyl]propanamide; SCHEMBL30137450	CC#Cc1cc(C(F)(F)F)ccc1NC(=O)C(C)(C)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)c(C#N)n1	C36H28F3N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-G19NE9	SCHEMBL25027213	N-[2-chloro-4-(trifluoromethyl)phenyl]-1-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-3,3-difluorocyclobutane-1-carboxamide; SCHEMBL30137269	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cnn(C6(C(=O)Nc7ccc(C(F)(F)F)cc7Cl)CC(F)(F)C6)c5)C4)cc3C2=O)C(=O)N1	C33H24ClF5N6O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-WGPFAU	SCHEMBL25024846	2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methyl-N-[2-prop-1-ynyl-4-(trifluoromethyl)phenyl]propanamide	CC#Cc1cc(C(F)(F)F)ccc1NC(=O)C(C)(C)n1cc(C#CC2CN(c3cc4c(cc3F)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C35H28F4N6O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-E0S950	SCHEMBL25026322	N-[2-chloro-4-(trifluoromethyl)phenyl]-1-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]-3-(trifluoromethyl)pyrazol-1-yl]cyclobutane-1-carboxamide	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cn(C6(C(=O)Nc7ccc(C(F)(F)F)cc7Cl)CCC6)nc5C(F)(F)F)C4)cc3C2=O)C(=O)N1	C34H25ClF6N6O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-MF51B4	SCHEMBL25026582	N-[2-cyclopropyl-4-(trifluoromethyl)phenyl]-2-[5-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]-4,6-dihydropyrrolo[3,4-c]pyrazol-1-yl]-2-methylpropanamide; SCHEMBL30137277	CC(C)(C(=O)Nc1ccc(C(F)(F)F)cc1C1CC1)n1ncc2c1CN(C1CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C1)C2	C35H34F3N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-O335VX	SCHEMBL25027202	N-[2-cyclopropyl-4-(trifluoromethyl)phenyl]-2-[5-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]methyl]-4,6-dihydropyrrolo[3,4-c]pyrazol-1-yl]-2-methylpropanamide; SCHEMBL30137481	CC(C)(C(=O)Nc1ccc(C(F)(F)F)cc1C1CC1)n1ncc2c1CN(CC1CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C1)C2	C36H36F3N7O5	AR-V7	P10275-3	CRBN	EP-4385985-A1
TPD-S1W1SA	EP4003979B1_25	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCOCCOCCN3C=C(CNC(=O)C4=CC(NC5=NNC(C6CC6)=C5)=NC(NC5=CC=C(CC#N)C=C5)=N4)N=N3)C(C)(C)C)C=C2)SC=N1	C51H61N15O7S	CHEK1	O14757	VHL	EP-4003979-B1
TPD-OT3IAO	EP4003979B1_26	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCOCCOCCOCCN3C=C(CNC(=O)C4=CC(NC5=NNC(C6CC6)=C5)=NC(NC5=CC=C(CC#N)C=C5)=N4)N=N3)C(C)(C)C)C=C2)SC=N1	C53H65N15O8S	CHEK1	O14757	VHL	EP-4003979-B1
TPD-UMKS51	EP4003979B1_27	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCOCCOCCOCCOCCN3C=C(CNC(=O)C4=CC(NC5=NNC(C6CC6)=C5)=NC(NC5=CC=C(CC#N)C=C5)=N4)N=N3)C(C)(C)C)C=C2)SC=N1	C55H69N15O9S	CHEK1	O14757	VHL	EP-4003979-B1
TPD-ZL9TNC	EP4003979B1_28	.	N#CCC1=CC=C(NC2=NC(C(=O)NCC3=CN(CCOCCNC(=O)COC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)N=N3)=CC(NC3=NNC(C4CC4)=C3)=N2)C=C1	C41H40N14O8	CHEK1	O14757	CRBN	EP-4003979-B1
TPD-FKDK9Y	PROTAC Chk1 degrader-1	PROTAC Chk1 degrader-1; orb2565422; HY-161108; CS-0927652; 2597167-34-3	N#CCC1=CC=C(NC2=NC(C(=O)NCC3=CN(CCOCCOCCNC(=O)COC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)N=N3)=CC(NC3=NNC(C4CC4)=C3)=N2)C=C1	C43H44N14O9	CHEK1	O14757	CRBN	EP-4003979-B1
TPD-4BT3T9	EP4003979B1_30	.	N#CCC1=CC=C(NC2=NC(C(=O)NCC3=CN(CCOCCOCCOCCNC(=O)COC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)N=N3)=CC(NC3=NNC(C4CC4)=C3)=N2)C=C1	C45H48N14O10	CHEK1	O14757	CRBN	EP-4003979-B1
TPD-TYKKIF	EP4003979B1_31	.	N#CCC1=CC=C(NC2=NC(C(=O)NCC3=CN(CCOCCOCCOCCOCCNC(=O)COC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)N=N3)=CC(NC3=NNC(C4CC4)=C3)=N2)C=C1	C47H52N14O11	CHEK1	O14757	CRBN	EP-4003979-B1
TPD-S8O3RK	EP4023649A1_1	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCOC3=CC=C(C4CCN(C5=NN6C(=NN=C6C(F)(F)F)CC5)CC4)C=C3)C(C)(C)C)C=C2)SC=N1	C45H56F3N9O6S	AR	P10275	VHL	EP-4023649-A1
TPD-UUBKDB	EP4023649A1_2	(2S,4S)-1-[(2S)-3,3-dimethyl-2-[5-[4-[[4-[1-[3-(trifluoromethyl)-7,8-dihydro-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]piperidin-4-yl]phenoxy]methyl]phenyl]pent-4-ynoylamino]butanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@H](O)CN3C(=O)[C@@H](NC(=O)CCC#CC3=CC=C(COC4=CC=C(C5CCN(C6=NN7C(=NN=C7C(F)(F)F)CC6)CC5)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C51H56F3N9O5S	AR	P10275	VHL	EP-4023649-A1
TPD-45WEMQ	EP4023649A1_3	(2S,4S)-1-[(2S)-3,3-dimethyl-2-[[2-[3-[2-[[2-[4-[1-[3-(trifluoromethyl)-7,8-dihydro-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]piperidin-4-yl]phenoxy]acetyl]amino]ethoxy]propoxy]acetyl]amino]butanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@H](O)CN3C(=O)[C@@H](NC(=O)COCCCOCCNC(=O)COC3=CC=C(C4CCN(C5=NN6C(=NN=C6C(F)(F)F)CC5)CC4)C=C3)C(C)(C)C)C=C2)SC=N1	C48H61F3N10O8S	AR	P10275	VHL	EP-4023649-A1
TPD-DI6CID	EP4023649A1_4	(2S,4S)-1-[(2S)-3,3-dimethyl-2-[3-[2-[2-[4-[5-[2-[4-[1-[3-(trifluoromethyl)-7,8-dihydro-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]piperidin-4-yl]phenyl]ethynyl]pyridin-2-yl]piperazin-1-yl]ethoxy]ethoxy]propanoylamino]butanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@H](O)CN3C(=O)[C@@H](NC(=O)CCOCCOCCN3CCN(C4=NC=C(C#CC5=CC=C(C6CCN(C7=NN8C(=NN=C8C(F)(F)F)CC7)CC6)C=C5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C57H69F3N12O6S	AR	P10275	VHL	EP-4023649-A1
TPD-TEV980	EP4023649A1_5	(2S,4S)-1-[(2S)-3,3-dimethyl-2-[3-[2-[2-[4-[2-[4-[1-[3-(trifluoromethyl)-7,8-dihydro-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]piperidin-4-yl]phenoxy]acetyl]piperazin-1-yl]ethoxy]ethoxy]propanoylamino]butanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@H](O)CN3C(=O)[C@@H](NC(=O)CCOCCOCCN3CCN(C(=O)COC4=CC=C(C5CCN(C6=NN7C(=NN=C7C(F)(F)F)CC6)CC5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C52H68F3N11O8S	AR	P10275	VHL	EP-4023649-A1
TPD-SFP28C	SCHEMBL24592103	(4R)-4-hydroxy-1-[(2R)-3-methyl-2-(3-methyl-1,2-oxazol-5-yl)butanoyl]-N-[1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]-3-oxo-3-[2-[4-[4-[1-[3-(trifluoromethyl)-7,8-dihydro-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]piperidin-4-yl]phenoxy]butoxy]ethylamino]propyl]pyrrolidine-2-carboxamide	CC1=NOC([C@H](C(=O)N2C[C@H](O)CC2C(=O)NC(CC(=O)NCCOCCCCOC2=CC=C(C3CCN(C4=NN5C(=NN=C5C(F)(F)F)CC4)CC3)C=C2)C2=CC=C(C3=C(C)N=CS3)C=C2)C(C)C)=C1	C50H61F3N10O7S	AR	P10275	VHL	EP-4023649-A1
TPD-U5N0HH	EP4023649A1_7	(2S,4S)-1-[2-[[2-[(3R,4S,5R)-3,4-dihydroxy-5-[[[2-[4-[1-[3-(trifluoromethyl)-7,8-dihydro-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]piperidin-4-yl]phenoxy]acetyl]amino]methyl]oxolan-2-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@H](O)CN3C(=O)C(NC(=O)CC3O[C@H](CNC(=O)COC4=CC=C(C5CCN(C6=NN7C(=NN=C7C(F)(F)F)CC6)CC5)C=C4)[C@@H](O)[C@H]3O)C(C)(C)C)C=C2)SC=N1	C48H59F3N10O9S	AR	P10275	VHL	EP-4023649-A1
TPD-9OOM53	EP4023649A1_8	(2S,4S)-1-[(2S)-3,3-dimethyl-2-[[2-[4-[4-[1-[3-[4-(trifluoromethyl)phenyl]-7,8-dihydro-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]piperidin-4-yl]phenoxy]butoxy]acetyl]amino]butanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCOC3=CC=C(C4CCN(C5=NN6C(=NN=C6C6=CC=C(C(F)(F)F)C=C6)CC5)CC4)C=C3)C(C)(C)C)C=C2)SC=N1	C51H60F3N9O6S	AR	P10275	VHL	EP-4023649-A1
TPD-O9IIW5	SCHEMBL24592128	(4R)-4-hydroxy-1-[(2R)-3-methyl-2-(3-methyl-1,2-oxazol-5-yl)butanoyl]-N-[1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]-3-oxo-3-[4-[4-[2-[4-[1-[3-(trifluoromethyl)-7,8-dihydro-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]piperidin-4-yl]phenyl]ethynyl]piperidin-1-yl]piperidin-1-yl]propyl]pyrrolidine-2-carboxamide	CC1=NOC([C@H](C(=O)N2C[C@H](O)CC2C(=O)NC(CC(=O)N2CCC(N3CCC(C#CC4=CC=C(C5CCN(C6=NN7C(=NN=C7C(F)(F)F)CC6)CC5)C=C4)CC3)CC2)C2=CC=C(C3=C(C)N=CS3)C=C2)C(C)C)=C1	C56H66F3N11O5S	AR	P10275	VHL	EP-4023649-A1
TPD-A8G1DF	EP4023649A1_10	(2S,4S)-1-[(2S)-3,3-dimethyl-2-[[4-[4-[5-[2-[4-[1-[3-(trifluoromethyl)-7,8-dihydro-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]piperidin-4-yl]phenyl]ethynyl]pyridin-2-yl]piperazin-1-yl]cyclohexanecarbonyl]amino]butanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@H](O)CN3C(=O)[C@@H](NC(=O)C3CCC(N4CCN(C5=NC=C(C#CC6=CC=C(C7CCN(C8=NN9C(=NN=C9C(F)(F)F)CC8)CC7)C=C6)C=C5)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C57H67F3N12O4S	AR	P10275	VHL	EP-4023649-A1
TPD-ZSKT4L	EP4023649A1_11	(2S,4S)-1-[(2S)-3,3-dimethyl-2-[[2-[4-[5-[2-[4-[1-[3-(trifluoromethyl)-7,8-dihydro-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]piperidin-4-yl]phenyl]ethynyl]pyridin-2-yl]piperazin-1-yl]acetyl]amino]butanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCN(C4=NC=C(C#CC5=CC=C(C6CCN(C7=NN8C(=NN=C8C(F)(F)F)CC7)CC6)C=C5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C52H59F3N12O4S	AR	P10275	VHL	EP-4023649-A1
TPD-IBWJZ6	SCHEMBL24592105	5-[2-[1-[1-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]acetyl]piperidin-4-yl]piperidin-4-yl]ethynyl]-N-[4-[1-[3-(trifluoromethyl)-7,8-dihydro-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]piperidin-4-yl]phenyl]pyridine-2-carboxamide	O=C1CCC(N2C(=O)C3=CC=CC(NCC(=O)N4CCC(N5CCC(C#CC6=CC=C(C(=O)NC7=CC=C(C8CCN(C9=NN%10C(=NN=C%10C(F)(F)F)CC9)CC8)C=C7)N=C6)CC5)CC4)=C3C2=O)C(=O)N1	C50H51F3N12O6	AR	P10275	CRBN	EP-4023649-A1
TPD-4I8LC7	EP4023649A1_13	(2S,4S)-1-[(2S)-3,3-dimethyl-2-[4-[4-[2-[4-[1-[3-(trifluoromethyl)-7,8-dihydro-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]piperidin-4-yl]phenyl]ethynyl]piperidin-1-yl]butanoylamino]butanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@H](O)CN3C(=O)[C@@H](NC(=O)CCCN3CCC(C#CC4=CC=C(C5CCN(C6=NN7C(=NN=C7C(F)(F)F)CC6)CC5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C50H61F3N10O4S	AR	P10275	VHL	EP-4023649-A1
TPD-0HK63C	SCHEMBL24592216	(2S,4R)-4-hydroxy-1-[(2R)-3-methyl-2-(3-methyl-1,2-oxazol-5-yl)butanoyl]-N-[1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]-3-oxo-3-[4-[2-[4-[1-[3-(trifluoromethyl)-7,8-dihydro-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]piperidin-4-yl]phenyl]ethynyl]piperidin-1-yl]propyl]pyrrolidine-2-carboxamide	CC1=NOC([C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NC(CC(=O)N2CCC(C#CC3=CC=C(C4CCN(C5=NN6C(=NN=C6C(F)(F)F)CC5)CC4)C=C3)CC2)C2=CC=C(C3=C(C)N=CS3)C=C2)C(C)C)=C1	C51H57F3N10O5S	AR	P10275	VHL	EP-4023649-A1
TPD-JI3PJA	EP4023649A1_15	(2S,4S)-1-[(2S)-3,3-dimethyl-2-[3-[4-[5-[2-[4-[1-[3-(trifluoromethyl)-7,8-dihydro-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]piperidin-4-yl]phenyl]ethynyl]pyridin-2-yl]piperazin-1-yl]propanoylamino]butanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@H](O)CN3C(=O)[C@@H](NC(=O)CCN3CCN(C4=NC=C(C#CC5=CC=C(C6CCN(C7=NN8C(=NN=C8C(F)(F)F)CC7)CC6)C=C5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C53H61F3N12O4S	AR	P10275	VHL	EP-4023649-A1
TPD-B9KSHH	EP4023649A1_16	(2S,4S)-1-[(2S)-3,3-dimethyl-2-[4-[4-[5-[2-[4-[1-[3-(trifluoromethyl)-7,8-dihydro-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]piperidin-4-yl]phenyl]ethynyl]pyridin-2-yl]piperazin-1-yl]butanoylamino]butanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@H](O)CN3C(=O)[C@@H](NC(=O)CCCN3CCN(C4=NC=C(C#CC5=CC=C(C6CCN(C7=NN8C(=NN=C8C(F)(F)F)CC7)CC6)C=C5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C54H63F3N12O4S	AR	P10275	VHL	EP-4023649-A1
TPD-XOGIUO	EP4023649A1_17	(2S,4S)-1-[(2S)-3,3-dimethyl-2-[5-[4-[5-[2-[4-[1-[3-(trifluoromethyl)-7,8-dihydro-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]piperidin-4-yl]phenyl]ethynyl]pyridin-2-yl]piperazin-1-yl]pentanoylamino]butanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@H](O)CN3C(=O)[C@@H](NC(=O)CCCCN3CCN(C4=NC=C(C#CC5=CC=C(C6CCN(C7=NN8C(=NN=C8C(F)(F)F)CC7)CC6)C=C5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C55H65F3N12O4S	AR	P10275	VHL	EP-4023649-A1
TPD-A75XTT	EP4023649A1_18	(2S,4S)-1-[(2S)-3,3-dimethyl-2-[6-[4-[5-[2-[4-[1-[3-(trifluoromethyl)-7,8-dihydro-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]piperidin-4-yl]phenyl]ethynyl]pyridin-2-yl]piperazin-1-yl]hexanoylamino]butanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCN3CCN(C4=NC=C(C#CC5=CC=C(C6CCN(C7=NN8C(=NN=C8C(F)(F)F)CC7)CC6)C=C5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C56H67F3N12O4S	AR	P10275	VHL	EP-4023649-A1
TPD-MB0ESI	EP4023649A1_19	(2S,4S)-1-[(2S)-3,3-dimethyl-2-[[2-[2-[4-[1-[3-(trifluoromethyl)-7,8-dihydro-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]piperidin-4-yl]phenoxy]ethoxy]acetyl]amino]butanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@H](O)CN3C(=O)[C@@H](NC(=O)COCCOC3=CC=C(C4CCN(C5=NN6C(=NN=C6C(F)(F)F)CC5)CC4)C=C3)C(C)(C)C)C=C2)SC=N1	C43H52F3N9O6S	AR	P10275	VHL	EP-4023649-A1
TPD-COCE7G	EP4023649A1_20	(2S,4S)-1-[(2S)-3,3-dimethyl-2-[[2-[3-[4-[1-[3-(trifluoromethyl)-7,8-dihydro-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]piperidin-4-yl]phenoxy]propoxy]acetyl]amino]butanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@H](O)CN3C(=O)[C@@H](NC(=O)COCCCOC3=CC=C(C4CCN(C5=NN6C(=NN=C6C(F)(F)F)CC5)CC4)C=C3)C(C)(C)C)C=C2)SC=N1	C44H54F3N9O6S	AR	P10275	VHL	EP-4023649-A1
TPD-DXI1C9	EP4023649A1_21	(2S,4S)-1-[(2S)-3,3-dimethyl-2-[[2-[5-[4-[1-[3-(trifluoromethyl)-7,8-dihydro-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]piperidin-4-yl]phenoxy]pentoxy]acetyl]amino]butanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCCOC3=CC=C(C4CCN(C5=NN6C(=NN=C6C(F)(F)F)CC5)CC4)C=C3)C(C)(C)C)C=C2)SC=N1	C46H58F3N9O6S	AR	P10275	VHL	EP-4023649-A1
TPD-3SSGQ7	EP4023649A1_23	(2S,4S)-1-[(2S)-3,3-dimethyl-2-[[2-[7-[4-[1-[3-(trifluoromethyl)-7,8-dihydro-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]piperidin-4-yl]phenoxy]heptoxy]acetyl]amino]butanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCCCCOC3=CC=C(C4CCN(C5=NN6C(=NN=C6C(F)(F)F)CC5)CC4)C=C3)C(C)(C)C)C=C2)SC=N1	C48H62F3N9O6S	AR	P10275	VHL	EP-4023649-A1
TPD-PWA1RG	EP4023649A1_24	.	CC1=C(C2=CC=C([C@@H](CC(=O)NCCOCCCCOC3=CC=C(C4CCN(C5=NN6C(=NN=C6C(F)(F)F)CC5)CC4)C=C3)NC(=O)C3C[C@@H](O)CN3C(=O)C(NC(=O)C3(F)CC3)C(C)(C)C)C=C2)SC=N1	C51H64F4N10O7S	AR	P10275	VHL	EP-4023649-A1
TPD-G730HE	EP4023649A1_25	(4R)-4-hydroxy-1-[3-methyl-2-(3-methyl-1,2-oxazol-5-yl)butanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]-3-oxo-3-[2-[4-[4-[1-[3-(trifluoromethyl)-7,8-dihydro-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]piperidin-4-yl]phenoxy]butoxy]ethylamino]propyl]pyrrolidine-2-carboxamide	CC1=NOC(C(C(=O)N2C[C@H](O)CC2C(=O)N[C@@H](CC(=O)NCCOCCCCOC2=CC=C(C3CCN(C4=NN5C(=NN=C5C(F)(F)F)CC4)CC3)C=C2)C2=CC=C(C3=C(C)N=CS3)C=C2)C(C)C)=C1	C50H61F3N10O7S	AR	P10275	VHL	EP-4023649-A1
TPD-AT8ZE3	EP4023649A1_26	.	CC1=C(C2=CC=C([C@H](CC(=O)NCCOCCCCOC3=CC=C(C4CCN(C5=NN6C(=NN=C6C(F)(F)F)CC5)CC4)C=C3)NC(=O)C3C[C@@H](O)CN3C(=O)C(NC(=O)C3(F)CC3)C(C)(C)C)C=C2)SC=N1	C51H64F4N10O7S	AR	P10275	VHL	EP-4023649-A1
TPD-NTCG6L	EP4023649A1_27	(4R)-1-[(2S)-2-[(1-cyanocyclopropanecarbonyl)amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]-3-oxo-3-[2-[4-[4-[1-[3-(trifluoromethyl)-7,8-dihydro-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]piperidin-4-yl]phenoxy]butoxy]ethylamino]propyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CC(=O)NCCOCCCCOC3=CC=C(C4CCN(C5=NN6C(=NN=C6C(F)(F)F)CC5)CC4)C=C3)NC(=O)C3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3(C#N)CC3)C(C)(C)C)C=C2)SC=N1	C52H64F3N11O7S	AR	P10275	VHL	EP-4023649-A1
TPD-DIGHKA	EP4023649A1_28	(2S,4S)-1-[(2S)-3,3-dimethyl-2-[[2-[4-[2-[4-[1-[3-(trifluoromethyl)-7,8-dihydro-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]piperidin-4-yl]phenoxy]ethyl]piperazin-1-yl]acetyl]amino]butanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCN(CCOC4=CC=C(C5CCN(C6=NN7C(=NN=C7C(F)(F)F)CC6)CC5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C47H60F3N11O5S	AR	P10275	VHL	EP-4023649-A1
TPD-N1V0YU	SCHEMBL24592383	1-[2-[[2-[(3R,4S,5R)-3,4-dihydroxy-5-[[4-[1-[3-(trifluoromethyl)-7,8-dihydro-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]piperidin-4-yl]phenoxy]methyl]oxolan-2-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)C3CC(O)CN3C(=O)C(NC(=O)CC3O[C@H](COC4=CC=C(C5CCN(C6=NN7C(=NN=C7C(F)(F)F)CC6)CC5)C=C4)[C@@H](O)[C@H]3O)C(C)(C)C)C=C2)SC=N1	C46H56F3N9O8S	AR	P10275	VHL	EP-4023649-A1
TPD-YR4VER	SCHEMBL24592201	3-[3-oxo-7-[6-[4-[1-[3-(trifluoromethyl)-7,8-dihydro-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]piperidin-4-yl]phenoxy]hex-1-ynyl]-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C#CCCCCOC4=CC=C(C5CCN(C6=NN7C(=NN=C7C(F)(F)F)CC6)CC5)C=C4)C=CC=C3C2=O)C(=O)N1	C36H36F3N7O4	AR	P10275	CRBN	EP-4023649-A1
TPD-4H1DK5	SCHEMBL24592138	N-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]-2-[6-[4-[1-[3-(trifluoromethyl)-7,8-dihydro-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]piperidin-4-yl]phenoxy]hexoxy]acetamide	O=C1CCC(N2CC3=C(NC(=O)COCCCCCCOC4=CC=C(C5CCN(C6=NN7C(=NN=C7C(F)(F)F)CC6)CC5)C=C4)C=CC=C3C2=O)C(=O)N1	C38H43F3N8O6	AR	P10275	CRBN	EP-4023649-A1
TPD-ON5B9A	EP4023649A1_33	(2S,4S)-1-[(2S)-3,3-dimethyl-2-[[4-[4-[2-[4-[1-[3-(trifluoromethyl)-7,8-dihydro-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]piperidin-4-yl]phenyl]ethynyl]piperidine-1-carbonyl]benzoyl]amino]butanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@H](O)CN3C(=O)[C@@H](NC(=O)C3=CC=C(C(=O)N4CCC(C#CC5=CC=C(C6CCN(C7=NN8C(=NN=C8C(F)(F)F)CC7)CC6)C=C5)CC4)C=C3)C(C)(C)C)C=C2)SC=N1	C54H59F3N10O5S	AR	P10275	VHL	EP-4023649-A1
TPD-7HPVGA	EP4023649A1_34	(2S,4S)-1-[(2S)-3,3-dimethyl-2-[[4-[4-[2-[4-[1-[3-(trifluoromethyl)-7,8-dihydro-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]piperidin-4-yl]phenyl]ethynyl]piperidine-1-carbonyl]cyclohexanecarbonyl]amino]butanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@H](O)CN3C(=O)[C@@H](NC(=O)C3CCC(C(=O)N4CCC(C#CC5=CC=C(C6CCN(C7=NN8C(=NN=C8C(F)(F)F)CC7)CC6)C=C5)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C54H65F3N10O5S	AR	P10275	VHL	EP-4023649-A1
TPD-0VAKHK	EP4023649A1_35	(2S,4S)-1-[(2S)-3,3-dimethyl-2-[[2-[4-[4-[1-[3-(trifluoromethyl)-7,8-dihydro-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]piperidin-4-yl]phenoxy]butoxy]acetyl]amino]butanoyl]-4-hydroxy-N-[[2-hydroxy-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC(O)=C(CNC(=O)[C@@H]3C[C@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCOC3=CC=C(C4CCN(C5=NN6C(=NN=C6C(F)(F)F)CC5)CC4)C=C3)C(C)(C)C)C=C2)SC=N1	C45H56F3N9O7S	AR	P10275	VHL	EP-4023649-A1
TPD-MI9NCI	SCHEMBL24592231	(4R)-1-[(2S)-2-[(1-fluorocyclopropanecarbonyl)amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)-2-[7-[4-[1-[3-(trifluoromethyl)-7,8-dihydro-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]piperidin-4-yl]phenoxy]heptoxy]phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)C3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3(F)CC3)C(C)(C)C)C(OCCCCCCCOC3=CC=C(C4CCN(C5=NN6C(=NN=C6C(F)(F)F)CC5)CC4)C=C3)=C2)SC=N1	C50H63F4N9O6S	AR	P10275	VHL	EP-4023649-A1
TPD-4JYITD	SCHEMBL24592175	N-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]-2-[4-[4-[1-[3-(trifluoromethyl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]piperidin-4-yl]phenoxy]butoxy]acetamide	O=C1CCC(N2CC3=C(NC(=O)COCCCCOC4=CC=C(C5CCN(C6=NN7C(=NN=C7C(F)(F)F)C=C6)CC5)C=C4)C=CC=C3C2=O)C(=O)N1	C36H37F3N8O6	AR	P10275	CRBN	EP-4023649-A1
TPD-BWH55T	SCHEMBL24592250	N-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]-7-[4-[1-[3-(trifluoromethyl)-7,8-dihydro-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]piperidin-4-yl]phenoxy]heptanamide	O=C1CCC(N2CC3=C(NC(=O)CCCCCCOC4=CC=C(C5CCN(C6=NN7C(=NN=C7C(F)(F)F)CC6)CC5)C=C4)C=CC=C3C2=O)C(=O)N1	C37H41F3N8O5	AR	P10275	CRBN	EP-4023649-A1
TPD-Y32ZLH	SCHEMBL24592139	3-[3-oxo-6-[1-[2-[4-[4-[1-[3-(trifluoromethyl)-7,8-dihydro-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]piperidin-4-yl]phenoxy]butoxy]acetyl]-3,6-dihydro-2H-pyridin-4-yl]-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(C4=CCN(C(=O)COCCCCOC5=CC=C(C6CCN(C7=NN8C(=NN=C8C(F)(F)F)CC7)CC6)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C41H45F3N8O6	AR	P10275	CRBN	EP-4023649-A1
TPD-HKRG14	SCHEMBL24592156	3-[3-oxo-6-[1-[2-[4-[4-[1-[3-(trifluoromethyl)-7,8-dihydro-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]piperidin-4-yl]phenoxy]butoxy]acetyl]piperidin-4-yl]-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(C4CCN(C(=O)COCCCCOC5=CC=C(C6CCN(C7=NN8C(=NN=C8C(F)(F)F)CC7)CC6)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C41H47F3N8O6	AR	P10275	CRBN	EP-4023649-A1
TPD-CI1JIU	SCHEMBL24592183	3-[3-oxo-6-[3-[4-[4-[1-[3-(trifluoromethyl)-7,8-dihydro-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]piperidin-4-yl]phenoxy]butoxy]prop-1-ynyl]-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(C#CCOCCCCOC4=CC=C(C5CCN(C6=NN7C(=NN=C7C(F)(F)F)CC6)CC5)C=C4)=CC=C3C2=O)C(=O)N1	C37H38F3N7O5	AR	P10275	CRBN	EP-4023649-A1
TPD-IZUG2W	SCHEMBL24592119	2-(2,6-Dioxopiperidin-3-yl)-4-[[2-oxo-2-[4-[4-[2-[4-[1-[3-(trifluoromethyl)-7,8-dihydro-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]piperidin-4-yl]phenyl]ethynyl]piperidin-1-yl]piperidin-1-yl]ethyl]amino]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC=CC(NCC(=O)N4CCC(N5CCC(C#CC6=CC=C(C7CCN(C8=NN9C(=NN=C9C(F)(F)F)CC8)CC7)C=C6)CC5)CC4)=C3C2=O)C(=O)N1	C44H47F3N10O5	AR	P10275	CRBN	EP-4023649-A1
TPD-G9BR2U	SCHEMBL24592124	2-(2,6-Dioxopiperidin-3-yl)-4-[4-[4-[2-[4-[1-[3-(trifluoromethyl)-7,8-dihydro-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]piperidin-4-yl]phenyl]ethynyl]piperidin-1-yl]piperidin-1-yl]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC=CC(N4CCC(N5CCC(C#CC6=CC=C(C7CCN(C8=NN9C(=NN=C9C(F)(F)F)CC8)CC7)C=C6)CC5)CC4)=C3C2=O)C(=O)N1	C42H44F3N9O4	AR	P10275	CRBN	EP-4023649-A1
TPD-VOY34R	SCHEMBL24592123	2-(2,6-Dioxopiperidin-3-yl)-4-[4-[2-[4-[4-[1-[3-(trifluoromethyl)-7,8-dihydro-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]piperidin-4-yl]phenoxy]butoxy]acetyl]piperazin-1-yl]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC=CC(N4CCN(C(=O)COCCCCOC5=CC=C(C6CCN(C7=NN8C(=NN=C8C(F)(F)F)CC7)CC6)C=C5)CC4)=C3C2=O)C(=O)N1	C40H44F3N9O7	AR	P10275	CRBN	EP-4023649-A1
TPD-3ZWLX3	SCHEMBL24592181	4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperidin-4-yl]ethynyl]-N-[2,2,4,4-tetramethyl-3-[[3-(trifluoromethyl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]oxy]cyclobutyl]benzamide	CC1(C)[C@H](NC(=O)C2=CC=C(C#CC3CCN(C4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)C=C2)C(C)(C)[C@H]1OC1=NN2C(=NN=C2C(F)(F)F)C=C1	C41H39F3N8O6	AR	P10275	CRBN	EP-4023649-A1
TPD-VDOEHT	SCHEMBL24592133	6-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoinden-4-yl]piperazin-1-yl]-N-[4-[[3-(trifluoromethyl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]oxy]cyclohexyl]pyridine-3-carboxamide	O=C1CCC(C2C(=O)C3=CC=CC(N4CCN(C5=CC=C(C(=O)N[C@H]6CC[C@H](OC7=NN8C(=NN=C8C(F)(F)F)C=C7)CC6)C=N5)CC4)=C3C2=O)C(=O)N1	C36H34F3N9O6	AR	P10275	CRBN	EP-4023649-A1
TPD-GWL7CY	SCHEMBL24592144	6-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoinden-4-yl]piperidin-4-yl]methyl]piperazin-1-yl]-N-[4-[[3-(trifluoromethyl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]oxy]cyclohexyl]pyridine-3-carboxamide	O=C1CCC(C2C(=O)C3=CC=CC(N4CCC(CN5CCN(C6=CC=C(C(=O)N[C@H]7CC[C@H](OC8=NN9C(=NN=C9C(F)(F)F)C=C8)CC7)C=N6)CC5)CC4)=C3C2=O)C(=O)N1	C42H45F3N10O6	AR	P10275	CRBN	EP-4023649-A1
TPD-ZIRB7F	SCHEMBL24592174	4-[2-[1-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]acetyl]piperidin-4-yl]ethynyl]-N-[2,2,4,4-tetramethyl-3-[[3-(trifluoromethyl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]oxy]cyclobutyl]benzamide	CC1(C)[C@H](NC(=O)C2=CC=C(C#CC3CCN(C(=O)CNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)C=C2)C(C)(C)[C@H]1OC1=NN2C(=NN=C2C(F)(F)F)C=C1	C43H42F3N9O7	AR	P10275	CRBN	EP-4023649-A1
TPD-2XKUDL	SCHEMBL24592245	3-[1,3-dioxo-4-[4-[[4-[5-[(1S,5R)-3-[[3-(trifluoromethyl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]oxy]-8-azabicyclo[3.2.1]octane-8-carbonyl]pyridin-2-yl]piperazin-1-yl]methyl]piperidin-1-yl]inden-2-yl]piperidine-2,6-dione	O=C1CCC(C2C(=O)C3=CC=CC(N4CCC(CN5CCN(C6=CC=C(C(=O)N7[C@@H]8CC[C@H]7C[C@@H](OC7=NN9C(=NN=C9C(F)(F)F)C=C7)C8)C=N6)CC5)CC4)=C3C2=O)C(=O)N1	C43H45F3N10O6	AR	P10275	CRBN	EP-4023649-A1
TPD-KMNKMG	SCHEMBL24592219	4-[2-[1-[1-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]acetyl]piperidin-4-yl]piperidin-4-yl]ethynyl]-N-[2,2,4,4-tetramethyl-3-[[3-(trifluoromethyl)-7,8-dihydro-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]oxy]cyclobutyl]benzamide; SCHEMBL24592337	CC1(C)[C@H](NC(=O)C2=CC=C(C#CC3CCN(C4CCN(C(=O)CNC5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)CC4)CC3)C=C2)C(C)(C)[C@H]1OC1=NN2C(=NN=C2C(F)(F)F)CC1	C48H53F3N10O7	AR	P10275	CRBN	EP-4023649-A1
TPD-SEHKPQ	EP4023649A1_53	(2S,4S)-1-[(2S)-3,3-dimethyl-2-[[2-[4-[4-[[2,2,4,4-tetramethyl-3-[[3-(trifluoromethyl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]oxy]cyclobutyl]carbamoyl]phenoxy]butoxy]acetyl]amino]butanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCOC3=CC=C(C(=O)NC4C(C)(C)C(OC5=NN6C(=NN=C6C(F)(F)F)C=C5)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C49H60F3N9O8S	AR	P10275	VHL	EP-4023649-A1
TPD-2ZMH91	SCHEMBL24514304	2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-N-[2-[2-[2-[4-[(Z)-1-(4-hydroxyphenyl)-2-phenylbut-1-enyl]phenoxy]ethyl-methylamino]-2-oxoethoxy]ethyl]acetamide	CC/C(=C(\c1ccc(O)cc1)c1ccc(OCCN(C)C(=O)COCCNC(=O)Cc2ccc3c(c2)CN(C2CCC(=O)NC2=O)C3=O)cc1)c1ccccc1	C44H46N4O8	PKCβ1	P05771	CRBN	US-20240058318-A1
TPD-L94VZM	SCHEMBL24514318	3-[2-[[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]acetyl]amino]ethoxy]-N-[2-[4-[(Z)-1-(4-hydroxyphenyl)-2-phenylbut-1-enyl]phenoxy]ethyl]-N-methylpropanamide	CC/C(=C(\c1ccc(O)cc1)c1ccc(OCCN(C)C(=O)CCOCCNC(=O)Cc2ccc3c(c2)CN(C2CCC(=O)NC2=O)C3=O)cc1)c1ccccc1	C45H48N4O8	PKCβ1	P05771	CRBN	US-20240058318-A1
TPD-V4F0SE	SCHEMBL24514406	2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-N-[2-[2-[2-[2-[4-[(Z)-1-(4-hydroxyphenyl)-2-phenylbut-1-enyl]phenoxy]ethylamino]ethoxy]ethoxy]ethyl]acetamide	CC/C(=C(\c1ccc(O)cc1)c1ccc(OCCNCCOCCOCCNC(=O)Cc2ccc3c(c2)CN(C2CCC(=O)NC2=O)C3=O)cc1)c1ccccc1	C45H50N4O8	PKCβ1	P05771	CRBN	US-20240058318-A1
TPD-N6TIKA	SCHEMBL24514319	2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-N-[2-[2-[2-[2-[4-[(Z)-1-(4-hydroxyphenyl)-2-phenylbut-1-enyl]phenoxy]ethyl-methylamino]-2-oxoethoxy]ethoxy]ethyl]acetamide	CC/C(=C(\c1ccc(O)cc1)c1ccc(OCCN(C)C(=O)COCCOCCNC(=O)Cc2ccc3c(c2)CN(C2CCC(=O)NC2=O)C3=O)cc1)c1ccccc1	C46H50N4O9	PKCβ1	P05771	CRBN	US-20240058318-A1
TPD-HUUJFY	SCHEMBL24514376	2-(2,6-dioxopiperidin-3-yl)-N-[2-[2-[2-[2-[4-[(Z)-1-(4-hydroxyphenyl)-2-phenylbut-1-enyl]phenoxy]ethyl-methylamino]-2-oxoethoxy]ethoxy]ethyl]-1-oxo-3H-isoindole-5-carboxamide	CC/C(=C(\c1ccc(O)cc1)c1ccc(OCCN(C)C(=O)COCCOCCNC(=O)c2ccc3c(c2)CN(C2CCC(=O)NC2=O)C3=O)cc1)c1ccccc1	C45H48N4O9	PKCβ1	P05771	CRBN	US-20240058318-A1
TPD-S0M8ES	SCHEMBL24514427	2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-N-[2-[2-[2-[2-[4-[(Z)-1-(4-hydroxyphenyl)-2-phenylbut-1-enyl]phenoxy]ethyl-methylamino]-2-oxoethoxy]ethoxy]ethyl]-N-methylacetamide	CC/C(=C(\c1ccc(O)cc1)c1ccc(OCCN(C)C(=O)COCCOCCN(C)C(=O)Cc2ccc3c(c2)CN(C2CCC(=O)NC2=O)C3=O)cc1)c1ccccc1	C47H52N4O9	PKCβ1	P05771	CRBN	US-20240058318-A1
TPD-OF4WM5	SCHEMBL24514426	2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-N-[2-[2-[(2R)-2-[2-[4-[(Z)-1-(4-hydroxyphenyl)-2-phenylbut-1-enyl]phenoxy]ethylamino]propoxy]ethoxy]ethyl]acetamide	CC/C(=C(\c1ccc(O)cc1)c1ccc(OCCN[C@H](C)COCCOCCNC(=O)Cc2ccc3c(c2)CN(C2CCC(=O)NC2=O)C3=O)cc1)c1ccccc1	C46H52N4O8	PKCβ1	P05771	CRBN	US-20240058318-A1
TPD-FIPIDC	SCHEMBL24514283	2-[2-[(3R)-1-[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]acetyl]pyrrolidin-3-yl]oxyethoxy]-N-[2-[4-[(Z)-1-(4-hydroxyphenyl)-2-phenylbut-1-enyl]phenoxy]ethyl]-N-methylacetamide	CC/C(=C(\c1ccc(O)cc1)c1ccc(OCCN(C)C(=O)COCCO[C@@H]2CCN(C(=O)Cc3ccc4c(c3)CN(C3CCC(=O)NC3=O)C4=O)C2)cc1)c1ccccc1	C48H52N4O9	PKCβ1	P05771	CRBN	US-20240058318-A1
TPD-KHHAEQ	SCHEMBL24514309	tert-butyl [3-[6-[2-[2-[2-[2-[2-[4-[(Z)-1-(4-hydroxyphenyl)-2-phenylbut-1-enyl]phenoxy]ethyl-methylamino]-2-oxoethoxy]ethoxy]ethylamino]-2-oxoethyl]-3-oxo-1H-isoindol-2-yl]-2,6-dioxopiperidin-1-yl]methyl carbonate	CC/C(=C(\c1ccc(O)cc1)c1ccc(OCCN(C)C(=O)COCCOCCNC(=O)Cc2ccc3c(c2)CN(C2CCC(=O)N(COC(=O)OC(C)(C)C)C2=O)C3=O)cc1)c1ccccc1	C52H60N4O12	PKCβ1	P05771	CRBN	US-20240058318-A1
TPD-PXI0O5	SCHEMBL24514310	tert-butyl [3-[6-[2-[2-[2-[2-[2-[4-[(Z)-1-(4-hydroxyphenyl)-2-phenylbut-1-enyl]phenoxy]ethyl-methylamino]-2-oxoethoxy]ethoxy]ethyl-methylamino]-2-oxoethyl]-3-oxo-1H-isoindol-2-yl]-2,6-dioxopiperidin-1-yl]methyl carbonate	CC/C(=C(\c1ccc(O)cc1)c1ccc(OCCN(C)C(=O)COCCOCCN(C)C(=O)Cc2ccc3c(c2)CN(C2CCC(=O)N(COC(=O)OC(C)(C)C)C2=O)C3=O)cc1)c1ccccc1	C53H62N4O12	PKCβ1	P05771	CRBN	US-20240058318-A1
TPD-7QO8AQ	US20240058318A1_Analogs1	.	CC/C(=C(/c1ccc(O)cc1)c1ccc(OCCN(C)C(=O)COCCOCCN(C)C(=O)Cc2ccc3c(c2)CN([C@@H]2CCC(=O)NC2=O)C3=O)cc1)c1ccccc1	C47H52N4O9	PKCβ1	P05771	CRBN	US-20240058318-A1
TPD-7VSJIU	US20240058318A1_Analogs2	.	CC/C(=C(/c1ccc(O)cc1)c1ccc(OCCN[C@H](C)COCCOCCNC(=O)Cc2ccc3c(c2)CN([C@@H]2CCC(=O)NC2=O)C3=O)cc1)c1ccccc1	C46H52N4O8	PKCβ1	P05771	CRBN	US-20240058318-A1
TPD-23NHMX	US20240058318A1_Analogs3	.	CC/C(=C(/c1ccc(O)cc1)c1ccc(OCCNCCOCCOCCNC(=O)Cc2ccc3c(c2)CN([C@@H]2CCC(=O)NC2=O)C3=O)cc1)c1ccccc1	C45H50N4O8	PKCβ1	P05771	CRBN	US-20240058318-A1
TPD-FLRR65	US20240058318A1_Analogs4	.	CC/C(=C(/c1ccc(O)cc1)c1ccc(OCCN(C)C(=O)COCCO[C@@H]2CCN(C(=O)Cc3ccc4c(c3)CN([C@@H]3CCC(=O)NC3=O)C4=O)C2)cc1)c1ccccc1	C48H52N4O9	PKCβ1	P05771	CRBN	US-20240058318-A1
TPD-CZM572	US20240058318A1_Analogs5	.	CC/C(=C(/c1ccc(O)cc1)c1ccc(OCCN(C)C(=O)COCCOCCNC(=O)Cc2ccc3c(c2)CN([C@@H]2CCC(=O)N(COC(=O)OC(C)(C)C)C2=O)C3=O)cc1)c1ccccc1	C52H60N4O12	PKCβ1	P05771	CRBN	US-20240058318-A1
TPD-PQD80Y	US20240058318A1_Analogs6	.	CC/C(=C(/c1ccc(O)cc1)c1ccc(OCCN(C)C(=O)COCCOCCN(C)C(=O)Cc2ccc3c(c2)CN([C@@H]2CCC(=O)N(COC(=O)OC(C)(C)C)C2=O)C3=O)cc1)c1ccccc1	C53H62N4O12	PKCβ1	P05771	CRBN	US-20240058318-A1
TPD-L0TK6E	NSC833480	2-(2,6-dioxopiperidin-3-yl)-N-[2-[2-[2-[4-[(Z)-1-(4-hydroxyphenyl)-2-phenylbut-1-enyl]phenoxy]ethyl-methylamino]-2-oxoethoxy]ethyl]-1-oxo-3H-isoindole-4-carboxamide; NSC-833480	CC/C(=C(\c1ccc(O)cc1)c1ccc(OCCN(C)C(=O)COCCNC(=O)c2cccc3c2CN(C2CCC(=O)NC2=O)C3=O)cc1)c1ccccc1	C43H44N4O8	PKCβ1	P05771	CRBN	US-20240058318-A1
TPD-38QAAN	US20240058318A1_TC-Pr-002	.	CC/C(=C(\c1ccc(O)cc1)c1ccc(OCCN(C)C(=O)CCOCCNC(=O)c2cccc3c2CN(C2CCC(=O)NC2=O)C3=O)cc1)c1ccccc1	C44H46N4O8	PKCβ1	P05771	CRBN	US-20240058318-A1
TPD-883S5A	NSC833488	2-(2,6-dioxopiperidin-3-yl)-N-[2-[2-[2-[2-[4-[(Z)-1-(4-hydroxyphenyl)-2-phenylbut-1-enyl]phenoxy]ethyl-methylamino]-2-oxoethoxy]ethoxy]ethyl]-1-oxo-3H-isoindole-4-carboxamide; NSC-833488	CC/C(=C(\c1ccc(O)cc1)c1ccc(OCCN(C)C(=O)COCCOCCNC(=O)c2cccc3c2CN(C2CCC(=O)NC2=O)C3=O)cc1)c1ccccc1	C45H48N4O9	PKCβ1	P05771	CRBN	US-20240058318-A1
TPD-Z0KF9Z	US20240058318A1_TC-Pr-004	.	CC/C(=C(\c1ccc(O)cc1)c1ccc(OCCN(C)C(=O)COCCNC(=O)c2ccc3c(c2)CN(C2CCC(=O)NC2=O)C3=O)cc1)c1ccccc1	C43H44N4O8	PKCβ1	P05771	CRBN	US-20240058318-A1
TPD-N07DGJ	US20240058318A1_TC-Pr-005	.	CC/C(=C(\c1ccc(O)cc1)c1ccc(OCCN(C)C(=O)CCOCCNC(=O)c2ccc3c(c2)CN(C2CCC(=O)NC2=O)C3=O)cc1)c1ccccc1	C44H46N4O8	PKCβ1	P05771	CRBN	US-20240058318-A1
TPD-B8LKUW	US20240058318A1_TC-Pr-008	.	CC/C(=C(\c1ccc(O)cc1)c1ccc(OCCN(C)C(=O)CCOCCNC(=O)Cc2ccc3c(c2)CN([C@H]2CCC(=O)NC2=O)C3=O)cc1)c1ccccc1	C45H48N4O8	PKCβ1	P05771	CRBN	US-20240058318-A1
TPD-1V6CR1	US20240058318A1_TC-Pr-009	.	CC/C(=C(\c1ccc(O)cc1)c1ccc(OCCN(C)C(=O)COCCOCCNC(=O)Cc2ccc3c(c2)CN([C@H]2CCC(=O)NC2=O)C3=O)cc1)c1ccccc1	C46H50N4O9	PKCβ1	P05771	CRBN	US-20240058318-A1
TPD-MF2GJ9	SCHEMBL24598087	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[5-methyl-6-[(6-methylpyridin-2-yl)carbamoyl]pyridin-3-yl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31030008	CC1=NC(NC(=O)C2=C(C)C=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=N2)=CC=C1	C45H50N12O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-4VNR4X	SCHEMBL24598541	8-[4-[2-[4-(2,6-dioxopiperidin-3-yl)-3,5-difluorophenyl]ethyl]piperazin-1-yl]-2-[5-methyl-6-[(6-methylpyridin-2-yl)carbamoyl]pyridin-3-yl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31030004	CC1=NC(NC(=O)C2=C(C)C=C(C3=NN4CCC5=C(C=CC(N6CCN(CCC7=CC(F)=C(C8CCC(=O)NC8=O)C(F)=C7)CC6)=C5)NC4=C3C(N)=O)C=N2)=CC=C1	C42H42F2N10O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-WIYGP6	SCHEMBL24598282	8-[4-[3-[4-[(3R)-2,6-dioxopiperidin-3-yl]phenyl]cyclobutyl]piperazin-1-yl]-2-[5-methyl-6-[(6-methylpyridin-2-yl)carbamoyl]pyridin-3-yl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31030041	CC1=NC(NC(=O)C2=C(C)C=C(C3=NN4CCC5=C(C=CC(N6CCN(C7CC(C8=CC=C([C@H]9CCC(=O)NC9=O)C=C8)C7)CC6)=C5)NC4=C3C(N)=O)C=N2)=CC=C1	C44H46N10O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-6PYZZL	SCHEMBL31030012	8-[4-[3-[4-[(3S)-2,6-dioxopiperidin-3-yl]phenyl]cyclobutyl]piperazin-1-yl]-2-[5-methyl-6-[(6-methylpyridin-2-yl)carbamoyl]pyridin-3-yl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	CC1=NC(NC(=O)C2=C(C)C=C(C3=NN4CCC5=C(C=CC(N6CCN(C7CC(C8=CC=C([C@@H]9CCC(=O)NC9=O)C=C8)C7)CC6)=C5)NC4=C3C(N)=O)C=N2)=CC=C1	C44H46N10O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-FW64P4	SCHEMBL24598077	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[4-methyl-5-[(6-methylpyridin-2-yl)carbamoyl]pyridin-2-yl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31029968	CC1=NC(NC(=O)C2=C(C)C=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)N=C2)=CC=C1	C45H50N12O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-8C66Y6	SCHEMBL24598380	8-[4-[2-[4-(2,6-dioxopiperidin-3-yl)-3,5-difluorophenyl]ethyl]piperazin-1-yl]-2-[4-methyl-5-[(6-methylpyridin-2-yl)carbamoyl]pyridin-2-yl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31030026	CC1=NC(NC(=O)C2=C(C)C=C(C3=NN4CCC5=C(C=CC(N6CCN(CCC7=CC(F)=C(C8CCC(=O)NC8=O)C(F)=C7)CC6)=C5)NC4=C3C(N)=O)N=C2)=CC=C1	C42H42F2N10O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-W7JTC1	SCHEMBL24598079	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[6-methyl-5-[(6-methylpyridin-2-yl)carbamoyl]pyridin-2-yl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31029987	CC1=NC(NC(=O)C2=CC=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)N=C2C)=CC=C1	C45H50N12O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-BH2BH9	SCHEMBL24598083	8-[4-[2-[4-(2,6-dioxopiperidin-3-yl)-3,5-difluorophenyl]ethyl]piperazin-1-yl]-2-[6-methyl-5-[(6-methylpyridin-2-yl)carbamoyl]pyridin-2-yl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31030022	CC1=NC(NC(=O)C2=CC=C(C3=NN4CCC5=C(C=CC(N6CCN(CCC7=CC(F)=C(C8CCC(=O)NC8=O)C(F)=C7)CC6)=C5)NC4=C3C(N)=O)N=C2C)=CC=C1	C42H42F2N10O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-M0VNUB	SCHEMBL24598082	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[2-fluoro-3-methyl-4-[(6-methylpyrazin-2-yl)carbamoyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31030079	CC1=NC(NC(=O)C2=C(C)C(F)=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2)=CN=C1	C45H49FN12O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-LM9LFQ	SCHEMBL24598153	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[4-[(6-ethylpyridin-2-yl)carbamoyl]-2-fluoro-3-methylphenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31030013	CCC1=NC(NC(=O)C2=C(C)C(F)=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2)=CC=C1	C47H52FN11O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-EQKVLT	SCHEMBL24598108	8-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazine-1-carbonyl]-2-(4-phenoxyphenyl)-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	NC(=O)C1=C2NC3=C(C=C(C(=O)N4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C=C3)CCN2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C48H47N9O7	BTK	Q06187	CRBN	US-20240246977-A1
TPD-DC8LIT	SCHEMBL24598131	2-[4-[(4-chloro-6-methylpyridin-2-yl)carbamoyl]-2-fluoro-3-methylphenyl]-8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31029965	CC1=NC(NC(=O)C2=C(C)C(F)=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2)=CC(Cl)=C1	C46H49ClFN11O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-60X0NB	SCHEMBL24598533	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[2-fluoro-3-methyl-4-[(4-methylpyrimidin-2-yl)carbamoyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	CC1=NC(NC(=O)C2=C(C)C(F)=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2)=NC=C1	C45H49FN12O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-4YOC6F	SCHEMBL24598133	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[2-fluoro-4-[(5-fluoro-6-methylpyridin-2-yl)carbamoyl]-3-methylphenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	CC1=NC(NC(=O)C2=CC=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C(F)=C2C)=CC=C1F	C46H49F2N11O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-9Z79WK	SCHEMBL24598137	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[2-fluoro-3-methyl-4-(1H-pyrrolo[3,2-b]pyridin-5-ylcarbamoyl)phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	CC1=C(C(=O)NC2=CC=C3NC=CC3=N2)C=CC(C2=NN3CCC4=C(C=CC(N5CCN(CC6CCN(C7=CC=C(N8CCC(=O)NC8=O)C=C7)CC6)CC5)=C4)NC3=C2C(N)=O)=C1F	C47H49FN12O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-KL7Y1I	SCHEMBL24598136	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[2-fluoro-3-methyl-4-(3-pyridin-2-yl-1,2,4-oxadiazol-5-yl)phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31030051	CC1=C(C2=NC(C3=CC=CC=N3)=NO2)C=CC(C2=NN3CCC4=C(C=CC(N5CCN(CC6CCN(C7=CC=C(N8CCC(=O)NC8=O)C=C7)CC6)CC5)=C4)NC3=C2C(N)=O)=C1F	C46H47FN12O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-U9YKZI	SCHEMBL24598140	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[2-fluoro-3-methyl-4-(quinoxalin-2-ylcarbamoyl)phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31030035	CC1=C(C(=O)NC2=CN=C3C=CC=CC3=N2)C=CC(C2=NN3CCC4=C(C=CC(N5CCN(CC6CCN(C7=CC=C(N8CCC(=O)NC8=O)C=C7)CC6)CC5)=C4)NC3=C2C(N)=O)=C1F	C48H49FN12O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-K6VL61	SCHEMBL24598135	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[2-fluoro-3-methyl-4-[(6-phenylpyridin-2-yl)carbamoyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31030033	CC1=C(C(=O)NC2=CC=CC(C3=CC=CC=C3)=N2)C=CC(C2=NN3CCC4=C(C=CC(N5CCN(CC6CCN(C7=CC=C(N8CCC(=O)NC8=O)C=C7)CC6)CC5)=C4)NC3=C2C(N)=O)=C1F	C51H52FN11O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-K0YOI4	SCHEMBL24598156	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[2-fluoro-3-methyl-4-[(4-pyrrolidin-1-ylpyridin-2-yl)carbamoyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31030005	CC1=C(C(=O)NC2=CC(N3CCCC3)=CC=N2)C=CC(C2=NN3CCC4=C(C=CC(N5CCN(CC6CCN(C7=CC=C(N8CCC(=O)NC8=O)C=C7)CC6)CC5)=C4)NC3=C2C(N)=O)=C1F	C49H55FN12O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-CS1E8E	SCHEMBL24598143	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[2-fluoro-4-[(4-methoxypyridin-2-yl)carbamoyl]-3-methylphenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31029971	COC1=CC=NC(NC(=O)C2=C(C)C(F)=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2)=C1	C46H50FN11O5	BTK	Q06187	CRBN	US-20240246977-A1
TPD-QDXBTT	SCHEMBL24598139	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[4-[(4-ethoxypyridin-2-yl)carbamoyl]-2-fluoro-3-methylphenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31029953	CCOC1=CC=NC(NC(=O)C2=C(C)C(F)=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2)=C1	C47H52FN11O5	BTK	Q06187	CRBN	US-20240246977-A1
TPD-ZW3YZD	SCHEMBL24598060	8-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidine-1-carbonyl]-2-(4-phenoxyphenyl)-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31029973	NC(=O)C1=C2NC3=C(C=C(C(=O)N4CCC(CN5CCN(C6=CC7=C(C=C6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)C=C3)CCN2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C48H46FN9O7	BTK	Q06187	CRBN	US-20240246977-A1
TPD-7J392T	SCHEMBL24598138	2-[4-[(5-chloro-6-methylpyridin-2-yl)carbamoyl]-2-fluoro-3-methylphenyl]-8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	CC1=NC(NC(=O)C2=CC=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C(F)=C2C)=CC=C1Cl	C46H49ClFN11O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-TTSDSU	SCHEMBL24598132	2-[4-[(5-chloro-6-methylpyridin-2-yl)carbamoyl]-2-fluoro-3-methylphenyl]-8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]azetidin-3-yl]methyl]piperazin-1-yl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31030030	CC1=C(Cl)C=CC(NC(=O)C2=C(C)C(F)=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)C7)CC6)=C5)NC4=C3C(N)=O)C=C2)=N1	C44H45ClFN11O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-12FBZX	SCHEMBL24598499	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)-3-methylphenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[2-fluoro-3-methyl-4-[(6-methylpyridin-2-yl)carbamoyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	CC1=CC(N2CCC(CN3CCN(C4=CC5=C(C=C4)NC4=C(C(N)=O)C(C6=C(F)C(C)=C(C(=O)NC7=CC=CC(C)=N7)C=C6)=NN4CC5)CC3)CC2)=CC=C1N1CCC(=O)NC1=O	C47H52FN11O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-82L0V4	SCHEMBL24598090	8-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[2-fluoro-3-methyl-4-[(6-methylpyridin-2-yl)carbamoyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	CC1=CC=CC(NC(=O)C2=C(C)C(F)=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=C(F)C=C9C(=O)N(C%10CCC(=O)NC%10=O)C(=O)C9=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2)=N1	C49H49F2N11O6	BTK	Q06187	CRBN	US-20240246977-A1
TPD-420W5X	SCHEMBL24598092	8-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-3-oxo-1H-isoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[2-fluoro-3-methyl-4-[(6-methylpyridin-2-yl)carbamoyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	CC1=CC=CC(NC(=O)C2=C(C)C(F)=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=C(F)C=C9CN(C%10CCC(=O)NC%10=O)C(=O)C9=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2)=N1	C49H51F2N11O5	BTK	Q06187	CRBN	US-20240246977-A1
TPD-XT4S7I	SCHEMBL24598393	8-[4-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]azetidin-3-yl]piperazin-1-yl]-2-[2-fluoro-3-methyl-4-[(6-methylpyridin-2-yl)carbamoyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31030009	CC1=CC=CC(NC(=O)C2=C(C)C(F)=C(C3=NN4CCC5=C(C=CC(N6CCN(C7CN(C8CN(C9=CC%10=C(C=C9)C(=O)N(C9CCC(=O)NC9=O)C%10=O)C8)C7)CC6)=C5)NC4=C3C(N)=O)C=C2)=N1	C49H49FN12O6	BTK	Q06187	CRBN	US-20240246977-A1
TPD-Z6AZHG	SCHEMBL24598097	8-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[2-fluoro-3-methyl-4-[(6-methylpyridin-2-yl)carbamoyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	CC1=CC=CC(NC(=O)C2=C(C)C(F)=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C9C(=O)N(C%10CCC(=O)NC%10=O)CC9=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2)=N1	C49H52FN11O5	BTK	Q06187	CRBN	US-20240246977-A1
TPD-WD0TNT	SCHEMBL24598096	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]azetidin-3-yl]methyl]piperazin-1-yl]-2-[2-fluoro-3-methyl-4-[(6-methylpyridin-2-yl)carbamoyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31029977	CC1=NC(NC(=O)C2=C(C)C(F)=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)C7)CC6)=C5)NC4=C3C(N)=O)C=C2)=CC=C1	C44H46FN11O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-9YW6W8	SCHEMBL24598095	8-[4-[[1-(2,6-dioxopiperidin-3-yl)-3,3-dimethyl-2-oxoindol-5-yl]methyl]piperazin-1-yl]-2-[2-fluoro-3-methyl-4-[(6-methylpyridin-2-yl)carbamoyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	CC1=CC=CC(NC(=O)C2=C(C)C(F)=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7=CC=C8C(=C7)C(C)(C)C(=O)N8C7CCC(=O)NC7=O)CC6)=C5)NC4=C3C(N)=O)C=C2)=N1	C46H47FN10O5	BTK	Q06187	CRBN	US-20240246977-A1
TPD-Y6HVAL	US20240246977A1_129B59	.	CC1=NC(NC(=O)C2=C(C)C(F)=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7=CC=C8C(=C7)OC(=O)N8C7CCC(=O)NC7=O)CC6)=C5)NC4=C3C(N)=O)C=C2)=CC=C1	C43H41FN10O6	BTK	Q06187	CRBN	US-20240246977-A1
TPD-K89O95	SCHEMBL24598056	8-N-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]-2-(4-phenoxyphenyl)-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1,8-dicarboxamide; SCHEMBL29710534	NC(=O)C1=C2NC3=C(C=C(C(=O)NC4CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)CCN2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C43H38N8O7	BTK	Q06187	CRBN	US-20240246977-A1
TPD-P5OJ6K	SCHEMBL24598098	8-[4-[2-[4-(2,6-dioxopiperidin-3-yl)-3,5-difluorophenyl]ethyl]piperazin-1-yl]-2-[2-fluoro-3-methyl-4-[(6-methylpyridin-2-yl)carbamoyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	CC1=CC=CC(NC(=O)C2=C(C)C(F)=C(C3=NN4CCC5=C(C=CC(N6CCN(CCC7=CC(F)=C(C8CCC(=O)NC8=O)C(F)=C7)CC6)=C5)NC4=C3C(N)=O)C=C2)=N1	C43H42F3N9O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-SBD5EF	SCHEMBL24598091	8-[4-[2-[4-[(3R)-2,6-dioxopiperidin-3-yl]-3,5-difluorophenyl]ethyl]piperazin-1-yl]-2-[2-fluoro-3-methyl-4-[(6-methylpyridin-2-yl)carbamoyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	CC1=NC(NC(=O)C2=C(C)C(F)=C(C3=NN4CCC5=C(C=CC(N6CCN(CCC7=CC(F)=C([C@H]8CCC(=O)NC8=O)C(F)=C7)CC6)=C5)NC4=C3C(N)=O)C=C2)=CC=C1	C43H42F3N9O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-SL9PU9	SCHEMBL24598093	8-[4-[3-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]cyclobutyl]piperazin-1-yl]-2-[2-fluoro-3-methyl-4-[(6-methylpyridin-2-yl)carbamoyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	CC1=CC=CC(NC(=O)C2=C(C)C(F)=C(C3=NN4CCC5=C(C=CC(N6CCN(C7CC(C8=CC=C(N9CCC(=O)NC9=O)C=C8)C7)CC6)=C5)NC4=C3C(N)=O)C=C2)=N1	C44H45FN10O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-AZ96AL	SCHEMBL24598099	8-[4-[1-[1-[4-(2,6-dioxopiperidin-3-yl)phenyl]azetidin-3-yl]azetidin-3-yl]piperazin-1-yl]-2-[2-fluoro-3-methyl-4-[(6-methylpyridin-2-yl)carbamoyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	CC1=CC=CC(NC(=O)C2=C(C)C(F)=C(C3=NN4CCC5=C(C=CC(N6CCN(C7CN(C8CN(C9=CC=C(C%10CCC(=O)NC%10=O)C=C9)C8)C7)CC6)=C5)NC4=C3C(N)=O)C=C2)=N1	C47H50FN11O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-SBJC3J	SCHEMBL24598101	8-[4-[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]azetidin-3-yl]piperazin-1-yl]-2-[2-fluoro-3-methyl-4-[(6-methylpyridin-2-yl)carbamoyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	CC1=CC=CC(NC(=O)C2=C(C)C(F)=C(C3=NN4CCC5=C(C=CC(N6CCN(C7CN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)C7)CC6)=C5)NC4=C3C(N)=O)C=C2)=N1	C43H44FN11O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-IQJIY5	SCHEMBL24598245	8-[4-[3-[4-[(3R)-2,6-dioxopiperidin-3-yl]phenyl]cyclobutyl]piperazin-1-yl]-2-[2-fluoro-3-methyl-4-[(6-methylpyridin-2-yl)carbamoyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	CC1=CC=CC(NC(=O)C2=C(C)C(F)=C(C3=NN4CCC5=C(C=CC(N6CCN(C7CC(C8=CC=C([C@H]9CCC(=O)NC9=O)C=C8)C7)CC6)=C5)NC4=C3C(N)=O)C=C2)=N1	C45H46FN9O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-F5AQKT	SCHEMBL24598100	8-[4-[3-[4-[(3S)-2,6-dioxopiperidin-3-yl]phenyl]cyclobutyl]piperazin-1-yl]-2-[2-fluoro-3-methyl-4-[(6-methylpyridin-2-yl)carbamoyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	CC1=CC=CC(NC(=O)C2=C(C)C(F)=C(C3=NN4CCC5=C(C=CC(N6CCN(C7CC(C8=CC=C([C@@H]9CCC(=O)NC9=O)C=C8)C7)CC6)=C5)NC4=C3C(N)=O)C=C2)=N1	C45H46FN9O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-PQM8I7	SCHEMBL24598332	8-[4-[[1-[4-[(2,4-dioxo-1,3-diazinan-1-yl)methyl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[2-fluoro-3-methyl-4-[(6-methylpyridin-2-yl)carbamoyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31030064	CC1=NC(NC(=O)C2=C(C)C(F)=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(CN9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2)=CC=C1	C47H52FN11O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-FIWO8Y	SCHEMBL24598094	8-[4-[[1-[3-[(2,4-dioxo-1,3-diazinan-1-yl)methyl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[2-fluoro-3-methyl-4-[(6-methylpyridin-2-yl)carbamoyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31030024	CC1=NC(NC(=O)C2=C(C)C(F)=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=CC(CN9CCC(=O)NC9=O)=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2)=CC=C1	C47H52FN11O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-5HPRWD	SCHEMBL24598058	8-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidine-4-carbonyl]amino]-2-(4-phenoxyphenyl)-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL29710653	NC(=O)C1=C2NC3=C(C=C(NC(=O)C4CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)CCN2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C43H38N8O7	BTK	Q06187	CRBN	US-20240246977-A1
TPD-I9KTY1	SCHEMBL24598036	8-[4-[3-[4-[[(3R)-2,6-dioxopiperidin-3-yl]amino]phenyl]cyclobutyl]piperazin-1-yl]-2-[2-fluoro-3-methyl-4-[(6-methylpyridin-2-yl)carbamoyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31030045	CC1=NC(NC(=O)C2=C(C)C(F)=C(C3=NN4CCC5=C(C=CC(N6CCN(C7CC(C8=CC=C(N[C@@H]9CCC(=O)NC9=O)C=C8)C7)CC6)=C5)NC4=C3C(N)=O)C=C2)=CC=C1	C45H47FN10O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-Z0G65I	SCHEMBL24598040	8-[4-[3-[4-[[(3S)-2,6-dioxopiperidin-3-yl]amino]phenyl]cyclobutyl]piperazin-1-yl]-2-[2-fluoro-3-methyl-4-[(6-methylpyridin-2-yl)carbamoyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31030011	CC1=NC(NC(=O)C2=C(C)C(F)=C(C3=NN4CCC5=C(C=CC(N6CCN(C7CC(C8=CC=C(N[C@H]9CCC(=O)NC9=O)C=C8)C7)CC6)=C5)NC4=C3C(N)=O)C=C2)=CC=C1	C45H47FN10O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-1E53JD	SCHEMBL24598037	8-[4-[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidine-4-carbonyl]piperazin-1-yl]-2-[2-fluoro-3-methyl-4-[(6-methylpyridin-2-yl)carbamoyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31030039	CC1=NC(NC(=O)C2=C(C)C(F)=C(C3=NN4CCC5=C(C=CC(N6CCN(C(=O)C7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2)=CC=C1	C46H48FN11O5	BTK	Q06187	CRBN	US-20240246977-A1
TPD-EYNJXB	SCHEMBL24598039	8-[4-[[(3R)-1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]pyrrolidin-3-yl]methyl]piperazin-1-yl]-2-[2-fluoro-3-methyl-4-[(6-methylpyridin-2-yl)carbamoyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31030071	CC1=NC(NC(=O)C2=C(C)C(F)=C(C3=NN4CCC5=C(C=CC(N6CCN(C[C@H]7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)C7)CC6)=C5)NC4=C3C(N)=O)C=C2)=CC=C1	C45H48FN11O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-G33PHC	SCHEMBL24598045	8-[4-[2-[3-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]acetyl]piperazin-1-yl]-2-[2-fluoro-3-methyl-4-[(6-methylpyridin-2-yl)carbamoyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31029978	CC1=NC(NC(=O)C2=C(C)C(F)=C(C3=NN4CCC5=C(C=CC(N6CCN(C(=O)CC7=CC(N8CCC(=O)NC8=O)=CC=C7)CC6)=C5)NC4=C3C(N)=O)C=C2)=CC=C1	C42H41FN10O5	BTK	Q06187	CRBN	US-20240246977-A1
TPD-92MVC8	SCHEMBL24598347	tert-butyl 2-[3-[4-[4-[[4-[1-carbamoyl-2-[2-fluoro-3-methyl-4-[(6-methylpyridin-2-yl)carbamoyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepin-8-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]-2,6-dioxo-1,3-diazinan-1-yl]acetate; SCHEMBL31029986	CC1=NC(NC(=O)C2=C(C)C(F)=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)N(CC(=O)OC(C)(C)C)C9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2)=CC=C1	C52H60FN11O6	BTK	Q06187	CRBN	US-20240246977-A1
TPD-25X57G	benzyl 2-[3-[4-[4-[[4-[1-carbamoyl-2-[2-fluoro-3-methyl-4-[(6-methylpyridin-2-yl)carbamoyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepin-8-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]-2,6-dioxo-1,3-diazinan-1-yl]acetate	SCHEMBL31030043	CC1=NC(NC(=O)C2=C(C)C(F)=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)N(CC(=O)OCC%10=CC=CC=C%10)C9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2)=CC=C1	C55H58FN11O6	BTK	Q06187	CRBN	US-20240246977-A1
TPD-7VRDJG	SCHEMBL24598349	[3-[4-[4-[[4-[1-carbamoyl-2-[2-fluoro-3-methyl-4-[(6-methylpyridin-2-yl)carbamoyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepin-8-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]-2,6-dioxo-1,3-diazinan-1-yl]methyl 2,2-dimethylpropanoate; SCHEMBL31029990	CC1=NC(NC(=O)C2=C(C)C(F)=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)N(COC(=O)C(C)(C)C)C9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2)=CC=C1	C52H60FN11O6	BTK	Q06187	CRBN	US-20240246977-A1
TPD-27TCG0	US20240246977A1_149B79	tert-butyl 2-[3-[4-[4-[[4-[1-carbamoyl-2-[2-fluoro-3-methyl-4-[[2-[(2-methylpropan-2-yl)oxy]-2-oxoethyl]-(6-methylpyridin-2-yl)carbamoyl]phenyl]-6,11-dihydro-5H-pyrazolo[1,5-c][3]benzazepin-8-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]-2,6-dioxo-1,3-diazinan-1-yl]acetate	CC1=NC(N(CC(=O)OC(C)(C)C)C(=O)C2=C(C)C(F)=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)N(CC(=O)OC(C)(C)C)C9=O)C=C8)CC7)CC6)=C5)CC4=C3C(N)=O)C=C2)=CC=C1	C59H71FN10O8	BTK	Q06187	CRBN	US-20240246977-A1
TPD-89IG33	SCHEMBL24598070	8-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperidine-4-carbonyl]amino]-2-(4-phenoxyphenyl)-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL29710565	NC(=O)C1=C2NC3=C(C=C(NC(=O)C4CCN(C5=CC=CC6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)CCN2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C43H38N8O7	BTK	Q06187	CRBN	US-20240246977-A1
TPD-1BTTZP	benzyl 2-[3-[4-[4-[[4-[1-carbamoyl-2-[2-fluoro-3-methyl-4-[(6-methylpyridin-2-yl)-(2-oxo-2-phenylmethoxyethyl)carbamoyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepin-8-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]-2,6-dioxo-1,3-diazinan-1-yl]acetate	SCHEMBL24598352; SCHEMBL31029983	CC1=NC(N(CC(=O)OCC2=CC=CC=C2)C(=O)C2=C(C)C(F)=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)N(CC(=O)OCC%10=CC=CC=C%10)C9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2)=CC=C1	C64H66FN11O8	BTK	Q06187	CRBN	US-20240246977-A1
TPD-AFZGWI	SCHEMBL24598389	[3-[4-[4-[[4-[1-carbamoyl-2-[4-[2,2-dimethylpropanoyloxymethyl-(6-methylpyridin-2-yl)carbamoyl]-2-fluoro-3-methylphenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepin-8-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]-2,6-dioxo-1,3-diazinan-1-yl]methyl 2,2-dimethylpropanoate; SCHEMBL31029957	CC1=NC(N(COC(=O)C(C)(C)C)C(=O)C2=C(C)C(F)=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)N(COC(=O)C(C)(C)C)C9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2)=CC=C1	C58H70FN11O8	BTK	Q06187	CRBN	US-20240246977-A1
TPD-ACOAUW	SCHEMBL24598038	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[2-fluoro-3-methyl-4-[(1-methylpyrazol-3-yl)carbamoyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	CC1=C(C(=O)NC2=NN(C)C=C2)C=CC(C2=NN3CCC4=C(C=CC(N5CCN(CC6CCN(C7=CC=C(N8CCC(=O)NC8=O)C=C7)CC6)CC5)=C4)NC3=C2C(N)=O)=C1F	C44H49FN12O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-QE7ZW2	SCHEMBL24598041	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[2-fluoro-3-methyl-4-(1,3-thiazol-2-ylcarbamoyl)phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	CC1=C(C(=O)NC2=NC=CS2)C=CC(C2=NN3CCC4=C(C=CC(N5CCN(CC6CCN(C7=CC=C(N8CCC(=O)NC8=O)C=C7)CC6)CC5)=C4)NC3=C2C(N)=O)=C1F	C43H46FN11O4S	BTK	Q06187	CRBN	US-20240246977-A1
TPD-0W7M1N	SCHEMBL24598047	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[2-fluoro-3-methyl-4-[(1-methyl-1,2,4-triazol-3-yl)carbamoyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	CC1=C(C(=O)NC2=NN(C)C=N2)C=CC(C2=NN3CCC4=C(C=CC(N5CCN(CC6CCN(C7=CC=C(N8CCC(=O)NC8=O)C=C7)CC6)CC5)=C4)NC3=C2C(N)=O)=C1F	C43H48FN13O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-ONQLFB	SCHEMBL24598046	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[2-fluoro-3-methyl-4-[[5-(trifluoromethyl)-1H-1,2,4-triazol-3-yl]carbamoyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	CC1=C(C(=O)NC2=NC(C(F)(F)F)=NN2)C=CC(C2=NN3CCC4=C(C=CC(N5CCN(CC6CCN(C7=CC=C(N8CCC(=O)NC8=O)C=C7)CC6)CC5)=C4)NC3=C2C(N)=O)=C1F	C43H45F4N13O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-B30O21	SCHEMBL24598050	2-[4-[(1,5-dimethylpyrazol-3-yl)carbamoyl]-2-fluoro-3-methylphenyl]-8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	CC1=CC(NC(=O)C2=C(C)C(F)=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2)=NN1C	C45H51FN12O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-YH2U1M	SCHEMBL24598043	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[2-fluoro-3-methyl-4-[(1-methylimidazol-4-yl)carbamoyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	CC1=C(C(=O)NC2=CN(C)C=N2)C=CC(C2=NN3CCC4=C(C=CC(N5CCN(CC6CCN(C7=CC=C(N8CCC(=O)NC8=O)C=C7)CC6)CC5)=C4)NC3=C2C(N)=O)=C1F	C44H49FN12O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-G7TCNU	SCHEMBL24598042	8-[4-[2-[4-(2,6-dioxopiperidin-3-yl)-3,5-difluorophenyl]ethyl]piperazin-1-yl]-2-[2-fluoro-3-methyl-4-[(1-methylimidazol-4-yl)carbamoyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	CC1=C(C(=O)NC2=CN(C)C=N2)C=CC(C2=NN3CCC4=C(C=CC(N5CCN(CCC6=CC(F)=C(C7CCC(=O)NC7=O)C(F)=C6)CC5)=C4)NC3=C2C(N)=O)=C1F	C41H41F3N10O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-9H32M1	SCHEMBL24598590	8-[4-[2-[4-[(3R)-2,6-dioxopiperidin-3-yl]-3,5-difluorophenyl]ethyl]piperazin-1-yl]-2-[2-fluoro-3-methyl-4-[(1-methylimidazol-4-yl)carbamoyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	CC1=C(C(=O)NC2=CN(C)C=N2)C=CC(C2=NN3CCC4=C(C=CC(N5CCN(CCC6=CC(F)=C([C@H]7CCC(=O)NC7=O)C(F)=C6)CC5)=C4)NC3=C2C(N)=O)=C1F	C41H41F3N10O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-ARM1UK	SCHEMBL24598063	8-[[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methylamino]-2-(4-phenoxyphenyl)-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	NC(=O)C1=C2NC3=C(C=C(NCC4CCN(C5=C(F)C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)C=C3)CCN2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C43H39FN8O6	BTK	Q06187	CRBN	US-20240246977-A1
TPD-8BSYXG	SCHEMBL24598048	8-[4-[2-[3-(2,6-dioxopiperidin-3-yl)-2-oxo-1,3-benzoxazol-7-yl]ethyl]piperazin-1-yl]-2-[2-fluoro-3-methyl-4-[(1-methylimidazol-4-yl)carbamoyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31030007	CC1=C(C(=O)NC2=CN(C)C=N2)C=CC(C2=NN3CCC4=C(C=CC(N5CCN(CCC6=C7OC(=O)N(C8CCC(=O)NC8=O)C7=CC=C6)CC5)=C4)NC3=C2C(N)=O)=C1F	C42H42FN11O6	BTK	Q06187	CRBN	US-20240246977-A1
TPD-K2DJ6G	SCHEMBL24598051	8-[4-[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidine-4-carbonyl]piperazin-1-yl]-2-[2-fluoro-3-methyl-4-[(1-methylimidazol-4-yl)carbamoyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	CC1=C(C(=O)NC2=CN(C)C=N2)C=CC(C2=NN3CCC4=C(C=CC(N5CCN(C(=O)C6CCN(C7=CC=C(N8CCC(=O)NC8=O)C=C7)CC6)CC5)=C4)NC3=C2C(N)=O)=C1F	C44H47FN12O5	BTK	Q06187	CRBN	US-20240246977-A1
TPD-KG3ROD	SCHEMBL24598044	8-[4-[[(3R)-1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]pyrrolidin-3-yl]methyl]piperazin-1-yl]-2-[2-fluoro-3-methyl-4-[(1-methylimidazol-4-yl)carbamoyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	CC1=C(C(=O)NC2=CN(C)C=N2)C=CC(C2=NN3CCC4=C(C=CC(N5CCN(C[C@H]6CCN(C7=CC=C(N8CCC(=O)NC8=O)C=C7)C6)CC5)=C4)NC3=C2C(N)=O)=C1F	C43H47FN12O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-WDY5N9	SCHEMBL24598161	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[2-fluoro-3-methyl-4-[(2-methyl-1,2,4-triazol-3-yl)carbamoyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	CC1=C(C(=O)NC2=NC=NN2C)C=CC(C2=NN3CCC4=C(C=CC(N5CCN(CC6CCN(C7=CC=C(N8CCC(=O)NC8=O)C=C7)CC6)CC5)=C4)NC3=C2C(N)=O)=C1F	C43H48FN13O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-BGCUTN	SCHEMBL24598165	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[2-fluoro-3-methyl-4-(1,3-thiazol-4-ylcarbamoyl)phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	CC1=C(C(=O)NC2=CSC=N2)C=CC(C2=NN3CCC4=C(C=CC(N5CCN(CC6CCN(C7=CC=C(N8CCC(=O)NC8=O)C=C7)CC6)CC5)=C4)NC3=C2C(N)=O)=C1F	C43H46FN11O4S	BTK	Q06187	CRBN	US-20240246977-A1
TPD-LILPF4	SCHEMBL24598194	8-[4-[2-[4-[(3R)-2,6-dioxopiperidin-3-yl]-3,5-difluorophenyl]ethyl]piperazin-1-yl]-2-[2-fluoro-3-methyl-4-(1,3-thiazol-4-ylcarbamoyl)phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	CC1=C(C(=O)NC2=CSC=N2)C=CC(C2=NN3CCC4=C(C=CC(N5CCN(CCC6=CC(F)=C([C@H]7CCC(=O)NC7=O)C(F)=C6)CC5)=C4)NC3=C2C(N)=O)=C1F	C40H38F3N9O4S	BTK	Q06187	CRBN	US-20240246977-A1
TPD-Y4ODIZ	SCHEMBL24598197	8-[4-[2-[3-(2,6-dioxopiperidin-3-yl)-2-oxo-1,3-benzoxazol-7-yl]ethyl]piperazin-1-yl]-2-[2-fluoro-3-methyl-4-(1,3-thiazol-4-ylcarbamoyl)phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31030073	CC1=C(C(=O)NC2=CSC=N2)C=CC(C2=NN3CCC4=C(C=CC(N5CCN(CCC6=C7OC(=O)N(C8CCC(=O)NC8=O)C7=CC=C6)CC5)=C4)NC3=C2C(N)=O)=C1F	C41H39FN10O6S	BTK	Q06187	CRBN	US-20240246977-A1
TPD-GYSLII	SCHEMBL24598199	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]azetidin-3-yl]methyl]piperazin-1-yl]-2-[2-fluoro-3-methyl-4-(1,3-thiazol-4-ylcarbamoyl)phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	CC1=C(C(=O)NC2=CSC=N2)C=CC(C2=NN3CCC4=C(C=CC(N5CCN(CC6CN(C7=CC=C(N8CCC(=O)NC8=O)C=C7)C6)CC5)=C4)NC3=C2C(N)=O)=C1F	C41H42FN11O4S	BTK	Q06187	CRBN	US-20240246977-A1
TPD-A6WDLH	SCHEMBL24598175	8-[4-[[1-[4-[(2,4-dioxo-1,3-diazinan-1-yl)methyl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[2-fluoro-3-methyl-4-(1,3-thiazol-4-ylcarbamoyl)phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	CC1=C(C(=O)NC2=CSC=N2)C=CC(C2=NN3CCC4=C(C=CC(N5CCN(CC6CCN(C7=CC=C(CN8CCC(=O)NC8=O)C=C7)CC6)CC5)=C4)NC3=C2C(N)=O)=C1F	C44H48FN11O4S	BTK	Q06187	CRBN	US-20240246977-A1
TPD-TIIISA	SCHEMBL24598202	8-[4-[[1-[3-[(2,4-dioxo-1,3-diazinan-1-yl)methyl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[2-fluoro-3-methyl-4-(1,3-thiazol-4-ylcarbamoyl)phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	CC1=C(C(=O)NC2=CSC=N2)C=CC(C2=NN3CCC4=C(C=CC(N5CCN(CC6CCN(C7=CC=CC(CN8CCC(=O)NC8=O)=C7)CC6)CC5)=C4)NC3=C2C(N)=O)=C1F	C44H48FN11O4S	BTK	Q06187	CRBN	US-20240246977-A1
TPD-NXHFY3	SCHEMBL24598064	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-(4-phenoxyphenyl)-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	NC(=O)C1=C2NC3=C(C=C(N4CCN(CC5CCN(C6=CC=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)CCN2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C44H47N9O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-XXBD6E	SCHEMBL24598177	8-[4-[3-[4-[[(3R)-2,6-dioxopiperidin-3-yl]amino]phenyl]cyclobutyl]piperazin-1-yl]-2-[2-fluoro-3-methyl-4-(1,3-thiazol-4-ylcarbamoyl)phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	CC1=C(C(=O)NC2=CSC=N2)C=CC(C2=NN3CCC4=C(C=CC(N5CCN(C6CC(C7=CC=C(N[C@@H]8CCC(=O)NC8=O)C=C7)C6)CC5)=C4)NC3=C2C(N)=O)=C1F	C42H43FN10O4S	BTK	Q06187	CRBN	US-20240246977-A1
TPD-NK7VFR	SCHEMBL24598167	8-[4-[3-[4-[[(3S)-2,6-dioxopiperidin-3-yl]amino]phenyl]cyclobutyl]piperazin-1-yl]-2-[2-fluoro-3-methyl-4-(1,3-thiazol-4-ylcarbamoyl)phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	CC1=C(C(=O)NC2=CSC=N2)C=CC(C2=NN3CCC4=C(C=CC(N5CCN(C6CC(C7=CC=C(N[C@H]8CCC(=O)NC8=O)C=C7)C6)CC5)=C4)NC3=C2C(N)=O)=C1F	C42H43FN10O4S	BTK	Q06187	CRBN	US-20240246977-A1
TPD-3VTYHA	SCHEMBL24598180	8-[4-[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidine-4-carbonyl]piperazin-1-yl]-2-[2-fluoro-3-methyl-4-(1,3-thiazol-4-ylcarbamoyl)phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	CC1=C(C(=O)NC2=CSC=N2)C=CC(C2=NN3CCC4=C(C=CC(N5CCN(C(=O)C6CCN(C7=CC=C(N8CCC(=O)NC8=O)C=C7)CC6)CC5)=C4)NC3=C2C(N)=O)=C1F	C43H44FN11O5S	BTK	Q06187	CRBN	US-20240246977-A1
TPD-S8164J	SCHEMBL24598157	8-[4-[[(3R)-1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]pyrrolidin-3-yl]methyl]piperazin-1-yl]-2-[2-fluoro-3-methyl-4-(1,3-thiazol-4-ylcarbamoyl)phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	CC1=C(C(=O)NC2=CSC=N2)C=CC(C2=NN3CCC4=C(C=CC(N5CCN(C[C@H]6CCN(C7=CC=C(N8CCC(=O)NC8=O)C=C7)C6)CC5)=C4)NC3=C2C(N)=O)=C1F	C42H44FN11O4S	BTK	Q06187	CRBN	US-20240246977-A1
TPD-FI2JEZ	SCHEMBL31030074	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[4-[[(2-methoxy-3-methylbenzoyl)amino]methyl]-3-methylphenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	COC1=C(C(=O)NCC2=CC=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2C)C=CC=C1C	C49H56N10O5	BTK	Q06187	CRBN	US-20240246977-A1
TPD-YIAJVM	SCHEMBL24598383	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[4-[[(2-methoxy-4-methylbenzoyl)amino]methyl]-3-methylphenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31029969	COC1=C(C(=O)NCC2=CC=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2C)C=CC(C)=C1	C49H56N10O5	BTK	Q06187	CRBN	US-20240246977-A1
TPD-DZTTWF	SCHEMBL24598170	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[4-[[(2-methoxybenzoyl)amino]methyl]-3-methylphenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	COC1=C(C(=O)NCC2=C(C)C=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2)C=CC=C1	C48H54N10O5	BTK	Q06187	CRBN	US-20240246977-A1
TPD-3YI3C2	SCHEMBL24598348	2-[4-[[(4,5-difluoro-2-methoxybenzoyl)amino]methyl]-3-methylphenyl]-8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	COC1=C(C(=O)NCC2=C(C)C=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2)C=C(F)C(F)=C1	C48H52F2N10O5	BTK	Q06187	CRBN	US-20240246977-A1
TPD-IGM43J	SCHEMBL24598312	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[4-[[(2-methoxypyridine-3-carbonyl)amino]methyl]-3-methylphenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	COC1=C(C(=O)NCC2=C(C)C=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2)C=CC=N1	C47H53N11O5	BTK	Q06187	CRBN	US-20240246977-A1
TPD-XQ3J5R	SCHEMBL24598159	8-[4-[2-[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]ethyl]piperazin-1-yl]-2-(4-phenoxyphenyl)-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	NC(=O)C1=C2NC3=C(C=C(N4CCN(CCC5CCN(C6=CC=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)CCN2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C45H49N9O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-SXQ2DM	SCHEMBL24598575	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[4-[[(3-methoxypyridine-2-carbonyl)amino]methyl]-3-methylphenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	COC1=C(C(=O)NCC2=C(C)C=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2)N=CC=C1	C47H53N11O5	BTK	Q06187	CRBN	US-20240246977-A1
TPD-MGW94W	SCHEMBL24598316	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[4-[[(3-methoxypyridine-4-carbonyl)amino]methyl]-3-methylphenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	COC1=C(C(=O)NCC2=C(C)C=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2)C=CN=C1	C47H53N11O5	BTK	Q06187	CRBN	US-20240246977-A1
TPD-9L1GWD	SCHEMBL24598331	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[4-[[(2-methoxy-6-methylbenzoyl)amino]methyl]-3-methylphenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	COC1=C(C(=O)NCC2=C(C)C=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2)C(C)=CC=C1	C49H56N10O5	BTK	Q06187	CRBN	US-20240246977-A1
TPD-5B8C72	SCHEMBL24598319	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[4-[[(2-methoxy-5-methylbenzoyl)amino]methyl]-3-methylphenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31029994	COC1=C(C(=O)NCC2=CC=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2C)C=C(C)C=C1	C49H56N10O5	BTK	Q06187	CRBN	US-20240246977-A1
TPD-16TTW6	SCHEMBL24598351	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[4-[[(3-fluoro-2-methoxybenzoyl)amino]methyl]-3-methylphenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31030066	COC1=C(C(=O)NCC2=CC=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2C)C=CC=C1F	C48H53FN10O5	BTK	Q06187	CRBN	US-20240246977-A1
TPD-KW4OLL	SCHEMBL24598385	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[4-[[(4-fluoro-2-methoxybenzoyl)amino]methyl]-3-methylphenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31030025	COC1=C(C(=O)NCC2=CC=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2C)C=CC(F)=C1	C48H53FN10O5	BTK	Q06187	CRBN	US-20240246977-A1
TPD-7DC14I	SCHEMBL24598314	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[4-[[(5-fluoro-2-methoxybenzoyl)amino]methyl]-3-methylphenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31030063	COC1=C(C(=O)NCC2=CC=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2C)C=C(F)C=C1	C48H53FN10O5	BTK	Q06187	CRBN	US-20240246977-A1
TPD-3RZ903	SCHEMBL31030014	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[3-methyl-4-[[(2,3,4,5-tetrafluoro-6-methoxybenzoyl)amino]methyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	COC1=C(C(=O)NCC2=C(C)C=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2)C(F)=C(F)C(F)=C1F	C48H50F4N10O5	BTK	Q06187	CRBN	US-20240246977-A1
TPD-BDOFWH	SCHEMBL24598377	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[2-methoxy-4-[[(2-methoxybenzoyl)amino]methyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	COC1=C(C(=O)NCC2=CC(OC)=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2)C=CC=C1	C48H54N10O6	BTK	Q06187	CRBN	US-20240246977-A1
TPD-66Q3LA	SCHEMBL24598374	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[4-[[(2-methoxybenzoyl)amino]methyl]-3-(trifluoromethyl)phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31029975	COC1=C(C(=O)NCC2=CC=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2C(F)(F)F)C=CC=C1	C48H51F3N10O5	BTK	Q06187	CRBN	US-20240246977-A1
TPD-VLAT5H	SCHEMBL24598059	8-[2-[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]ethoxy]-2-(4-phenoxyphenyl)-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	NC(=O)C1=C2NC3=C(C=C(OCCC4CCN(C5=CC=C(N6CCC(=O)NC6=O)C=C5)CC4)C=C3)CCN2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C41H41N7O5	BTK	Q06187	CRBN	US-20240246977-A1
TPD-I5A0MH	SCHEMBL24598416	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[2-fluoro-4-[[(2-methoxybenzoyl)amino]methyl]-3-methylphenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31029984	COC1=C(C(=O)NCC2=CC=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C(F)=C2C)C=CC=C1	C48H53FN10O5	BTK	Q06187	CRBN	US-20240246977-A1
TPD-VER8MF	SCHEMBL24598355	2-[2,3-difluoro-4-[[(2-methoxybenzoyl)amino]methyl]phenyl]-8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	COC1=C(C(=O)NCC2=C(F)C(F)=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2)C=CC=C1	C47H50F2N10O5	BTK	Q06187	CRBN	US-20240246977-A1
TPD-94WOCI	SCHEMBL24598438	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[2-fluoro-4-[[(2-methoxybenzoyl)amino]methyl]-5-methylphenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31030040	COC1=C(C(=O)NCC2=C(C)C=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C(F)=C2)C=CC=C1	C48H53FN10O5	BTK	Q06187	CRBN	US-20240246977-A1
TPD-94FIQD	SCHEMBL24598067	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[2-fluoro-3-methyl-4-[[6-methyl-4-(trifluoromethyl)pyridin-2-yl]carbamoyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	CC1=CC(C(F)(F)F)=CC(NC(=O)C2=C(C)C(F)=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2)=N1	C47H49F4N11O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-1PHE6O	SCHEMBL24598266	8-[1-[2-[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]ethyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	NC(=O)C1=C2NC3=C(C=C(C4CCN(CCC5CCN(C6=CC=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)CCN2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C46H50N8O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-30WY6C	SCHEMBL24598255	8-[[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperidine-4-carbonyl]amino]-2-(4-phenoxyphenyl)-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	NC(=O)C1=C2NC3=C(C=C(NC(=O)C4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C=C3)CCN2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C49H49N9O7	BTK	Q06187	CRBN	US-20240246977-A1
TPD-QK8QWO	SCHEMBL24598065	8-[1-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	NC(=O)C1=C2NC3=C(C=C(C4CCN(CC5CCN(C6=CC=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)CCN2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C45H48N8O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-0IF6DK	SCHEMBL24598071	8-[2-[1-[4-[(2,6-dioxopiperidin-3-yl)amino]phenyl]piperidin-4-yl]ethyl]-2-(4-phenoxyphenyl)-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	NC(=O)C1=C2NC3=C(C=C(CCC4CCN(C5=CC=C(NC6CCC(=O)NC6=O)C=C5)CC4)C=C3)CCN2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C42H43N7O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-2BIM30	SCHEMBL24598072	N-[1-[4-carbamoyl-5-(4-phenoxyphenyl)-1H-pyrazol-3-yl]-2,3-dihydroindol-5-yl]-1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidine-4-carboxamide	NC(=O)C1=C(N2CCC3=C2C=CC(NC(=O)C2CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC2)=C3)NN=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C43H38N8O7	BTK	Q06187	CRBN	US-20240246977-A1
TPD-Y3Z06F	SCHEMBL24598362	2-[4-(4-tert-butylphenoxy)phenyl]-8-[1-[2-[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]ethyl]piperidin-4-yl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	CC(C)(C)C1=CC=C(OC2=CC=C(C3=NN4CCC5=C(C=CC(C6CCN(CCC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2)C=C1	C50H58N8O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-VBS5FH	SCHEMBL24598075	2-[4-(4-tert-butylphenoxy)phenyl]-8-[1-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperidin-4-yl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	CC(C)(C)C1=CC=C(OC2=CC=C(C3=NN4CCC5=C(C=CC(C6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2)C=C1	C49H56N8O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-6O1P9K	SCHEMBL24598408	9-N-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1,9-dicarboxamide; SCHEMBL31030000	NC(=O)C1=C2NC3=C(C=CC(C(=O)NC4CCN(CC5CCN(C6=C(F)C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)=C3)CCN2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C49H48FN9O7	BTK	Q06187	CRBN	US-20240246977-A1
TPD-TZ49J3	SCHEMBL24598410	9-[[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperidine-4-carbonyl]amino]-2-(4-phenoxyphenyl)-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31030049	NC(=O)C1=C2NC3=C(C=CC(NC(=O)C4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)=C3)CCN2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C49H49N9O7	BTK	Q06187	CRBN	US-20240246977-A1
TPD-GN3G8L	SCHEMBL24598084	9-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazine-1-carbonyl]-2-(4-phenoxyphenyl)-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31030034	NC(=O)C1=C2NC3=C(C=CC(C(=O)N4CCN(CC5CCN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)=C3)CCN2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C48H47N9O7	BTK	Q06187	CRBN	US-20240246977-A1
TPD-F4FVY6	SCHEMBL24598074	9-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidine-1-carbonyl]-2-(4-phenoxyphenyl)-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31029962	NC(=O)C1=C2NC3=C(C=CC(C(=O)N4CCC(CN5CCN(C6=CC7=C(C=C6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)=C3)CCN2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C48H46FN9O7	BTK	Q06187	CRBN	US-20240246977-A1
TPD-A2ZBSQ	SCHEMBL24598076	9-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]-2-(4-phenoxyphenyl)-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31030067	NC(=O)C1=C2NC3=C(C=CC(N4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)=C3)CCN2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C47H47N9O6	BTK	Q06187	CRBN	US-20240246977-A1
TPD-E5R1M4	SCHEMBL24598196	8-[[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperidin-4-yl]amino]-2-(4-phenoxyphenyl)-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	NC(=O)C1=C2NC3=C(C=C(NC4CCN(CC5CCN(C6=C(F)C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C=C3)CCN2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C48H48FN9O6	BTK	Q06187	CRBN	US-20240246977-A1
TPD-MR50TK	SCHEMBL24598335	9-[1-[2-[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]ethyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31029981	NC(=O)C1=C2NC3=C(C=CC(C4CCN(CCC5CCN(C6=CC=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)=C3)CCN2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C46H50N8O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-BXNBCH	SCHEMBL24598154	9-[1-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31030061	NC(=O)C1=C2NC3=C(C=CC(C4CCN(CC5CCN(C6=CC=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)=C3)CCN2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C45H48N8O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-WBNB8B	US20240246977A1_32A25	.	NC(=O)C1=C2NC3=C(C=CC(OCCC4CCN(C5=CC=C(N6CCC(=O)NC6=O)C=C5)CC4)=C3)CCC2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C42H42N6O5	BTK	Q06187	CRBN	US-20240246977-A1
TPD-9G1R0T	SCHEMBL24598125	9-[1-[3-[4-[(2,6-dioxopiperidin-3-yl)amino]phenoxy]propyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31030032	NC(=O)C1=C2NC3=C(C=CC(C4CCN(CCCOC5=CC=C(NC6CCC(=O)NC6=O)C=C5)CC4)=C3)CCN2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C43H45N7O5	BTK	Q06187	CRBN	US-20240246977-A1
TPD-CPRX8Z	SCHEMBL24598085	9-[1-[2-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]ethyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL29710549	NC(=O)C1=C2NC3=C(C=CC(C4CCN(CCC5=CC=C(N6CCC(=O)NC6=O)C=C5)CC4)=C3)CCN2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C41H41N7O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-Y62IQ3	SCHEMBL24598224	9-[1-[2-[4-(2,6-dioxopiperidin-3-yl)phenyl]ethyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL29710558	NC(=O)C1=C2NC3=C(C=CC(C4CCN(CCC5=CC=C(C6CCC(=O)NC6=O)C=C5)CC4)=C3)CCN2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C42H42N6O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-4Q018U	SCHEMBL24598186	9-[1-[[1-[4-[(2,6-dioxopiperidin-3-yl)amino]phenyl]piperidin-4-yl]methyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31029999	NC(=O)C1=C2NC3=C(C=CC(C4CCN(CC5CCN(C6=CC=C(NC7CCC(=O)NC7=O)C=C6)CC5)CC4)=C3)CCN2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C46H50N8O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-6IDU1P	SCHEMBL24598269	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-(6-phenoxypyridin-3-yl)-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	NC(=O)C1=C2NC3=C(C=C(N4CCN(CC5CCN(C6=CC=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)CCN2N=C1C1=CC=C(OC2=CC=CC=C2)N=C1	C43H46N10O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-FTEVTA	SCHEMBL24598121	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-(2-methoxy-4-phenoxyphenyl)-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	COC1=C(C2=NN3CCC4=C(C=CC(N5CCN(CC6CCN(C7=CC=C(N8CCC(=O)NC8=O)C=C7)CC6)CC5)=C4)NC3=C2C(N)=O)C=CC(OC2=CC=CC=C2)=C1	C45H49N9O5	BTK	Q06187	CRBN	US-20240246977-A1
TPD-24OPD1	SCHEMBL24598271	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-(2-fluoro-4-phenoxyphenyl)-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	NC(=O)C1=C2NC3=C(C=C(N4CCN(CC5CCN(C6=CC=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)CCN2N=C1C1=C(F)C=C(OC2=CC=CC=C2)C=C1	C44H46FN9O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-TQN26T	SCHEMBL24598195	8-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]-2-(4-phenoxyphenyl)-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	NC(=O)C1=C2NC3=C(C=C(N4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C=C3)CCN2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C47H47N9O6	BTK	Q06187	CRBN	US-20240246977-A1
TPD-LZR6HD	SCHEMBL24598272	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-(4-phenylmethoxyphenyl)-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	NC(=O)C1=C2NC3=C(C=C(N4CCN(CC5CCN(C6=CC=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)CCN2N=C1C1=CC=C(OCC2=CC=CC=C2)C=C1	C45H49N9O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-UXGRJW	SCHEMBL24598160	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[4-[[4-(trifluoromethyl)pyridin-2-yl]carbamoyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	NC(=O)C1=C2NC3=C(C=C(N4CCN(CC5CCN(C6=CC=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)CCN2N=C1C1=CC=C(C(=O)NC2=NC=CC(C(F)(F)F)=C2)C=C1	C45H46F3N11O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-TDOTF4	SCHEMBL24598226	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)-3-methylphenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[4-[[4-(trifluoromethyl)pyridin-2-yl]carbamoyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31030036	CC1=CC(N2CCC(CN3CCN(C4=CC5=C(C=C4)NC4=C(C(N)=O)C(C6=CC=C(C(=O)NC7=NC=CC(C(F)(F)F)=C7)C=C6)=NN4CC5)CC3)CC2)=CC=C1N1CCC(=O)NC1=O	C46H48F3N11O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-SFAFK1	SCHEMBL24598225	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[4-[(4-methoxypyridin-2-yl)carbamoyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31029961	COC1=CC=NC(NC(=O)C2=CC=C(C3=NN4CCC5=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=CC=C5NC4=C3C(N)=O)C=C2)=C1	C45H49N11O5	BTK	Q06187	CRBN	US-20240246977-A1
TPD-M2H8YC	SCHEMBL24598229	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[4-[(4-methylpyridin-2-yl)carbamoyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31030020	CC1=CC=NC(NC(=O)C2=CC=C(C3=NN4CCC5=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=CC=C5NC4=C3C(N)=O)C=C2)=C1	C45H49N11O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-T4WNUV	SCHEMBL24598275	2-[4-[(4-cyclopropylpyridin-2-yl)carbamoyl]phenyl]-8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31030046	NC(=O)C1=C2NC3=CC=C(N4CCN(CC5CCN(C6=CC=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3CCN2N=C1C1=CC=C(C(=O)NC2=CC(C3CC3)=CC=N2)C=C1	C47H51N11O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-DKO6OG	SCHEMBL24598250	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[4-(pyridin-2-ylcarbamoyl)phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31030055	NC(=O)C1=C2NC3=CC=C(N4CCN(CC5CCN(C6=CC=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3CCN2N=C1C1=CC=C(C(=O)NC2=CC=CC=N2)C=C1	C44H47N11O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-KRI9CT	SCHEMBL24598354	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[4-[[6-(trifluoromethyl)pyridin-2-yl]carbamoyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31029989	NC(=O)C1=C2NC3=CC=C(N4CCN(CC5CCN(C6=CC=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3CCN2N=C1C1=CC=C(C(=O)NC2=CC=CC(C(F)(F)F)=N2)C=C1	C45H46F3N11O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-U606A8	US20240246977A1_4A3	.	C=C1CCC(N2C(=O)C3=C(C=C(N4CCC(CNC5=CC6=C(C=C5)NC5=C(C(N)=O)C(C7=CC=C(OC8=CC=CC=C8)C=C7)=NN5CC6)CC4)C=C3)C2=O)C(=O)N1	C44H42N8O5	BTK	Q06187	CRBN	US-20240246977-A1
TPD-00MKD6	SCHEMBL24598405	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[4-[[5-(trifluoromethyl)pyridin-2-yl]carbamoyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31029988	NC(=O)C1=C2NC3=CC=C(N4CCN(CC5CCN(C6=CC=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3CCN2N=C1C1=CC=C(C(=O)NC2=CC=C(C(F)(F)F)C=N2)C=C1	C45H46F3N11O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-3JKR2P	SCHEMBL24598205	2-[4-[[4-(difluoromethyl)pyridin-2-yl]carbamoyl]phenyl]-8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31030056	NC(=O)C1=C2NC3=CC=C(N4CCN(CC5CCN(C6=CC=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3CCN2N=C1C1=CC=C(C(=O)NC2=CC(C(F)F)=CC=N2)C=C1	C45H47F2N11O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-VCSMGW	SCHEMBL24598407	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[4-[(6-methylpyridin-2-yl)carbamoyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31030076	CC1=NC(NC(=O)C2=CC=C(C3=NN4CCC5=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=CC=C5NC4=C3C(N)=O)C=C2)=CC=C1	C45H49N11O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-B3I4QX	SCHEMBL24598340	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[2-fluoro-4-[[4-(trifluoromethyl)pyridin-2-yl]carbamoyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31030028	NC(=O)C1=C2NC3=C(C=C(N4CCN(CC5CCN(C6=CC=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)CCN2N=C1C1=C(F)C=C(C(=O)NC2=CC(C(F)(F)F)=CC=N2)C=C1	C45H45F4N11O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-EYLQUD	SCHEMBL24598187	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[3-fluoro-4-[[4-(trifluoromethyl)pyridin-2-yl]carbamoyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	NC(=O)C1=C2NC3=C(C=C(N4CCN(CC5CCN(C6=CC=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)CCN2N=C1C1=CC(F)=C(C(=O)NC2=NC=CC(C(F)(F)F)=C2)C=C1	C45H45F4N11O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-Y5HPPI	SCHEMBL24598010	2-[3,5-difluoro-4-[[4-(trifluoromethyl)pyridin-2-yl]carbamoyl]phenyl]-8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31030018	NC(=O)C1=C2NC3=C(C=C(N4CCN(CC5CCN(C6=CC=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)CCN2N=C1C1=CC(F)=C(C(=O)NC2=NC=CC(C(F)(F)F)=C2)C(F)=C1	C45H44F5N11O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-RPOR54	SCHEMBL24598172	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[2-methyl-4-[[4-(trifluoromethyl)pyridin-2-yl]carbamoyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	CC1=C(C2=NN3CCC4=C(C=CC(N5CCN(CC6CCN(C7=CC=C(N8CCC(=O)NC8=O)C=C7)CC6)CC5)=C4)NC3=C2C(N)=O)C=CC(C(=O)NC2=NC=CC(C(F)(F)F)=C2)=C1	C46H48F3N11O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-U2XQRY	SCHEMBL24598213	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[2-methoxy-4-[(6-methylpyridin-2-yl)carbamoyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	COC1=C(C2=NN3CCC4=C(C=CC(N5CCN(CC6CCN(C7=CC=C(N8CCC(=O)NC8=O)C=C7)CC6)CC5)=C4)NC3=C2C(N)=O)C=CC(C(=O)NC2=NC(C)=CC=C2)=C1	C46H51N11O5	BTK	Q06187	CRBN	US-20240246977-A1
TPD-0PM9UB	SCHEMBL24598208	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[2-methoxy-4-[[4-(trifluoromethyl)pyridin-2-yl]carbamoyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	COC1=C(C2=NN3CCC4=C(C=CC(N5CCN(CC6CCN(C7=CC=C(N8CCC(=O)NC8=O)C=C7)CC6)CC5)=C4)NC3=C2C(N)=O)C=CC(C(=O)NC2=NC=CC(C(F)(F)F)=C2)=C1	C46H48F3N11O5	BTK	Q06187	CRBN	US-20240246977-A1
TPD-VDSU3X	SCHEMBL24598491	2-[3,5-dimethyl-4-[[4-(trifluoromethyl)pyridin-2-yl]carbamoyl]phenyl]-8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	CC1=CC(C2=NN3CCC4=C(C=CC(N5CCN(CC6CCN(C7=CC=C(N8CCC(=O)NC8=O)C=C7)CC6)CC5)=C4)NC3=C2C(N)=O)=CC(C)=C1C(=O)NC1=NC=CC(C(F)(F)F)=C1	C47H50F3N11O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-U6QK56	SCHEMBL24598053	8-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]amino]-2-(4-phenoxyphenyl)-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL29710608	NC(=O)C1=C2NC3=C(C=C(NC4CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)CCN2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C42H38N8O6	BTK	Q06187	CRBN	US-20240246977-A1
TPD-95641H	SCHEMBL24598430	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[3-methyl-4-[[4-(trifluoromethyl)pyridin-2-yl]carbamoyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	CC1=C(C(=O)NC2=NC=CC(C(F)(F)F)=C2)C=CC(C2=NN3CCC4=C(C=CC(N5CCN(CC6CCN(C7=CC=C(N8CCC(=O)NC8=O)C=C7)CC6)CC5)=C4)NC3=C2C(N)=O)=C1	C46H48F3N11O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-RPAIFS	SCHEMBL24598146	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[3-methyl-4-[(6-methylpyridin-2-yl)carbamoyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	CC1=CC=CC(NC(=O)C2=C(C)C=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2)=N1	C46H51N11O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-OESHCQ	SCHEMBL24598493	2-[4-[(4,6-dimethylpyridin-2-yl)carbamoyl]-3-methylphenyl]-8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	CC1=CC(NC(=O)C2=C(C)C=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2)=NC(C)=C1	C47H53N11O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-YFT9QN	SCHEMBL24598215	2-[3-chloro-4-[(6-methylpyridin-2-yl)carbamoyl]phenyl]-8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31029966	CC1=CC=CC(NC(=O)C2=C(Cl)C=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2)=N1	C45H48ClN11O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-HKO21Q	SCHEMBL24598398	2-[2-chloro-4-[(6-methylpyridin-2-yl)carbamoyl]phenyl]-8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	CC1=CC=CC(NC(=O)C2=CC(Cl)=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2)=N1	C45H48ClN11O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-V831SC	SCHEMBL24598212	2-[3-chloro-4-[[4-(trifluoromethyl)pyridin-2-yl]carbamoyl]phenyl]-8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31029980	NC(=O)C1=C2NC3=C(C=C(N4CCN(CC5CCN(C6=CC=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)CCN2N=C1C1=CC(Cl)=C(C(=O)NC2=NC=CC(C(F)(F)F)=C2)C=C1	C45H45ClF3N11O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-XG5BSA	SCHEMBL24598190	2-[2-chloro-4-[[4-(trifluoromethyl)pyridin-2-yl]carbamoyl]phenyl]-8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	NC(=O)C1=C2NC3=C(C=C(N4CCN(CC5CCN(C6=CC=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)CCN2N=C1C1=C(Cl)C=C(C(=O)NC2=NC=CC(C(F)(F)F)=C2)C=C1	C45H45ClF3N11O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-YA2U8Y	SCHEMBL24598248	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[2-fluoro-3-methyl-4-[[4-(trifluoromethyl)pyridin-2-yl]carbamoyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	CC1=C(C(=O)NC2=NC=CC(C(F)(F)F)=C2)C=CC(C2=NN3CCC4=C(C=CC(N5CCN(CC6CCN(C7=CC=C(N8CCC(=O)NC8=O)C=C7)CC6)CC5)=C4)NC3=C2C(N)=O)=C1F	C46H47F4N11O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-M0KVMJ	SCHEMBL24598241	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[2-fluoro-3-methyl-4-[(6-methylpyridin-2-yl)carbamoyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	CC1=CC=CC(NC(=O)C2=C(C)C(F)=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2)=N1	C46H50FN11O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-5OJK3E	SCHEMBL24598246	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[4-[[(2-methoxybenzoyl)amino]methyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	COC1=C(C(=O)NCC2=CC=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2)C=CC=C1	C47H52N10O5	BTK	Q06187	CRBN	US-20240246977-A1
TPD-ZXDPCU	SCHEMBL24598252	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[4-[[(2-methoxy-5-methylbenzoyl)amino]methyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	COC1=C(C(=O)NCC2=CC=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2)C=C(C)C=C1	C48H54N10O5	BTK	Q06187	CRBN	US-20240246977-A1
TPD-Z0LVI6	SCHEMBL24598214	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[4-[[(2-methoxynaphthalene-1-carbonyl)amino]methyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31030059	COC1=C(C(=O)NCC2=CC=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2)C2=C(C=CC=C2)C=C1	C51H54N10O5	BTK	Q06187	CRBN	US-20240246977-A1
TPD-5JZUQ7	SCHEMBL24598105	8-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]-2-(4-phenoxyphenyl)-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	NC(=O)C1=C2NC3=C(C=C(N4CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)CCN2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C41H36N8O6	BTK	Q06187	CRBN	US-20240246977-A1
TPD-LB31M6	SCHEMBL24598211	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[4-[[[2-methoxy-5-(trifluoromethyl)benzoyl]amino]methyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	COC1=C(C(=O)NCC2=CC=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2)C=C(C(F)(F)F)C=C1	C48H51F3N10O5	BTK	Q06187	CRBN	US-20240246977-A1
TPD-EXPH3C	SCHEMBL24598232	2-[4-[[(2,6-dimethoxybenzoyl)amino]methyl]phenyl]-8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	COC1=CC=CC(OC)=C1C(=O)NCC1=CC=C(C2=NN3CCC4=C(C=CC(N5CCN(CC6CCN(C7=CC=C(N8CCC(=O)NC8=O)C=C7)CC6)CC5)=C4)NC3=C2C(N)=O)C=C1	C48H54N10O6	BTK	Q06187	CRBN	US-20240246977-A1
TPD-6DDGGQ	SCHEMBL24598305	2-[4-[[(2,4-dimethoxybenzoyl)amino]methyl]phenyl]-8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	COC1=CC(OC)=C(C(=O)NCC2=CC=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2)C=C1	C48H54N10O6	BTK	Q06187	CRBN	US-20240246977-A1
TPD-KV0GR5	SCHEMBL24598238	2-[4-[[(2,3-difluoro-6-methoxybenzoyl)amino]methyl]phenyl]-8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31030010	COC1=C(C(=O)NCC2=CC=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2)C(F)=C(F)C=C1	C47H50F2N10O5	BTK	Q06187	CRBN	US-20240246977-A1
TPD-OT4VE6	SCHEMBL24598532	2-[4-[[(5-cyclopropyl-2-methoxybenzoyl)amino]methyl]phenyl]-8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31029955	COC1=C(C(=O)NCC2=CC=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2)C=C(C2CC2)C=C1	C50H56N10O5	BTK	Q06187	CRBN	US-20240246977-A1
TPD-J8XFB0	SCHEMBL24598436	2-[4-[[(4,5-difluoro-2-methoxybenzoyl)amino]methyl]phenyl]-8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	COC1=C(C(=O)NCC2=CC=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2)C=C(F)C(F)=C1	C47H50F2N10O5	BTK	Q06187	CRBN	US-20240246977-A1
TPD-XF0D8P	SCHEMBL24598243	3-tert-butyl-N-[[4-[1-carbamoyl-8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepin-2-yl]phenyl]methyl]-1,2,4-oxadiazole-5-carboxamide	CC(C)(C)C1=NOC(C(=O)NCC2=CC=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2)=N1	C46H54N12O5	BTK	Q06187	CRBN	US-20240246977-A1
TPD-O399MR	SCHEMBL24598216	5-tert-butyl-N-[[4-[1-carbamoyl-8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepin-2-yl]-2-methylphenyl]methyl]-1,2,4-oxadiazole-3-carboxamide	CC1=C(CNC(=O)C2=NOC(C(C)(C)C)=N2)C=CC(C2=NN3CCC4=C(C=CC(N5CCN(CC6CCN(C7=CC=C(N8CCC(=O)NC8=O)C=C7)CC6)CC5)=C4)NC3=C2C(N)=O)=C1	C47H56N12O5	BTK	Q06187	CRBN	US-20240246977-A1
TPD-8W8Y6E	SCHEMBL24598021	3-tert-butyl-N-[[4-[1-carbamoyl-8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepin-2-yl]-2-methylphenyl]methyl]-1,2,4-oxadiazole-5-carboxamide	CC1=C(CNC(=O)C2=NC(C(C)(C)C)=NO2)C=CC(C2=NN3CCC4=C(C=CC(N5CCN(CC6CCN(C7=CC=C(N8CCC(=O)NC8=O)C=C7)CC6)CC5)=C4)NC3=C2C(N)=O)=C1	C47H56N12O5	BTK	Q06187	CRBN	US-20240246977-A1
TPD-3YFAKW	SCHEMBL24598200	8-[[2-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]-2-(4-phenoxyphenyl)-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	NC(=O)C1=C2NC3=C(C=C(NC(=O)COCCOCCOCCOCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C3)CCN2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C47H48N8O11	BTK	Q06187	CRBN	US-20240246977-A1
TPD-X63QHQ	SCHEMBL24598015	2-[4-[[(1-tert-butylpyrazole-3-carbonyl)amino]methyl]-3-methylphenyl]-8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	CC1=C(CNC(=O)C2=NN(C(C)(C)C)C=C2)C=CC(C2=NN3CCC4=C(C=CC(N5CCN(CC6CCN(C7=CC=C(N8CCC(=O)NC8=O)C=C7)CC6)CC5)=C4)NC3=C2C(N)=O)=C1	C48H58N12O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-H9ZDEO	SCHEMBL24598016	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[4-[[(2-methoxynaphthalene-1-carbonyl)amino]methyl]-3-methylphenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31030015	COC1=C(C(=O)NCC2=C(C)C=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2)C2=C(C=CC=C2)C=C1	C52H56N10O5	BTK	Q06187	CRBN	US-20240246977-A1
TPD-605JW7	SCHEMBL24598019	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[4-[[[2-methoxy-5-(trifluoromethyl)benzoyl]amino]methyl]-3-methylphenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	COC1=C(C(=O)NCC2=C(C)C=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2)C=C(C(F)(F)F)C=C1	C49H53F3N10O5	BTK	Q06187	CRBN	US-20240246977-A1
TPD-QTKG7F	SCHEMBL24598022	2-[4-[[(5-chloro-2-methoxybenzoyl)amino]methyl]-3-methylphenyl]-8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31030057	COC1=C(C(=O)NCC2=C(C)C=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2)C=C(Cl)C=C1	C48H53ClN10O5	BTK	Q06187	CRBN	US-20240246977-A1
TPD-YRM8WT	SCHEMBL24598023	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[3-fluoro-4-[[(2-methoxybenzoyl)amino]methyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31029991	COC1=C(C(=O)NCC2=CC=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2F)C=CC=C1	C47H51FN10O5	BTK	Q06187	CRBN	US-20240246977-A1
TPD-1K3IAD	SCHEMBL24598017	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[3-fluoro-4-[[(2-methoxynaphthalene-1-carbonyl)amino]methyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31030069	COC1=C(C(=O)NCC2=CC=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2F)C2=C(C=CC=C2)C=C1	C51H53FN10O5	BTK	Q06187	CRBN	US-20240246977-A1
TPD-J6MU79	SCHEMBL24598158	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[3-fluoro-4-[[[2-methoxy-5-(trifluoromethyl)benzoyl]amino]methyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	COC1=C(C(=O)NCC2=C(F)C=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2)C=C(C(F)(F)F)C=C1	C48H50F4N10O5	BTK	Q06187	CRBN	US-20240246977-A1
TPD-E9ZMYM	SCHEMBL24598555	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[2-methoxy-4-[[[2-methoxy-5-(trifluoromethyl)benzoyl]amino]methyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	COC1=C(C(=O)NCC2=CC(OC)=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2)C=C(C(F)(F)F)C=C1	C49H53F3N10O6	BTK	Q06187	CRBN	US-20240246977-A1
TPD-1ZPNWU	SCHEMBL24598258	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[2-fluoro-4-[[[2-methoxy-5-(trifluoromethyl)benzoyl]amino]methyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	COC1=C(C(=O)NCC2=CC(F)=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2)C=C(C(F)(F)F)C=C1	C48H50F4N10O5	BTK	Q06187	CRBN	US-20240246977-A1
TPD-1QZGWG	SCHEMBL24598026	2-[2,3-difluoro-4-[[[2-methoxy-5-(trifluoromethyl)benzoyl]amino]methyl]phenyl]-8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	COC1=C(C(=O)NCC2=C(F)C(F)=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2)C=C(C(F)(F)F)C=C1	C48H49F5N10O5	BTK	Q06187	CRBN	US-20240246977-A1
TPD-N0GQDX	SCHEMBL24598141	8-N-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1,8-dicarboxamide	NC(=O)C1=C2NC3=C(C=C(C(=O)NC4CCN(CC5CCN(C6=C(F)C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C=C3)CCN2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C49H48FN9O7	BTK	Q06187	CRBN	US-20240246977-A1
TPD-66PL0A	SCHEMBL24598027	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[4-[1-[[4-(trifluoromethyl)pyridin-2-yl]amino]ethyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	CC(NC1=NC=CC(C(F)(F)F)=C1)C1=CC=C(C2=NN3CCC4=C(C=CC(N5CCN(CC6CCN(C7=CC=C(N8CCC(=O)NC8=O)C=C7)CC6)CC5)=C4)NC3=C2C(N)=O)C=C1	C46H50F3N11O3	BTK	Q06187	CRBN	US-20240246977-A1
TPD-GAM0P6	SCHEMBL24598028	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[4-[1-[[4-(trifluoromethyl)pyridin-2-yl]amino]cyclopropyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	NC(=O)C1=C2NC3=C(C=C(N4CCN(CC5CCN(C6=CC=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)CCN2N=C1C1=CC=C(C2(NC3=NC=CC(C(F)(F)F)=C3)CC2)C=C1	C47H50F3N11O3	BTK	Q06187	CRBN	US-20240246977-A1
TPD-773QF3	SCHEMBL24598024	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[4-[1-[[4-(trifluoromethyl)pyridin-2-yl]amino]propyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	CCC(NC1=NC=CC(C(F)(F)F)=C1)C1=CC=C(C2=NN3CCC4=C(C=CC(N5CCN(CC6CCN(C7=CC=C(N8CCC(=O)NC8=O)C=C7)CC6)CC5)=C4)NC3=C2C(N)=O)C=C1	C47H52F3N11O3	BTK	Q06187	CRBN	US-20240246977-A1
TPD-1KS36P	SCHEMBL24598020	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[4-[(1R)-1-[(4-methoxypyridine-3-carbonyl)amino]ethyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31029979	COC1=C(C(=O)N[C@H](C)C2=CC=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2)C=NC=C1	C47H53N11O5	BTK	Q06187	CRBN	US-20240246977-A1
TPD-5AOPV3	SCHEMBL24598421	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[4-[1-[(2-methoxybenzoyl)amino]ethyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	COC1=C(C(=O)NC(C)C2=CC=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2)C=CC=C1	C48H54N10O5	BTK	Q06187	CRBN	US-20240246977-A1
TPD-KBJBT3	SCHEMBL24598295	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[4-[(1R)-1-[(2-methoxybenzoyl)amino]ethyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	COC1=C(C(=O)N[C@H](C)C2=CC=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2)C=CC=C1	C48H54N10O5	BTK	Q06187	CRBN	US-20240246977-A1
TPD-73IENL	SCHEMBL24598498	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[4-[(1R)-1-[(2-methoxynaphthalene-1-carbonyl)amino]ethyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide; SCHEMBL31030023	COC1=C(C(=O)N[C@H](C)C2=CC=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C=C2)C2=C(C=CC=C2)C=C1	C52H56N10O5	BTK	Q06187	CRBN	US-20240246977-A1
TPD-7SR6AF	SCHEMBL24598086	3-[3-(4,4-dimethyl-9-oxo-1,10-diazatricyclo[6.4.0.02,6]dodeca-2(6),7-dien-10-yl)-2-methylphenyl]-8-[3-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenoxy]propoxy]-6,11-dihydro-5H-imidazo[5,1-b][1,3]benzodiazepine-1-carboxamide	CC1=C(N2CCN3C(=CC4=C3CC(C)(C)C4)C2=O)C=CC=C1C1=NC(C(N)=O)=C2NC3=CC=C(OCCCOC4=CC=C(N5CCC(=O)NC5=O)C=C4)C=C3CCN12	C44H46N8O6	BTK	Q06187	CRBN	US-20240246977-A1
TPD-TC6UBY	SCHEMBL27342420	8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-[2-fluoro-5-methyl-4-[(6-methylpyridin-2-yl)carbamoyl]phenyl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepine-1-carboxamide	CC1=CC=CC(NC(=O)C2=C(C)C=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C(N)=O)C(F)=C2)=N1	C46H50FN11O4	BTK	Q06187	CRBN	US-20240246977-A1
TPD-C18YTB	SCHEMBL24598080	5-[1-cyano-8-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-6,11-dihydro-5H-pyrazolo[5,1-b][1,3]benzodiazepin-2-yl]-3-methyl-N-(6-methylpyridin-2-yl)pyridine-2-carboxamide; SCHEMBL31030029	CC1=NC(NC(=O)C2=C(C)C=C(C3=NN4CCC5=C(C=CC(N6CCN(CC7CCN(C8=CC=C(N9CCC(=O)NC9=O)C=C8)CC7)CC6)=C5)NC4=C3C#N)C=N2)=CC=C1	C45H48N12O3	BTK	Q06187	CRBN	US-20240246977-A1
TPD-GN1PPE	US20240246977A1_9A12	.	NC(=O)C1=C2NC3=C(C=C(C(=O)NC4CCN(CN5CCN(C6=C(F)C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C=C3)CCN2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C48H47FN10O7	BTK	Q06187	CRBN	US-20240246977-A1
TPD-QJ9G78	CHEMBL5396974	(2S,4S)-1-[(2S)-3,3-dimethyl-2-[3-[2-[methyl-[6-methyl-2-[4-[(2-phenylacetyl)amino]anilino]pyrimidin-4-yl]amino]ethoxy]propanoylamino]butanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL31032332	Cc1cc(N(C)CCOCCC(=O)N[C@H](C(=O)N2C[C@@H](O)C[C@H]2C(=O)NCc2ccc(-c3scnc3C)cc2)C(C)(C)C)nc(Nc2ccc(NC(=O)Cc3ccccc3)cc2)n1	C47H57N9O6S	TG2	P21980	VHL	US-20240287033-A1
TPD-3I746V	CHEMBL5437985	(2S,4S)-1-[(2S)-3,3-dimethyl-2-[3-[2-[2-[2-[2-[2-[methyl-[6-methyl-2-[4-[(2-phenylacetyl)amino]anilino]pyrimidin-4-yl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]propanoylamino]butanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL31032289	Cc1cc(N(C)CCOCCOCCOCCOCCOCCC(=O)N[C@H](C(=O)N2C[C@@H](O)C[C@H]2C(=O)NCc2ccc(-c3scnc3C)cc2)C(C)(C)C)nc(Nc2ccc(NC(=O)Cc3ccccc3)cc2)n1	C55H73N9O10S	TG2	P21980	VHL	US-20240287033-A1
TPD-72HOLP	SCHEMBL31032338	N-[4-[[4-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]amino]ethoxy]ethyl-methylamino]-6-methylpyrimidin-2-yl]amino]phenyl]-2-phenylacetamide	Cc1cc(N(C)CCOCCNc2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)nc(Nc2ccc(NC(=O)Cc3ccccc3)cc2)n1	C37H38N8O6	TG2	P21980	CRBN	US-20240287033-A1
TPD-WLOQ54	US20240287033A1_NUCC-0227324	.	Cc1cc(N(C)CCOCCOCCOCCNc2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)nc(Nc2ccc(NC(=O)Cc3ccccc3)cc2)n1	C41H46N8O8	TG2	P21980	CRBN	US-20240287033-A1
TPD-S065VI	US20240287033A1_NUCC-0227325	.	Cc1cc(N(C)CCOCCOCCOCCOCCOCCNc2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)nc(Nc2ccc(NC(=O)Cc3ccccc3)cc2)n1	C45H54N8O10	TG2	P21980	CRBN	US-20240287033-A1
TPD-RYXO1R	US20240287033A1_NUCC-0227350	.	Cc1cc(N(C)CCOCCOc2cc(-c3scnc3C)ccc2CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)C)nc(Nc2ccc(NC(=O)Cc3ccccc3)cc2)n1	C50H60FN9O7S	TG2	P21980	VHL	US-20240287033-A1
TPD-AWRW65	US20240287033A1_NUCC-0227351	.	Cc1cc(N(C)CCOCCOCCOc2cc(-c3scnc3C)ccc2CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)C)nc(Nc2ccc(NC(=O)Cc3ccccc3)cc2)n1	C52H64FN9O8S	TG2	P21980	VHL	US-20240287033-A1
TPD-A9PSEG	US20240287033A1_NUCC-0227352	.	Cc1cc(N(C)CCOCCOCCOCCOc2cc(-c3scnc3C)ccc2CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)C)nc(Nc2ccc(NC(=O)Cc3ccccc3)cc2)n1	C54H68FN9O9S	TG2	P21980	VHL	US-20240287033-A1
TPD-PY3VML	US20240287033A1_NUCC-0227374	.	Cc1cc(N(C)CCOCCOCCSC(C)(C)[C@H](NC(=O)C2(F)CC2)C(=O)N2C[C@H](O)C[C@H]2C(=O)NCc2ccc(-c3scnc3C)cc2)nc(Nc2ccc(NC(=O)Cc3ccccc3)cc2)n1	C51H62FN9O7S2	TG2	P21980	VHL	US-20240287033-A1
TPD-QNR1ZT	US20240287033A1_NUCC-0227404	.	Cc1cc(N(C)CCOCCOCCOCCSC(C)(C)[C@H](NC(=O)C2(F)CC2)C(=O)N2C[C@H](O)C[C@H]2C(=O)NCc2ccc(-c3scnc3C)cc2)nc(Nc2ccc(NC(=O)Cc3ccccc3)cc2)n1	C53H66FN9O8S2	TG2	P21980	VHL	US-20240287033-A1
TPD-E8E6S6	US20240287033A1_NUCC-0227405	.	Cc1cc(N(C)CCOCCSC(C)(C)[C@H](NC(=O)C2(F)CC2)C(=O)N2C[C@H](O)C[C@H]2C(=O)NCc2ccc(-c3scnc3C)cc2)nc(Nc2ccc(NC(=O)Cc3ccccc3)cc2)n1	C49H58FN9O6S2	TG2	P21980	VHL	US-20240287033-A1
TPD-UE0MGQ	US20240287033A1_NUCC-0228723	.	Cc1cc(N(C)CCCCCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCc2ccc(-c3scnc3C)cc2)C(C)(C)C)nc(Nc2ccc(NC(=O)Cc3ccccc3)cc2)n1	C48H59N9O5S	TG2	P21980	VHL	US-20240287033-A1
TPD-N4I1G7	US20240287033A1_NUCC-0228741	.	Cc1cc(N(C)CCCCCCCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCc2ccc(-c3scnc3C)cc2)C(C)(C)C)nc(Nc2ccc(NC(=O)Cc3ccccc3)cc2)n1	C50H63N9O5S	TG2	P21980	VHL	US-20240287033-A1
TPD-O8KMV6	US20240287101A1_1	.	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CC4CCC(C1)N4)=NC(OCCN1CCC(CN4CC5(C4)CN(C4=CC6=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)C5)CC1)=N3)=CC(O)=C2	C51H55FN10O6	KRAS	P01116	CRBN	US-20240287101-A1
TPD-T6LK61	US20240287101A1_2	3-[6-[2-[[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]-2,7-diazaspiro[3.5]nonan-7-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CC4CCC(C1)N4)=NC(OCCN1CCC(CN4CC5(CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)CC5)C4)CC1)=N3)=CC(O)=C2	C53H61FN10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-6OFMGM	US20240287101A1_3	3-[7-[7-[[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]-2,7-diazaspiro[3.5]nonan-2-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CC4CCC(C1)N4)=NC(OCCN1CCC(CN4CCC5(CC4)CN(C4=C6CN(C7CCC(=O)NC7=O)C(=O)C6=CC=C4)C5)CC1)=N3)=CC(O)=C2	C53H61FN10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-K88OED	US20240287101A1_4	5-[3-[2-[4-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperazin-1-yl]ethyl-methylamino]cyclobutyl]oxy-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CC4CCC(C1)N4)=NC(OCCN1CCN(CCN(C)[C@H]4C[C@H](OC5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC1)=N3)=CC(O)=C2	C51H57FN10O7	KRAS	P01116	CRBN	US-20240287101-A1
TPD-44VJMG	US20240287101A1_5	.	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CC4CCC(C1)N4)=NC(OCCN1CCN(C4=NC=NC(N5CCN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)=C4)CC1)=N3)=CC(O)=C2	C52H54FN13O6	KRAS	P01116	CRBN	US-20240287101-A1
TPD-3PRKDE	US20240287101A1_6	.	CCC1=CC=CC2=C1C(C1=C(N)C3=C(C=N1)C(N1CC4CCC(C1)N4)=NC(OCCN1CCN(CC4CCN(C(=O)C5=CC=C(OC)C(N6CCC(=O)NC6=O)=C5)CC4)CC1)=N3)=CC(O)=C2	C49H59N11O6	KRAS	P01116	CRBN	US-20240287101-A1
TPD-5L122B	US20240287101A1_7	6-[4-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)-4-methoxyisoindole-1,3-dione	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CC4CCC(C1)N4)=NC(OCCN1CCN(C4=CC(OC)=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC1)=N3)=CC(O)=C2	C45H46FN9O7	KRAS	P01116	CRBN	US-20240287101-A1
TPD-02EGRP	US20240287101A1_8	5-[1-[[1-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-4-yl]oxy-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CC4CCC(C1)N4)=NC(OCCN1CCC(CN4CCC(OC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC1)=N3)=CC(O)=C2	C51H56FN9O7	KRAS	P01116	CRBN	US-20240287101-A1
TPD-IRPP7U	US20240287101A1_9	3-[7-[4-[[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CCC1=CC=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCCN5CCC(CN6CCN(C7=CC=CC8=C7CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)=NC4=C3F)=C21	C50H57FN10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-ZVICTJ	US20240287101A1_10	5-[4-[3-[1-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]propyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CC4CCC(C1)N4)=NC(OCCN1CCC(CCCN4CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC1)=N3)=CC(O)=C2	C52H59FN10O6	KRAS	P01116	CRBN	US-20240287101-A1
TPD-F49OG3	US20240287101A1_11	.	CCC1=CC=CC(/C=C(O)\C=C\C2=C(F)C3=C(C=N2)C(N2CC4CCC(C2)N4)=NC(OCCN2CCC(CN(C)[C@H]4C[C@H](OC5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC2)=N3)=C1	C51H58FN9O7	KRAS	P01116	CRBN	US-20240287101-A1
TPD-L0QB46	US20240287101A1_12	5-[4-[2-[1-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]ethyl]piperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CC4CCC(C1)N4)=NC(OCCN1CCC(CCC4CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC1)=N3)=CC(O)=C2	C52H58FN9O6	KRAS	P01116	CRBN	US-20240287101-A1
TPD-CKTMWA	US20240287101A1_13	5-[4-[2-[1-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]propan-2-yl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CC4CCC(C1)N4)=NC(OCCN1CCC(C(C)(C)N4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC1)=N3)=CC(O)=C2	C52H59FN10O6	KRAS	P01116	CRBN	US-20240287101-A1
TPD-DDXBB5	US20240287101A1_14	.	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CC4CCC(C1)N4)=NC(OCCN1CCN(CC4CCN(C5=CC(F)=C(N6CCC(=O)NC6=O)C=C5)CC4)CC1)=N3)=CC(O)=C2	C47H54F2N10O4	KRAS	P01116	CRBN	US-20240287101-A1
TPD-W4P07X	US20240287101A1_15	.	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CC4CCC(C1)N4)=NC(OCCN1CCN(CC4CCN(C5=CC=C(OC)C(C(=O)NC6CCC(=O)NC6=O)=C5)CC4)CC1)=N3)=CC(O)=C2	C50H59FN10O6	KRAS	P01116	CRBN	US-20240287101-A1
TPD-WL36AJ	US20240287101A1_16	.	CCC1=CC=CC2=C1C(C1=C(F)C3=C(CN1)C(N1CC4CCC(C1)N4)=NC(OCCN1CCC(CN4C=CC=C(CN5CCC(=O)NC5=O)C4=O)CC1)=N3)=CC(O)=C2	C43H50FN9O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-CFC2WY	US20240287101A1_17	5-[4-[[4-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperazin-1-yl]methyl]piperidin-1-yl]-N-(2,6-dioxopiperidin-3-yl)-2-fluorobenzamide	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CC4CCC(C1)N4)=NC(OCCN1CCN(CC4CCN(C5=CC=C(F)C(C(=O)NC6CCC(=O)NC6=O)=C5)CC4)CC1)=N3)=CC(O)=C2	C49H56F2N10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-6MBSPI	US20240287101A1_18	4-[1-[[1-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-4-yl]oxy-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CC4CCC(C1)N4)=NC(OCCN1CCC(CN4CCC(OC5=CC=CC6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC1)=N3)=CC(O)=C2	C51H56FN9O7	KRAS	P01116	CRBN	US-20240287101-A1
TPD-QGNLF1	US20240287101A1_19	.	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CC4CCC(C1)N4)=NC(OCCN1CCC4(CC1)CCN(C1=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C1)CC4)=N3)=CC(O)=C2	C49H52FN9O6	KRAS	P01116	CRBN	US-20240287101-A1
TPD-AV27N3	US20240287101A1_20	5-[4-[[4-[[1-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperazin-1-yl]methyl]piperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CC4CCC(C1)N4)=NC(OCCN1CCC(CN4CCN(CC5CCN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)CC1)=N3)=CC(O)=C2	C56H66FN11O6	KRAS	P01116	CRBN	US-20240287101-A1
TPD-UANFZ3	US20240287101A1_21	5-[4-[[4-[[4-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]morpholin-2-yl]methyl]piperazin-1-yl]methyl]piperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CC4CCC(C1)N4)=NC(OCCN1CCOC(CN4CCN(CC5CCN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)C1)=N3)=CC(O)=C2	C55H64FN11O7	KRAS	P01116	CRBN	US-20240287101-A1
TPD-HHVF58	US20240287101A1_22	5-[9-[[1-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CC4CCC(C1)N4)=NC(OCCN1CCC(CN4CCC5(CC4)CCN(C4=CC6=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC5)CC1)=N3)=CC(O)=C2	C55H63FN10O6	KRAS	P01116	CRBN	US-20240287101-A1
TPD-23OLRL	US20240287101A1_23	3-[7-[4-[4-[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]oxycyclohexyl]oxypiperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CCC1=CC=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCCN5CCC(O[C@H]6CC[C@H](OC7CCN(C8=CC=CC9=C8CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)=NC4=C3F)=C21	C56H66FN9O7	KRAS	P01116	CRBN	US-20240287101-A1
TPD-U8Q1CA	US20240287101A1_24	3-[7-[4-[3-[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]oxycyclobutyl]oxypiperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CCC1=CC=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCCN5CCC(O[C@H]6C[C@H](OC7CCN(C8=CC=CC9=C8CN(C8CCC(=O)NC8=O)C9=O)CC7)C6)CC5)=NC4=C3F)=C21	C54H62FN9O7	KRAS	P01116	CRBN	US-20240287101-A1
TPD-N5DW64	US20240287101A1_25	5-[4-[[9-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]-3,9-diazaspiro[5.5]undecan-3-yl]methyl]piperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CC4CCC(C1)N4)=NC(OCCN1CCC4(CC1)CCN(CC1CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC1)CC4)=N3)=CC(O)=C2	C55H63FN10O6	KRAS	P01116	CRBN	US-20240287101-A1
TPD-JRVDGM	US20240287101A1_26	5-[4-[[1-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methoxymethyl]piperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CC4CCC(C1)N4)=NC(OCCN1CCC(COCC4CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC1)=N3)=CC(O)=C2	C52H58FN9O7	KRAS	P01116	CRBN	US-20240287101-A1
TPD-WJJ6J0	US20240287101A1_27	5-[4-[1-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]piperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CC4CCC(C1)N4)=NC(OCCN1CCC(C4CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC1)=N3)=CC(O)=C2	C50H54FN9O6	KRAS	P01116	CRBN	US-20240287101-A1
TPD-LNA722	SCHEMBL31129401	3-[4-[4-[[1-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-1-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	CCC1=CC=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCCN5CCC(CC6CCN(C7=CC=CC8=C7N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC5)=NC4=C3F)=C21	C51H59FN10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-LO4VPK	US20240287101A1_29	3-[7-[4-[[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]-4-fluoropiperidin-4-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CCC1=CC=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCCN5CCC(F)(CC6CCN(C7=CC=CC8=C7CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)=NC4=C3F)=C21	C51H57F2N9O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-1HGRQR	US20240287101A1_30	3-[7-[4-[[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]-3-methylpiperidine-2,6-dione	CCC1=CC=CC2=CC(O)=CC(C3=C(F)C4=NC(OCCN5CCC(CC6CCN(C7=CC=CC8=C7CN(C7(C)CCC(=O)NC7=O)C8=O)CC6)CC5)=NC(N5CC6CCC(C5)N6)=C4C=N3)=C21	C52H60FN9O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-HJ6WUX	US20240287101A1_31	.	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CC4CCC(C1)N4)=NC(OCCN1CCC(CCN4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC1)=N3)=CC(O)=C2	C51H57FN10O6	KRAS	P01116	CRBN	US-20240287101-A1
TPD-57Z33O	US20240287101A1_32	5-[4-[[1-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CC4CCC(C1)N4)=NC(OCCN1CCC(CN4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC1)=N3)=CC(O)=C2	C50H55FN10O6	KRAS	P01116	CRBN	US-20240287101-A1
TPD-0IYWAH	US20240287101A1_33	.	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CC4CCC(C1)N4)=NC(OCCN1CCN([C@H]4CC[C@H](NC5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC1)=N3)=CC(O)=C2	C50H55FN10O6	KRAS	P01116	CRBN	US-20240287101-A1
TPD-8W1LYV	US20240287101A1_34	5-[1-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CC4CCC(C1)N4)=NC(OCCN1CCC(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC1)=N3)=CC(O)=C2	C45H45FN8O6	KRAS	P01116	CRBN	US-20240287101-A1
TPD-V7C9UD	SCHEMBL31129361	3-[7-[4-[[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCCN5CCC(CC6CCN(C7=CC=CC8=C7CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)=NC4=C3F)=C21	C51H53F2N9O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-0KAGOR	SCHEMBL31129381	3-[5-[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CC4CCC(C1)N4)=NC(OCCN1CCC(C4=CC=C5CN(C6CCC(=O)NC6=O)C(=O)C5=C4)CC1)=N3)=CC(O)=C2	C45H47FN8O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-A27P01	US20240287101A1_37	4-[4-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperazin-1-yl]-N-(2,6-dioxopiperidin-3-yl)-2-fluorobenzamide	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CC4CCC(C1)N4)=NC(OCCN1CCN(C4=CC(F)=C(C(=O)NC5CCC(=O)NC5=O)C=C4)CC1)=N3)=CC(O)=C2	C43H45F2N9O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-RJMQPP	US20240287101A1_38	3-[6-[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CC4CCC(C1)N4)=NC(OCCN1CCC(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5)CC1)=N3)=CC(O)=C2	C45H47FN8O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-6U19M4	US20240287101A1_39	3-[6-[4-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CC4CCC(C1)N4)=NC(OCCN1CCN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5)CC1)=N3)=CC(O)=C2	C44H46FN9O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-ZJ3X8M	US20240287101A1_40	.	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CC4CCC(C1)N4)=NC(OCCN1CCN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC1)=N3)=CC(O)=C2	C44H44FN9O6	KRAS	P01116	CRBN	US-20240287101-A1
TPD-U210OU	SCHEMBL31129400	3-[7-[4-[[1-[2-[7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoro-4-(8-methyl-3,8-diazabicyclo[3.2.1]octan-3-yl)pyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CCC1=CC=CC2=CC(O)=CC(C3=C(F)C4=NC(OCCN5CCC(CC6CCN(C7=CC=CC8=C7CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)=NC(N5CC6CCC(C5)N6C)=C4C=N3)=C21	C52H60FN9O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-MEK3NP	SCHEMBL31129731	3-[7-[4-[[4-[[1-[2-[7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoro-4-(8-methyl-3,8-diazabicyclo[3.2.1]octan-3-yl)pyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-1-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CCC1=CC=CC2=CC(O)=CC(C3=C(F)C4=NC(OCCN5CCC(CC6CCN(CC7CCN(C8=CC=CC9=C8CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)=NC(N5CC6CCC(C5)N6C)=C4C=N3)=C21	C58H71FN10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-LD9W6T	SCHEMBL31129462	3-[7-[4-[[4-[[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-1-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=NC(OCCN5CCC(CC6CCN(CC7CCN(C8=CC=CC9=C8CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)=NC(N5CC6CCC(C5)N6)=C4C=N3)=C21	C57H64F2N10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-QCSWGB	US20240287101A1_44	3-[7-[4-[[4-[[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-1-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]-3-methylpiperidine-2,6-dione	CCC1=CC=CC2=CC(O)=CC(C3=C(F)C4=NC(OCCN5CCC(CC6CCN(CC7CCN(C8=CC=CC9=C8CN(C8(C)CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)=NC(N5CC6CCC(C5)N6)=C4C=N3)=C21	C58H71FN10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-KLZURP	US20240287101A1_45	3-[7-[4-[[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]-1-methylpiperidine-2,6-dione	CCC1=CC=CC2=CC(O)=CC(C3=C(F)C4=NC(OCCN5CCC(CC6CCN(C7=CC=CC8=C7CN(C7CCC(=O)N(C)C7=O)C8=O)CC6)CC5)=NC(N5CC6CCC(C5)N6)=C4C=N3)=C21	C52H60FN9O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-UPAVR5	US20240287101A1_46	3-[7-[4-[[4-[[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-1-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]-1-methylpiperidine-2,6-dione	CCC1=CC=CC2=CC(O)=CC(C3=C(F)C4=NC(OCCN5CCC(CC6CCN(CC7CCN(C8=CC=CC9=C8CN(C8CCC(=O)N(C)C8=O)C9=O)CC7)CC6)CC5)=NC(N5CC6CCC(C5)N6)=C4C=N3)=C21	C58H71FN10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-V08AON	US20240287101A1_47	[(3S,8S)-8-[[7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoro-4-(8-methyl-3,8-diazabicyclo[3.2.1]octan-3-yl)pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazine-1-carboxylate	CCC1=CC=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6C)=NC(OC[C@@]56CCCN5[C@H](COC(=O)N5CCN(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8)CC5)CC6)=NC4=C3F)=C21	C53H59FN10O7	KRAS	P01116	CRBN	US-20240287101-A1
TPD-7U6A42	US20240287101A1_48	[(3R,8R)-8-[[7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoro-4-(8-methyl-3,8-diazabicyclo[3.2.1]octan-3-yl)pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazine-1-carboxylate	CCC1=CC=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6C)=NC(OC[C@]56CCCN5[C@@H](COC(=O)N5CCN(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8)CC5)CC6)=NC4=C3F)=C21	C53H59FN10O7	KRAS	P01116	CRBN	US-20240287101-A1
TPD-TEZZO8	US20240287101A1_49	[(3S,8S)-8-[[7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoro-4-(8-methyl-3,8-diazabicyclo[3.2.1]octan-3-yl)pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]piperazine-1-carboxylate	CCC1=CC=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6C)=NC(OC[C@@]56CCCN5[C@H](COC(=O)N5CCN(C7=C8CN(C9CCC(=O)NC9=O)C(=O)C8=CC=C7)CC5)CC6)=NC4=C3F)=C21	C53H59FN10O7	KRAS	P01116	CRBN	US-20240287101-A1
TPD-B3JJRL	US20240287101A1_50	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 4-[2-(1-methyl-2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazine-1-carboxylate	[H]N1C2CCC1CN(C1=NC(OC[C@@]34CCCN3[C@H](COC(=O)N3CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)N(C)C5=O)C6)CC3)CC4)=NC3=C(F)C(C4=C5C(=CC(O)=C4)C=CC=C5CC)=NC=C13)C2	C53H59FN10O7	KRAS	P01116	CRBN	US-20240287101-A1
TPD-0U8K1A	US20240287101A1_51	[(3R,8R)-8-[[7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoro-4-(8-methyl-3,8-diazabicyclo[3.2.1]octan-3-yl)pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]piperazine-1-carboxylate	CCC1=CC=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6C)=NC(OC[C@]56CCCN5[C@@H](COC(=O)N5CCN(C7=C8CN(C9CCC(=O)NC9=O)C(=O)C8=CC=C7)CC5)CC6)=NC4=C3F)=C21	C53H59FN10O7	KRAS	P01116	CRBN	US-20240287101-A1
TPD-8C9JZ9	US20240287101A1_52	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 4-[2-(1-methyl-2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]piperazine-1-carboxylate	[H]N1C2CCC1CN(C1=NC(OC[C@@]34CCCN3[C@H](COC(=O)N3CCN(C5=C6CN(C7CCC(=O)N(C)C7=O)C(=O)C6=CC=C5)CC3)CC4)=NC3=C(F)C(C4=C5C(=CC(O)=C4)C=CC=C5CC)=NC=C13)C2	C53H59FN10O7	KRAS	P01116	CRBN	US-20240287101-A1
TPD-AV7C80	US20240287101A1_53	[(3R,8R)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazine-1-carboxylate	[H]N1C2CCC1CN(C1=NC(OC[C@]34CCCN3[C@@H](COC(=O)N3CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6)CC3)CC4)=NC3=C(F)C(C4=C5C(=CC(O)=C4)C=CC=C5CC)=NC=C13)C2	C52H57FN10O7	KRAS	P01116	CRBN	US-20240287101-A1
TPD-DEXL0Z	US20240287101A1_54	[(3R,8R)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 4-[2-(1-methyl-2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]piperazine-1-carboxylate	[H]N1C2CCC1CN(C1=NC(OC[C@]34CCCN3[C@@H](COC(=O)N3CCN(C5=C6CN(C7CCC(=O)N(C)C7=O)C(=O)C6=CC=C5)CC3)CC4)=NC3=C(F)C(C4=C5C(=CC(O)=C4)C=CC=C5CC)=NC=C13)C2	C53H59FN10O7	KRAS	P01116	CRBN	US-20240287101-A1
TPD-KSJ0ZP	SCHEMBL31129514	3-[7-[4-[[4-[[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-1-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CCC1=CC=CC2=CC(O)=CC(C3=C(F)C4=NC(OCCN5CCC(CC6CCN(CC7CCN(C8=CC=CC9=C8CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)=NC(N5CC6CCC(C5)N6)=C4C=N3)=C21	C57H69FN10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-OOK3ID	SCHEMBL31129442	3-[7-[4-[[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CCC1=CC=CC2=CC(O)=CC(C3=C(F)C4=NC(OCCN5CCC(CC6CCN(C7=CC=CC8=C7CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)=NC(N5CC6CCC(C5)N6)=C4C=N3)=C21	C51H58FN9O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-6IIMHY	SCHEMBL31129686	4-[4-[[4-[[1-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-1-yl]methyl]piperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	[H]N1C2CCC1CN(C1=C3C=NC(C4=C5C(=CC(O)=C4)C=CC=C5CC)=C(F)C3=NC(OCCN3CCC(CC4CCN(CC5CCN(C6=CC=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)CC3)=N1)C2	C57H67FN10O6	KRAS	P01116	CRBN	US-20240287101-A1
TPD-68FXM3	US20240287101A1_58	.	[H]N1C2CCC1CN(C1NC(OC[C@@]34CCCN3[C@H](COC(=O)N3CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6)CC3)CC4)=NC3=C(F)C(C4=C5C(=CC(O)=C4)C=CC=C5CC)=NC=C31)C2	C52H59FN10O7	KRAS	P01116	CRBN	US-20240287101-A1
TPD-PZIA8S	US20240287101A1_60	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]piperazine-1-carboxylate	[H]N1C2CCC1CN(C1=NC(OC[C@@]34CCCN3[C@H](COC(=O)N3CCN(C5=C6CN(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)CC3)CC4)=NC3=C(F)C(C4=C5C(=CC(O)=C4)C=CC=C5CC)=NC=C13)C2	C52H57FN10O7	KRAS	P01116	CRBN	US-20240287101-A1
TPD-EOD51F	US20240287101A1_61	.	[H]N1C2CCC1CN(C1=NC(OC[C@]34CCCN3[C@@H](COC(=O)N3CCN(C5=C6CN(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)CC3)CC4)=NC3=C(F)C(C4=C5C(CC)=CC=CC5CC(O)=C4)=NC=C13)C2	C52H59FN10O7	KRAS	P01116	CRBN	US-20240287101-A1
TPD-TPAJXW	US20240287101A1_62	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazine-1-carboxylate	[H]N1C2CCC1CN(C1=NC(OC[C@@]34CCCN3[C@H](COC(=O)N3CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC3)CC4)=NC3=C(F)C(C4=C5C(=CC(O)=C4)C=CC=C5CC)=NC=C13)C2	C52H55FN10O8	KRAS	P01116	CRBN	US-20240287101-A1
TPD-D6LLOK	US20240287101A1_63	.	[H]N1C2CCC1CN(C1=NC(OC[C@]34CCCN3C(OC(=O)N3CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)N(I)C5=O)C6=O)CC3)CC4)=NC3=C(F)C(C4=C5C(=CC(O)=C4)C=CC=C5CC)=NC=C13)C2	C51H52FIN10O8	KRAS	P01116	CRBN	US-20240287101-A1
TPD-J8KJTR	US20240287101A1_64	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperazine-1-carboxylate	[H]N1C2CCC1CN(C1=NC(OC[C@@]34CCCN3[C@H](COC(=O)N3CCN(C5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)CC3)CC4)=NC3=C(F)C(C4=C5C(=CC(O)=C4)C=CC=C5CC)=NC=C13)C2	C52H55FN10O8	KRAS	P01116	CRBN	US-20240287101-A1
TPD-YRB2RE	US20240287101A1_65	[(3R,8R)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperazine-1-carboxylate	[H]N1C2CCC1CN(C1=NC(OC[C@]34CCCN3[C@@H](COC(=O)N3CCN(C5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)CC3)CC4)=NC3=C(F)C(C4=C5C(=CC(O)=C4)C=CC=C5CC)=NC=C13)C2	C52H55FN10O8	KRAS	P01116	CRBN	US-20240287101-A1
TPD-2ZETZ3	SCHEMBL31129524	4-[4-[[1-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	[H]N1C2CCC1CN(C1=NC(OCCN3CCC(CC4CCN(C5=CC=CC6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)=NC3=C(F)C(C4=CC(O)=CC5=C4C(CC)=CC=C5)=NC=C13)C2	C51H56FN9O6	KRAS	P01116	CRBN	US-20240287101-A1
TPD-GDQDNK	US20240287101A1_67	.	[H]N1C2CCC1CN(C1=NC(OCCN3CCC(CC4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6C5)CC4)CC3)=NC3=C(F)C(C4=CC(O)=CC5=C4C(CC)=CC=C5)=NC=C13)C2	C51H58FN9O6	KRAS	P01116	CRBN	US-20240287101-A1
TPD-CG7LEG	US20240287101A1_68	3-[6-[4-[[4-[[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-1-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=NC(OCCN5CCC(CC6CCN(CC7CCN(C8=CC=C9C(=O)N(C%10CCC(=O)NC%10=O)CC9=C8)CC7)CC6)CC5)=NC(N5CC6CCC(C5)N6)=C4C=N3)=C21	C57H64F2N10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-TT5SIC	orb2802253	3-[6-[4-[[4-[[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-1-yl]methyl]piperidin-1-yl]-7-fluoro-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31129346; 3052745-16-8	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=NC(OCCN5CCC(CC6CCN(CC7CCN(C8=CC=C9C(=O)N(C%10CCC(=O)NC%10=O)CC9=C8F)CC7)CC6)CC5)=NC(N5CC6CCC(C5)N6)=C4C=N3)=C21	C57H63F3N10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-DB173P	US20240287101A1_70	3-[6-[4-[[9-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]-3,9-diazaspiro[5.5]undecan-3-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=NC(OCCN5CCC6(CC5)CCN(CC5CCN(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8)CC5)CC6)=NC(N5CC6CCC(C5)N6)=C4C=N3)=C21	C55H60F2N10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-QFOIZZ	US20240287101A1_71	3-[6-[4-[[4-[(3R,5S)-5-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1-methylpyrrolidin-3-yl]oxypiperidin-1-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CCC1=CC=CC2=CC(O)=CC(C3=C(F)C4=NC(OC[C@@H]5C[C@@H](OC6CCN(CC7CCN(C8=CC=C9C(=O)N(C%10CCC(=O)NC%10=O)CC9=C8)CC7)CC6)CN5C)=NC(N5CC6CCC(C5)N6)=C4C=N3)=C21	C55H65FN10O6	KRAS	P01116	CRBN	US-20240287101-A1
TPD-KNMIFV	US20240287101A1_72	.	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=NC(OCCN5CCC(CN6CC7(CCN(C8=CC9=C(C=C8)C(=O)N(C8CCC(=O)NC8=O)C9)CC7)C6)CC5)=NC(N5CC6CCC(C5)N6)=C4C=N3)C21	C53H58F2N10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-W7WWLJ	US20240287101A1_73	3-[6-[4-[[4-[(3R,5S)-5-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1-methylpyrrolidin-3-yl]oxypiperidin-1-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=NC(OC[C@@H]5C[C@@H](OC6CCN(CC7CCN(C8=CC=C9C(=O)N(C%10CCC(=O)NC%10=O)CC9=C8)CC7)CC6)CN5C)=NC(N5CC6CCC(C5)N6)=C4C=N3)=C21	C55H60F2N10O6	KRAS	P01116	CRBN	US-20240287101-A1
TPD-HJUALJ	US20240287101A1_74	5-[4-[[4-[[1-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-1-yl]methyl]piperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=NC(OCCN5CCC(CC6CCN(CC7CCN(C8=CC=C9C(=O)N(C%10CCC(=O)NC%10=O)C(=O)C9=C8)CC7)CC6)CC5)=NC(N5CC6CCC(C5)N6)=C4C=N3)=C21	C57H62F2N10O6	KRAS	P01116	CRBN	US-20240287101-A1
TPD-MMWOWI	US20240287101A1_75	4-[4-[[4-[[1-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-1-yl]methyl]piperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=NC(OCCN5CCC(CC6CCN(CC7CCN(C8=CC=CC9=C8C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)=NC(N5CC6CCC(C5)N6)=C4C=N3)=C21	C57H62F2N10O6	KRAS	P01116	CRBN	US-20240287101-A1
TPD-0FSLGV	US20240287101A1_76	5-[4-[[9-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]-3,9-diazaspiro[5.5]undecan-3-yl]methyl]piperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=NC(OCCN5CCC6(CC5)CCN(CC5CCN(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC5)CC6)=NC(N5CC6CCC(C5)N6)=C4C=N3)=C21	C55H58F2N10O6	KRAS	P01116	CRBN	US-20240287101-A1
TPD-QGWJ3P	US20240287101A1_77	3-[6-[4-[(3R,5S)-5-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1-methylpyrrolidin-3-yl]oxypiperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CCC1=CC=CC2=CC(O)=CC(C3=C(F)C4=NC(OC[C@@H]5C[C@@H](OC6CCN(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8)CC6)CN5C)=NC(N5CC6CCC(C5)N6)=C4C=N3)=C21	C49H54FN9O6	KRAS	P01116	CRBN	US-20240287101-A1
TPD-HXUYXG	US20240287101A1_78	3-[6-[4-[(3R,5S)-5-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1-methylpyrrolidin-3-yl]oxypiperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=NC(OC[C@@H]5C[C@@H](OC6CCN(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8)CC6)CN5C)=NC(N5CC6CCC(C5)N6)=C4C=N3)=C21	C49H49F2N9O6	KRAS	P01116	CRBN	US-20240287101-A1
TPD-KXDNXH	SCHEMBL31129666	3-[6-[4-[[4-[[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]-difluoromethyl]piperidin-1-yl]methyl]piperidin-1-yl]-7-fluoro-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCCN5CCC(C(F)(F)C6CCN(CC7CCN(C8=CC=C9C(=O)N(C%10CCC(=O)NC%10=O)CC9=C8F)CC7)CC6)CC5)=NC4=C3F)=C21	C57H61F5N10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-UCZD2X	SCHEMBL31129736	3-[5-[4-[[1-[[1-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-4-yl]methyl]piperidin-1-yl]-2-oxo-3-propan-2-ylbenzimidazol-1-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OCCN4CCC(CN5CCC(CC6CCN(C7=CC8=C(C=C7)N(C7CCC(=O)NC7=O)C(=O)N8C(C)C)CC6)CC5)CC4)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC(O)=C2	C59H69F2N11O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-19X5F4	SCHEMBL31129500	3-[7-chloro-6-[4-[[1-[[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-4-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	[H]N1C2CCC1CN(C1=C3C=NC(C4=CC(O)=CC5=C4C(C#C)=C(F)C=C5)=C(F)C3=NC(OCCN3CCC(CN4CCC(CC5CCN(C6=C(Cl)C7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)CC5)CC4)CC3)=N1)C2	C57H63ClF2N10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-WLM3I0	SCHEMBL31129380	3-[5-[4-[[1-[[1-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-4-yl]methyl]piperidin-1-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	[H]N1C2CCC1CN(C1=C3C=NC(C4=CC(O)=CC5=C4C(C#C)=C(F)C=C5)=C(F)C3=NC(OCCN3CCC(CN4CCC(CC5CCN(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC5)CC4)CC3)=N1)C2	C57H65F2N11O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-1YVOIU	SCHEMBL31129646	3-[4-[4-[[9-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]-3,9-diazaspiro[5.5]undecan-3-yl]methyl]piperidin-1-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCCN5CCC6(CC5)CCN(CC5CCN(C7=C8C(=CC=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)CC5)CC6)=NC4=C3F)=C21	C55H61F2N11O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-BVQQCB	US20240287101A1_84	.	[H]N1C2CCC1CN(C1=NC(OC[C@]34CCCN3[C@H](CN3CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7C6)CC5)CC3)CC4)=NC3=C(F)C(C4=CC(O)=CC5=C4C(C#C)=C(F)C=C5)=NC=C13)C2	C57H65F2N11O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-FL0YKF	SCHEMBL31129397	3-[6-[4-[[4-[(3R,5S)-5-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1-methylpyrrolidin-3-yl]oxypiperidin-1-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CCC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OC[C@@H]5C[C@@H](OC6CCN(CC7CCN(C8=CC9=C(C=C8)C(=O)N(C8CCC(=O)NC8=O)C9)CC7)CC6)CN5C)=NC4=C3F)=C21	C55H64F2N10O6	KRAS	P01116	CRBN	US-20240287101-A1
TPD-1II0JK	SCHEMBL31129480	3-[6-[4-[[4-[[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-1-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CCC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCCN5CCC(CC6CCN(CC7CCN(C8=CC=C9C(=O)N(C%10CCC(=O)NC%10=O)CC9=C8)CC7)CC6)CC5)=NC4=C3F)=C21	C57H68F2N10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-Q2WEYB	SCHEMBL31129367	3-[6-[4-[[1-[[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-4-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCCN5CCC(CN6CCC(CC7CCN(C8=CC=C9C(=O)N(C%10CCC(=O)NC%10=O)CC9=C8)CC7)CC6)CC5)=NC4=C3F)=C21	C57H64F2N10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-KRBKAY	US20240287101A1_88	.	C#CC1=C(N)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCCN5CCC(CN6CCC(CC7CCN(C8=CC=C9C(=O)N(C%10CCC(=O)NC%10=O)CC9=C8F)CC7)CC6)CC5)=NC4=C3F)=C21	C57H65F2N11O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-VAWW17	SCHEMBL31129439	3-[5-[4-[[1-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-1-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione; SCHEMBL31129450	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCCN5CCC(CC6CCN(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC5)=NC4=C3F)=C21	C51H54F2N10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-I74NY7	SCHEMBL31129385	3-[6-[4-[[4-[[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]-4-fluoropiperidin-1-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCCN5CCC(CC6(F)CCN(CC7CCN(C8=CC=C9C(=O)N(C%10CCC(=O)NC%10=O)CC9=C8)CC7)CC6)CC5)=NC4=C3F)=C21	C57H63F3N10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-TL1AUI	SCHEMBL31129431	3-[6-[4-[[4-[[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]-4-fluoropiperidin-4-yl]methyl]piperidin-1-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCCN5CCC(F)(CC6CCN(CC7CCN(C8=CC=C9C(=O)N(C%10CCC(=O)NC%10=O)CC9=C8)CC7)CC6)CC5)=NC4=C3F)=C21	C57H63F3N10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-B48E9S	SCHEMBL31129627	3-[6-[9-[[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]-3,9-diazaspiro[5.5]undecan-3-yl]-7-fluoro-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCCN5CCC(CN6CCC7(CC6)CCN(C6=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C6F)CC7)CC5)=NC4=C3F)=C21	C55H59F3N10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-8L5JX6	SCHEMBL31129662	3-[6-[9-[[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]-3,9-diazaspiro[5.5]undecan-3-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCCN5CCC(CN6CCC7(CC6)CCN(C6=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C6)CC7)CC5)=NC4=C3F)=C21	C55H60F2N10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-JDYH2G	SCHEMBL31129589	3-[4-[4-[[4-[[1-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-1-yl]methyl]piperidin-1-yl]-2-oxo-3-propan-2-ylbenzimidazol-1-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCCN5CCC(CC6CCN(CC7CCN(C8=C9C(=CC=C8)N(C8CCC(=O)NC8=O)C(=O)N9C(C)C)CC7)CC6)CC5)=NC4=C3F)=C21	C59H69F2N11O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-U2I4PX	SCHEMBL31129507	3-[5-[4-[[4-[(3R,5S)-5-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1-methylpyrrolidin-3-yl]oxypiperidin-1-yl]methyl]piperidin-1-yl]-2-oxo-3-propan-2-ylbenzimidazol-1-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OC[C@@H]5C[C@@H](OC6CCN(CC7CCN(C8=CC9=C(C=C8)N(C8CCC(=O)NC8=O)C(=O)N9C(C)C)CC7)CC6)CN5C)=NC4=C3F)=C21	C57H65F2N11O6	KRAS	P01116	CRBN	US-20240287101-A1
TPD-458Z7V	SCHEMBL31129477	3-[5-[4-[[4-[(3R,5S)-5-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1-methylpyrrolidin-3-yl]oxypiperidin-1-yl]methyl]piperidin-1-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OC[C@@H]5C[C@@H](OC6CCN(CC7CCN(C8=CC9=C(C=C8)N(C8CCC(=O)NC8=O)C(=O)N9C)CC7)CC6)CN5C)=NC4=C3F)=C21	C55H61F2N11O6	KRAS	P01116	CRBN	US-20240287101-A1
TPD-FSH3GZ	US20240287101A1_97	3-[6-[4-[[4-[[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-1-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]-3-methylpiperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCCN5CCC(CC6CCN(CC7CCN(C8=CC=C9C(=O)N(C%10(C)CCC(=O)NC%10=O)CC9=C8)CC7)CC6)CC5)=NC4=C3F)=C21	C58H66F2N10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-CDCJFV	SCHEMBL31129374	3-[5-[4-[[4-[[1-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-1-yl]methyl]piperidin-1-yl]-2-oxo-3-propan-2-ylbenzimidazol-1-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCCN5CCC(CC6CCN(CC7CCN(C8=CC9=C(C=C8)N(C8CCC(=O)NC8=O)C(=O)N9C(C)C)CC7)CC6)CC5)=NC4=C3F)=C21	C59H69F2N11O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-3KCYVJ	US20240287101A1_99	.	[H]N1C2CCC1CN(C1=NC(OCC3(CN4CCC(CC5CCN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)CC5)CC4)CC3)=NC3=C(F)C(C4CC(O)=CC5=C4C(C#C)=C(F)C=C5)=NC=C13)C2	C54H59F2N9O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-C0IRIA	US20240287101A1_100	.	[H]N1C=CN(C2=NC(OC[C@@]34CCCN3[C@H](CN3CCN(CC5CCN(C6=CCC7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)CC5)CC3)CC4)=NC3=C(F)C(C4=CC(O)=CC5=C4C(C#C)=C(F)C=C5)=NC=C23)CC1	C55H61F2N11O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-22YXMP	SCHEMBL31129611	3-[6-[4-[[4-[[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperazin-1-yl]methyl]piperidin-1-yl]-7-fluoro-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCCN5CCC(CN6CCN(CC7CCN(C8=CC=C9C(=O)N(C%10CCC(=O)NC%10=O)CC9=C8F)CC7)CC6)CC5)=NC4=C3F)=C21	C56H62F3N11O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-96F648	US20240287101A1_102	.	C#CC1=C(F)C=CC2=CC(OI)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCCN5CCC(CC6CCN(CC7CCN(C8=CC9=C(C=C8)N(C8CCC(=O)NC8=O)C(=O)N9C)CC7)CC6)CC5)=NC4=C3F)=C21	C57H64F2IN11O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-EJNYCF	SCHEMBL31129348	3-[6-[4-[(3R,5S)-5-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1-methylpyrrolidin-3-yl]oxypiperidin-1-yl]-7-fluoro-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OC[C@@H]5C[C@@H](OC6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7F)CC6)CN5C)=NC4=C3F)=C21	C49H48F3N9O6	KRAS	P01116	CRBN	US-20240287101-A1
TPD-UFEVAB	US20240287101A1_104	.	C#CC1=C(F)C=CC2=CC(OI)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OC[C@@H]5C[C@@H](OC6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7)CC6)CN5C)=NC4=C3F)=C21	C49H48F2IN9O6	KRAS	P01116	CRBN	US-20240287101-A1
TPD-K9O0IY	US20240287101A1_105	3-[6-[4-[[4-[[1-[2-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]-methylamino]ethyl]piperidin-4-yl]methyl]piperidin-1-yl]methyl]piperidin-1-yl]-7-fluoro-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	[H]N1C2CCC1CN(C1=C3C=NC(C4=CC(O)=CC5=C4C(C#C)=C(F)C=C5)=C(F)C3=NC(N(C)CCN3CCC(CC4CCN(CC5CCN(C6=C(F)C7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)CC5)CC4)CC3)=N1)C2	C58H66F3N11O4	KRAS	P01116	CRBN	US-20240287101-A1
TPD-L767G3	SCHEMBL31129530	3-[6-[4-[[4-[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]oxypiperidin-1-yl]methyl]piperidin-1-yl]-7-fluoro-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCCN5CCC(OC6CCN(CC7CCN(C8=CC=C9C(=O)N(C%10CCC(=O)NC%10=O)CC9=C8F)CC7)CC6)CC5)=NC4=C3F)=C21	C56H61F3N10O6	KRAS	P01116	CRBN	US-20240287101-A1
TPD-KKBPVW	US20240287101A1_107	3-[6-[4-[[4-[[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)pyrido[3,2-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-1-yl]methyl]piperidin-1-yl]-7-fluoro-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	[H]N1C2CCC1CN(C1=C3N=CC(C4=CC(O)=CC5=C4C(C#C)=C(F)C=C5)=CC3=NC(OCCN3CCC(CC4CCN(CC5CCN(C6=C(F)C7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)CC5)CC4)CC3)=N1)C2	C57H64F2N10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-5RN2G4	US20240287101A1_108	3-[6-[4-[[4-[[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)quinazolin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-1-yl]methyl]piperidin-1-yl]-7-fluoro-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	[H]N1C2CCC1CN(C1=C3C=CC(C4=CC(O)=CC5=C4C(C#C)=C(F)C=C5)=CC3=NC(OCCN3CCC(CC4CCN(CC5CCN(C6=C(F)C7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)CC5)CC4)CC3)=N1)C2	C58H65F2N9O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-0L6WSZ	SCHEMBL31129349	3-[7-chloro-6-[4-[[4-[[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-1-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	[H]N1C2CCC1CN(C1=C3C=NC(C4=CC(O)=CC5=C4C(C#C)=C(F)C=C5)=C(F)C3=NC(OCCN3CCC(CC4CCN(CC5CCN(C6=C(Cl)C7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)CC5)CC4)CC3)=N1)C2	C57H63ClF2N10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-DVK1VI	SCHEMBL31129550	3-[5-[4-[[4-[[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-1-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	[H]N1C2CCC1CN(C1=C3C=NC(C4=CC(O)=CC5=C4C(C#C)=C(F)C=C5)=C(F)C3=NC(OCCN3CCC(CC4CCN(CC5CCN(C6=CC7=C(C=C6)CN(C6CCC(=O)NC6=O)C7=O)CC5)CC4)CC3)=N1)C2	C57H64F2N10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-WBU3ZM	SCHEMBL31129468	3-[6-[4-[[4-[[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperazin-1-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCCN5CCC(CN6CCN(CC7CCN(C8=CC=C9C(=O)N(C%10CCC(=O)NC%10=O)CC9=C8)CC7)CC6)CC5)=NC4=C3F)=C21	C56H63F2N11O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-Z6KG0Z	SCHEMBL31129335	3-[6-[4-[[4-[(3R,5S)-5-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1-methylpyrrolidin-3-yl]oxypiperidin-1-yl]methyl]-4-fluoropiperidin-1-yl]-7-fluoro-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OC[C@@H]5C[C@@H](OC6CCN(CC7(F)CCN(C8=C(F)C9=C(C=C8)C(=O)N(C8CCC(=O)NC8=O)C9)CC7)CC6)CN5C)=NC4=C3F)=C21	C55H58F4N10O6	KRAS	P01116	CRBN	US-20240287101-A1
TPD-WZH3A6	US20240287101A1_113	3-[7-chloro-6-[4-[[4-[(3R,5S)-5-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1-methylpyrrolidin-3-yl]oxypiperidin-1-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OC[C@@H]5C[C@@H](OC6CCN(CC7CCN(C8=C(Cl)C9=C(C=C8)C(=O)N(C8CCC(=O)NC8=O)C9)CC7)CC6)CN5C)=NC4=C3F)=C21	C55H59ClF2N10O6	KRAS	P01116	CRBN	US-20240287101-A1
TPD-5G7YGG	US20240287101A1_114	.	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=NC(OC[C@@H]5CC[C@@H](COC(=O)N6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7)CC6)N5C)=NC(N5CC6CCC(C5)N6)=C4C=C3)=C21	C51H51F2N9O7	KRAS	P01116	CRBN	US-20240287101-A1
TPD-BH27WC	SCHEMBL31129596	3-[7-[4-[[4-[(3R,5S)-5-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1-methylpyrrolidin-3-yl]oxypiperidin-1-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OC[C@@H]5C[C@@H](OC6CCN(CC7CCN(C8=C9CN(C%10CCC(=O)NC%10=O)C(=O)C9=CC=C8)CC7)CC6)CN5C)=NC4=C3F)=C21	C55H60F2N10O6	KRAS	P01116	CRBN	US-20240287101-A1
TPD-QS48WP	SCHEMBL31129427	[(2S,5S)-5-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1-methylpyrrolidin-2-yl]methyl 4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]piperazine-1-carboxylate	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=NC(OC[C@@H]5CC[C@@H](COC(=O)N6CCN(C7=C8CN(C9CCC(=O)NC9=O)C(=O)C8=CC=C7)CC6)N5C)=NC(N5CC6CCC(C5)N6)=C4C=N3)=C21	C50H50F2N10O7	KRAS	P01116	CRBN	US-20240287101-A1
TPD-K0HDJ7	SCHEMBL31129740	3-[7-[4-[(3R,5S)-5-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1-methylpyrrolidin-3-yl]oxypiperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CCC1=CC=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OC[C@@H]5C[C@@H](OC6CCN(C7=CC=CC8=C7CN(C7CCC(=O)NC7=O)C8=O)CC6)CN5C)=NC4=C3F)=C21	C49H54FN9O6	KRAS	P01116	CRBN	US-20240287101-A1
TPD-0AOCHP	SCHEMBL31129700	3-[6-[4-[[7-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]-2,7-diazaspiro[3.5]nonan-2-yl]methyl]-4-fluoropiperidin-1-yl]-7-fluoro-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCCN5CCC6(CC5)CN(CC5(F)CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7F)CC5)C6)=NC4=C3F)=C21	C53H54F4N10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-6RU45G	SCHEMBL31129602	3-[6-[4-[[9-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]-3,9-diazaspiro[5.5]undecan-3-yl]methyl]-4-fluoropiperidin-1-yl]-7-fluoro-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCCN5CCC6(CC5)CCN(CC5(F)CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7F)CC5)CC6)=NC4=C3F)=C21	C55H58F4N10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-T49R0P	SCHEMBL31129566	3-[6-[4-[[9-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]-3,9-diazaspiro[5.5]undecan-3-yl]methyl]piperidin-1-yl]-7-fluoro-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCCN5CCC6(CC5)CCN(CC5CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7F)CC5)CC6)=NC4=C3F)=C21	C55H59F3N10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-N7NIUZ	SCHEMBL31129703	3-[6-[4-[[4-[(3R,5S)-5-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1-methylpyrrolidin-3-yl]oxypiperidin-1-yl]methyl]piperidin-1-yl]-7-fluoro-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OC[C@@H]5C[C@@H](OC6CCN(CC7CCN(C8=C(F)C9=C(C=C8)C(=O)N(C8CCC(=O)NC8=O)C9)CC7)CC6)CN5C)=NC4=C3F)=C21	C55H59F3N10O6	KRAS	P01116	CRBN	US-20240287101-A1
TPD-8ZJOCJ	SCHEMBL31129620	3-[7-[4-[[4-[[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]-4-fluoropiperidin-4-yl]methyl]piperidin-1-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCCN5CCC(F)(CC6CCN(CC7CCN(C8=CC=CC9=C8CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)=NC4=C3F)=C21	C57H63F3N10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-OTGOIU	SCHEMBL31129359	3-[7-[4-[[4-[[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-1-yl]methyl]-4-fluoropiperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCCN5CCC(CC6CCN(CC7(F)CCN(C8=CC=CC9=C8CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)=NC4=C3F)=C21	C57H63F3N10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-S34GUU	SCHEMBL31129720	3-[7-[4-[[1-[[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-4-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCCN5CCC(CN6CCC(CC7CCN(C8=CC=CC9=C8CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)=NC4=C3F)=C21	C57H64F2N10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-8K2FMZ	US20240287101A1_127	3-[6-[4-[[7-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]-2,7-diazaspiro[3.5]nonan-2-yl]methyl]piperidin-1-yl]-7-fluoro-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCCN5CCC6(CC5)CN(CC5CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7F)CC5)C6)=NC4=C3F)=C21	C53H55F3N10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-ZJW327	SCHEMBL31129717	3-[7-[4-[2-[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]ethyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=NC(OCCN5CCC(CCC6CCN(C7=C8CN(C9CCC(=O)NC9=O)C(=O)C8=CC=C7)CC6)CC5)=NC(N5CC6CCC(C5)N6)=C4C=N3)=C21	C52H55F2N9O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-XJJP8C	SCHEMBL31129660	3-[4-[4-[[1-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-1-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=NC(OCCN5CCC(CC6CCN(C7=C8C(=CC=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)CC6)CC5)=NC(N5CC6CCC(C5)N6)=C4C=N3)=C21	C51H54F2N10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-JTHEA3	SCHEMBL31129690	3-[7-[4-[[4-[[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-1-yl]methyl]piperidin-1-yl]-5-fluoro-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCCN5CCC(CC6CCN(CC7CCN(C8=CC(F)=CC9=C8CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)=NC4=C3F)=C21	C57H63F3N10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-7YN10F	SCHEMBL31129667	3-[7-[4-[[4-[[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]-4-fluoropiperidin-1-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCCN5CCC(CC6(F)CCN(CC7CCN(C8=CC=CC9=C8CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)=NC4=C3F)=C21	C57H63F3N10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-HI562O	US20240287101A1_132	.	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=CC(OCCN5CCC6(CC5)CCN(CC5CCN(C7=C8CN(C9CCC(=O)NC9=O)C(=O)C8=CC=C7)CC5)CC6)=NC(N5CC6CCC(C5)N6)=C4C=N3)=C21	C56H61F2N9O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-KKA5QI	SCHEMBL31129671	3-[4-[4-[[4-[[1-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-1-yl]methyl]piperidin-1-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=NC(OCCN5CCC(CC6CCN(CC7CCN(C8=C9C(=CC=C8)N(C8CCC(=O)NC8=O)C(=O)N9C)CC7)CC6)CC5)=NC(N5CC6CCC(C5)N6)=C4C=N3)=C21	C57H65F2N11O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-3Y05HL	SCHEMBL31129654	3-[7-[4-[[7-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]-2,7-diazaspiro[3.5]nonan-2-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=NC(OCCN5CCC6(CC5)CN(CC5CCN(C7=C8CN(C9CCC(=O)NC9=O)C(=O)C8=CC=C7)CC5)C6)=NC(N5CC6CCC(C5)N6)=C4C=N3)=C21	C53H56F2N10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-XOD6KS	SCHEMBL31129738	3-[7-[4-[[4-[[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperazin-1-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCCN5CCC(CN6CCN(CC7CCN(C8=CC=CC9=C8CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)=NC4=C3F)=C21	C56H63F2N11O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-4DZVVH	SCHEMBL31129518	3-[7-[4-[[4-[[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-1-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CCC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCCN5CCC(CC6CCN(CC7CCN(C8=CC=CC9=C8CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)=NC4=C3F)=C21	C57H68F2N10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-RHE7YM	SCHEMBL31129520	3-[7-[4-[[4-[(3R,5S)-5-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1-methylpyrrolidin-3-yl]oxypiperidin-1-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CCC1=CC=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OC[C@@H]5C[C@@H](OC6CCN(CC7CCN(C8=C9CN(C%10CCC(=O)NC%10=O)C(=O)C9=CC=C8)CC7)CC6)CN5C)=NC4=C3F)=C21	C55H65FN10O6	KRAS	P01116	CRBN	US-20240287101-A1
TPD-7HJ75S	SCHEMBL31129746	3-[7-[2-[[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]-2,7-diazaspiro[3.5]nonan-7-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=NC(OCCN5CCC(CN6CC7(CCN(C8=CC=CC9=C8CN(C8CCC(=O)NC8=O)C9=O)CC7)C6)CC5)=NC(N5CC6CCC(C5)N6)=C4C=N3)=C21	C53H56F2N10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-5NRWRK	US20240287101A1_141	3-[7-[7-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]-2,7-diazaspiro[3.5]nonan-2-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CC4CCC(C1)N4)=NC(OCCN1CCC4(CC1)CN(C1=C5CN(C6CCC(=O)NC6=O)C(=O)C5=CC=C1)C4)=N3)=CC(O)=C2	C47H50FN9O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-RDWAR7	US20240287101A1_142	3-[6-[4-[[4-[[1-[2-[7-(3-chloro-2-cyclopropyl-5-hydroxyphenyl)-4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-1-yl]methyl]piperidin-1-yl]-7-fluoro-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	[H]N1C2CCC1CN(C1=C3C=NC(C4=CC(O)=CC(Cl)=C4C4CC4)=C(F)C3=NC(OCCN3CCC(CC4CCN(CC5CCN(C6=C(F)C7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)CC5)CC4)CC3)=N1)C2	C54H65ClF2N10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-CVQJCD	US20240287101A1_143	3-[6-[4-[[4-[[(3S,8R)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl]piperazin-1-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	[H]N1C2CCC1CN(C1=NC(OC[C@]34CCCN3[C@H](CN3CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)CC5)CC3)CC4)=NC3=C(F)C(C4=CC=CC5=C4C(C#C)=C(F)C=C5)=NC=C13)C2	C57H63F2N11O4	KRAS	P01116	CRBN	US-20240287101-A1
TPD-4DLAAL	US20240287101A1_144	3-[6-[4-[[4-[(3R,5S)-5-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1-methylpyrrolidin-3-yl]oxypiperidin-1-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	[H]N1C2CCC1CN(C1=C3C=NC(C4=C5C(=CC=C4)C=CC(F)=C5C#C)=C(F)C3=NC(OC[C@@H]3C[C@@H](OC4CCN(CC5CCN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)CC5)CC4)CN3C)=N1)C2	C55H60F2N10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-GQTAE5	US20240287101A1_145	3-[6-[4-[[(3S,8R)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	[H]N1C2CCC1CN(C1=NC(OC[C@]34CCCN3[C@H](CN3CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6)CC3)CC4)=NC3=C(F)C(C4=CC=CC5=C4C(C#C)=C(F)C=C5)=NC=C13)C2	C51H52F2N10O4	KRAS	P01116	CRBN	US-20240287101-A1
TPD-0D5SKE	US20240287101A1_146	3-[6-[4-[[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	[H]N1C2CCC1CN(C1=NC(OC[C@@]34CCCN3[C@H](CN3CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6)CC3)CC4)=NC3=C(F)C(C4=CC=CC5=C4C(C#C)=C(F)C=C5)=NC=C13)C2	C51H52F2N10O4	KRAS	P01116	CRBN	US-20240287101-A1
TPD-P4I80L	US20240287101A1_147	3-[6-[4-[[4-[[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl]piperazin-1-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	[H]N1C(=O)CCC(N2CC3=CC(N4CCC(CN5CCN(C[C@@H]6CC[C@]7(COC8=NC9=C(F)C(C%10=CC=CC%11=C%10C(C#C)=C(F)C=C%11)=NC=C9C(N9CC%10CCC(C9)N%10[H])=N8)CCCN67)CC5)CC4)=CC=C3C2=O)C1=O	C57H63F2N11O4	KRAS	P01116	CRBN	US-20240287101-A1
TPD-7T4D6N	SCHEMBL31129781	3-[6-[4-[[4-[[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperazin-1-yl]methyl]piperidin-1-yl]-7-fluoro-4-methyl-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCCN5CCC(CN6CCN(CC7CCN(C8=CC(C)=C9C(=O)N(C%10CCC(=O)NC%10=O)CC9=C8F)CC7)CC6)CC5)=NC4=C3F)=C21	C57H64F3N11O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-OWQNW0	SCHEMBL31129501	3-[6-[4-[[4-[[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-1-yl]methyl]piperidin-1-yl]-7-fluoro-4-methyl-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCCN5CCC(CC6CCN(CC7CCN(C8=C(F)C9=C(C(=O)N(C%10CCC(=O)NC%10=O)C9)C(C)=C8)CC7)CC6)CC5)=NC4=C3F)=C21	C58H65F3N10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-8Z741U	US20240287101A1_150	3-[6-[4-[[7-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]-2,7-diazaspiro[3.5]nonan-2-yl]methyl]piperidin-1-yl]-7-fluoro-4-methyl-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCCN5CCC6(CC5)CN(CC5CCN(C7=C(F)C8=C(C(=O)N(C9CCC(=O)NC9=O)C8)C(C)=C7)CC5)C6)=NC4=C3F)=C21	C54H57F3N10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-KIYNM4	SCHEMBL31129351	3-[6-[4-[[4-[(3R,5S)-5-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1-methylpyrrolidin-3-yl]oxypiperidin-1-yl]methyl]piperidin-1-yl]-7-fluoro-4-methyl-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OC[C@@H]5C[C@@H](OC6CCN(CC7CCN(C8=C(F)C9=C(C(=O)N(C%10CCC(=O)NC%10=O)C9)C(C)=C8)CC7)CC6)CN5C)=NC4=C3F)=C21	C56H61F3N10O6	KRAS	P01116	CRBN	US-20240287101-A1
TPD-RPBM5N	US20240287101A1_152	3-[6-[4-[[4-[[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoroquinazolin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-1-yl]methyl]piperidin-1-yl]-7-fluoro-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	[H]N1C2CCC1CN(C1=C3C=CC(C4=CC(O)=CC5=C4C(C#C)=C(F)C=C5)=C(F)C3=NC(OCCN3CCC(CC4CCN(CC5CCN(C6=C(F)C7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)CC5)CC4)CC3)=N1)C2	C58H64F3N9O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-Y2L4KH	SCHEMBL31129372	3-[6-[4-[[9-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]-3,9-diazaspiro[5.5]undecan-3-yl]methyl]piperidin-1-yl]-7-fluoro-4-methyl-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCCN5CCC6(CC5)CCN(CC5CCN(C7=C(F)C8=C(C(=O)N(C9CCC(=O)NC9=O)C8)C(C)=C7)CC5)CC6)=NC4=C3F)=C21	C56H61F3N10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-WN466Y	SCHEMBL31129416	3-[6-[2-[[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]-2,7-diazaspiro[3.5]nonan-7-yl]-7-fluoro-4-methyl-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCCN5CCC(CN6CC7(CCN(C8=C(F)C9=C(C(=O)N(C%10CCC(=O)NC%10=O)C9)C(C)=C8)CC7)C6)CC5)=NC4=C3F)=C21	C54H57F3N10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-AYUODN	US20240287101A1_155	3-[6-[2-[[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]-2,7-diazaspiro[3.5]nonan-7-yl]-7-fluoro-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCCN5CCC(CN6CC7(CCN(C8=C(F)C9=C(C=C8)C(=O)N(C8CCC(=O)NC8=O)C9)CC7)C6)CC5)=NC4=C3F)=C21	C53H55F3N10O4	KRAS	P01116	CRBN	US-20240287101-A1
TPD-VJYSLE	US20240287101A1_156	.	[H]N1C2CCC1CN(C1=C(/C=N\C)C(/C(F)=C/C3=C4C(=CC=C3)C=CC(F)C4C#C)=NC(OCCN3CCC4(CC3)CCN(CC3CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)CC6=C5F)CC3)CC4)=N1)C2	C56H65F3N10O4	KRAS	P01116	CRBN	US-20240287101-A1
TPD-30XMQ6	US20240287101A1_157	3-[7-[4-[[4-[[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-1-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC=CC(C3=C(F)C4=NC(OCCN5CCC(CC6CCN(CC7CCN(C8=C9CN(C%10CCC(=O)NC%10=O)C(=O)C9=CC=C8)CC7)CC6)CC5)=NC(N5CC6CCC(C5)N6)=C4C=N3)=C21	C57H64F2N10O4	KRAS	P01116	CRBN	US-20240287101-A1
TPD-GX6LQB	US20240287101A1_158	.	CCC1=CC=CC2=C(F)C(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCCN5CCC(CC6CCN(C7=CC=CC8=C7CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)=NC4=C3F)=C12	C51H57F2N9O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-O6CHSG	SCHEMBL31129426	3-[5-[4-[[4-[[1-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperazin-1-yl]methyl]piperidin-1-yl]-4-fluoro-2-oxo-3-propan-2-ylbenzimidazol-1-yl]piperidine-2,6-dione	[H]N1C2CCC1CN(C1=C3C=NC(C4=CC(O)=CC5=C4C(C#C)=C(F)C=C5)=C(F)C3=NC(OCCN3CCC(CN4CCN(CC5CCN(C6=C(F)C7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)N7C(C)C)CC5)CC4)CC3)=N1)C2	C58H67F3N12O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-S6TK07	SCHEMBL31129649	3-[5-[4-[[4-[[1-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]-4-methylpiperidin-4-yl]methyl]piperazin-1-yl]methyl]piperidin-1-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	[H]N1C2CCC1CN(C1=C3C=NC(C4=CC(O)=CC5=C4C(C#C)=C(F)C=C5)=C(F)C3=NC(OCCN3CCC(C)(CN4CCN(CC5CCN(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC5)CC4)CC3)=N1)C2	C57H66F2N12O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-GVXR4S	SCHEMBL31129395	3-[5-[4-[[4-[[1-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]-4-methylpiperidin-4-yl]methyl]piperidin-1-yl]methyl]piperidin-1-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=NC(OCCN5CCC(C)(CC6CCN(CC7CCN(C8=CC9=C(C=C8)N(C8CCC(=O)NC8=O)C(=O)N9C)CC7)CC6)CC5)=NC(N5CC6CCC(C5)N6)=C4C=N3)=C21	C58H67F2N11O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-EJ1GUC	SCHEMBL31129487	3-[5-[4-[[4-[[4-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]-3,3-dimethylpiperazin-1-yl]methyl]piperidin-1-yl]methyl]piperidin-1-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=NC(OCCN5CCN(CC6CCN(CC7CCN(C8=CC9=C(C=C8)N(C8CCC(=O)NC8=O)C(=O)N9C)CC7)CC6)CC5(C)C)=NC(N5CC6CCC(C5)N6)=C4C=N3)=C21	C58H68F2N12O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-05R3J7	SCHEMBL31129664	(3R)-3-[6-[4-[[4-[[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-1-yl]methyl]piperidin-1-yl]-7-fluoro-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCCN5CCC(CC6CCN(CC7CCN(C8=C(F)C9=C(C=C8)C(=O)N([C@@H]8CCC(=O)NC8=O)C9)CC7)CC6)CC5)=NC4=C3F)=C21	C57H63F3N10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-E3NKBU	SCHEMBL31129563	3-[6-[3-[[4-[(3R,5S)-5-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1-methylpyrrolidin-3-yl]oxypiperidin-1-yl]methyl]azetidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	[H]N1C2CCC1CN(C1=C3C=NC(C4=C5C(=CC(O)=C4)C=CC(F)=C5C#C)=C(F)C3=NC(OC[C@@H]3C[C@@H](OC4CCN(CC5CN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)C5)CC4)CN3C)=N1)C2	C53H56F2N10O6	KRAS	P01116	CRBN	US-20240287101-A1
TPD-D2LT4S	SCHEMBL31129419	3-[6-[4-[[4-[(3R,5S)-5-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1-ethylpyrrolidin-3-yl]oxypiperidin-1-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OC[C@@H]5C[C@@H](OC6CCN(CC7CCN(C8=CC9=C(C=C8)C(=O)N(C8CCC(=O)NC8=O)C9)CC7)CC6)CN5CC)=NC4=C3F)=C21	C56H62F2N10O6	KRAS	P01116	CRBN	US-20240287101-A1
TPD-A6NPRZ	SCHEMBL31129496	3-[5-[4-[[1-[[1-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-4-yl]methyl]piperidin-1-yl]-4-fluoro-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	[H]N1C2CCC1CN(C1=C3C=NC(C4=CC(O)=CC5=C4C(C#C)=C(F)C=C5)=C(F)C3=NC(OCCN3CCC(CN4CCC(CC5CCN(C6=C(F)C7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC5)CC4)CC3)=N1)C2	C57H64F3N11O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-UPBT27	SCHEMBL31129516	3-[5-[4-[[1-[[1-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-4-yl]methyl]piperidin-1-yl]-4-fluoro-2-oxo-3-propan-2-ylbenzimidazol-1-yl]piperidine-2,6-dione	[H]N1C2CCC1CN(C1=C3C=NC(C4=CC(O)=CC5=C4C(C#C)=C(F)C=C5)=C(F)C3=NC(OCCN3CCC(CN4CCC(CC5CCN(C6=C(F)C7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)N7C(C)C)CC5)CC4)CC3)=N1)C2	C59H68F3N11O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-86KRVH	SCHEMBL31129455	3-[6-[4-[[4-[[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]-2,2-dimethylpiperidin-4-yl]methyl]piperazin-1-yl]methyl]piperidin-1-yl]-7-fluoro-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	[H]N1C2CCC1CN(C1=C3C=NC(C4=C5C(=CC(O)=C4)C=CC(F)=C5C#C)=C(F)C3=NC(OCCN3CCC(CN4CCN(CC5CCN(C6=C(F)C7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)CC5)CC4)CC3(C)C)=N1)C2	C58H66F3N11O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-CG6NNI	SCHEMBL31129436	3-[6-[4-[[4-[[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]-2,2-dimethylpiperazin-1-yl]methyl]piperidin-1-yl]-7-fluoro-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	[H]N1C2CCC1CN(C1=C3C=NC(C4=C5C(=CC(O)=C4)C=CC(F)=C5C#C)=C(F)C3=NC(OCCN3CCC(CN4CCN(CC5CCN(C6=C(F)C7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)CC5)C(C)(C)C4)CC3)=N1)C2	C58H66F3N11O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-NWW0OI	SCHEMBL31129616	3-[6-[4-[[1-[[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-4-yl]methyl]piperidin-1-yl]-7-fluoro-4-methyl-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	[H]N1C2CCC1CN(C1=C3C=NC(C4=C5C(=CC(O)=C4)C=CC(F)=C5C#C)=C(F)C3=NC(OCCN3CCC(CN4CCC(CC5CCN(C6=C(F)C7=C(C(=O)N(C8CCC(=O)NC8=O)C7)C(C)=C6)CC5)CC4)CC3)=N1)C2	C58H65F3N10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-J2HLA9	SCHEMBL31129677	3-[5-[4-[[9-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]-3,9-diazaspiro[5.5]undecan-3-yl]methyl]piperidin-1-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	CCC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=NC(OCCN5CCC6(CC5)CCN(CC5CCN(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC5)CC6)=NC(N5CC6CCC(C5)N6)=C4C=N3)=C21	C55H65F2N11O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-F2J5V7	SCHEMBL31129734	3-[4-[4-[[4-[[1-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-1-yl]methyl]piperidin-1-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	CCC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCCN5CCC(CC6CCN(CC7CCN(C8=CC=CC9=C8N(C)C(=O)N9C8CCC(=O)NC8=O)CC7)CC6)CC5)=NC4=C3F)=C21	C57H69F2N11O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-PI2LH2	SCHEMBL31129582	3-[5-[4-[[4-[[4-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperazin-1-yl]methyl]piperidin-1-yl]methyl]piperidin-1-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=NC(OCCN5CCN(CC6CCN(CC7CCN(C8=CC9=C(C=C8)N(C8CCC(=O)NC8=O)C(=O)N9C)CC7)CC6)CC5)=NC(N5CC6CCC(C5)N6)=C4C=N3)=C21	C56H64F2N12O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-RU8DRI	SCHEMBL31129718	3-[6-[4-[[4-[[4-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]-3,3-dimethylpiperazin-1-yl]methyl]piperidin-1-yl]methyl]piperidin-1-yl]-7-fluoro-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	[H]N1C2CCC1CN(C1=C3C=NC(C4=C5C(=CC(O)=C4)C=CC(F)=C5C#C)=C(F)C3=NC(OCCN3CCN(CC4CCN(CC5CCN(C6=C(F)C7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)CC5)CC4)CC3(C)C)=N1)C2	C58H66F3N11O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-VODSDU	SCHEMBL31129724	3-[5-[4-[[1-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-1-yl]-2-oxo-3-propan-2-ylbenzimidazol-1-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCCN5CCC(CC6CCN(C7=CC=C8C(=C7)N(C(C)C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC5)=NC4=C3F)=C21	C53H58F2N10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-SFUNCX	SCHEMBL31129585	3-[5-[4-[[(2S,5S)-5-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1-methylpyrrolidin-2-yl]methyl]piperazin-1-yl]-2-oxo-3-propan-2-ylbenzimidazol-1-yl]piperidine-2,6-dione	[H]N1C2CCC1CN(C1=C3C=NC(C4=CC(O)=CC5=C4C(C#C)=C(F)C=C5)=C(F)C3=NC(OC[C@@H]3CC[C@@H](CN4CCN(C5=CC=C6C(=C5)N(C(C)C)C(=O)N6C5CCC(=O)NC5=O)CC4)N3C)=N1)C2	C51H55F2N11O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-9S7WJ1	SCHEMBL31129344	3-[7-chloro-6-[4-[[4-[(3R,5S)-5-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1-methylpyrrolidin-3-yl]oxypiperidin-1-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CCC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OC[C@@H]5C[C@@H](OC6CCN(CC7CCN(C8=C(Cl)C9=C(C=C8)C(=O)N(C8CCC(=O)NC8=O)C9)CC7)CC6)CN5C)=NC4=C3F)=C21	C55H63ClF2N10O6	KRAS	P01116	CRBN	US-20240287101-A1
TPD-F1NMOS	SCHEMBL31129774	3-[6-[4-[[4-[(3R,5S)-5-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1-methylpyrrolidin-3-yl]oxypiperidin-1-yl]methyl]piperidin-1-yl]-7-fluoro-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CCC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OC[C@@H]5C[C@@H](OC6CCN(CC7CCN(C8=C(F)C9=C(C=C8)C(=O)N(C8CCC(=O)NC8=O)C9)CC7)CC6)CN5C)=NC4=C3F)=C21	C55H63F3N10O6	KRAS	P01116	CRBN	US-20240287101-A1
TPD-KYGHTU	SCHEMBL31129577	3-[5-[4-[[4-[[1-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]-4-methylpiperidin-4-yl]methyl]piperidin-1-yl]methyl]piperidin-1-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	CCC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=NC(OCCN5CCC(C)(CC6CCN(CC7CCN(C8=CC9=C(C=C8)N(C8CCC(=O)NC8=O)C(=O)N9C)CC7)CC6)CC5)=NC(N5CC6CCC(C5)N6)=C4C=N3)=C21	C58H71F2N11O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-4BX1RH	SCHEMBL31129692	3-[5-[4-[[4-[[1-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]-4-methylpiperidin-4-yl]methyl]piperazin-1-yl]methyl]piperidin-1-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	CCC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=NC(OCCN5CCC(C)(CN6CCN(CC7CCN(C8=CC9=C(C=C8)N(C8CCC(=O)NC8=O)C(=O)N9C)CC7)CC6)CC5)=NC(N5CC6CCC(C5)N6)=C4C=N3)=C21	C57H70F2N12O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-XV9NHS	SCHEMBL31129658	3-[5-[4-[[4-[[1-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]-4-fluoropiperidin-4-yl]methyl]piperazin-1-yl]methyl]piperidin-1-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	CCC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=NC(OCCN5CCC(F)(CN6CCN(CC7CCN(C8=CC9=C(C=C8)N(C8CCC(=O)NC8=O)C(=O)N9C)CC7)CC6)CC5)=NC(N5CC6CCC(C5)N6)=C4C=N3)=C21	C56H67F3N12O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-HHTCPU	SCHEMBL31129598	3-[5-[4-[[4-[[1-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]-4-fluoropiperidin-4-yl]methyl]piperidin-1-yl]methyl]piperidin-1-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	CCC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=NC(OCCN5CCC(F)(CC6CCN(CC7CCN(C8=CC9=C(C=C8)N(C8CCC(=O)NC8=O)C(=O)N9C)CC7)CC6)CC5)=NC(N5CC6CCC(C5)N6)=C4C=N3)=C21	C57H68F3N11O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-1DZVVP	SCHEMBL31129741	3-[5-[4-[[1-[[1-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]-4-fluoropiperidin-4-yl]methyl]piperidin-4-yl]methyl]piperidin-1-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=NC(OCCN5CCC(F)(CN6CCC(CC7CCN(C8=CC9=C(C=C8)N(C8CCC(=O)NC8=O)C(=O)N9C)CC7)CC6)CC5)=NC(N5CC6CCC(C5)N6)=C4C=N3)=C21	C57H64F3N11O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-ADX36M	SCHEMBL31129590	3-[5-[4-[[4-[[1-[(2R)-1-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxypropan-2-yl]piperidin-4-yl]methyl]piperidin-1-yl]methyl]piperidin-1-yl]-2-oxo-3-propan-2-ylbenzimidazol-1-yl]piperidine-2,6-dione	[H]N1C2CCC1CN(C1=C3C=NC(C4=C5C(=CC(O)=C4)C=CC(F)=C5C#C)=C(F)C3=NC(OC[C@@H](C)N3CCC(CC4CCN(CC5CCN(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)N7C(C)C)CC5)CC4)CC3)=N1)C2	C60H71F2N11O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-6Z49NS	SCHEMBL31129645	3-[6-[4-[[4-[[1-[(2R)-1-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxypropan-2-yl]piperidin-4-yl]methyl]piperidin-1-yl]methyl]piperidin-1-yl]-7-fluoro-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	[H]N1C2CCC1CN(C1=C3C=NC(C4=C5C(=CC(O)=C4)C=CC(F)=C5C#C)=C(F)C3=NC(OC[C@@H](C)N3CCC(CC4CCN(CC5CCN(C6=C(F)C7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)CC5)CC4)CC3)=N1)C2	C58H65F3N10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-20MANA	SCHEMBL31129656	3-[7-chloro-6-[4-[[4-[[1-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperazin-1-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCC5(CN6CCN(CC7CCN(C8=C(Cl)C9=C(C=C8)C(=O)N(C8CCC(=O)NC8=O)C9)CC7)CC6)CC5)=NC4=C3F)=C21	C53H55ClF2N10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-NX1FMO	SCHEMBL31129466	3-[7-chloro-6-[4-[[1-[[1-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCC5(CN6CCC(CN7CCN(C8=C(Cl)C9=C(C=C8)C(=O)N(C8CCC(=O)NC8=O)C9)CC7)CC6)CC5)=NC4=C3F)=C21	C53H55ClF2N10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-X8LSW3	SCHEMBL31129765	3-[5-[4-[[4-[[1-[[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperazin-1-yl]methyl]piperidin-1-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCC5(CN6CCN(CC7CCN(C8=CC9=C(C=C8)N(C8CCC(=O)NC8=O)C(=O)N9C)CC7)CC6)CC5)=NC4=C3F)=C21	C53H57F2N11O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-1B0JIE	SCHEMBL31129558	3-[5-[4-[[1-[[1-[[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCC5(CN6CCC(CN7CCN(C8=CC9=C(C=C8)N(C8CCC(=O)NC8=O)C(=O)N9C)CC7)CC6)CC5)=NC4=C3F)=C21	C53H57F2N11O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-J0JCCA	SCHEMBL31129363	3-[7-chloro-6-[4-[[1-[[1-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCC5(CN6CCC(CC7CCN(C8=C(Cl)C9=C(C=C8)C(=O)N(C8CCC(=O)NC8=O)C9)CC7)CC6)CC5)=NC4=C3F)=C21	C54H56ClF2N9O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-J3NBI8	SCHEMBL31129678	3-[5-[4-[[1-[[1-[[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]methyl]piperidin-1-yl]-2-oxo-3-propan-2-ylbenzimidazol-1-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCC5(CN6CCC(CC7CCN(C8=CC9=C(C=C8)N(C8CCC(=O)NC8=O)C(=O)N9C(C)C)CC7)CC6)CC5)=NC4=C3F)=C21	C56H62F2N10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-MB2UYU	SCHEMBL31129375	3-[6-[4-[[1-[[1-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]methyl]piperidin-1-yl]-7-fluoro-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCC5(CN6CCC(CC7CCN(C8=C(F)C9=C(C=C8)C(=O)N(C8CCC(=O)NC8=O)C9)CC7)CC6)CC5)=NC4=C3F)=C21	C54H56F3N9O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-SRVRGO	SCHEMBL31129569	3-[5-[4-[[3-[[1-[[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-3,9-diazaspiro[5.5]undecan-9-yl]methyl]piperidin-1-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCC5(CN6CCC7(CCN(CC8CCN(C9=CC%10=C(C=C9)N(C9CCC(=O)NC9=O)C(=O)N%10C)CC8)CC7)CC6)CC5)=NC4=C3F)=C21	C58H65F2N11O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-MVNTUX	SCHEMBL31129556	3-[6-[4-[[4-[[1-[(2S)-1-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxypropan-2-yl]piperidin-4-yl]methyl]piperidin-1-yl]methyl]piperidin-1-yl]-7-fluoro-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	[H]N1C2CCC1CN(C1=C3C=NC(C4=C5C(=CC(O)=C4)C=CC(F)=C5C#C)=C(F)C3=NC(OC[C@H](C)N3CCC(CC4CCN(CC5CCN(C6=C(F)C7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)CC5)CC4)CC3)=N1)C2	C58H65F3N10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-TTFA69	SCHEMBL31129631	3-[5-[4-[[4-[[1-[(2S)-1-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxypropan-2-yl]piperidin-4-yl]methyl]piperidin-1-yl]methyl]piperidin-1-yl]-2-oxo-3-propan-2-ylbenzimidazol-1-yl]piperidine-2,6-dione	[H]N1C2CCC1CN(C1=C3C=NC(C4=C5C(=CC(O)=C4)C=CC(F)=C5C#C)=C(F)C3=NC(OC[C@H](C)N3CCC(CC4CCN(CC5CCN(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)N7C(C)C)CC5)CC4)CC3)=N1)C2	C60H71F2N11O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-RQWILK	SCHEMBL31129603	3-[5-[4-[[4-[[1-[[1-[[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]methyl]piperidin-1-yl]methyl]piperidin-1-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCC5(CN6CCC(CC7CCN(CC8CCN(C9=CC%10=C(C=C9)N(C9CCC(=O)NC9=O)C(=O)N%10C)CC8)CC7)CC6)CC5)=NC4=C3F)=C21	C60H69F2N11O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-PYMPHQ	US20240287101A1_197	.	[H]C1=C(C#C)C2=C(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCCN5CCC6(CC5)CCN(CC5CCN(C7=CC=C8C(=C7F)N(C)C(=O)N8C7CCC(=O)NC7=O)CC5)CC6)=NC4=C3F)C=C(O)C=C2C=C1	C55H61F2N11O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-3J5XGV	SCHEMBL31129420	3-[5-[4-[[4-[[1-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]-4-fluoropiperidin-4-yl]methyl]piperidin-1-yl]methyl]piperidin-1-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	[H]N1C2CCC1CN(C1=C3C=NC(C4=C5C(=CC(O)=C4)C=CC(F)=C5C#C)=C(F)C3=NC(OCCN3CCC(F)(CC4CCN(CC5CCN(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC5)CC4)CC3)=N1)C2	C57H64F3N11O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-VXMK0V	SCHEMBL31129564	3-[5-[4-[[4-[[1-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-1-yl]methyl]piperidin-1-yl]-4,7-difluoro-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCCN5CCC(CC6CCN(CC7CCN(C8=C(F)C9=C(C(F)=C8)N(C8CCC(=O)NC8=O)C(=O)N9C)CC7)CC6)CC5)=NC4=C3F)=C21	C57H63F4N11O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-PV3DUX	SCHEMBL31129357	3-[5-[4-[[4-[[1-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]-4-fluoropiperidin-4-yl]methyl]piperazin-1-yl]methyl]piperidin-1-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCCN5CCC(F)(CN6CCN(CC7CCN(C8=CC9=C(C=C8)N(C8CCC(=O)NC8=O)C(=O)N9C)CC7)CC6)CC5)=NC4=C3F)=C21	C56H63F3N12O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-EL66KF	SCHEMBL31129555	3-[5-[4-[[4-[(3R,5S)-5-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1-methylpyrrolidin-3-yl]oxypiperidin-1-yl]methyl]piperidin-1-yl]-4,7-difluoro-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OC[C@@H]5C[C@@H](OC6CCN(CC7CCN(C8=C(F)C9=C(C(F)=C8)N(C8CCC(=O)NC8=O)C(=O)N9C)CC7)CC6)CN5C)=NC4=C3F)=C21	C55H59F4N11O6	KRAS	P01116	CRBN	US-20240287101-A1
TPD-7UAL61	SCHEMBL31129609	3-[5-[4-[[9-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]-3,9-diazaspiro[5.5]undecan-3-yl]methyl]piperidin-1-yl]-2-oxo-3-propan-2-ylbenzimidazol-1-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCCN5CCC6(CC5)CCN(CC5CCN(C7=CC=C8C(=C7)N(C(C)C)C(=O)N8C7CCC(=O)NC7=O)CC5)CC6)=NC4=C3F)=C21	C57H65F2N11O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-73L1QO	SCHEMBL31129572	3-[5-[4-[[9-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]-3,9-diazaspiro[5.5]undecan-3-yl]methyl]piperidin-1-yl]-4-fluoro-2-oxo-3-propan-2-ylbenzimidazol-1-yl]piperidine-2,6-dione	[H]N1C2CCC1CN(C1=C3C=NC(C4=C5C(=CC(O)=C4)C=CC(F)=C5C#C)=C(F)C3=NC(OCCN3CCC4(CC3)CCN(CC3CCN(C5=CC=C6C(=C5F)N(C(C)C)C(=O)N6C5CCC(=O)NC5=O)CC3)CC4)=N1)C2	C57H64F3N11O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-1T8ZRY	US20240287101A1_204	3-[5-[4-[[4-[[(3S,8R)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl]piperazin-1-yl]methyl]piperidin-1-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	[H]N1C2CCC1CN(C1=NC(OC[C@]34CCCN3[C@H](CN3CCN(CC5CCN(C6=CC=C7C(=C6)N(C)C(=O)N7C6CCC(=O)NC6=O)CC5)CC3)CC4)=NC3=C(F)C(C4=CC(O)=CC5=C4C(C#C)=C(F)C=C5)=NC=C13)C2	C57H64F2N12O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-JFX6VU	SCHEMBL31129434	3-[5-[4-[[4-[[1-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-1-yl]methyl]piperidin-1-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	CCC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCCN5CCC(CC6CCN(CC7CCN(C8=CC9=C(C=C8)N(C8CCC(=O)NC8=O)C(=O)N9C)CC7)CC6)CC5)=NC4=C3F)=C21	C57H69F2N11O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-7C2G9F	SCHEMBL31129373	3-[5-[4-[[4-[[1-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-1-yl]methyl]piperidin-1-yl]-4-fluoro-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCCN5CCC(CC6CCN(CC7CCN(C8=C(F)C9=C(C=C8)N(C8CCC(=O)NC8=O)C(=O)N9C)CC7)CC6)CC5)=NC4=C3F)=C21	C57H64F3N11O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-2Z73GM	SCHEMBL31129537	3-[5-[4-[[4-[(3R,5S)-5-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1-methylpyrrolidin-3-yl]oxypiperidin-1-yl]methyl]piperidin-1-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	CCC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OC[C@@H]5C[C@@H](OC6CCN(CC7CCN(C8=CC9=C(C=C8)N(C8CCC(=O)NC8=O)C(=O)N9C)CC7)CC6)CN5C)=NC4=C3F)=C21	C55H65F2N11O6	KRAS	P01116	CRBN	US-20240287101-A1
TPD-OMDCWZ	US20240287101A1_208	3-[5-[4-[[4-[[(3S,8R)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl]piperazin-1-yl]methyl]piperidin-1-yl]-2-oxo-3-propan-2-ylbenzimidazol-1-yl]piperidine-2,6-dione	[H]N1C2CCC1CN(C1=NC(OC[C@]34CCCN3[C@H](CN3CCN(CC5CCN(C6=CC=C7C(=C6)N(C(C)C)C(=O)N7C6CCC(=O)NC6=O)CC5)CC3)CC4)=NC3=C(F)C(C4=CC(O)=CC5=C4C(C#C)=C(F)C=C5)=NC=C13)C2	C59H68F2N12O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-GZGL8L	SCHEMBL31129583	3-[5-[4-[[4-[(3R,5S)-5-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1-methylpyrrolidin-3-yl]oxypiperidin-1-yl]methyl]piperidin-1-yl]-2-oxo-3-propan-2-ylbenzimidazol-1-yl]piperidine-2,6-dione	CCC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OC[C@@H]5C[C@@H](OC6CCN(CC7CCN(C8=CC9=C(C=C8)N(C8CCC(=O)NC8=O)C(=O)N9C(C)C)CC7)CC6)CN5C)=NC4=C3F)=C21	C57H69F2N11O6	KRAS	P01116	CRBN	US-20240287101-A1
TPD-SWLX13	SCHEMBL31129465	3-[5-[4-[[1-[[1-[[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]methyl]piperidin-1-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCC5(CN6CCC(CC7CCN(C8=CC9=C(C=C8)N(C8CCC(=O)NC8=O)C(=O)N9C)CC7)CC6)CC5)=NC4=C3F)=C21	C54H58F2N10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-6ZMNLK	SCHEMBL31129525	3-[5-[4-[[4-[[(2S,5S)-5-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1-methylpyrrolidin-2-yl]methyl]piperazin-1-yl]methyl]piperidin-1-yl]-2-oxo-3-propan-2-ylbenzimidazol-1-yl]piperidine-2,6-dione	[H]N1C2CCC1CN(C1=C3C=NC(C4=CC(O)=CC5=C4C(C#C)=C(F)C=C5)=C(F)C3=NC(OC[C@@H]3CC[C@@H](CN4CCN(CC5CCN(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)N7C(C)C)CC5)CC4)N3C)=N1)C2	C57H66F2N12O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-P3OJAD	SCHEMBL31129491	3-[5-[4-[[4-[[1-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-1-yl]methyl]piperidin-1-yl]-2-oxo-3-propan-2-ylbenzimidazol-1-yl]piperidine-2,6-dione	CCC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCCN5CCC(CC6CCN(CC7CCN(C8=CC9=C(C=C8)N(C8CCC(=O)NC8=O)C(=O)N9C(C)C)CC7)CC6)CC5)=NC4=C3F)=C21	C59H73F2N11O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-ISPK20	SCHEMBL31129745	3-[5-[4-[[4-[(3R,5S)-5-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1-methylpyrrolidin-3-yl]oxypiperidin-1-yl]methyl]piperidin-1-yl]-4-fluoro-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OC[C@@H]5C[C@@H](OC6CCN(CC7CCN(C8=C(F)C9=C(C=C8)N(C8CCC(=O)NC8=O)C(=O)N9C)CC7)CC6)CN5C)=NC4=C3F)=C21	C55H60F3N11O6	KRAS	P01116	CRBN	US-20240287101-A1
TPD-9F6541	SCHEMBL31129633	(3S)-3-[6-[4-[[4-[[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-1-yl]methyl]piperidin-1-yl]-7-fluoro-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCCN5CCC(CC6CCN(CC7CCN(C8=C(F)C9=C(C=C8)C(=O)N([C@H]8CCC(=O)NC8=O)C9)CC7)CC6)CC5)=NC4=C3F)=C21	C57H63F3N10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-J7VR9H	SCHEMBL31129744	(3S)-3-[6-[4-[[4-[[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-1-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCCN5CCC(CC6CCN(CC7CCN(C8=CC9=C(C=C8)C(=O)N([C@H]8CCC(=O)NC8=O)C9)CC7)CC6)CC5)=NC4=C3F)=C21	C57H64F2N10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-ZPS0OP	SCHEMBL31129523	(3R)-3-[6-[4-[[4-[[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-1-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCCN5CCC(CC6CCN(CC7CCN(C8=CC9=C(C=C8)C(=O)N([C@@H]8CCC(=O)NC8=O)C9)CC7)CC6)CC5)=NC4=C3F)=C21	C57H64F2N10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-NTF4PN	SCHEMBL31129600	3-[5-[4-[[4-[[1-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-1-yl]methyl]piperidin-1-yl]-4-fluoro-2-oxo-3-propan-2-ylbenzimidazol-1-yl]piperidine-2,6-dione	[H]N1C2CCC1CN(C1=C3C=NC(C4=CC(O)=CC5=C4C(C#C)=C(F)C=C5)=C(F)C3=NC(OCCN3CCC(CC4CCN(CC5CCN(C6=C(F)C7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)N7C(C)C)CC5)CC4)CC3)=N1)C2	C59H68F3N11O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-MRTA8Q	SCHEMBL31129345	3-[5-[4-[[9-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]-3,9-diazaspiro[5.5]undecan-3-yl]methyl]piperidin-1-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCCN5CCC6(CC5)CCN(CC5CCN(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC5)CC6)=NC4=C3F)=C21	C55H61F2N11O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-FMVYY7	SCHEMBL31129448	3-[7-chloro-6-[4-[[4-[[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperazin-1-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	[H]N1C2CCC1CN(C1=C3C=NC(C4=CC(O)=CC5=C4C(C#C)=C(F)C=C5)=C(F)C3=NC(OCCN3CCC(CN4CCN(CC5CCN(C6=C(Cl)C7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)CC5)CC4)CC3)=N1)C2	C56H62ClF2N11O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-GSNZZG	SCHEMBL31129407	3-[7-chloro-6-[4-[[9-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]-3,9-diazaspiro[5.5]undecan-3-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	[H]N1C2CCC1CN(C1=C3C=NC(C4=CC(O)=CC5=C4C(C#C)=C(F)C=C5)=C(F)C3=NC(OCCN3CCC4(CC3)CCN(CC3CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)CC6=C5Cl)CC3)CC4)=N1)C2	C55H59ClF2N10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-QDAMZJ	SCHEMBL31129676	3-[5-[4-[[4-[[1-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperazin-1-yl]methyl]piperidin-1-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	[H]N1C2CCC1CN(C1=C3C=NC(C4=CC(O)=CC5=C4C(C#C)=C(F)C=C5)=C(F)C3=NC(OCCN3CCC(CN4CCN(CC5CCN(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC5)CC4)CC3)=N1)C2	C56H64F2N12O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-WL6WAI	SCHEMBL31129699	3-[5-[4-[[4-[[1-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperazin-1-yl]methyl]piperidin-1-yl]-2-oxo-3-propan-2-ylbenzimidazol-1-yl]piperidine-2,6-dione	[H]N1C2CCC1CN(C1=C3C=NC(C4=CC(O)=CC5=C4C(C#C)=C(F)C=C5)=C(F)C3=NC(OCCN3CCC(CN4CCN(CC5CCN(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)N7C(C)C)CC5)CC4)CC3)=N1)C2	C58H68F2N12O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-S5KXU1	SCHEMBL31129424	3-[6-[4-[[1-[[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]-7-fluoro-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	[H]N1C2CCC1CN(C1=C3C=NC(C4=C5C(=CC(O)=C4)C=CC(F)=C5C#C)=C(F)C3=NC(OCCN3CCC(CN4CCC(CN5CCN(C6=C(F)C7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)CC5)CC4)CC3)=N1)C2	C56H62F3N11O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-Q7C38C	SCHEMBL31129421	3-[5-[4-[[4-[(3R,5S)-5-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1-methylpyrrolidin-3-yl]oxypiperidin-1-yl]methyl]piperidin-1-yl]-4-fluoro-2-oxo-3-propan-2-ylbenzimidazol-1-yl]piperidine-2,6-dione	[H]N1C2CCC1CN(C1=C3C=NC(C4=C5C(=CC(O)=C4)C=CC(F)=C5C#C)=C(F)C3=NC(OC[C@@H]3C[C@@H](OC4CCN(CC5CCN(C6=C(F)C7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)N7C(C)C)CC5)CC4)CN3C)=N1)C2	C57H64F3N11O6	KRAS	P01116	CRBN	US-20240287101-A1
TPD-N4HODP	US20240287101A1_225	.	C#CC1=C(F)C=CC2=CC(O)=CC(C3=CC=C4C(N5CC6CCC(C5)N6)=NC(OCCN5CCC6(CC5)CCN(CC5CCN(C7=CC=C8C(=C7F)N(C)C(=O)N8C7CCC(=O)NC7=O)CC5)CC6)=NC4=C3F)=C21	C56H61F3N10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-AGGFYV	SCHEMBL31129682	3-[5-[4-[[4-[[1-[3-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxypropyl]piperidin-4-yl]methyl]piperidin-1-yl]methyl]piperidin-1-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCCCN5CCC(CC6CCN(CC7CCN(C8=CC9=C(C=C8)N(C8CCC(=O)NC8=O)C(=O)N9C)CC7)CC6)CC5)=NC4=C3F)=C21	C58H67F2N11O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-DHC7XV	US20240287101A1_227	3-[5-[4-[[4-[[4-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoroquinazolin-2-yl]oxyethyl]-3,3-dimethylpiperazin-1-yl]methyl]piperidin-1-yl]methyl]piperidin-1-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=NC(OCCN5CCN(CC6CCN(CC7CCN(C8=CC9=C(C=C8)N(C8CCC(=O)NC8=O)C(=O)N9C)CC7)CC6)CC5(C)C)=NC(N5CC6CCC(C5)N6)=C4C=C3)=C21	C59H69F2N11O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-FG5HNA	SCHEMBL31129452	3-[5-[4-[[1-[[1-[[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-4-fluoropiperidin-4-yl]methyl]piperazin-1-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OCC4(CN5CCC(F)(CN6CCN(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC5)CC4)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C53H56F3N11O4	KRAS	P01116	CRBN	US-20240287101-A1
TPD-EFC0KG	SCHEMBL31129422	3-[5-[3-[[4-[[1-[[1-[[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]methyl]piperidin-1-yl]methyl]azetidin-1-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(OCC5(CN6CCC(CC7CCN(CC8CN(C9=CC%10=C(C=C9)N(C9CCC(=O)NC9=O)C(=O)N%10C)C8)CC7)CC6)CC5)=NC4=C3F)=C21	C58H65F2N11O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-Y0AZXX	orb2802159	3-[5-[4-[[4-[[1-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-1-yl]methyl]piperidin-1-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione; SCHEMBL31129456; 3052745-46-4	[H]N1C2CCC1CN(C1=NC(OCCN3CCC(CC4CCN(CC5CCN(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC5)CC4)CC3)=NC3=C(F)C(C4=CC(O)=CC5=C4C(C#C)=C(F)C=C5)=NC=C13)C2	C57H65F2N11O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-QO9L9C	US20240287101A1_232	3-[5-[4-[[4-[[1-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoroquinazolin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-1-yl]methyl]piperidin-1-yl]-4-fluoro-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	[H]N1C2CCC1CN(C1=NC(OCCN3CCC(CC4CCN(CC5CCN(C6=C(F)C7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC5)CC4)CC3)=NC3=C(F)C(C4=CC(O)=CC5=C4C(C#C)=C(F)C=C5)=CC=C13)C2	C58H65F3N10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-SBB5AQ	US20240287101A1_233	3-[5-[4-[[1-[[1-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoroquinazolin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-4-yl]methyl]piperidin-1-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	[H]N1C2CCC1CN(C1=NC(OCCN3CCC(CN4CCC(CC5CCN(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC5)CC4)CC3)=NC3=C(F)C(C4=CC(O)=CC5=C4C(C#C)=C(F)C=C5)=CC=C13)C2	C58H66F2N10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-IGNN2M	US20240287101A1_234	3-[5-[4-[[4-[[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl]piperazin-1-yl]methyl]piperidin-1-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	[H]N1C2CCC1CN(C1=NC(OC[C@@]34CCCN3[C@H](CN3CCN(CC5CCN(C6=CC=C7C(=C6)N(C)C(=O)N7C6CCC(=O)NC6=O)CC5)CC3)CC4)=NC3=C(F)C(C4=CC=CC5=C4C(C#C)=C(F)C=C5)=NC=C13)C2	C57H64F2N12O4	KRAS	P01116	CRBN	US-20240287101-A1
TPD-RN56GO	SCHEMBL31129411	3-[6-[3-[[4-[[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]piperidin-1-yl]methyl]azetidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	[H]N1C2CCC1CN(C1=C3C=NC(C4=CC(O)=CC5=C4C(C#C)=C(F)C=C5)=C(F)C3=NC(OCCN3CCC(CC4CCN(CC5CN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)C5)CC4)CC3)=N1)C2	C55H60F2N10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-FX3RPM	SCHEMBL31129390	3-[5-[4-[[1-[(3R)-1-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]pyrrolidin-3-yl]piperidin-4-yl]methyl]piperidin-1-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=NC=C4C(N5CC6CCC(C5)N6)=NC(N5CC[C@@H](N6CCC(CC7CCN(C8=CC=C9C(=C8)N(C)C(=O)N9C8CCC(=O)NC8=O)CC7)CC6)C5)=NC4=C3F)=C21	C53H57F2N11O4	KRAS	P01116	CRBN	US-20240287101-A1
TPD-AN2SKK	US20240287101A1_237	.	C#CC1=C(F)C=CC2=CC(O)=CC(C3=CC=C4C(N5CC6CCC(C5)N6)=NC(OCCN5CCC(CC6CCN(CC7CCN(C8=CC9=C(C=C8)N(C8CCC(=O)NC8=O)C(=O)N9C)CC7)CC6)CC5)=NC4=C3F)=C21	C58H66F2N10O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-7HHUFV	US20240287101A1_238	3-[6-[4-[[4-[[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl]piperazin-1-yl]methyl]piperidin-1-yl]-7-fluoro-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	[H]N1C2CCC1CN(C1=NC(OC[C@@]34CCCN3[C@H](CN3CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6F)CC5)CC3)CC4)=NC3=C(F)C(C4=CC=CC5=C4C(C#C)=C(F)C=C5)=NC=C13)C2	C57H62F3N11O4	KRAS	P01116	CRBN	US-20240287101-A1
TPD-UJ0R7A	SCHEMBL31129701	3-[6-[4-[[4-[[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperidin-4-yl]methyl]-3,3-dimethylpiperazin-1-yl]methyl]piperidin-1-yl]-7-fluoro-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	[H]N1C2CCC1CN(C1=C3C=NC(C4=C5C(=CC(O)=C4)C=CC(F)=C5C#C)=C(F)C3=NC(OCCN3CCC(CN4CCN(CC5CCN(C6=C(F)C7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)CC5)CC4(C)C)CC3)=N1)C2	C58H66F3N11O5	KRAS	P01116	CRBN	US-20240287101-A1
TPD-6E0LIY	SCHEMBL24851843	4-[[(7R)-8-cyclopentyl-7-ethyl-6-oxo-5,7-dihydropteridin-2-yl]amino]-N-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethyl]-3-methoxybenzamide	CC[C@@H]1C(=O)Nc2cnc(Nc3ccc(C(=O)NCCOCCOCCNc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)cc3OC)nc2N1C1CCCC1	C40H47N9O9	PLK1	P53350	CRBN	US-20240316054-A1
TPD-MQH1NK	US20240316054A1_2	.	CCC[C@@H]1C(=O)N(C)c2cnc(Nc3ccc(C(=O)NCCOCCOCCNC4C=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C54)cc3OC)nc2N1C1CCCC1	C42H53N9O9	PLK1	P53350	CRBN	US-20240316054-A1
TPD-I8ZNZW	SCHEMBL24851360	4-[[(7R)-8-cyclopentyl-7-ethyl-5-methyl-6-oxo-7H-pteridin-2-yl]amino]-N-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethyl]-3-methylbenzamide	CC[C@@H]1C(=O)N(C)c2cnc(Nc3ccc(C(=O)NCCOCCOCCNc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)cc3C)nc2N1C1CCCC1	C41H49N9O8	PLK1	P53350	CRBN	US-20240316054-A1
TPD-35ZJIK	SCHEMBL24851681	4-[[(7R)-8-cyclopentyl-7-ethyl-5-methyl-6-oxo-7H-pteridin-2-yl]amino]-N-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethyl]benzamide	CC[C@@H]1C(=O)N(C)c2cnc(Nc3ccc(C(=O)NCCOCCOCCNc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)cc3)nc2N1C1CCCC1	C40H47N9O8	PLK1	P53350	CRBN	US-20240316054-A1
TPD-Z70IRD	SCHEMBL31098162	4-[[(7R)-8-cyclopentyl-7-ethyl-5-methyl-6-oxo-7H-pteridin-2-yl]amino]-N-[2-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethyl]-3-methoxybenzamide; PD141857	CC[C@@H]1C(=O)N(C)c2cnc(Nc3ccc(C(=O)NCCOCCOCCOCCOCCNc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)cc3OC)nc2N1C1CCCC1	C45H57N9O11	PLK1	P53350	CRBN	US-20240316054-A1
TPD-MF6H8X	SCHEMBL24851392	4-[[(7R)-8-cyclopentyl-7-ethyl-5-methyl-6-oxo-7H-pteridin-2-yl]amino]-N-[(3S)-1-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperazin-1-yl]-4-oxobutanoyl]pyrrolidin-3-yl]-3-methoxybenzamide; SCHEMBL31098117	CC[C@@H]1C(=O)N(C)c2cnc(Nc3ccc(C(=O)N[C@H]4CCN(C(=O)CCC(=O)N5CCN(c6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)cc3OC)nc2N1C1CCCC1	C47H55N11O9	PLK1	P53350	CRBN	US-20240316054-A1
TPD-8WFJK6	SCHEMBL31098094	4-[[(7R)-8-cyclopentyl-7-ethyl-5-methyl-6-oxo-7H-pteridin-2-yl]amino]-N-[1-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperazin-1-yl]propanoyl]piperidin-4-yl]-3-methoxybenzamide	CC[C@@H]1C(=O)N(C)c2cnc(Nc3ccc(C(=O)NC4CCN(C(=O)CCN5CCN(c6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3OC)nc2N1C1CCCC1	C47H57N11O8	PLK1	P53350	CRBN	US-20240316054-A1
TPD-6Q72H3	SCHEMBL31098122	4-[[(7R)-8-cyclopentyl-7-ethyl-5-methyl-6-oxo-7H-pteridin-2-yl]amino]-N-[1-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]butanoyl]piperidin-4-yl]-3-methoxybenzamide	CC[C@@H]1C(=O)N(C)c2cnc(Nc3ccc(C(=O)NC4CCN(C(=O)CCCNc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)cc3OC)nc2N1C1CCCC1	C44H52N10O8	PLK1	P53350	CRBN	US-20240316054-A1
TPD-W8GF84	SCHEMBL24852311	4-[[(7R)-8-cyclohexyl-5,7-dimethyl-6-oxo-7H-pteridin-2-yl]amino]-N-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethyl]-3-methoxybenzamide	COc1cc(C(=O)NCCOCCOCCNc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)ccc1Nc1ncc2c(n1)N(C1CCCCC1)[C@H](C)C(=O)N2C	C41H49N9O9	PLK1	P53350	CRBN	US-20240316054-A1
TPD-3R73WH	SCHEMBL24851805	4-[[(7R)-8-cyclopentyl-7-ethyl-5-methyl-6-oxo-7H-pteridin-2-yl]amino]-N-[4-[4-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethyl]piperazin-1-yl]cyclohexyl]-3-methoxybenzamide; SCHEMBL31098126	CC[C@@H]1C(=O)N(C)c2cnc(Nc3ccc(C(=O)N[C@H]4CC[C@H](N5CCN(CCOCCNc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3OC)nc2N1C1CCCC1	C49H63N11O8	PLK1	P53350	CRBN	US-20240316054-A1
TPD-H515JM	US20240316054A1_11	.	CC[C@@H]1C(=O)N(C)c2cnc(Nc3ccc(C(=O)N[C@H]4CC[C@H](N5CCN(CCNc6cccc7c6C(=O)N(C6CCC(=O)NC6O)C7=O)CC5)CC4)cc3OC)nc2N1C1CCCC1	C47H61N11O7	PLK1	P53350	CRBN	US-20240316054-A1
TPD-NZ8PPS	PZ15227	4-[4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[(2R)-4-[4-[4-[4-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxymethyl]triazol-1-yl]butanoyl]piperazin-1-yl]-1-phenylsulfanylbutan-2-yl]amino]-3-(trifluoromethylsulfonyl)phenyl]sulfonylbenzamide; orb2813997; SCHEMBL19475680; SCHEMBL19475686; OWEARFNXBBNNKR-ADXOFTSBSA-N; 4-[4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[(2R)-4-[4-[4-[4-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxymethyl]triazol-1-yl]butanoyl]piperazin-1-yl]-1-phenylsulfanylbutan-2-yl]amino]-3-(trifluoromethylsulfonyl)phenyl]sulfonylbenzamide	CC1(C)CCC(c2ccc(Cl)cc2)=C(CN2CCN(c3ccc(C(=O)NS(=O)(=O)c4ccc(N[C@H](CCN5CCN(C(=O)CCCn6cc(COCCOCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)CC5)CSc5ccccc5)c(S(=O)(=O)C(F)(F)F)c4)cc3)CC2)C1	C71H82ClF3N12O12S3	BCL-2;BCL2L1	P10415/Q07817	VHL	US-20240398764-A1
TPD-VO68X8	PROTAC Bcl-xL degrader-3	PROTAC Bcl-xL degrader-3; 2471970-60-0; orb1983289; CHEMBL5418789; SCHEMBL22325102; EX-A8706; DA-66944; PD173425; HY-132997; CS-0311713	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCC(=O)N2CCN(C[C@]3(C)CCC(c4ccc(Cl)cc4)=C(CN4CCN(c5ccc(C(=O)NS(=O)(=O)c6ccc(N[C@H](CCN7CCOCC7)CSc7ccccc7)c(S(=O)(=O)C(F)(F)F)c6)cc5)CC4)C3)CC2)C(C)(C)C)cc1	C82H105ClF3N11O11S4	BCL-2;BCL2L1	P10415/Q07817	VHL	US-20240398764-A1
TPD-Y451PI	US20240398764A1_3	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CC2C(=O)[C@@H](NC(=O)CCCCCCC(=O)N2CCN(C[C@]3(C)CCC(c4ccc(Cl)cc4)=C(CN4CCN(c5ccc(C(=O)NS(=O)(=O)c6ccc(N[C@H](CCN7CCOCC7)CSc7ccccc7)c(S(=O)(=O)C(F)(F)F)c6)cc5)CC4)C3)CC2)C(C)(C)C)cc1	C83H106ClF3N10O11S4	BCL-2;BCL2L1	P10415/Q07817	VHL	US-20240398764-A1
TPD-AENNB5	SCHEMBL23959089	4-[4-[[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]methyl]phenyl]-N-[(1S,3S)-3-[(5-pentan-3-ylpyrazolo[1,5-a]pyrimidin-7-yl)amino]cyclopentyl]benzamide	CCC(CC)c1cc(N[C@H]2CC[C@H](NC(=O)c3ccc(-c4ccc(CNc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6=O)cc4)cc3)C2)n2nccc2n1	C43H44N8O5	CDK9	P50750	CRBN	WO-2021216828-A1
TPD-5N32RQ	SCHEMBL25477379	3-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]-N-[(1R,3R)-3-[(5-propylpyrazolo[1,5-a]pyrimidin-7-yl)amino]cyclopentyl]propanamide	CCCc1cc(N[C@@H]2CC[C@@H](NC(=O)CCOCCNc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)n2nccc2n1	C32H38N8O6	CDK9	P50750	CRBN	WO-2021216828-A1
TPD-0IMODV	SCHEMBL25477382	3-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]-N-[(1R,3R)-3-[(5-propylpyrazolo[1,5-a]pyrimidin-7-yl)amino]cyclopentyl]propanamide	CCCc1cc(N[C@@H]2CC[C@@H](NC(=O)CCOCCOCCNc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)n2nccc2n1	C34H42N8O7	CDK9	P50750	CRBN	WO-2021216828-A1
TPD-6167ZH	SCHEMBL25187677	3-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]-N-[(1R,3R)-3-[(5-propylpyrazolo[1,5-a]pyrimidin-7-yl)amino]cyclopentyl]propanamide	CCCc1cc(N[C@@H]2CC[C@@H](NC(=O)CCOCCOCCOCCNc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)n2nccc2n1	C36H46N8O8	CDK9	P50750	CRBN	WO-2021216828-A1
TPD-EQD7BO	SCHEMBL25193168	3-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethoxy]-N-[(1R,3R)-3-[(5-propylpyrazolo[1,5-a]pyrimidin-7-yl)amino]cyclopentyl]propanamide	CCCc1cc(N[C@@H]2CC[C@@H](NC(=O)CCOCCOCCOCCOCCNc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)n2nccc2n1	C38H50N8O9	CDK9	P50750	CRBN	WO-2021216828-A1
TPD-NJB8U8	SCHEMBL25477384	7-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]-N-[(1R,3R)-3-[(5-propylpyrazolo[1,5-a]pyrimidin-7-yl)amino]cyclopentyl]heptanamide	CCCc1cc(N[C@@H]2CC[C@@H](NC(=O)CCCCCCNc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)n2nccc2n1	C34H42N8O5	CDK9	P50750	CRBN	WO-2021216828-A1
TPD-1M0ZRA	SCHEMBL25189702	4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]-N-[(1R,3R)-3-[(5-propylpyrazolo[1,5-a]pyrimidin-7-yl)amino]cyclopentyl]butanamide	CCCc1cc(N[C@@H]2CC[C@@H](NC(=O)CCCNc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)n2nccc2n1	C31H36N8O5	CDK9	P50750	CRBN	WO-2021216828-A1
TPD-DHQW24	SCHEMBL25183569	10-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]-N-[(1R,3R)-3-[(5-propylpyrazolo[1,5-a]pyrimidin-7-yl)amino]cyclopentyl]decanamide	CCCc1cc(N[C@@H]2CC[C@@H](NC(=O)CCCCCCCCCNc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)n2nccc2n1	C37H48N8O5	CDK9	P50750	CRBN	WO-2021216828-A1
TPD-4U3JTR	SCHEMBL25197903	4-[4-[[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]methyl]phenyl]-N-[(1R,3R)-3-[(5-propylpyrazolo[1,5-a]pyrimidin-7-yl)amino]cyclopentyl]benzamide; SCHEMBL31291559	CCCc1cc(N[C@@H]2CC[C@@H](NC(=O)c3ccc(-c4ccc(CNc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6=O)cc4)cc3)C2)n2nccc2n1	C41H40N8O5	CDK9	P50750	CRBN	WO-2021216828-A1
TPD-VO48YM	SCHEMBL23959027	(2S,4R)-1-[(2S)-3,3-dimethyl-2-[2-[3-oxo-3-[[(1R,3R)-3-[(5-propylpyrazolo[1,5-a]pyrimidin-7-yl)amino]cyclopentyl]amino]propoxy]ethylamino]butanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CCCc1cc(N[C@@H]2CC[C@@H](NC(=O)CCOCCN[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCc3ccc(-c4scnc4C)cc3)C(C)(C)C)C2)n2nccc2n1	C41H57N9O5S	CDK9	P50750	VHL	WO-2021216828-A1
TPD-HO82KB	SCHEMBL23959182	(2S,4R)-1-[(2S)-3,3-dimethyl-2-[2-[2-[3-oxo-3-[[(1R,3R)-3-[(5-propylpyrazolo[1,5-a]pyrimidin-7-yl)amino]cyclopentyl]amino]propoxy]ethoxy]ethylamino]butanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CCCc1cc(N[C@@H]2CC[C@@H](NC(=O)CCOCCOCCN[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCc3ccc(-c4scnc4C)cc3)C(C)(C)C)C2)n2nccc2n1	C43H61N9O6S	CDK9	P50750	VHL	WO-2021216828-A1
TPD-SZWUHQ	SCHEMBL23959464	(2S,4R)-1-[(2S)-3,3-dimethyl-2-[2-[2-[2-[3-oxo-3-[[(1R,3R)-3-[(5-propylpyrazolo[1,5-a]pyrimidin-7-yl)amino]cyclopentyl]amino]propoxy]ethoxy]ethoxy]ethylamino]butanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CCCc1cc(N[C@@H]2CC[C@@H](NC(=O)CCOCCOCCOCCN[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCc3ccc(-c4scnc4C)cc3)C(C)(C)C)C2)n2nccc2n1	C45H65N9O7S	CDK9	P50750	VHL	WO-2021216828-A1
TPD-M79HR3	WO-2021216828-A1_KI-ARv3-D14	.	CCCc1cc(N[C@@H]2CC[C@@H](NC(=O)CCOCCOCCOCCOCCN[C@H](C(=O)N3C[C@H](O)CC3C(=O)NCc3ccc(-c4scnc4C)cc3)C(C)(C)C)C2)n2nccc2n1	C47H69N9O8S	CDK9	P50750	VHL	WO-2021216828-A1
TPD-CQ2G93	WO-2021216828-A1_KI-ARv3-D15	.	CCCc1cc(N[C@@H]2CC[C@@H](NC(=O)CCCCCCN[C@H](C(=O)N3C[C@H](O)CC3C(=O)NCc3ccc(-c4scnc4C)cc3)C(C)(C)C)C2)n2nccc2n1	C43H61N9O4S	CDK9	P50750	VHL	WO-2021216828-A1
TPD-FU8XEC	WO-2021216828-A1_KI-ARv3-D16	.	CCCc1cc(N[C@@H]2CC[C@@H](NC(=O)CCCCCCCN[C@H](C(=O)N3C[C@H](O)CC3C(=O)NCc3ccc(-c4scnc4C)cc3)C(C)(C)C)C2)n2nccc2n1	C44H63N9O4S	CDK9	P50750	VHL	WO-2021216828-A1
TPD-LE2OKS	WO-2021216828-A1_KI-ARv3-D17	.	CCCc1cc(N[C@@H]2CC[C@@H](NC(=O)CCCCCCCCCN[C@H](C(=O)N3C[C@H](O)CC3C(=O)NCc3ccc(-c4scnc4C)cc3)C(C)(C)C)C2)n2nccc2n1	C46H67N9O4S	CDK9	P50750	VHL	WO-2021216828-A1
TPD-XUNBVR	WO-2021216828-A1_KI-ARv3-D18	.	CCCc1cc(N[C@@H]2CC[C@@H](NC(=O)c3ccc(-c4ccc(CN[C@H](C(=O)N5C[C@H](O)CC5C(=O)NCc5ccc(-c6scnc6C)cc5)C(C)(C)C)cc4)cc3)C2)n2nccc2n1	C50H59N9O4S	CDK9	P50750	VHL	WO-2021216828-A1
TPD-D3XCMQ	WO-2022101603-A1_MN674	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](C)NC(=O)COCC(C)(COCCOCCNC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)COCCOCCNC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)cc1	C72H84Cl2N14O11S3	BRD2	P25440	CRBN	WO-2022101603-A1
TPD-9OQQ9U	WO-2022101603-A1_SIM1	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](O)NC(=O)COCC(C)(COCCOCCOCCNC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)COCCOCCOCCNC(=O)C[C@@H]2N=C(c3ccc(CI)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)cc1	C76H92ClIN14O14S3	BRD2	P25440	VHL	WO-2022101603-A1
TPD-SB4FWO	WO-2022101603-A1_SIM2	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](C)NC(=O)COCCOCC(C)(COCCOCCOCCNC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)COCCOCCOCCNC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)cc1	C78H96Cl2N14O14S3	BRD2	P25440	VHL	WO-2022101603-A1
TPD-Q8Q34M	WO-2022101603-A1_SIM3	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](C)NC(=O)COCC(C)(COCCOCCOCCOCCN=NC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)COCCOCCOCCOCCNC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)cc1	C80H99Cl2N15O15S3	BRD2	P25440	VHL	WO-2022101603-A1
TPD-V5EEF0	WO-2022101603-A1_SIM4	.	Cc1sc2c(c1C)C(c1ccc(Cl)cc1)=N[C@@H](CC(=O)NCCOCCOCCOCC(C)(COCCOCCOCCNC(=O)C[C@@H]1N=C(c3ccc(CI)cc3)c3c(sc(C)c3C)-n3c(C)nnc31)COCC(=O)NCCNc1cccc3c1C(=O)N(C1CCC(=O)NC1=O)C3=O)c1nnc(C)n1-2	C73H86ClIN14O14S2	BRD2	P25440	CRBN	WO-2022101603-A1
TPD-HCECB9	SIM5	2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]-N-[2-[2-[2-[2-[2-[2-[2-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]ethoxy]ethoxy]ethoxymethyl]-3-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethylamino]-2-oxoethoxy]ethoxy]-2-methylpropoxy]ethoxy]ethoxy]ethyl]acetamide; SCHEMBL29780150	Cc1sc2c(c1C)C(c1ccc(Cl)cc1)=N[C@@H](CC(=O)NCCOCCOCCOCC(C)(COCCOCCOCCNC(=O)C[C@@H]1N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc31)COCCOCC(=O)NCCNc1cccc3c1C(=O)N(C1CCC(=O)NC1=O)C3=O)c1nnc(C)n1-2	C74H88Cl2N14O15S2	BRD2	P25440	CRBN	WO-2022101603-A1
TPD-Q5S8N3	WO-2022101603-A1_SIM6	.	C=C1CCC(N2C(=O)c3cccc(NCCNC(=O)COCC(C)(COCCOCCOCCOCCNC(=O)C[C@@H]4N=C(c5ccc(Cl)cc5)c5c(sc(C)c5C)-n5c(C)nnc54)COCCOCCOCCOCCNC(=O)C[C@@H]4N=C(c5ccc(Cl)cc5)c5c(sc(C)c5C)-n5c(C)nnc54)c3C2=O)C(=O)N1	C77H94Cl2N14O15S2	BRD2	P25440	CRBN	WO-2022101603-A1
TPD-64RZD0	SCHEMBL30298154	(2S,4R)-1-[(2S)-2-[[2-[4-[2-[2,3-difluoro-6-(2-morpholin-4-yl-1,3-thiazol-4-yl)phenoxy]acetyl]piperazin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CN2CCN(C(=O)COc3c(-c4csc(N5CCOCC5)n4)ccc(F)c3F)CC2)C(C)(C)C)cc1	C44H54F2N8O7S2	AR-V7	P10275-3	VHL	WO-2023039601-A1
TPD-Q2M4VY	SCHEMBL30298157	(2S,4R)-1-[(2S)-2-[3-[4-[2-[2,3-difluoro-6-(2-morpholin-4-yl-1,3-thiazol-4-yl)phenoxy]acetyl]piperazin-1-yl]propanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCN2CCN(C(=O)COc3c(-c4csc(N5CCOCC5)n4)ccc(F)c3F)CC2)C(C)(C)C)cc1	C45H56F2N8O7S2	AR-V7	P10275-3	VHL	WO-2023039601-A1
TPD-DGL49A	WO-2023039601-A1_3	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)C2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCC(=O)N2CCCC(NC(=O)COc3c(-c4csc(N5CCOCC5)n4)ccc(F)c3F)C2)C(C)(C)C)cc1	C47H58F2N8O8S2	AR-V7	P10275-3	VHL	WO-2023039601-A1
TPD-F4IZDJ	WO-2023039601-A1_4	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)C2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCn2nncc2CCOc2c(-c3csc(N4CCOCC4)n3)ccc(F)c2F)C(C)(C)C)cc1	C45H55F2N9O6S2	AR-V7	P10275-3	VHL	WO-2023039601-A1
TPD-Q6ICBY	SCHEMBL30298155	N-[3-[2,3-difluoro-6-(2-morpholin-4-yl-1,3-thiazol-4-yl)phenoxy]cyclobutyl]-N'-[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]butanediamide; SCHEMBL31289439	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCC(=O)N[C@H]2C[C@H](Oc3c(-c4csc(N5CCOCC5)n4)ccc(F)c3F)C2)C(C)(C)C)cc1	C44H53F2N7O7S2	AR-V7	P10275-3	VHL	WO-2023039601-A1
TPD-U7K8MV	WO-2023039601-A1_6	.	COc1cc(C(=O)NCC2CN(C(=O)COc3c(-c4csc(N5CCOCC5)n4)ccc(F)c3F)C2)ccc1NC(=O)[C@@H]1N[C@@H](CC(C)(C)C)[C@](C#N)(c2ccc(Cl)cc2F)C1c1cccc(Cl)c1F	C50H49Cl2F4N7O6S	AR-V7	P10275-3	VHL	WO-2023039601-A1
TPD-SLO6YE	SCHEMBL30298159	(2R,3S,4R,5S)-3-(3-chloro-2-fluorophenyl)-4-(4-chloro-2-fluorophenyl)-4-cyano-N-[4-[[1-[2-[2,3-difluoro-6-(2-morpholin-4-yl-1,3-thiazol-4-yl)phenoxy]acetyl]piperidin-4-yl]methylcarbamoyl]-2-methoxyphenyl]-5-(2,2-dimethylpropyl)pyrrolidine-2-carboxamide	COc1cc(C(=O)NCC2CCN(C(=O)COc3c(-c4csc(N5CCOCC5)n4)ccc(F)c3F)CC2)ccc1NC(=O)[C@@H]1N[C@@H](CC(C)(C)C)[C@](C#N)(c2ccc(Cl)cc2F)[C@H]1c1cccc(Cl)c1F	C52H53Cl2F4N7O6S	AR-V7	P10275-3	VHL	WO-2023039601-A1
TPD-Y24E24	SCHEMBL30298142	(2R,3S,4R,5S)-3-(3-chloro-2-fluorophenyl)-4-(4-chloro-2-fluorophenyl)-4-cyano-N-[4-[2-[4-[2-[2,3-difluoro-6-(2-morpholin-4-yl-1,3-thiazol-4-yl)phenoxy]acetyl]piperazin-1-yl]ethylcarbamoyl]-2-methoxyphenyl]-5-(2,2-dimethylpropyl)pyrrolidine-2-carboxamide	COc1cc(C(=O)NCCN2CCN(C(=O)COc3c(-c4csc(N5CCOCC5)n4)ccc(F)c3F)CC2)ccc1NC(=O)[C@@H]1N[C@@H](CC(C)(C)C)[C@](C#N)(c2ccc(Cl)cc2F)[C@H]1c1cccc(Cl)c1F	C52H54Cl2F4N8O6S	AR-V7	P10275-3	VHL	WO-2023039601-A1
TPD-DJRR8H	WO-2023039601-A1_9	.	COc1cc(C(=O)N2CCC(NC(=O)COc3c(-c4csc(N5CCOCC5)n4)ccc(F)c3F)CC2)ccc1NC(=O)[C@@H]1NC(C(C)(C)C)[C@](C#N)(c2ccc(Cl)cc2F)[C@H]1c1cccc(Cl)c1F	C50H49Cl2F4N7O6S	AR-V7	P10275-3	VHL	WO-2023039601-A1
TPD-QIWT0V	SCHEMBL30298158	(2R,3S,4R,5S)-3-(3-chloro-2-fluorophenyl)-4-(4-chloro-2-fluorophenyl)-4-cyano-N-[4-[2-[2-[4-[2-[2,3-difluoro-6-(2-morpholin-4-yl-1,3-thiazol-4-yl)phenoxy]ethyl]triazol-1-yl]ethoxy]ethylcarbamoyl]-2-methoxyphenyl]-5-(2,2-dimethylpropyl)pyrrolidine-2-carboxamide	COc1cc(C(=O)NCCOCCn2cc(CCOc3c(-c4csc(N5CCOCC5)n4)ccc(F)c3F)nn2)ccc1NC(=O)[C@@H]1N[C@@H](CC(C)(C)C)[C@](C#N)(c2ccc(Cl)cc2F)[C@H]1c1cccc(Cl)c1F	C52H53Cl2F4N9O6S	AR-V7	P10275-3	VHL	WO-2023039601-A1
TPD-VF4GWW	WO-2023039601-A1_11	.	C[C@@H]1CN(CC(=O)N2CC(C)(C)c3nc(CO)c(Cc4ccc(F)cc4)cc32)C(C(=O)N2CCN(C(=O)COCOCCOc3cc(-c4csc(N5CCOCC5)n4)cc(F)c3F)CC2)CN1	C47H57F3N8O8S	AR-V7	P10275-3	VHL	WO-2023039601-A1
TPD-2VAG9Y	WO-2023039601-A1_12	.	C[C@@H]1CN(CC(=O)N2CC(C)(C)c3nc(CO)c(Cc4ccc(F)cc4)cc32)C(C(=O)N2CCOCC2C(=O)NCCOCOCCOc2cc(-c3csc(N4CCOCC4)n3)cc(F)c2F)CN1	C48H59F3N8O9S	AR-V7	P10275-3	VHL	WO-2023039601-A1
TPD-A1VICZ	WO-2023039601-A1_13	.	C[C@@H]1CN(CC(=O)N2CC(C)(C)c3nc(CO)c(Cc4ccc(F)cc4)cc32)[C@@H](CN2CCOCC2C(=O)NCCOCCOc2c(-c3csc(N4CCOCC4)n3)ccc(F)c2F)CN1	C47H59F3N8O7S	AR-V7	P10275-3	VHL	WO-2023039601-A1
TPD-3P8CI5	WO-2023039601-A1_14	(3S)-N-[2-[2-[2-[2,3-difluoro-6-(2-morpholin-4-yl-1,3-thiazol-4-yl)phenoxy]ethoxy]ethoxy]ethyl]-4-[[(2R,5R)-1-[2-[6-[(4-fluorophenyl)methyl]-5-(hydroxymethyl)-3,3-dimethyl-2H-pyrrolo[3,2-b]pyridin-1-yl]-2-oxoethyl]-5-methylpiperazin-2-yl]methyl]morpholine-3-carboxamide	C[C@@H]1CN(CC(=O)N2CC(C)(C)c3nc(CO)c(Cc4ccc(F)cc4)cc32)[C@@H](CN2CCOC[C@H]2C(=O)NCCOCCOCCOc2c(-c3csc(N4CCOCC4)n3)ccc(F)c2F)CN1	C49H63F3N8O8S	AR-V7	P10275-3	VHL	WO-2023039601-A1
TPD-V8KM0F	WO-2023039601-A1_15	.	C[C@@H]1CN(CC(=O)N2CC(C)(C)c3nc(CO)c(Cc4ccc(F)cc4)cc32)[C@@H](CN2CCOC[C@H]2C(=O)NCCOCCOCCCOCCOc2c(-c3csc(N4CCOCC4)n3)ccc(F)c2F)CN1	C52H69F3N8O9S	AR-V7	P10275-3	VHL	WO-2023039601-A1
TPD-XTIZT5	WO-2023039601-A1_16	.	C[C@@H]1CN(CC(=O)N2CC(C)(C)c3nc(CO)c(Cc4ccc(F)cc4)cc32)[C@@H](CN2CCOC[C@H]2C(=O)NCCCNC(=O)COc2c(-c3csc(N4CCOCC4)n3)ccc(F)c2F)CN1	C48H60F3N9O7S	AR-V7	P10275-3	VHL	WO-2023039601-A1
TPD-PMGQ3I	WO-2023039601-A1_17	.	C[C@@H]1CN(CC(=O)N2CC(C)(C)c3nc(CO)c(Cc4ccc(F)cc4)cc32)[C@@H](CN2CCOCC2C(=O)NCCCCNC(=O)COc2c(-c3csc(N4CCOCC4)n3)ccc(F)c2F)CN1	C49H62F3N9O7S	AR-V7	P10275-3	VHL	WO-2023039601-A1
TPD-J16FV7	WO-2023039601-A1_18	.	C[C@@H]1CN(CC(=O)N2CC(C)(C)c3nc(CO)c(Cc4ccc(F)cc4)cc32)[C@@H](CN2CCOCC2C(=O)NCCCCCCNC(=O)COc2c(-c3csc(N4CCOCC4)n3)ccc(F)c2F)CN1	C51H66F3N9O7S	AR-V7	P10275-3	VHL	WO-2023039601-A1
TPD-1AA258	WO-2023039601-A1_20	.	C[C@@H]1CN(CC(=O)N2CC(C)(C)c3nc(CO)c(Cc4ccc(F)cc4)cc32)[C@@H](CN2CCOCC2C(=O)NCCCCCCCCCCNC(=O)COc2c(-c3csc(N4CCOCC4)n3)ccc(F)c2F)CN1	C55H74F3N9O7S	AR-V7	P10275-3	VHL	WO-2023039601-A1
TPD-RGPF6Y	WO-2023039601-A1_21	.	C[C@@H]1CN(CC(=O)N2CC(C)(C)c3nc(CO)c(Cc4ccc(F)cc4)cc32)[C@@H](CN2CCOC[C@H]2C(=O)NCCCCCCCCCCCCCCNC(=O)COc2c(-c3csc(N4CCOCC4)n3)ccc(F)c2F)CN1	C59H82F3N9O7S	AR-V7	P10275-3	VHL	WO-2023039601-A1
TPD-O36CXE	WO-2023039601-A1_22	(4R)-N-[3-[2-[4-[2-[2,3-difluoro-6-(2-morpholin-4-yl-1,3-thiazol-4-yl)phenoxy]acetyl]piperazin-1-yl]ethylamino]-1-[4-(4-methyl-1,2-thiazol-5-yl)phenyl]-3-oxopropyl]-1-[(2S)-2-[(1-fluorocyclopropanecarbonyl)amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide	Cc1cnsc1-c1ccc(C(CC(=O)NCCN2CCN(C(=O)COc3c(-c4csc(N5CCOCC5)n4)ccc(F)c3F)CC2)NC(=O)C2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)C)cc1	C49H60F3N9O8S2	AR-V7	P10275-3	VHL	WO-2023039601-A1
TPD-8MILP0	WO-2023039601-A1_23	(4R)-N-[3-[[4-[3-[[2-[2,3-difluoro-6-(2-morpholin-4-yl-1,3-thiazol-4-yl)phenoxy]acetyl]amino]piperidin-1-yl]-4-oxobutyl]amino]-1-[4-(4-methyl-1,2-thiazol-5-yl)phenyl]-3-oxopropyl]-1-[(2S)-2-[(1-fluorocyclopropanecarbonyl)amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide	Cc1cnsc1-c1ccc(C(CC(=O)NCCCC(=O)N2CCCC(NC(=O)COc3c(-c4csc(N5CCOCC5)n4)ccc(F)c3F)C2)NC(=O)C2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)C)cc1	C52H64F3N9O9S2	AR-V7	P10275-3	VHL	WO-2023039601-A1
TPD-VQA3ER	WO-2023039601-A1_24	.	Cc1cnsc1-c1ccc(C(CC(=O)NCCCCn2nncc2CCOC2C(c3csc(N4CCOCC4)n3)=CC=C(F)C2F)NC(=O)C2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)C)cc1	C49H61F3N10O7S2	AR-V7	P10275-3	VHL	WO-2023039601-A1
TPD-8E0D8Q	WO-2023039601-A1_25	(4R)-N-[3-[[2-[[3-[2,3-difluoro-6-(2-morpholin-4-yl-1,3-thiazol-4-yl)phenoxy]cyclobutyl]amino]-2-oxoethyl]amino]-1-[4-(4-methyl-1,2-thiazol-5-yl)phenyl]-3-oxopropyl]-1-[(2S)-2-[(1-fluorocyclopropanecarbonyl)amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide	Cc1cnsc1-c1ccc(C(CC(=O)NCC(=O)N[C@H]2C[C@H](Oc3c(-c4csc(N5CCOCC5)n4)ccc(F)c3F)C2)NC(=O)C2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)C)cc1	C47H55F3N8O8S2	AR-V7	P10275-3	VHL	WO-2023039601-A1
TPD-T65HLD	SCHEMBL31289531	4-[2-[4-[2-[2,3-Difluoro-6-(2-morpholin-4-yl-1,3-thiazol-4-yl)phenoxy]acetyl]piperazin-1-yl]ethylamino]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	O=C1CCC(N2C(=O)c3cccc(NCCN4CCN(C(=O)COc5c(-c6csc(N7CCOCC7)n6)ccc(F)c5F)CC4)c3C2=O)C(=O)N1	C34H35F2N7O7S	AR-V7	P10275-3	CRBN	WO-2023039601-A1
TPD-D0PB14	SCHEMBL31289429	2-[2,3-difluoro-6-(2-morpholin-4-yl-1,3-thiazol-4-yl)phenoxy]-N-[1-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]butanoyl]piperidin-3-yl]acetamide	O=C1CCC(N2C(=O)c3cccc(NCCCC(=O)N4CCCC(NC(=O)COc5c(-c6csc(N7CCOCC7)n6)ccc(F)c5F)C4)c3C2=O)C(=O)N1	C37H39F2N7O8S	AR-V7	P10275-3	CRBN	WO-2023039601-A1
TPD-P734UQ	SCHEMBL31289444	4-[4-[5-[2-[2,3-Difluoro-6-(2-morpholin-4-yl-1,3-thiazol-4-yl)phenoxy]ethyl]triazol-1-yl]butylamino]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	O=C1CCC(N2C(=O)c3cccc(NCCCCn4nncc4CCOc4c(-c5csc(N6CCOCC6)n5)ccc(F)c4F)c3C2=O)C(=O)N1	C34H34F2N8O6S	AR-V7	P10275-3	CRBN	WO-2023039601-A1
TPD-Z94MBE	SCHEMBL31289430	N-[3-[2,3-difluoro-6-(2-morpholin-4-yl-1,3-thiazol-4-yl)phenoxy]cyclobutyl]-4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]butanamide	O=C1CCC(N2C(=O)c3cccc(NCCCC(=O)N[C@H]4C[C@H](Oc5c(-c6csc(N7CCOCC7)n6)ccc(F)c5F)C4)c3C2=O)C(=O)N1	C34H34F2N6O7S	AR-V7	P10275-3	CRBN	WO-2023039601-A1
TPD-MOY0R4	SCHEMBL31203642	2-[2,3-difluoro-6-(2-morpholin-4-yl-1,3-thiazol-4-yl)phenoxy]-N-[5-[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]-5-oxopentyl]acetamide	O=C(COc1c(-c2csc(N3CCOCC3)n2)ccc(F)c1F)NCCCCC(=O)N1CCN(c2cc3c(cc2F)C(=O)N(C2CCC(=O)NC2=O)C3=O)CC1	C37H38F3N7O8S	AR-V7	P10275-3	CRBN	WO-2023039604-A1
TPD-2CAT6Y	SCHEMBL31203634	5-[4-[2-[2-[2-[2-[2,3-Difluoro-6-(2-morpholin-4-yl-1,3-thiazol-4-yl)phenoxy]ethoxy]ethoxy]ethoxy]acetyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)-6-fluoroisoindole-1,3-dione	O=C1CCC(N2C(=O)c3cc(F)c(N4CCN(C(=O)COCCOCCOCCOc5c(-c6csc(N7CCOCC7)n6)ccc(F)c5F)CC4)cc3C2=O)C(=O)N1	C38H41F3N6O10S	AR-V7	P10275-3	CRBN	WO-2023039604-A1
TPD-Y9U216	SCHEMBL31203525	5-[4-[4-[2-[2,3-Difluoro-6-(2-morpholin-4-yl-1,3-thiazol-4-yl)phenoxy]ethylamino]butanoyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)-6-fluoroisoindole-1,3-dione	O=C1CCC(N2C(=O)c3cc(F)c(N4CCN(C(=O)CCCNCCOc5c(-c6csc(N7CCOCC7)n6)ccc(F)c5F)CC4)cc3C2=O)C(=O)N1	C36H38F3N7O7S	AR-V7	P10275-3	CRBN	WO-2023039604-A1
TPD-KR7BOD	SCHEMBL31203627	5-[4-[5-[2-[2,3-Difluoro-6-(2-morpholin-4-yl-1,3-thiazol-4-yl)phenoxy]ethylamino]pentanoyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)-6-fluoroisoindole-1,3-dione	O=C1CCC(N2C(=O)c3cc(F)c(N4CCN(C(=O)CCCCNCCOc5c(-c6csc(N7CCOCC7)n6)ccc(F)c5F)CC4)cc3C2=O)C(=O)N1	C37H40F3N7O7S	AR-V7	P10275-3	CRBN	WO-2023039604-A1
TPD-LPRQSQ	SCHEMBL31203601	5-[4-[6-[2-[2,3-Difluoro-6-(2-morpholin-4-yl-1,3-thiazol-4-yl)phenoxy]ethylamino]hexanoyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)-6-fluoroisoindole-1,3-dione	O=C1CCC(N2C(=O)c3cc(F)c(N4CCN(C(=O)CCCCCNCCOc5c(-c6csc(N7CCOCC7)n6)ccc(F)c5F)CC4)cc3C2=O)C(=O)N1	C38H42F3N7O7S	AR-V7	P10275-3	CRBN	WO-2023039604-A1
TPD-0YMFL0	SCHEMBL31203643	5-[4-[7-[2-[2,3-Difluoro-6-(2-morpholin-4-yl-1,3-thiazol-4-yl)phenoxy]ethylamino]heptanoyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)-6-fluoroisoindole-1,3-dione	O=C1CCC(N2C(=O)c3cc(F)c(N4CCN(C(=O)CCCCCCNCCOc5c(-c6csc(N7CCOCC7)n6)ccc(F)c5F)CC4)cc3C2=O)C(=O)N1	C39H44F3N7O7S	AR-V7	P10275-3	CRBN	WO-2023039604-A1
TPD-RVMHFJ	SCHEMBL31203615	5-[4-[11-[2-[2,3-Difluoro-6-(2-morpholin-4-yl-1,3-thiazol-4-yl)phenoxy]ethylamino]undecanoyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)-6-fluoroisoindole-1,3-dione	O=C1CCC(N2C(=O)c3cc(F)c(N4CCN(C(=O)CCCCCCCCCCNCCOc5c(-c6csc(N7CCOCC7)n6)ccc(F)c5F)CC4)cc3C2=O)C(=O)N1	C43H52F3N7O7S	AR-V7	P10275-3	CRBN	WO-2023039604-A1
TPD-1UQBQR	SCHEMBL31203556	5-[4-[2-[2-[2-[2-[2,3-Difluoro-6-(2-morpholin-4-yl-1,3-thiazol-4-yl)phenoxy]ethylamino]ethoxy]ethoxy]acetyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)-6-fluoroisoindole-1,3-dione	O=C1CCC(N2C(=O)c3cc(F)c(N4CCN(C(=O)COCCOCCNCCOc5c(-c6csc(N7CCOCC7)n6)ccc(F)c5F)CC4)cc3C2=O)C(=O)N1	C38H42F3N7O9S	AR-V7	P10275-3	CRBN	WO-2023039604-A1
TPD-PAA1Q2	SCHEMBL31203628	5-[4-[5-[2,3-Difluoro-6-(2-morpholin-4-yl-1,3-thiazol-4-yl)phenoxy]pentyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)-6-fluoroisoindole-1,3-dione	O=C1CCC(N2C(=O)c3cc(F)c(N4CCN(CCCCCOc5c(-c6csc(N7CCOCC7)n6)ccc(F)c5F)CC4)cc3C2=O)C(=O)N1	C35H37F3N6O6S	AR-V7	P10275-3	CRBN	WO-2023039604-A1
TPD-QK8EOK	SCHEMBL31203620	5-[4-[7-[2,3-Difluoro-6-(2-morpholin-4-yl-1,3-thiazol-4-yl)phenoxy]heptyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)-6-fluoroisoindole-1,3-dione	O=C1CCC(N2C(=O)c3cc(F)c(N4CCN(CCCCCCCOc5c(-c6csc(N7CCOCC7)n6)ccc(F)c5F)CC4)cc3C2=O)C(=O)N1	C37H41F3N6O6S	AR-V7	P10275-3	CRBN	WO-2023039604-A1
TPD-FYVX39	SCHEMBL31203633	2-[2,3-difluoro-6-(2-morpholin-4-yl-1,3-thiazol-4-yl)phenoxy]-N-[7-[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]heptyl]acetamide	O=C(COc1c(-c2csc(N3CCOCC3)n2)ccc(F)c1F)NCCCCCCCN1CCN(c2cc3c(cc2F)C(=O)N(C2CCC(=O)NC2=O)C3=O)CC1	C39H44F3N7O7S	AR-V7	P10275-3	CRBN	WO-2023039604-A1
TPD-FW70CM	SCHEMBL31203651	2-[2,3-difluoro-6-(2-morpholin-4-yl-1,3-thiazol-4-yl)phenoxy]-N-[7-[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]-7-oxoheptyl]acetamide	O=C(COc1c(-c2csc(N3CCOCC3)n2)ccc(F)c1F)NCCCCCCC(=O)N1CCN(c2cc3c(cc2F)C(=O)N(C2CCC(=O)NC2=O)C3=O)CC1	C39H42F3N7O8S	AR-V7	P10275-3	CRBN	WO-2023039604-A1
TPD-AKBEIB	SCHEMBL31203644	5-[4-[[1-[2-[2,3-Difluoro-6-(2-morpholin-4-yl-1,3-thiazol-4-yl)phenoxy]acetyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)-6-fluoroisoindole-1,3-dione	O=C1CCC(N2C(=O)c3cc(F)c(N4CCN(CC5CCN(C(=O)COc6c(-c7csc(N8CCOCC8)n7)ccc(F)c6F)CC5)CC4)cc3C2=O)C(=O)N1	C38H40F3N7O7S	AR-V7	P10275-3	CRBN	WO-2023039604-A1
TPD-D22SRJ	SCHEMBL31203624	5-[4-[[1-[6-[2,3-Difluoro-6-(2-morpholin-4-yl-1,3-thiazol-4-yl)phenoxy]pyridazin-3-yl]piperidin-4-yl]methyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)-6-fluoroisoindole-1,3-dione	O=C1CCC(N2C(=O)c3cc(F)c(N4CCN(CC5CCN(c6ccc(Oc7c(-c8csc(N9CCOCC9)n8)ccc(F)c7F)nn6)CC5)CC4)cc3C2=O)C(=O)N1	C40H40F3N9O6S	AR-V7	P10275-3	CRBN	WO-2023039604-A1
TPD-2NDOY0	SCHEMBL31203607	2-[2,3-difluoro-6-(2-morpholin-4-yl-1,3-thiazol-4-yl)phenoxy]-N-[4-[[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]amino]butyl]acetamide	O=C(COc1c(-c2csc(N3CCOCC3)n2)ccc(F)c1F)NCCCCNc1cc2c(cc1F)C(=O)N(C1CCC(=O)NC1=O)C2=O	C32H31F3N6O7S	AR-V7	P10275-3	CRBN	WO-2023039604-A1
TPD-YU4E1C	SCHEMBL31203598	2-[2,3-difluoro-6-(2-morpholin-4-yl-1,3-thiazol-4-yl)phenoxy]-N-[6-[[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]amino]hexyl]acetamide	O=C(COc1c(-c2csc(N3CCOCC3)n2)ccc(F)c1F)NCCCCCCNc1cc2c(cc1F)C(=O)N(C1CCC(=O)NC1=O)C2=O	C34H35F3N6O7S	AR-V7	P10275-3	CRBN	WO-2023039604-A1
TPD-V1XVJ4	SCHEMBL31203579	2-[2,3-difluoro-6-(2-morpholin-4-yl-1,3-thiazol-4-yl)phenoxy]-N-[8-[[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]amino]octyl]acetamide	O=C(COc1c(-c2csc(N3CCOCC3)n2)ccc(F)c1F)NCCCCCCCCNc1cc2c(cc1F)C(=O)N(C1CCC(=O)NC1=O)C2=O	C36H39F3N6O7S	AR-V7	P10275-3	CRBN	WO-2023039604-A1
TPD-YHZ5R6	SCHEMBL31203614	2-[2,3-difluoro-6-(2-morpholin-4-yl-1,3-thiazol-4-yl)phenoxy]-N-[10-[[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]amino]decyl]acetamide	O=C(COc1c(-c2csc(N3CCOCC3)n2)ccc(F)c1F)NCCCCCCCCCCNc1cc2c(cc1F)C(=O)N(C1CCC(=O)NC1=O)C2=O	C38H43F3N6O7S	AR-V7	P10275-3	CRBN	WO-2023039604-A1
TPD-9E26U6	SCHEMBL31203557	2-[2,3-difluoro-6-(2-morpholin-4-yl-1,3-thiazol-4-yl)phenoxy]-N-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]amino]ethoxy]ethoxy]ethyl]acetamide	O=C(COc1c(-c2csc(N3CCOCC3)n2)ccc(F)c1F)NCCOCCOCCNc1cc2c(cc1F)C(=O)N(C1CCC(=O)NC1=O)C2=O	C34H35F3N6O9S	AR-V7	P10275-3	CRBN	WO-2023039604-A1
TPD-WAB12S	SCHEMBL31203645	2-[2,3-difluoro-6-(2-morpholin-4-yl-1,3-thiazol-4-yl)phenoxy]-N-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]amino]ethoxy]ethoxy]ethoxy]ethyl]acetamide	O=C(COc1c(-c2csc(N3CCOCC3)n2)ccc(F)c1F)NCCOCCOCCOCCNc1cc2c(cc1F)C(=O)N(C1CCC(=O)NC1=O)C2=O	C36H39F3N6O10S	AR-V7	P10275-3	CRBN	WO-2023039604-A1
TPD-SRSB4V	SCHEMBL31203573	2-[2,3-difluoro-6-[2-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)-1,3-thiazol-4-yl]phenoxy]-N-[5-[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]-5-oxopentyl]acetamide	O=C(COc1c(-c2csc(N3CC4CCC(C3)O4)n2)ccc(F)c1F)NCCCCC(=O)N1CCN(c2cc3c(cc2F)C(=O)N(C2CCC(=O)NC2=O)C3=O)CC1	C39H40F3N7O8S	AR-V7	P10275-3	CRBN	WO-2023039604-A1
TPD-67VH02	SCHEMBL31203611	2-[2,3-difluoro-6-[2-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)-1,3-thiazol-4-yl]phenoxy]-N-[7-[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]-7-oxoheptyl]acetamide	O=C(COc1c(-c2csc(N3CC4CCC(C3)O4)n2)ccc(F)c1F)NCCCCCCC(=O)N1CCN(c2cc3c(cc2F)C(=O)N(C2CCC(=O)NC2=O)C3=O)CC1	C41H44F3N7O8S	AR-V7	P10275-3	CRBN	WO-2023039604-A1
TPD-QHFF54	SCHEMBL31203763	2-[2,3-difluoro-6-(2-morpholin-4-yl-1,3-thiazol-4-yl)phenoxy]-N-[11-[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]-11-oxoundecyl]acetamide	O=C(COc1c(-c2csc(N3CCOCC3)n2)ccc(F)c1F)NCCCCCCCCCCC(=O)N1CCN(c2cc3c(cc2F)C(=O)N(C2CCC(=O)NC2=O)C3=O)CC1	C43H50F3N7O8S	AR-V7	P10275-3	CRBN	WO-2023039604-A1
TPD-ERZ7PM	SCHEMBL31203650	2-[2,3-difluoro-6-[2-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)-1,3-thiazol-4-yl]phenoxy]-N-[11-[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]-11-oxoundecyl]acetamide	O=C(COc1c(-c2csc(N3CC4CCC(C3)O4)n2)ccc(F)c1F)NCCCCCCCCCCC(=O)N1CCN(c2cc3c(cc2F)C(=O)N(C2CCC(=O)NC2=O)C3=O)CC1	C45H52F3N7O8S	AR-V7	P10275-3	CRBN	WO-2023039604-A1
TPD-3127SW	SCHEMBL31203616	2-[2,3-difluoro-6-[2-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)-1,3-thiazol-4-yl]phenoxy]-N-[10-[[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]amino]decyl]acetamide	O=C(COc1c(-c2csc(N3CC4CCC(C3)O4)n2)ccc(F)c1F)NCCCCCCCCCCNc1cc2c(cc1F)C(=O)N(C1CCC(=O)NC1=O)C2=O	C40H45F3N6O7S	AR-V7	P10275-3	CRBN	WO-2023039604-A1
TPD-U3KXQI	SCHEMBL31203589	5-[4-[2-[2-[2-[2,3-Difluoro-6-(2-morpholin-4-yl-1,3-thiazol-4-yl)phenoxy]ethoxy]ethoxy]ethoxy]butylamino]-2-(2,6-dioxopiperidin-3-yl)-6-fluoroisoindole-1,3-dione	O=C1CCC(N2C(=O)c3cc(F)c(NCCCCOCCOCCOCCOc4c(-c5csc(N6CCOCC6)n5)ccc(F)c4F)cc3C2=O)C(=O)N1	C36H40F3N5O9S	AR-V7	P10275-3	CRBN	WO-2023039604-A1
TPD-68CCA1	SCHEMBL31203530	2-[2,3-difluoro-6-(2-morpholin-4-yl-1,3-thiazol-4-yl)phenoxy]-N-[2-[2-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]-2-oxoethoxy]ethoxy]ethyl]acetamide	O=C(COc1c(-c2csc(N3CCOCC3)n2)ccc(F)c1F)NCCOCCOCC(=O)N1CCN(c2cc3c(cc2F)C(=O)N(C2CCC(=O)NC2=O)C3=O)CC1	C38H40F3N7O10S	AR-V7	P10275-3	CRBN	WO-2023039604-A1
TPD-MIJCXN	SCHEMBL31203656	5-[4-[5-[2,3-Difluoro-6-(2-morpholin-4-yl-1,3-thiazol-4-yl)phenoxy]pentanoyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)-6-fluoroisoindole-1,3-dione	O=C1CCC(N2C(=O)c3cc(F)c(N4CCN(C(=O)CCCCOc5c(-c6csc(N7CCOCC7)n6)ccc(F)c5F)CC4)cc3C2=O)C(=O)N1	C35H35F3N6O7S	AR-V7	P10275-3	CRBN	WO-2023039604-A1
TPD-1M3I0B	SCHEMBL31203547	5-[4-[7-[2,3-Difluoro-6-(2-morpholin-4-yl-1,3-thiazol-4-yl)phenoxy]heptanoyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)-6-fluoroisoindole-1,3-dione	O=C1CCC(N2C(=O)c3cc(F)c(N4CCN(C(=O)CCCCCCOc5c(-c6csc(N7CCOCC7)n6)ccc(F)c5F)CC4)cc3C2=O)C(=O)N1	C37H39F3N6O7S	AR-V7	P10275-3	CRBN	WO-2023039604-A1
TPD-DMNKJV	SCHEMBL31203662	5-[4-[8-[2,3-Difluoro-6-(2-morpholin-4-yl-1,3-thiazol-4-yl)phenoxy]octanoyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)-6-fluoroisoindole-1,3-dione	O=C1CCC(N2C(=O)c3cc(F)c(N4CCN(C(=O)CCCCCCCOc5c(-c6csc(N7CCOCC7)n6)ccc(F)c5F)CC4)cc3C2=O)C(=O)N1	C38H41F3N6O7S	AR-V7	P10275-3	CRBN	WO-2023039604-A1
TPD-2J7HAI	SCHEMBL31203759	5-[4-[11-[2,3-Difluoro-6-(2-morpholin-4-yl-1,3-thiazol-4-yl)phenoxy]undecanoyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)-6-fluoroisoindole-1,3-dione	O=C1CCC(N2C(=O)c3cc(F)c(N4CCN(C(=O)CCCCCCCCCCOc5c(-c6csc(N7CCOCC7)n6)ccc(F)c5F)CC4)cc3C2=O)C(=O)N1	C41H47F3N6O7S	AR-V7	P10275-3	CRBN	WO-2023039604-A1
TPD-A67QCB	SCHEMBL31203565	5-[4-[2-[2-[2-[2,3-Difluoro-6-(2-morpholin-4-yl-1,3-thiazol-4-yl)phenoxy]ethoxy]ethoxy]acetyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)-6-fluoroisoindole-1,3-dione	O=C1CCC(N2C(=O)c3cc(F)c(N4CCN(C(=O)COCCOCCOc5c(-c6csc(N7CCOCC7)n6)ccc(F)c5F)CC4)cc3C2=O)C(=O)N1	C36H37F3N6O9S	AR-V7	P10275-3	CRBN	WO-2023039604-A1
TPD-JUK1Q9	WO-2023039604-A1_Scheme3.Example10	.	O=C1CCC(N2C(=O)c3ccc(N4CCN(C(=O)COCCOCCOCCOc5c(-c6csc(N7CCOCC7)n6)ccc(F)c5F)CC4)cc3C2=O)C(=O)N1	C38H42F2N6O10S	AR-V7	P10275-3	CRBN	WO-2023039604-A1
TPD-M9EPDY	SCHEMBL25143321	4-[2-[2-[2-[2-[2-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethylamino]-2-methyl-N-(5-phenyl-1,3-thiazol-2-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCOCCOCCOCCNc5ccc(C(=O)Nc6ncc(-c7ccccc7)s6)c(C)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C55H69N11O9S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-NH1DUN	SCHEMBL25143286	4-[2-[2-[2-[2-[2-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethylamino]-2-methyl-N-(5-methyl-1,3-thiazol-2-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCOCCOCCOCCNc5ccc(C(=O)Nc6ncc(C)s6)c(C)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C50H67N11O9S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-33VX2X	WO-2023061440-A1_CPD-003	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCOCCOCCOCCNc5ccc(C(=O)Nc6ncc(C(F)(F)F)s6)c(C)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C50H64F3N11O9S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-TT41DV	SCHEMBL25142802	4-[2-[2-[2-[2-[2-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethylamino]-2-methyl-N-(1,3-thiazol-2-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCOCCOCCOCCNc5ccc(C(=O)Nc6nccs6)c(C)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C49H65N11O9S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-WEHTRJ	SCHEMBL25142784	4-[2-[2-[2-[2-[2-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethylamino]-N-(5-chloro-1,3-thiazol-2-yl)-2-methylbenzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCOCCOCCOCCNc5ccc(C(=O)Nc6ncc(Cl)s6)c(C)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C49H64ClN11O9S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-8BHQT6	SCHEMBL25143227	4-[2-[2-[2-[2-[2-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethylamino]-2-methyl-N-(5-propan-2-yl-1,3-thiazol-2-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCOCCOCCOCCNc5ccc(C(=O)Nc6ncc(C(C)C)s6)c(C)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C52H71N11O9S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-792MGW	SCHEMBL25142769	4-[2-[2-[2-[2-[2-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethylamino]-2-methyl-N-(4-phenyl-1,3-thiazol-2-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCOCCOCCOCCNc5ccc(C(=O)Nc6nc(-c7ccccc7)cs6)c(C)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C55H69N11O9S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-ZWX00H	SCHEMBL25142936	4-N-[2-[2-[2-[2-[2-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethyl]-2-methyl-1-N-(5-methyl-1,3-thiazol-2-yl)benzene-1,4-dicarboxamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCOCCOCCOCCNC(=O)c5ccc(C(=O)Nc6ncc(C)s6)c(C)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C51H67N11O10S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-V6C648	WO-2023061440-A1_CPD-009	4-N-[5-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]pentyl]-2-methyl-1-N-(5-methyl-1,3-thiazol-2-yl)benzene-1,4-dicarboxamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCCCCNC(=O)c5ccc(C(=O)Nc6ncc(C)s6)c(C)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C44H53N11O5S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-NB48T8	SCHEMBL25142749	4-N-[2-[2-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]ethyl]-2-methyl-1-N-(5-methyl-1,3-thiazol-2-yl)benzene-1,4-dicarboxamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCNC(=O)c5ccc(C(=O)Nc6ncc(C)s6)c(C)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H55N11O7S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-5ZGTCZ	SCHEMBL25142971	4-N-[2-[2-[2-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]ethoxy]ethyl]-2-methyl-1-N-(5-methyl-1,3-thiazol-2-yl)benzene-1,4-dicarboxamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCOCCNC(=O)c5ccc(C(=O)Nc6ncc(C)s6)c(C)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H59N11O8S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-WQ9PKA	WO-2023061440-A1_CPD-012	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCOCCOCCOCCNC(=O)c5ccc(C)c(C(=O)Nc6ncc(C)s6)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C51H67N11O10S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-F8FKH8	SCHEMBL25142729	4-[[2-[2-[2-[2-[2-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethylamino]-2-oxoethyl]amino]-2-methyl-N-(5-methyl-1,3-thiazol-2-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCOCCOCCNC(=O)CNc5ccc(C(=O)Nc6ncc(C)s6)c(C)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C50H66N12O9S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-H5CQHM	SCHEMBL25142731	4-[[2-[2-[2-[2-[2-[2-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethylamino]-2-oxoethyl]amino]-2-methyl-N-(5-methyl-1,3-thiazol-2-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCOCCOCCOCCNC(=O)CNc5ccc(C(=O)Nc6ncc(C)s6)c(C)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C52H70N12O10S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-J5LH05	WO-2023061440-A1_CPD-015	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCCCCNC(=O)CNc5ccc(C(=O)Nc6ncc(C)s6)c(C)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H56N12O5S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-GYG8TJ	SCHEMBL25142734	4-[[2-[7-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]heptylamino]-2-oxoethyl]amino]-2-methyl-N-(5-methyl-1,3-thiazol-2-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCCCCCCNC(=O)CNc5ccc(C(=O)Nc6ncc(C)s6)c(C)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H60N12O5S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-T1M21O	SCHEMBL25143263	4-[[2-[2-[2-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]ethylamino]-2-oxoethyl]amino]-2-methyl-N-(5-methyl-1,3-thiazol-2-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCNC(=O)CNc5ccc(C(=O)Nc6ncc(C)s6)c(C)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C46H58N12O7S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-I1QEJQ	SCHEMBL25142984	4-[[2-[2-[2-[2-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]ethoxy]ethylamino]-2-oxoethyl]amino]-2-methyl-N-(5-methyl-1,3-thiazol-2-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCOCCNC(=O)CNc5ccc(C(=O)Nc6ncc(C)s6)c(C)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C48H62N12O8S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-JO2TG1	SCHEMBL25143033	4-[2-[2-[2-[2-[2-[2-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethylamino]-2-oxoethoxy]-2-methyl-N-(5-methyl-1,3-thiazol-2-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCOCCOCCOCCNC(=O)COc5ccc(C(=O)Nc6ncc(C)s6)c(C)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C52H69N11O11S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-K7C6G5	SCHEMBL25143283	4-[2-[2-[2-[2-[2-[2-[[2-[4-[[6-[[5-fluoro-4-(7-fluoro-2-methyl-3-propan-2-ylbenzimidazol-5-yl)pyrimidin-2-yl]amino]pyridin-3-yl]methyl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethylamino]-2-methyl-N-(5-methyl-1,3-thiazol-2-yl)benzamide	Cc1cnc(NC(=O)c2ccc(NCCOCCOCCOCCOCCOCCNC(=O)CN3CCN(Cc4ccc(Nc5ncc(F)c(-c6cc(F)c7nc(C)n(C(C)C)c7c6)n5)nc4)CC3)cc2C)s1	C51H66F2N12O7S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-A3RU10	SCHEMBL25142922	4-[2-[2-[2-[2-[2-[2-[[2-[4-[6-[[5-fluoro-4-(7-fluoro-2-methyl-3-propan-2-ylbenzimidazol-5-yl)pyrimidin-2-yl]amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethylamino]-2-methyl-N-(5-methyl-1,3-thiazol-2-yl)benzamide	Cc1cnc(NC(=O)c2ccc(NCCOCCOCCOCCOCCOCCNC(=O)CN3CCN(c4ccc(Nc5ncc(F)c(-c6cc(F)c7nc(C)n(C(C)C)c7c6)n5)nc4)CC3)cc2C)s1	C50H64F2N12O7S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-0VAL13	SCHEMBL25143131	2-methyl-N-(5-methyl-1,3-thiazol-2-yl)-4-[2-[2-[2-[2-[2-[2-[[2-[4-[6-[(10-oxospiro[1,3,5,11-tetrazatricyclo[7.4.0.02,7]trideca-2,4,6,8-tetraene-13,1'-cyclohexane]-4-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethylamino]benzamide	Cc1cnc(NC(=O)c2ccc(NCCOCCOCCOCCOCCOCCNC(=O)CN3CCN(c4ccc(Nc5ncc6cc7n(c6n5)C5(CCCCC5)CNC7=O)nc4)CC3)cc2C)s1	C49H66N12O8S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-7SZJ5V	SCHEMBL25143028	7-cyclopentyl-N,N-dimethyl-2-[[5-[4-[2-[2-[2-[2-[2-[2-[2-[3-methyl-4-[(5-methyl-1,3-thiazol-2-yl)carbamoyl]anilino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethylamino]-2-oxoethyl]piperazin-1-yl]pyridin-2-yl]amino]pyrrolo[2,3-d]pyrimidine-6-carboxamide	Cc1cnc(NC(=O)c2ccc(NCCOCCOCCOCCOCCOCCNC(=O)CN3CCN(c4ccc(Nc5ncc6cc(C(=O)N(C)C)n(C7CCCC7)c6n5)nc4)CC3)cc2C)s1	C49H68N12O8S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-C3Y1OS	SCHEMBL25143287	4-N-[9-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]nonyl]-2-methyl-1-N-(5-methyl-1,3-thiazol-2-yl)benzene-1,4-dicarboxamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCCCCCCCCNC(=O)c5ccc(C(=O)Nc6ncc(C)s6)c(C)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C48H61N11O5S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-IP4FXO	SCHEMBL25143027	4-[2-[2-[2-[2-[2-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethylamino]-2-methyl-N-(4-methylphenyl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCOCCOCCOCCNc5ccc(C(=O)Nc6ccc(C)cc6)c(C)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C53H70N10O9	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-582K3H	SCHEMBL25143289	4-[2-[2-[2-[2-[2-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethylamino]-2-methyl-N-(5-methylpyridin-2-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCOCCOCCOCCNc5ccc(C(=O)Nc6ccc(C)cn6)c(C)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C52H69N11O9	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-EGMKSP	WO-2023061440-A1_CPD-027	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCOCCOCCOCCNc5ccc(C(=O)Nc6ccccn6)c(C)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C51H67N11O9	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-GB9Q69	WO-2023061440-A1_CPD-028	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCOCCOCCOCCNc5ccc(C(=O)Nc6ncc(F)s6)c(C)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C49H64FN11O9S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-GB7ZZC	SCHEMBL25142970	4-[2-[2-[2-[2-[2-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethylamino]-N-(5-cyclopropyl-1,3-thiazol-2-yl)-2-methylbenzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCOCCOCCOCCNc5ccc(C(=O)Nc6ncc(C7CC7)s6)c(C)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C52H69N11O9S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-5DZ6ND	SCHEMBL25142654	4-[2-[2-[2-[2-[2-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethylamino]-N-(5-methoxy-1,3-thiazol-2-yl)-2-methylbenzamide	COc1cnc(NC(=O)c2ccc(NCCOCCOCCOCCOCCOCCNC(=O)CN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)cc2C)s1	C50H67N11O10S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-LG54I9	SCHEMBL25142657	4-[2-[2-[2-[2-[2-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-methylbenzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCOCCOCCOCCNc5ccc(C(=O)Nc6nc(C)c(C)s6)c(C)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C51H69N11O9S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-F7OT09	SCHEMBL25142912	Methyl 2-[[4-[2-[2-[2-[2-[2-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethylamino]-2-methylbenzoyl]amino]-1,3-thiazole-5-carboxylate	COC(=O)c1cnc(NC(=O)c2ccc(NCCOCCOCCOCCOCCOCCNC(=O)CN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)cc2C)s1	C51H67N11O11S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-9A8Y3S	WO-2023061440-A1_CPD-033	.	COC(=O)c1nc(NC(=O)c2ccc(NCCOCCOCCOCCOCCOCCNC(=O)CN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)cc2C)sc1C	C52H69N11O11S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-GXH57U	SCHEMBL25142505	4-[2-[2-[2-[2-[2-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethylamino]-2-methyl-N-(5-methyl-4-phenyl-1,3-thiazol-2-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCOCCOCCOCCNc5ccc(C(=O)Nc6nc(-c7ccccc7)c(C)s6)c(C)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C56H71N11O9S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-UFVUK4	SCHEMBL25143528	4-[[2-[9-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]nonylamino]-2-oxoethyl]amino]-2-methyl-N-(5-methyl-1,3-thiazol-2-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCCCCCCCCNC(=O)CNc5ccc(C(=O)Nc6ncc(C)s6)c(C)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C49H64N12O5S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-MPM04C	WO-2023061440-A1_CPD-036	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCCCCNC(=O)COc5ccc(C(=O)Nc6ncc(C)s6)c(C)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H55N11O6S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-GW0OZS	SCHEMBL25142433	4-[2-[7-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]heptylamino]-2-oxoethoxy]-2-methyl-N-(5-methyl-1,3-thiazol-2-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCCCCCCNC(=O)COc5ccc(C(=O)Nc6ncc(C)s6)c(C)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H59N11O6S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-I4K1HI	SCHEMBL25142938	4-[2-[9-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]nonylamino]-2-oxoethoxy]-2-methyl-N-(5-methyl-1,3-thiazol-2-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCCCCCCCCNC(=O)COc5ccc(C(=O)Nc6ncc(C)s6)c(C)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C49H63N11O6S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-S59M05	WO-2023061440-A1_CPD-039	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCNC(=O)COc5ccc(C(=O)Nc6ncc(C)s6)c(C)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C46H57N11O8S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-RDXBSA	SCHEMBL25142900	4-[2-[2-[2-[2-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]ethoxy]ethylamino]-2-oxoethoxy]-2-methyl-N-(5-methyl-1,3-thiazol-2-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCOCCNC(=O)COc5ccc(C(=O)Nc6ncc(C)s6)c(C)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C48H61N11O9S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-KIXAA0	SCHEMBL25142705	4-[2-[2-[2-[2-[2-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethylamino]-2-oxoethoxy]-2-methyl-N-(5-methyl-1,3-thiazol-2-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCOCCOCCNC(=O)COc5ccc(C(=O)Nc6ncc(C)s6)c(C)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C50H65N11O10S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-NKZZKU	SCHEMBL25142656	4-[2-[2-[2-[2-[2-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethylamino]-2-methyl-N-(5-methyl-4-propan-2-yl-1,3-thiazol-2-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCOCCOCCOCCNc5ccc(C(=O)Nc6nc(C(C)C)c(C)s6)c(C)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C53H73N11O9S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-A2TEI5	SCHEMBL25143295	4-[2-[2-[2-[2-[2-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethylamino]-N-(4-bromo-5-methyl-1,3-thiazol-2-yl)-2-methylbenzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCOCCOCCOCCNc5ccc(C(=O)Nc6nc(Br)c(C)s6)c(C)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C50H66BrN11O9S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-D4UFCL	SCHEMBL25143008	4-[2-[2-[2-[2-[2-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethylamino]-N-(4-acetyl-5-methyl-1,3-thiazol-2-yl)-2-methylbenzamide	CC(=O)c1nc(NC(=O)c2ccc(NCCOCCOCCOCCOCCOCCNC(=O)CN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)cc2C)sc1C	C52H69N11O10S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-AUD0TP	SCHEMBL25142950	4-[2-[2-[2-[2-[2-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethylamino]-N-(4-cyclopropyl-5-methyl-1,3-thiazol-2-yl)-2-methylbenzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCOCCOCCOCCNc5ccc(C(=O)Nc6nc(C7CC7)c(C)s6)c(C)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C53H71N11O9S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-PRI95V	SCHEMBL25143298	4-[2-[2-[2-[2-[2-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethylamino]-N-(4-ethyl-5-methyl-1,3-thiazol-2-yl)-2-methylbenzamide	CCc1nc(NC(=O)c2ccc(NCCOCCOCCOCCOCCOCCNC(=O)CN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)cc2C)sc1C	C52H71N11O9S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-HIDQ5M	SCHEMBL25142916	4-N-[7-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]heptyl]-2-methyl-1-N-(5-methyl-1,3-thiazol-2-yl)benzene-1,4-dicarboxamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCCCCCCNC(=O)c5ccc(C(=O)Nc6ncc(C)s6)c(C)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C46H57N11O5S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-UDMWB9	WO-2023061440-A1_CPD-050	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCOCCOCCOCCNc5ccc(C(=O)Nc6cc(C)n(C)n6)c(C)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C51H70N12O9	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-VCZXZV	SCHEMBL25143034	2-[3-[2-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]propanoylamino]-N-(5-methyl-1,3-thiazol-2-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)Nc5ccccc5C(=O)Nc5ncc(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C44H53N11O7S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-9413RY	WO-2023061440-A1_CPD-052	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)Nc5ccccc5C(=O)Nc5cc(C)n(C)n5)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H56N12O7	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-1167BF	WO-2023061440-A1_CPD-053	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)Nc5ccccc5C(=O)Nc5ccccn5)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H53N11O7	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-PYD7IF	SCHEMBL25142658	2-[3-[2-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]propanoylamino]-N-(5-methylpyrazin-2-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)Nc5ccccc5C(=O)Nc5cnc(C)cn5)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H54N12O7	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-BMEDK1	WO-2023061440-A1_CPD-055	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)Nc5ccccc5C(=O)Nc5ncc(C)cn5)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H54N12O7	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-01URO9	WO-2023061440-A1_CPD-056	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)Nc5ccccc5C(=O)Nc5ccc(C)nn5)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H54N12O7	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-FPRGQM	SCHEMBL25142903	2-[3-[2-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]propanoylamino]-N-(4-cyclopropyl-5-methyl-1,3-thiazol-2-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)Nc5ccccc5C(=O)Nc5nc(C6CC6)c(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H57N11O7S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-APZBRP	WO-2023061440-A1_CPD-058	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)Nc5ccccc5C(=O)Nc5nc(C)ns5)CC4)cn3)nc2n(C2CCCC2)c1=O	C43H52N12O7S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-VOXOM6	WO-2023061440-A1_CPD-059	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)Nc5ccccc5C(=O)Nc5nc(C6CC6)ns5)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H54N12O7S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-U6SRU2	SCHEMBL25142554	2-[3-[2-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]propanoylamino]-N-(6-methylpyridin-3-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)Nc5ccccc5C(=O)Nc5ccc(C)nc5)CC4)cn3)nc2n(C2CCCC2)c1=O	C46H55N11O7	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-SR3TN5	WO-2023061440-A1_CPD-061	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)Nc5ccccc5C(=O)Nc5ccc(C)cn5)CC4)cn3)nc2n(C2CCCC2)c1=O	C46H55N11O7	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-2H6E17	SCHEMBL25142826	2-[3-[2-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]propanoylamino]-N-[5-methyl-4-(oxan-4-yl)-1,3-thiazol-2-yl]benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)Nc5ccccc5C(=O)Nc5nc(C6CCOCC6)c(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C49H61N11O8S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-MTASRZ	SCHEMBL25142944	2-[3-[2-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]propanoylamino]-N-(1-methylimidazol-4-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)Nc5ccccc5C(=O)Nc5cn(C)cn5)CC4)cn3)nc2n(C2CCCC2)c1=O	C44H54N12O7	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-3NH04T	SCHEMBL25143258	2-[3-[2-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]propanoylamino]-N-(5-methyl-1H-imidazol-2-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)Nc5ccccc5C(=O)Nc5ncc(C)[nH]5)CC4)cn3)nc2n(C2CCCC2)c1=O	C44H54N12O7	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-OAB0Q3	SCHEMBL25142798	2-[3-[2-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]propanoylamino]-N-(5-methylthiophen-2-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)Nc5ccccc5C(=O)Nc5ccc(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H54N10O7S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-3JE28P	WO-2023061440-A1_CPD-066	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)Nc5ccccc5C(=O)Nc5ncc(C)o5)CC4)cn3)nc2n(C2CCCC2)c1=O	C44H53N11O8	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-3PIETS	SCHEMBL25143307	2-[3-[2-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]propanoylamino]-N-(1-methylpyrazol-3-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)Nc5ccccc5C(=O)Nc5ccn(C)n5)CC4)cn3)nc2n(C2CCCC2)c1=O	C44H54N12O7	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-DWQEWC	SCHEMBL25142870	2-[3-[2-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]propanoylamino]-N-[1-methyl-5-(trifluoromethyl)pyrazol-3-yl]benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)Nc5ccccc5C(=O)Nc5cc(C(F)(F)F)n(C)n5)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H53F3N12O7	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-BXR354	SCHEMBL25143262	2-[3-[2-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]propanoylamino]-N-(5-methyl-4-propan-2-yl-1,3-thiazol-2-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)Nc5ccccc5C(=O)Nc5nc(C(C)C)c(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H59N11O7S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-MKMLWZ	WO-2023061440-A1_CPD-071	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)Nc5ccccc5C(=O)Nc5nc(Br)c(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C44H52BrN11O7S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-46W2QX	WO-2023061440-A1_CPD-072	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)Nc5ccccc5C(=O)Nc5nc(C6CCNCC6)c(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C49H62N12O7S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-DVBLJ4	WO-2023061440-A1_CPD-073	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)Nc5ccccc5C(=O)Nc5cc[nH]n5)CC4)cn3)nc2n(C2CCCC2)c1=O	C43H52N12O7	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-IOKJ61	WO-2023061440-A1_CPD-074	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)Nc5ccccc5C(=O)Nc5cc(C)[nH]n5)CC4)cn3)nc2n(C2CCCC2)c1=O	C44H54N12O7	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-RXK4C4	WO-2023061440-A1_CPD-075	.	CCc1nc(NC(=O)c2ccccc2NC(=O)CCOCCOCCNC(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)sc1C	C46H57N11O7S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-J2LK9B	WO-2023061440-A1_CPD-076	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)Nc5ccccc5C(=O)Nc5cc(C)n(C(C)C)n5)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H60N12O7	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-WB0K8B	SCHEMBL25143082	2-[3-[2-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]propanoylamino]-N-[5-methyl-4-(trifluoromethyl)-1,3-thiazol-2-yl]benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)Nc5ccccc5C(=O)Nc5nc(C(F)(F)F)c(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H52F3N11O7S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-BYWWH7	WO-2023061440-A1_CPD-078	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCCCCCCCCNc5cccc(C(=O)Nc6nc(C)c(C)s6)c5C)CC4)cn3)nc2n(C2CCCC2)c1=O	C48H63N11O4S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-CDKD64	WO-2023061440-A1_CPD-079	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)Nc5ccccc5C(=O)Nc5cc(C6CC6)n(C)n5)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H58N12O7	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-829TAE	SCHEMBL25142419	2-[3-[2-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]propanoylamino]-N-[5-methyl-4-(1-methylpiperidin-4-yl)-1,3-thiazol-2-yl]benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)Nc5ccccc5C(=O)Nc5nc(C6CCN(C)CC6)c(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C50H64N12O7S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-GROTPE	SCHEMBL25142426	2-[3-[2-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]propanoylamino]-N-(5-fluoropyridin-2-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)Nc5ccccc5C(=O)Nc5ccc(F)cn5)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H52FN11O7	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-9ECK11	SCHEMBL25142509	2-[3-[2-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]propanoylamino]-N-(5-chloropyridin-2-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)Nc5ccccc5C(=O)Nc5ccc(Cl)cn5)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H52ClN11O7	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-Y9VA36	SCHEMBL25142893	2-[3-[2-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]propanoylamino]-N-(5-cyanopyridin-2-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)Nc5ccccc5C(=O)Nc5ccc(C#N)cn5)CC4)cn3)nc2n(C2CCCC2)c1=O	C46H52N12O7	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-QA8J59	SCHEMBL25142762	2-[3-[2-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]propanoylamino]-N-[5-(trifluoromethyl)pyridin-2-yl]benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)Nc5ccccc5C(=O)Nc5ccc(C(F)(F)F)cn5)CC4)cn3)nc2n(C2CCCC2)c1=O	C46H52F3N11O7	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-IWD4A1	WO-2023061440-A1_CPD-085	.	COc1ccc(NC(=O)c2ccccc2NC(=O)CCOCCOCCNC(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)nn1	C45H54N12O8	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-DWG7OX	SCHEMBL25142790	3-[2-[2-[2-[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]ethylamino]ethoxy]ethoxy]ethylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-methylbenzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CCNCCOCCOCCNc5cccc(C(=O)Nc6nc(C)c(C)s6)c5C)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H59N11O5S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-B97VZF	SCHEMBL25142813	5-[3-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]propylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-methylbenzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCCNc5ccc(C)c(C(=O)Nc6nc(C)c(C)s6)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C42H51N11O4S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-NQOMEG	WO-2023061440-A1_CPD-088	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCCCNc5ccc(C)c(C(=O)Nc6nc(C)c(C)s6)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C43H53N11O4S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-6Z1NPR	WO-2023061440-A1_CPD-089	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCNc5ccc(C)c(C(=O)Nc6nc(C)c(C)s6)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H57N11O6S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-CVCDO5	WO-2023061440-A1_CPD-090	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCCCCCCCNc5cccc(C(=O)Nc6nc(C)c(C)s6)c5C)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H61N11O4S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-0C7IP3	WO-2023061440-A1_CPD-091	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(=O)CCNc5ccc(C)c(C(=O)Nc6nc(C)c(C)s6)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C40H46N10O4S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-CAKRFO	WO-2023061440-A1_CPD-092	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCNc5cccc(C(=O)Nc6nc(C)c(C)s6)c5C)CC4)cn3)nc2n(C2CCCC2)c1=O	C41H49N11O4S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-2Q0SA8	SCHEMBL25143501	5-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-methylbenzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCNc5ccc(C)c(C(=O)Nc6nc(C)c(C)s6)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C41H49N11O4S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-KY09CO	SCHEMBL25143539	5-[6-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]hexylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-methylbenzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCCCCCNc5ccc(C)c(C(=O)Nc6nc(C)c(C)s6)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H57N11O4S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-1CESCZ	SCHEMBL25143503	5-[8-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]octylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-methylbenzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCCCCCCCNc5ccc(C)c(C(=O)Nc6nc(C)c(C)s6)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H61N11O4S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-4FI4FX	SCHEMBL25143541	5-[2-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-methylbenzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCNc5ccc(C)c(C(=O)Nc6nc(C)c(C)s6)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C43H53N11O5S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-T1KH5J	SCHEMBL25143526	5-[2-[2-[2-[2-[2-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-methylbenzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCOCCOCCOCCNc5ccc(C)c(C(=O)Nc6nc(C)c(C)s6)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C51H69N11O9S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-Y0JPB3	WO-2023061440-A1_CPD-098	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCCNc5cccc(C(=O)Nc6nc(C)c(C)s6)c5C)CC4)cn3)nc2n(C2CCCC2)c1=O	C42H51N11O4S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-28H9K0	WO-2023061440-A1_CPD-099	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCCCNc5cccc(C(=O)Nc6nc(C)c(C)s6)c5C)CC4)cn3)nc2n(C2CCCC2)c1=O	C43H53N11O4S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-O8Y9N7	SCHEMBL25142493	3-[5-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]pentylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-methylbenzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCCCCNc5cccc(C(=O)Nc6nc(C)c(C)s6)c5C)CC4)cn3)nc2n(C2CCCC2)c1=O	C44H55N11O4S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-T9VO2G	SCHEMBL25142495	3-[6-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]hexylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-methylbenzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCCCCCNc5cccc(C(=O)Nc6nc(C)c(C)s6)c5C)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H57N11O4S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-5Q5PX7	WO-2023061440-A1_CPD-102	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCCCCCCNc5cccc(C(=O)Nc6nc(C)c(C)s6)c5C)CC4)cn3)nc2n(C2CCCC2)c1=O	C46H59N11O4S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-1IEJW6	WO-2023061440-A1_CPD-103	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCNc5cccc(C(=O)Nc6nc(C)c(C)s6)c5C)CC4)cn3)nc2n(C2CCCC2)c1=O	C43H53N11O5S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-Y7A96N	WO-2023061440-A1_CPD-104	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCNc5cccc(C(=O)Nc6nc(C)c(C)s6)c5C)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H57N11O6S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-M6IC9R	WO-2023061440-A1_CPD-105	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCOCCNc5cccc(C(=O)Nc6nc(C)c(C)s6)c5C)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H61N11O7S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-6ZUFB4	WO-2023061440-A1_CPD-106	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCOCCOCCNc5cccc(C(=O)Nc6nc(C)c(C)s6)c5C)CC4)cn3)nc2n(C2CCCC2)c1=O	C49H65N11O8S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-4QNFLM	SCHEMBL25142780	3-[2-[2-[2-[2-[2-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-methylbenzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCOCCOCCOCCNc5cccc(C(=O)Nc6nc(C)c(C)s6)c5C)CC4)cn3)nc2n(C2CCCC2)c1=O	C51H69N11O9S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-FADAWK	SCHEMBL25142797	5-[[5-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]-5-oxopentyl]amino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-methylbenzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(=O)CCCCNc5ccc(C)c(C(=O)Nc6nc(C)c(C)s6)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C42H50N10O4S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-2O5541	WO-2023061440-A1_CPD-109	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(=O)CCCCCCNc5ccc(C)c(C(=O)Nc6nc(C)c(C)s6)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C44H54N10O4S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-OB2S7Q	WO-2023061440-A1_CPD-110	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(=O)CCOCCNc5ccc(C)c(C(=O)Nc6nc(C)c(C)s6)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C42H50N10O5S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-QPXQQQ	SCHEMBL25143248	5-[2-[2-[2-[3-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]-3-oxopropoxy]ethoxy]ethoxy]ethylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-methylbenzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(=O)CCOCCOCCOCCNc5ccc(C)c(C(=O)Nc6nc(C)c(C)s6)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C46H58N10O7S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-70JYK0	WO-2023061440-A1_CPD-112	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(=O)CCNc5cccc(C(=O)Nc6nc(C)c(C)s6)c5C)CC4)cn3)nc2n(C2CCCC2)c1=O	C40H46N10O4S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-RL162Y	WO-2023061440-A1_CPD-113	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCCCCCCCC(=O)Nc5ccccc5C(=O)Nc5nc(C)c(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H59N11O5S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-PDSR35	SCHEMBL25142886	2-[3-[2-[2-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]ethoxy]propanoylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)benzamide; SCHEMBL31110157	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCOCCC(=O)Nc5ccccc5C(=O)Nc5nc(C)c(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H59N11O8S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-TUMUK0	WO-2023061440-A1_CPD-115	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)Nc5ccccc5C(=O)Nc5nc(C)c(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H55N11O7S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-3XSO2Z	SCHEMBL25142772	5-[5-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]pentylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-methylbenzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCCCCNc5ccc(C)c(C(=O)Nc6nc(C)c(C)s6)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C44H55N11O4S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-P113JA	SCHEMBL25142888	5-[7-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]heptylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-methylbenzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCCCCCCNc5ccc(C)c(C(=O)Nc6nc(C)c(C)s6)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C46H59N11O4S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-CH9Z4G	WO-2023061440-A1_CPD-118	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCOCCOCCNc5ccc(C)c(C(=O)Nc6nc(C)c(C)s6)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C49H65N11O8S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-XLQ6WS	SCHEMBL25142892	5-[2-[2-[2-[2-[3-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]-3-oxopropoxy]ethoxy]ethoxy]ethoxy]ethylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-methylbenzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(=O)CCOCCOCCOCCOCCNc5ccc(C)c(C(=O)Nc6nc(C)c(C)s6)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C48H62N10O8S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-VXC5MO	SCHEMBL25142714	3-[2-[3-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]-3-oxopropoxy]ethylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-methylbenzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(=O)CCOCCNc5cccc(C(=O)Nc6nc(C)c(C)s6)c5C)CC4)cn3)nc2n(C2CCCC2)c1=O	C42H50N10O5S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-FZEHR4	WO-2023061440-A1_CPD-121	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(=O)CCOCCOCCNc5cccc(C(=O)Nc6nc(C)c(C)s6)c5C)CC4)cn3)nc2n(C2CCCC2)c1=O	C44H54N10O6S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-13K5XL	SCHEMBL25142883	3-[2-[2-[2-[3-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]-3-oxopropoxy]ethoxy]ethoxy]ethylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-methylbenzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(=O)CCOCCOCCOCCNc5cccc(C(=O)Nc6nc(C)c(C)s6)c5C)CC4)cn3)nc2n(C2CCCC2)c1=O	C46H58N10O7S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-10OCUO	WO-2023061440-A1_CPD-123	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(=O)CCOCCOCCOCCOCCNc5cccc(C(=O)Nc6nc(C)c(C)s6)c5C)CC4)cn3)nc2n(C2CCCC2)c1=O	C48H62N10O8S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-HGTS63	SCHEMBL25142532	3-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]-2-oxoethyl]amino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-methylbenzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(=O)CNc5cccc(C(=O)Nc6nc(C)c(C)s6)c5C)CC4)cn3)nc2n(C2CCCC2)c1=O	C39H44N10O4S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-6DWAPR	SCHEMBL25143007	3-[[8-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]-8-oxooctyl]amino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-methylbenzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(=O)CCCCCCCNc5cccc(C(=O)Nc6nc(C)c(C)s6)c5C)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H56N10O4S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-A7F3S7	SCHEMBL25143584	3-[2-[2-[2-[2-[2-[3-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]-3-oxopropoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-methylbenzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(=O)CCOCCOCCOCCOCCOCCNc5cccc(C(=O)Nc6nc(C)c(C)s6)c5C)CC4)cn3)nc2n(C2CCCC2)c1=O	C50H66N10O9S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-OBQ6LI	SCHEMBL25142462	2-[3-[2-[3-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]-3-oxopropoxy]ethoxy]propanoylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(=O)CCOCCOCCC(=O)Nc5ccccc5C(=O)Nc5nc(C)c(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C44H52N10O7S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-LJLH0A	WO-2023061440-A1_CPD-129	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(=O)CCCCCNc5ccc(C)c(C(=O)Nc6nc(C)c(C)s6)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C43H52N10O4S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-DLQ2UU	WO-2023061440-A1_CPD-130	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(=O)CCOCCOCCNc5ccc(C)c(C(=O)Nc6nc(C)c(C)s6)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C44H54N10O6S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-5KANL9	WO-2023061440-A1_CPD-131	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(=O)CCOCCOCCOCCOCCOCCOCCNc5ccc(C)c(C(=O)Nc6nc(C)c(C)s6)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C52H70N10O10S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-JX6O74	WO-2023061440-A1_CPD-133	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(=O)CCOCCOCCOCCOCCOCCOCCNc5cccc(C(=O)Nc6nc(C)c(C)s6)c5C)CC4)cn3)nc2n(C2CCCC2)c1=O	C52H70N10O10S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-WMIOYX	SCHEMBL25143157	5-[2-[2-[2-[2-[2-[3-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]-3-oxopropoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-methylbenzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(=O)CCOCCOCCOCCOCCOCCNc5ccc(C)c(C(=O)Nc6nc(C)c(C)s6)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C50H66N10O9S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-V2K8T1	WO-2023061440-A1_CPD-135	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(=O)CNc5ccc(C)c(C(=O)Nc6nc(C)c(C)s6)c5)CC4)cn3)nc2n(C2CC=CC2)c1=O	C39H42N10O4S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-GHFR8W	SCHEMBL25142748	2-[8-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]octanoylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCCCCCCC(=O)Nc5ccccc5C(=O)Nc5nc(C)c(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C46H57N11O5S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-K7QK5O	SCHEMBL25143344	3-[[6-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]-6-oxohexyl]amino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-methylbenzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(=O)CCCCCNc5cccc(C(=O)Nc6nc(C)c(C)s6)c5C)CC4)cn3)nc2n(C2CCCC2)c1=O	C43H52N10O4S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-VXS35S	WO-2023061440-A1_CPD-138	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(=O)CCCCCCNc5cccc(C(=O)Nc6nc(C)c(C)s6)c5C)CC4)cn3)nc2n(C2CCCC2)c1=O	C44H54N10O4S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-CHXGT7	SCHEMBL25142649	2-[3-[2-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]propanoylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)-6-methylbenzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)Nc5cccc(C)c5C(=O)Nc5nc(C)c(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C46H57N11O7S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-JCVZV2	WO-2023061440-A1_CPD-140	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)Nc5cc(Cl)ccc5C(=O)Nc5nc(C)c(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H54ClN11O7S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-JAZCLU	WO-2023061440-A1_CPD-141	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)Nc5ccc(C)cc5C(=O)Nc5nc(C)c(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C46H57N11O7S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-9Q8XWN	WO-2023061440-A1_CPD-142	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)Nc5ccc(Cl)cc5C(=O)Nc5nc(C)c(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H54ClN11O7S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-3ZS2BD	WO-2023061440-A1_CPD-143	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)Nc5cc(F)ccc5C(=O)Nc5nc(C)c(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H54FN11O7S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-6GBXPI	WO-2023061440-A1_CPD-144	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)Nc5cc(Br)ccc5C(=O)Nc5nc(C)c(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H54BrN11O7S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-74PTQG	SCHEMBL25143445	2-[3-[2-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]propanoylamino]-5-bromo-N-(4,5-dimethyl-1,3-thiazol-2-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)Nc5ccc(Br)cc5C(=O)Nc5nc(C)c(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H54BrN11O7S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-H3BI3V	SCHEMBL25143448	2-[3-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]propanoylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCC(=O)Nc5ccccc5C(=O)Nc5nc(C)c(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C41H47N11O5S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-I5YWEX	SCHEMBL25143439	2-[3-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]propanoylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCC(=O)Nc5ccccc5C(=O)Nc5nc(C)c(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C43H51N11O6S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-4IEEK9	WO-2023061440-A1_CPD-148	.	CCCCNc1ccc(NC(=O)CCOCCOCCNC(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)c(C(=O)Nc2nc(C)c(C)s2)c1	C49H64N12O7S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-AQV74A	WO-2023061440-A1_CPD-149	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)Nc5cc(C)ccc5C(=O)Nc5nc(C)c(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C46H57N11O7S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-O5WAUQ	WO-2023061440-A1_CPD-150	.	CNc1ccc(NC(=O)CCOCCOCCNC(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)c(C(=O)Nc2nc(C)c(C)s2)c1	C46H58N12O7S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-O90SK2	WO-2023061440-A1_CPD-151	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)Nc5ccc(N(C)C)cc5C(=O)Nc5nc(C)c(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H60N12O7S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-T5TFS2	WO-2023061440-A1_CPD-152	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)Nc5ccc(F)cc5C(=O)Nc5nc(C)c(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H54FN11O7S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-4FEEDV	SCHEMBL31110118	2-[[4-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]-4-oxobutanoyl]amino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(=O)CCC(=O)Nc5ccccc5C(=O)Nc5nc(C)c(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C40H44N10O5S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-U85IZA	WO-2023061440-A1_CPD-154	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)Nc5ccccc5CNc5nc(C)c(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H57N11O6S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-4VGV5R	WO-2023061440-A1_CPD-155	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)Nc5cc(N(C)C)ccc5C(=O)Nc5nc(C)c(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H60N12O7S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-BG9BK0	SCHEMBL31110007	2-[[6-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]-6-oxohexanoyl]amino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(=O)CCCCC(=O)Nc5ccccc5C(=O)Nc5nc(C)c(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C42H48N10O5S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-FL0OH8	SCHEMBL31110009	2-[[7-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]-7-oxoheptanoyl]amino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(=O)CCCCCC(=O)Nc5ccccc5C(=O)Nc5nc(C)c(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C43H50N10O5S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-I9FN04	SCHEMBL25142588	2-[[3-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]-3-oxopropanoyl]amino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)benzamide; SCHEMBL31110174	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(=O)CC(=O)Nc5ccccc5C(=O)Nc5nc(C)c(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C39H42N10O5S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-N8JXUI	SCHEMBL25143626	2-[[5-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]-5-oxopentanoyl]amino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)benzamide; SCHEMBL31110289	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(=O)CCCC(=O)Nc5ccccc5C(=O)Nc5nc(C)c(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C41H46N10O5S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-69SDVG	SCHEMBL31110246	2-[[9-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]-9-oxononanoyl]amino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(=O)CCCCCCCC(=O)Nc5ccccc5C(=O)Nc5nc(C)c(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H54N10O5S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-FH6I5G	SCHEMBL25142985	2-[[8-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]-8-oxooctanoyl]amino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)benzamide; SCHEMBL31110266	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(=O)CCCCCCC(=O)Nc5ccccc5C(=O)Nc5nc(C)c(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C44H52N10O5S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-QKRD6G	SCHEMBL31110090	2-[[10-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]-10-oxodecanoyl]amino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(=O)CCCCCCCCC(=O)Nc5ccccc5C(=O)Nc5nc(C)c(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C46H56N10O5S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-XFG7MK	SCHEMBL25142988	2-[3-[2-[2-[2-[2-[3-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]-3-oxopropoxy]ethoxy]ethoxy]ethoxy]ethoxy]propanoylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(=O)CCOCCOCCOCCOCCOCCC(=O)Nc5ccccc5C(=O)Nc5nc(C)c(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C50H64N10O10S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-X7LE87	WO-2023061440-A1_CPD-164	.	CNc1ccc(C(=O)Nc2nc(C)c(C)s2)c(NC(=O)CCOCCOCCNC(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)c1	C46H58N12O7S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-X5AEF2	SCHEMBL25142917	5-[[4-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]-4-oxobutyl]amino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-methylbenzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(=O)CCCNc5ccc(C)c(C(=O)Nc6nc(C)c(C)s6)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C41H48N10O4S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-8MQ45S	WO-2023061440-A1_CPD-166	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCOCCOCCOCCNc5ccc(CNc6nc(C)c(C)s6)c(C)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C51H71N11O8S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-PDQB41	SCHEMBL25142684	2-[3-[2-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]propanoylamino]-4-(butylamino)-N-(4,5-dimethyl-1,3-thiazol-2-yl)benzamide	CCCCNc1ccc(C(=O)Nc2nc(C)c(C)s2)c(NC(=O)CCOCCOCCNC(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)c1	C49H64N12O7S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-MNGTLE	SCHEMBL25142761	2-[7-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]heptanoylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCCCCCC(=O)Nc5ccccc5C(=O)Nc5nc(C)c(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H55N11O5S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-6PU66F	SCHEMBL31110252	2-[3-[2-[2-[2-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]propanoylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCOCCOCCC(=O)Nc5ccccc5C(=O)Nc5nc(C)c(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C49H63N11O9S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-95M21L	SCHEMBL25142612	2-[4-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]butanoylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCCC(=O)Nc5ccccc5C(=O)Nc5nc(C)c(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C42H49N11O5S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-IW4Q3F	WO-2023061440-A1_CPD-172	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCCCCC(=O)Nc5ccccc5C(=O)Nc5nc(C)c(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C44H53N11O5S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-E4LIZ8	WO-2023061440-A1_CPD-173	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCOCCOCCOCCOCCC(=O)Nc5ccccc5C(=O)Nc5nc(C)c(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C53H71N11O11S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-8CWMFY	SCHEMBL25142615	2-[5-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]pentanoylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCCCC(=O)Nc5ccccc5C(=O)Nc5nc(C)c(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C43H51N11O5S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-9PT7YC	SCHEMBL25142814	2-[3-[2-[2-[2-[2-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]propanoylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCOCCOCCOCCC(=O)Nc5ccccc5C(=O)Nc5nc(C)c(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C51H67N11O10S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-HP0UPO	WO-2023061440-A1_CPD-176	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(=O)CCOCCOCCOCCOCCC(=O)Nc5ccccc5C(=O)Nc5nc(C)c(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C48H60N10O9S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-ZXD69V	SCHEMBL25142659	2-[12-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]dodecanoylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CCCCCCCCCCCC(=O)Nc5ccccc5C(=O)Nc5nc(C)c(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C48H62N10O4S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-0XP8LY	SCHEMBL25143052	2-[3-[2-[2-[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]ethoxy]ethoxy]ethoxy]propanoylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CCOCCOCCOCCC(=O)Nc5ccccc5C(=O)Nc5nc(C)c(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H56N10O7S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-GDZTHW	WO-2023061440-A1_CPD-179	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)NC5CCCCC5C(=O)Nc5nc(C)c(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H61N11O7S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-029L19	WO-2023061440-A1_CPD-180	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCC(=O)Nc5ccccc5C(=O)Nc5nc(C)c(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C40H45N11O5S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-K0S7QV	SCHEMBL25142990	2-[3-[3-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]-3-oxopropoxy]propanoylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(=O)CCOCCC(=O)Nc5ccccc5C(=O)Nc5nc(C)c(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C42H48N10O6S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-F4BVIY	SCHEMBL25143017	2-[3-[2-[2-[2-[2-[2-[3-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]-3-oxopropoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]propanoylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(=O)CCOCCOCCOCCOCCOCCOCCC(=O)Nc5ccccc5C(=O)Nc5nc(C)c(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C52H68N10O11S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-6LPGBO	SCHEMBL25142804	2-[8-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]octanoylamino]-N-(5-methylpyridin-2-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CCCCCCCC(=O)Nc5ccccc5C(=O)Nc5ccc(C)cn5)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H54N10O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-E7ZN30	WO-2023061440-A1_CPD-184	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)Nc5ccccc5C(=O)Nc5ccc(C6CC6)cn5)CC4)cn3)nc2n(C2CCCC2)c1=O	C48H57N11O7	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-K9EZC5	WO-2023061440-A1_CPD-185	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)Nc5ccccc5C(=O)Nc5ccc(N(C)C)nn5)CC4)cn3)nc2n(C2CCCC2)c1=O	C46H57N13O7	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-USFYU3	WO-2023061440-A1_CPD-186	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)Nc5ccccc5C(=O)Nc5cnc(C)nc5)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H54N12O7	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-6YAEZC	WO-2023061440-A1_CPD-187	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CCNCCOCCOCCC(=O)Nc5ccccc5C(=O)Nc5nc(C)c(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H57N11O6S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-W6JWXJ	SCHEMBL25142875	3-[7-[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]ethylamino]heptylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-methylbenzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CCNCCCCCCCNc5cccc(C(=O)Nc6nc(C)c(C)s6)c5C)CC4)cn3)nc2n(C2CCCC2)c1=O	C46H61N11O3S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-WLLJ02	WO-2023061440-A1_CPD-189	.	CC(=O)N1CCc2c(c(N3CCCc4cc(-c5cnn(C)c5)c(C(F)F)cc43)nn2C2CCN(CC(=O)NCCNc3ccc(C(=O)Nc4ncc(C)s4)c(C)c3)CC2)C1	C43H51F2N11O3S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-RQXBKS	WO-2023061440-A1_CPD-190	.	CC(=O)N1CCc2c(c(N3CCCc4cc(-c5cnn(C)c5)c(C(F)F)cc43)nn2C2CCN(CC(=O)NCCCNc3ccc(C(=O)Nc4ncc(C)s4)c(C)c3)CC2)C1	C44H53F2N11O3S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-862BDH	WO-2023061440-A1_CPD-191	.	CC(=O)N1CCc2c(c(N3CCCc4cc(-c5cnn(C)c5)c(C(F)F)cc43)nn2C2CCN(CC(=O)NCCCCNc3ccc(C(=O)Nc4ncc(C)s4)c(C)c3)CC2)C1	C45H55F2N11O3S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-U4UFRT	WO-2023061440-A1_CPD-192	.	CC(=O)N1CCc2c(c(N3CCCc4cc(-c5cnn(C)c5)c(C(F)F)cc43)nn2C2CCN(CC(=O)NCCCCCNc3ccc(C(=O)Nc4ncc(C)s4)c(C)c3)CC2)C1	C46H57F2N11O3S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-N4FMNR	WO-2023061440-A1_CPD-193	.	CC(=O)N1CCc2c(c(N3CCCc4cc(-c5cnn(C)c5)c(C(F)F)cc43)nn2C2CCN(CC(=O)NCCCCCCNc3ccc(C(=O)Nc4ncc(C)s4)c(C)c3)CC2)C1	C47H59F2N11O3S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-CLCTC6	WO-2023061440-A1_CPD-194	.	CC(=O)N1CCc2c(c(N3CCCc4cc(-c5cnn(C)c5)c(C(F)F)cc43)nn2C2CCN(CC(=O)NCCCCCCCNc3ccc(C(=O)Nc4ncc(C)s4)c(C)c3)CC2)C1	C48H61F2N11O3S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-K0W2V7	WO-2023061440-A1_CPD-195	.	CC(=O)N1CCc2c(c(N3CCCc4cc(-c5cnn(C)c5)c(C(F)F)cc43)nn2C2CCN(CC(=O)NCCCCCCCCNc3ccc(C(=O)Nc4ncc(C)s4)c(C)c3)CC2)C1	C49H63F2N11O3S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-8J6TIG	WO-2023061440-A1_CPD-196	.	CC(=O)N1CCc2c(c(N3CCCc4cc(-c5cnn(C)c5)c(C(F)F)cc43)nn2C2CCN(CC(=O)NCCCCCCCCCNc3ccc(C(=O)Nc4ncc(C)s4)c(C)c3)CC2)C1	C50H65F2N11O3S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-V6HU1M	WO-2023061440-A1_CPD-197	.	CC(=O)N1CCc2c(c(N3CCCc4cc(-c5cnn(C)c5)c(C(F)F)cc43)nn2C2CCN(CC(=O)NCCOCCNc3ccc(C(=O)Nc4ncc(C)s4)c(C)c3)CC2)C1	C45H55F2N11O4S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-3SI4NU	WO-2023061440-A1_CPD-198	.	CC(=O)N1CCc2c(c(N3CCCc4cc(-c5cnn(C)c5)c(C(F)F)cc43)nn2C2CCN(CC(=O)NCCOCCOCCNc3ccc(C(=O)Nc4ncc(C)s4)c(C)c3)CC2)C1	C47H59F2N11O5S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-3HLBZ3	SCHEMBL31110217	2-[[4-[4-[5-acetyl-3-[7-(difluoromethyl)-6-(1-methylpyrazol-4-yl)-3,4-dihydro-2H-quinolin-1-yl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]piperidin-1-yl]-4-oxobutanoyl]amino]-N-(4-methyl-5-nitro-1,3-thiazol-2-yl)benzamide	CC(=O)N1CCc2c(c(N3CCCc4cc(-c5cnn(C)c5)c(C(F)F)cc43)nn2C2CCN(C(=O)CCC(=O)Nc3ccccc3C(=O)Nc3nc(C)c([N+](=O)[O-])s3)CC2)C1	C42H45F2N11O6S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-0N9MP4	SCHEMBL31110130	2-[[5-[4-[5-acetyl-3-[7-(difluoromethyl)-6-(1-methylpyrazol-4-yl)-3,4-dihydro-2H-quinolin-1-yl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]piperidin-1-yl]-5-oxopentanoyl]amino]-N-(4-methyl-5-nitro-1,3-thiazol-2-yl)benzamide	CC(=O)N1CCc2c(c(N3CCCc4cc(-c5cnn(C)c5)c(C(F)F)cc43)nn2C2CCN(C(=O)CCCC(=O)Nc3ccccc3C(=O)Nc3nc(C)c([N+](=O)[O-])s3)CC2)C1	C43H47F2N11O6S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-4HJ5BI	SCHEMBL31110085	2-[[6-[4-[5-acetyl-3-[7-(difluoromethyl)-6-(1-methylpyrazol-4-yl)-3,4-dihydro-2H-quinolin-1-yl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]piperidin-1-yl]-6-oxohexanoyl]amino]-N-(4-methyl-5-nitro-1,3-thiazol-2-yl)benzamide	CC(=O)N1CCc2c(c(N3CCCc4cc(-c5cnn(C)c5)c(C(F)F)cc43)nn2C2CCN(C(=O)CCCCC(=O)Nc3ccccc3C(=O)Nc3nc(C)c([N+](=O)[O-])s3)CC2)C1	C44H49F2N11O6S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-7MCX85	SCHEMBL31110164	2-[[7-[4-[5-acetyl-3-[7-(difluoromethyl)-6-(1-methylpyrazol-4-yl)-3,4-dihydro-2H-quinolin-1-yl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]piperidin-1-yl]-7-oxoheptanoyl]amino]-N-(4-methyl-5-nitro-1,3-thiazol-2-yl)benzamide	CC(=O)N1CCc2c(c(N3CCCc4cc(-c5cnn(C)c5)c(C(F)F)cc43)nn2C2CCN(C(=O)CCCCCC(=O)Nc3ccccc3C(=O)Nc3nc(C)c([N+](=O)[O-])s3)CC2)C1	C45H51F2N11O6S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-MHCJI8	SCHEMBL31110193	2-[[8-[4-[5-acetyl-3-[7-(difluoromethyl)-6-(1-methylpyrazol-4-yl)-3,4-dihydro-2H-quinolin-1-yl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]piperidin-1-yl]-8-oxooctanoyl]amino]-N-(4-methyl-5-nitro-1,3-thiazol-2-yl)benzamide	CC(=O)N1CCc2c(c(N3CCCc4cc(-c5cnn(C)c5)c(C(F)F)cc43)nn2C2CCN(C(=O)CCCCCCC(=O)Nc3ccccc3C(=O)Nc3nc(C)c([N+](=O)[O-])s3)CC2)C1	C46H53F2N11O6S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-M0JSG5	SCHEMBL31110257	2-[[9-[4-[5-acetyl-3-[7-(difluoromethyl)-6-(1-methylpyrazol-4-yl)-3,4-dihydro-2H-quinolin-1-yl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]piperidin-1-yl]-9-oxononanoyl]amino]-N-(4-methyl-5-nitro-1,3-thiazol-2-yl)benzamide	CC(=O)N1CCc2c(c(N3CCCc4cc(-c5cnn(C)c5)c(C(F)F)cc43)nn2C2CCN(C(=O)CCCCCCCC(=O)Nc3ccccc3C(=O)Nc3nc(C)c([N+](=O)[O-])s3)CC2)C1	C47H55F2N11O6S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-KF8XTV	SCHEMBL31110215	2-[[10-[4-[5-acetyl-3-[7-(difluoromethyl)-6-(1-methylpyrazol-4-yl)-3,4-dihydro-2H-quinolin-1-yl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]piperidin-1-yl]-10-oxodecanoyl]amino]-N-(4-methyl-5-nitro-1,3-thiazol-2-yl)benzamide	CC(=O)N1CCc2c(c(N3CCCc4cc(-c5cnn(C)c5)c(C(F)F)cc43)nn2C2CCN(C(=O)CCCCCCCCC(=O)Nc3ccccc3C(=O)Nc3nc(C)c([N+](=O)[O-])s3)CC2)C1	C48H57F2N11O6S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-RQ2QX1	SCHEMBL31110269	2-[[11-[4-[5-acetyl-3-[7-(difluoromethyl)-6-(1-methylpyrazol-4-yl)-3,4-dihydro-2H-quinolin-1-yl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]piperidin-1-yl]-11-oxoundecanoyl]amino]-N-(4-methyl-5-nitro-1,3-thiazol-2-yl)benzamide	CC(=O)N1CCc2c(c(N3CCCc4cc(-c5cnn(C)c5)c(C(F)F)cc43)nn2C2CCN(C(=O)CCCCCCCCCC(=O)Nc3ccccc3C(=O)Nc3nc(C)c([N+](=O)[O-])s3)CC2)C1	C49H59F2N11O6S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-SHCCFB	WO-2023061440-A1_CPD-207	.	CC(=O)N1CCc2c(c(N3CCCc4cc(-c5cnn(C)c5)c(C(F)F)cc43)nn2C2CCN(C(=O)CCCCCCCCCCC(=O)Nc3ccccc3C(=O)Nc3nc(C)c([N+](=O)[O-])s3)CC2)C1	C50H61F2N11O6S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-LIOAI6	SCHEMBL31110146	2-[[13-[4-[5-acetyl-3-[7-(difluoromethyl)-6-(1-methylpyrazol-4-yl)-3,4-dihydro-2H-quinolin-1-yl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]piperidin-1-yl]-13-oxotridecanoyl]amino]-N-(4-methyl-5-nitro-1,3-thiazol-2-yl)benzamide	CC(=O)N1CCc2c(c(N3CCCc4cc(-c5cnn(C)c5)c(C(F)F)cc43)nn2C2CCN(C(=O)CCCCCCCCCCCC(=O)Nc3ccccc3C(=O)Nc3nc(C)c([N+](=O)[O-])s3)CC2)C1	C51H63F2N11O6S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-XGGFKR	WO-2023061440-A1_CPD-209	.	CC(=O)N1CCc2c(c(N3CCCc4cc(-c5cnn(C)c5)c(C(F)F)cc43)nn2C2CCN(CC(=O)NCC(=O)Nc3ccccc3C(=O)Nc3nc(C)c([N+](=O)[O-])s3)CC2)C1	C42H46F2N12O6S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-KXLXBZ	WO-2023061440-A1_CPD-210	.	CC(=O)N1CCc2c(c(N3CCCc4cc(-c5cnn(C)c5)c(C(F)F)cc43)nn2C2CCN(CC(=O)NCCC(=O)Nc3ccccc3C(=O)Nc3nc(C)c([N+](=O)[O-])s3)CC2)C1	C43H48F2N12O6S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-ZO5LW3	WO-2023061440-A1_CPD-211	.	CC(=O)N1CCc2c(c(N3CCCc4cc(-c5cnn(C)c5)c(C(F)F)cc43)nn2C2CCN(CC(=O)NCCCC(=O)Nc3ccccc3C(=O)Nc3nc(C)c([N+](=O)[O-])s3)CC2)C1	C44H50F2N12O6S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-5J9UMT	WO-2023061440-A1_CPD-212	.	CC(=O)N1CCc2c(c(N3CCCc4cc(-c5cnn(C)c5)c(C(F)F)cc43)nn2C2CCN(CC(=O)NCCCCC(=O)Nc3ccccc3C(=O)Nc3nc(C)c([N+](=O)[O-])s3)CC2)C1	C45H52F2N12O6S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-4TVMHY	WO-2023061440-A1_CPD-213	.	CC(=O)N1CCc2c(c(N3CCCc4cc(-c5cnn(C)c5)c(C(F)F)cc43)nn2C2CCN(CC(=O)NCCCCCC(=O)Nc3ccccc3C(=O)Nc3nc(C)c([N+](=O)[O-])s3)CC2)C1	C46H54F2N12O6S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-WZCX5M	WO-2023061440-A1_CPD-214	.	CC(=O)N1CCc2c(c(N3CCCc4cc(-c5cnn(C)c5)c(C(F)F)cc43)nn2C2CCN(CC(=O)NCCCCCCC(=O)Nc3ccccc3C(=O)Nc3nc(C)c([N+](=O)[O-])s3)CC2)C1	C47H56F2N12O6S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-AWJKIN	WO-2023061440-A1_CPD-215	.	CC(=O)N1CCc2c(c(N3CCCc4cc(-c5cnn(C)c5)c(C(F)F)cc43)nn2C2CCN(CC(=O)NCCCCCCCC(=O)Nc3ccccc3C(=O)Nc3nc(C)c([N+](=O)[O-])s3)CC2)C1	C48H58F2N12O6S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-FB7SW1	WO-2023061440-A1_CPD-216	.	CC(=O)N1CCc2c(c(N3CCCc4cc(-c5cnn(C)c5)c(C(F)F)cc43)nn2C2CCN(CC(=O)NCCCCCCCCC(=O)Nc3ccccc3C(=O)Nc3nc(C)c([N+](=O)[O-])s3)CC2)C1	C49H60F2N12O6S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-JAXMY1	WO-2023061440-A1_CPD-217	.	CC(=O)N1CCc2c(c(N3CCCc4cc(-c5cnn(C)c5)c(C(F)F)cc43)nn2C2CCN(CC(=O)NCCCCCCCCCC(=O)Nc3ccccc3C(=O)Nc3nc(C)c([N+](=O)[O-])s3)CC2)C1	C50H62F2N12O6S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-E6PCJL	WO-2023061440-A1_CPD-218	.	CC(=O)N1CCc2c(c(N3CCCc4cc(-c5cnn(C)c5)c(C(F)F)cc43)nn2C2CCN(CC(=O)NCCCCCCCCCCC(=O)Nc3ccccc3C(=O)Nc3nc(C)c([N+](=O)[O-])s3)CC2)C1	C51H64F2N12O6S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-MQT3SU	WO-2023061440-A1_CPD-219	2-[5-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]pentanoylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)benzamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCCCNC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)sc1C	C36H37ClN8O3S2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-ILWETL	WO-2023061440-A1_CPD-220	3-[2-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]ethylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-methylbenzamide	Cc1nc(NC(=O)c2cccc(NCCNC(=O)C[C@@H]3N=C(c4ccc(Cl)cc4)c4c(sc(C)c4C)-n4c(C)nnc43)c2C)sc1C	C34H35ClN8O2S2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-D0ONPS	SCHEMBL25142642	3-[3-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]propylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-methylbenzamide	Cc1nc(NC(=O)c2cccc(NCCCNC(=O)C[C@@H]3N=C(c4ccc(Cl)cc4)c4c(sc(C)c4C)-n4c(C)nnc43)c2C)sc1C	C35H37ClN8O2S2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-FE1BKU	SCHEMBL25142651	3-[4-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]butylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-methylbenzamide	Cc1nc(NC(=O)c2cccc(NCCCCNC(=O)C[C@@H]3N=C(c4ccc(Cl)cc4)c4c(sc(C)c4C)-n4c(C)nnc43)c2C)sc1C	C36H39ClN8O2S2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-GJDF02	WO-2023061440-A1_CPD-223	3-[5-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]pentylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-methylbenzamide	Cc1nc(NC(=O)c2cccc(NCCCCCNC(=O)C[C@@H]3N=C(c4ccc(Cl)cc4)c4c(sc(C)c4C)-n4c(C)nnc43)c2C)sc1C	C37H41ClN8O2S2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-31WA0N	SCHEMBL25143513	3-[6-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]hexylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-methylbenzamide	Cc1nc(NC(=O)c2cccc(NCCCCCCNC(=O)C[C@@H]3N=C(c4ccc(Cl)cc4)c4c(sc(C)c4C)-n4c(C)nnc43)c2C)sc1C	C38H43ClN8O2S2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-L6O0YU	WO-2023061440-A1_CPD-225	3-[7-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]heptylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-methylbenzamide	Cc1nc(NC(=O)c2cccc(NCCCCCCCNC(=O)C[C@@H]3N=C(c4ccc(Cl)cc4)c4c(sc(C)c4C)-n4c(C)nnc43)c2C)sc1C	C39H45ClN8O2S2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-TO1RW4	WO-2023061440-A1_CPD-226	3-[8-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]octylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-methylbenzamide	Cc1nc(NC(=O)c2cccc(NCCCCCCCCNC(=O)C[C@@H]3N=C(c4ccc(Cl)cc4)c4c(sc(C)c4C)-n4c(C)nnc43)c2C)sc1C	C40H47ClN8O2S2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-0DS0FH	SCHEMBL25143544	3-[2-[2-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]ethoxy]ethylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-methylbenzamide	Cc1nc(NC(=O)c2cccc(NCCOCCNC(=O)C[C@@H]3N=C(c4ccc(Cl)cc4)c4c(sc(C)c4C)-n4c(C)nnc43)c2C)sc1C	C36H39ClN8O3S2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-KZ2DJ2	WO-2023061440-A1_CPD-228	.	Cc1nc(NC(=O)c2cccc(NCCOCCOCCNCC[C@@H]3N=C(c4ccc(Cl)cc4)c4c(sc(C)c4C)-n4c(C)nnc43)c2C)sc1C	C38H45ClN8O3S2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-9BCNAT	WO-2023061440-A1_CPD-229	3-[2-[2-[2-[2-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]ethoxy]ethoxy]ethoxy]ethylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-methylbenzamide	Cc1nc(NC(=O)c2cccc(NCCOCCOCCOCCNC(=O)C[C@@H]3N=C(c4ccc(Cl)cc4)c4c(sc(C)c4C)-n4c(C)nnc43)c2C)sc1C	C40H47ClN8O5S2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-X5F1AT	WO-2023061440-A1_CPD-230	3-[2-[2-[2-[2-[2-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-methylbenzamide	Cc1nc(NC(=O)c2cccc(NCCOCCOCCOCCOCCNC(=O)C[C@@H]3N=C(c4ccc(Cl)cc4)c4c(sc(C)c4C)-n4c(C)nnc43)c2C)sc1C	C42H51ClN8O6S2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-ZN2XSB	WO-2023061440-A1_CPD-231	.	Cc1nc(NC(=O)c2cccc(NCCOCCOCCOCCOCCOCCNC(=O)C[C@@H]3NC(c4ccc(Cl)cc4)c4c(sc(C)c4C)-n4c(C)nnc43)c2C)sc1C	C44H57ClN8O7S2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-XKB11C	WO-2023061440-A1_CPD-232	2-[3-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]propanoylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)benzamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCNC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)sc1C	C34H33ClN8O3S2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-4SQORT	WO-2023061440-A1_CPD-233	2-[4-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]butanoylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)benzamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCCNC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)sc1C	C35H35ClN8O3S2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-V12IZJ	WO-2023061440-A1_CPD-234	2-[6-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]hexanoylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)benzamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCCCCNC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)sc1C	C37H39ClN8O3S2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-PB1TM3	WO-2023061440-A1_CPD-235	2-[7-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]heptanoylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)benzamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCCCCCNC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)sc1C	C38H41ClN8O3S2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-DLF7X0	WO-2023061440-A1_CPD-236	2-[3-[2-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]ethoxy]propanoylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)benzamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCOCCNC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)sc1C	C36H37ClN8O4S2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-1D9K92	WO-2023061440-A1_CPD-237	2-[3-[2-[2-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]ethoxy]ethoxy]propanoylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)benzamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCOCCOCCNC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)sc1C	C38H41ClN8O5S2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-Z7MJGL	WO-2023061440-A1_CPD-238	.	Cc1nc(NC(=O)c2ccccc2NC(=O)CCOCCOCCOCCNC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3cnnc32)sc1C	C39H43ClN8O6S2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-D56RL3	WO-2023061440-A1_CPD-239	2-[3-[2-[2-[2-[2-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]propanoylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)benzamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCOCCOCCOCCOCCNC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)sc1C	C42H49ClN8O7S2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-1TOHCE	SCHEMBL25143510	2-[3-[2-[2-[2-[2-[2-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]propanoylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)benzamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCOCCOCCOCCOCCOCCNC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)sc1C	C44H53ClN8O8S2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-LK43LL	SCHEMBL25143638	2-[3-[2-[2-[2-[2-[2-[2-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]propanoylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)benzamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCOCCOCCOCCOCCOCCOCCNC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)sc1C	C46H57ClN8O9S2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-RLG75K	SCHEMBL25143643	N-[2-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]ethyl]-N'-[2-[(4,5-dimethyl-1,3-thiazol-2-yl)carbamoyl]phenyl]propanediamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CC(=O)NCCNC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)sc1C	C36H36ClN9O4S2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-JT0307	WO-2023061440-A1_CPD-243	N-[2-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]ethyl]-N'-[2-[(4,5-dimethyl-1,3-thiazol-2-yl)carbamoyl]phenyl]butanediamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCC(=O)NCCNC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)sc1C	C37H38ClN9O4S2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-KN2TC7	SCHEMBL25142432	N-[2-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]ethyl]-N'-[2-[(4,5-dimethyl-1,3-thiazol-2-yl)carbamoyl]phenyl]pentanediamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCCC(=O)NCCNC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)sc1C	C38H40ClN9O4S2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-XN307N	WO-2023061440-A1_CPD-245	N-[2-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]ethyl]-N'-[2-[(4,5-dimethyl-1,3-thiazol-2-yl)carbamoyl]phenyl]hexanediamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCCCC(=O)NCCNC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)sc1C	C39H42ClN9O4S2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-J41NTJ	WO-2023061440-A1_CPD-246	.	Cc1nc(NC(=O)c2ccccc2NC(=O)CCCCCC(=O)NCCNC(=O)C[C@@H]2NC(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)sc1C	C40H46ClN9O4S2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-UTEZV7	WO-2023061440-A1_CPD-247	N-[2-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]ethyl]-N'-[2-[(4,5-dimethyl-1,3-thiazol-2-yl)carbamoyl]phenyl]octanediamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCCCCCC(=O)NCCNC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)sc1C	C41H46ClN9O4S2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-XH4YXP	WO-2023061440-A1_CPD-248	.	Cc1nc(NC(=O)c2ccccc2NC(=O)CCCCCCCC(=O)NCCNC(=O)C[C@@H]2NC(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)sc1C	C42H50ClN9O4S2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-EV7XM5	WO-2023061440-A1_CPD-249	.	Cc1ccc(C2=N[C@@H](CC(=O)NCCNC(=O)CCCCCCCCC(=O)Nc3ccccc3C(=O)Nc3nc(C)c(C)s3)c3nnc(C)n3-c3sc(C)c(C)c32)cc1	C44H53N9O4S2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-H4TJHG	SCHEMBL25142534	2-[3-[2-[3-[2-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]ethylamino]-3-oxopropoxy]ethoxy]propanoylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)benzamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCOCCOCCC(=O)NCCNC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)sc1C	C41H46ClN9O6S2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-AP18I0	WO-2023061440-A1_CPD-251	.	Cc1nc(NC(=O)c2ccccc2NC(=O)CCOCCOCCOCCOCCC(=O)NCCNC(=O)CC2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)sc1C	C45H54ClN9O8S2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-YCTBHB	WO-2023061440-A1_CPD-252	2-[3-[2-[2-[2-[2-[3-[2-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]ethylamino]-3-oxopropoxy]ethoxy]ethoxy]ethoxy]ethoxy]propanoylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)benzamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCOCCOCCOCCOCCOCCC(=O)NCCNC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)sc1C	C47H58ClN9O9S2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-LL42UB	WO-2023061440-A1_CPD-253	2-[12-[2-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]ethylamino]dodecanoylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)benzamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCCCCCCCCCCNCCNC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)sc1C	C45H56ClN9O3S2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-4BL8G5	SCHEMBL25142810	2-[3-[2-[2-[2-[2-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]ethylamino]ethoxy]ethoxy]ethoxy]propanoylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)benzamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCOCCOCCOCCNCCNC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)sc1C	C42H50ClN9O6S2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-ET2Q2K	SCHEMBL25142819	2-[[2-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]acetyl]amino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)benzamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CNC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)sc1C	C33H31ClN8O3S2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-2KGUCW	WO-2023061440-A1_CPD-256	2-[8-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]octanoylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)benzamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCCCCCCNC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)sc1C	C39H43ClN8O3S2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-HL335P	WO-2023061440-A1_CPD-257	2-[3-[3-[2-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]ethylamino]-3-oxopropoxy]propanoylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)benzamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCOCCC(=O)NCCNC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)sc1C	C39H42ClN9O5S2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-0EZTL7	SCHEMBL25143500	2-[9-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]nonanoylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)benzamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCCCCCCCNC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)sc1C	C40H45ClN8O3S2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-JIX68N	SCHEMBL25143519	2-[9-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]nonylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)benzamide	Cc1nc(NC(=O)c2ccccc2NCCCCCCCCCNC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)sc1C	C40H47ClN8O2S2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-WU3N5Y	WO-2023061440-A1_CPD-260	.	Cc1nc(NC(=O)c2ccccc2NC(=O)CCOCCCCCOCCC(=O)NCCNC(=O)C[C@@H]2NC(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)sc1C	C44H54ClN9O6S2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-OR61PE	SCHEMBL25143208	2-[3-[2-[2-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]ethoxy]ethoxy]propylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)benzamide	Cc1nc(NC(=O)c2ccccc2NCCCOCCOCCNC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)sc1C	C38H43ClN8O4S2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-08PQ2F	WO-2023061440-A1_CPD-263	2-acetamido-4-[3-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]propylamino]-N-(4-methyl-5-nitro-1,3-thiazol-2-yl)benzamide	CC(=O)Nc1cc(NCCCNC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)ccc1C(=O)Nc1nc(C)c([N+](=O)[O-])s1	C35H35ClN10O5S2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-01LPOR	WO-2023061440-A1_CPD-264	.	CC(=O)Nc1cc(NCCCCCNC(=O)C[C@@H]2NC(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)ccc1C(=O)Nc1nc(C)c([N+](=O)[O-])s1	C37H41ClN10O5S2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-U19Q65	WO-2023061440-A1_CPD-265	.	CC(=O)Nc1cc(NCCCCCCCCCNC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)ccc1C(=O)Nc1nc(C)c(OON=O)s1	C41H47ClN10O6S2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-NOSRVE	WO-2023061440-A1_CPD-266	2-acetamido-4-[11-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]undecylamino]-N-(4-methyl-5-nitro-1,3-thiazol-2-yl)benzamide	CC(=O)Nc1cc(NCCCCCCCCCCCNC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)ccc1C(=O)Nc1nc(C)c([N+](=O)[O-])s1	C43H51ClN10O5S2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-YRSX57	SCHEMBL25142414	2-[3-[2-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]propylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCCNc5ccccc5C(=O)Nc5nc(C)c(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H57N11O6S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-3CQ6ER	SCHEMBL25143276	2-[9-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]nonylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCCCCCCCCNc5ccccc5C(=O)Nc5nc(C)c(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H61N11O4S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-OGI5C6	SCHEMBL25143020	2-[5-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]pentanoylamino]-N-(5-methylpyridin-2-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCCCC(=O)Nc5ccccc5C(=O)Nc5ccc(C)cn5)CC4)cn3)nc2n(C2CCCC2)c1=O	C44H51N11O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-EIS150	WO-2023061440-A1_CPD-270	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)Nc5ccccc5C(=O)Nc5ccc(C)c(C6CC6)n5)CC4)cn3)nc2n(C2CC=CC2)c1=O	C49H57N11O7	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-UN4209	SCHEMBL25143172	3-[2-[2-[5-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]pentoxy]ethoxy]ethylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-methylbenzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CCCCCOCCOCCNc5cccc(C(=O)Nc6nc(C)c(C)s6)c5C)CC4)cn3)nc2n(C2CCCC2)c1=O	C46H60N10O5S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-WCOR8O	SCHEMBL25143166	N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-[[2-[[2-[4-[[6-[[5-fluoro-4-(7-fluoro-2-methyl-3-propan-2-ylbenzimidazol-5-yl)pyrimidin-2-yl]amino]pyridin-3-yl]methyl]piperazin-1-yl]acetyl]amino]acetyl]amino]benzamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CNC(=O)CN2CCN(Cc3ccc(Nc4ncc(F)c(-c5cc(F)c6nc(C)n(C(C)C)c6c5)n4)nc3)CC2)sc1C	C41H44F2N12O3S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-8TWJ7L	SCHEMBL25142562	N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-[3-[[2-[4-[[6-[[5-fluoro-4-(7-fluoro-2-methyl-3-propan-2-ylbenzimidazol-5-yl)pyrimidin-2-yl]amino]pyridin-3-yl]methyl]piperazin-1-yl]acetyl]amino]propanoylamino]benzamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCNC(=O)CN2CCN(Cc3ccc(Nc4ncc(F)c(-c5cc(F)c6nc(C)n(C(C)C)c6c5)n4)nc3)CC2)sc1C	C42H46F2N12O3S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-EWPSMG	SCHEMBL25143065	N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-[4-[[2-[4-[[6-[[5-fluoro-4-(7-fluoro-2-methyl-3-propan-2-ylbenzimidazol-5-yl)pyrimidin-2-yl]amino]pyridin-3-yl]methyl]piperazin-1-yl]acetyl]amino]butanoylamino]benzamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCCNC(=O)CN2CCN(Cc3ccc(Nc4ncc(F)c(-c5cc(F)c6nc(C)n(C(C)C)c6c5)n4)nc3)CC2)sc1C	C43H48F2N12O3S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-8G4HE9	WO-2023061440-A1_CPD-275	N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-[5-[[2-[4-[[6-[[5-fluoro-4-(7-fluoro-2-methyl-3-propan-2-ylbenzimidazol-5-yl)pyrimidin-2-yl]amino]pyridin-3-yl]methyl]piperazin-1-yl]acetyl]amino]pentanoylamino]benzamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCCCNC(=O)CN2CCN(Cc3ccc(Nc4ncc(F)c(-c5cc(F)c6nc(C)n(C(C)C)c6c5)n4)nc3)CC2)sc1C	C44H50F2N12O3S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-QYSDS3	WO-2023061440-A1_CPD-276	N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-[6-[[2-[4-[[6-[[5-fluoro-4-(7-fluoro-2-methyl-3-propan-2-ylbenzimidazol-5-yl)pyrimidin-2-yl]amino]pyridin-3-yl]methyl]piperazin-1-yl]acetyl]amino]hexanoylamino]benzamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCCCCNC(=O)CN2CCN(Cc3ccc(Nc4ncc(F)c(-c5cc(F)c6nc(C)n(C(C)C)c6c5)n4)nc3)CC2)sc1C	C45H52F2N12O3S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-UOVSBX	WO-2023061440-A1_CPD-277	N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-[7-[[2-[4-[[6-[[5-fluoro-4-(7-fluoro-2-methyl-3-propan-2-ylbenzimidazol-5-yl)pyrimidin-2-yl]amino]pyridin-3-yl]methyl]piperazin-1-yl]acetyl]amino]heptanoylamino]benzamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCCCCCNC(=O)CN2CCN(Cc3ccc(Nc4ncc(F)c(-c5cc(F)c6nc(C)n(C(C)C)c6c5)n4)nc3)CC2)sc1C	C46H54F2N12O3S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-J54VJE	WO-2023061440-A1_CPD-278	N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-[8-[[2-[4-[[6-[[5-fluoro-4-(7-fluoro-2-methyl-3-propan-2-ylbenzimidazol-5-yl)pyrimidin-2-yl]amino]pyridin-3-yl]methyl]piperazin-1-yl]acetyl]amino]octanoylamino]benzamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCCCCCCNC(=O)CN2CCN(Cc3ccc(Nc4ncc(F)c(-c5cc(F)c6nc(C)n(C(C)C)c6c5)n4)nc3)CC2)sc1C	C47H56F2N12O3S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-2WW4ZT	WO-2023061440-A1_CPD-279	N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-[9-[[2-[4-[[6-[[5-fluoro-4-(7-fluoro-2-methyl-3-propan-2-ylbenzimidazol-5-yl)pyrimidin-2-yl]amino]pyridin-3-yl]methyl]piperazin-1-yl]acetyl]amino]nonanoylamino]benzamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCCCCCCCNC(=O)CN2CCN(Cc3ccc(Nc4ncc(F)c(-c5cc(F)c6nc(C)n(C(C)C)c6c5)n4)nc3)CC2)sc1C	C48H58F2N12O3S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-BUV1JQ	WO-2023061440-A1_CPD-280	N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-[3-[2-[[2-[4-[[6-[[5-fluoro-4-(7-fluoro-2-methyl-3-propan-2-ylbenzimidazol-5-yl)pyrimidin-2-yl]amino]pyridin-3-yl]methyl]piperazin-1-yl]acetyl]amino]ethoxy]propanoylamino]benzamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCOCCNC(=O)CN2CCN(Cc3ccc(Nc4ncc(F)c(-c5cc(F)c6nc(C)n(C(C)C)c6c5)n4)nc3)CC2)sc1C	C44H50F2N12O4S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-4GIFCT	WO-2023061440-A1_CPD-281	N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-[3-[2-[2-[[2-[4-[[6-[[5-fluoro-4-(7-fluoro-2-methyl-3-propan-2-ylbenzimidazol-5-yl)pyrimidin-2-yl]amino]pyridin-3-yl]methyl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]propanoylamino]benzamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCOCCOCCNC(=O)CN2CCN(Cc3ccc(Nc4ncc(F)c(-c5cc(F)c6nc(C)n(C(C)C)c6c5)n4)nc3)CC2)sc1C	C46H54F2N12O5S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-5O70WA	WO-2023061440-A1_CPD-282	N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-[3-[2-[2-[2-[[2-[4-[[6-[[5-fluoro-4-(7-fluoro-2-methyl-3-propan-2-ylbenzimidazol-5-yl)pyrimidin-2-yl]amino]pyridin-3-yl]methyl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]ethoxy]propanoylamino]benzamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCOCCOCCOCCNC(=O)CN2CCN(Cc3ccc(Nc4ncc(F)c(-c5cc(F)c6nc(C)n(C(C)C)c6c5)n4)nc3)CC2)sc1C	C48H58F2N12O6S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-9O2HHK	WO-2023061440-A1_CPD-283	N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-[3-[2-[2-[2-[2-[[2-[4-[[6-[[5-fluoro-4-(7-fluoro-2-methyl-3-propan-2-ylbenzimidazol-5-yl)pyrimidin-2-yl]amino]pyridin-3-yl]methyl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]propanoylamino]benzamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCOCCOCCOCCOCCNC(=O)CN2CCN(Cc3ccc(Nc4ncc(F)c(-c5cc(F)c6nc(C)n(C(C)C)c6c5)n4)nc3)CC2)sc1C	C50H62F2N12O7S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-HVKURT	WO-2023061440-A1_CPD-284	.	Cc1nc(NC(=O)c2ccccc2NC(=O)CCOCCOCCOCCOCCOCCNC(=O)CN2CCN(Cc3ccc(Nc4ncc(F)c(-c5cc(F)c6nc(C)n(C(C)C)c6c5)n4)nc3)CC2)sc1C	C52H66F2N12O8S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-HINCLB	WO-2023061440-A1_CPD-285	N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-[3-[2-[2-[2-[2-[2-[2-[[2-[4-[[6-[[5-fluoro-4-(7-fluoro-2-methyl-3-propan-2-ylbenzimidazol-5-yl)pyrimidin-2-yl]amino]pyridin-3-yl]methyl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]propanoylamino]benzamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCOCCOCCOCCOCCOCCOCCNC(=O)CN2CCN(Cc3ccc(Nc4ncc(F)c(-c5cc(F)c6nc(C)n(C(C)C)c6c5)n4)nc3)CC2)sc1C	C54H70F2N12O9S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-77VSYC	WO-2023061440-A1_CPD-286	.	Cc1nc(NC(=O)c2ccccc2NC(=O)CNC(=O)CN2CCN(c3ccc(Nc4ncc5cc(C(=O)N(C)C)n(C6CCCC6)c5n4)nc3)CC2)sc1C	C39H46N12O4S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-K88D69	WO-2023061440-A1_CPD-287	.	Cc1nc(NC(=O)c2ccccc2NC(=O)CCNC(=O)CN2CCN(c3ccc(Nc4ncc5cc(C(=O)N(C)C)n(C6CCCC6)c5n4)nc3)CC2)sc1C	C40H48N12O4S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-VWYC0M	WO-2023061440-A1_CPD-288	.	Cc1nc(NC(=O)c2ccccc2NC(=O)CCCNC(=O)CN2CCN(c3ccc(Nc4ncc5cc(C(=O)N(C)C)n(C6CCCC6)c5n4)nc3)CC2)sc1C	C41H50N12O4S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-F0TNTL	SCHEMBL25142991	7-cyclopentyl-2-[[5-[4-[2-[[5-[2-[(4,5-dimethyl-1,3-thiazol-2-yl)carbamoyl]anilino]-5-oxopentyl]amino]-2-oxoethyl]piperazin-1-yl]pyridin-2-yl]amino]-N,N-dimethylpyrrolo[2,3-d]pyrimidine-6-carboxamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5cc(C(=O)N(C)C)n(C6CCCC6)c5n4)nc3)CC2)sc1C	C42H52N12O4S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-W68ALF	WO-2023061440-A1_CPD-290	.	CNC(=O)c1cc2cnc(Nc3ccc(N4CCN(CC(=O)NCCCCCC(=O)Nc5ccccc5C(=O)Nc5nc(C)c(C)s5)CC4)cn3)nc2n1C1CCCC1	C42H52N12O4S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-T6XQPC	SCHEMBL25142964	7-cyclopentyl-2-[[5-[4-[2-[[7-[2-[(4,5-dimethyl-1,3-thiazol-2-yl)carbamoyl]anilino]-7-oxoheptyl]amino]-2-oxoethyl]piperazin-1-yl]pyridin-2-yl]amino]-N,N-dimethylpyrrolo[2,3-d]pyrimidine-6-carboxamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5cc(C(=O)N(C)C)n(C6CCCC6)c5n4)nc3)CC2)sc1C	C44H56N12O4S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-9E7IW8	WO-2023061440-A1_CPD-292	.	Cc1nc(NC(=O)c2ccccc2NC(=O)CCCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5cc(C(=O)N(C)C)n(C6CCCC6)c5n4)nc3)CC2)sc1C	C45H58N12O4S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-9FR8LB	SCHEMBL25142980	7-cyclopentyl-2-[[5-[4-[2-[[9-[2-[(4,5-dimethyl-1,3-thiazol-2-yl)carbamoyl]anilino]-9-oxononyl]amino]-2-oxoethyl]piperazin-1-yl]pyridin-2-yl]amino]-N,N-dimethylpyrrolo[2,3-d]pyrimidine-6-carboxamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCCCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5cc(C(=O)N(C)C)n(C6CCCC6)c5n4)nc3)CC2)sc1C	C46H60N12O4S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-2NDN7A	SCHEMBL25142896	7-cyclopentyl-2-[[5-[4-[2-[2-[3-[2-[(4,5-dimethyl-1,3-thiazol-2-yl)carbamoyl]anilino]-3-oxopropoxy]ethylamino]-2-oxoethyl]piperazin-1-yl]pyridin-2-yl]amino]-N,N-dimethylpyrrolo[2,3-d]pyrimidine-6-carboxamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCOCCNC(=O)CN2CCN(c3ccc(Nc4ncc5cc(C(=O)N(C)C)n(C6CCCC6)c5n4)nc3)CC2)sc1C	C42H52N12O5S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-W4LPGH	SCHEMBL25142719	7-cyclopentyl-2-[[5-[4-[2-[2-[2-[3-[2-[(4,5-dimethyl-1,3-thiazol-2-yl)carbamoyl]anilino]-3-oxopropoxy]ethoxy]ethylamino]-2-oxoethyl]piperazin-1-yl]pyridin-2-yl]amino]-N,N-dimethylpyrrolo[2,3-d]pyrimidine-6-carboxamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCOCCOCCNC(=O)CN2CCN(c3ccc(Nc4ncc5cc(C(=O)N(C)C)n(C6CCCC6)c5n4)nc3)CC2)sc1C	C44H56N12O6S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-E7CM1A	WO-2023061440-A1_CPD-296	.	Cc1nc(NC(=O)c2ccccc2NC(=O)CCOCCOCCOCCNC(=O)CN2CCN(c3ccc(Nc4ncc5cc(C(=O)N(C)C)n(C6CCCC6)c5n4)nc3)CC2)sc1C	C46H60N12O7S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-EE00SF	WO-2023061440-A1_CPD-297	.	Cc1nc(NC(=O)c2ccccc2NC(=O)CCOCCOCCOCCOCCNC(=O)CN2CCN(c3ccc(Nc4ncc5cc(C(=O)N(C)C)n(C6CCCC6)c5n4)nc3)CC2)sc1C	C48H64N12O8S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-RW225X	WO-2023061440-A1_CPD-298	.	Cc1nc(NC(=O)c2ccccc2NC(=O)CCOCCOCCOCCOCCOCCNC(=O)CN2CCN(c3ccc(Nc4ncc5cc(C(=O)N(C)C)n(C6CCCC6)c5n4)nc3)CC2)sc1C	C50H68N12O9S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-XA1EPE	WO-2023061440-A1_CPD-299	.	Cc1nc(NC(=O)c2ccccc2NC(=O)CCOCCOCCOCCOCCOCCOCCNC(=O)CN2CCN(c3ccc(Nc4ncc5cc(C(=O)N(C)C)n(C6CCCC6)c5n4)nc3)CC2)sc1C	C52H72N12O10S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-BZ4F7W	WO-2023061440-A1_CPD-300	N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-[[2-[[2-[4-[6-[[5-fluoro-4-(7-fluoro-2-methyl-3-propan-2-ylbenzimidazol-5-yl)pyrimidin-2-yl]amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]acetyl]amino]benzamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CNC(=O)CN2CCN(c3ccc(Nc4ncc(F)c(-c5cc(F)c6nc(C)n(C(C)C)c6c5)n4)nc3)CC2)sc1C	C40H42F2N12O3S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-25X0G5	SCHEMBL25143296	N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-[3-[[2-[4-[6-[[5-fluoro-4-(7-fluoro-2-methyl-3-propan-2-ylbenzimidazol-5-yl)pyrimidin-2-yl]amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]propanoylamino]benzamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCNC(=O)CN2CCN(c3ccc(Nc4ncc(F)c(-c5cc(F)c6nc(C)n(C(C)C)c6c5)n4)nc3)CC2)sc1C	C41H44F2N12O3S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-9SUIZL	WO-2023061440-A1_CPD-302	N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-[4-[[2-[4-[6-[[5-fluoro-4-(7-fluoro-2-methyl-3-propan-2-ylbenzimidazol-5-yl)pyrimidin-2-yl]amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]butanoylamino]benzamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCCNC(=O)CN2CCN(c3ccc(Nc4ncc(F)c(-c5cc(F)c6nc(C)n(C(C)C)c6c5)n4)nc3)CC2)sc1C	C42H46F2N12O3S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-TGQM9E	WO-2023061440-A1_CPD-303	N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-[5-[[2-[4-[6-[[5-fluoro-4-(7-fluoro-2-methyl-3-propan-2-ylbenzimidazol-5-yl)pyrimidin-2-yl]amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]pentanoylamino]benzamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCCCNC(=O)CN2CCN(c3ccc(Nc4ncc(F)c(-c5cc(F)c6nc(C)n(C(C)C)c6c5)n4)nc3)CC2)sc1C	C43H48F2N12O3S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-XN2PDU	WO-2023061440-A1_CPD-304	N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-[6-[[2-[4-[6-[[5-fluoro-4-(7-fluoro-2-methyl-3-propan-2-ylbenzimidazol-5-yl)pyrimidin-2-yl]amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]hexanoylamino]benzamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc(F)c(-c5cc(F)c6nc(C)n(C(C)C)c6c5)n4)nc3)CC2)sc1C	C44H50F2N12O3S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-DVDIZA	WO-2023061440-A1_CPD-305	N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-[7-[[2-[4-[6-[[5-fluoro-4-(7-fluoro-2-methyl-3-propan-2-ylbenzimidazol-5-yl)pyrimidin-2-yl]amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]heptanoylamino]benzamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc(F)c(-c5cc(F)c6nc(C)n(C(C)C)c6c5)n4)nc3)CC2)sc1C	C45H52F2N12O3S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-MAI1TP	WO-2023061440-A1_CPD-306	N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-[8-[[2-[4-[6-[[5-fluoro-4-(7-fluoro-2-methyl-3-propan-2-ylbenzimidazol-5-yl)pyrimidin-2-yl]amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]octanoylamino]benzamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc(F)c(-c5cc(F)c6nc(C)n(C(C)C)c6c5)n4)nc3)CC2)sc1C	C46H54F2N12O3S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-31D3JC	SCHEMBL25142793	N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-[9-[[2-[4-[6-[[5-fluoro-4-(7-fluoro-2-methyl-3-propan-2-ylbenzimidazol-5-yl)pyrimidin-2-yl]amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]nonanoylamino]benzamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCCCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc(F)c(-c5cc(F)c6nc(C)n(C(C)C)c6c5)n4)nc3)CC2)sc1C	C47H56F2N12O3S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-MGLLVN	SCHEMBL25142987	N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-[3-[2-[[2-[4-[6-[[5-fluoro-4-(7-fluoro-2-methyl-3-propan-2-ylbenzimidazol-5-yl)pyrimidin-2-yl]amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]propanoylamino]benzamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCOCCNC(=O)CN2CCN(c3ccc(Nc4ncc(F)c(-c5cc(F)c6nc(C)n(C(C)C)c6c5)n4)nc3)CC2)sc1C	C43H48F2N12O4S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-Z92T8Y	WO-2023061440-A1_CPD-309	.	Cc1nc(NC(=O)c2ccccc2NC(=O)CCOCCOCCNC(=O)CN2CCN(c3ccc(Nc4ncc(F)c(-c5cc(F)c6c(c5)N(C(C)C)C(C)N6)n4)nc3)CC2)sc1C	C45H54F2N12O5S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-3W8QWZ	WO-2023061440-A1_CPD-310	.	Cc1cnc(Nc2ccc(N3CCN(CC(=O)NCCOCCOCCOCCC(=O)Nc4ccccc4C(=O)Nc4nc(C)c(C)s4)CC3)cn2)nc1-c1cc(F)c2nc(C)n(C(C)C)c2c1	C48H59FN12O6S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-N3K66I	SCHEMBL25143481	N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-[3-[2-[2-[2-[2-[[2-[4-[6-[[5-fluoro-4-(7-fluoro-2-methyl-3-propan-2-ylbenzimidazol-5-yl)pyrimidin-2-yl]amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]propanoylamino]benzamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCOCCOCCOCCOCCNC(=O)CN2CCN(c3ccc(Nc4ncc(F)c(-c5cc(F)c6nc(C)n(C(C)C)c6c5)n4)nc3)CC2)sc1C	C49H60F2N12O7S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-RHL838	SCHEMBL25143466	N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-[3-[2-[2-[2-[2-[2-[[2-[4-[6-[[5-fluoro-4-(7-fluoro-2-methyl-3-propan-2-ylbenzimidazol-5-yl)pyrimidin-2-yl]amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]propanoylamino]benzamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCOCCOCCOCCOCCOCCNC(=O)CN2CCN(c3ccc(Nc4ncc(F)c(-c5cc(F)c6nc(C)n(C(C)C)c6c5)n4)nc3)CC2)sc1C	C51H64F2N12O8S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-7QUAN1	SCHEMBL25143496	N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-[3-[2-[2-[2-[2-[2-[2-[[2-[4-[6-[[5-fluoro-4-(7-fluoro-2-methyl-3-propan-2-ylbenzimidazol-5-yl)pyrimidin-2-yl]amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]propanoylamino]benzamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCOCCOCCOCCOCCOCCOCCNC(=O)CN2CCN(c3ccc(Nc4ncc(F)c(-c5cc(F)c6nc(C)n(C(C)C)c6c5)n4)nc3)CC2)sc1C	C53H68F2N12O9S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-I9D2EE	WO-2023061440-A1_CPD-314	N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-[[2-[[2-[4-[6-[(10-oxospiro[1,3,5,11-tetrazatricyclo[7.4.0.02,7]trideca-2,4,6,8-tetraene-13,1'-cyclohexane]-4-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]acetyl]amino]benzamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CNC(=O)CN2CCN(c3ccc(Nc4ncc5cc6n(c5n4)C4(CCCCC4)CNC6=O)nc3)CC2)sc1C	C39H44N12O4S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-LT7GC0	SCHEMBL25143473	N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-[3-[[2-[4-[6-[(10-oxospiro[1,3,5,11-tetrazatricyclo[7.4.0.02,7]trideca-2,4,6,8-tetraene-13,1'-cyclohexane]-4-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]propanoylamino]benzamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCNC(=O)CN2CCN(c3ccc(Nc4ncc5cc6n(c5n4)C4(CCCCC4)CNC6=O)nc3)CC2)sc1C	C40H46N12O4S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-3IGCFN	WO-2023061440-A1_CPD-316	N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-[4-[[2-[4-[6-[(10-oxospiro[1,3,5,11-tetrazatricyclo[7.4.0.02,7]trideca-2,4,6,8-tetraene-13,1'-cyclohexane]-4-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]butanoylamino]benzamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCCNC(=O)CN2CCN(c3ccc(Nc4ncc5cc6n(c5n4)C4(CCCCC4)CNC6=O)nc3)CC2)sc1C	C41H48N12O4S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-CS92GC	WO-2023061440-A1_CPD-317	N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-[5-[[2-[4-[6-[(10-oxospiro[1,3,5,11-tetrazatricyclo[7.4.0.02,7]trideca-2,4,6,8-tetraene-13,1'-cyclohexane]-4-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]pentanoylamino]benzamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5cc6n(c5n4)C4(CCCCC4)CNC6=O)nc3)CC2)sc1C	C42H50N12O4S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-NNLPFG	WO-2023061440-A1_CPD-318	N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-[6-[[2-[4-[6-[(10-oxospiro[1,3,5,11-tetrazatricyclo[7.4.0.02,7]trideca-2,4,6,8-tetraene-13,1'-cyclohexane]-4-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]hexanoylamino]benzamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5cc6n(c5n4)C4(CCCCC4)CNC6=O)nc3)CC2)sc1C	C43H52N12O4S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-YP6NM8	WO-2023061440-A1_CPD-319	N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-[7-[[2-[4-[6-[(10-oxospiro[1,3,5,11-tetrazatricyclo[7.4.0.02,7]trideca-2,4,6,8-tetraene-13,1'-cyclohexane]-4-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]heptanoylamino]benzamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5cc6n(c5n4)C4(CCCCC4)CNC6=O)nc3)CC2)sc1C	C44H54N12O4S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-VWYBRE	WO-2023061440-A1_CPD-320	N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-[8-[[2-[4-[6-[(10-oxospiro[1,3,5,11-tetrazatricyclo[7.4.0.02,7]trideca-2,4,6,8-tetraene-13,1'-cyclohexane]-4-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]octanoylamino]benzamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5cc6n(c5n4)C4(CCCCC4)CNC6=O)nc3)CC2)sc1C	C45H56N12O4S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-KUXXRA	SCHEMBL25142752	N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-[9-[[2-[4-[6-[(10-oxospiro[1,3,5,11-tetrazatricyclo[7.4.0.02,7]trideca-2,4,6,8-tetraene-13,1'-cyclohexane]-4-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]nonanoylamino]benzamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCCCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5cc6n(c5n4)C4(CCCCC4)CNC6=O)nc3)CC2)sc1C	C46H58N12O4S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-4CYC92	SCHEMBL25142741	N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-[3-[2-[[2-[4-[6-[(10-oxospiro[1,3,5,11-tetrazatricyclo[7.4.0.02,7]trideca-2,4,6,8-tetraene-13,1'-cyclohexane]-4-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]propanoylamino]benzamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCOCCNC(=O)CN2CCN(c3ccc(Nc4ncc5cc6n(c5n4)C4(CCCCC4)CNC6=O)nc3)CC2)sc1C	C42H50N12O5S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-XF8CFF	WO-2023061440-A1_CPD-323	.	Cc1nc(NC(=O)c2ccccc2NC(=O)CCOCCOCCNC(=O)CN2CCN(c3ccc(Nc4ncc5cc6n(c5n4)C4(CC=CCC4)CNC6=O)nc3)CC2)sc1C	C44H52N12O6S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-LHCRZ4	SCHEMBL25142696	N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-[3-[2-[2-[2-[[2-[4-[6-[(10-oxospiro[1,3,5,11-tetrazatricyclo[7.4.0.02,7]trideca-2,4,6,8-tetraene-13,1'-cyclohexane]-4-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]ethoxy]propanoylamino]benzamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCOCCOCCOCCNC(=O)CN2CCN(c3ccc(Nc4ncc5cc6n(c5n4)C4(CCCCC4)CNC6=O)nc3)CC2)sc1C	C46H58N12O7S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-A3JEGP	WO-2023061440-A1_CPD-325	N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-[3-[2-[2-[2-[2-[[2-[4-[6-[(10-oxospiro[1,3,5,11-tetrazatricyclo[7.4.0.02,7]trideca-2,4,6,8-tetraene-13,1'-cyclohexane]-4-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]propanoylamino]benzamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCOCCOCCOCCOCCNC(=O)CN2CCN(c3ccc(Nc4ncc5cc6n(c5n4)C4(CCCCC4)CNC6=O)nc3)CC2)sc1C	C48H62N12O8S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-SWF246	WO-2023061440-A1_CPD-326	.	Cc1nc(NC(=O)c2ccccc2NC(=O)CCOCCOCCOCCOCCOCCNC(=O)CN2CCN(c3ccc(Nc4ncc5cc6n(c5n4)C4(CC=CCC4)CNC6=O)nc3)CC2)sc1C	C50H64N12O9S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-DHNXDV	WO-2023061440-A1_CPD-327	N-(4,5-dimethyl-1,3-thiazol-2-yl)-2-[3-[2-[2-[2-[2-[2-[2-[[2-[4-[6-[(10-oxospiro[1,3,5,11-tetrazatricyclo[7.4.0.02,7]trideca-2,4,6,8-tetraene-13,1'-cyclohexane]-4-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]propanoylamino]benzamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCOCCOCCOCCOCCOCCOCCNC(=O)CN2CCN(c3ccc(Nc4ncc5cc6n(c5n4)C4(CCCCC4)CNC6=O)nc3)CC2)sc1C	C52H70N12O10S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-9S4EIL	WO-2023061440-A1_CPD-328	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCCCCCCNc5cccc(C(=O)Nc6ccc(C)nc6)c5C)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H59N11O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-21AGU7	WO-2023061440-A1_CPD-329	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCCCCCCNc5cccc(C(=O)Nc6cc(C)n(C)n6)c5C)CC4)cn3)nc2n(C2CCCC2)c1=O	C46H60N12O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-WN5DFL	SCHEMBL25143120	2-[5-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]pentylamino]-N-(5-methylpyridin-2-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCCCCNc5ccccc5C(=O)Nc5ccc(C)cn5)CC4)cn3)nc2n(C2CCCC2)c1=O	C44H53N11O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-X03VLM	WO-2023061440-A1_CPD-331	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCCCCCCNc5cccc(C(=O)Nc6ccc(C)nn6)c5C)CC4)cn3)nc2n(C2CCCC2)c1=O	C46H58N12O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-ZG8QF4	WO-2023061440-A1_CPD-332	.	COc1ccc(NC(=O)c2ccccc2NC(=O)CCOCCOCCN(C)C(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)nn1	C46H56N12O8	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-LU82N2	SCHEMBL25142428	3-[7-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]heptylamino]-2-methyl-N-(5-methylpyridin-2-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCCCCCCNc5cccc(C(=O)Nc6ccc(C)cn6)c5C)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H59N11O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-GUSXIV	WO-2023061440-A1_CPD-334	.	COc1ccc(NC(=O)c2cccc(NCCCCCCCNC(=O)CN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)c2C)nn1	C46H58N12O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-48D24O	WO-2023061440-A1_CPD-335	.	CNc1ccc(NC(=O)c2ccccc2NC(=O)CCOCCOCCNC(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)nn1	C45H55N13O7	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-E8B2PG	SCHEMBL25143091	2-[3-[2-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]propanoylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)-6-methylpyridine-3-carboxamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)Nc5nc(C)ccc5C(=O)Nc5nc(C)c(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H56N12O7S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-WQ1CR8	SCHEMBL25143121	2-[3-[2-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]ethoxy]ethoxy]propanoylamino]-6-chloro-N-(5-methylpyridin-2-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)Nc5cccc(Cl)c5C(=O)Nc5ccc(C)cn5)CC4)cn3)nc2n(C2CCCC2)c1=O	C46H54ClN11O7	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-VJZFRD	WO-2023061440-A1_CPD-338	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCCCCCCNc5nc(C)ccc5C(=O)Nc5nc(C)c(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H58N12O4S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-DWAYZW	WO-2023061440-A1_CPD-339	.	CNc1ccc(C(=O)Nc2ccc(C)cn2)c(NC(=O)CCOCCOCCNC(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)c1	C47H58N12O7	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-JBQ27M	WO-2023061440-A1_CPD-340	.	CNC(=O)c1ccc(C)nc1NCCCCCCCNC(=O)CN1CCN(c2ccc(Nc3ncc4c(C)c(C(C)=O)c(=O)n(C5CCCC5)c4n3)nc2)CC1	C41H55N11O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-F26EYX	WO-2023061440-A1_CPD-341	.	COc1ccc(NC(=O)c2cccc(NCCOCCOCCNC(=O)CN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)c2C)nn1	C45H56N12O7	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-ZZ63UR	WO-2023061440-A1_CPD-342	.	COc1ccc(NC(=O)c2ccccc2NC(=O)CCOCCOCCNC(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)nc1	C46H55N11O8	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-XASYMN	WO-2023061440-A1_CPD-343	.	CNc1ccc(C(=O)Nc2ccc(OC)nn2)c(NC(=O)CCOCCOCCNC(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)c1	C46H57N13O8	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-VVW4XP	WO-2023061440-A1_CPD-345	.	COc1ccc(NC(=O)c2ccccc2NC(=O)CCN2CCN(CCNC(=O)CN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)CC2)nn1	C47H58N14O6	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-NIZW5U	WO-2023061440-A1_CPD-346	.	COc1ccc(NC(=O)c2ccccc2NC(=O)CCCCN2CCC(NC(=O)CN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)CC2)nn1	C48H59N13O6	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-L6NI5Q	WO-2023061440-A1_CPD-347	.	COc1ccc(NC(=O)c2ccccc2NC(=O)COCCN2CCC(NC(=O)CN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)CC2)nn1	C47H57N13O7	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-KSPUFO	SCHEMBL25143281	2-[3-[2-[4-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]piperidin-1-yl]ethoxy]propanoylamino]-N-(6-methoxypyridazin-3-yl)benzamide	COc1ccc(NC(=O)c2ccccc2NC(=O)CCOCCN2CCC(NC(=O)CN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)CC2)nn1	C48H59N13O7	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-YPY2TV	WO-2023061440-A1_CPD-349	.	COc1ccc(NC(=O)c2ccccc2NC(=O)COCCOC2CCC(NC(=O)CN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)CC2)nn1	C48H58N12O8	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-GLLFQ6	WO-2023061440-A1_CPD-350	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)Nc5ccccc5C(=O)Nc5ccc(OC6CC6)nn5)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H56N12O8	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-REMG9H	WO-2023061440-A1_CPD-351	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)Nc5ccccc5C(=O)Nc5ccc(OC(C)C)nn5)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H58N12O8	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-CZZ9C6	WO-2023061440-A1_CPD-352	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)Nc5ccccc5C(=O)Nc5ccc(OC(F)(F)F)nn5)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H51F3N12O8	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-62GG2Z	WO-2023061440-A1_CPD-353	2-[10-[2-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]ethylamino]decanoylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)benzamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCCCCCCCCNCCNC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)sc1C	C43H52ClN9O3S2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-M80ZVC	WO-2023061440-A1_CPD-354	2-[8-[2-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]ethylamino]octanoylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)benzamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCCCCCCNCCNC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)sc1C	C41H48ClN9O3S2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-CCW6X9	WO-2023061440-A1_CPD-355	2-[6-[2-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]ethylamino]hexanoylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)benzamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCCCCNCCNC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)sc1C	C39H44ClN9O3S2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-7L9ASJ	SCHEMBL25142488	2-[4-[2-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]ethylamino]butanoylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)benzamide	Cc1nc(NC(=O)c2ccccc2NC(=O)CCCNCCNC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)sc1C	C37H40ClN9O3S2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-6PF1HR	SCHEMBL25142468	2-[3-[2-[2-[3-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]-3-oxopropoxy]ethoxy]ethoxy]propanoylamino]-N-(4,5-dimethyl-1,3-thiazol-2-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(=O)CCOCCOCCOCCC(=O)Nc5ccccc5C(=O)Nc5nc(C)c(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C46H56N10O8S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-3ZP4V1	WO-2023061440-A1_CPD-358	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)Nc5cc6c(cc5C(=O)Nc5ccc(C)cn5)CCCN6)CC4)cn3)nc2n(C2CCCC2)c1=O	C49H60N12O7	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-CFRC1G	WO-2023061440-A1_CPD-359	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)Nc5c(C(=O)Nc6ccc(C)cn6)ccc6[nH]ncc56)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H55N13O7	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-91WM1M	WO-2023061440-A1_CPD-360	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)Nc5cc6c(cc5C(=O)Nc5ccc(C)cn5)CCN6)CC4)cn3)nc2n(C2CCCC2)c1=O	C48H58N12O7	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-CUUSN3	WO-2023061440-A1_CPD-361	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)Nc5c(C(=O)Nc6ccc(C)cn6)ccc6[nH]ccc56)CC4)cn3)nc2n(C2CCCC2)c1=O	C48H56N12O7	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-5ET7GQ	WO-2023061440-A1_CPD-362	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)Nc5c(C(=O)Nc6ccc(C)cn6)ccc6ncccc56)CC4)cn3)nc2n(C2CCCC2)c1=O	C49H56N12O7	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-IFI84F	WO-2023061440-A1_CPD-363	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCCCCNc5ccccc5C(=O)Nc5nc(C)c(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C43H53N11O4S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-52IR46	WO-2023061440-A1_CPD-364	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCCCCCCNc5ccccc5C(=O)Nc5nc(C)c(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H57N11O4S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-DSJ2QC	WO-2023061440-A1_CPD-365	.	COc1ccc(NC(=O)c2ccc(N(C)C)cc2NC(=O)CCOCCOCCNC(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)nn1	C47H59N13O8	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-FOEAJB	WO-2023061440-A1_CPD-366	.	COc1ccc(NC(=O)c2ccccc2NC(=O)COCCO[C@H]2CC[C@H](NC(=O)CN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)CC2)nn1	C48H58N12O8	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-S2HCN9	WO-2023061440-A1_CPD-367	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)Nc5ccccc5C(=O)Nc5nnc(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C43H52N12O7S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-QS8FH0	WO-2023061440-A1_CPD-368	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCCCCCCNc5cc(C)ccc5C(=O)N/C(C)=N/C(C)=C(/C)S)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H63N11O4S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-JMDKJS	WO-2023061440-A1_CPD-369	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCOCCOCCC(=O)Nc5ccccc5C(=O)Nc5ccc(C#N)nn5)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H51N13O7	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-EGGPR2	WO-2023061440-A1_CPD-370	.	CNc1ccc(C(=O)Nc2nc(C)c(C)s2)c(NCCCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)c1	C46H60N12O4S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-QXAYSZ	WO-2023061440-A1_CPD-371	.	CNc1ccc(C(=O)Nc2ccc(C)c(C3CC3)n2)c(NCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)c1	C48H60N12O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-R2CXKG	WO-2023061440-A1_CPD-372	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCCCCNc5cc(F)ccc5C(=O)Nc5ccc(N(C)C)nn5)CC4)cn3)nc2n(C2CCCC2)c1=O	C44H54FN13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-AYG3CX	WO-2023061440-A1_CPD-373	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCCCCNc5cc(C)ccc5C(=O)Nc5ccc(N(C)C)nn5)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H57N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-RLQAM4	WO-2023061440-A1_CPD-374	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCCCCNc5cc(Cl)ccc5C(=O)Nc5ccc(N(C)C)nn5)CC4)cn3)nc2n(C2CCCC2)c1=O	C44H54ClN13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-4B3FYU	WO-2023061440-A1_CPD-375	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCCCNc5cc(C)ccc5C(=O)Nc5ccc(N(C)C)nn5)CC4)cn3)nc2n(C2CCCC2)c1=O	C44H55N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-4UNEPH	WO-2023061440-A1_CPD-376	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCCCCNc5cc(C#N)ccc5C(=O)Nc5ccc(N(C)C)nn5)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H54N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-ECCWE4	SCHEMBL25142502	2-[5-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]pentylamino]-4-chloro-N-(6-cyclopropyl-5-methylpyridin-2-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCCCCNc5cc(Cl)ccc5C(=O)Nc5ccc(C)c(C6CC6)n5)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H56ClN11O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-ADE92K	SCHEMBL25142423	2-[5-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]hexylamino]-4-chloro-N-(6-cyclopropyl-5-methylpyridin-2-yl)benzamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NC(C)CCCCNc5cc(Cl)ccc5C(=O)Nc5ccc(C)c(C6CC6)n5)CC4)cn3)nc2n(C2CCCC2)c1=O	C48H58ClN11O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-XKAKHQ	WO-2023061440-A1_CPD-380	.	CNc1ccc(C(=O)Nc2ccc(OC)nn2)c(NC(=O)CCOCCOCCNC(=O)CN2CCN(c3ccc(N(C)c4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)c1	C47H59N13O8	CDK4;CDK6	P11802/Q00534	DDB1	WO-2023061440-A1
TPD-U30U0F	SCHEMBL26091724	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[[3-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26094815; SCHEMBL30351554	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5C6CCC5CN(c5cc7c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)nn3)CC2)cc1Cl	C43H45ClFN9O6	IKZF1;IKZF3	Q13422/Q9UKT9	CRBN	WO-2023066350-A1
TPD-V4AWVK	SCHEMBL26092554	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[[8-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]-3,8-diazabicyclo[3.2.1]octan-3-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26092556; SCHEMBL30352143	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CC6CCC(C5)N6c5cc6c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)nn3)CC2)cc1Cl	C43H45ClFN9O6	IKZF1;IKZF3	Q13422/Q9UKT9	CRBN	WO-2023066350-A1
TPD-1EFE29	Bavdegalutamide	Bavdegalutamide; 2222112-77-6; ARV-110; 3-Pyridazinecarboxamide, N-[trans-4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[[4-[2-(2,6-dioxo-3-piperidinyl)-6-fluoro-2,3-dihydro-1,3-dioxo-1H-isoindol-5-yl]-1-piperazinyl]methyl]-1-piperidinyl]-; ARV110; N-(trans-4-(3-Chloro-4-cyanophenoxy)cyclohexyl)-6-(4-((4-(2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindolin-5-yl)piperazin-1-yl)methyl)piperidin-1-yl)pyridazine-3-carboxamide; Bavdegalutamide [INN]; Bavdegalutamide [USAN]; H6NYM0V650; Bavdegalutamide (USAN); N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; 3-Pyridazinecarboxamide, N-(trans-4-(3-chloro-4-cyanophenoxy)cyclohexyl)-6-(4-((4-(2-(2,6-dioxo-3-piperidinyl)-6-fluoro-2,3-dihydro-1,3-dioxo-1H-isoindol-5-yl)-1-piperazinyl)methyl)-1-piperidinyl)-; 6-[4-({4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxo-2,3-dihydro-1H-isoindol-5-yl]piperazin-1-yl}methyl)piperidin-1-yl]-N-[(1r,4r)-4-(3-chloro-4-cyanophenoxy)cyclohexyl]pyridazine-3-carboxamide; N-((1R,4R)-4-(3-Chloro-4-cyanophenoxy)cyclohexyl)-6-(4-((4-(2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxo-2,3-dihydro-1H-isoindol-5-yl)piperazin-1-yl)methyl)piperidin-1-yl)pyridazine-3-carboxamide; N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-({4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxo-2,3-dihydro-1H-isoindol-5-yl]piperazin-1-yl}methyl)piperidin-1-yl]pyridazine-3-carboxamide; starbld0008416; Bavdegalutamide [WHO-DD]; UNII-H6NYM0V650; Bavdegalutamide [USAN:INN]; ARV-110 (PROTAC); orb1306042; CHEMBL4862963; SCHEMBL20046698; SCHEMBL25328627; SCHEMBL26645696; SCHEMBL29382105; GTPL11512; ARV-110?; EX-A5017; BDBM50620120; s6965; WHO 11542; AKOS040745012; AT25206; AC-37002; AS-84821; BP-28371; compound 406 [WO2018071606A1]; DB-384510; HY-138641; CS-0159884; D12316; EN300-28235534	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)nn3)CC2)cc1Cl	C41H43ClFN9O6	IKZF1;IKZF3	Q13422/Q9UKT9	CRBN	WO-2023066350-A1
TPD-WLOKAI	SCHEMBL26094702	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[[6-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-3,6-diazabicyclo[3.1.1]heptan-3-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26094703; SCHEMBL30352019	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CC6CC(C5)N6c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)nn3)CC2)cc1Cl	C42H44ClN9O6	IKZF1;IKZF3	Q13422/Q9UKT9	CRBN	WO-2023066350-A1
TPD-I5Q350	SCHEMBL30351706	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[[8-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]-3,8-diazabicyclo[3.2.1]octan-3-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide	CC1(C)[C@H](NC(=O)c2ccc(N3CCC(CN4CC5CCC(C4)N5c4cc5c(cc4F)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)nn2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C45H49ClFN9O6	IKZF1;IKZF3	Q13422/Q9UKT9	CRBN	WO-2023066350-A1
TPD-N6VA4O	SCHEMBL31033647	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide	CC1(C)[C@H](NC(=O)c2ccc(N3CCC(CN4C5CCC4CN(c4ccc6c(c4)C(=O)N(C4CCC(=O)NC4=O)C6=O)C5)CC3)nn2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C45H50ClN9O6	IKZF1;IKZF3	Q13422/Q9UKT9	CRBN	WO-2023066350-A1
TPD-9X1YSH	SCHEMBL31034019	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[[6-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-3,6-diazabicyclo[3.1.1]heptan-3-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide	CC1(C)[C@H](NC(=O)c2ccc(N3CCC(CN4CC5CC(C4)N5c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)nn2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C44H48ClN9O6	IKZF1;IKZF3	Q13422/Q9UKT9	CRBN	WO-2023066350-A1
TPD-P08IKW	SCHEMBL31034001	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-3,6-diazabicyclo[3.1.1]heptan-6-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide	CC1(C)C(NC(=O)c2ccc(N3CCC(CN4C5CC4CN(c4ccc6c(c4)C(=O)N(C4CCC(=O)NC4=O)C6=O)C5)CC3)nn2)C(C)(C)C1Oc1ccc(C#N)c(Cl)c1	C44H48ClN9O6	IKZF1;IKZF3	Q13422/Q9UKT9	CRBN	WO-2023066350-A1
TPD-0OSRUC	SCHEMBL30352324	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[[8-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]-3,8-diazabicyclo[3.2.1]octan-3-yl]methyl]piperidin-1-yl]pyridine-3-carboxamide	CC1(C)[C@H](NC(=O)c2ccc(N3CCC(CN4CC5CCC(C4)N5c4cc5c(cc4F)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)nc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C46H50ClFN8O6	IKZF1;IKZF3	Q13422/Q9UKT9	CRBN	WO-2023066350-A1
TPD-56OLM1	SCHEMBL30352185	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[[6-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]-3,6-diazabicyclo[3.1.1]heptan-3-yl]methyl]piperidin-1-yl]pyridine-3-carboxamide	CC1(C)[C@H](NC(=O)c2ccc(N3CCC(CN4CC5CC(C4)N5c4cc5c(cc4F)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)nc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C45H48ClFN8O6	IKZF1;IKZF3	Q13422/Q9UKT9	CRBN	WO-2023066350-A1
TPD-S6NY2P	SCHEMBL30352149	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[[3-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]-3,6-diazabicyclo[3.1.1]heptan-6-yl]methyl]piperidin-1-yl]pyridine-3-carboxamide	CC1(C)[C@H](NC(=O)c2ccc(N3CCC(CN4C5CC4CN(c4cc6c(cc4F)C(=O)N(C4CCC(=O)NC4=O)C6=O)C5)CC3)nc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C45H48ClFN8O6	IKZF1;IKZF3	Q13422/Q9UKT9	CRBN	WO-2023066350-A1
TPD-0V9Y0A	SCHEMBL31033953	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[[8-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-3,8-diazabicyclo[3.2.1]octan-3-yl]methyl]piperidin-1-yl]pyridine-3-carboxamide	CC1(C)[C@H](NC(=O)c2ccc(N3CCC(CN4CC5CCC(C4)N5c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)nc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C46H51ClN8O6	IKZF1;IKZF3	Q13422/Q9UKT9	CRBN	WO-2023066350-A1
TPD-GG29HM	SCHEMBL31033999	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]methyl]piperidin-1-yl]pyridine-3-carboxamide	CC1(C)[C@H](NC(=O)c2ccc(N3CCC(CN4C5CCC4CN(c4ccc6c(c4)C(=O)N(C4CCC(=O)NC4=O)C6=O)C5)CC3)nc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C46H51ClN8O6	IKZF1;IKZF3	Q13422/Q9UKT9	CRBN	WO-2023066350-A1
TPD-TSUWKE	SCHEMBL31033747	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[[6-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-3,6-diazabicyclo[3.1.1]heptan-3-yl]methyl]piperidin-1-yl]pyridine-3-carboxamide	CC1(C)[C@H](NC(=O)c2ccc(N3CCC(CN4CC5CC(C4)N5c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)nc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C45H49ClN8O6	IKZF1;IKZF3	Q13422/Q9UKT9	CRBN	WO-2023066350-A1
TPD-0NE7OT	SCHEMBL26095276	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[3-[[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]-3,8-diazabicyclo[3.2.1]octan-8-yl]pyridazine-3-carboxamide; SCHEMBL30352346	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4C5CCC4CN(CC4CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC4)C5)nn3)CC2)cc1Cl	C43H45ClFN9O6	IKZF1;IKZF3	Q13422/Q9UKT9	CRBN	WO-2023066350-A1
TPD-HMV8D4	SCHEMBL26094808	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[8-[[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]-3,8-diazabicyclo[3.2.1]octan-3-yl]pyridazine-3-carboxamide; SCHEMBL30352178	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CC5CCC(C4)N5CC4CCN(c5cc6c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)nn3)CC2)cc1Cl	C43H45ClFN9O6	IKZF1;IKZF3	Q13422/Q9UKT9	CRBN	WO-2023066350-A1
TPD-HBQCGP	WO-2023066350-A1_GT-03451	.	Cc1cc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4C5CC4CN(CC4CCC(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC4)C5)nn3)CC2)ccc1C#N	C44H47FN8O6	IKZF1;IKZF3	Q13422/Q9UKT9	CRBN	WO-2023066350-A1
TPD-26SSBI	SCHEMBL26091525	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[6-[[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]-3,6-diazabicyclo[3.1.1]heptan-3-yl]pyridazine-3-carboxamide; SCHEMBL30351442	N#Cc1ccc(OC2CCC(NC(=O)c3ccc(N4CC5CC(C4)N5CC4CCN(c5cc6c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)nn3)CC2)cc1Cl	C42H43ClFN9O6	IKZF1;IKZF3	Q13422/Q9UKT9	CRBN	WO-2023066350-A1
TPD-WZEN1T	SCHEMBL31034073	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-3,6-diazabicyclo[3.1.1]heptan-6-yl]methyl]piperidin-1-yl]pyridine-3-carboxamide	CC1(C)[C@H](NC(=O)c2ccc(N3CCC(CN4C5CC4CN(c4ccc6c(c4)C(=O)N(C4CCC(=O)NC4=O)C6=O)C5)CC3)nc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C45H49ClN8O6	IKZF1;IKZF3	Q13422/Q9UKT9	CRBN	WO-2023066350-A1
TPD-5MALGQ	WO-2023066350-A1_GT-03481	.	CCC1CCC(Nc2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)CN1CC1CCN(c2ccc(C(=O)N[C@H]3C(C)(C)[C@H](Oc4ccc(C#N)c(Cl)c4)C3(C)C)cn2)CC1	C47H55ClN8O6	IKZF1;IKZF3	Q13422/Q9UKT9	CRBN	WO-2023066350-A1
TPD-YEDPQT	SCHEMBL30351597	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[[3-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]methyl]piperidin-1-yl]pyridine-3-carboxamide	CC1(C)[C@H](NC(=O)c2ccc(N3CCC(CN4C5CCC4CN(c4cc6c(cc4F)C(=O)N(C4CCC(=O)NC4=O)C6=O)C5)CC3)nc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C46H50ClFN8O6	IKZF1;IKZF3	Q13422/Q9UKT9	CRBN	WO-2023066350-A1
TPD-ILM7YF	SCHEMBL26094210	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[[6-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]-3,6-diazabicyclo[3.1.1]heptan-3-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26094213; SCHEMBL30351401	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CC6CC(C5)N6c5cc6c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)nn3)CC2)cc1Cl	C42H43ClFN9O6	IKZF1;IKZF3	Q13422/Q9UKT9	CRBN	WO-2023066350-A1
TPD-EYBAUZ	SCHEMBL26091332	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[[3-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]-3,6-diazabicyclo[3.1.1]heptan-6-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26093494; SCHEMBL30351972	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5C6CC5CN(c5cc7c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)nn3)CC2)cc1Cl	C42H43ClFN9O6	IKZF1;IKZF3	Q13422/Q9UKT9	CRBN	WO-2023066350-A1
TPD-NX7WYS	SCHEMBL26090501	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[[8-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-3,8-diazabicyclo[3.2.1]octan-3-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26090509; SCHEMBL30351416	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CC6CCC(C5)N6c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)nn3)CC2)cc1Cl	C43H46ClN9O6	IKZF1;IKZF3	Q13422/Q9UKT9	CRBN	WO-2023066350-A1
TPD-IP4NXW	SCHEMBL26093995	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26093996; SCHEMBL30351617	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5C6CCC5CN(c5ccc7c(c5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)nn3)CC2)cc1Cl	C43H46ClN9O6	IKZF1;IKZF3	Q13422/Q9UKT9	CRBN	WO-2023066350-A1
TPD-VT0NUI	SCHEMBL26091174	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-3,6-diazabicyclo[3.1.1]heptan-6-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26091178; SCHEMBL30352360	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5C6CC5CN(c5ccc7c(c5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)nn3)CC2)cc1Cl	C42H44ClN9O6	IKZF1;IKZF3	Q13422/Q9UKT9	CRBN	WO-2023066350-A1
TPD-9YF1IU	SCHEMBL30351925	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[[5-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]-2,5-diazabicyclo[2.2.2]octan-2-yl]methyl]piperidin-1-yl]pyridine-3-carboxamide	CC1(C)[C@H](NC(=O)c2ccc(N3CCC(CN4CC5CCC4CN5c4cc5c(cc4F)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)nc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C46H50ClFN8O6	IKZF1;IKZF3	Q13422/Q9UKT9	CRBN	WO-2023066350-A1
TPD-URY47H	SCHEMBL31033716	7-cyclopentyl-2-[[5-[4-[[8-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-3,8-diazabicyclo[3.2.1]octan-3-yl]methyl]piperidin-1-yl]pyridin-2-yl]amino]-N,N-dimethylpyrrolo[2,3-d]pyrimidine-6-carboxamide	CN(C)C(=O)c1cc2cnc(Nc3ccc(N4CCC(CN5CC6CCC(C5)N6c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)cn3)nc2n1C1CCCC1	C44H51N11O5	IKZF1;IKZF3	Q13422/Q9UKT9	CRBN	WO-2023066350-A1
TPD-ESPV9V	SCHEMBL31033754	7-cyclopentyl-2-[[5-[4-[[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]methyl]piperidin-1-yl]pyridin-2-yl]amino]-N,N-dimethylpyrrolo[2,3-d]pyrimidine-6-carboxamide	CN(C)C(=O)c1cc2cnc(Nc3ccc(N4CCC(CN5C6CCC5CN(c5ccc7c(c5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)cn3)nc2n1C1CCCC1	C44H51N11O5	IKZF1;IKZF3	Q13422/Q9UKT9	CRBN	WO-2023066350-A1
TPD-AO8RPC	SCHEMBL30352401	7-cyclopentyl-2-[[5-[4-[[6-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]-3,6-diazabicyclo[3.1.1]heptan-3-yl]methyl]piperidin-1-yl]pyridin-2-yl]amino]-N,N-dimethylpyrrolo[2,3-d]pyrimidine-6-carboxamide	CN(C)C(=O)c1cc2cnc(Nc3ccc(N4CCC(CN5CC6CC(C5)N6c5cc6c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)cn3)nc2n1C1CCCC1	C43H48FN11O5	IKZF1;IKZF3	Q13422/Q9UKT9	CRBN	WO-2023066350-A1
TPD-Z07Y4T	SCHEMBL30352271	7-cyclopentyl-2-[[5-[4-[[8-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]-3,8-diazabicyclo[3.2.1]octan-3-yl]methyl]piperidin-1-yl]pyridin-2-yl]amino]-N,N-dimethylpyrrolo[2,3-d]pyrimidine-6-carboxamide	CN(C)C(=O)c1cc2cnc(Nc3ccc(N4CCC(CN5CC6CCC(C5)N6c5cc6c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)cn3)nc2n1C1CCCC1	C44H50FN11O5	IKZF1;IKZF3	Q13422/Q9UKT9	CRBN	WO-2023066350-A1
TPD-5P1VZI	SCHEMBL26091389	7-cyclopentyl-2-[[5-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]pyridin-2-yl]amino]-N,N-dimethylpyrrolo[2,3-d]pyrimidine-6-carboxamide; SCHEMBL30351737	CN(C)C(=O)c1cc2cnc(Nc3ccc(N4CCC(CN5CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cn3)nc2n1C1CCCC1	C42H48FN11O5	IKZF1;IKZF3	Q13422/Q9UKT9	CRBN	WO-2023066350-A1
TPD-SBV5Q1	WO-2023066350-A1_GT-03657	.	CN(C)C(=O)c1cc2cnc(Nc3ccc(N4CCC(CN5C6CC5CN(c5cc7c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)cn3)cc2n1C1CCCC1	C44H49FN10O5	IKZF1;IKZF3	Q13422/Q9UKT9	CRBN	WO-2023066350-A1
TPD-6MN1ET	SCHEMBL30351434	7-cyclopentyl-2-[[5-[4-[[3-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]methyl]piperidin-1-yl]pyridin-2-yl]amino]-N,N-dimethylpyrrolo[2,3-d]pyrimidine-6-carboxamide	CN(C)C(=O)c1cc2cnc(Nc3ccc(N4CCC(CN5C6CCC5CN(c5cc7c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)cn3)nc2n1C1CCCC1	C44H50FN11O5	IKZF1;IKZF3	Q13422/Q9UKT9	CRBN	WO-2023066350-A1
TPD-MLX50Q	SCHEMBL31033946	7-cyclopentyl-2-[[5-[4-[[6-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-3,6-diazabicyclo[3.1.1]heptan-3-yl]methyl]piperidin-1-yl]pyridin-2-yl]amino]-N,N-dimethylpyrrolo[2,3-d]pyrimidine-6-carboxamide	CN(C)C(=O)c1cc2cnc(Nc3ccc(N4CCC(CN5CC6CC(C5)N6c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)cn3)nc2n1C1CCCC1	C43H49N11O5	IKZF1;IKZF3	Q13422/Q9UKT9	CRBN	WO-2023066350-A1
TPD-ZMRL98	WO-2023066350-A1_GT-03660	.	CN(C)C(=O)c1cc2ccc(Nc3ccc(N4CCC(CN5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cn3)nc2n1C1CCCC1	C43H50N10O5	IKZF1;IKZF3	Q13422/Q9UKT9	CRBN	WO-2023066350-A1
TPD-9DJGI7	SCHEMBL31034071	7-cyclopentyl-2-[[5-[4-[[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-3,6-diazabicyclo[3.1.1]heptan-6-yl]methyl]piperidin-1-yl]pyridin-2-yl]amino]-N,N-dimethylpyrrolo[2,3-d]pyrimidine-6-carboxamide	CN(C)C(=O)c1cc2cnc(Nc3ccc(N4CCC(CN5C6CC5CN(c5ccc7c(c5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)cn3)nc2n1C1CCCC1	C43H49N11O5	IKZF1;IKZF3	Q13422/Q9UKT9	CRBN	WO-2023066350-A1
TPD-GJFI18	SCHEMBL26091974	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[[5-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]-2,5-diazabicyclo[2.2.2]octan-2-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26091978; SCHEMBL30352104	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CC6CCC5CN6c5cc6c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)nn3)CC2)cc1Cl	C43H45ClFN9O6	IKZF1;IKZF3	Q13422/Q9UKT9	CRBN	WO-2023066350-A1
TPD-I9WRS5	SCHEMBL26091766	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[[5-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-2,5-diazabicyclo[2.2.2]octan-2-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26091771; SCHEMBL30352150	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CC6CCC5CN6c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)nn3)CC2)cc1Cl	C43H46ClN9O6	IKZF1;IKZF3	Q13422/Q9UKT9	CRBN	WO-2023066350-A1
TPD-5NDY43	WO-2023208165-A1_1	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cnn(C6(C(=O)N7CCc8cc(C(F)(F)F)ccc87)CCC6)c5)C4)cc3C2=O)C(=O)N1	C35H29F3N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-RB5QG9	WO-2023208165-A1_2	.	CN(C(=O)C1(n2cc(C#CC3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)cn2)CCC1)c1ccc(C(F)(F)F)cc1Cl	C34H28ClF3N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-QVP4VQ	WO-2023208165-A1_3	.	CCN(C(=O)C1(n2cc(C#CC3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)cn2)CCC1)c1ccc(C(F)(F)F)cc1Cl	C35H30ClF3N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-GVN3WG	WO-2023208165-A1_4	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cnn(C(C(=O)Nc6ccc(C(F)(F)F)cc6Cl)C6CC6)c5)C4)cc3C2=O)C(=O)N1	C33H26ClF3N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-UEDLTM	WO-2023208165-A1_5	.	CC(C(=O)Nc1ccc(C(F)(F)F)cc1Cl)(C1CC1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C34H28ClF3N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-RGUQB2	WO-2023208165-A1_6	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cnn(C(F)(F)C(=O)Nc6ccc(C(F)(F)F)cc6Cl)c5)C4)cc3C2=O)C(=O)N1	C30H20ClF5N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-Z9KJCM	WO-2023208165-A1_7	.	CC(C)(C(=O)N1CCc2cc(C(F)(F)F)ccc21)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C34H29F3N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-QIVAFO	WO-2023208165-A1_8	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cnn(C6(C(=O)N7Cc8ccc(C(F)(F)F)cc8C7)CCC6)c5)C4)cc3C2=O)C(=O)N1	C35H29F3N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-KS3PJC	WO-2023208165-A1_9	.	CC(C)(C(=O)N1CCc2cc(C#N)ccc21)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C34H29N7O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-621JCS	WO-2023208165-A1_10	.	N#Cc1ccc2c(c1)CCN2C(=O)C1(n2cc(C#CC3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)cn2)CCC1	C35H29N7O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-5QMH26	WO-2023208165-A1_11	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cnn(C6(C(=O)N7CCC(c8ccc(C(F)(F)F)cc8)CC7)CCC6)c5)C4)cc3C2=O)C(=O)N1	C38H35F3N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-NIYQ9L	WO-2023208165-A1_12	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cnn(C6(C(=O)N7CCC(c8ccc(C(F)(F)F)cc8)C7)CCC6)c5)C4)cc3C2=O)C(=O)N1	C37H33F3N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-RR7JXM	WO-2023208165-A1_13	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cnn(C6(C(=O)N7CCCC7c7ccc(C(F)(F)F)cc7)CCC6)c5)C4)cc3C2=O)C(=O)N1	C37H33F3N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-3MQPLA	WO-2023208165-A1_14	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cnn(C6(C(=O)N7CCc8cc(C(F)(F)F)ccc8C7)CCC6)c5)C4)cc3C2=O)C(=O)N1	C36H31F3N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-OJIDNQ	WO-2023208165-A1_15	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cnn(C6(C(=O)n7c8ccccc8c8cc(CF)ccc87)CCC6)c5)C4)cc3C2=O)C(=O)N1	C39H31FN6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-Y279WP	WO-2023208165-A1_16	.	N#Cc1ccc(NC(=O)C2(n3cc(C#CC4CN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)c(C4CC4)n3)CCC2)c(C2CC2)c1	C39H35N7O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-30Z60L	WO-2023208165-A1_17	.	CC#Cc1cc(C(F)(F)F)ccc1NC(=O)C1(n2cc(C#CC3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)c(C3CC3)n2)CCC1	C39H33F3N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-ULD3RO	WO-2023208165-A1_18	.	CC(C)(C(=O)Nc1ccc(C#N)cc1-n1cc(F)cn1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C35H28FN9O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-R17TT2	WO-2023208165-A1_19	.	CC#Cc1cc(N)ccc1NC(=O)C(C)(C)N/C=C(/C#CC1CN(c2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)C1)C=N	C34H33N7O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-NTAQK8	WO-2023208165-A1_20	.	CC(C)(C(=O)Nc1ccc(C(F)(F)F)cc1C#CC(F)(F)F)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C35H26F6N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-V0JMDQ	WO-2023208165-A1_21	.	CC(C)C#Cc1cc(C(F)(F)F)ccc1NC(=O)C(C)(C)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C37H33F3N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-I0PQ3G	WO-2023208165-A1_22	.	CN(C)Cc1ccc(NC(=O)C2(n3cc(C#CC4CN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)cn3)CCC2)c(Cl)c1	C35H34ClN7O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-9DB8X7	WO-2023208165-A1_23	.	C#Cc1ccc(NC(=O)C(C)(C)n2cc(C#CC3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)cn2)c(Cl)c1	C33H27ClN6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-177M1F	WO-2023208165-A1_24	.	CC(C)(O)C#Cc1cc(C(F)(F)F)ccc1NC(=O)C(C)(C)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C37H33F3N6O6	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-M7XOMQ	WO-2023208165-A1_25	.	CC(CC1CC1)(C(=O)Nc1ccc(C(F)(F)F)cc1Cl)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C35H30ClF3N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-WS5DFR	WO-2023208165-A1_26	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cnn(C6(C(=O)Nc7ccc(C(F)(F)F)cc7Cl)CC(O)C6)c5)C4)cc3C2=O)C(=O)N1	C33H26ClF3N6O6	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-07Y65R	WO-2023208165-A1_27	.	C#CCc1cc(C(F)(F)F)ccc1NC(=O)C(C)(C)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C35H29F3N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-0RAJPB	WO-2023208165-A1_28	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cn(C6(C(=O)Nc7ccc(C(F)(F)F)cc7Cl)CCC6)nc5C(=O)O)C4)cc3C2=O)C(=O)N1	C34H26ClF3N6O7	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-Y4OSY0	WO-2023208165-A1_29	.	CC(C)(C(=O)Nc1ccc(C#N)cc1C1CC1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)c(C(F)(F)F)n1	C36H30F3N7O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-EZ3ZN4	WO-2023208165-A1_30	.	CC#Cc1cc(C(F)(F)F)ccc1NC(=O)C(C)(C)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)c(C(F)(F)F)n1	C36H28F6N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-6MLASO	WO-2023208165-A1_31	.	CN(C)CCc1ccc(NC(=O)C2(n3cc(C#CC4CN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)cn3)CCC2)c(Cl)c1	C36H36ClN7O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-41RTTA	WO-2023208165-A1_32	.	CCC#Cc1cc(C(F)(F)F)ccc1NC(=O)C(C)(C)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C36H31F3N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-0NDMAQ	WO-2023208165-A1_33	.	CN(C)C#Cc1cc(C(F)(F)F)ccc1NC(=O)C(C)(C)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C36H32F3N7O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-78W9JY	WO-2023208165-A1_34	.	CC#Cc1cc(C(F)(F)F)ccc1NC(=O)C(C)(C)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)c(C2CC2)n1	C38H33F3N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-ST9H3Z	WO-2023208165-A1_35	.	CC(C)(C(=O)Nc1ccc(C#N)cc1C1CC1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)c(C2CC2)n1	C38H35N7O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-SUQCW0	WO-2023208165-A1_36	.	CC#Cc1ccccc1NC(=O)C(C)(C)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C34H30N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-L74O00	WO-2023208165-A1_37	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cnn(C6(CC(=O)Nc7ccc(C(F)(F)F)cc7Cl)CCC6)c5)C4)cc3C2=O)C(=O)N1	C34H28ClF3N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-11B5ZV	WO-2023208165-A1_38	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cnc(C6(NC(=O)c7ccc(C(F)(F)F)cc7CI)CCC6)s5)C4)cc3C2=O)C(=O)N1	C34H27F3IN5O5S	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-VQ54J9	WO-2023208165-A1_39	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cc6n(c5)CCN(C(=O)c5ccc(C(F)(F)F)cc5Cl)C6)C4)cc3C2=O)C(=O)N1	C33H25ClF3N5O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-TEKWLD	WO-2023208165-A1_40	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cn(C6(C(=O)Nc7ccc(C(F)(F)F)cc7Cl)CCC6)nc5CN5CCOCC5)C4)cc3C2=O)C(=O)N1	C38H35ClF3N7O6	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-HD1YDP	SCHEMBL25026330	N-[2-chloro-4-(trifluoromethyl)phenyl]-1-[3-(difluoromethyl)-4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]cyclobutane-1-carboxamide	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cn(C6(C(=O)Nc7ccc(C(F)(F)F)cc7Cl)CCC6)nc5C(F)F)C4)cc3C2=O)C(=O)N1	C34H26ClF5N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-EMEK0R	WO-2023208165-A1_42	.	CN(C)Cc1nn(C2(C(=O)Nc3ccc(C(F)(F)F)cc3Cl)CCC2)cc1C#CC1CN(c2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)C1	C36H33ClF3N7O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-CR343W	WO-2023208165-A1_43	.	CC(C)(Oc1ccc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cc1)C(=O)Nc1ccc(C#N)cc1C1CC1	C38H33N5O6	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-7D6PFE	WO-2023208165-A1_44	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cccc(C(=O)Nc6ccc(C(F)(F)F)cc6Cl)c5)C4)cc3C2=O)C(=O)N1	C32H22ClF3N4O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-IOQ2IB	WO-2023208165-A1_45	.	CC(C)(C(=O)Nc1ccc(C#N)cc1C1CC1)c1ccc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cc1	C38H33N5O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-WBTCYR	WO-2023208165-A1_46	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5ccc(C6(C(=O)Nc7ccc(C(F)(F)F)cc7Cl)CCC6)cc5)C4)cc3C2=O)C(=O)N1	C36H28ClF3N4O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-BQ6BSK	WO-2023208165-A1_47	.	CC(C)(Cn1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1)C(=O)Nc1ccc(C#N)cc1C1CC1	C36H33N7O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-J2QLWF	WO-2023208165-A1_48	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5ccn(C6(C(=O)Nc7ccc(C(F)(F)F)cc7Cl)CCC6)n5)C4)cc3C2=O)C(=O)N1	C33H26ClF3N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-CCSI3R	WO-2023208165-A1_49	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5ccnn5C5(C(=O)Nc6ccc(C(F)(F)F)cc6Cl)CCC5)C4)cc3C2=O)C(=O)N1	C33H26ClF3N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-Z9LPQQ	WO-2023208165-A1_50	.	O=C1CCC(N2C(=O)c3ccc(N4CC(c5ccc(-c6cnn(C7(C(=O)Nc8ccc(C(F)(F)F)cc8Cl)CCC7)c6)cc5)C4)cc3C2=O)C(=O)N1	C37H30ClF3N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-ZP5BVN	WO-2023208165-A1_51	.	CC(C)c1csc(-c2cc(C(F)(F)F)ccc2NC(=O)C(C)(C)n2cc(C#CC3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)cn2)n1	C38H34F3N7O5S	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-JJ3U83	WO-2023208165-A1_52	.	CC(C)(C(=O)Nc1ccc(C(F)(F)F)cc1C#CC(F)F)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C35H27F5N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-UE2V0S	WO-2023208165-A1_53	.	CC(C)(C(=O)Nc1ccc(C#N)cc1C1CC1)n1cc(N2CC(C#Cc3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C35H31N7O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-FQJDEK	WO-2023208165-A1_54	.	CC(C)(C(=O)Nc1ccccc1C1CC1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C34H32N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-FI46PS	WO-2023208165-A1_55	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5ccccc5C(=O)Nc5ccc(C(F)(F)F)cc5Cl)C4)cc3C2=O)C(=O)N1	C32H22ClF3N4O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-6ST6NE	WO-2023208165-A1_56	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cnn(C6(C(=O)Nc7ccc(C(F)(F)F)cc7C(F)(F)F)CCC6)c5)C4)cc3C2=O)C(=O)N1	C34H26F6N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-MRWBEG	WO-2023208165-A1_57	.	O=C1CCC(N2C(=O)c3ccc(-n4cc(C#Cc5cnn(C6(C(=O)Nc7ccc(C(F)(F)F)cc7Cl)CCC6)c5)cn4)cc3C2=O)C(=O)N1	C33H23ClF3N7O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-9BJ4UP	WO-2023208165-A1_58	.	O=C1CCC(N2C(=O)c3ccc(N4CC(n5cc(-c6cnn(C7(C(=O)Nc8ccc(C(F)(F)F)cc8Cl)CCC7)c6)nn5)C4)cc3C2=O)C(=O)N1	C33H27ClF3N9O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-CVZIAF	WO-2023208165-A1_59	.	CC(C)(C(=O)Nc1ccc(C#N)cc1C1CC1(F)F)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C35H29F2N7O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-YCRMYD	WO-2023208165-A1_60	.	CC(C)(C(=O)Nc1ccc(C(F)(F)F)cc1C1CC1(F)F)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C35H29F5N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-F9FHGQ	WO-2023208165-A1_61	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5nn(C6(C(=O)Nc7ccc(C(F)(F)F)cc7Cl)CCC6)c6ccccc56)C4)cc3C2=O)C(=O)N1	C37H28ClF3N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-NV7EQG	WO-2023208165-A1_62	.	CC(C)(C(=O)N1CC2(CC2)c2cc(C#N)ccc21)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C36H31N7O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-RX2S0P	WO-2023208165-A1_63	.	CC(C)(C(=O)Nc1ccc(C2CC2)cc1C#N)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C35H31N7O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-VPIMT4	WO-2023208165-A1_64	.	CC(C)(C(=O)Nc1ccc(N=O)cc1CC(F)(F)F)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C33H28F3N7O6	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-0M6NYB	WO-2023208165-A1_65	.	CC(C)(C(=O)Nc1ccc(C2CC2)cc1C1CC1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C37H36N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-RLCHRF	WO-2023208165-A1_66	.	CC(C)(C(=O)Nc1ccc(C#N)cc1C1CC1)n1cc(C#CC2CN(c3ccc4c(c3)CN(C3CCC(=O)NC3=O)C4=O)C2)cn1	C35H33N7O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-SAJD71	WO-2023208165-A1_67	.	O=C1CCC(N2C(=O)c3ccc(N4CC(CC#Cc5cnn(C6(C(=O)Nc7ccc(C(F)(F)F)cc7Cl)CCC6)c5)C4)cc3C2=O)C(=O)N1	C34H28ClF3N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-7K6PGE	WO-2023208165-A1_68	.	CC(C)(C(=O)Nc1ccc(C#N)cc1C1CC1)n1ccc(C#CCC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)c1	C37H34N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-1KAS4Y	WO-2023208165-A1_69	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5ccn(C6(C(=O)Nc7ccccc7)CCC6)c5)C4)cc3C2=O)C(=O)N1	C33H29N5O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-ZL761X	WO-2023208165-A1_70	.	O=C1CCC(N2C(=O)c3ccc(C#CC#Cc4cnn(C5(C(=O)Nc6ccc(C(F)(F)F)cc6Cl)CCC5)c4)cc3C2=O)C(=O)N1	C32H21ClF3N5O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-8MM747	WO-2023208165-A1_71	.	O=C1CCC(n2cc3cc(N4CC(C#Cc5cnn(C6(C(=O)Nc7ccc(C(F)(F)F)cc7Cl)CCC6)c5)C4)ccc3n2)C(=O)N1	C32H27ClF3N7O3	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-XDMDSU	WO-2023208165-A1_72	.	O=C1CCC(n2ncc3cc(N4CC(C#Cc5cnn(C6(C(=O)Nc7ccc(C(F)(F)F)cc7Cl)CCC6)c5)C4)ccc32)C(=O)N1	C32H27ClF3N7O3	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-BZ8ANR	WO-2023208165-A1_73	.	CC(C)(C(=O)N1CCc2cc(C(F)(F)F)ccc21)c1ccc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cc1	C37H31F3N4O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-LLKJBA	WO-2023208165-A1_74	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cc(Cl)cc(C(=O)Nc6ccc(C(F)(F)F)cc6Cl)c5)C4)cc3C2=O)C(=O)N1	C32H21Cl2F3N4O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-XZJB8A	WO-2023208165-A1_75	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cc(F)cc(C(=O)Nc6ccc(C(F)(F)F)cc6Cl)c5)C4)cc3C2=O)C(=O)N1	C32H21ClF4N4O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-LVMU3U	WO-2023208165-A1_76	.	CC(C)(C(=O)Nc1ccc(CC(F)(F)F)cc1Cl)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C33H28ClF3N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-WTJFUK	WO-2023208165-A1_77	.	CC(C)(C(=O)Nc1ccc(C#N)cc1C1CC1)n1cc(C#CC2CN(c3ccc4c(cnn4C4CCC(=O)NC4=O)c3)C2)cn1	C34H32N8O3	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-X8SXWZ	WO-2023208165-A1_78	.	CC(C)(C(=O)Nc1ccc(C#N)cc1C1CC1)n1cc(C#CC2CN(c3ccc4nn(C5CCC(=O)NC5=O)cc4c3)C2)cn1	C34H32N8O3	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-VYJ57C	WO-2023208165-A1_79	.	CC(C)(C(=O)Nc1ccc(C2CC2)cc1C(F)(F)F)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C35H31F3N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-HOC43X	WO-2023208165-A1_80	.	CC(C)(C(=O)Nc1ccc(C2CC2)cc1Cl)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C34H31ClN6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-WZX6NS	WO-2023208165-A1_81	.	CC(C)(C(=O)Nc1ccc(C#N)cc1C1CC1)c1ccc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)c(C(F)(F)F)c1	C39H32F3N5O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-LR94MH	WO-2023208165-A1_82	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cn(C6(C(=O)Nc7ccc(C(F)(F)F)cc7Cl)CCC6)nc5-c5ccccc5)C4)cc3C2=O)C(=O)N1	C39H30ClF3N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-QY012C	WO-2023208165-A1_83	.	CC(C)(C(=O)Nc1ccc(N=O)cc1C1CC1)n1nccc1C#CC1CN(c2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)C1	C34H31N7O6	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-3L0BYX	WO-2023208165-A1_84	.	CC(C(=O)Nc1ccc(C#N)cc1C1CC1)n1ccc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)n1	C34H29N7O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-GKLJIQ	WO-2023208165-A1_85	.	CC(C)(C(=O)Nc1ccc(C#N)cc1C1CC1)c1ccc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cc1F	C38H32FN5O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-FGGXKN	WO-2023208165-A1_86	.	CC(C)(C(=O)Nc1ccc(C#N)cc1C1CC1)n1cc(-c2ccc(C3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)cc2)cn1	C40H37N7O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-XB2EUG	WO-2023208165-A1_87	.	O=C1CCC(N2C(=O)c3ccc(N4CCC(c5ccc(-c6cnn(C7(C(=O)Nc8ccc(C(F)(F)F)cc8Cl)CCC7)c6)cc5)CC4)cc3C2=O)C(=O)N1	C39H34ClF3N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-8DG1ZJ	WO-2023208165-A1_88	.	O=C1CCC(N2C(=O)c3ccc(N4CCC(c5ccc(-c6cnn(C7(C(=O)Nc8ccc(C(F)(F)F)cc8Cl)CCC7)c6)cc5)C4)cc3C2=O)C(=O)N1	C38H32ClF3N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-5SWBX7	WO-2023208165-A1_89	.	CC(C)(C(=O)Nc1ccc(C#N)cc1C1CC1)c1ccc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C37H32N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-1ZRL43	WO-2023208165-A1_90	.	CC(C)(C(=O)Nc1ccc(C#N)cc1C1CC1)n1cc(-c2ccc(C3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)cc2)cn1	C41H39N7O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-YWJII8	WO-2023208165-A1_91	.	CC(C)(C(=O)Nc1ccc(N2CC(F)C2)cc1Cl)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C34H31ClFN7O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-HIYY07	WO-2023208165-A1_92	.	CC(C)c1ccc(NC(=O)C(C)(C)n2cc(C#CC3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)cn2)c(Cl)c1	C34H33ClN6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-9ML727	WO-2023208165-A1_93	.	CC(C)Cc1ccc(NC(=O)C(C)(C)n2cc(C#CC3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)cn2)c(Cl)c1	C35H35ClN6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-OK0VX0	WO-2023208165-A1_94	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5ccc(NC(=O)Nc6ccc(C(F)(F)F)cc6Cl)cc5)C4)cc3C2=O)C(=O)N1	C32H23ClF3N5O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-19NE64	WO-2023208165-A1_95	.	CC(C)(C(=O)Nc1ccc(-c2ccccc2)cc1Cl)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C37H31ClN6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-69DGFT	WO-2023208165-A1_96	.	CC(C)(C(=O)Nc1ccc2ccccc2c1Cl)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C35H29ClN6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-SR3YOY	WO-2023208165-A1_97	.	CC(C)(C(=O)Nc1ccc(-n2cccn2)cc1Cl)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C34H29ClN8O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-2U6TD8	WO-2023208165-A1_98	.	N#Cc1cn(C2(C(=O)Nc3ccc(C(F)(F)F)cc3Cl)CCC2)nc1C#CC1CN(c2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)C1	C34H25ClF3N7O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-5ZWQR2	WO-2023208165-A1_99	.	CCc1ccc(NC(=O)C(C)(C)n2cc(C#CC3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)cn2)c(Cl)c1	C33H31ClN6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-XQ17L8	WO-2023208165-A1_100	.	Cc1cnn(C(C)(C)C(=O)Nc2ccc(C#N)cc2C2CC2)c1C#CC1CN(c2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)C1	C36H33N7O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-FYXNTH	WO-2023208165-A1_101	.	Cc1cn(C(C)(C)C(=O)Nc2ccc(C#N)cc2C2CC2)nc1C#CC1CN(c2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)C1	C36H33N7O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-7M5FJB	WO-2023208165-A1_102	.	CC(C)(C(=O)Nc1ccc(C#N)cc1C1CC1)n1cc(-c2cc(F)c(C3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)cc2F)cn1	C39H33F2N7O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-87O85H	WO-2023208165-A1_103	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cccc(NC(=O)c6ccc(C(F)(F)F)cc6Cl)c5)C4)cc3C2=O)C(=O)N1	C32H22ClF3N4O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-30NFPF	WO-2023208165-A1_104	.	Cc1cc(C#N)cc(C2CC2)c1NC(=O)C(C)(C)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C36H33N7O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-DCW2PP	WO-2023208165-A1_105	.	CC(C)(C(=O)Nc1cccc(C#N)c1C1CC1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C35H31N7O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-TV0TST	WO-2023208165-A1_106	.	CC(C)(C(=O)Nc1cc(C#N)ccc1C1CC1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C35H31N7O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-6YXTDO	WO-2023208165-A1_107	.	CC(C)(C(=O)Nc1ccc(C#N)c(F)c1C1CC1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C35H30FN7O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-3QWHKS	WO-2023208165-A1_108	.	CC(C)(C(=O)Nc1c(F)cc(C#N)cc1C1CC1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C35H30FN7O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-AY6783	WO-2023208165-A1_109	.	CC(C)(C(=O)Nc1ccc(C2CC2)cc1-n1cccn1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C37H34N8O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-ZLY9I3	WO-2023208165-A1_110	.	CC(C)(C(=O)Nc1ccc(C#N)cc1C1CC1)n1cc(-c2ccc(C3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)cc2F)cn1	C39H34FN7O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-H4V1EM	WO-2023208165-A1_111	.	Cc1cc(-c2cnn(C(C)(C)C(=O)Nc3ccc(C#N)cc3C3CC3)c2)ccc1C1CN(c2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)C1	C40H37N7O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-IACXX6	WO-2023208165-A1_112	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cnn(C6(C(=O)Nc7ccc(C8CC8)cc7Cl)CCC6)c5)C4)cc3C2=O)C(=O)N1	C35H31ClN6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-3R4DQT	WO-2023208165-A1_113	.	CC(C)(C(=O)Nc1ccc(C2CC2)cc1Cl)n1cc(C#CC2CN(c3cc4c(cc3F)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C34H30ClFN6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-12QFBG	WO-2023208165-A1_114	.	Cc1cn(C2(C(=O)Nc3ccc(C(F)(F)F)cc3Cl)CCC2)nc1C#CC1CN(c2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)C1	C34H28ClF3N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-7PC89W	WO-2023208165-A1_115	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5ccc(C6(C(=O)Nc7ccc(C(F)(F)F)cc7Cl)CCC6)c(F)c5)C4)cc3C2=O)C(=O)N1	C36H27ClF4N4O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-8LO4J9	WO-2023208165-A1_116	.	CC(C)(C(=O)Nc1ccc(C#N)cc1C1CC1)n1cc(-c2ccc(C3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)c3ccccc23)cn1	C43H37N7O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-MUI1ZA	WO-2023208165-A1_117	.	CC(C)(C(=O)Nc1ccc(C#N)cc1C1CC1)n1cc(-c2ccc(C3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)c3c2CCC3)cn1	C42H39N7O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-HDDWSL	WO-2023208165-A1_118	.	O=C1CCC(N2C(=O)c3cc4c(cc3C2=O)CC(C#Cc2cnn(C3(C(=O)Nc5ccc(C(F)(F)F)cc5Cl)CCC3)c2)C4)C(=O)N1	C33H25ClF3N5O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-T70LGD	WO-2023208165-A1_119	.	CC#Cc1ccc(NC(=O)C(C)(C)n2cc(C#CC3Cc4cc5c(cc4C3)C(=O)N(C3CCC(=O)NC3=O)C5=O)cn2)c(C2CC2)c1	C37H33N5O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-FH5LFC	WO-2023208165-A1_120	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5c(F)cnn5C5(C(=O)Nc6ccc(C(F)(F)F)cc6Cl)CCC5)C4)cc3C2=O)C(=O)N1	C33H25ClF4N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-Q706A1	WO-2023208165-A1_121	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5nn(C6(C(=O)Nc7ccc(C(F)(F)F)cc7Cl)CCC6)cc5F)C4)cc3C2=O)C(=O)N1	C33H25ClF4N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-QBTQSC	WO-2023208165-A1_122	.	CC(C)(C(=O)Nc1ccc(C#N)cc1C1CC1)n1ncc(F)c1C#CC1CN(c2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)C1	C35H30FN7O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-2Z6ASM	WO-2023208165-A1_123	.	CC(C)(C(=O)Nc1ccc(C#N)cc1C1CC1)n1cc(F)c(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)n1	C35H30FN7O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-RN9YAP	WO-2023208165-A1_124	.	CC(C)(C(=O)Nc1ccc(C(F)(F)F)cc1Cl)c1ccc(-c2ccc(C3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)cc2)cc1	C39H32ClF3N4O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-DPSU4K	WO-2023208165-A1_125	.	CC(C)c1cc(C2CC2)ccc1NC(=O)C(C)(C)n1cc(C#CC2CN(c3cc4c(cc3F)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C37H37FN6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-HJCPQX	WO-2023208165-A1_126	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cnn(C6(C(=O)Nc7ccc(C8CC8)cc7C7CC7)CCC6)c5)C4)cc3C2=O)C(=O)N1	C38H36N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-AO2GUJ	WO-2023208165-A1_127	.	CC(C)(C(=O)Nc1ccc(C#N)cc1C1CC1)n1cc(C#CCN2Cc3cc4c(cc3C2)C(=O)N(C2CCC(=O)NC2=O)C4=O)cn1	C35H31N7O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-6M4CCX	WO-2023208165-A1_128	.	CC(C)(C(=O)Nc1ccc(CC2CC2)cc1Cl)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C35H33ClN6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-B86LN2	WO-2023208165-A1_129	.	CC(C)(C(=O)Nc1ccc(C#N)cc1C1CC1)c1ccc(-c2ccc(C3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)cc2)cn1	C41H36N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-GWR68W	WO-2023208165-A1_130	.	CC(C)(C(=O)Nc1ccc(C#N)cc1C1CC1)n1cc(-c2ccc(C3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)cc2)cn1	C39H35N7O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-P5VBO4	WO-2023208165-A1_131	.	Cc1cc(C2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cc(F)c1-c1cnn(C(C)(C)C(=O)Nc2ccc(C#N)cc2C2CC2)c1	C40H36FN7O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-VB34BU	WO-2023208165-A1_132	.	CC(C)(C(=O)Nc1ccc(C#N)cc1C1CC1)n1cc(-c2ccc(C3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)c(F)c2F)cn1	C39H33F2N7O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-7SS152	WO-2023208165-A1_133	.	O=C1CCC(N2C(=O)c3cc4c(cc3C2=O)CN(CC#Cc2cnn(C3(C(=O)Nc5ccc(C(F)(F)F)cc5Cl)CCC3)c2)C4)C(=O)N1	C33H26ClF3N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-QVV6BK	WO-2023208165-A1_134	.	CC(C)(C(=O)Nc1ccc(C2CC2)cc1Cl)n1cc(C#CC2CN(c3ccc4c(c3)CN(C3CCC(=O)NC3=O)C4=O)C2)cn1	C34H33ClN6O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-IV75QY	WO-2023208165-A1_135	.	CC#Cc1ccc(NC(=O)C(C)(C)n2cc(C#CC3CN(c4cc5c(cc4F)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)cn2)c(Cl)c1	C34H28ClFN6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-JEE87A	WO-2023208165-A1_136	.	O=C1CCC(N2C(=O)c3cc4c(cc3C2=O)CN(CC2CN(c3cnn(C5(C(=O)Nc6ccc(C(F)(F)F)cc6Cl)CCC5)c3)C2)C4)C(=O)N1	C34H31ClF3N7O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-AZN6GK	WO-2023208165-A1_137	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5ccc(C(=O)Nc6ccc(C(F)(F)F)cc6Cl)cc5F)C4)cc3C2=O)C(=O)N1	C32H21ClF4N4O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-ZP98X3	WO-2023208165-A1_138	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5ccnc(C(=O)Nc6ccc(C(F)(F)F)cc6Cl)c5)C4)cc3C2=O)C(=O)N1	C31H21ClF3N5O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-AFASTA	WO-2023208165-A1_139	.	N#Cc1ccc(NC(=O)c2cccc(C#CC3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)c2)c(C2CC2)c1	C35H27N5O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-WO9SKI	WO-2023208165-A1_140	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5ccc(OC(C(=O)N6CCc7cc(C(F)(F)F)ccc76)C6CC6)cc5)C4)cc3C2=O)C(=O)N1	C38H31F3N4O6	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-OCLJY2	WO-2023208165-A1_141	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5ccc6c(c5)CN(C(=O)Nc5ccc(CF)cc5Cl)CC6)C4)cc3C2=O)C(=O)N1	C35H29ClFN5O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-RQUO1D	WO-2023208165-A1_142	.	CC(C)(C(=O)Nc1ccc2c(c1Cl)CCC2)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C34H31ClN6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-GYM4MR	WO-2023208165-A1_143	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cc(F)cc(NC(=O)c6ccc(C(F)(F)F)cc6Cl)c5)C4)cc3C2=O)C(=O)N1	C32H21ClF4N4O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-AF48YO	WO-2023208165-A1_144	.	Cc1cc(F)cc(C)c1NC(=O)C(C)(C)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C33H31FN6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-J1AP3I	WO-2023208165-A1_145	.	Cc1ccc(NC(=O)C(C)(C)n2cc(C#CC3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)cn2)c(C)c1	C33H32N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-HY197E	WO-2023208165-A1_146	.	CC(C)(C(=O)Nc1ccc(C#N)cc1C1CC1)n1cc(-c2ccc(C3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)c(F)c2)cn1	C39H34FN7O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-U2ZI4M	WO-2023208165-A1_147	.	CC(C)(C(=O)Nc1c(Cl)cc(C2CC2)cc1C1CC1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C37H35ClN6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-NZOQCH	WO-2023208165-A1_148	.	CC(C)(C(=O)Nc1c(C2CC2)cc(C#N)cc1C1CC1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C38H35N7O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-YUB9GN	WO-2023208165-A1_149	.	CC(C)(C(=O)Nc1c(C2CC2)cc(C2CC2)cc1C1CC1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C40H40N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-NYKRL8	WO-2023208165-A1_150	.	CC(C)(C(=O)Nc1ccc(C2CC2)cc1F)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C34H31FN6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-98JSJO	WO-2023208165-A1_151	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cc(F)cc(NC(=O)Nc6ccc(C(F)(F)F)cc6Cl)c5)C4)cc3C2=O)C(=O)N1	C32H22ClF4N5O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-90OZ78	WO-2023208165-A1_152	.	CC(C)(C(=O)Nc1cc(C2CC2)ccc1C1CC1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C37H36N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-9K2JZB	WO-2023208165-A1_153	.	O=C1CCC(N2C(=O)c3cc(F)c(N4CC(C#Cc5cc(Cl)cc(C(=O)Nc6ccc(C(F)(F)F)cc6Cl)c5)C4)cc3C2=O)C(=O)N1	C32H20Cl2F4N4O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-RGJ0IX	WO-2023208165-A1_154	.	CC(C)(C(=O)Nc1c(Cl)cc(C#N)cc1C1CC1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C35H30ClN7O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-MPXY0Q	WO-2023208165-A1_156	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cc(F)cc(C(=O)N6CCc7cc(C(F)(F)F)ccc76)c5)C4)cc3C2=O)C(=O)N1	C34H24F4N4O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-THV8NW	WO-2023208165-A1_157	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5ccc(C(=O)Nc6ccc(C7CC7)cc6C6CC6)cc5F)C4)cc3C2=O)C(=O)N1	C37H31FN4O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-VTN0WM	WO-2023208165-A1_158	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5ccnc(C(=O)Nc6ccc(C7CC7)cc6C6CC6)c5)C4)cc3C2=O)C(=O)N1	C36H31N5O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-8OX0PS	WO-2023208165-A1_159	.	CC(C)(C(=O)Nc1c(Cl)cc(Cl)cc1C1CC1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C34H30Cl2N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-3PR0YK	WO-2023208165-A1_160	.	CC(C)(C(=O)Nc1cc(C2CC2)cc(C2CC2)c1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C37H36N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-QOA2MQ	WO-2023208165-A1_161	.	CC(C)(C(=O)Nc1ccc(C2CC2)c(C2CC2)c1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C37H36N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-MB22AB	WO-2023208165-A1_162	.	Cc1cc(C#CC2CN(c3ccc4c(c3)CN(C3CCC(=O)NC3=O)C4=O)C2)cc(C(=O)Nc2ccc(C(F)(F)F)cc2Cl)c1	C33H26ClF3N4O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-TG28SL	WO-2023208165-A1_163	.	CC(C)(C(=O)Nc1ccc(-c2ccc(F)cc2)cc1C1CC1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C40H35FN6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-ZH6SFV	WO-2023208165-A1_164	.	CC(C)(C(=O)Nc1cc2oc3ccccc3c2cc1C1CC1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C40H34N6O6	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-JXLJFG	WO-2023208165-A1_165	.	Cc1cc(C2CC2)ccc1NC(=O)C(C)(C)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C35H34N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-F6UCKS	WO-2023208165-A1_166	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cc(F)cc(C(=O)Nc6ccc(C7CC7)cc6C6CC6)c5)C4)cc3C2=O)C(=O)N1	C37H31FN4O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-ZAHN7Y	WO-2023208165-A1_167	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cc(Cl)cc(C(=O)Nc6ccc(C7CC7)cc6C6CC6)c5)C4)cc3C2=O)C(=O)N1	C37H31ClN4O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-B0YF04	WO-2023208165-A1_168	.	N#Cc1ccc(NC(=O)c2cc(F)cc(C#CC3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)c2)c2ccccc12	C36H24FN5O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-HJ8MTN	WO-2023208165-A1_169	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cc(F)cc(NC(=O)Nc6ccc(C7CC7)cc6C6CC6)c5)C4)cc3C2=O)C(=O)N1	C37H32FN5O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-MRFKEF	WO-2023208165-A1_170	.	O=C1CCC(N2C(=O)c3cc(F)c(N4CC(C#Cc5cc(F)cc(C(=O)Nc6ccc(C(F)(F)F)cc6Cl)c5)C4)cc3C2=O)C(=O)N1	C32H20ClF5N4O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-2UEHKW	WO-2023208165-A1_171	.	O=C1CCC(N2Cc3cc(N4CC(C#Cc5cc(F)cc(C(=O)Nc6ccc(C(F)(F)F)cc6Cl)c5)C4)ccc3C2=O)C(=O)N1	C32H23ClF4N4O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-DICETB	WO-2023208165-A1_172	.	CC(C)(C(=O)Nc1ccc(F)cc1C1CC1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C34H31FN6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-235VQX	WO-2023208165-A1_173	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5csc(C(=O)Nc6ccc(C7CC7)cc6C6CC6)c5)C4)cc3C2=O)C(=O)N1	C35H30N4O5S	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-9K80Y0	WO-2023208165-A1_174	.	Cc1ccc(NC(=O)C(C)(C)n2cc(C#CC3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)cn2)c(C2CC2)c1	C35H34N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-GXA7OA	WO-2023208165-A1_175	.	CC(C)(C(=O)Nc1ccc(C2CC2)cc1C1CC1)c1ccc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)c(C(F)(F)F)c1	C41H37F3N4O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-O2TO4M	WO-2023208165-A1_176	.	CC(C)(C(=O)Nc1ccc(C2CC2)cc1C1CC1)n1cc(C#CC2CN(c3ccc4c(c3)CN(C3CCC(=O)NC3=O)C4=O)C2)cn1	C37H38N6O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-BUT5MU	WO-2023208165-A1_177	.	CC(C)(C(=O)Nc1cc(C2CC2)ccc1Cl)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C34H31ClN6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-Y70R2J	WO-2023208165-A1_178	.	CC(C)(C(=O)Nc1c(Cl)cccc1C1CC1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C34H31ClN6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-UP3EXV	WO-2023208165-A1_179	.	CC(C)(C(=O)Nc1c(C2CC2)cccc1C1CC1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C37H36N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-2GL05E	WO-2023208165-A1_180	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5nc6ccc(C(=O)Nc7ccc(C8CC8)cc7C7CC7)cc6s5)C4)cc3C2=O)C(=O)N1	C38H31N5O5S	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-T5WBZM	WO-2023208165-A1_181	.	CC(C)(C(=O)Nc1ccc(C2CC2)c2c1CCO2)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C36H34N6O6	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-PJAZNB	WO-2023208165-A1_182	.	O=C1CCC(N2C(=O)c3ccc(NCC#Cc4cnn(C5(C(=O)Nc6ccc(CF)cc6Cl)CCC5)c4)cc3C2=O)C(=O)N1	C31H26ClFN6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-6Y4KUQ	WO-2023208165-A1_183	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cc(C(=O)Nc6ccc(C7CC7)cc6C6CC6)cc6ccccc56)C4)cc3C2=O)C(=O)N1	C41H34N4O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-QYQHSZ	WO-2023208165-A1_184	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cc(C(=O)Nc6ccc(C(F)(F)F)cc6Cl)cc6ccccc56)C4)cc3C2=O)C(=O)N1	C36H24ClF3N4O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-UNRB1I	WO-2023208165-A1_185	.	C#Cc1ccc(NC(=O)c2cc(F)cc(C#CC3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)c2)c(Cl)c1	C33H22ClFN4O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-ESOF7C	WO-2023208165-A1_186	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5ccc6c(c5)CC(C(=O)Nc5ccc(C(F)(F)F)cc5Cl)C6)C4)cc3C2=O)C(=O)N1	C35H26ClF3N4O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-MDS052	WO-2023208165-A1_187	.	Cc1cc(C(C)C)cc(C2CC2)c1NC(=O)C(C)(C)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C38H40N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-Z5DL2P	WO-2023208165-A1_188	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cnn(C6(C(=O)Nc7ccc(OC(F)(F)F)cc7Cl)CCC6)c5)C4)cc3C2=O)C(=O)N1	C33H26ClF3N6O6	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-J16I56	WO-2023208165-A1_189	.	CC(C)(C(=O)Nc1cccc(C2CC2)c1Cl)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C34H31ClN6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-NYWD03	WO-2023208165-A1_190	.	CC(C)(C(=O)Nc1ccc2c(c1C1CC1)CCC2)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C37H36N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-TTPR5X	WO-2023208165-A1_191	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5nc6ccc(C(=O)Nc7ccc(C(F)(F)F)cc7Cl)cc6s5)C4)cc3C2=O)C(=O)N1	C33H21ClF3N5O5S	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-J49Q9H	WO-2023208165-A1_192	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cc(C(=O)Nc6ccc(C(F)(F)F)cc6Cl)cc(C6CC6)c5)C4)cc3C2=O)C(=O)N1	C35H26ClF3N4O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-NYGL4U	WO-2023208165-A1_193	.	CC(C)(C(=O)Nc1ccc(C2CC2)cc1Cl)c1ccc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)c(C(F)(F)F)c1	C38H32ClF3N4O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-909HED	WO-2023208165-A1_194	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cc(F)cc(C(=O)Nc6ccc(C7CC7)cc6Cl)c5)C4)cc3C2=O)C(=O)N1	C34H26ClFN4O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-M0N1Q1	WO-2023208165-A1_195	.	CC(C)(C(=O)Nc1ccc(-n2cccn2)cc1C1CC1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C37H34N8O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-QFDVR9	WO-2023208165-A1_196	.	CC(C)(C(=O)Nc1cc2c(cc1C1CC1)-c1ccccc1C2)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C41H36N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-YZVGB7	WO-2023208165-A1_197	.	CC(C)(C(=O)Nc1ccc(-c2ccccc2F)cc1Cl)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C37H30ClFN6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-JNI20P	WO-2023208165-A1_198	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cc(C(=O)Nc6ccc(C(F)(F)F)cc6Cl)cc(C(F)(F)F)c5)C4)cc3C2=O)C(=O)N1	C33H21ClF6N4O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-AYB2ZE	WO-2023208165-A1_199	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5ccc6cc(C(=O)Nc7ccc(C(F)(F)F)cc7Cl)ccc6c5)C4)cc3C2=O)C(=O)N1	C36H24ClF3N4O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-GU2LSY	WO-2023208165-A1_200	.	CC(C)(C(=O)Nc1c(Cl)cc(C2CC2)cc1Cl)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C34H30Cl2N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-2IZJ0N	WO-2023208165-A1_201	.	N#Cc1ccc(NC(=O)C2CCCN(c3ccc(C4CN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)cc3)C2)c(C2CC2)c1	C38H36N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-XV3NWC	WO-2023208165-A1_202	.	O=C1CCC(N2C(=O)c3ccc(N4CC(c5ccc(-c6cnn(C7(C(=O)Nc8ccc(C(F)(F)F)cc8Cl)CCC7)c6)cc5F)C4)cc3C2=O)C(=O)N1	C37H29ClF4N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2023208165-A1
TPD-6WGJ0T	SCHEMBL24891516	3-[6-[1-[[4-[4-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]butoxy]phenyl]methyl]piperidin-4-yl]-3-oxo-1H-isoindol-2-yl]-1-methylpiperidine-2,6-dione; SCHEMBL31137782	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CCCCOc5ccc(CN6CCC(c7ccc8c(c7)CN(C7CCC(=O)N(C)C7=O)C8=O)CC6)cc5)CC4)cn3)nc2n(C2CCCC2)c1=O	C54H64N10O6	CDK4;CDK6;IKZF2	P11802/Q00534/Q9UKS7	CRBN	WO-2023288305-A1
TPD-NO96GD	SCHEMBL24891530	3-[6-[1-[[4-[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]ethoxy]phenyl]methyl]piperidin-4-yl]-3-oxo-1H-isoindol-2-yl]-1-methylpiperidine-2,6-dione; SCHEMBL30121143	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CCOc5ccc(CN6CCC(c7ccc8c(c7)CN(C7CCC(=O)N(C)C7=O)C8=O)CC6)cc5)CC4)cn3)nc2n(C2CCCC2)c1=O	C52H60N10O6	CDK4;CDK6;IKZF2	P11802/Q00534/Q9UKS7	CRBN	WO-2023288305-A1
TPD-HDECC1	SCHEMBL24891401	3-[6-[1-[[3-[2-[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]ethoxy]ethoxy]phenyl]methyl]piperidin-4-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30121159	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CCOCCOc5cccc(CN6CCC(c7ccc8c(c7)CN(C7CCC(=O)NC7=O)C8=O)CC6)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C53H62N10O7	CDK4;CDK6;IKZF2	P11802/Q00534/Q9UKS7	CRBN	WO-2023288305-A1
TPD-S98MSM	SCHEMBL24891340	3-[6-[1-[[4-[2-[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]ethoxy]ethoxy]phenyl]methyl]piperidin-4-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30121163; PD216400	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CCOCCOc5ccc(CN6CCC(c7ccc8c(c7)CN(C7CCC(=O)NC7=O)C8=O)CC6)cc5)CC4)cn3)nc2n(C2CCCC2)c1=O	C53H62N10O7	CDK4;CDK6;IKZF2	P11802/Q00534/Q9UKS7	CRBN	WO-2023288305-A1
TPD-1YEKF1	WO-2023288305-A1_Ia-3	.	CC(=O)c1c(C)c2ccc(Nc3ccc(N4CCN(CCOCCOCCOc5cccc(CN6CCC(c7ccc8c(c7)CN(C7CCC(=O)NC7=O)C8=O)CC6)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C56H67N9O8	CDK4;CDK6;IKZF2	P11802/Q00534/Q9UKS7	CRBN	WO-2023288305-A1
TPD-J0LU2F	SCHEMBL24891339	3-[6-[1-[[4-[2-[2-[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]ethoxy]ethoxy]ethoxy]phenyl]methyl]piperidin-4-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30121112; PD216402	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CCOCCOCCOc5ccc(CN6CCC(c7ccc8c(c7)CN(C7CCC(=O)NC7=O)C8=O)CC6)cc5)CC4)cn3)nc2n(C2CCCC2)c1=O	C55H66N10O8	CDK4;CDK6;IKZF2	P11802/Q00534/Q9UKS7	CRBN	WO-2023288305-A1
TPD-8HQCBT	SCHEMBL24891479	3-[6-[1-[[3-[4-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]butoxy]phenyl]methyl]piperidin-4-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30121191; PD216403	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CCCCOc5cccc(CN6CCC(c7ccc8c(c7)CN(C7CCC(=O)NC7=O)C8=O)CC6)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C53H62N10O6	CDK4;CDK6;IKZF2	P11802/Q00534/Q9UKS7	CRBN	WO-2023288305-A1
TPD-Z7FUNP	SCHEMBL24891341	3-[6-[1-[[4-[4-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]butoxy]phenyl]methyl]piperidin-4-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30121104; PD216404	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CCCCOc5ccc(CN6CCC(c7ccc8c(c7)CN(C7CCC(=O)NC7=O)C8=O)CC6)cc5)CC4)cn3)nc2n(C2CCCC2)c1=O	C53H62N10O6	CDK4;CDK6;IKZF2	P11802/Q00534/Q9UKS7	CRBN	WO-2023288305-A1
TPD-PSYB9W	SCHEMBL24891343	3-[6-[1-[[3-[6-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]hexoxy]phenyl]methyl]piperidin-4-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; PD216405	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CCCCCCOc5cccc(CN6CCC(c7ccc8c(c7)CN(C7CCC(=O)NC7=O)C8=O)CC6)c5)CC4)cn3)nc2n(C2CCCC2)c1=O	C55H66N10O6	CDK4;CDK6;IKZF2	P11802/Q00534/Q9UKS7	CRBN	WO-2023288305-A1
TPD-X3RDJF	SCHEMBL24891344	3-[6-[1-[[4-[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]ethoxy]phenyl]methyl]piperidin-4-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30121126; PD216406	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CCOc5ccc(CN6CCC(c7ccc8c(c7)CN(C7CCC(=O)NC7=O)C8=O)CC6)cc5)CC4)cn3)nc2n(C2CCCC2)c1=O	C51H58N10O6	CDK4;CDK6;IKZF2	P11802/Q00534/Q9UKS7	CRBN	WO-2023288305-A1
TPD-3LWDRW	WO-2024001839-A1_1	(2S,4R)-1-[(2S)-2-[[2-[[1-[[1-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]methoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(COCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8scnc8C)cc7)C(C)(C)C)CC6)CC5)nc4c3F)c12	C61H70F2N10O7S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-6IKBM1	WO-2024001839-A1_2	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(OCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8scnc8C)cc7)C(C)(C)C)CC6)CC5)nc4c3F)c12	C60H68F2N10O7S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-Q0G4PW	WO-2024001839-A1_3	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CC(COCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8scnc8C)cc7)C(C)(C)C)C6)CC5)nc4c3F)c12	C59H66F2N10O7S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-T8WTSH	WO-2024001839-A1_4	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CC[C@@H](OCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8scnc8C)cc7)C(C)(C)C)C6)CC5)nc4c3F)c12	C59H66F2N10O7S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-J034W1	WO-2024001839-A1_5	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CC[C@H](OCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8scnc8C)cc7)C(C)(C)C)C6)CC5)nc4c3F)c12	C59H66F2N10O7S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-UASRAB	WO-2024001839-A1_6	(2S,4R)-1-[(2S)-2-[[2-[1-[[1-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(CC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8scnc8C)cc7)C(C)(C)C)CC6)CC5)nc4c3F)c12	C60H68F2N10O6S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-1B1CER	WO-2024001839-A1_7	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(CCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8scnc8C)cc7)C(C)(C)C)CC6)CC5)nc4c3F)c12	C61H70F2N10O6S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-W0MKLD	WO-2024001839-A1_8	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CC(OCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8scnc8C)cc7)C(C)(C)C)C6)CC5)nc4c3F)c12	C58H64F2N10O7S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-PX7KTX	WO-2024001839-A1_9	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(OCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8scnc8C)cc7)C(C)(C)C)CC6)CC5)nc4c3F)c12	C60H72F2N10O7S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-AF0LYZ	WO-2024001839-A1_10	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COC2CCN(CC3(COc4nc(N5CC6CCC(C5)N6)c5cnc(-c6cc(O)cc7ccc(F)c(Cl)c67)c(F)c5n4)CC3)CC2)C(C)(C)C)cc1	C58H67ClF2N10O7S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-QVQH7O	WO-2024001839-A1_11	.	CCc1cccc2cc(O)cc(N3CCc4c(nc(OCC5(CN6CCC(OCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8scnc8C)cc7)C(C)(C)C)CC6)CC5)nc4N4CC5CCC(C4)N5)C3)c12	C60H78N10O7S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-9R17TL	WO-2024001839-A1_12	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(OCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8scnc8C)cc7)C(C)(C)C)CC6)CCC5)nc4c3F)c12	C61H70F2N10O7S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-S2LQ78	WO-2024001839-A1_13	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC5(CN6CC(CC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8scnc8C)cc7)C(C)(C)C)C6)CC5)nc4c3F)c12	C57H62F2N10O6S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-6UV06K	WO-2024001839-A1_14	.	C#Cc1c(F)ccc2cc(O)cc(-c3ccc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(OCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8scnc8C)cc7)C(C)(C)C)CC6)CC5)nc4c3F)c12	C61H69F2N9O7S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-ZXQSR3	WO-2024001839-A1_15	.	C#Cc1c(F)ccc2cc(O)cc(-c3c(Cl)cc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(OCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8scnc8C)cc7)C(C)(C)C)CC6)CC5)nc4c3F)c12	C61H68ClF2N9O7S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-AKWI5V	WO-2024001839-A1_16	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CC7CC(OCC(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)CC7C6)CC5)nc4c3F)c12	C62H70F2N10O7S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-T0W8KD	WO-2024001839-A1_17	.	C#Cc1c(F)ccc2cc(O)cc(-c3ccc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CC7(CCC(OCC(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)CC7)C6)CC5)nc4c3F)c12	C64H73F2N9O7S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-7Q31HY	WO-2024001839-A1_18	.	C#Cc1c(N)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC7(CCC(OCC(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)CC7)CC6)CC5)nc4c3F)c12	C65H78FN11O7S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-0F4O72	WO-2024001839-A1_19	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CC7(CC(OCC(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)C7)C6)CC5)nc4c3F)c12	C61H68F2N10O7S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-R6Z19E	WO-2024001839-A1_20	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC7(CC(OCC(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)C7)C6)CC5)nc4c3F)c12	C62H70F2N10O7S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-A7HZJC	WO-2024001839-A1_22	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CNC6CC7(CCC(OCC(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)C7)C6)CC5)nc4c3F)c12	C63H72F2N10O7S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-W9HPSI	WO-2024001839-A1_23	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6C7CCC6CC(COCC(=O)N[C@H](C(=O)N6C[C@H](O)CC6C(=O)N[C@@H](C)c6ccc(-c8scnc8C)cc6)C(C)(C)C)C7)CC5)nc4c3F)c12	C63H72F2N10O7S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-3FX649	WO-2024001839-A1_24	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6C7CCC6CC(OCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)c6ccc(-c8scnc8C)cc6)C(C)(C)C)C7)CC5)nc4c3F)c12	C62H70F2N10O7S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-TV56OD	WO-2024001839-A1_25	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6C7CCCC6CC(OCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)c6ccc(-c8scnc8C)cc6)C(C)(C)C)C7)CC5)nc4c3F)c12	C63H72F2N10O7S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-KM6FKP	WO-2024001839-A1_26	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CC7CCC6CC7OCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)c6ccc(-c7scnc7C)cc6)C(C)(C)C)CC5)nc4c3F)c12	C62H70F2N10O7S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-0CTFAX	WO-2024001839-A1_27	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CC7CC6CC7OCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)c6ccc(-c7scnc7C)cc6)C(C)(C)C)CC5)nc4c3F)c12	C61H68F2N10O7S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-Q63BWS	WO-2024001839-A1_28	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6[C@@H]7CC[C@H]6C[C@@H](OCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)c6ccc(-c8scnc8C)cc6)C(C)(C)C)C7)CC5)nc4c3F)c12	C62H70F2N10O7S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-C6JHDO	WO-2024001839-A1_30	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6[C@@H]7C[C@H](OCC(=O)N[C@H](C(=O)N8C[C@H](O)CC8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)C[C@H]6C7)CC5)nc4c3F)c12	C61H68F2N10O7S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-L4M3BI	WO-2024001839-A1_31	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CC7(CCC(CC(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)CC7)C6)CC5)nc4c3F)c12	C63H72F2N10O6S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-91HKSE	WO-2024001839-A1_32	(2S,4R)-1-[(2S)-2-[[2-[7-[[1-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC7(CC6)CC(CC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)c6ccc(-c8scnc8C)cc6)C(C)(C)C)C7)CC5)nc4c3F)c12	C63H72F2N10O6S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-QY0B07	WO-2024001839-A1_33	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCN(CCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8scnc8C)cc7)C(C)(C)C)CC6)CC5)cc4c3F)c12	C61H70F2N10O6S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-VSNB89	WO-2024001839-A1_34	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCCCCCN5CCC(OCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)c6ccc(Cl)cc6)C(C)(C)C)CC5)nc4c3F)c12	C56H66ClF2N9O7	KRAS	P01116	VHL	WO-2024001839-A1
TPD-2LY2AR	WO-2024001839-A1_35	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(OCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8ccccc8F)cc7)C(C)(C)C)CC6)CC5)nc4c3F)c12	C62H68F3N9O7	KRAS	P01116	VHL	WO-2024001839-A1
TPD-SS8PHP	WO-2024001839-A1_36	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(OCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)NCc7ccc8ccccc8c7)C(C)(C)C)CC6)CC5)nc4c3F)c12	C59H65F2N9O7	KRAS	P01116	VHL	WO-2024001839-A1
TPD-7WPX0Z	WO-2024001839-A1_37	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(OCC(=O)NC(C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8scnc8C)cc7)C7CCCCC7)CC6)CC5)nc4c3F)c12	C62H70F2N10O7S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-WRBWQX	WO-2024001839-A1_38	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC7(CC6)CC(OCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)c6ccc(-c8scnc8C)cc6)C(C)(C)C)C7)CC5)nc4c3F)c12	C63H76F2N10O7S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-HCOASM	WO-2024001839-A1_39	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC7(CCC(CC(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)CC7)CC6)CC5)nc4c3F)c12	C65H80F2N10O6S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-1KCAN4	WO-2024001839-A1_40	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC7(CCC(OCC(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)CC7)CC6)CC5)nc4c3F)c12	C65H80F2N10O7S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-CNK49O	WO-2024001839-A1_41	(2S,4R)-1-[(2S)-2-[[2-[[2-[[1-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-2-azaspiro[3.5]nonan-7-yl]oxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CC7(CCC(OCC(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)CC7)C6)CC5)nc4c3F)c12	C63H76F2N10O7S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-E4VGP7	WO-2024001839-A1_42	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CC7(CCC(COCC(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)CC7)C6)CC5)nc4c3F)c12	C64H80F2N10O7S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-A83GCF	WO-2024001839-A1_43	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CC7(CCC(CCC(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)CC7)C6)CC5)nc4c3F)c12	C64H78F2N10O6S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-0YVLYE	WO-2024001839-A1_44	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CC7(CCC(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)CC7)C6)CC5)nc4c3F)c12	C62H74F2N10O6S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-2G9A28	WO-2024001839-A1_45	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC7(CC6)CC(CCC(=O)N[C@H](C(=O)N6C[C@H](O)CC6C(=O)N[C@@H](C)c6ccc(-c8scnc8C)cc6)C(C)(C)C)C7)CC5)nc4c3F)c12	C64H78F2N10O6S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-6YQ22Q	WO-2024001839-A1_46	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCCCCCN5CC6(CCC(OCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8scnc8C)cc7)C(C)(C)C)C6)C5)nc4c3F)c12	C62H76F2N10O7S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-51R7JD	WO-2024001839-A1_47	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CC7(CC(CCC(=O)N[C@H](C(=O)N8C[C@H](O)CC8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)C7)C6)CC5)nc4c3F)c12	C62H74F2N10O6S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-3LM15Y	WO-2024001839-A1_48	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CC7(CC(CC(=O)N[C@H](C(=O)N8C[C@H](O)CC8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)C7)C6)CC5)nc4c3F)c12	C61H72F2N10O6S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-G0OB9I	WO-2024001839-A1_49	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CC7(CC(COCC(=O)N[C@H](C(=O)N8C[C@H](O)CC8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)C7)C6)CC5)nc4c3F)c12	C62H74F2N10O7S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-FVCD1D	WO-2024001839-A1_50	.	Cc1ccsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COC2CCN(CC3(COc4nc(N5CC6CCC(C5)N6)c5cnc(-c6ccc(F)c7sc(N)nc67)c(F)c5n4)CC3)CC2)C(C)(C)C)cc1	C56H67F2N11O6S2	KRAS	P01116	VHL	WO-2024001839-A1
TPD-N9TXZU	WO-2024001839-A1_51	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COC2CCN(CC3(COc4nc(N5CC6CCC(C5)N6)c5cnc(-c6c(C)c(F)cc7[nH]ncc67)c(F)c5n4)CC3)CC2)C(C)(C)C)cc1	C56H68F2N12O6S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-HX6KYX	WO-2024001839-A1_52	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCO[C@H](COCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8scnc8C)cc7)C(C)(C)C)C6)CC5)nc4c3F)c12	C60H72F2N10O8S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-EET59V	WO-2024001839-A1_53	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCO[C@@H](COCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8scnc8C)cc7)C(C)(C)C)C6)CC5)nc4c3F)c12	C60H72F2N10O8S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-MGW9PQ	WO-2024001839-A1_54	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)cc(OCC5(CN6CCC(OCC(=O)N[C@H](C(=O)N7C[C@H](O)CC7C(=O)N[C@@H](C)c7ccc(-c8scnc8C)cc7)C(C)(C)C)CC6)CCC5)nc4c3F)c12	C62H75F2N9O7S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-18KO0X	WO-2024001839-A1_55	(2S,4R)-1-[(2S)-2-[[2-[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-(3-oxa-7,9-diazabicyclo[3.3.1]nonan-7-yl)pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]oxyacetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6COCC(C5)N6)nc(OCC5(CN6CCC(OCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8scnc8C)cc7)C(C)(C)C)CC6)CC5)nc4c3F)c12	C60H72F2N10O8S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-6UDJS1	WO-2024001839-A1_56	(2S,4R)-1-[(2S)-2-[[2-[1-[[1-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]oxyacetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(2-methylpyrazol-3-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(OCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8ccnn8C)cc7)C(C)(C)C)CC6)CC5)nc4c3F)c12	C60H73F2N11O7	KRAS	P01116	VHL	WO-2024001839-A1
TPD-GBBYGH	WO-2024001839-A1_57	(2S,4R)-1-[(2S)-2-[[2-[1-[[1-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]oxyacetyl]amino]-3,3-dimethylbutanoyl]-N-[(1S)-1-[4-(2-ethylpyrazol-3-yl)phenyl]ethyl]-4-hydroxypyrrolidine-2-carboxamide	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(OCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8ccnn8CC)cc7)C(C)(C)C)CC6)CC5)nc4c3F)c12	C61H75F2N11O7	KRAS	P01116	VHL	WO-2024001839-A1
TPD-84KMW5	WO-2024001839-A1_58	(2S,4R)-1-[(2S)-2-[[2-[1-[[1-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]oxyacetyl]amino]-3,3-dimethylbutanoyl]-N-[(1S)-1-[2-fluoro-4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]-4-hydroxypyrrolidine-2-carboxamide	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(OCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8scnc8C)cc7F)C(C)(C)C)CC6)CC5)nc4c3F)c12	C60H71F3N10O7S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-1BITNL	WO-2024001839-A1_59	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(OCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8scnc8C)cc7O)C(C)(C)C)CC6)CC5)nc4c3F)c12	C60H72F2N10O8S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-H8T5R6	WO-2024001839-A1_60	.	CCc1c(F)ccc2cc(O)cc(-c3c(Cl)cc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(OCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8scnc8C)cc7)C(C)(C)C)CC6)CC5)nc4c3F)c12	C61H72ClF2N9O7S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-3UVDN1	WO-2024001839-A1_61	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(OCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8ccccc8F)cc7)C(C)(C)C)CC6)CC5)cc4c3F)c12	C63H73F3N8O7	KRAS	P01116	VHL	WO-2024001839-A1
TPD-S2XHYH	WO-2024001839-A1_62	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(OCC(=O)N[C@H](C(=O)N7C[C@H](O)CC7C(=O)NCc7ccc8ccccc8c7)C(C)(C)C)CC6)CC5)nc4c3F)c12	C59H69F2N9O7	KRAS	P01116	VHL	WO-2024001839-A1
TPD-ABD9L9	WO-2024001839-A1_63	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC7(CC6)CC(OCC(=O)N[C@H](C(=O)N6CC(O)C[C@H]6C(=O)N[C@@H](C)c6ccc(-c8ccccc8F)cc6)C(C)(C)C)C7)CC5)nc4c3F)c12	C65H76F3N9O7	KRAS	P01116	VHL	WO-2024001839-A1
TPD-GBKE2B	WO-2024001839-A1_64	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC7(CC6)CC(OCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)NCc6ccc8ccccc8c6)C(C)(C)C)C7)CC5)cc4c3F)c12	C63H74F2N8O7	KRAS	P01116	VHL	WO-2024001839-A1
TPD-5T3H86	WO-2024001839-A1_65	(2S,4R)-N-[(1S)-1-[4-(2-chlorophenyl)phenyl]ethyl]-1-[(2S)-2-[[2-[1-[[1-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]oxyacetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(OCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8ccccc8Cl)cc7)C(C)(C)C)CC6)CC5)nc4c3F)c12	C62H72ClF2N9O7	KRAS	P01116	VHL	WO-2024001839-A1
TPD-VRJAEB	WO-2024001839-A1_66	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(OCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)NCc7ccc8cc(F)ccc8c7)C(C)(C)C)CC6)CC5)nc4c3F)c12	C59H68F3N9O7	KRAS	P01116	VHL	WO-2024001839-A1
TPD-M2A45A	WO-2024001839-A1_67	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(OCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)NCc7ccc8cc(Cl)ccc8c7)C(C)(C)C)CC6)CC5)nc4c3F)c12	C59H68ClF2N9O7	KRAS	P01116	VHL	WO-2024001839-A1
TPD-7MY1FV	WO-2024001839-A1_68	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(OCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc8ccccc8c7)C(C)(C)C)CC6)CC5)nc4c3F)c12	C60H71F2N9O7	KRAS	P01116	VHL	WO-2024001839-A1
TPD-5TIAMC	WO-2024001839-A1_69	(2S,4R)-N-[(1S)-1-[4-(2-chlorophenyl)phenyl]ethyl]-1-[(2S)-2-[[2-[[7-[[1-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]oxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC7(CC6)CC(OCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)c6ccc(-c8ccccc8Cl)cc6)C(C)(C)C)C7)CC5)nc4c3F)c12	C65H76ClF2N9O7	KRAS	P01116	VHL	WO-2024001839-A1
TPD-32DKXU	WO-2024001839-A1_70	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC7(CC6)CC(OCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)NCc6ccc8cc(F)ccc8c6)C(C)(C)C)C7)CC5)nc4c3F)c12	C62H72F3N9O7	KRAS	P01116	VHL	WO-2024001839-A1
TPD-G6EZRZ	WO-2024001839-A1_71	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC7(CC6)CC(OCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)NCc6ccc8cc(Cl)ccc8c6)C(C)(C)C)C7)CC5)nc4c3F)c12	C62H72ClF2N9O7	KRAS	P01116	VHL	WO-2024001839-A1
TPD-RB8X38	WO-2024001839-A1_72	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC7(CC6)CC(OCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)c6ccc8ccccc8c6)C(C)(C)C)C7)CC5)nc4c3F)c12	C63H75F2N9O7	KRAS	P01116	VHL	WO-2024001839-A1
TPD-QSFG03	WO-2024001839-A1_73	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CC7(CC(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)C7)C6)CC5)nc4c3F)c12	C60H70F2N10O6S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-USEJ27	WO-2024001839-A1_74	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC7(CC6)CC(C(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)c6ccc(-c8scnc8C)cc6)C(C)(C)C)C7)CC5)nc4c3F)c12	C62H74F2N10O6S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-PRFSVF	WO-2024001839-A1_75	3-[[1-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-N-[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]-3-azaspiro[5.5]undecane-9-carboxamide	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC7(CCC(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)CC7)CC6)CC5)nc4c3F)c12	C64H78F2N10O6S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-2T3QTR	WO-2024001839-A1_76	.	C=C(N[C@@H](C)c1ccc(-c2scnc2C)cc1)[C@@H]1C[C@@H](O)CN1C(O)[C@@H](NC(=O)CCC1CCC2(CC1)CCN(CC1(COc3nc(N4CC5CCC(C4)N5)c4cnc(-c5cc(O)cc6ccc(F)c(CC)c56)c(F)c4n3)CC1)CC2)C(C)(C)C	C67H86F2N10O5S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-5MO0ZZ	WO-2024001839-A1_77	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CC2CCC3(CC2)CCN(CC2(COc4nc(N5CC6CCC(C5)N6)c5cnc(-c6cc(O)cc7ccc(F)c(C)c67)c(F)c5n4)CC2)CC3)C(C)(C)C)cc1	C64H78F2N10O6S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-5GHZID	WO-2024001839-A1_78	(2S,4R)-1-[(2S)-2-[[2-[[7-[[1-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]oxy]acetyl]amino]-3,3-dimethylbutanoyl]-N-[(1S)-1-(6-fluoronaphthalen-2-yl)ethyl]-4-hydroxypyrrolidine-2-carboxamide	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC7(CC6)CC(OCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)c6ccc8cc(F)ccc8c6)C(C)(C)C)C7)CC5)nc4c3F)c12	C63H74F3N9O7	KRAS	P01116	VHL	WO-2024001839-A1
TPD-A6IKM6	WO-2024001839-A1_79	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC7(CC6)CC(OCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)c6ccc8cc(Cl)ccc8c6)C(C)(C)C)C7)CC5)nc4c3F)c12	C63H74ClF2N9O7	KRAS	P01116	VHL	WO-2024001839-A1
TPD-7O8YLG	WO-2024001839-A1_80	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC7(CC6)CC(OCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)NCc6ccc8c(Cl)cccc8c6)C(C)(C)C)C7)CC5)nc4c3F)c12	C62H72ClF2N9O7	KRAS	P01116	VHL	WO-2024001839-A1
TPD-RA071U	WO-2024001839-A1_81	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(CCC5(CN6CC7(CCC(OCC(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)NCc8ccc9ccccc9c8)C(C)(C)C)CC7)C6)CC5)nc4c3F)c12	C63H75F2N9O6	KRAS	P01116	VHL	WO-2024001839-A1
TPD-8V21P9	WO-2024001839-A1_82	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CC7(CCC(OCC(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc9ccccc9c8)C(C)(C)C)CC7)C6)CC5)nc4c3F)c12	C63H75F2N9O7	KRAS	P01116	VHL	WO-2024001839-A1
TPD-A7LPCT	WO-2024001839-A1_83	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2CC(=O)CN2C(=O)[C@@H](NC(=O)COC2CC3(CCN(CC4(COc5nc(N6CC7CCC(C6)N7)c6cnc(-c7ccc(F)c8sc(N)nc78)c(F)c6n5)CC4)CC3)C2)C(C)(C)C)cc1	C58H68F2N12O6S2	KRAS	P01116	VHL	WO-2024001839-A1
TPD-KR9PW5	WO-2024001839-A1_84	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC[C@@H](OCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8scnc8C)cc7)C(C)(C)C)C6)CC5)nc4c3F)c12	C60H72F2N10O7S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-0E07SZ	WO-2024001839-A1_85	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(N6CCC[C@H](OCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8scnc8C)cc7)C(C)(C)C)C6)CC5)nc4c3F)c12	C59H70F2N10O7S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-RAPC7U	WO-2024001839-A1_86	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCCCCN5CCC6(CC5)CC(OCC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)c5ccc(-c7ccccc7F)cc5)C(C)(C)C)C6)nc4c3F)c12	C64H72F3N9O7	KRAS	P01116	VHL	WO-2024001839-A1
TPD-OGZF5N	WO-2024001839-A1_87	(2S,4R)-N-[(1S)-1-[4-(2-chlorophenyl)phenyl]ethyl]-1-[(2S)-2-[[2-[1-[[1-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]oxyacetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(OCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8ccccc8Cl)cc7)C(C)(C)C)CC6)CC5)nc4c3F)c12	C62H68ClF2N9O7	KRAS	P01116	VHL	WO-2024001839-A1
TPD-M1666B	WO-2024001839-A1_88	.	C#CC1=C(F)C=CC2C=C(O)C=C(c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(OCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc8ccccc8c7)C(C)(C)C)CC6)CC5)nc4c3F)C12	C60H69F2N9O7	KRAS	P01116	VHL	WO-2024001839-A1
TPD-SUVB27	WO-2024001839-A1_89	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(OCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc8cc(Cl)ccc8c7)C(C)(C)C)CC6)CC5)nc4c3F)c12	C60H66ClF2N9O7	KRAS	P01116	VHL	WO-2024001839-A1
TPD-7JQR8U	WO-2024001839-A1_90	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(OCC(=O)NC(C(=O)N7C[C@H](O)C[C@H]7C(=O)NCc7ccc8c(Cl)cccc8c7)C(C)(C)C)CC6)CC5)nc4c3F)c12	C59H64ClF2N9O7	KRAS	P01116	VHL	WO-2024001839-A1
TPD-FB58WE	WO-2024001839-A1_91	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(OCC(=O)N[C@H](C(=O)N7C[C@H](O)CC7C(=O)N[C@@H](C)c7ccc8cc(Cl)ccc8c7)C(C)(C)C)CC6)CC5)nc4c3F)c12	C60H70ClF2N9O7	KRAS	P01116	VHL	WO-2024001839-A1
TPD-851WUF	WO-2024001839-A1_92	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(OCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)NCc7ccc8c(Cl)cccc8c7)C(C)(C)C)CC6)CC5)nc4c3F)c12	C59H68ClF2N9O7	KRAS	P01116	VHL	WO-2024001839-A1
TPD-HKL55I	WO-2024001839-A1_93	(2S,4R)-1-[(2S)-2-[[2-[(3S)-1-[[1-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-3-yl]oxyacetyl]amino]-3,3-dimethylbutanoyl]-N-[(1S)-1-[4-(2-fluorophenyl)phenyl]ethyl]-4-hydroxypyrrolidine-2-carboxamide	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC[C@H](OCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8ccccc8F)cc7)C(C)(C)C)C6)CC5)nc4c3F)c12	C62H72F3N9O7	KRAS	P01116	VHL	WO-2024001839-A1
TPD-IKUB3B	WO-2024001839-A1_94	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC[C@H](OCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)NCc7ccc8ccccc8c7)C(C)C)C6)CC5)nc4c3F)c12	C58H67F2N9O7	KRAS	P01116	VHL	WO-2024001839-A1
TPD-NJ1YXG	WO-2024001839-A1_95	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC[C@H](OCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8scnc8C)cc7)C(C)(C)C)C6)CC5)nc4c3F)c12	C60H68F2N10O7S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-MFBB2C	WO-2024001839-A1_96	(2S,4R)-1-[(2S)-2-[[2-[(3S)-1-[[1-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-3-yl]oxyacetyl]amino]-3,3-dimethylbutanoyl]-N-[(1S)-1-[4-(2-fluorophenyl)phenyl]ethyl]-4-hydroxypyrrolidine-2-carboxamide	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC[C@H](OCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8ccccc8F)cc7)C(C)(C)C)C6)CC5)nc4c3F)c12	C62H68F3N9O7	KRAS	P01116	VHL	WO-2024001839-A1
TPD-2V7OYO	WO-2024001839-A1_97	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC[C@H](OCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)NCc7ccc8ccccc8c7)C(C)(C)C)C6)CC5)nc4c3F)c12	C59H65F2N9O7	KRAS	P01116	VHL	WO-2024001839-A1
TPD-RJBT11	WO-2024001839-A1_98	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC7(CC6)CC(OCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](CO)c6ccc(-c8ccccc8F)cc6)C(C)(C)C)C7)CC5)nc4c3F)c12	C65H76F3N9O8	KRAS	P01116	VHL	WO-2024001839-A1
TPD-AKY4QE	WO-2024001839-A1_99	.	Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(OCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](CO)c7ccc(-c8ccccc8F)cc7)C(C)(C)C)CC6)CC5)nc4c3F)c12	C61H70F3N9O8	KRAS	P01116	VHL	WO-2024001839-A1
TPD-ETAAR9	WO-2024001839-A1_100	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC7(CC6)CC(OCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](CO)c6ccc(-c8ccccc8F)cc6)C(C)(C)C)C7)CC5)nc4c3F)c12	C65H72F3N9O8	KRAS	P01116	VHL	WO-2024001839-A1
TPD-TGCSJP	WO-2024001839-A1_101	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(OCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](CO)c7ccc(-c8ccccc8Cl)cc7)C(C)(C)C)CC6)CC5)cc4c3F)c12	C63H69ClF2N8O8	KRAS	P01116	VHL	WO-2024001839-A1
TPD-FJGBJH	WO-2024001839-A1_102	(2S,4R)-N-[(1R)-1-[4-(2-chlorophenyl)phenyl]-2-hydroxyethyl]-1-[(2S)-2-[[2-[[7-[[1-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]oxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC7(CC6)CC(OCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](CO)c6ccc(-c8ccccc8Cl)cc6)C(C)(C)C)C7)CC5)nc4c3F)c12	C65H72ClF2N9O8	KRAS	P01116	VHL	WO-2024001839-A1
TPD-U1F93R	WO-2024001839-A1_103	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(OCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](CO)c7ccc(-c8scnc8C)cc7)C(C)(C)C)CC6)CC5)nc4c3F)c12	C60H68F2N10O8S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-4NEZZS	WO-2024001839-A1_104	(2S,4R)-N-[(1R)-1-[4-(2-chlorophenyl)phenyl]-2-hydroxyethyl]-1-[(2S)-2-[[2-[1-[[1-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]oxyacetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(OCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](CO)c7ccc(-c8ccccc8Cl)cc7)C(C)(C)C)CC6)CC5)nc4c3F)c12	C62H72ClF2N9O8	KRAS	P01116	VHL	WO-2024001839-A1
TPD-IBLK6L	WO-2024001839-A1_105	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(OCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](CO)c7ccc(-c8ccccc8F)cc7)C(C)(C)C)CC6)CC5)nc4c3F)c12	C62H72F3N9O8	KRAS	P01116	VHL	WO-2024001839-A1
TPD-XQX0ML	WO-2024001839-A1_106	.	CCc1c(F)ccc2cc(O)cc(-c3ccc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(OCC(O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8scnc8C)cc7)C(C)(C)C)CC6)CC5)nc4c3F)c12	C61H75F2N9O7S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-47ECVV	WO-2024001839-A1_107	(2S,4R)-1-[(2S)-2-[[2-[1-[[1-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]oxyacetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1R)-2-hydroxy-1-naphthalen-2-ylethyl]pyrrolidine-2-carboxamide	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(OCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](CO)c7ccc8ccccc8c7)C(C)(C)C)CC6)CC5)nc4c3F)c12	C60H67F2N9O8	KRAS	P01116	VHL	WO-2024001839-A1
TPD-8LG976	WO-2024001839-A1_108	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(OCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)NCc7ccc8cc(Cl)ccc8c7)C(C)(C)C)CC6)CC5)nc4c3F)c12	C59H64ClF2N9O7	KRAS	P01116	VHL	WO-2024001839-A1
TPD-ZLQKC7	WO-2024001839-A1_109	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCCCCN5CCC[C@H](OCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](CO)c6ccc(-c7ccccc7F)cc6)C(C)(C)C)C5)nc4c3F)c12	C61H72F3N9O8	KRAS	P01116	VHL	WO-2024001839-A1
TPD-3CPBB6	WO-2024001839-A1_110	(2S,4R)-1-[(2S)-2-[[2-[(3S)-1-[[1-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-3-yl]oxyacetyl]amino]-3,3-dimethylbutanoyl]-N-[(1R)-1-[4-(2-fluorophenyl)phenyl]-2-hydroxyethyl]-4-hydroxypyrrolidine-2-carboxamide	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC[C@H](OCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](CO)c7ccc(-c8ccccc8F)cc7)C(C)(C)C)C6)CC5)nc4c3F)c12	C62H68F3N9O8	KRAS	P01116	VHL	WO-2024001839-A1
TPD-RP2H1I	WO-2024001839-A1_111	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC[C@H](OCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)NCc7ccc8cc(Cl)ccc8c7)C(C)(C)C)C6)CC5)nc4c3F)c12	C59H68ClF2N9O7	KRAS	P01116	VHL	WO-2024001839-A1
TPD-MZPL4A	WO-2024001839-A1_112	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC[C@H](OCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)NCc7ccc8c(Cl)cccc8c7)C(C)(C)C)C6)CC5)nc4c3F)c12	C59H68ClF2N9O7	KRAS	P01116	VHL	WO-2024001839-A1
TPD-09TFGU	WO-2024001839-A1_113	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC[C@H](OCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc8ccccc8c7)C(C)(C)C)C6)CC5)nc4c3F)c12	C60H71F2N9O7	KRAS	P01116	VHL	WO-2024001839-A1
TPD-PG8SE9	WO-2024001839-A1_114	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC[C@H](OCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc8cc(Cl)ccc8c7)C(C)(C)C)C6)CC5)nc4c3F)c12	C60H70ClF2N9O7	KRAS	P01116	VHL	WO-2024001839-A1
TPD-HCV9TW	WO-2024001839-A1_115	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC[C@H](OCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc8c(Cl)cccc8c7)C(C)(C)C)C6)CC5)nc4c3F)c12	C60H70ClF2N9O7	KRAS	P01116	VHL	WO-2024001839-A1
TPD-8EUGVE	WO-2024001839-A1_117	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC[C@H](OCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)NCc7ccc8cc(Cl)ccc8c7)C(C)(C)C)C6)CC5)nc4c3F)c12	C59H64ClF2N9O7	KRAS	P01116	VHL	WO-2024001839-A1
TPD-JWA8MD	WO-2024001839-A1_118	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC[C@H](OCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)NCc7ccc8c(Cl)cccc8c7)C(C)(C)C)C6)CC5)nc4c3F)c12	C59H64ClF2N9O7	KRAS	P01116	VHL	WO-2024001839-A1
TPD-L1UYZO	WO-2024001839-A1_119	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC[C@H](OCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc8ccccc8c7)C(C)(C)C)C6)CC5)nc4c3F)c12	C60H67F2N9O7	KRAS	P01116	VHL	WO-2024001839-A1
TPD-0G74F1	WO-2024001839-A1_120	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC[C@H](OCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc8cc(Cl)ccc8c7)C(C)(C)C)C6)CC5)nc4c3F)c12	C60H66ClF2N9O7	KRAS	P01116	VHL	WO-2024001839-A1
TPD-1WG4K9	WO-2024001839-A1_121	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC[C@H](OCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc8c(Cl)cccc8c7)C(C)(C)C)C6)CC5)nc4c3F)c12	C60H66ClF2N9O7	KRAS	P01116	VHL	WO-2024001839-A1
TPD-I88F66	WO-2024001839-A1_122	(2S)-4-[[1-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-N-[(2S)-1-[(2S,4R)-2-[[(1S)-1-[4-(2-fluorophenyl)phenyl]ethyl]carbamoyl]-4-hydroxypyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]morpholine-2-carboxamide	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCO[C@H](C(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8ccccc8F)cc7)C(C)(C)C)C6)CC5)nc4c3F)c12	C60H68F3N9O7	KRAS	P01116	VHL	WO-2024001839-A1
TPD-MN9NDT	WO-2024001839-A1_123	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCOC(C(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8ccccc8F)cc7)C(C)(C)C)C6)CC5)nc4c3F)c12	C60H68F3N9O7	KRAS	P01116	VHL	WO-2024001839-A1
TPD-W3WCXZ	WO-2024001839-A1_124	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCO[C@@H](CC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8ccccc8F)cc7)C(C)(C)C)C6)CC5)nc4c3F)c12	C61H70F3N9O7	KRAS	P01116	VHL	WO-2024001839-A1
TPD-GMDH68	WO-2024001839-A1_125	(2S,4R)-1-[(2S)-2-[[2-[(2R)-4-[[1-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]morpholin-2-yl]acetyl]amino]-3,3-dimethylbutanoyl]-N-[(1S)-1-[4-(2-fluorophenyl)phenyl]ethyl]-4-hydroxypyrrolidine-2-carboxamide	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCO[C@H](CC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8ccccc8F)cc7)C(C)(C)C)C6)CC5)nc4c3F)c12	C61H70F3N9O7	KRAS	P01116	VHL	WO-2024001839-A1
TPD-M2M31O	WO-2024001839-A1_126	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCOC(CCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8ccccc8F)cc7)C(C)(C)C)C6)CC5)nc4c3F)c12	C62H72F3N9O7	KRAS	P01116	VHL	WO-2024001839-A1
TPD-BM2KAE	WO-2024001839-A1_127	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCCCC6C(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)c6ccc(-c7ccccc7F)cc6)C(C)(C)C)CC5)nc4c3F)c12	C61H70F3N9O6	KRAS	P01116	VHL	WO-2024001839-A1
TPD-Y9DIM7	WO-2024001839-A1_128	(2R)-1-[[1-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-N-[(2S)-1-[(2S,4R)-2-[[(1S)-1-[4-(2-fluorophenyl)phenyl]ethyl]carbamoyl]-4-hydroxypyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]piperidine-2-carboxamide	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCCC[C@@H]6C(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)c6ccc(-c7ccccc7F)cc6)C(C)(C)C)CC5)nc4c3F)c12	C61H70F3N9O6	KRAS	P01116	VHL	WO-2024001839-A1
TPD-3MSZF4	WO-2024001839-A1_129	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCCC[C@H]6CC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)c6ccc(-c7ccccc7F)cc6)C(C)(C)C)CC5)nc4c3F)c12	C62H72F3N9O6	KRAS	P01116	VHL	WO-2024001839-A1
TPD-OMME0H	WO-2024001839-A1_130	(2S,4R)-1-[(2S)-2-[[2-[(2R)-1-[[1-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-2-yl]acetyl]amino]-3,3-dimethylbutanoyl]-N-[(1S)-1-[4-(2-fluorophenyl)phenyl]ethyl]-4-hydroxypyrrolidine-2-carboxamide	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCCC[C@@H]6CC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)c6ccc(-c7ccccc7F)cc6)C(C)(C)C)CC5)nc4c3F)c12	C62H72F3N9O6	KRAS	P01116	VHL	WO-2024001839-A1
TPD-AMCTMA	WO-2024001839-A1_131	(3R)-1-[[1-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-N-[(2S)-1-[(2S,4R)-2-[[(1S)-1-[4-(2-fluorophenyl)phenyl]ethyl]carbamoyl]-4-hydroxypyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]piperidine-3-carboxamide	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC[C@@H](C(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8ccccc8F)cc7)C(C)(C)C)C6)CC5)nc4c3F)c12	C61H70F3N9O6	KRAS	P01116	VHL	WO-2024001839-A1
TPD-9VC144	WO-2024001839-A1_132	(3S)-1-[[1-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-N-[(2S)-1-[(2S,4R)-2-[[(1S)-1-[4-(2-fluorophenyl)phenyl]ethyl]carbamoyl]-4-hydroxypyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]piperidine-3-carboxamide	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC[C@H](C(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8ccccc8F)cc7)C(C)(C)C)C6)CC5)nc4c3F)c12	C61H70F3N9O6	KRAS	P01116	VHL	WO-2024001839-A1
TPD-R97I9L	WO-2024001839-A1_133	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC[C@@H](CC(=O)N[C@H](C(=O)N7CC(=O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8ccccc8F)cc7)C(C)(C)C)C6)CC5)nc4c3F)c12	C62H70F3N9O6	KRAS	P01116	VHL	WO-2024001839-A1
TPD-QPAAUV	WO-2024001839-A1_134	(2S,4R)-1-[(2S)-2-[[2-[(3R)-1-[[1-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-3-yl]acetyl]amino]-3,3-dimethylbutanoyl]-N-[(1S)-1-[4-(2-fluorophenyl)phenyl]ethyl]-4-hydroxypyrrolidine-2-carboxamide	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC[C@H](CC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8ccccc8F)cc7)C(C)(C)C)C6)CC5)nc4c3F)c12	C62H72F3N9O6	KRAS	P01116	VHL	WO-2024001839-A1
TPD-P4W981	WO-2024001839-A1_135	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCCC(CCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8ccccc8F)cc7)C(C)(C)C)C6)CC5)nc4c3F)c12	C63H74F3N9O6	KRAS	P01116	VHL	WO-2024001839-A1
TPD-5J73GR	WO-2024001839-A1_136	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(OCc7cn([C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)nn7)CC6)CC5)nc4c3F)c12	C61H68F2N12O6S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-HGWD41	WO-2024001839-A1_137	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(Cc7cn([C@H](C(=O)N8C[C@H](O)C[C@H]8C(O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)nn7)CC6)CC5)nc4c3F)c12	C61H70F2N12O5S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-CZ4GCR	WO-2024001839-A1_138	(2S,4R)-1-[(2S)-2-[6-[1-[[1-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]oxy-3-oxo-1H-isoindol-2-yl]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(Oc7ccc8c(c7)CN([C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c9scnc9C)cc7)C(C)(C)C)C8=O)CC6)CC5)nc4c3F)c12	C66H74F2N10O7S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-5GTCR8	WO-2024001839-A1_139	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCN(c7ccc8c(c7)CN([C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c9scnc9C)cc7)C(C)(C)C)C8=O)CC6)CC5)nc4c3C)c12	C66H76FN11O6S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-LAAP24	WO-2024001839-A1_140	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCN(c7ccc8c(c7)C(=O)N([C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c9scnc9C)cc7)C(C)(C)C)C8)CC6)CC5)nc4c3F)c12	C65H73F2N11O6S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-E592Q7	WO-2024001839-A1_141	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(Oc7ccc8c(c7)C(=O)N([C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c9scnc9C)cc7)C(C)(C)C)C8)CC6)CC5)nc4c3F)c12	C66H74F2N10O7S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-XHJYWF	WO-2024001839-A1_142	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(Oc7cccc8c7CN([C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c9scnc9C)cc7)C(C)(C)C)C8=O)CC6)CC5)nc4c3F)c12	C66H74F2N10O7S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-8O3RJT	WO-2024001839-A1_143	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC7(CC6)CC(Oc6cccc8c6CN([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)c6ccc(-c9scnc9C)cc6)C(C)(C)C)C8=O)C7)CC5)nc4c3F)c12	C69H78F2N10O7S	KRAS	P01116	VHL	WO-2024001839-A1
TPD-8B0Z6V	WO-2024001839-A1_144	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC7(CCC(CCC(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](CO)c8ccc(-c9ccccc9Cl)cc8)C(C)(C)C)CC7)CC6)CC5)nc4c3F)c12	C68H82ClF2N9O7	KRAS	P01116	VHL	WO-2024001839-A1
TPD-DBC1UG	WO-2024001839-A1_145	(2S,4R)-N-[(1R)-1-[4-(2-chlorophenyl)phenyl]-2-hydroxyethyl]-1-[(2S)-2-[[2-[[7-[[1-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]oxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC7(CC6)CC(OCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](CO)c6ccc(-c8ccccc8Cl)cc6)C(C)(C)C)C7)CC5)nc4c3F)c12	C65H76ClF2N9O8	KRAS	P01116	VHL	WO-2024001839-A1
TPD-G79ECX	WO-2024001839-A1_146	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC[C@H](OCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](CO)c7ccc(-c8ccccc8Cl)cc7)C(C)(C)C)C6)CC5)nc4c3F)c12	C62H72ClF2N9O8	KRAS	P01116	VHL	WO-2024001839-A1
TPD-3NI8G2	WO-2024001839-A1_147	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC[C@H](OCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](CO)c7ccc(-c8ccccc8Cl)cc7)C(C)(C)C)C6)CC5)nc4c3F)c12	C62H68ClF2N9O8	KRAS	P01116	VHL	WO-2024001839-A1
TPD-R4AZYH	WO-2024001839-A1_148	(2S,4R)-N-[(1R)-1-[4-(2-chlorophenyl)phenyl]-2-hydroxyethyl]-1-[(2S)-2-[[2-[[3-[[1-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-3-azaspiro[5.5]undecan-9-yl]oxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC7(CCC(OCC(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](CO)c8ccc(-c9ccccc9Cl)cc8)C(C)(C)C)CC7)CC6)CC5)nc4c3F)c12	C67H80ClF2N9O8	KRAS	P01116	VHL	WO-2024001839-A1
TPD-0PTLM8	WO-2024001839-A1_149	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC7(CCC(OCC(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)NC(CO)c8ccc(-c9ccccc9Cl)cc8)C(C)(C)C)CC7)CC6)CC5)nc4c3F)c12	C67H76ClF2N9O8	KRAS	P01116	VHL	WO-2024001839-A1
TPD-ISZ69Z	WO-2024001839-A1_150	(2S,4R)-N-[(1R)-1-[4-(2-chlorophenyl)phenyl]-2-hydroxyethyl]-1-[(2S)-2-[[2-[[2-[[1-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-2-azaspiro[3.5]nonan-7-yl]oxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CC7(CCC(OCC(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](CO)c8ccc(-c9ccccc9Cl)cc8)C(C)(C)C)CC7)C6)CC5)nc4c3F)c12	C65H76ClF2N9O8	KRAS	P01116	VHL	WO-2024001839-A1
TPD-TNQRDR	WO-2024001839-A1_151	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCCCCCN5CC6(CCC(OCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](CO)c7ccc(-c8ccccc8Cl)cc7)C(C)(C)C)CC6)C5)nc4c3F)c12	C65H74ClF2N9O8	KRAS	P01116	VHL	WO-2024001839-A1
TPD-KE7JLU	WO-2024001839-A1_152	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC7(CCC(CCC(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9ccccc9F)cc8)C(C)(C)C)CC7)CC6)CC5)nc4c3F)c12	C68H82F3N9O6	KRAS	P01116	VHL	WO-2024001839-A1
TPD-I8JDKB	WO-2024001839-A1_153	(2S,4R)-1-[(2S)-2-[3-[3-[[1-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-3-azaspiro[5.5]undecan-9-yl]propanoylamino]-3,3-dimethylbutanoyl]-N-[(1S)-1-[4-(2-fluorophenyl)phenyl]ethyl]-4-hydroxypyrrolidine-2-carboxamide	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC7(CCC(CCC(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9ccccc9F)cc8)C(C)(C)C)CC7)CC6)CC5)nc4c3F)c12	C68H78F3N9O6	KRAS	P01116	VHL	WO-2024001839-A1
TPD-3UU0GC	WO-2024001839-A1_154	(2S,4R)-1-[(2S)-2-[7-[(3S)-1-[[1-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-3-yl]oxy-3-oxo-1H-isoindol-2-yl]-3,3-dimethylbutanoyl]-N-[(1S)-1-[4-(2-fluorophenyl)phenyl]ethyl]-4-hydroxypyrrolidine-2-carboxamide	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC[C@H](Oc7cccc8c7CN([C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c9ccccc9F)cc7)C(C)(C)C)C8=O)C6)CC5)nc4c3F)c12	C68H74F3N9O7	KRAS	P01116	VHL	WO-2024001839-A1
TPD-JQKNX6	WO-2024001839-A1_155	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC[C@@H](Oc7cccc8c7CN([C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c9ccccc9F)cc7)C(C)(C)C)C8=O)C6)CC5)nc4c3F)c12	C68H74F3N9O7	KRAS	P01116	VHL	WO-2024001839-A1
TPD-IJM88A	WO-2024001839-A1_156	(2S,4R)-1-[(2S)-2-[7-[[1-[[1-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]methoxy]-3-oxo-1H-isoindol-2-yl]-3,3-dimethylbutanoyl]-N-[(1S)-1-[4-(2-fluorophenyl)phenyl]ethyl]-4-hydroxypyrrolidine-2-carboxamide	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(COc7cccc8c7CN([C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c9ccccc9F)cc7)C(C)(C)C)C8=O)CC6)CC5)nc4c3F)c12	C69H76F3N9O7	KRAS	P01116	VHL	WO-2024001839-A1
TPD-1PFKQR	WO-2024001839-A1_157	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CC6CCC(Oc7cccc8c7CN([C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c9ccccc9F)cc7)C(C)(C)C)C8=O)CC6)CC5)nc4c3F)c12	C69H75F3N8O7	KRAS	P01116	VHL	WO-2024001839-A1
TPD-3V6SD2	WO-2024001839-A1_158	(2S,4R)-1-[(2S)-2-[7-[4-[[1-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]-3,3-dimethylbutanoyl]-N-[(1S)-1-[4-(2-fluorophenyl)phenyl]ethyl]-4-hydroxypyrrolidine-2-carboxamide	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCN(c7cccc8c7CN([C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c9ccccc9F)cc7)C(C)(C)C)C8=O)CC6)CC5)nc4c3F)c12	C67H73F3N10O6	KRAS	P01116	VHL	WO-2024001839-A1
TPD-57F7LD	WO-2024001839-A1_159	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC56CC5C6N5CCC6(CCC(OCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8ccccc8F)cc7)C(C)(C)C)CC6)CC5)nc4c3F)c12	C67H78F3N9O7	KRAS	P01116	VHL	WO-2024001839-A1
TPD-LICLFU	WO-2024001839-A1_160	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC7(CCC(CC(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9ccccc9F)cc8)C(C)(C)C)CC7)CC6)CC5)nc4c3F)c12	C67H80F3N9O6	KRAS	P01116	VHL	WO-2024001839-A1
TPD-CPFG7O	WO-2024001839-A1_161	(2S,4R)-1-[(2S)-2-[[2-[[2-[[1-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-2-azaspiro[3.5]nonan-7-yl]oxy]acetyl]amino]-3,3-dimethylbutanoyl]-N-[(1S)-1-[4-(2-fluorophenyl)phenyl]ethyl]-4-hydroxypyrrolidine-2-carboxamide	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CC7(CCC(OCC(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9ccccc9F)cc8)C(C)(C)C)CC7)C6)CC5)nc4c3F)c12	C65H76F3N9O7	KRAS	P01116	VHL	WO-2024001839-A1
TPD-XWFYV8	WO-2024001839-A1_162	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCO[C@H](COCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8ccccc8F)cc7)C(C)(C)C)C6)CC5)nc4c3F)c12	C62H72F3N9O8	KRAS	P01116	VHL	WO-2024001839-A1
TPD-CFC7OY	WO-2024001839-A1_163	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(c7cn([C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9ccccc9F)cc8)C(C)(C)C)nn7)CC6)CC5)nc4c3F)c12	C62H70F3N11O5	KRAS	P01116	VHL	WO-2024001839-A1
TPD-Z0W5ZG	WO-2024001839-A1_164	(2S,4R)-1-[(2S)-2-[[2-[1-[[1-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]oxyacetyl]amino]-3,3-dimethylbutanoyl]-N-[(1S)-1-[4-(2,6-difluorophenyl)phenyl]ethyl]-4-hydroxypyrrolidine-2-carboxamide	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(OCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8c(F)cccc8F)cc7)C(C)(C)C)CC6)CC5)nc4c3F)c12	C62H71F4N9O7	KRAS	P01116	VHL	WO-2024001839-A1
TPD-MK36YV	WO-2024001839-A1_165	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(OCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8ccccc8F)cc7)C(C)(C)C)CC6)CCC5)nc4c3F)c12	C63H74F3N9O7	KRAS	P01116	VHL	WO-2024001839-A1
TPD-722B99	WO-2024012570-A1_1	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cnn(-c6cnn(-c7c(Cl)cc(C(F)(F)F)cc7Cl)c6)c5)C4)cc3C2=O)C(=O)N1	C31H20Cl2F3N7O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-1NGDHQ	WO-2024012570-A1_10	.	N#Cc1ccc(-n2cc(-n3cc(C#CC4CN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)cn3)cn2)c(C2CC2)c1	C34H26N8O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-RP7Y7Q	WO-2024012570-A1_11	.	CC#Cc1cc(C(F)(F)F)ccc1-n1cc(-n2cc(C#CC3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)cn2)cn1	C34H24F3N7O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-F7MLC1	WO-2024012570-A1_12	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cnn(-c6cnn(Cc7ccc(C(F)(F)F)cc7Cl)c6)c5)C4)cc3C2=O)C(=O)N1	C32H23ClF3N7O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-JSU327	WO-2024012570-A1_13	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cnn(-c6cn(-c7c(Cl)cc(C(F)(F)F)cc7Cl)cn6)c5)C4)cc3C2=O)C(=O)N1	C31H20Cl2F3N7O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-S5MXL0	WO-2024012570-A1_14	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cnn(C6CCC(c7ccc(C(F)(F)F)cc7Cl)C6)c5)C4)cc3C2=O)C(=O)N1	C33H27ClF3N5O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-ZL6HOO	WO-2024012570-A1_15	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cnn(C6CCN(c7ccc(C(F)(F)F)cc7Cl)C6)c5)C4)cc3C2=O)C(=O)N1	C32H26ClF3N6O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-35BTGQ	WO-2024012570-A1_16	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cnn(C6CCN(c7ccc(C(F)(F)F)cc7Cl)C6=O)c5)C4)cc3C2=O)C(=O)N1	C32H24ClF3N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-DNBJJ4	WO-2024012570-A1_17	.	N#Cc1ccc(-n2cc(-n3cc(C#CC4CN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)cn3)cn2)c2ccccc12	C35H24N8O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-FYKCKA	WO-2024012570-A1_18	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cnn(-c6cnn(-c7ccc(C(F)(F)F)cc7C7CC7)c6)c5)C4)cc3C2=O)C(=O)N1	C34H26F3N7O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-FEVNKL	WO-2024012570-A1_19	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cnn(C6CCN(c7ccc(C(F)(F)F)cc7Cl)CC6)c5)C4)cc3C2=O)C(=O)N1	C33H28ClF3N6O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-39UV8T	WO-2024012570-A1_2	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5csc(N6CCN(c7ccc(C(F)(F)F)cc7Cl)C6=O)n5)C4)cc3C2=O)C(=O)N1	C31H22ClF3N6O5S	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-9XWN82	WO-2024012570-A1_20	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cnn(C6CCN(Cc7ccc(C(F)(F)F)cc7Cl)C6)c5)C4)cc3C2=O)C(=O)N1	C33H28ClF3N6O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-VA0XD7	WO-2024012570-A1_21	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cnn(C6CCN(Cc7ccc(C(F)(F)F)cc7Cl)CC6)c5)C4)cc3C2=O)C(=O)N1	C34H30ClF3N6O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-AIPCNJ	WO-2024012570-A1_22	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cnn(-c6cnn(-c7ccc(C(F)(F)F)cc7Cl)c6)c5)C4)cc3C2=O)C(=O)N1	C31H21ClF3N7O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-Q3UMON	WO-2024012570-A1_23	.	CC1(C)C(=O)N(c2ccc(C(F)(F)F)cc2Cl)c2ccc(-n3cc(C#CC4CN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)cn3)cc21	C38H28ClF3N6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-Q0KTJM	WO-2024012570-A1_24	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cnn(Cc6cnn(Cc7ccc(C(F)(F)F)cc7Cl)c6)c5)C4)cc3C2=O)C(=O)N1	C33H25ClF3N7O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-S97DT1	WO-2024012570-A1_25	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cnn(-c6ccc7[nH]c8ccc(C(F)(F)F)cc8c7c6)c5)C4)cc3C2=O)C(=O)N1	C34H23F3N6O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-1EBXSK	WO-2024012570-A1_26	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cnn(CC6CN(c7ccc(C(F)(F)F)cc7Cl)C6)c5)C4)cc3C2=O)C(O)N1	C32H28ClF3N6O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-5PUN72	WO-2024012570-A1_27	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cnn(C6CN(c7ccc(C(F)(F)F)cc7Cl)C6)c5)C4)cc3C2=O)C(=O)N1	C31H24ClF3N6O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-4JPQC2	WO-2024012570-A1_29	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cnn(C6(CNc7ccc(C(F)(F)F)cc7Cl)CCC6)c5)C4)cc3C2=O)C(=O)N1	C33H28ClF3N6O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-51K260	WO-2024012570-A1_3	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cnn(C6(c7nc8cc(C(F)(F)F)ccc8[nH]7)CCC6)c5)C4)cc3C2=O)C(=O)N1	C33H26F3N7O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-7N81FJ	WO-2024012570-A1_30	.	CC1(C)C(=O)N(c2ccc(C#N)cc2Cl)c2ccc(-n3cc(C#CC4CN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)cn3)cc21	C38H28ClN7O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-DRD3TA	WO-2024012570-A1_31	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cnn(Cc6cnn(-c7c(Cl)cc(C(F)(F)F)cc7Cl)c6)c5)C4)cc3C2=O)C(=O)N1	C32H22Cl2F3N7O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-KPWGG7	WO-2024012570-A1_32	.	CC1(C)C(=O)N(c2ccc(C#N)c(Cl)c2)c2ccc(-n3cc(C#CC4CN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)cn3)cc21	C38H28ClN7O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-LKWEIC	WO-2024012570-A1_33	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5ccc(-c6cnn(-c7ccc(C(F)(F)F)cc7Cl)c6)cc5)C4)cc3C2=O)C(=O)N1	C34H23ClF3N5O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-11YE33	WO-2024012570-A1_34	.	Cc1c(C#N)c(-c2ccc(C#N)cc2)c(C)n1Cc1ccc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cc1	C39H30N6O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-LE1Q11	WO-2024012570-A1_35	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cnn(C6CN(Cc7ccc(C(F)(F)F)cc7Cl)C6)c5)C4)cc3C2=O)C(=O)N1	C32H26ClF3N6O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-G6VYLS	WO-2024012570-A1_36-A	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cnn([C@H]6C[C@@H](CNc7ccc(C(F)(F)F)cc7Cl)C6)c5)C4)cc3C2=O)C(=O)N1	C33H28ClF3N6O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-51CQP2	WO-2024012570-A1_36-B	.	Cc1cc(C(F)(F)F)ccc1NC[C@H]1C[C@H](n2cc(C#CC3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)cn2)C1	C34H31F3N6O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-2YAMGE	WO-2024012570-A1_38	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cnn(C6CCC6CNc6ccc(C(F)(F)F)cc6Cl)c5)C4)cc3C2=O)C(=O)N1	C33H28ClF3N6O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-IO8NVU	WO-2024012570-A1_39	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cccc(-c6cnn(-c7ccc(C(F)(F)F)cc7Cl)c6)c5)C4)cc3C2=O)C(=O)N1	C34H23ClF3N5O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-JKI9HE	WO-2024012570-A1_40-A	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cnn([C@H]6CC[C@@H](Oc7ccc(C(F)(F)F)cc7Cl)CC6)c5)C4)cc3C2=O)C(=O)N1	C34H29ClF3N5O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-JBLN0X	WO-2024012570-A1_40-B	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cnn([C@H]6CC[C@H](Oc7ccc(C(F)(F)F)cc7Cl)CC6)c5)C4)cc3C2=O)C(=O)N1	C34H29ClF3N5O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-TXN89L	WO-2024012570-A1_41	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5nn(-c6cnn(-c7ccc(C(F)(F)F)cc7Cl)c6)c6ccccc56)C4)cc3C2=O)C(=O)N1	C35H23ClF3N7O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-OXNHBT	WO-2024012570-A1_42	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cccc(-c6nc7cc(C(F)(F)F)cc(Cl)c7[nH]6)c5)C4)cc3C2=O)C(=O)N1	C32H21ClF3N5O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-7OIEO1	WO-2024012570-A1_43	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5ccc6nc(-c7ccc(C(F)(F)F)cc7Cl)[nH]c6c5)C4)cc3C2=O)C(=O)N1	C32H21ClF3N5O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-KCCVO1	WO-2024012570-A1_44	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cccc6c5cnn6-c5cnn(-c6ccc(CF)cc6Cl)c5)C4)cc3C2=O)C(=O)N1	C35H25ClFN7O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-IMXLVM	WO-2024012570-A1_45	.	CC1(C)C(=O)N(c2ccc(C#N)c(Cl)c2)c2ccc(C#CC3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)cc21	C35H26ClN5O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-V4622Y	WO-2024012570-A1_46	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cnn(C6CC7CN(c8ccc(C(F)(F)F)cc8Cl)CC7C6)c5)C4)cc3C2=O)C(=O)N1	C35H30ClF3N6O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-TZ3HRI	WO-2024012570-A1_47	.	Cc1nn(-c2cnn(-c3c(Cl)cc(C(F)(F)F)cc3Cl)c2)cc1C#CC1CN(c2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)C1	C32H22Cl2F3N7O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-LUU8YJ	WO-2024012570-A1_48	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5ccc(CN6C7CCC6CC(Oc6ccc(C(F)(F)F)cc6Cl)C7)cc5)C4)cc3C2=O)C(=O)N1	C39H34ClF3N4O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-GZKA2R	WO-2024012570-A1_49	.	O=C1CCC(N2C(=O)c3ccc(N4CC(n5ncc6cc(-c7nc8c(C9CC9)cc(C9CC9)cc8[nH]7)ccc65)C4)cc3C2=O)C(=O)N1	C36H31N7O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-BIKWG8	WO-2024012570-A1_5	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cnn(C6(Cn7ncc8cc(C(F)(F)F)ccc87)CCC6)c5)C4)cc3C2=O)C(=O)N1	C34H28F3N7O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-264VKD	WO-2024012570-A1_50	.	O=C1CCC(N2C(=O)c3ccc(N4CC(n5cc6cc(-c7nc8c(C9CC9)cc(C9CC9)cc8[nH]7)ccc6n5)C4)cc3C2=O)C(=O)N1	C36H31N7O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-JFY9K0	WO-2024012570-A1_51	.	CC(Oc1cc(F)cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)c1)c1ccc(C(F)(F)F)cc1Cl	C33H24ClF4N3O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-LXZ8BM	WO-2024012570-A1_52	.	C[C@@H](Oc1ccc(C(F)(F)F)cc1Cl)c1cc(F)ccc1C#CC1CN(c2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)C1	C33H24ClF4N3O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-EQTQCR	WO-2024012570-A1_53	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cc(F)cc(Oc6ccc(C(F)(F)F)cc6Cl)c5)C4)cc3C2=O)C(=O)N1	C31H20ClF4N3O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-LC5Q8H	WO-2024012570-A1_54	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cnn(C6(c7ncc(-c8ccc(C(F)(F)F)cc8Cl)[nH]7)CCC6)c5)C4)cc3C2=O)C(=O)N1	C35H27ClF3N7O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-8WWJRZ	WO-2024012570-A1_55	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cc(F)cc(-c6ccc(C(F)(F)F)cc6Cl)c5)C4)cc3C2=O)C(=O)N1	C31H20ClF4N3O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-MKP1A7	WO-2024012570-A1_56	.	Cc1c(C#N)c(-c2ccc(C#N)cc2)c(C)n1Cc1ccc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cc1F	C39H29FN6O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-2259C2	WO-2024012570-A1_57	.	Cc1c(C#N)c(-c2ccc(C#N)cc2)c(C)n1Cc1ccc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)c(F)c1	C39H29FN6O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-AL2MLQ	WO-2024012570-A1_58	.	CC(C)(c1ccc(-c2ccc(C(F)(F)F)cc2Cl)cc1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C37H29ClF3N5O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-OLPGVZ	WO-2024012570-A1_59	.	CC(c1ccc(-c2ccc(C(F)(F)F)cc2Cl)c(F)c1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C36H26ClF4N5O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-6EP0MG	WO-2024012570-A1_6	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cnn(-c6csc(-c7ccc(C(F)(F)F)cc7Cl)n6)c5)C4)cc3C2=O)C(=O)N1	C31H20ClF3N6O4S	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-HFHITL	WO-2024012570-A1_60	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cnn(Cc6ccc(-c7ccc(C(F)(F)F)cc7Cl)c(F)c6)c5)C4)cc3C2=O)C(=O)N1	C35H24ClF4N5O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-JRK5TN	WO-2024012570-A1_61	.	CC(C)(c1ccc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cc1)c1ccc(-c2ccc(C(F)(F)F)cc2Cl)cc1	C40H31ClF3N3O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-388BM1	WO-2024012570-A1_62	.	Cc1c(C#N)c(-c2ccc(C#N)cc2)c(C)n1Cc1ccc(-c2ccc(C3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)c(F)c2)cc1F	C43H32F2N6O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-BUU6W7	WO-2024012570-A1_7	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cnn(-c6csc(N7CCOCC7)n6)c5)C4)cc3C2=O)C(=O)N1	C28H25N7O5S	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-L8W9UK	WO-2024012570-A1_8	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cnn(-c6ccc(-c7ccc(C(F)(F)F)cc7Cl)cc6)c5)C4)cc3C2=O)C(=O)N1	C34H23ClF3N5O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-T83PYS	WO-2024012570-A1_9	.	O=C1CCC(N2C(=O)c3ccc(N4CC(C#Cc5cnn(-c6cccc(-c7ccc(C(F)(F)F)cc7Cl)c6)c5)C4)cc3C2=O)C(=O)N1	C34H23ClF3N5O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2024012570-A1
TPD-3K93R9	WO-2024148257-A1_YX-02-030	.	CCOc1cc(C(C)(C)C)ccc1C1=N[C@](C)(c2ccc(Cl)cc2)[C@](C)(c2ccc(Cl)cc2)N1C(=O)N1CCN(CC(=O)NCCOCCOCCOCC(=O)N[C@@H](C)C(=O)N2C[C@H](O)C[C@H]2C(=O)NCc2ccc(-c3scnc3C)cc2)CC1	C63H79Cl2N9O10S	MDM2	Q00987	VHL	WO-2024148257-A1
TPD-RAYZQW	WO-2024148257-A1_YX-02-041	.	CCOc1cc(C(C)(C)C)ccc1C1=N[C@@](C)(c2ccc(Cl)cc2)[C@@](C)(c2ccc(Cl)cc2)N1C(=O)N1CCN(CC(=O)NCCCCNC(=O)COc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)CC1	C55H62Cl2N8O9	MDM2	Q00987	CRBN	WO-2024148257-A1
TPD-4DHA9K	WO-2024148257-A1_YX-02-052	.	CCOc1cc(C(C)(C)C)ccc1C1=N[C@@](C)(c2ccc(Cl)cc2)[C@@](C)(c2ccc(Cl)cc2)N1C(=O)N1CCN(CC(=O)NCCOCCOCCNC(=O)CN2CCN(C(=O)N3C(c4ccc(C(C)(C)C)cc4OCC)=N[C@](C)(c4ccc(Cl)cc4)[C@]3(C)c3ccc(Cl)cc3)CC2)CC1	C78H96Cl4N10O8	MDM2	Q00987	MDM2	WO-2024148257-A1
TPD-KHPDIH	WO-2024148257-A1_YX-02-062	.	CCOc1cc(C(C)(C)C)ccc1C1=N[C@@](C)(c2ccc(Cl)cc2)[C@@](C)(c2ccc(Cl)cc2)N1C(=O)N1CCN(CC(=O)NCCOCCOCCOCNC(=O)CN2CCN(C(=O)N3C(c4ccc(C(C)(C)C)cc4OCC)=N[C@](C)(c4ccc(Cl)cc4)[C@]3(C)c3ccc(CI)cc3)CC2)CC1	C80H100Cl3IN10O9	MDM2	Q00987	MDM2	WO-2024148257-A1
TPD-0ESXC2	WO-2024148257-A1_YX-02-228	.	CCOc1cc(C(C)(C)C)ccc1C1=N[C@](C)(c2ccc(Cl)cc2)[C@](C)(c2ccc(Cl)cc2)N1C(=O)N1CCN(CC(=O)NCCCNC(=O)COc2ccc3c(c2)CN(C(=O)[C@H](NC(=O)[C@@H](C)NC)C(C)(C)C)[C@@H](C(=O)N[C@H]2CCCc4ccccc42)C3)CC1	C71H90Cl2N10O8	MDM2	Q00987	VHL	WO-2024148257-A1
TPD-RD5S96	WO-2024148257-A1_YX-02-230	.	CCOc1cc(C(C)C)ccc1C1=N[C@](C)(c2ccc(Cl)cc2)[C@](C)(c2ccc(Cl)cc2)N1C(=O)N1CCN(CC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCc2ccc(-c3scnc3C)cc2)C(C)(C)C)CC1	C57H68Cl2N8O6S	MDM2	Q00987	VHL	WO-2024148257-A1
TPD-IJ24YV	orb2802390	2-[7-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]heptylamino]-N-[6-(dimethylamino)pyridazin-3-yl]-6-(methylamino)pyridine-3-carboxamide; 3055471-57-0	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)n1	C46H61N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-XK8102	WO-2024183798-A1_CPD--100	.	CNc1ccc(C(=O)Nc2cc[nH]n2)c(NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C43H52N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-3OUB3X	WO-2024183798-A1_CPD--101	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC(CC(=O)NCCN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)C2)n1	C45H57N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-IE9XOX	WO-2024183798-A1_CPD--102	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCC2CN(C(=O)CN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)C2)n1	C45H57N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-EOMHF1	WO-2024183798-A1_CPD--103	.	CNc1ccc(C(=O)Nc2cccc(C3CC3)n2)c(NC2CC3(C2)CN(C(=O)CCN2CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC2)C3)n1	C48H57N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-E21Y9G	WO-2024183798-A1_CPD--104	.	CNc1ccc(C(=O)Nc2ccc(N)nn2)c(NCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)n1	C42H53N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-EWJBIO	WO-2024183798-A1_CPD--105	.	CNc1ccc(C(=O)Nc2ccc(C)nn2)c(NCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)n1	C43H54N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-5BP1BJ	WO-2024183798-A1_CPD--106	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CCN(CCNC(=O)CN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)C2)n1	C45H58N16O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-XVU1BG	WO-2024183798-A1_CPD--107	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CN(CCNC(=O)CN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)C2)n1	C44H56N16O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-Q20QAW	WO-2024183798-A1_CPD--108	.	CNc1ccc(C(=O)Nc2ccc(OC)nn2)c(NCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)n1	C43H54N14O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-3SZY6K	WO-2024183798-A1_CPD--109	.	CNc1ccc(C(=O)Nc2ccc(C)c(C)n2)c(NCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)n1	C45H57N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-CA9VOP	WO-2024183798-A1_CPD--11	.	CNc1ccc(C(=O)Nc2ccc(OC)nn2)c(NCCCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)n1	C45H58N14O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-TH3BXO	WO-2024183798-A1_CPD--110	.	CNc1ccc(NC(=O)c2ccc(NC)nc2NCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)nn1	C43H55N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-M9HC1K	WO-2024183798-A1_CPD--111	.	CNc1ccc(C(=O)Nc2ccc(C)c(C(C)C)n2)c(NCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)n1	C47H61N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-0OL7SJ	WO-2024183798-A1_CPD--112	.	CNc1ccc(C(=O)Nc2ccc(Cl)c(C3CC3)n2)c(NCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)n1	C46H56ClN13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-MXFPTN	WO-2024183798-A1_CPD--113	.	CNc1ccc(C(=O)Nc2ccc(F)c(C3CC3)n2)c(NCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)n1	C46H56FN13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-KLTWGY	WO-2024183798-A1_CPD--114	.	CNc1ccc(C(=O)Nc2nc(C3CC3)ccc2F)c(NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C48H56FN13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-0IYC16	WO-2024183798-A1_CPD--115	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC3(C2)CN(C(=O)C2(CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)CC2)C3)n1	C48H59N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-3YM8GX	WO-2024183798-A1_CPD--116	.	CNc1ccc(C(=O)Nc2ccc(C)c(OC)n2)c(NCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)n1	C45H57N13O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-6LFE5I	WO-2024183798-A1_CPD--117	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC3(C2)CN(C(=O)C(C)CN2CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC2)C3)n1	C47H59N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-8LCPVG	WO-2024183798-A1_CPD--118	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC3(C2)CN(C(=O)C(C)(C)CN2CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC2)C3)n1	C48H61N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-1OIQWJ	WO-2024183798-A1_CPD--119	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NC5CC6(C5)CC(Nc5nc(C(C)C)ccc5C(=O)Nc5cccc(C7CC7)n5)C6)CC4)cn3)nc2n(C2CCCC2)c1=O	C50H60N12O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-LYIZ2I	WO-2024183798-A1_CPD--12	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCCCNC(=O)C(C)N2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)n1	C45H59N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-2WCI2S	WO-2024183798-A1_CPD--120	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NC5CC6(C5)CC(Nc5nc(C)ccc5C(=O)Nc5cccc(C7CC7)n5)C6)CC4)cn3)nc2n(C2CCCC2)c1=O	C48H56N12O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-N5XRAK	WO-2024183798-A1_CPD--121	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NC5CC6(C5)CC(Nc5nc(C(F)(F)F)ccc5C(=O)Nc5cccc(C7CC7)n5)C6)CC4)cn3)nc2n(C2CCCC2)c1=O	C48H53F3N12O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-ABUM20	WO-2024183798-A1_CPD--122	.	CNc1ccc(C(=O)Nc2cccc(=O)[nH]2)c(NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C45H53N13O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-PQHJI7	WO-2024183798-A1_CPD--123	.	CNc1ccc(C(=O)Nc2ccc(C)c(=O)[nH]2)c(NCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)n1	C44H55N13O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-ETRLRA	WO-2024183798-A1_CPD--124	.	CCc1ccc(C(=O)Nc2cccc(C3CC3)n2)c(NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C49H58N12O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-JLQIK8	WO-2024183798-A1_CPD--125	.	CNc1ccc(C(=O)Nc2ccc(OC)c(C3CC3)n2)c(NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C49H59N13O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-NEZZW3	WO-2024183798-A1_CPD--126	.	CNc1ccc(C(=O)Nc2cccc(C)n2)c(NC[C@H]2CC[C@H](NC(=O)CN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)CC2)n1	C46H57N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-T9HCKQ	WO-2024183798-A1_CPD--127	.	CNc1ccc(C(=O)Nc2cc(C(F)(F)F)n(C)n2)c(NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C45H53F3N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-NR3BZQ	WO-2024183798-A1_CPD--128	.	CNc1ccc(C(=O)Nc2ccc(F)c(C3CC3)n2)c(NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C48H56FN13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-5OI19Q	WO-2024183798-A1_CPD--129	.	CNc1ccc(C(=O)Nc2cc(C)n(C)n2)c(NC2CC3(C2)CN(C(=O)CCN2CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC2)C3)n1	C45H56N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-MXEM5P	WO-2024183798-A1_CPD--130	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CCC(NC(=O)CN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)CC2)n1	C45H57N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-TICHGO	WO-2024183798-A1_CPD--131	.	CNc1ccc(C(=O)Nc2cc(C)n(C)n2)c(NC[C@H]2CC[C@H](NC(=O)CN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)CC2)n1	C45H58N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-Y7AGNH	WO-2024183798-A1_CPD--132	.	CNc1ccc(C(=O)Nc2ccc(C#N)c(C3CC3)n2)c(NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C49H56N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-IV9DUY	WO-2024183798-A1_CPD--133	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC3(C2)CN(C(=O)N2CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC2)C3)n1	C44H53N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-8JZKAZ	WO-2024183798-A1_CPD--134	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC3(CC(NC(=O)N4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C45H55N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-OE2VYO	WO-2024183798-A1_CPD--135	.	CNc1ccc(C(=O)Nc2cn(C)c(C3CC3)n2)c(NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C47H58N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-TW5KO0	WO-2024183798-A1_CPD--136	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CCC(CCNC(=O)CN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)C2)n1	C46H59N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-KCE8P2	WO-2024183798-A1_CPD--137	.	CNc1ccc(C(=O)Nc2ccccn2)c(NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C45H53N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-7OCYSG	WO-2024183798-A1_CPD--138	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NC5CC6(C5)CC(Nc5nc(C7CC7)ccc5C(=O)Nc5cccc(C7CC7)n5)C6)CC4)cn3)nc2n(C2CCCC2)c1=O	C50H58N12O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-DLZLIN	WO-2024183798-A1_CPD--139	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NC5CC6(C5)CC(Nc5nc(NC(C)C)ccc5C(=O)Nc5cccc(C7CC7)n5)C6)CC4)cn3)nc2n(C2CCCC2)c1=O	C50H61N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-VO47X9	WO-2024183798-A1_CPD--140	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC3(C2)CC(C(=O)N2CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC2)C3)n1	C45H54N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-COMBFR	WO-2024183798-A1_CPD--141	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NC5CC6(C5)CC(Nc5nc(C#N)ccc5C(=O)Nc5cccc(C7CC7)n5)C6)CC4)cn3)nc2n(C2CCCC2)c1=O	C48H53N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-VCE72T	WO-2024183798-A1_CPD--142	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCCCCCCNc5nc(-c6ccc(C#N)nc6)ccc5C(=O)Nc5nc(C)c(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C50H58N14O4S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-LXH1GH	WO-2024183798-A1_CPD--143	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCC5CC(Nc6cc(Cl)ccc6C(=O)Nc6ccc(C)c(C7CC7)n6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C48H56ClN11O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-ZZF0EO	WO-2024183798-A1_CPD--144	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(=O)NCCC5CC(Nc6cc(Cl)ccc6C(=O)Nc6ccc(C)c(C7CC7)n6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H54ClN11O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-WF6KJF	WO-2024183798-A1_CPD--145	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCC5CC(Nc6cc(Cl)ccc6C(=O)Nc6ccc(N(C)C)nn6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H54ClN13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-4VAUQT	WO-2024183798-A1_CPD--146	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCC2CCN(C(=O)CCN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)CC2)n1	C46H59N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-CH3YUF	WO-2024183798-A1_CPD--147	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC3(CC(CC(=O)N4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C46H56N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-XL2LM5	WO-2024183798-A1_CPD--148	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC(CC(=O)N3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)C2)n1	C43H52N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-O9Y48G	WO-2024183798-A1_CPD--149	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC(NC(=O)CN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)C2)n1	C43H53N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-K5NCI9	WO-2024183798-A1_CPD--150	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC(NC(=O)CCN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)C2)n1	C44H55N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-JL3M08	WO-2024183798-A1_CPD--151	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC(NC(=O)N3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)C2)n1	C42H51N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-ATRTOD	WO-2024183798-A1_CPD--152	.	CNc1ccc(C(=O)Nc2cn(C)cn2)c(NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C44H54N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-F30VOS	WO-2024183798-A1_CPD--153	.	CNc1ccc(C(=O)Nc2ccnn2C)c(NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C44H54N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-QPIMYH	WO-2024183798-A1_CPD--154	.	CNc1ccc(C(=O)Nc2cccc(C3CC3)n2)c(NC[C@H]2CC[C@H](NC(=O)CN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)CC2)n1	C48H59N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-Z6U3P3	WO-2024183798-A1_CPD--155	.	CNc1ccc(C(=O)Nc2cccc(C)n2)c(NC2CC3(C2)CN(C(=O)CCN2CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC2)C3)n1	C46H55N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-PIGBAB	WO-2024183798-A1_CPD--156	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC(CCCC(=O)N3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)C2)n1	C45H56N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-HJ8OSW	WO-2024183798-A1_CPD--157	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC(C(=O)NCCN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)C2)n1	C44H55N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-7IS8IH	WO-2024183798-A1_CPD--158	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CCC3(C2)CN(C(=O)CCN2CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC2)C3)n1	C47H59N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-LIMGI8	WO-2024183798-A1_CPD--159	.	CNc1ccc(C(=O)Nc2ccon2)c(NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C43H51N13O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-B262BA	WO-2024183798-A1_CPD--16	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCCCCNc5nc(C)ccc5C(=O)Nc5ccc(N(C)C)nn5)CC4)cn3)nc2n(C2CCCC2)c1=O	C44H56N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-J72YW1	WO-2024183798-A1_CPD--160	.	CNc1ccc(C(=O)Nc2cc(C)on2)c(NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C44H53N13O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-QJ1CI8	WO-2024183798-A1_CPD--161	.	CNc1ccc(C(=O)Nc2cccc(OC)n2)c(NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C46H55N13O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-8S3TND	WO-2024183798-A1_CPD--162	.	CNc1ccc(C(=O)Nc2cccc(C3CC3)n2)c(NC2CC(CNC(=O)CN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)C2)n1	C46H55N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-EQRCUZ	WO-2024183798-A1_CPD--164	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC(COCC(=O)N3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)C2)n1	C44H54N14O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-P85TYV	WO-2024183798-A1_CPD--165	.	CNc1ccc(C(=O)Nc2cc(C)n(C)n2)c(NC2CC(CNC(=O)CN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)C2)n1	C43H54N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-P86NKH	WO-2024183798-A1_CPD--166	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC(CNC(=O)N3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)C2)n1	C43H53N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-GQ6HTW	WO-2024183798-A1_CPD--167	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC(CNC(=O)C(C)(C)N3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)C2)n1	C46H59N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-32JI55	WO-2024183798-A1_CPD--168	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC(OCC(=O)N3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)C2)n1	C43H52N14O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-G0WJHA	WO-2024183798-A1_CPD--169	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC[C@H]2CC[C@H](CNC(=O)N3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)CC2)n1	C46H59N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-9PKUDE	WO-2024183798-A1_CPD--17	.	CNc1ccc(C(=O)Nc2ccc(N3CCCC3)nn2)c(NCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)n1	C46H59N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-HHJYFD	WO-2024183798-A1_CPD--170	.	CNc1ccc(C(=O)Nc2cccc(C)n2)c(NC2CC(CNC(=O)CN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)C2)n1	C44H53N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-ON6VOF	WO-2024183798-A1_CPD--171	.	CNc1ccc(C(=O)Nc2cccc(C)n2)c(NC2CC3(C2)CN(C(=O)C2(CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)CC2)C3)n1	C48H57N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-EBR486	WO-2024183798-A1_CPD--172	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC(CNC(=O)C3(CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)CC3)C2)n1	C47H59N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-VTD787	WO-2024183798-A1_CPD--173	.	CNc1ccc(C(=O)Nc2cccc(C3CC3)n2)c(NC2CC3(C2)CN(C(=O)C2(CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)CC2)C3)n1	C50H59N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-BI6T95	WO-2024183798-A1_CPD--174	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC3(CC(NC(=O)C(C)(C)N4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C48H61N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-1HH5J5	WO-2024183798-A1_CPD--175	.	CNc1ccc(C(=O)Nc2cccc(C3CC3)n2)c(NC2CC3(C2)CN(C(=O)C(C)(C)N2CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC2)C3)n1	C49H59N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-5TQG8J	WO-2024183798-A1_CPD--176	.	CNc1ccc(C(=O)Nc2cccc(C)n2)c(NC2CC3(C2)CN(C(=O)C(C)(C)N2CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC2)C3)n1	C47H57N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-61Y64M	WO-2024183798-A1_CPD--177	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)c(C3CC3)n2)c(NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C50H62N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-X1I2V6	WO-2024183798-A1_CPD--178	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC(OCCC(=O)N3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)C2)n1	C44H54N14O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-YWDKJE	WO-2024183798-A1_CPD--179	.	CNc1ccc(C(=O)Nc2cn(C)c(C)n2)c(NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C45H56N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-M1RAOG	WO-2024183798-A1_CPD--18	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCCCCNc5nc(NC(C)C)ccc5C(=O)Nc5ccc(N(C)C)nn5)CC4)cn3)nc2n(C2CCCC2)c1=O	C46H61N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-17ATXA	WO-2024183798-A1_CPD--180	.	CNc1ccc(C(=O)Nc2cccc(N)n2)c(NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C45H54N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-IG3L57	WO-2024183798-A1_CPD--181	.	CNc1cccc(NC(=O)c2ccc(NC)nc2NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C46H56N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-52O8TR	WO-2024183798-A1_CPD--182	.	CNc1ccc(C(=O)Nc2ccc(C)c(C)n2)c(NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C47H57N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-J47LXM	WO-2024183798-A1_CPD--183	.	CNc1ccc(C(=O)Nc2ccn(C)c2)c(NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C45H55N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-C1XL1A	WO-2024183798-A1_CPD--184	.	CNc1ccc(C(=O)Nc2cccc(C(F)F)n2)c(NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C46H53F2N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-JVASDN	WO-2024183798-A1_CPD--185	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC(CCC(=O)N3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)C2)n1	C44H54N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-2P2Q9E	WO-2024183798-A1_CPD--186	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CN(C(=O)CCN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)C2)n1	C43H53N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-SPHQ5D	WO-2024183798-A1_CPD--187	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CN(C(=O)CN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)C2)n1	C42H51N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-KH8KDZ	WO-2024183798-A1_CPD--188	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCC2CC(CCC(=O)CN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)C2)n1	C46H58N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-FRW1OP	WO-2024183798-A1_CPD--189	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC3(C2)CC(OC(C)C(=O)N2CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC2)C3)n1	C47H58N14O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-324LAX	WO-2024183798-A1_CPD--19	.	CNc1ccc(C(=O)Nc2ccc(C(F)(F)F)nn2)c(NCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)n1	C43H51F3N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-G9U010	WO-2024183798-A1_CPD--190	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NC5CC6(C5)CC(Nc5nc(NC(C)C)ccc5C(=O)Nc5cccc(C)n5)C6)CC4)cn3)nc2n(C2CCCC2)c1=O	C48H59N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-6XO6LC	WO-2024183798-A1_CPD--191	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NC5CC6(C5)CC(Nc5nc(C)ccc5C(=O)Nc5cccc(C)n5)C6)CC4)cn3)nc2n(C2CCCC2)c1=O	C46H54N12O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-VKIBD2	WO-2024183798-A1_CPD--192	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NC5CC6(C5)CC(Nc5nc(C)ccc5C(=O)Nc5cc(C)on5)C6)CC4)cn3)nc2n(C2CCCC2)c1=O	C44H52N12O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-E2QPUP	WO-2024183798-A1_CPD--193	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC[C@H]2CC[C@@H](NC(=O)CN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)CC2)n1	C46H59N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-RYYT6N	WO-2024183798-A1_CPD--194	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)n1	C39H46N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-KSB47K	WO-2024183798-A1_CPD--195	.	CNc1ccc(C(=O)Nc2cn(C)c(C(C)C)n2)c(NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C47H60N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-1AYRQ9	WO-2024183798-A1_CPD--196	.	CNc1ccc(C(=O)Nc2cccc(C)n2)c(NC2CC(NC(=O)CN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)C2)n1	C43H51N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-HGSI98	WO-2024183798-A1_CPD--197	.	CNc1ccc(C(=O)Nc2cc(C)n(C)n2)c(NC2CC(NC(=O)CN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)C2)n1	C42H52N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-4P6BY0	WO-2024183798-A1_CPD--198	.	CNc1ccc(C(=O)Nc2cc(C)on2)c(NC2CC(NC(=O)CN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)C2)n1	C41H49N13O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-2PYE4K	WO-2024183798-A1_CPD--199	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NC5CC6(C5)CC(Nc5nc(NC(C)C)ccc5C(=O)Nc5cc(C)on5)C6)CC4)cn3)nc2n(C2CCCC2)c1=O	C46H57N13O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-GUR1II	WO-2024183798-A1_CPD--20	.	CNc1ccc(C(=O)Nc2ccc(Cl)cn2)c(NCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)n1	C43H52ClN13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-U123IQ	WO-2024183798-A1_CPD--200	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CCN(C(=O)CN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)CC2)n1	C44H55N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-TY0V5L	WO-2024183798-A1_CPD--201	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CCN(C(=O)CN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)C2)n1	C43H53N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-TA22TX	WO-2024183798-A1_CPD--21	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCCCNCCN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)n1	C44H59N15O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-TAWAGK	WO-2024183798-A1_CPD--22	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCCC(C)NC(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)n1	C45H59N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-9Z4J62	WO-2024183798-A1_CPD--23	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(N(C)CCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)n1	C45H59N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-GAYH2Z	WO-2024183798-A1_CPD--24	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(Nc2cnn(CCNC(=O)CN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)c2)n1	C44H53N17O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-MUWNKM	WO-2024183798-A1_CPD--25	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(Nc2cnn(CCNC(=O)CN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)n2)n1	C43H52N18O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-WPHP19	WO-2024183798-A1_CPD--26	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(Nc2cc(CCNC(=O)CN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)no2)n1	C44H52N16O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-IAU5AV	WO-2024183798-A1_CPD--27	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCCCCNc5nc(C6CC6)ccc5C(=O)Nc5ccc(N(C)C)nn5)CC4)cn3)nc2n(C2CCCC2)c1=O	C46H58N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-H277UZ	WO-2024183798-A1_CPD--28	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCCCCNc5nc(C#N)ccc5C(=O)Nc5ccc(N(C)C)nn5)CC4)cn3)nc2n(C2CCCC2)c1=O	C44H53N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-61QRGN	WO-2024183798-A1_CPD--29	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC(C)CCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)n1	C45H59N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-3R3W3U	WO-2024183798-A1_CPD--30	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCCn2cc(CN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)nn2)n1	C44H55N17O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-PAWY6C	WO-2024183798-A1_CPD--31	.	CNc1ccc(C(=O)Nc2ccc(C3CC3)nn2)c(NCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)n1	C45H56N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-LXV9LC	WO-2024183798-A1_CPD--32	.	CNc1ccc(C(=O)Nc2ccc3c(cnn3C)n2)c(NCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)n1	C45H55N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-WSJUEC	WO-2024183798-A1_CPD--33	.	CNc1ccc(C(=O)Nc2ccc3c(ccn3C)n2)c(NCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)n1	C46H56N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-SRT5RF	WO-2024183798-A1_CPD--34	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC(CCNC(=O)CN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)C2)n1	C45H57N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-AVE3EJ	WO-2024183798-A1_CPD--35	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC(CCNC(=O)N3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)C2)n1	C44H55N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-WNM7KF	WO-2024183798-A1_CPD--36	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCCC(=O)NCCN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)n1	C44H57N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-UZP0NR	WO-2024183798-A1_CPD--37	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCCNC(=O)CCN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)n1	C44H57N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-CRGUWX	WO-2024183798-A1_CPD--38	.	CNc1ccc(C(=O)Nc2ccc3ncn(C)c3n2)c(NCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)n1	C45H55N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-CPSB7T	orb2802234	2-[[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]acetyl]amino]spiro[3.3]heptan-6-yl]amino]-N-[6-(dimethylamino)pyridazin-3-yl]-6-(methylamino)pyridine-3-carboxamide; 3055472-38-0	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C46H57N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-YI13XV	WO-2024183798-A1_CPD--40	.	CNc1ccc(C(=O)Nc2ccc3c(n2)CCC3)c(NCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)n1	C46H57N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-0Y2QW4	WO-2024183798-A1_CPD--41	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCC2CC(NC(=O)CN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)C2)n1	C45H57N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-FRUB8W	WO-2024183798-A1_CPD--42	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(N2CCC(CCNC(=O)CN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)CC2)n1	C46H59N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-IE4O0G	WO-2024183798-A1_CPD--43	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(CC2CCC(CNC(=O)CN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)CC2)n1	C47H60N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-887EU8	WO-2024183798-A1_CPD--44	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCCCCNc5nc(C6CC6)ccc5C(=O)Nc5ccc(C)c(C6CC6)n5)CC4)cn3)nc2n(C2CCCC2)c1=O	C49H60N12O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-BJXLOT	WO-2024183798-A1_CPD--45	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCC5CC(Nc6nc(C7CC7)ccc6C(=O)Nc6ccc(C)c(C7CC7)n6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C50H60N12O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-UBUMCY	WO-2024183798-A1_CPD--46	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)cc2)c(NCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)n1	C46H59N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-EGV1H2	WO-2024183798-A1_CPD--47	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)cn2)c(NCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)n1	C45H58N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-6L0R8D	WO-2024183798-A1_CPD--48	.	CNc1ccc(C(=O)NC2CCC(N(C)C)CC2)c(NCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)n1	C46H65N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-NG71RA	WO-2024183798-A1_CPD--49	.	CNc1ccc(C(=O)Nc2ccn(C)n2)c(NCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)n1	C42H54N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-GXUWG4	WO-2024183798-A1_CPD--50	.	CNc1ccc(C(=O)Nc2cc(C)n(C)n2)c(NCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)n1	C43H56N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-E96LZJ	WO-2024183798-A1_CPD--51	.	CNc1ccc(C(=O)Nc2cccc(C3CC3)n2)c(NCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)n1	C46H57N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-HYLBKL	WO-2024183798-A1_CPD--52	.	CNc1ccc(C(=O)Nc2cc(Cl)cc(C3CC3)n2)c(NCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)n1	C46H56ClN13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-X7QWDP	WO-2024183798-A1_CPD--53	.	CNc1ccc(C(=O)Nc2cc(C)cc(C3CC3)n2)c(NCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)n1	C47H59N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-L883XK	WO-2024183798-A1_CPD--54	.	CCc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)n1	C45H58N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-Z559W5	WO-2024183798-A1_CPD--55	.	CNc1ccc(C(=O)NC2CCC(N(C)C)C2)c(NCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)n1	C45H63N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-E56EZT	WO-2024183798-A1_CPD--56	.	CNc1ccc(C(=O)Nc2nc(C3CC3)c(C)s2)c(NCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)n1	C45H57N13O4S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-AC6NJF	WO-2024183798-A1_CPD--57	.	CNc1ccc(C(=O)Nc2ccc(C)c(C3CC3)n2)c(NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C49H59N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-ZF7JFE	WO-2024183798-A1_CPD--58	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nc2)c(NCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)n1	C45H58N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-X5XG8F	WO-2024183798-A1_CPD--59	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCCCCNc5nc(NC6CCC6)ccc5C(=O)Nc5ccc(N(C)C)nn5)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H61N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-WYHO5D	WO-2024183798-A1_CPD--6	.	CNc1ccc(C(=O)Nc2ccc(C)c(C3CC3)n2)c(NCCCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)n1	C49H63N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-UY35HF	WO-2024183798-A1_CPD--60	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NC(C)CCCCNc5nc(C6CC6)ccc5C(=O)Nc5ccc(C)c(C6CC6)n5)CC4)cn3)nc2n(C2CCCC2)c1=O	C50H62N12O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-ZTE5QO	WO-2024183798-A1_CPD--61	.	CNc1ccc(C(=O)Nc2nc(C3CC3)ccc2C)c(NCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)n1	C47H59N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-EWB0FH	WO-2024183798-A1_CPD--62	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC3(C2)CN(C(=O)CCN2CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC2)C3)n1	C46H57N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-QVIPWZ	WO-2024183798-A1_CPD--63	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCCCCNc5nc(C(C)C)ccc5C(=O)Nc5ccc(N(C)C)nn5)CC4)cn3)nc2n(C2CCCC2)c1=O	C46H60N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-E4EE29	WO-2024183798-A1_CPD--64	.	CNc1ccc(C(=O)NC2CC(N(C)C)C2)c(NCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)n1	C44H61N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-A2ET8F	WO-2024183798-A1_CPD--65	.	CNc1ccc(C(=O)NC2CC(CN(C)C)C2)c(NCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)n1	C45H63N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-XOSL3A	WO-2024183798-A1_CPD--67	.	CNc1ccc(C(=O)NC2CC3(C2)CC(N(C)C)C3)c(NCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)n1	C47H65N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-451V5V	WO-2024183798-A1_CPD--68	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCCCCNc5nc(C(F)(F)F)ccc5C(=O)Nc5ccc(N(C)C)nn5)CC4)cn3)nc2n(C2CCCC2)c1=O	C44H53F3N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-HZ50E1	WO-2024183798-A1_CPD--69	.	CNc1ccc(C(=O)Nc2ccc3c(n2)CCC3)c(NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C48H57N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-BAP6VQ	WO-2024183798-A1_CPD--7	.	CNc1ccc(C(=O)Nc2ccc(C)c(C3CC3)n2)c(NCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)n1	C47H59N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-UCRQBW	WO-2024183798-A1_CPD--70	.	CNc1ccc(C(=O)Nc2cc(C)n(C)n2)c(NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C45H56N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-9I8G6F	WO-2024183798-A1_CPD--71	.	CNc1ccc(C(=O)N(C)c2ccc(N(C)C)nn2)c(NCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)n1	C45H59N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-I0P6HX	WO-2024183798-A1_CPD--72	.	CNc1ccc(C(=O)Nc2cccc(C3CC3)n2)c(NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C48H57N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-R0LECW	WO-2024183798-A1_CPD--73	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCC2CCC(NC(=O)CN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)CC2)n1	C46H59N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-NRLOX7	WO-2024183798-A1_CPD--74	.	CNc1ccc(C(=O)Nc2ccc(C3CC3)nc2)c(NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C48H57N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-Y6SXCI	WO-2024183798-A1_CPD--75	.	CNc1ccc(C(=O)Nc2cccc(C)n2)c(NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C46H55N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-PHSWWZ	WO-2024183798-A1_CPD--76	.	CNc1ccc(C(=O)Nc2cccc(C(C)C)n2)c(NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C48H59N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-Q31DRN	WO-2024183798-A1_CPD--77	.	CNc1ccc(C(=O)Nc2ccc(=O)[nH]n2)c(NCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)n1	C42H52N14O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-X3SAOO	WO-2024183798-A1_CPD--78	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC3(CC(NCC(=O)N4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C46H57N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-2186PT	WO-2024183798-A1_CPD--79	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC(CNC(=O)CN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)C2)n1	C44H55N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-Z6PD7L	WO-2024183798-A1_CPD--80	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC(CNC(=O)CCN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)C2)n1	C45H57N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-RLC8CR	WO-2024183798-A1_CPD--81	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC3(CC(CNC(=O)N4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C46H57N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-EY4Q6W	WO-2024183798-A1_CPD--82	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC3(CC(CCC(=O)N4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C47H58N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-BZC8D4	WO-2024183798-A1_CPD--83	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC3(CC(CCCN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C47H60N14O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-R8CN6D	WO-2024183798-A1_CPD--84	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC3(C2)CC(OCC(=O)N2CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC2)C3)n1	C46H56N14O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-LNM2XB	WO-2024183798-A1_CPD--85	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCCCCNc5nc(NC(C)(C)C)ccc5C(=O)Nc5ccc(N(C)C)nn5)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H63N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-KHIB23	WO-2024183798-A1_CPD--86	.	CNc1ccc(C(=O)Nc2ccnc(C3CC3)c2)c(NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C48H57N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-NZLA63	WO-2024183798-A1_CPD--87	.	CNc1ccc(C(=O)Nc2ccc(C(F)(F)F)c(C3CC3)n2)c(NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C49H56F3N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-BX7HDD	WO-2024183798-A1_CPD--88	.	CNc1ccc(C(=O)Nc2cccc(N(C)C)n2)c(NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C47H58N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-C7SOGC	WO-2024183798-A1_CPD--89	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCC2CCN(C(=O)CN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)CC2)n1	C46H59N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-ZOIRYY	WO-2024183798-A1_CPD--9	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCCCCCCNc5nc(C)ccc5C(=O)Nc5ccc(C)c(C6CC6)n5)CC4)cn3)nc2n(C2CCCC2)c1=O	C49H62N12O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-36RMF1	WO-2024183798-A1_CPD--90	.	CNc1ccc(C(=O)Nc2cccc(C#N)n2)c(NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C46H52N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-XVOMI9	WO-2024183798-A1_CPD--91	.	CNc1ccc(C(=O)Nc2cccc(C(F)(F)F)n2)c(NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C46H52F3N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-SZKW4D	WO-2024183798-A1_CPD--92	.	CNc1ccc(C(=O)Nc2cc(C)[nH]n2)c(NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C44H54N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-HY0QVW	WO-2024183798-A1_CPD--93	.	CNc1ccc(C(=O)Nc2ccn(C)n2)c(NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C44H54N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-RI2DRB	WO-2024183798-A1_CPD--94	.	CNc1ccc(C(=O)Nc2cnn(C)c2)c(NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C44H54N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-JK4XCQ	WO-2024183798-A1_CPD--95	.	CNc1ccc(C(=O)Nc2cc(C(C)C)n(C)n2)c(NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C47H60N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-S39XQQ	WO-2024183798-A1_CPD--96	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC3(CC(NCCN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C46H59N15O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-JFXOE8	WO-2024183798-A1_CPD--97	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC3(C2)CN(C(=O)CN2CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC2)C3)n1	C45H55N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-SEGK7W	WO-2024183798-A1_CPD--98	.	CNc1ccc(C(=O)Nc2cc(C3CC3)n(C)n2)c(NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C47H58N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-21S82O	WO-2024183798-A1_CPD--99	.	CNc1ccc(C(=O)Nc2cc(C)n(C(C)C)n2)c(NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C47H60N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-OCSPQ9	WO-2024183798-A1_CPD-1	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCCNc5nc(C)ccc5C(=O)Nc5nc(C)c(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C41H50N12O4S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-B8FNO0	WO-2024183798-A1_CPD-2	.	COc1ccc(NC(=O)c2ccc(C)nc2NCCCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)nn1	C45H57N13O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-20ZZVM	WO-2024183798-A1_CPD-202	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC(Cn3cc(CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)nn3)C2)n1	C45H55N17O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-XPJ5U9	WO-2024183798-A1_CPD-203	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CCN(C(=O)CCN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)CC2)n1	C45H57N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-M4T1P8	WO-2024183798-A1_CPD-204	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NNC2CCC(CCC(=O)N3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)CC2)n1	C46H59N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-QQQ609	WO-2024183798-A1_CPD-205	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCC5CC(Nc6nc(NC(C)C)ccc6C(=O)Nc6cc(C)n(C)n6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H58N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-ZOC73I	WO-2024183798-A1_CPD-206	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCC5CC(Nc6nc(C)ccc6C(=O)Nc6cc(C)n(C)n6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C43H53N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-802RZ7	WO-2024183798-A1_CPD-207	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NC5CC6(C5)CC(Nc5nc(C)ccc5C(=O)Nc5cn(C)c(C7CC7)n5)C6)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H57N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-8JYY7L	WO-2024183798-A1_CPD-208	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC3(C2)CC(C(=O)C(F)(F)CN2CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC2)C3)n1	C47H56F2N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-BMTRK1	WO-2024183798-A1_CPD-210	.	CCc1ccc(C(=O)Nc2cc(C)n(C)n2)c(NC2CC(CNC(=O)CN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)C2)n1	C44H55N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-NZ8HVL	WO-2024183798-A1_CPD-211	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CN(C(=O)CCCN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)C2)n1	C44H55N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-8EZQAX	WO-2024183798-A1_CPD-212	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCC5CC(Nc6nc(C(C)C)ccc6C(=O)Nc6cc(C)n(C)n6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H57N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-S8XRA1	WO-2024183798-A1_CPD-213	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCC5CC(Nc6nc(C7CC7)ccc6C(=O)Nc6cc(C)n(C)n6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H55N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-Z3PIEO	WO-2024183798-A1_CPD-214	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCC2CCC(OCC(=O)N3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)CC2)n1	C46H58N14O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-ARTNBL	WO-2024183798-A1_CPD-215	.	CNc1ccc(C(=O)Nc2cc(C3CC3)on2)c(NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C46H55N13O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-WZLDH9	WO-2024183798-A1_CPD-216	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC3(C2)CC(OC(C)(C)C(=O)N2CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC2)C3)n1	C48H60N14O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-HXRZWL	WO-2024183798-A1_CPD-217	.	CNc1ccc(C(=O)Nc2cn(C)c(C3CC3)n2)c(NC2CC(NC(=O)CN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)C2)n1	C44H54N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-ZM543V	WO-2024183798-A1_CPD-218	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CCN(C(=O)CCN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)C2)n1	C44H55N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-W9H84A	WO-2024183798-A1_CPD-219	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CCC(NC(=O)CN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)C2)n1	C44H55N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-6QW8SI	WO-2024183798-A1_CPD-220	.	CNc1ccc(C(=O)Nc2ccc(OC)c(C)n2)c(NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C47H57N13O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-RSDSK1	WO-2024183798-A1_CPD-221	.	CNc1ccc(C(=O)Nc2ccc(F)c(C)n2)c(NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C46H54FN13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-P42HO6	WO-2024183798-A1_CPD-222	.	CC(=O)c1c(C)c2ccc(Nc3ccc(N4CCN(CC(=O)NC5CC6(C5)CC(Nc5nc(NC(C)C)ccc5C(=O)Nc5cn(C)c(C7CC7)n5)C6)CC4)cn3)nc2n(C2CCCC2)c1=O	C50H63N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-TEAP70	WO-2024183798-A1_CPD-223	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CCC(NC(=O)CCN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)CC2)n1	C46H59N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-ESIP79	WO-2024183798-A1_CPD-224	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC3(C2)CN(C(=O)CC(C)N2CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC2)C3)n1	C47H59N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-PCQRRD	WO-2024183798-A1_CPD-226	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(=O)C(C)(C)OC5CC6(CC(Nc7nc(C)ccc7C(=O)Nc7cccc(C)n7)C6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C48H57N11O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-Q7GBDK	WO-2024183798-A1_CPD-227	.	CNc1ccc(C(=O)Nc2cc(C(C)C)on2)c(NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C46H57N13O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-POL8PU	WO-2024183798-A1_CPD-228	.	CNc1ccc(C(=O)Nc2cc(C)[nH]n2)c(NC2CCN(C(=O)CN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)CC2)n1	C42H52N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-BPFOV5	WO-2024183798-A1_CPD-229	.	CNc1ccc(C(=O)Nc2cc(C)on2)c(NC2CCN(C(=O)CN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)CC2)n1	C42H51N13O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-7IT5I5	WO-2024183798-A1_CPD-230	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)N5CCC(Nc6nc(C)ccc6C(=O)Nc6cc(C)n(C)n6)CC5)CC4)cn3)nc2n(C2CCCC2)c1=O	C43H53N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-455CRH	WO-2024183798-A1_CPD-231	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)N5CCC(Nc6nc(C)ccc6C(=O)Nc6cc(C)on6)CC5)CC4)cn3)nc2n(C2CCCC2)c1=O	C42H50N12O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-NN31P3	WO-2024183798-A1_CPD-233	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(F)(F)C(=O)N5CC(Nc6nc(C)ccc6C(=O)Nc6cc(C)n(C)n6)C5)CC4)cn3)cc2n(C2CCCC2)c1=O	C43H50F2N12O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-IXD6YF	WO-2024183798-A1_CPD-234	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(F)(F)C(=O)N5CC(Nc6nc(C)ccc6C(=O)Nc6cc(C)on6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C41H46F2N12O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-B79D21	WO-2024183798-A1_CPD-235	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CCC3(C2)CN(C(=O)CN2CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC2)C3)n1	C46H57N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-ZNAUAH	WO-2024183798-A1_CPD-236	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)N5CCC(Nc6nc(C)ccc6C(=O)Nc6cn(C)c(C7CC7)n6)CC5)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H55N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-VF97XQ	WO-2024183798-A1_CPD-238	.	CNc1ccc(C(=O)Nc2cn(C(C)C)c(C)n2)c(NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C47H60N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-9SGUB0	WO-2024183798-A1_CPD-239	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NC5CC6(C5)CC(Nc5nc(C)ccc5C(=O)Nc5ccc(F)c(C7CC7)n5)C6)CC4)cn3)nc2n(C2CCCC2)c1=O	C48H55FN12O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-DCT8MU	WO-2024183798-A1_CPD-240	.	CNc1ccc(C(=O)Nc2cccc(C3CC3)n2)c(NC2CC(NC(=O)CN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)C2)n1	C45H53N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-VKR8RJ	WO-2024183798-A1_CPD-241	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NC5CC6(C5)CC(Nc5nc(C)ccc5C(=O)Nc5ccc(N(C)C)nn5)C6)CC4)cn3)nc2n(C2CCCC2)c1=O	C46H56N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-MO4FXI	WO-2024183798-A1_CPD-242	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC(NC(=O)C(C)N3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)C2)n1	C44H55N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-GPJYPX	WO-2024183798-A1_CPD-243	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC(NC(=O)C(C)(C)N3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)C2)n1	C45H57N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-TU59FQ	WO-2024183798-A1_CPD-244	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NC5CC6(C5)CC(Nc5nc(C)ccc5C(=O)Nc5cc(C)n(C)n5)C6)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H55N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-JRPV8B	WO-2024183798-A1_CPD-245	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NC5CC(Nc6nc(C)ccc6C(=O)Nc6ccc(N(C)C)nn6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C43H52N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-869CU1	WO-2024183798-A1_CPD-246	.	CNc1ccc(C(=O)Nc2ncc(C)o2)c(NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C44H53N13O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-W8LTJE	WO-2024183798-A1_CPD-247	.	CNc1ccc(C(=O)Nc2nc(C)c(C)o2)c(NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C45H55N13O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-3MF73D	WO-2024183798-A1_CPD-248	.	C=C(C)c1c(C)c2ccc(Nc3ccc(N4CCN(CC(F)(F)C(=O)N5CC(Nc6nc(C)ccc6C(=O)Nc6ccc(N(C)C)nn6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H53F2N13O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-6C81U1	WO-2024183798-A1_CPD-249	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(F)(F)C(=O)N5CC6(CC(Nc7nc(C)ccc7C(=O)Nc7ccc(N(C)C)nn7)C6)C5)CC4)cc3)nc2n(C2CCCC2)c1=O	C47H55F2N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-74F6WF	WO-2024183798-A1_CPD-250	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)N5CCC(Nc6nc(C)ccc6C(=O)Nc6ccc(N(C)C)nn6)CC5)CC4)cn3)nc2n(C2CCCC2)c1=O	C44H54N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-YQX3C9	WO-2024183798-A1_CPD-251	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCCCCNc5nc6[nH]ccc6cc5C(=O)Nc5ccc(N(C)C)nn5)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H55N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-TVBS8X	WO-2024183798-A1_CPD-252	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)N5CCC(Nc6nc(C)ccc6C(=O)Nc6cccc(C7CC7)n6)CC5)CC4)cn3)nc2n(C2CCCC2)c1=O	C46H54N12O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-VRUJ6D	WO-2024183798-A1_CPD-253	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NC5CC6(CC(Cc7nc(NC(C)C)ccc7C(=O)Nc7cc(C)n(C)n7)C6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C48H61N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-VD5AD5	WO-2024183798-A1_CPD-254	.	CNc1ccc(C(=O)Nc2cn(C)c(C3CC3)n2)c(NC2CC(CNC(=O)CN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)C2)n1	C45H56N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-DNTWNO	WO-2024183798-A1_CPD-259	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NC5CC6(C5)CC(Nc5cc(Cl)ccc5C(=O)Nc5cc(C)on5)C6)CC4)cn3)nc2n(C2CCCC2)c1=O	C44H50ClN11O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-FSFSXM	WO-2024183798-A1_CPD-260	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NC5CC6(C5)CC(Nc5cc(F)ccc5C(=O)Nc5cc(C)on5)C6)CC4)cn3)nc2n(C2CCCC2)c1=O	C44H50FN11O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-GPEKW6	WO-2024183798-A1_CPD-261	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCC5CC(Nc6cc(C(F)(F)F)ccc6C(=O)Nc6cc(C)n(C)n6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C44H51F3N12O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-1VIBU5	WO-2024183798-A1_CPD-262	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)CCC5CC(Nc6ccc(C(F)(F)F)cc6C(=O)Nc6cc(C)n(C)n6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H52F3N11O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-4D09P6	WO-2024183798-A1_CPD-263	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCC5CC(Nc6ccc(F)cc6C(=O)Nc6cc(C)n(C)n6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C43H51FN12O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-4CJC55	WO-2024183798-A1_CPD-264	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCC5CC(Nc6cc(F)ccc6C(=O)Nc6cc(C)n(C)n6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C43H51FN12O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-ZGN0R0	WO-2024183798-A1_CPD-265	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCC5CC(Nc6c(F)cccc6C(=O)Nc6cc(C)n(C)n6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C43H51FN12O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-G64F5E	WO-2024183798-A1_CPD-266	.	CC(=O)c1c(C)c2ccc(Nc3ccc(N4CCN(CC(=O)NCC5CC(Nc6c(C(=O)Nc7cc(C)n(C)n7)cccc6C(F)(F)F)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H52F3N11O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-H9VU62	WO-2024183798-A1_CPD-267	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC3(C2)CN(C(=O)CCN2CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC2(C)C)C3)n1	C48H61N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-1I0RT9	WO-2024183798-A1_CPD-268	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC3(C2)CN(C(=O)CN2CCN(Cc4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC2)C3)n1	C46H57N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-PRRC0G	WO-2024183798-A1_CPD-269	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CN(C(=O)CN3CCN(Cc4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)C2)n1	C43H53N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-23KIVH	WO-2024183798-A1_CPD-270	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)N5CCC(Nc6nc(C)ccc6C(=O)Nc6cccc(C)n6)CC5)CC4)cn3)nc2n(C2CCCC2)c1=O	C44H52N12O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-0EHIW1	WO-2024183798-A1_CPD-271	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CCC(CNC(=O)CN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)C2)n1	C45H57N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-P59TVH	WO-2024183798-A1_CPD-272	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NC5CC6(C5)CC(Nc5nc(NC(C)C)ccc5C(=O)Nc5ccc(N(C)C)nn5)C6)CC4)cn3)nc2n(C2CCCC2)c1=O	C48H61N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-JCVUO0	WO-2024183798-A1_CPD-273	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CCC(=O)N5CCC(Nc6nc(C)ccc6C(=O)Nc6cn(C)c(C7CC7)n6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H55N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-V7G7HQ	WO-2024183798-A1_CPD-274	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CCC(=O)N5CCC(Nc6nc(NC(C)C)ccc6C(=O)Nc6cn(C)c(C7CC7)n6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H60N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-RUR60M	WO-2024183798-A1_CPD-275	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)N[C@H]5CC[C@H](CNc6nc(NC(C)C)ccc6C(=O)Nc6cn(C)c(C7CC7)n6)CC5)CC4)cn3)nc2n(C2CCCC2)c1=O	C49H64N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-3DH16K	WO-2024183798-A1_CPD-276	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)N[C@H]5CC[C@H](CNc6nc(C)ccc6C(=O)Nc6cn(C)c(C7CC7)n6)CC5)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H59N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-D0ECKA	WO-2024183798-A1_CPD-277	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCC5CC(Nc6nc(NC(C)C)ccc6C(=O)Nc6cn(C)c(C7CC7)n6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H60N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-D8FWXH	WO-2024183798-A1_CPD-278	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCC5CC(Nc6nc(C)ccc6C(=O)Nc6cn(C)c(C7CC7)n6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H55N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-9CZ0ER	WO-2024183798-A1_CPD-279	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)N5CCC(Nc6nc(NC(C)C)ccc6C(=O)Nc6cn(C)c(C7CC7)n6)CC5)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H60N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-I5WCG7	WO-2024183798-A1_CPD-280	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NC5CC(Nc6nc(NC(C)C)ccc6C(=O)Nc6ccc(N(C)C)nn6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H57N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-PAHD1W	WO-2024183798-A1_CPD-281	.	CNc1ccc(C(=O)Nc2cc(C)on2)c(NC2CC(CNC(=O)CN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)C2)n1	C42H51N13O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-19P7BA	WO-2024183798-A1_CPD-282	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCC5CC(Nc6nc(NC(C)C)ccc6C(=O)Nc6cc(C)on6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C44H55N13O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-FM058I	WO-2024183798-A1_CPD-283	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCC5CC(Nc6nc(C)ccc6C(=O)Nc6cc(C)on6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C42H50N12O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-ZKAU1J	WO-2024183798-A1_CPD-284	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NC5CCC(Nc6nc(NC(C)C)ccc6C(=O)Nc6cn(C)c(C7CC7)n6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H60N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-9UZWF5	WO-2024183798-A1_CPD-285	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NC5CCC(Nc6nc(C)ccc6C(=O)Nc6cn(C)c(C7CC7)n6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H55N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-LMZ84D	WO-2024183798-A1_CPD-286	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NC5CC6(C5)CC(Nc5cc(C)ccc5C(=O)Nc5cc(C)on5)C6)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H53N11O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-48OBP4	WO-2024183798-A1_CPD-287	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(=O)NC5CC(Nc6nc(C)ccc6C(=O)Nc6cn(C)c(C7CC7)n6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C43H51N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-4ZUKXB	WO-2024183798-A1_CPD-288	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NC5CC(Nc6nc(NC(C)C)ccc6C(=O)Nc6cn(C)c(C7CC7)n6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C46H58N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-WHGHI3	WO-2024183798-A1_CPD-289	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(=O)NC5CC(Nc6nc(NC(C)C)ccc6C(=O)Nc6cn(C)c(C7CC7)n6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H56N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-ZWXO9A	WO-2024183798-A1_CPD-290	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)N5CCC(Nc6nc(NC(C)C)ccc6C(=O)Nc6cc(C)on6)CC5)CC4)cn3)nc2n(C2CCCC2)c1=O	C44H55N13O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-QD0CIJ	WO-2024183798-A1_CPD-291	.	C=C(C)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NC5CC6(C5)CC(Nc5nc(N(C)C)ccc5C(=O)Nc5cn(C)c(C7CC7)n5)C6)CC4)cn3)nc2n(C2CCCC2)c1=O	C49H62N14O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-0R0DO9	WO-2024183798-A1_CPD-292	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NC5CC6(C5)CC(Nc5nc(OC(C)C)ccc5C(=O)Nc5cn(C)c(C7CC7)n5)C6)CC4)cn3)nc2n(C2CCCC2)c1=O	C49H61N13O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-ZFFN4M	WO-2024183798-A1_CPD-293	.	CCNc1ccc(C(=O)Nc2cn(C)c(C3CC3)n2)c(NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C48H60N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-4CZOZZ	WO-2024183798-A1_CPD-294	.	C=C(C)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NC5CCC(Nc6ncccc6C(=O)Nc6cc(C)on6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C42H50N12O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-Y5JHOF	WO-2024183798-A1_CPD-295	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NC5CCC(Nc6nc(NC(C)C)ccc6C(=O)Nc6cc(C)on6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C44H55N13O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-3GS480	WO-2024183798-A1_CPD-296	.	CNc1ccc(C(=O)Nc2cn(C)c(C3CCCC3)n2)c(NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)c1	C50H63N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-TDY58A	WO-2024183798-A1_CPD-297	.	CNc1ccc(C(=O)Nc2cc(C)n(C3CCC3)n2)c(NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C48H60N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-9J3XIC	WO-2024183798-A1_CPD-298	.	CCCNc1ccc(C(=O)Nc2cn(C)c(C3CC3)n2)c(NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C49H62N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-1HQU3F	WO-2024183798-A1_CPD-299	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CCN(C(=O)CNC3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)CC2)n1	C45H57N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-C3X9L1	WO-2024183798-A1_CPD-3	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCCCCCNc5nc(C)ccc5C(=O)Nc5nc(C)c(C)s5)CC4)cn3)nc2n(C2CCCC2)c1=O	C43H54N12O4S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-CW0EIL	WO-2024183798-A1_CPD-300	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CCN(C(=O)CN3CCN(Cc4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)CC2)n1	C45H57N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-HMNL5D	WO-2024183798-A1_CPD-301	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CCC(=O)N5CCC(Nc6nc(NC(C)C)ccc6C(=O)Nc6ccc(N(C)C)nn6)CC5)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H61N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-RBC0YU	WO-2024183798-A1_CPD-302	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CCC(=O)N5CC6(CC(Nc7nc(NC(C)C)ccc7C(=O)Nc7cc(C)n(C)n7)C6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H60N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-5CQOV9	WO-2024183798-A1_CPD-303	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CCC(=O)N5CC(Nc6nc(NC(C)C)ccc6C(=O)Nc6ccc(N(C)C)nn6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H57N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-25ERT2	WO-2024183798-A1_CPD-304	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CCC(=O)N5CC(Nc6nc(NC(C)C)ccc6C(=O)Nc6cn(C)c(C7CC7)n6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C46H58N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-XKCBZQ	WO-2024183798-A1_CPD-305	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CCC(=O)N5CC6(CC(Nc7nc(NC(C)C)ccc7C(=O)Nc7ccc(N(C)C)nn7)C6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C48H61N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-1I4009	WO-2024183798-A1_CPD-306	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC5(C(=O)N6CC7(CC(Nc8nc(NC(C)C)ccc8C(=O)Nc8ccc(N(C)C)nn8)C7)C6)CC5)CC4)cn3)nc2n(C2CCCC2)c1=O	C50H63N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-FPG6C1	WO-2024183798-A1_CPD-307	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NC5CC(Nc6nc(C)ccc6C(=O)Nc6cn(C)c(C7CC7)n6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C44H53N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-BBRFMO	WO-2024183798-A1_CPD-308	.	CCc1nc(NC(=O)c2ccc(NC)nc2NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)cn1C	C46H58N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-KCOTTJ	WO-2024183798-A1_CPD-309	.	CCCc1nc(NC(=O)c2ccc(NC)nc2NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)c[nH]1	C46H58N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-L8HG4J	WO-2024183798-A1_CPD-310	.	CNc1ccc(C(=O)Nc2cn(C)c(C3CCC3)n2)c(NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C48H60N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-CQGAUL	WO-2024183798-A1_CPD-311	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC(OC(=O)N3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)C2)n1	C42H50N14O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-MTC3WD	WO-2024183798-A1_CPD-312	.	CCn1nc(NC(=O)c2ccc(NC)nc2NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)cc1C	C46H58N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-Z3IG8F	WO-2024183798-A1_CPD-313	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CCC(=O)N5CCC(Nc6nc(NC(C)C)ccc6C(=O)Nc6c[nH]c(C7CC7)n6)CC5)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H60N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-NMIAJ9	WO-2024183798-A1_CPD-314	.	CCCn1nc(NC(=O)c2ccc(NC)nc2NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)cc1C	C47H60N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-Z97BU7	WO-2024183798-A1_CPD-315	.	CNc1ccc(C(=O)Nc2cc(C)n(C3CC3)n2)c(NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C47H58N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-Y0AONU	WO-2024183798-A1_CPD-316	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCC5CC(Nc6nc(NC(C)C)ccc6C(=O)Nc6ccc(N(C)C)nn6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C46H59N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-IW93YX	WO-2024183798-A1_CPD-317	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NC5CC6(C5)CC(Oc5nc(NC(C)C)ccc5C(=O)Nc5cn(C)c(C7CC7)n5)C6)CC4)cn3)nc2n(C2CCCC2)c1=O	C49H61N13O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-8NURK1	WO-2024183798-A1_CPD-318	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NC5CC6(C5)CC(Nc5nc(CC(C)C)ccc5C(=O)Nc5cn(C)c(C7CC7)n5)C6)CC4)cn3)nc2n(C2CCCC2)c1=O	C50H63N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-443VB7	WO-2024183798-A1_CPD-319	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC(N3CCC(CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C46H59N15O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-EMIDET	WO-2024183798-A1_CPD-320	.	CNc1ccc(C(=O)Nc2cn(C)c(C3CC3)n2)c(NC2CC3(C2)CN(C(=O)C2CC24CCN(c2ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc2)CC4)C3)n1	C48H57N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-H5Z3PN	WO-2024183798-A1_CPD-321	.	CNc1ccc(C(=O)Nc2cn(C)c(C3CC3)n2)c(NC2CC3(C2)CN(C(=O)C2CC4(CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C2)C3)n1	C49H59N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-38AFGT	WO-2024183798-A1_CPD-322	.	CC(=O)c1c(C)c2ccc(Nc3ccc(N4CCN(CC5(C(=O)N6CC7(CC(Nc8nc(NC(C)C)ccc8C(=O)Nc8cn(C)c(C9CC9)n8)C7)C6)CC5)CC4)cn3)nc2n(C2CCCC2)c1=O	C52H65N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-4MAFG5	WO-2024183798-A1_CPD-323	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CCC(=O)N5CC6(CC(Nc7nc(NC(C)C)ccc7C(=O)Nc7cn(C)c(C8CC8)n7)C6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C49H62N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-UHTKXW	WO-2024183798-A1_CPD-324	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC3(C2)CN(C(=O)C2CC24CCN(c2ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc2)CC4)C3)n1	C47H56N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-K9EOB0	WO-2024183798-A1_CPD-325	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC3(C2)CN(C(=O)C2CC4(CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C2)C3)n1	C48H58N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-DE4307	WO-2024183798-A1_CPD-326	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(C)C(=O)NC5CC(Nc6nc(NC(C)C)ccc6C(=O)Nc6ccc(N(C)C)nn6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C46H59N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-WMNTPN	WO-2024183798-A1_CPD-327	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(C)C(=O)NC5CC(Nc6nc(NC(C)C)ccc6C(=O)Nc6cn(C)c(C7CC7)n6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H60N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-Y66OH2	WO-2024183798-A1_CPD-328	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CCN(C(=O)C3CC34CCN(c3ccc(Nc5cc6c(cn5)c(C)c(C(C)=O)c(=O)n6C5CCCC5)nc3)CC4)CC2)n1	C47H57N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-QULPIT	WO-2024183798-A1_CPD-329	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CCN(C(=O)C3CC4(CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)CC2)n1	C47H58N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-Z7BAY1	WO-2024183798-A1_CPD-330	.	CNc1ccc(C(=O)Nc2cn(C)c(C(C)O)n2)c(NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C46H58N14O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-IDFWNG	WO-2024183798-A1_CPD-331	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC(C(=O)N3CC4(CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C45H54N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-CWSC6K	WO-2024183798-A1_CPD-332	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC(C(=O)N3CC(N4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C45H55N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-UMY51C	WO-2024183798-A1_CPD-333	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC(C(=O)N3CCC(N4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C46H57N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-BT5IH0	WO-2024183798-A1_CPD-334	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC(C(=O)N3CCC(N4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)CC3)C2)n1	C47H59N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-6ZWFYJ	WO-2024183798-A1_CPD-335	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC(n3cc(CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)nn3)C2)n1	C44H53N17O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-6V789S	WO-2024183798-A1_CPD-336	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC(CN3CCC(CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C47H61N15O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-2257GZ	WO-2024183798-A1_CPD-337	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC(C(=O)N3CCC4(CC3)CCN(c3ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc3)CC4)C2)n1	C47H58N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-ZUI26M	WO-2024183798-A1_CPD-338	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(C)CC(=O)N5CC6(CC(Nc7nc(NC(C)C)ccc7C(=O)Nc7cn(C)c(C8CC8)n7)C6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C50H64N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-U2EJJC	WO-2024183798-A1_CPD-339	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(C)CC(=O)N5CC6(CC(Nc7nc(C)ccc7C(=O)Nc7cn(C)c(C8CC8)n7)C6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C48H59N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-PV136D	WO-2024183798-A1_CPD-340	.	CNc1ccc(C(=O)Nc2cn(C)c(C(C)(C)O)n2)c(NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C47H60N14O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-ZWLO5T	WO-2024183798-A1_cpd-341	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(C)CC(=O)N5CC6(CC(Nc7nc(C)ccc7C(=O)Nc7ccc(N(C)C)nn7)C6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H58N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-XPCG8Z	WO-2024183798-A1_CPD-342	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(CC(=O)N5CC6(CC(Nc7nc(C)ccc7C(=O)Nc7ccc(N(C)C)nn7)C6)C5)C(F)(F)F)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H55F3N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-CKKUIN	WO-2024183798-A1_CPD-343	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCC5CC(Nc6nc(C)ccc6C(=O)Nc6ccc(N(C)C)nn6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C44H54N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-ZWOF1M	WO-2024183798-A1_CPD-344	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCC2(F)CN(C(=O)CN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)C2)n1	C43H52FN15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-XGLSCG	WO-2024183798-A1_CPD-345	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCC23CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)(C2)C3)n1	C45H55N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-84CCLS	WO-2024183798-A1_CPD-346	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC23CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)(C2)C3)n1	C44H53N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-85D7OJ	WO-2024183798-A1_CPD-347	.	CNc1ccc(C(=O)Nc2cn(C)c(C3CC3)n2)c(NC2CCC3(CC2)CC(NC(=O)CN2CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC2)C3)n1	C49H62N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-HT1DSM	WO-2024183798-A1_CPD-348	.	CNc1ccc(C(=O)Nc2ccc(CN(C)C)nn2)c(NC2CC3(C2)CN(C(=O)C2CC(N4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C2)C3)n1	C49H61N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-JBUIVB	WO-2024183798-A1_CPD-349	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NC5CC6(C5)CC(Nc5nc(C(C)O)ccc5C(=O)Nc5cn(C)c(C7CC7)n5)C6)CC4)cn3)nc2n(C2CCCC2)c1=O	C48H59N13O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-CZ0WXO	WO-2024183798-A1_CPD-350	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CCC(C(=O)N3CCC4(CC3)CCN(c3ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc3)CC4)CC2)n1	C49H62N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-ZTOXGY	WO-2024183798-A1_CPD-351	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CCC(C(=O)N3CC4(CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)CC2)n1	C47H58N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-OZ2C4N	WO-2024183798-A1_CPD-352	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NC5CC6(C5)CC(Nc5nc(C(C)(C)O)ccc5C(=O)Nc5cn(C)c(C7CC7)n5)C6)CC4)cn3)nc2n(C2CCCC2)c1=O	C49H61N13O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-A802YB	WO-2024183798-A1_CPD-353	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NC(C)C5CC(Nc6nc(C)ccc6C(=O)Nc6cc(C)n(C)n6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C44H55N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-VESZ0X	WO-2024183798-A1_CPD-354	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCC2COC3(C2)CN(C(=O)CN2CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC2)C3)n1	C46H57N15O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-PF1T1N	WO-2024183798-A1_CPD-355	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(C)CC(=O)N5CC(Nc6nc(NC(C)C)ccc6C(=O)Nc6ccc(N(C)C)nn6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C46H59N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-X04L2K	WO-2024183798-A1_CPD-356	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCC(NCC(=O)N5CC(Nc6nc(NC(C)C)ccc6C(=O)Nc6ccc(N(C)C)nn6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H57N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-ZNK908	WO-2024183798-A1_CPD-357	.	C=C(C)c1c(C)c2cnc(Nc3ccc(N4CCC(NCC(=O)N5CCC(Nc6nc(NC(C)C)ccc6C(=O)Nc6ccc(N(C)C)nn6)CC5)CC4)cn3)nc2n(C2CCCC2)c1=O	C48H63N15O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-EBFUED	WO-2024183798-A1_CPD-358	.	CC(=O)c1c(C)c2cnc(Nc3ccc(CN4CCN(CC(=O)N5CCC(Nc6nc(NC(C)C)ccc6C(=O)Nc6ccc(N(C)C)nn6)CC5)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H61N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-VYJTO9	WO-2024183798-A1_CPD-359	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(C)CC(=O)N5CCC(Nc6nc(NC(C)C)ccc6C(=O)Nc6ccc(N(C)C)nn6)CC5)CC4)cn3)nc2n(C2CCCC2)c1=O	C48H63N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-WOPOYE	WO-2024183798-A1_CPD-360	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCC(N(C)CC(=O)N5CCC(Nc6nc(NC(C)C)ccc6C(=O)Nc6ccc(N(C)C)nn6)CC5)CC4)cn3)nc2n(C2CCCC2)c1=O	C48H63N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-ZZGVDY	WO-2024183798-A1_CPD-361	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NC(C)C5CC(Nc6nc(C)ccc6C(=O)Nc6cc(C)on6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C43H52N12O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-EN0PM5	WO-2024183798-A1_CPD-362	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CCC(C(=O)N3CC(N4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)CC2)n1	C47H59N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-YGLQLM	WO-2024183798-A1_CPD-363	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC3(C2)CC(C(=O)N2CC4(CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C2)C3)n1	C48H58N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-R7I747	WO-2024183798-A1_CPD-364	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC3(C2)CN(C(=O)C2CN(C4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C2)C3)n1	C48H59N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-HPBZY0	WO-2024183798-A1_CPD-365	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(C)CC(=O)NC5CC(Nc6nc(NC(C)C)ccc6C(=O)Nc6ccc(N(C)C)nn6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H61N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-5WRZ8J	WO-2024183798-A1_CPD-366	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C5(C(=O)NC6CC7(C6)CC(Nc6nc(NC(C)C)ccc6C(=O)Nc6cn(C)c(C8CC8)n6)C7)CC5)CC4)cn3)nc2n(C2CCCC2)c1=O	C51H64N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-J5WHF3	WO-2024183798-A1_CPD-367	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(CC(=O)N5CC6(CC(Nc7nc(NC(C)C)ccc7C(=O)Nc7ccc(N(C)C)nn7)C6)C5)C(F)(F)F)CC4)cn3)nc2n(C2CCCC2)c1=O	C49H60F3N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-I0T8WG	WO-2024183798-A1_CPD-368	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(C)CC(=O)N5CC6(CC(Nc7nc(NC(C)C)ccc7C(=O)Nc7ccc(N(C)C)nn7)C6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C49H63N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-8FUC9N	WO-2024183798-A1_CPD-369	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)N5CCC(Nc6nc(NC(C)C)ccc6C(=O)Nc6ccc(N(C)C)nn6)CC5)CC4)cn3)nc2n(C2CCCC2)c1=O	C46H59N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-PG5NOD	WO-2024183798-A1_CPD-370	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(C)CC(=O)N5CCC(Nc6nc(NC(C)C)ccc6C(=O)Nc6ccc(N(C)C)nn6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H61N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-TDO6A2	WO-2024183798-A1_CPD-371	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C5(C(=O)NC6CC7(C6)CC(Nc6nc(NC(C)C)ccc6C(=O)Nc6cc(C)on6)C7)CC5)CC4)cn3)nc2n(C2CCCC2)c1=O	C48H59N13O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-MSY3N4	WO-2024183798-A1_CPD-372	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCC(NCC(=O)N5CCC(Nc6nc(NC(C)C)ccc6C(=O)Nc6ccc(N(C)C)nn6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C46H59N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-Z9OAX1	WO-2024183798-A1_CPD-373	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCC5(CN(CC(=O)N6CC7(CC(Nc8nc(C)ccc8C(=O)Nc8ccc(N(C)C)nn8)C7)C6)C5)C4)cn3)nc2n(C2CCCC2)c1=O	C47H56N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-RQV398	WO-2024183798-A1_CPD-374	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC3(C2)CC(C(=O)NC2CC4(CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C2)C3)n1	C49H60N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-HMWALQ	WO-2024183798-A1_CPD-375	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC(C(=O)NC3CC4(CCN(c5ccc(N/C(C)=N/c6c(C=N)c(C)c(C(C)=O)c(=O)n6C6CCCC6)nc5)CC4)C3)C2)n1	C47H60N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-W6OLQJ	WO-2024183798-A1_CPD-376	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC3(C2)CC(C(=O)N2CC(C4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C2)C3)n1	C49H60N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-S1JQE4	WO-2024183798-A1_CPD-377	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NC(C)C5CC(Nc6nc(NC(C)C)ccc6C(=O)Nc6cc(C)on6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H57N13O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-N36Q2L	WO-2024183798-A1_CPD-378	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCC5(CN(C(=O)C6CC7(CC(Nc8nc(C)ccc8C(=O)Nc8ccc(N(C)C)nn8)C7)C6)C5)C4)cn3)nc2n(C2CCCC2)c1=O	C47H55N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-GTRZQG	WO-2024183798-A1_CPD-379	.	Cc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC3(C2)CC(C(=O)N2CCC4(CCN(c5ccc(Nc6ncc7c(C)c(C=O)c(=O)n(C8CCCC8)c7n6)nc5)C4)C2)C3)n1	C47H55N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-7XITP5	WO-2024183798-A1_CPD-380	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCC5(CCN(C(=O)C6CC7(CC(Nc8nc(C)ccc8C(=O)Nc8ccc(N(C)C)nn8)C7)C6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C49H59N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-XBJERE	WO-2024183798-A1_CPD-381	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC(C(=O)N3CCC4(CCN(c5ccc(Nc6ncc7c(n6)N(C6CCCC6)C(=O)C(C(C)=O)C7C)nc5)CC4)C3)C2)n1	C46H58N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-Z30VWH	WO-2024183798-A1_CPD-382	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCC(NCC(=O)NC5CC(Nc6nc(NC(C)C)ccc6C(=O)Nc6ccc(N(C)C)nn6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C46H59N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-FJ6K7B	WO-2024183798-A1_CPD-383	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(C)CC(=O)N5CCC6(CC5)CC6Nc5nc(C)ccc5C(=O)Nc5ccc(N(C)C)nn5)CC4)cn3)nc2n(C2CCCC2)c1=O	C48H60N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-2QJ00I	WO-2024183798-A1_CPD-384	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCC5(CCN(CC(=O)N6CC7(CC(Nc8nc(C)ccc8C(=O)Nc8ccc(N(C)C)nn8)C7)C6)C5)C4)cn3)nc2n(C2CCCC2)c1=O	C48H58N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-6BVQRQ	WO-2024183798-A1_CPD-385	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CCC(C(=O)N3CCC4(CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)CC2)n1	C48H60N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-M1BK2B	WO-2024183798-A1_CPD-386	.	C=C(C)c1c(C)c2cnc(Nc3ccc(CC4CCN(CC(=O)N5CCC(Nc6nc(NC(C)C)ccc6C(=O)Nc6ccc(N(C)C)nn6)CC5)CC4)cn3)cc2n(C2CCCC2)c1=O	C50H65N13O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-5PRL4C	WO-2024183798-A1_CPD-387	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NC(C)(C)C5CC(Nc6nc(NC(C)C)ccc6C(=O)Nc6cc(C)n(C)n6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H62N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-1F3SOL	WO-2024183798-A1_CPD-388	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nc2)c(NC2CC(C(=O)NC3CCC4(CC3)CCN(c3ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc3)CC4)C2)n1	C49H61N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-XQM729	WO-2024183798-A1_CPD-389	.	CC(=O)c1c(C)c2cnc(Nc3ccc(C4CCC(NCC(=O)N5CCC(Nc6nc(NC(C)C)ccc6C(=O)Nc6ccc(N(C)C)nn6)CC5)CC4)cn3)nc2n(C2CCCC2)c1=O	C48H62N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-UJTAUA	WO-2024183798-A1_CPD-390	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCC(N5CC(C(=O)N6CCC(Nc7nc(NC(C)C)ccc7C(=O)Nc7ccc(N(C)C)nn7)CC6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C49H63N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-LIW262	WO-2024183798-A1_CPD-391	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCC(N5CC(C(=O)N6CC7(CC(Nc8nc(NC(C)C)ccc8C(=O)Nc8ccc(N(C)C)nn8)C7)C6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C50H63N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-LQLSU1	WO-2024183798-A1_CPD-392	.	CC(=O)c1c(C)c2cnc(Nc3ccc(CN4CCC(CC(=O)N5CCC(Nc6nc(NC(C)C)ccc6C(=O)Nc6ccc(N(C)C)nn6)CC5)CC4)cn3)nc2n(C2CCCC2)c1=O	C48H62N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-ZUBTTH	WO-2024183798-A1_CPD-393	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCC(N5CC(C(=O)NC6CC7(C6)CC(Nc6nc(NC(C)C)ccc6C(=O)Nc6ccc(N(C)C)nn6)C7)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C51H65N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-GMPI6S	WO-2024183798-A1_CPD-394	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCC(N5CCC(C(=O)N6CC(Nc7nc(NC(C)C)ccc7C(=O)Nc7ccc(N(C)C)nn7)C6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C48H61N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-I24OJU	WO-2024183798-A1_CPD-395	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCC(N5CCC(C(=O)N6CCC(Nc7nc(NC(C)C)ccc7C(=O)Nc7ccc(N(C)C)nn7)C6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C49H63N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-VWV6SI	WO-2024183798-A1_CPD-396	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCC(N5CCC(C(=O)N6CCC(Nc7nc(NC(C)C)ccc7C(=O)Nc7ccc(N(C)C)nn7)CC6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C50H65N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-I6V9KT	WO-2024183798-A1_CPD-397	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCC(N5CCC(C(=O)NC6CC7(C6)CC(Nc6nc(NC(C)C)ccc6C(=O)Nc6ccc(N(C)C)nn6)C7)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C52H67N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-TFS7UG	WO-2024183798-A1_CPD-398	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCC(N5CCC(C(=O)N6CC7(CC(Nc8nc(NC(C)C)ccc8C(=O)Nc8ccc(N(C)C)nn8)C7)C6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C51H65N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-K2S1KQ	WO-2024183798-A1_CPD-399	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C5CCN(C(=O)[C@H]6CC[C@H](Nc7nc(NC(C)C)ccc7C(=O)Nc7ccc(N(C)C)nn7)CC6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C50H65N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-CNPZG3	WO-2024183798-A1_CPD-4	.	CNc1ccc(C(=O)Nc2nc(C)c(C)s2)c(NCCCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)n1	C45H59N13O4S	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-CVZ8KG	WO-2024183798-A1_CPD-400	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C5CCN(C(=O)C6CC7(CC(Nc8nc(NC(C)C)ccc8C(=O)Nc8ccc(N(C)C)nn8)C7)C6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C51H65N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-D59VJX	WO-2024183798-A1_CPD-401	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C5CN(C(=O)C6CC7(CC(Nc8nc(NC(C)C)ccc8C(=O)Nc8ccc(N(C)C)nn8)C7)C6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C50H63N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-60AXYR	WO-2024183798-A1_CPD-402	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C5CCN(C(=O)C6CC(Nc7nc(NC(C)C)ccc7C(=O)Nc7ccc(N(C)C)nn7)C6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C48H61N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-QFQGEU	WO-2024183798-A1_CPD-403	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C5CCN(C(=O)[C@H]6CC[C@@H](Nc7nc(NC(C)C)ccc7C(=O)Nc7ccc(N(C)C)nn7)C6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C49H63N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-7L5FKS	WO-2024183798-A1_CPD-404	.	CC(=O)c1c(C)c2cnc(N(C)c3ccc(N4CCN(CCC(=O)N5CC6(CC(Nc7nc(NC(C)C)ccc7C(=O)Nc7cc(C)n(C)n7)C6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C48H62N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-WM9GAT	WO-2024183798-A1_CPD-405	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(C)C(=O)NC5CC6(C5)CC(Nc5nc(C)ccc5C(=O)Nc5cn(C)c(C7CC7)n5)C6)CC4)cn3)cc2n(C2CCCC2)c1=O	C49H60N12O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-3GF1XR	WO-2024183798-A1_CPD-406	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(C)C(=O)NC5CC6(C5)CC(Nc5nc(NC(C)C)ccc5C(=O)Nc5ccc(CN(C)C)nn5)C6)CC4)cn3)nc2n(C2CCCC2)c1=O	C50H65N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-Q0OI8Q	WO-2024183798-A1_CPD-407	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCC5(CC4)CC5C(=O)N4CCC(Nc5nc(NC(C)C)ccc5C(=O)Nc5ccc(N(C)C)nn5)CC4)cn3)nc2n(C2CCCC2)c1=O	C48H60N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-7HTRDV	WO-2024183798-A1_CPD-408	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCC5(CC4)CC5C(=O)N4CCC(Nc5nc(NC(C)C)ccc5C(=O)Nc5cc(C)n(C)n5)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H59N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-Q5IORA	WO-2024183798-A1_CPD-409	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCC5(CC4)CC5C(=O)N4CCC(Nc5nc(NC(C)C)ccc5C(=O)Nc5cn(C)c(C6CC6)n5)CC4)cn3)nc2n(C2CCCC2)c1=O	C49H61N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-CTO54S	WO-2024183798-A1_CPD-410	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NC(C)(C)C5CC(Nc6nc(NC(C)C)ccc6C(=O)Nc6cc(C)on6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C46H59N13O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-H149EB	WO-2024183798-A1_CPD-411	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCC5(CC4)CC5C(=O)N4CC5(CC(Nc6nc(NC(C)C)ccc6C(=O)Nc6ccc(N(C)C)nn6)C5)C4)cn3)nc2n(C2CCCC2)c1=O	C49H60N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-8HBYE0	WO-2024183798-A1_CPD-412	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCC5(CC4)CC5C(=O)N4CC5(CC(Nc6nc(NC(C)C)ccc6C(=O)Nc6cn(C)c(C7CC7)n6)C5)C4)cn3)nc2n(C2CCCC2)c1=O	C50H61N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-O9BW6T	WO-2024183798-A1_CPD-413	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCC5(CC4)CC5C(=O)NC4CC(Nc5nc(NC(C)C)ccc5C(=O)Nc5ccc(N(C)C)nn5)C4)cn3)nc2n(C2CCCC2)c1=O	C47H58N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-1FJTNN	WO-2024183798-A1_CPD-414	.	CC(=O)c1c(C)c2ccc(Nc3ccc(N4CCC5(CC4)CC5C(=O)NC4CC5(C4)CC(Nc4nc(NC(C)C)ccc4C(=O)Nc4ccc(N(C)C)nn4)C5)cn3)nc2n(C2CCCC2)c1=O	C51H63N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-JPDEH2	WO-2024183798-A1_CPD-415	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCC5(CC4)CC5C(=O)N4CC5(CC(Nc6nc(NC(C)C)ccc6C(=O)Nc6cc(C)n(C)n6)C5)C4)cn3)nc2n(C2CCCC2)c1=O	C48H59N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-AKVHGX	WO-2024183798-A1_CPD-416	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CCC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C47H59N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-C4JQS4	WO-2024183798-A1_CPD-417	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCC5(CC4)CC5C(=O)NC4CCC(Nc5nc(NC(C)C)ccc5C(=O)Nc5ccc(N(C)C)nn5)C4)cn3)nc2n(C2CCCC2)c1=O	C48H60N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-P2YZQJ	WO-2024183798-A1_CPD-418	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CC5(CN(CC(=O)N6CCC(Nc7nc(NC(C)C)ccc7C(=O)Nc7ccc(N(C)C)nn7)CC6)C5)C4)cn3)nc2n(C2CCCC2)c1=O	C47H59N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-RSBBAF	WO-2024183798-A1_CPD-419	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCC5(CC4)CC5C(=O)N4CCC(Nc5nc(NC(C)C)ccc5C(=O)Nc5cc(C)on5)CC4)cn3)nc2n(C2CCCC2)c1=O	C46H56N12O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-4ML2YB	WO-2024183798-A1_CPD-420	.	CC(=O)c1c(C)c2cnc(Nc3ccc(CN4CCN(CC(=O)N5CCC(Nc6nc(NC(C)C)ccc6C(=O)Nc6cn(C)c(C7CC7)n6)CC5)CC4)cn3)nc2n(C2CCCC2)c1=O	C48H62N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-IYSS31	WO-2024183798-A1_CPD-421	.	CC(=O)c1c(C)c2cnc(Nc3ccc(CN4CCN(CC(=O)N5CCC(Nc6nc(NC(C)C)ccc6C(=O)Nc6cc(C)n(C)n6)CC5)CC4)cn3)nc2n(C2CCCC2)c1=O	C46H60N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-I02TX6	WO-2024183798-A1_CPD-422	.	CC(=O)c1c(C)c2cnc(Nc3ccc(CN4CCN(CC(=O)N5CC6(CC(Nc7nc(NC(C)C)ccc7C(=O)Nc7ccc(N(C)C)nn7)C6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C48H61N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-FE172G	WO-2024183798-A1_CPD-423	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CC5(CN(CC(=O)N6CC7(CC(Nc8nc(NC(C)C)ccc8C(=O)Nc8ccc(N(C)C)nn8)C7)C6)C5)C4)cn3)nc2n(C2CCCC2)c1=O	C48H59N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-DKQQVL	WO-2024183798-A1_CPD-424	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CC5(CN(CC(=O)N6CCC(Nc7nc(NC(C)C)ccc7C(=O)Nc7ccc(N(C)C)nn7)C6)C5)C4)cn3)nc2n(C2CCCC2)c1=O	C46H57N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-RVIU8U	WO-2024183798-A1_CPD-425	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCC(N(C)CC(=O)N5CC6(CC(Nc7nc(NC(C)C)ccc7C(=O)Nc7ccc(N(C)C)nn7)C6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C49H63N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-X4PKKR	WO-2024183798-A1_CPD-426	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCC(N(C)CC(=O)N5CCC(Nc6nc(NC(C)C)ccc6C(=O)Nc6ccc(N(C)C)nn6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H61N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-YPK78R	WO-2024183798-A1_CPD-427	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCC(N(C)CC(=O)N5CC(Nc6nc(NC(C)C)ccc6C(=O)Nc6ccc(N(C)C)nn6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C46H59N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-GFP5F8	WO-2024183798-A1_CPD-428	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC(C(=O)NC3CCC4(CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C47H58N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-RHIWI4	WO-2024183798-A1_CPD-429	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NCC56CC(Nc7nc(NC(C)C)ccc7C(=O)Nc7ccc(N(C)C)nn7)(C5)C6)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H59N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-U99LY5	WO-2024183798-A1_CPD-430	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CCC(N(C)C(=O)CN3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)C2)n1	C45H57N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-8LDMZT	WO-2024183798-A1_CPD-431	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(C)CC(=O)N5CCC(Nc6nc(NC(C)C)ccc6C(=O)Nc6cn(C)c(C7CC7)n6)CC5)CC4)cn3)nc2n(C2CCCC2)c1=O	C49H64N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-TZARCQ	WO-2024183798-A1_CPD-432	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CCC(=O)N5CC6(CC(Nc7nc(C)ccc7C(=O)Nc7ccc(N(C)C)nn7)C6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C46H56N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-YJZ0S9	WO-2024183798-A1_CPD-433	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(CC(=O)N5CC6(CC(Nc7nc(NC(C)C)ccc7C(=O)Nc7cc(C)n(C)n7)C6)C5)C(F)(F)F)CC4)cn3)nc2n(C2CCCC2)c1=O	C48H59F3N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-6YHHBW	WO-2024183798-A1_CPD-434	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(CF)CC(=O)N5CC6(CC(Nc7nc(C)ccc7C(=O)Nc7cc(C)n(C)n7)C6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C46H56FN13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-0PBWOD	WO-2024183798-A1_CPD-435	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(CC(=O)N5CC6(CC(Nc7nc(C)ccc7C(=O)Nc7cn(C)c(C8CC8)n7)C6)C5)C(F)(F)F)CC4)cn3)nc2n(C2CCCC2)c1=O	C48H56F3N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-INFE3F	WO-2024183798-A1_CPD-436	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(CC(=O)N5CC6(CC(Nc7nc(NC(C)C)ccc7C(=O)Nc7cn(C)c(C8CC8)n7)C6)C5)C(F)(F)F)CC4)cn3)nc2n(C2CCCC2)c1=O	C50H61F3N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-EV6AUZ	WO-2024183798-A1_CPD-437	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCC5(CC4)CC(C(=O)NC4CC6(C4)CC(Nc4nc(NC(C)C)ccc4C(=O)Nc4ccc(N(C)C)nn4)C6)C5)cn3)nc2n(C2CCCC2)c1=O	C51H64N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-77O547	WO-2024183798-A1_CPD-438	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(C)C(=O)NC5CC6(C5)CC(Nc5nc(C)ccc5C(=O)Nc5ccc(N(C)C)nn5)C6)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H58N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-ONR0OA	WO-2024183798-A1_CPD-439	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCC5(CC4)CC5C(=O)NC4CC5(C4)CC(Nc4nc(C)ccc4C(=O)Nc4ccc(N(C)C)nn4)C5)cn3)nc2n(C2CCCC2)c1=O	C48H57N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-PEORV0	WO-2024183798-A1_CPD-440	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NC5CC6(C5)CC(Nc5nc(NC(C)C)ccc5C(=O)Nc5cc7n(n5)CCC7)C6)CC4)cn3)nc2n(C2CCCC2)c1=O	C48H60N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-53VKIT	WO-2024183798-A1_CPD-441	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCC5(CCN(CC(=O)N6CCC(Nc7nc(C)ccc7C(=O)Nc7ccc(N(C)C)nn7)CC6)C5)C4)cn3)nc2n(C2CCCC2)c1=O	C47H58N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-6IRWSE	WO-2024183798-A1_CPD-442	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCC5(CCN(CC(=O)N6CC(Nc7nc(C)ccc7C(=O)Nc7ccc(N(C)C)nn7)C6)C5)C4)cn3)nc2n(C2CCCC2)c1=O	C45H54N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-4MDJHJ	WO-2024183798-A1_CPD-443	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCC5(CCN(CC(=O)N6CC7(CC(Nc8nc(C)ccc8C(=O)Nc8cn(C)c(C9CC9)n8)C7)C6)C5)C4)cn3)nc2n(C2CCCC2)c1=O	C49H59N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-Y7R2LO	WO-2024183798-A1_CPD-444	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCC5(CCN(CC(=O)N6CC7(CC(Nc8nc(NC(C)C)ccc8C(=O)Nc8cn(C)c(C9CC9)n8)C7)C6)C5)C4)cn3)nc2n(C2CCCC2)c1=O	C51H64N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-189WOS	WO-2024183798-A1_CPD-445	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCC5(CCN(CC(=O)NCC6CC(Nc7nc(C)ccc7C(=O)Nc7ccc(N(C)C)nn7)C6)C5)C4)cn3)nc2n(C2CCCC2)c1=O	C47H58N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-16QQVW	WO-2024183798-A1_CPD-446	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCC5(CCN(CC(=O)N6CC7(CC(Nc8nc(NC(C)C)ccc8C(=O)Nc8cc(C)n(C)n8)C7)C6)C5)C4)cn3)nc2n(C2CCCC2)c1=O	C49H62N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-G586CL	WO-2024183798-A1_CPD-447	.	C=C(C)c1c(C)c2cnc(Nc3ccc(N4CCC5(CCN(CC(=O)N6CC7(CC(Nc8nc(C)ccc8C(=O)Nc8cc(C)n(C)n8)C7)C6)C5)C4)cn3)nc2n(C2CCCC2)c1=O	C48H59N13O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-18D0LM	WO-2024183798-A1_CPD-448	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCC5(CCN(CC(=O)N6CC7(CC(Nc8nc(NC(C)C)ccc8C(=O)Nc8ccc(N(C)C)nn8)C7)C6)C5)C4)cn3)nc2n(C2CCCC2)c1=O	C50H63N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-135J47	WO-2024183798-A1_CPD-449	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCC5(CCN(CC(=O)NC6CC7(C6)CC(Nc6nc(C)ccc6C(=O)Nc6ccc(N(C)C)nn6)C7)C5)C4)cn3)nc2n(C2CCCC2)c1=O	C49H60N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-MC38UA	WO-2024183798-A1_CPD-450	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCC5(CCN(CC(=O)NC6CC(Nc7nc(C)ccc7C(=O)Nc7ccc(N(C)C)nn7)C6)C5)C4)cn3)nc2n(C2CCCC2)c1=O	C46H56N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-C2P5UK	WO-2024183798-A1_CPD-451	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCC5(CC4)CC5C(=O)NC4CC5(C4)CC(Nc4nc(NC(C)C)ccc4C(=O)Nc4cc(C)n(C)n4)C5)cn3)nc2n(C2CCCC2)c1=O	C49H61N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-KAC7WN	WO-2024183798-A1_CPD-452	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NC5CC6(C5)CC(Nc5nc(NC(C)C)ccc5C(=O)Nc5cc(C)n(C7CC7)n5)C6)CC4)cn3)nc2n(C2CCCC2)c1=O	C49H62N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-S7BTXD	WO-2024183798-A1_CPD-453	.	COc1cccc(NC(=O)c2ccc(NC(C)C)nc2NC2CC3(CC(NC(=O)CN4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C48H59N13O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-OLX7NV	WO-2024183798-A1_CPD-454	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CC5(CN(CCC(=O)N6CCC(Nc7nc(NC(C)C)ccc7C(=O)Nc7ccc(N(C)C)nn7)CC6)C5)C4)cn3)nc2n(C2CCCC2)c1=O	C48H61N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-8KXPO0	WO-2024183798-A1_CPD-455	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CC5(CN(CCC(=O)N6CC7(CC(Nc8nc(NC(C)C)ccc8C(=O)Nc8ccc(N(C)C)nn8)C7)C6)C5)C4)cn3)nc2n(C2CCCC2)c1=O	C49H61N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-Q1QV6W	WO-2024183798-A1_CPD-456	.	CC(=O)c1c(C)c2cnc(Nc3ccc(CN4CCN(C(C)C(=O)N5CC6(CC(Nc7nc(C)ccc7C(=O)Nc7ccc(N(C)C)nn7)C6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H58N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-8I8K3A	WO-2024183798-A1_CPD-457	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCC5(CC4)CC5C(=O)NC4CC5(C4)CC(Nc4nc(NC(C)C)ccc4C(=O)Nc4cn(C)c(C6CC6)n4)C5)cn3)nc2n(C2CCCC2)c1=O	C51H63N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-DODCBF	WO-2024183798-A1_CPD-458	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CCC(=O)N5CC6(CC(Nc7nc(C)ccc7C(=O)Nc7ccc(N(C)C)nn7)C6)C5)C(C)(C)C4)cn3)nc2n(C2CCCC2)c1=O	C48H60N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-GCXLSM	WO-2024183798-A1_CPD-459	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CCC(=O)N5CC6(CC(Nc7nc(NC(C)C)ccc7C(=O)Nc7ccc(N(C)C)nn7)C6)C5)C(C)(C)C4)cn3)nc2n(C2CCCC2)c1=O	C50H65N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-5U5DLU	WO-2024183798-A1_CPD-460	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCC(N5CCC(C(=O)NC6CC(Nc7nc(NC(C)C)ccc7C(=O)Nc7ccc(N(C)C)nn7)C6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C49H63N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-SDEMUS	WO-2024183798-A1_CPD-461	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCC(N5CCC(C(=O)NCC6CC(Nc7nc(NC(C)C)ccc7C(=O)Nc7ccc(CN(C)C)nn7)C6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C51H67N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-8NM1T0	WO-2024183798-A1_CPD-462	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCC(N5CCC(C(=O)NC6CCC(Nc7nc(NC(C)C)ccc7C(=O)Nc7ccc(N(C)C)nn7)CC6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C51H67N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-U6RC83	WO-2024183798-A1_CPD-463	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCC(N(C)CC(=O)N5CCC(Nc6nc(C)ccc6C(=O)Nc6ccc(N(C)C)nn6)CC5)CC4)cn3)nc2n(C2CCCC2)c1=O	C46H58N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-A5LU1S	WO-2024183798-A1_CPD-464	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCC(N(C)CC(=O)N5CC6(CC(Nc7nc(C)ccc7C(=O)Nc7ccc(N(C)C)nn7)C6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H58N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-RP74CV	WO-2024183798-A1_CPD-465	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCC(NCC(=O)N5CCC(Nc6nc(NC(C)C)ccc6C(=O)Nc6cc(C)n(C)n6)CC5)CC4)cn3)nc2n(C2CCCC2)c1=O	C46H60N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-0LLBEB	WO-2024183798-A1_CPD-466	.	CC(=O)c1c(C)c2ccc(Nc3ccc(N4CCC(N(C)CC(=O)N5CCC(Nc6nc(NC(C)C)ccc6C(=O)Nc6cn(C)c(C7CC7)n6)CC5)CC4)cn3)nc2n(C2CCCC2)c1=O	C50H65N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-09POP9	WO-2024183798-A1_CPD-467	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CC5(CN(CC(=O)NC6CC7(C6)CC(Nc6nc(NC(C)C)ccc6C(=O)Nc6ccc(N(C)C)nn6)C7)C5)C4)cn3)nc2n(C2CCCC2)c1=O	C49H61N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-VVNING	WO-2024183798-A1_CPD-468	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CC5(CN(CC(=O)NCC6CC(Nc7nc(NC(C)C)ccc7C(=O)Nc7ccc(N(C)C)nn7)C6)C5)C4)cn3)nc2n(C2CCCC2)c1=O	C47H59N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-DYWPW3	WO-2024183798-A1_CPD-469	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C5CCN(C(=O)N6CCC(Nc7nc(NC(C)C)ccc7C(=O)Nc7ccc(N(C)C)nn7)CC6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C49H64N16O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-41C46G	WO-2024183798-A1_CPD-470	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C5CCN(C(=O)NC6CC7(C6)CC(Nc6nc(NC(C)C)ccc6C(=O)Nc6ccc(N(C)C)nn6)C7)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C51H66N16O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-OLG5D0	WO-2024183798-A1_CPD-471	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C5CCN(C(=O)C6CC(Nc7nc(C)ccc7C(=O)Nc7ccc(N(C)C)nn7)C6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C46H56N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-9PSEP6	WO-2024183798-A1_CPD-472	.	CC(=O)c1c(C)c2cnc(Nc3ccc(CN4CCN(CC(=O)NC5CC6(C5)CC(Nc5nc(NC(C)C)ccc5C(=O)Nc5ccc(N(C)C)nn5)C6)CC4)cn3)nc2n(C2CCCC2)c1=O	C49H63N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-R1EDCO	WO-2024183798-A1_CPD-473	.	CC(=O)c1c(C)c2cnc(Nc3ccc(CN4CCN(CC(=O)NC5CCC(Nc6nc(NC(C)C)ccc6C(=O)Nc6ccc(N(C)C)nn6)CC5)CC4)cn3)nc2n(C2CCCC2)c1=O	C48H63N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-DBOIO1	WO-2024183798-A1_CPD-474	.	CC(=O)c1c(C)c2ccc(Nc3ccc(CN4CCN(CC(=O)N5CCC(Nc6nc(C)ccc6C(=O)Nc6ccc(N(C)C)nn6)CC5)CC4)cn3)nc2n(C2CCCC2)c1=O	C46H57N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-5MHUPH	WO-2024183798-A1_CPD-475	.	CC(=O)c1c(C)c2cnc(Nc3ccc(CN4CCN(CC(=O)NC5CC(Nc6nc(NC(C)C)ccc6C(=O)Nc6ccc(N(C)C)nn6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C46H59N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-8ZQ4NX	WO-2024183798-A1_CPD-476	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C5CCN(C(=O)[C@H]6CC[C@H](Nc7nc(C)ccc7C(=O)Nc7ccc(N(C)C)nn7)CC6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C48H60N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-JL2PT2	WO-2024183798-A1_CPD-477	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C5CCN(C(=O)[C@H]6CC[C@H](Nc7nc(C)ccc7C(=O)Nc7cc(C)n(C)n7)CC6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H59N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-IWLGCG	WO-2024183798-A1_CPD-478	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C5CCN(C(=O)[C@H]6CC[C@H](Nc7nc(NC(C)C)ccc7C(=O)Nc7cc(C)n(C)n7)CC6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C49H64N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-103KSR	WO-2024183798-A1_CPD-479	.	CC(=O)c1c(C)c2cnc(Nc3ccc(CN4CCN(CC(=O)NCC56CC(Nc7nc(NC(C)C)ccc7C(=O)Nc7ccc(N(C)C)nn7)(C5)C6)CC4)cn3)nc2n(C2CCCC2)c1=O	C48H61N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-2PJY67	WO-2024183798-A1_CPD-480	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C5CCN(C(=O)[C@H]6CC[C@H](Nc7nc(C)ccc7C(=O)Nc7cn(C)c(C8CC8)n7)CC6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C49H61N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-9GXUIB	WO-2024183798-A1_CPD-481	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C5CCN(C(=O)[C@H]6CC[C@H](Nc7nc(NC(C)C)ccc7C(=O)Nc7cn(C)c(C8CC8)n7)CC6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C51H66N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-OO09RL	WO-2024183798-A1_CPD-482	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C5CCN(C(=O)N6CCC(Nc7nc(C)ccc7C(=O)Nc7ccc(N(C)C)nn7)CC6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H59N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-WM6S6J	WO-2024183798-A1_CPD-483	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C5CCN(C(=O)NC6CCC(Nc7nc(NC(C)C)ccc7C(=O)Nc7ccc(N(C)C)nn7)CC6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C50H66N16O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-DMY451	WO-2024183798-A1_CPD-484	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CC5(CC(N(C)CC(=O)N6CCC(Nc7nc(NC(C)C)ccc7C(=O)Nc7ccc(N(C)C)nn7)CC6)C5)C4)cn3)nc2n(C2CCCC2)c1=O	C49H63N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-TR7NU0	WO-2024183798-A1_CPD-485	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCC5(CCN(CC(=O)NCC67CC(Nc8nc(NC(C)C)ccc8C(=O)Nc8ccc(N(C)C)nn8)(C6)C7)C5)C4)cn3)nc2n(C2CCCC2)c1=O	C50H63N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-JJDWEP	WO-2024183798-A1_CPD-486	.	CC(=O)c1c(C)c2cnc(Nc3ccc(CN4CCC(NC(=O)C5CC6(CC(Nc7nc(NC(C)C)ccc7C(=O)Nc7ccc(N(C)C)nn7)C6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C49H62N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-PCXBNT	WO-2024183798-A1_CPD-487	.	CC(=O)c1c(C)c2cnc(Nc3ccc(CN4CCN(CC(=O)N5CCC6(CCC(Nc7nc(NC(C)C)ccc7C(=O)Nc7ccc(N(C)C)nn7)C6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C50H65N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-FLDPTT	WO-2024183798-A1_CPD-488	.	CC(=O)c1c(C)c2cnc(Nc3ccc(C(C)N4CCN(CC(=O)N5CC6(CC(Nc7nc(C)ccc7C(=O)Nc7ccc(N(C)C)nn7)C6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H58N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-Q43X2N	WO-2024183798-A1_CPD-489	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CC5(CN(CC(=O)N6CC7(CC(Nc8nc(C)ccc8C(=O)Nc8ccc(N(C)C)nn8)C7)C6)C5)C4)cn3)nc2n(C2CCCC2)c1=O	C46H54N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-KCBW9K	WO-2024183798-A1_CPD-490	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CC5(CN(CC(=O)N6CCC(Nc7nc(C)ccc7C(=O)Nc7ccc(N(C)C)nn7)CC6)C5)C4)cn3)nc2n(C2CCCC2)c1=O	C45H54N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-WKLRWY	WO-2024183798-A1_CPD-491	.	CC(=O)c1c(C)c2cnc(Nc3ccc(CN4CCN(C(=O)CN5CCC(Nc6nc(C)ccc6C(=O)Nc6ccc(N(C)C)nn6)CC5)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H56N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-60ENBW	WO-2024183798-A1_CPD-492	.	CCc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(N[C@H]2CC[C@H](C(=O)N3CCC(N4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)CC2)n1	C49H62N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-S6Z3FW	WO-2024183798-A1_CPD-493	.	CC(=O)c1c(C)c2cnc(Nc3ccc(CN4CCN(CC(=O)NCC5CC(Nc6nc(NC(C)C)ccc6C(=O)Nc6ccc(N(C)C)nn6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H61N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-019R8S	WO-2024183798-A1_CPD-494	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C5CCN(C(=O)NC6CC(Nc7nc(C)ccc7C(=O)Nc7ccc(N(C)C)nn7)C6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C46H57N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-KYCEE3	WO-2024183798-A1_CPD-495	.	CC(=O)c1c(C)c2cnc(Nc3ccc(CN4CCN(C(=O)[C@H]5CC[C@H](Nc6nc(C)ccc6C(=O)Nc6ccc(N(C)C)nn6)CC5)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H55N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-JRSTI6	WO-2024183798-A1_CPD-496	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCC5(CCN(CC(=O)NC67CC(Nc8nc(NC(C)C)ccc8C(=O)Nc8ccc(N(C)C)nn8)(C6)C7)C5)C4)cn3)nc2n(C2CCCC2)c1=O	C49H61N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-NNQ1GS	WO-2024183798-A1_CPD-497	.	CC(=O)c1c(C)c2cnc(Nc3ccc(CN4CC5(C4)CN(C(=O)CN4CC6(CC(Nc7nc(NC(C)C)ccc7C(=O)Nc7ccc(N(C)C)nn7)C6)C4)C5)cn3)nc2n(C2CCCC2)c1=O	C49H61N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-6DX4MB	WO-2024183798-A1_CPD-498	.	CC(=O)c1c(C)c2cnc(Nc3ccc(CN4CC5(C4)CN(C(=O)CN4CCC(Nc6nc(NC(C)C)ccc6C(=O)Nc6ccc(N(C)C)nn6)CC4)C5)cn3)nc2n(C2CCCC2)c1=O	C48H61N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-OFN85L	WO-2024183798-A1_CPD-499	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C5CCN(C(=O)C6CCC(Nc7nc(C(C)C)ccc7C(=O)Nc7ccc(N(C)C)nn7)CC6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C50H64N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-FB07LU	WO-2024183798-A1_CPD-5	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)n1	C44H57N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-OPKLCV	WO-2024183798-A1_CPD-500	.	COc1ccc(NC(=O)c2ccc(NC(C)C)nc2N[C@H]2CC[C@H](C(=O)N3CCC(N4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)CC2)nn1	C49H62N14O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-JXA9I4	WO-2024183798-A1_CPD-501	.	CC(=O)c1c(C)c2cnc(Nc3ccc(CN4CCN(CC(=O)NC5CCC(Nc6nc(NC(C)C)ccc6C(=O)Nc6ccc(N(C)C)nn6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H61N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-S25ONW	WO-2024183798-A1_CPD-502	.	CC(=O)c1c(C)c2cnc(Nc3ccc(CN4CCN(CC(=O)NC56CC(Nc7nc(NC(C)C)ccc7C(=O)Nc7ccc(N(C)C)nn7)(C5)C6)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H59N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-D625VX	WO-2024183798-A1_CPD-503	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CCC(=O)NC56CC(Nc7nc(NC(C)C)ccc7C(=O)Nc7ccc(N(C)C)nn7)(C5)C6)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H59N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-S6QI0G	WO-2024183798-A1_CPD-504	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(C)CC(=O)NC56CC(Nc7nc(NC(C)C)ccc7C(=O)Nc7ccc(N(C)C)nn7)(C5)C6)CC4)cn3)nc2n(C2CCCC2)c1=O	C48H61N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-Q9MPSK	WO-2024183798-A1_CPD-505	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCC(N(C)CC(=O)NC56CC(Nc7nc(NC(C)C)ccc7C(=O)Nc7ccc(N(C)C)nn7)(C5)C6)CC4)cn3)nc2n(C2CCCC2)c1=O	C48H61N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-DOB6MF	WO-2024183798-A1_CPD-506	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CCCNC(=O)C56CC(Nc7nc(NC(C)C)ccc7C(=O)Nc7ccc(N(C)C)nn7)(C5)C6)CC4)cn3)nc2n(C2CCCC2)c1=O	C48H61N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-IF8JJX	WO-2024183798-A1_CPD-507	.	CC(=O)c1c(C)c2cnc(Nc3ccc(CN4CCC5(CCN(C(=O)CN6CC7(CC(Nc8nc(C)ccc8C(=O)Nc8ccc(N(C)C)nn8)C7)C6)C5)C4)cn3)nc2n(C2CCCC2)c1=O	C49H60N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-3G2U7N	WO-2024183798-A1_CPD-508	.	CC(=O)c1c(C)c2cnc(Nc3ccc(CN4CC5(CN(CC(=O)N6CC7(CC(Nc8nc(NC(C)C)ccc8C(=O)Nc8ccc(N(C)C)nn8)C7)C6)C5)C4)cn3)nc2n(C2CCCC2)c1=O	C49H61N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-J0L3NI	WO-2024183798-A1_CPD-509	.	C=C(C)c1c(C)c2cnc(Nc3ccc(CN4CC5(CN(CC(=O)N6CCC(Nc7nc(NC(C)C)ccc7C(=O)Nc7ccc(N(C)C)nn7)CC6)C5)C4)cn3)nc2n(C2CCCC2)c1=O	C49H63N15O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-R35Z7J	WO-2024183798-A1_CPD-510	.	CC(=O)c1c(C)c2cnc(Nc3ccc(CN4CCN(C5CCN(C(=O)C6CC(Nc7nc(NC(C)C)ccc7C(=O)Nc7ccc(N(C)C)nn7)C6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C49H63N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-P4HPHU	WO-2024183798-A1_CPD-511	.	CC(=O)c1c(C)c2cnc(Nc3ccc(CN4CCN(C5CCN(C(=O)C6CCC(Nc7nc(NC(C)C)ccc7C(=O)Nc7ccc(N(C)C)nn7)C6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C50H65N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-U4RUTX	WO-2024183798-A1_CPD-512	.	CC(=O)c1c(C)c2cnc(Nc3ccc(CN4CCN(C5CCN(C(=O)[C@H]6CC[C@H](Nc7nc(NC(C)C)ccc7C(=O)Nc7ccc(N(C)C)nn7)CC6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C51H67N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-N0O2GQ	WO-2024183798-A1_CPD-513	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CN(CC(=O)N3CCN(Cc4ccc(Nc5ncc6cc(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)C2)n1	C42H51N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-NIQNCW	WO-2024183798-A1_CPD-514	.	CC(=O)c1cc2cnc(Nc3ccc(N4CCN(CC(=O)NC5CC6(C5)CC(Nc5nc(NC(C)C)ccc5C(=O)Nc5cc(C)n(C(F)(F)F)n5)C6)CC4)cn3)nc2n(C2CCCC2)c1=O	C46H55F3N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-KUFHYO	WO-2024183798-A1_CPD-515	.	CC(=O)c1cc2cnc(Nc3ccc(CN4CCN(CC(=O)N5CC6(CCC(Nc7nc(NC(C)C)ccc7C(=O)Nc7ccc(N(C)C)nn7)C6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C48H61N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-O2ZB18	WO-2024183798-A1_CPD-516	.	CC(=O)c1cc2cnc(Nc3ccc(N4CCN(C5CCN(C(=O)C6(C)CCC(Nc7nc(NC(C)C)ccc7C(=O)Nc7ccc(N(C)C)nn7)CC6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C50H65N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-75SNMP	WO-2024183798-A1_CPD-517	.	CC(=O)c1cc2cnc(Nc3ccc(N4CCC(N(C)C(=O)CN5CC(Nc6nc(NC(C)C)ccc6C(=O)Nc6ccc(N(C)C)nn6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H57N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-4Q5KE8	WO-2024183798-A1_CPD-518	.	CC(=O)c1cc2cnc(Nc3ccc(N4CCN(C5CCN(C(=O)CN6CC7(CC(Nc8nc(NC(C)C)ccc8C(=O)Nc8ccc(N(C)C)nn8)C7)C6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C50H64N16O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-SO04VP	WO-2024183798-A1_CPD-519	.	CC(=O)c1cc2cnc(Nc3ccc(CN4CCC5(CCN(CC(=O)N6CC7(CC(Nc8nc(C)ccc8C(=O)Nc8ccc(N(C)C)nn8)C7)C6)C5)C4)cn3)nc2n(C2CCCC2)c1=O	C48H58N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-Y14FL8	WO-2024183798-A1_CPD-520	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C5CCN(C(=O)[C@H]6CC[C@H](Nc7nc(NC(C)C)ccc7C(=O)Nc7cc8n(n7)CCC8)CC6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C50H64N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-S56MHZ	WO-2024183798-A1_CPD-521	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C5CCN(C(=O)[C@H]6CC[C@H](Nc7nc(C)ccc7C(=O)Nc7cc8n(n7)CCC8)CC6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C48H59N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-O3ESG8	WO-2024183798-A1_CPD-522	.	COc1cccc(NC(=O)c2ccc(NC(C)C)nc2N[C@H]2CC[C@H](C(=O)N3CCC(N4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)CC2)n1	C50H63N13O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-3O8BBA	WO-2024183798-A1_CPD-523	.	COc1cccc(NC(=O)c2ccc(C)nc2N[C@H]2CC[C@H](C(=O)N3CCC(N4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)CC2)n1	C48H58N12O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-3433P6	WO-2024183798-A1_CPD-524	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(CC(=O)N5CC6(CC(Nc7nc(C)ccc7C(=O)Nc7cc8n(n7)CCC8)C6)C5)C(F)(F)F)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H54F3N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-BKN7OB	WO-2024183798-A1_CPD-525	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)N(C)CC56CC(Nc7nc(NC(C)C)ccc7C(=O)Nc7ccc(N(C)C)nn7)(C5)C6)CC4)cn3)nc2n(C2CCCC2)c1=O	C48H61N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-7SOZPV	WO-2024183798-A1_CPD-526	.	CCc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(N[C@H]2CC[C@H](C(=O)N3CCC(N4CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)CC2)c1	C50H63N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-05AFJM	WO-2024183798-A1_CPD-527	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C5CCN(C(=O)[C@H]6CC[C@H](Nc7cc(NC(C)C)ccc7C(=O)Nc7ccc(N(C)C)nn7)CC6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C51H66N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-FI5FQH	WO-2024183798-A1_CPD-528	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C5CCN(C(=O)[C@H]6CC[C@H](Nc7cc(C(C)C)ccc7C(=O)Nc7ccc(N(C)C)nn7)CC6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C51H65N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-JE7BN6	WO-2024183798-A1_CPD-529	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCC5(CCN(CC(=O)N6CC7(CC(Nc8nc(NC(C)C)ccc8C(=O)Nc8cc9n(n8)CCC9)C7)C6)C5)C4)cn3)nc2n(C2CCCC2)c1=O	C50H62N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-H8OIDH	WO-2024183798-A1_CPD-530	.	CC(=O)c1c(C)c2cnc(Nc3ccc(CN4CCN(CC(=O)N5CCC(Nc6nc(NC(C)C)ccc6C(=O)Nc6cc7n(n6)CCC7)CC5)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H60N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-YZ10U3	WO-2024183798-A1_CPD-531	.	COc1cccc(NC(=O)c2ccc(C)nc2NC2CC3(C2)CN(C(=O)CC(N2CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC2)C(F)(F)F)C3)n1	C47H53F3N12O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-P71ITX	WO-2024183798-A1_CPD-532	.	COc1cccc(NC(=O)c2ccc(NC(C)C)nc2NC2CC3(C2)CN(C(=O)CN2CCC4(CCN(c5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)C4)C2)C3)n1	C50H61N13O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-HTHQM5	WO-2024183798-A1_CPD-533	.	COC1=CC=CC(NC(=O)c2ccc(NC(C)C)nc2NC2CCN(C(=O)CN3CCN(Cc4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)CC2)N1	C47H61N13O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-4RSE8N	WO-2024183798-A1_CPD-534	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C5CCN(C(=O)C67CC(Nc8nc(NC(C)C)ccc8C(=O)Nc8ccc(N(C)C)nn8)(C6)C7)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C49H61N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-BEHKUC	WO-2024183798-A1_CPD-535	.	CC(C)Nc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(N[C@H]2CC[C@H](C(=O)N3CCC(N4CCN(c5ccc(Nc6ncc7ccc(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)CC2)n1	C47H61N15O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-8G2IE6	WO-2024183798-A1_CPD-536	.	COC1(C(=O)N2CCC(N3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)C2)CCC(Nc2nc(NC(C)C)ccc2C(=O)Nc2ccc(N(C)C)nn2)CC1	C51H67N15O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-2FLNBN	WO-2024183798-A1_CPD-537	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C5CCN(C(=O)CC67CC(Nc8nc(NC(C)C)ccc8C(=O)Nc8ccc(N(C)C)nn8)(C6)C7)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C50H63N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-S0LNEY	WO-2024183798-A1_CPD-538	.	CC(=O)c1c(C)c2cnc(Nc3ccc(CN4CCN(C(=O)CN5CC6(CC(Nc7nc(NC(C)C)ccc7C(=O)Nc7ccc(N(C)C)nn7)C6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C48H61N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-XFOA9K	WO-2024183798-A1_CPD-539	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C5CCN(C(=O)N6CCC7(CC(Nc8nc(NC(C)C)ccc8C(=O)Nc8ccc(N(C)C)nn8)C7)C6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C51H66N16O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-DMJEQN	WO-2024183798-A1_CPD-540	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C5CCN(C(=O)C6CCC(Nc7nc(NC(C)C)ccc7-c7nc8cc(N(C)C)ccc8[nH]7)CC6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C52H66N14O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-I9FJ93	WO-2024183798-A1_CPD-541	.	CC(=O)c1c(C)c2cnc(Nc3ccc(CN4CCN(C(=O)CN5CCC(Nc6nc(NC(C)C)ccc6C(=O)Nc6ccc(N(C)C)nn6)CC5)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H61N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-KN516G	WO-2024183798-A1_CPD-542	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCC(N5CCC[C@H]5C(=O)NCC5CC(Nc6nc(NC(C)C)ccc6C(=O)Nc6ccc(N(C)C)nn6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C50H65N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-R4TXBC	WO-2024183798-A1_CPD-543	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCC(N5CCC[C@H]5C(=O)NC5CC6(C5)CC(Nc5nc(NC(C)C)ccc5C(=O)Nc5ccc(N(C)C)nn5)C6)CC4)cn3)nc2n(C2CCCC2)c1=O	C52H67N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-7Z2OT4	WO-2024183798-A1_CPD-544	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCC(N5CCC[C@H]5C(=O)N5CC6(CC(Nc7nc(NC(C)C)ccc7C(=O)Nc7ccc(N(C)C)nn7)C6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C51H65N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-8UNBZ3	WO-2024183798-A1_CPD-545	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C5CCN(C(=O)N6CC7(CCC(Nc8nc(NC(C)C)ccc8C(=O)Nc8ccc(N(C)C)nn8)C7)C6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C51H66N16O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-SS34ZX	WO-2024183798-A1_CPD-546	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C5CCN(C(=O)C6CCC(Nc7nc(NC(C)C)ccc7-c7nc8ccc(N(C)C)nc8[nH]7)CC6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C51H65N15O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-IOYEO5	WO-2024183798-A1_CPD-547	.	CC(=O)c1c(C)c2cnc(Nc3ccc(CN4CCN(CC(=O)N5CCC6(CCC(Nc7nc(NC(C)C)ccc7C(=O)Nc7cc(C)n(C)n7)C6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C49H64N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-ALXJPC	WO-2024183798-A1_CPD-548	.	CC(=O)c1c(C)c2cnc(Nc3ccc(CN4CCN(CC(=O)N5CCC6(CCC(Nc7nc(NC(C)C)ccc7C(=O)Nc7cn(C)c(C8CC8)n7)C6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C51H66N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-T6XO3I	WO-2024183798-A1_CPD-549	.	CC(=O)c1c(C)c2cnc(Nc3ccc(CN4CCN(CC(=O)N5CCC6(CCC(Nc7nc(NC(C)C)ccc7C(=O)Nc7cc8n(n7)CCC8)C6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C50H64N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-56AY1J	WO-2024183798-A1_CPD-550	.	CC(=O)c1c(C)c2cnc(Nc3ccc(CN4CCN(C(C)C(=O)N5CCC6(CCC(Nc7nc(NC(C)C)ccc7C(=O)Nc7ccc(N(C)C)nn7)C6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C51H67N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-B340FD	WO-2024183798-A1_CPD-551	.	CC(=O)c1c(C)c2cnc(Nc3ccc(C(C)N4CCN(CC(=O)N5CCC6(CCC(Nc7nc(NC(C)C)ccc7C(=O)Nc7ccc(N(C)C)nn7)C6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C51H67N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-AZW8HE	WO-2024183798-A1_CPD-552	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C5CCN(C(=O)C6CCC(Nc7nc(NC(C)C)ccc7-c7nc8cnc(N(C)C)cc8[nH]7)CC6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C51H65N15O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-DN9JKX	WO-2024183798-A1_CPD-553	.	CCN1CCc2cc(-c3nc(Nc4ccc(CN5CCN(CC(=O)N6CC7(CC(Nc8nc(NC(C)C)ccc8C(=O)Nc8ccc(N(C)C)nn8)C7)C6)CC5)cn4)ncc3F)ccc2C1=O	C48H58FN15O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-VXOAX8	WO-2024183798-A1_CPD-554	.	CCN1CCc2cc(-c3nc(Nc4ccc(CN5CCN(CC(=O)NC6CC7(C6)CC(Nc6nc(NC(C)C)ccc6C(=O)Nc6ccc(N(C)C)nn6)C7)CC5)cn4)ncc3F)ccc2C1=O	C49H60FN15O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-29UW7I	WO-2024183798-A1_CPD-555	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C5CCN(C(=O)N6CC7(CCC(Nc8nc(NC(C)C)ccc8C(=O)Nc8ccc(N(C)C)nn8)CC7)C6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C52H68N16O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-G9TSDB	WO-2024183798-A1_CPD-556	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C5CCN(C(=O)C6CCC7(CC(Nc8nc(NC(C)C)ccc8C(=O)Nc8ccc(N(C)C)nn8)C7)C6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C52H67N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-VELU1Z	WO-2024183798-A1_CPD-557	.	CC(C)Nc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC3(C2)CN(C(=O)CN2CCN(Cc4ccc(Nc5ncc6cc7n(c6n5)C5(CCCCC5)CNC7=O)nc4)CC2)C3)n1	C47H60N16O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-X4W6I4	WO-2024183798-A1_CPD-558	.	CC(C)Nc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC3(CC(NC(=O)CN4CCN(Cc5ccc(Nc6ncc7cc8n(c7n6)C6(CCCCC6)CNC8=O)nc5)CC4)C3)C2)n1	C48H62N16O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-DE2EWE	WO-2024183798-A1_CPD-559	.	CC(C)Nc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(N[C@H]2CC[C@H](C(=O)N3CCC(N4CCN(c5ccc(Nc6ncc7cc(C(F)F)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)CC2)n1	C48H61F2N15O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-LF9VYG	WO-2024183798-A1_CPD-560	.	CC(=O)c1cc2cnc(Nc3ccc(N4CCN(C5CCN(C(=O)[C@H]6CC[C@H](Nc7nc(NC(C)C)ccc7C(=O)Nc7ccc(N(C)C)nn7)CC6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C49H63N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-9P8MA8	WO-2024183798-A1_CPD-561	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C5CCN(C(=O)N6CCC7(CCC(Nc8nc(NC(C)C)ccc8C(=O)Nc8ccc(N(C)C)nn8)C7)C6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C52H68N16O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-9HL2C4	WO-2024183798-A1_CPD-562	.	CC(C)Nc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC3(CC(NC(=O)CN4CCN(Cc5ccc(Nc6ncc7cc(C(=O)N(C)C)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C48H64N16O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-47SIA1	WO-2024183798-A1_CPD-563	.	CC(C)Nc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC3(C2)CN(C(=O)CN2CCN(Cc4ccc(Nc5ncc6cc(C(=O)N(C)C)n(C7CCCC7)c6n5)nc4)CC2)C3)n1	C47H62N16O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-K7VL57	WO-2024183798-A1_CPD-564	.	CC(=O)c1c(C)c2cnc(Nc3ccc(CN4CCN(CC(=O)N5CCC(Nc6nc(NC(C)C)ccc6C(=O)Nc6cn7c(n6)CCC7)CC5)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H60N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-MOY2B3	WO-2024183798-A1_CPD-565	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCC5(CCN(CC(=O)N6CC7(CC(Nc8nc(NC(C)C)ccc8C(=O)Nc8cn9c(n8)CCC9)C7)C6)C5)C4)cn3)nc2n(C2CCCC2)c1=O	C50H62N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-3D7Z65	WO-2024183798-A1_CPD-566	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CC(=O)NC5CC6(C5)CC(Nc5nc(NC(C)C)ccc5C(=O)Nc5cn7c(n5)CCC7)C6)CC4)cn3)nc2n(C2CCCC2)c1=O	C48H60N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-BE5CDM	WO-2024183798-A1_CPD-567	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(CC(=O)N5CC6(CC(Nc7nc(C)ccc7C(=O)Nc7cn8c(n7)CCC8)C6)C5)C(F)(F)F)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H54F3N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-X4ZFPU	WO-2024183798-A1_CPD-568	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C5CCN(C(=O)[C@H]6CC[C@H](Nc7nc(NC(C)C)ccc7C(=O)Nc7cn8c(n7)CCC8)CC6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C50H64N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-MVOOW9	WO-2024183798-A1_CPD-569	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C5CCN(C(=O)[C@H]6CC[C@H](Nc7nc(C)ccc7C(=O)Nc7cn8c(n7)CCC8)CC6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C48H59N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-YMI14Q	WO-2024183798-A1_CPD-570	.	CC(=O)c1c(C)c2cnc(Nc3ccc(CN4CCN(CC(=O)N5CCC6(CC(Nc7nc(NC(C)C)ccc7C(=O)Nc7ccc(N(C)C)nn7)C6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C49H63N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-FGMTWV	WO-2024183798-A1_CPD-571	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C5CCN(C(=O)[C@H]6CC[C@H](Nc7nc(C(F)(F)F)ccc7C(=O)Nc7ccc(N(C)C)nn7)CC6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C48H57F3N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-MS5D38	WO-2024183798-A1_CPD-572	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C5CCN(C(=O)C6(F)CCC(Nc7nc(NC(C)C)ccc7C(=O)Nc7ccc(N(C)C)nn7)CC6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C50H64FN15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-OYJBKF	WO-2024183798-A1_CPD-573	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C5CCN(C(=O)[C@H]6CC[C@H](Nc7nc(C8CC8)ccc7C(=O)Nc7ccc(N(C)C)nn7)CC6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C50H62N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-22BBNG	WO-2024183798-A1_CPD-574	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C5CCN(C(=O)C6(O)CCC(Nc7nc(NC(C)C)ccc7C(=O)Nc7ccc(N(C)C)nn7)CC6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C50H65N15O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-NAUMFA	WO-2024183798-A1_CPD-577	.	CCc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC23CC(C(=O)N4CCC(N5CCN(c6ccc(Nc7ncc8c(C)c(C(C)=O)c(=O)n(C9CCCC9)c8n7)nc6)CC5)C4)(C2)C3)n1	C48H58N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-5628E9	WO-2024183798-A1_CPD-578	.	CCc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC3(CC(NC(=O)CN4CCN(Cc5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C48H60N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-LB14JE	WO-2024183798-A1_CPD-579	.	CC(=O)c1c(C)c2cnc(Nc3ccc(CN4CCN(CC(=O)NC5CC6(C5)CC(Nc5nc(C(C)C)ccc5C(=O)Nc5ccc(N(C)C)nn5)C6)CC4)cn3)nc2n(C2CCCC2)c1=O	C49H62N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-NYF722	WO-2024183798-A1_CPD-580	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C5CCN(C(=O)C67CC(Nc8nc(C(C)C)ccc8C(=O)Nc8ccc(N(C)C)nn8)(C6)C7)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C49H60N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-DG9TEF	WO-2024183798-A1_CPD-581	.	CC(=O)c1c(C)c2cnc(Nc3ccc(CN4CCN(CC(=O)N5CCC6(CCC(Nc7nc(C8CC8)ccc7C(=O)Nc7ccc(N(C)C)nn7)C6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C50H62N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-1SY0ES	WO-2024183798-A1_CPD-582	.	CCc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CCC3(CCN(C(=O)CN4CCN(Cc5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)n1	C49H62N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-66LB3Z	WO-2024183798-A1_CPD-583	.	CC(=O)c1c(C)c2cnc(Nc3ccc(CN4CCN(CC(=O)N5CCC6(CCC(Nc7nc(C(C)C)ccc7C(=O)Nc7ccc(N(C)C)nn7)C6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C50H64N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-R4IIF9	WO-2024183798-A1_CPD-584	.	CC(=O)c1c(C)c2cnc(Nc3ccc(CN4CCN(CC(=O)NC5CC6(C5)CC(Nc5nc(NC(C)C)ccc5C(=O)Nc5cc7n(n5)CCC7)C6)CC4)cn3)nc2n(C2CCCC2)c1=O	C49H62N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-JN75EN	WO-2024183798-A1_CPD-585	.	CC(=O)c1c(C)c2cnc(Nc3ccc(CN4CCN(C(C)C(=O)NC5CC6(C5)CC(Nc5nc(NC(C)C)ccc5C(=O)Nc5ccc(N(C)C)nn5)C6)CC4)cn3)nc2n(C2CCCC2)c1=O	C50H65N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-6O5J95	WO-2024183798-A1_CPD-586	.	CC(=O)c1c(C)c2cnc(Nc3ccc(C(C)N4CCN(CC(=O)NC5CC6(C5)CC(Nc5nc(NC(C)C)ccc5C(=O)Nc5ccc(N(C)C)nn5)C6)CC4)cn3)nc2n(C2CCCC2)c1=O	C50H65N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-96U28D	WO-2024183798-A1_CPD-587	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C5CCN(C(=O)C67CC(Nc8nc(NC(C)C)ccc8C(=O)Nc8cc(C)n(C)n8)(C6)C7)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C48H60N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-EL9YJ7	WO-2024183798-A1_CPD-588	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C5CCN(C(=O)C67CC(Nc8nc(NC(C)C)ccc8C(=O)Nc8cn(C)c(C9CC9)n8)(C6)C7)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C50H62N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-EPMGXH	WO-2024183798-A1_CPD-589	.	CC(=O)c1c(C)c2cnc(Nc3ccc(CN4CCN(CC(=O)NC5CC6(C5)CC(Nc5nc(NC(C)C)ccc5C(=O)Nc5cn(C)c(C7CC7)n5)C6)CC4)cn3)nc2n(C2CCCC2)c1=O	C50H64N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-CK17ZZ	WO-2024183798-A1_CPD-590	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C5CCN(C(=O)C67CC(Nc8nc(C)ccc8C(=O)Nc8ccc(N(C)C)nn8)(C6)C7)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H56N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-9SUMN1	WO-2024183798-A1_CPD-591	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C5CCN(C(=O)C67CC(Nc8nc(NC(C)C)ccc8C(=O)Nc8cc(C)on8)(C6)C7)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H57N13O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-KA63AE	WO-2024183798-A1_CPD-592	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C5CCN(C(=O)C67CC(Nc8nc(NC(C)C)ccc8C(=O)Nc8cc9n(n8)CCC9)(C6)C7)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C49H60N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-LA0QLS	WO-2024183798-A1_CPD-593	.	CC(=O)c1c(C)c2cnc(Nc3ccc(CN4CCC(CC(=O)NC5CC6(C5)CC(Nc5nc(NC(C)C)ccc5C(=O)Nc5ccc(N(C)C)nn5)C6)CC4)cn3)nc2n(C2CCCC2)c1=O	C50H64N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-DPUEHC	WO-2024183798-A1_CPD-594	.	CC(=O)c1c(C)c2cnc(Nc3ccc(CN4CCN(CC(=O)N(C)C5CC6(CC(Nc7nc(NC(C)C)ccc7C(=O)Nc7ccc(N(C)C)nn7)C6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C50H65N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-BNR5QC	WO-2024183798-A1_CPD-595	.	CC(=O)c1c(C)c2cnc(Nc3ccc(CN4CCC(N(C)C(=O)C5CC6(CC(Nc7nc(NC(C)C)ccc7C(=O)Nc7ccc(N(C)C)nn7)C6)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C50H64N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-PRW72J	WO-2024183798-A1_CPD-596	.	CC(=O)c1c(C)c2cnc(Nc3ccc(CN4CCC(CC(=O)NC5CC6(C5)CC(Nc5nc(NC(C)C)ccc5C(=O)Nc5ccc(N(C)C)nn5)C6)C4)cn3)nc2n(C2CCCC2)c1=O	C49H62N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-KYKPEV	WO-2024183798-A1_CPD-597	.	CCc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(N[C@H]2CC[C@H](C(=O)N3CCC(N4CCN(C5CCC(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)CC5)CC4)C3)CC2)n1	C50H69N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-VA7GD8	WO-2024183798-A1_CPD-598	.	CCc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NC2CC3(CC(NC(=O)CN4CCN(Cc5ccc(Nc6ncc7c(C)c(C(C)=O)c(=O)n(C8CCCC8)c7n6)nc5)CC4)C3)C2)c1	C49H61N13O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-P10F9W	WO-2024183798-A1_CPD-599	.	CC(=O)c1c(C)c2cnc(Nc3ccc(CC4CCN(CC(=O)NC5CC6(C5)CC(Nc5nc(NC(C)C)ccc5C(=O)Nc5ccc(N(C)C)nn5)C6)CC4)cn3)nc2n(C2CCCC2)c1=O	C50H64N14O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-OP5UMA	WO-2024183798-A1_CPD-600	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCC(=O)N2CCN(Cc3ccc(Nc4ncc(F)c(-c5cc(F)c6nc(C)n(C(C)C)c6c5)n4)nc3)CC2)n1	C41H47F2N15O2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-7ZQZC3	WO-2024183798-A1_CPD-601	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCC(=O)N2CCN(Cc3ccc(Nc4ncc(F)c(-c5cc(F)c6nc(C)n(C(C)C)c6c5)n4)nc3)CC2)n1	C42H49F2N15O2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-D1HZLC	WO-2024183798-A1_CPD-602	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCCC(=O)N2CCN(Cc3ccc(Nc4ncc(F)c(-c5cc(F)c6nc(C)n(C(C)C)c6c5)n4)nc3)CC2)n1	C43H51F2N15O2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-F25PDQ	WO-2024183798-A1_CPD-603	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCCCC(=O)N2CCN(Cc3ccc(Nc4ncc(F)c(-c5cc(F)c6nc(C)n(C(C)C)c6c5)n4)nc3)CC2)n1	C44H53F2N15O2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-LE8VD9	WO-2024183798-A1_CPD-604	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCCCCC(=O)N2CCN(Cc3ccc(Nc4ncc(F)c(-c5cc(F)c6nc(C)n(C(C)C)c6c5)n4)nc3)CC2)n1	C45H55F2N15O2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-HRWT65	WO-2024183798-A1_CPD-605	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCCCCCC(=O)N2CCN(Cc3ccc(Nc4ncc(F)c(-c5cc(F)c6nc(C)n(C(C)C)c6c5)n4)nc3)CC2)n1	C46H57F2N15O2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-JKNULG	WO-2024183798-A1_CPD-606	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCOCCC(=O)N2CCN(Cc3ccc(Nc4ncc(C)c(-c5cc(F)c6nc(C)n(C(C)C)c6c5)n4)nc3)CC2)n1	C44H54FN15O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-8YI40L	WO-2024183798-A1_CPD-607	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCOCCOCCC(=O)N2CCN(Cc3ccc(Nc4ncc(F)c(-c5cc(F)c6nc(C)n(C(C)C)c6c5)n4)nc3)CC2)n1	C45H55F2N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-2MCSBY	WO-2024183798-A1_CPD-608	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCNC(=O)CN2CCN(Cc3ccc(Nc4ncc(F)c(-c5cc(F)c6nc(C)n(C(C)C)c6c5)n4)nc3)CC2)n1	C42H50F2N16O2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-DNI5Y3	WO-2024183798-A1_CPD-609	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCNC(=O)CN2CCN(Cc3ccc(Nc4ncc(F)c(-c5cc(F)c6nc(C)n(C(C)C)c6c5)n4)nc3)CC2)n1	C43H52F2N16O2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-CMCBJH	WO-2024183798-A1_CPD-610	.	CNc1ccc(CNc2ccc(N(C)C)nn2)c(NCCCCNC(=O)CN2CCN(Cc3ccc(Nc4ncc(F)c(-c5cc(F)c6nc(C)n(C(C)C)c6c5)n4)nc3)CC2)n1	C44H56F2N16O	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-1E6S88	WO-2024183798-A1_CPD-611	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCCCNC(=O)CN2CCN(Cc3ccc(Nc4ncc(F)c(-c5cc(F)c6nc(C)n(C(C)C)c6c5)n4)nc3)CC2)n1	C45H56F2N16O2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-T5STF4	WO-2024183798-A1_CPD-612	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCCCCNC(=O)CN2CCN(Cc3ccc(Nc4ncc(F)c(-c5cc(F)c6nc(C)n(C(C)C)c6c5)n4)nc3)CC2)n1	C46H58F2N16O2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-5VJE1O	WO-2024183798-A1_CPD-613	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCCCCCNC(=O)CN2CCN(Cc3ccc(Nc4ncc(F)c(-c5cc(F)c6nc(C)n(C(C)C)c6c5)n4)nc3)CC2)n1	C47H60F2N16O2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-PKB2SD	WO-2024183798-A1_CPD-614	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCCCCCCNC(=O)CN2CCN(Cc3ccc(Nc4ncc(F)c(-c5cc(F)c6nc(C)n(C(C)C)c6c5)n4)nc3)CC2)n1	C48H62F2N16O2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-2P2Y10	WO-2024183798-A1_CPD-615	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCOCCNC(=O)CN2CCN(Cc3ccc(Nc4ncc(F)c(-c5cc(F)c6nc(C)n(C(C)C)c6c5)n4)nc3)CC2)n1	C44H54F2N16O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-ROR2JO	WO-2024183798-A1_CPD-616	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCC(=O)N2CCN(c3ccc(Nc4ncc5cc(C(=O)N(C)C)n(C6CCCC6)c5n4)nc3)CC2)n1	C39H49N15O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-2XU25I	WO-2024183798-A1_CPD-617	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCC(=O)N2CCN(c3ccc(Nc4ncc5cc(C(=O)N(C)C)n(C6CCCC6)c5n4)nc3)CC2)n1	C40H51N15O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-NUPA2X	WO-2024183798-A1_CPD-618	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCCC(=O)N2CCN(c3ccc(Nc4ncc5cc(C(=O)N(C)C)n(C6CCCC6)c5n4)nc3)CC2)n1	C41H53N15O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-N2J2N5	WO-2024183798-A1_CPD-619	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCCCC(=O)N2CCN(c3ccc(Nc4ncc5cc(C(=O)N(C)C)n(C6CCCC6)c5n4)nc3)CC2)n1	C42H55N15O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-JS5X4Z	WO-2024183798-A1_CPD-620	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCCCCC(=O)N2CCN(c3ccc(Nc4ncc5cc(C(=O)N(C)C)n(C6CCCC6)c5n4)nc3)CC2)n1	C43H57N15O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-VQ9FSZ	WO-2024183798-A1_CPD-621	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCCCCCC(=O)N2CCN(c3ccc(Nc4ncc5cc(C(=O)N(C)C)n(C6CCCC6)c5n4)nc3)CC2)n1	C44H59N15O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-28BHOP	WO-2024183798-A1_CPD-622	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCOCCC(=O)N2CCN(c3ccc(Nc4ncc5cc(C(=O)N(C)C)n(C6CCCC6)c5n4)nc3)CC2)n1	C41H53N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-0IIUDN	WO-2024183798-A1_CPD-623	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCOCCOCCC(=O)N2CCN(c3ccc(Nc4ncc5cc(C(=O)N(C)C)n(C6CCCC6)c5n4)nc3)CC2)n1	C43H57N15O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-YABATP	WO-2024183798-A1_CPD-624	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCNC(=O)CN2CCN(c3ccc(Nc4ncc5cc(C(=O)N(C)C)n(C6CCCC6)c5n4)nc3)CC2)n1	C40H52N16O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-YUIG5Q	WO-2024183798-A1_CPD-625	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5cc(C(=O)N(C)C)n(C6CCCC6)c5n4)nc3)CC2)n1	C41H54N16O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-C2NVTP	WO-2024183798-A1_CPD-626	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5cc(C(=O)N(C)C)n(C6CCCC6)c5n4)nc3)CC2)n1	C42H56N16O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-FM6DII	WO-2024183798-A1_CPD-627	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5cc(C(=O)N(C)C)n(C6CCCC6)c5n4)nc3)CC2)n1	C43H58N16O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-0MOQQD	WO-2024183798-A1_CPD-628	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5cc(C(=O)N(C)C)n(C6CCCC6)c5n4)nc3)CC2)n1	C44H60N16O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-GG66CF	WO-2024183798-A1_CPD-629	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5cc(C(=O)N(C)C)n(C6CCCC6)c5n4)nc3)CC2)n1	C45H62N16O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-YLKHCU	WO-2024183798-A1_CPD-630	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5cc(C(=O)N(C)C)n(C6CCCC6)c5n4)nc3)CC2)n1	C46H64N16O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-X98RYW	WO-2024183798-A1_CPD-631	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCOCCNC(=O)CN2CCN(c3ccc(Nc4ncc5cc(C(=O)N(C)C)n(C6CCCC6)c5n4)nc3)CC2)n1	C42H56N16O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-H2Z9KL	WO-2024183798-A1_CPD-632	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCC(=O)N2CCN(c3ccc(Nc4ncc5cc6n(c5n4)C4(CCCCC4)CNC6=O)nc3)CC2)n1	C39H47N15O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-PU2GT1	WO-2024183798-A1_CPD-633	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCC(=O)N2CCN(c3ccc(Nc4ncc5cc6n(c5n4)C4(CCCCC4)CNC6=O)nc3)CC2)n1	C40H49N15O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-EBIDHF	WO-2024183798-A1_CPD-634	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCCC(=O)N2CCN(c3ccc(Nc4ncc5cc6n(c5n4)C4(CCCCC4)CNC6=O)nc3)CC2)n1	C41H51N15O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-FD6YGS	WO-2024183798-A1_CPD-635	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCCCCC(=O)N2CCN(c3ccc(Nc4ncc5cc6n(c5n4)C4(CCCCC4)CNC6=O)nc3)CC2)n1	C43H55N15O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-MD64ZQ	WO-2024183798-A1_CPD-637	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCCCCCC(=O)N2CCN(c3ccc(Nc4ncc5cc6n(c5n4)C4(CCCCC4)CNC6=O)nc3)CC2)n1	C44H57N15O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-Q16BOQ	WO-2024183798-A1_CPD-638	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCOCCC(=O)N2CCN(c3ccc(Nc4ncc5cc6n(c5n4)C4(CCCCC4)CNC6=O)nc3)CC2)n1	C41H51N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-I8A1FC	WO-2024183798-A1_CPD-639	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCOCCOCCC(=O)N2CCN(c3ccc(Nc4ncc5cc6n(c5n4)C4(CCCCC4)CNC6=O)nc3)CC2)n1	C43H55N15O5	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-O573EZ	WO-2024183798-A1_CPD-640	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCNC(=O)CN2CCN(c3ccc(Nc4ncc5cc6n(c5n4)C4(CCCCC4)CNC6=O)nc3)CC2)n1	C40H50N16O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-G0659L	WO-2024183798-A1_CPD-641	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5cc6n(c5n4)C4(CCCCC4)CNC6=O)nc3)CC2)n1	C41H52N16O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-XOOC9R	WO-2024183798-A1_CPD-642	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5cc6n(c5n4)C4(CCCCC4)CNC6O)nc3)CC2)n1	C42H56N16O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-DUKMRZ	WO-2024183798-A1_CPD-643	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5cc6n(c5n4)C4(CCCCC4)CNC6=O)nc3)CC2)n1	C43H56N16O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-V652AS	WO-2024183798-A1_CPD-644	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5cc6n(c5n4)C4(CCCCC4)CNC6=O)nc3)CC2)n1	C44H58N16O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-9UX07B	WO-2024183798-A1_CPD-645	.	CNc1ccc(C(=O)Nc2ccc(CN(C)C)nn2)c(NCCCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5cc6n(c5n4)C4(CCCCC4)CNC6=O)nc3)CC2)n1	C46H62N16O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-CKVK73	WO-2024183798-A1_CPD-646	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc5cc6n(c5n4)C4(CCCCC4)CNC6=O)nc3)CC2)n1	C46H62N16O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-3LM553	WO-2024183798-A1_CPD-647	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCOCCNC(=O)CN2CCN(c3ccc(Nc4ncc5cc6n(c5n4)C4(CCCCC4)CNC6=O)nc3)CC2)n1	C42H54N16O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-BWBIMO	WO-2024183798-A1_CPD-648	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCC(=O)N2CCN(c3ccc(Nc4ncc(F)c(-c5cc(F)c6nc(C)n(C(C)C)c6c5)n4)nc3)CC2)n1	C40H45F2N15O2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-67S3RM	WO-2024183798-A1_CPD-649	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCC(=O)N2CCN(c3ccc(Nc4ncc(F)c(-c5cc(F)c6nc(C)n(C(C)C)c6c5)n4)nc3)CC2)n1	C41H47F2N15O2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-BT6XUA	WO-2024183798-A1_CPD-650	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCCC(=O)N2CCN(c3ccc(Nc4ncc(F)c(-c5cc(F)c6nc(C)n(C(C)C)c6c5)n4)nc3)CC2)n1	C42H49F2N15O2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-JSDQ58	WO-2024183798-A1_CPD-651	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCCCC(=O)N2CCN(c3ccc(Nc4ncc(F)c(-c5cc(F)c6nc(C)n(C(C)C)c6c5)n4)nc3)CC2)n1	C43H51F2N15O2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-MT9A4G	WO-2024183798-A1_CPD-652	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCCCCC(=O)N2CCN(c3ccc(Nc4ncc(C)c(-c5cc(F)c6nc(C)n(C(C)C)c6c5)n4)nc3)CC2)n1	C45H56FN15O2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-ZCGL36	WO-2024183798-A1_CPD-653	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCCCCCC(=O)N2CCN(c3ccc(Nc4ncc(F)c(-c5cc(F)c6nc(C)n(C(C)C)c6c5)n4)nc3)CC2)n1	C45H55F2N15O2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-6CX5J2	WO-2024183798-A1_CPD-654	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCOCCC(=O)N2CCN(c3ccc(Nc4ncc(F)c(-c5cc(F)c6nc(C)n(C(C)C)c6c5)n4)nc3)CC2)n1	C42H49F2N15O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-8G4UDR	WO-2024183798-A1_CPD-655	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCOCCOCCC(=O)N2CCN(c3ccc(Nc4ncc(F)c(-c5cc(F)c6nc(C)n(C(C)C)c6c5)n4)nc3)CC2)n1	C44H53F2N15O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-6WC2FI	WO-2024183798-A1_CPD-656	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCC(=O)N2CCN(Cc3ccc(Nc4ncc(F)c(-c5cc(F)c6nc(C)n(C(C)C)c6c5)n4)nc3)CC2)n1	C40H45F2N15O2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-O9663A	WO-2024183798-A1_CPD-657	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCC(=O)N2CCN(c3ccc(Nc4ncc5cc(C(=O)N(C)C)n(C6CCCC6)c5n4)nc3)CC2)n1	C38H47N15O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-TQLIX6	WO-2024183798-A1_CPD-658	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCNC(=O)CN2CCN(c3ccc(Nc4ncc(F)c(-c5cc(F)c6nc(C)n(C(C)C)c6c5)n4)nc3)CC2)n1	C41H48F2N16O2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-QQO118	WO-2024183798-A1_CPD-659	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCNC(=O)CN2CCN(c3ccc(Nc4ncc(F)c(-c5cc(F)c6nc(C)n(C(C)C)c6c5)n4)nc3)CC2)n1	C42H50F2N16O2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-HQWP9F	WO-2024183798-A1_CPD-660	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc(F)c(-c5cc(F)c6nc(C)n(C(C)C)c6c5)n4)nc3)CC2)n1	C43H52F2N16O2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-5QWHSN	WO-2024183798-A1_CPD-661	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc(F)c(-c5cc(F)c6nc(C)n(C(C)C)c6c5)n4)nc3)CC2)n1	C44H54F2N16O2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-LFPJXY	WO-2024183798-A1_CPD-662	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc(F)c(-c5cc(F)c6nc(C)n(C(C)C)c6c5)n4)nc3)CC2)n1	C45H56F2N16O2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-IFYJVM	WO-2024183798-A1_CPD-663	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc(C)c(-c5cc(F)c6nc(C)n(C(C)C)c6c5)n4)nc3)CC2)n1	C47H61FN16O2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-ERIAZW	WO-2024183798-A1_CPD-664	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCCCCCCNC(=O)CN2CCN(c3ccc(Nc4ncc(F)c(-c5cc(F)c6nc(C)n(C(C)C)c6c5)n4)nc3)CC2)n1	C47H60F2N16O2	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-I5GSU4	WO-2024183798-A1_CPD-665	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCOCCNC(=O)CN2CCN(c3ccc(Nc4ncc(F)c(-c5cc(F)c6nc(C)n(C(C)C)c6c5)n4)nc3)CC2)n1	C43H52F2N16O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-RXE0LE	WO-2024183798-A1_CPD-666	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCC(=O)NC2CCC(Nc3ncc4ccc(=O)n(C5CCCC5)c4n3)CC2)n1	C34H44N12O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-GN9VIZ	WO-2024183798-A1_CPD-667	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCC(=O)NC2CCC(Nc3ncc4ccc(=O)n(C5CCCC5)c4n3)CC2)n1	C35H46N12O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-07SCF0	WO-2024183798-A1_CPD-668	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCCC(=O)NC2CCC(Nc3ncc4ccc(=O)n(C5CCCC5)c4n3)CC2)n1	C36H48N12O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-7KLMXQ	WO-2024183798-A1_CPD-669	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCCCC(=O)NC2CCC(Nc3ncc4ccc(=O)n(C5CCCC5)c4n3)CC2)n1	C37H50N12O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-7ELN53	WO-2024183798-A1_CPD-670	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCCCCC(=O)NC2CCC(Nc3ncc4ccc(=O)n(C5CCCC5)c4n3)CC2)n1	C38H52N12O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-GJOXDI	WO-2024183798-A1_CPD-671	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCCCCCC(=O)NC2CCC(Nc3ncc4ccc(=O)n(C5CCCC5)c4n3)CC2)n1	C39H54N12O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-G0GIY2	WO-2024183798-A1_CPD-672	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCOCCC(=O)NC2CCC(Nc3ncc4ccc(=O)n(C5CCCC5)c4n3)CC2)n1	C36H48N12O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-WP0GS2	WO-2024183798-A1_CPD-673	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCC(=O)NC2CCC3(CC2)CC(Nc2ncc4ccc(=O)n(C5CCCC5)c4n2)C3)n1	C37H48N12O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-1JQ1TA	WO-2024183798-A1_CPD-674	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCC(=O)NC2CCC3(CC2)CC(Nc2ncc4ccc(=O)n(C5CCCC5)c4n2)C3)n1	C38H50N12O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-QPL3HI	WO-2024183798-A1_CPD-675	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCCC(=O)NC2CCC3(CC2)CC(Nc2ncc4ccc(=O)n(C5CCCC5)c4n2)C3)n1	C39H52N12O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-9Q1971	WO-2024183798-A1_CPD-676	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCCCC(=O)NC2CCC3(CC2)CC(Nc2ncc4ccc(=O)n(C5CCCC5)c4n2)C3)n1	C40H54N12O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-MOJARO	WO-2024183798-A1_CPD-677	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCCCCC(=O)NC2CCC3(CC2)CC(Nc2ncc4ccc(=O)n(C5CCCC5)c4n2)C3)n1	C41H56N12O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-6FH56S	WO-2024183798-A1_CPD-678	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCCCCCCC(=O)NC2CCC3(CC2)CC(NC2=Nc4c(ccc(=O)n4C4CCCC4)CN2)C3)n1	C42H60N12O3	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-8XG2HB	WO-2024183798-A1_CPD-679	.	CNc1ccc(C(=O)Nc2ccc(N(C)C)nn2)c(NCCOCCC(=O)NC2CCC3(CC2)CC(Nc2ncc4ccc(=O)n(C5CCCC5)c4n2)C3)n1	C39H52N12O4	CDK4;CDK6	P11802/Q00534	DDB1	WO-2024183798-A1
TPD-6A33LW	MZ 1	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[2-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; 1797406-69-9; MZ1; (2S,4R)-1-[(2S)-2-[[2-[2-[2-[2-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; CHEMBL4226570; (2S,4R)-1-((S)-2-(tert-butyl)-17-((S)-4-(4-chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl)-4,16-dioxo-6,9,12-trioxa-3,15-diazaheptadecanoyl)-4-hydroxy-N-(4-(4-methylthiazol-5-yl)benzyl)pyrrolidine-2-carboxamide; orb1301791; SCHEMBL18076362; GTPL10728; MZ1; MZ-1; CHEBI:189652; BCP31482; EX-A3902; MZ 1( MZ-1); XWC40669; BDBM50459880; s8889; AKOS032947179; AT14161; AC-36493; BP-27846; DA-65741; HY-107425; CS-0028453; EN300-22213039; ethylthiazol-5-yl)benzyl)pyrrolidine-2-carboxamide; Z2967326564; (2S,4R)-1-((S)-2-(tert-butyl)-17-((S)-4-(4-chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl)-4,16-dioxo-6,9,12-trioxa-3,15-diazaheptadecan-1-oyl)-4-hydroxy-N-(4-(4-methylthiazol-5-yl)benzyl)pyrrolidine-2-carboxamide; (2S,4R)-1-((S)-2-(tert-butyl)-17-((S)-4-(4-chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl)-4,16-dioxo-6,9,12-trioxa-3,15-diazaheptadecanoyl)-4-hydroxy-N-(4-(4-m; (2S,4R)-1-[(2S)-2-(2-{2-[2-(2-{2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetraazatricyclo[8.3.0.0,2,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetamido}ethoxy)ethoxy]ethoxy}acetamido)-3,3-dimethylbutanoyl]-4-hydroxy-N-{[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl}pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCNC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)C(C)(C)C)cc1	C49H60ClN9O8S2	BRD4	O60885	VHL	WO-2016146985-A1
TPD-CEOP6W	CHEMBL4227226	(2S,4R)-1-((S)-2-(tert-butyl)-20-((S)-4-(4-chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl)-4,19-dioxo-6,9,12,15-tetraoxa-3,18-diazaicosanoyl)-4-hydroxy-N-(4-(4-methylthiazol-5-yl)benzyl)pyrrolidine-2-carboxamide; (2S,4R)-1-((S)-2-(tert-butyl)-20-((S)-4-(4-chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl)-4,19-dioxo-6,9,12,15-tetraoxa-3,18-diazaicosanoyl)-4-hydroxy-N-(4-(4-methylthiazol-5-yl)benzyl)pyrrolidine-2-carboxamide; SCHEMBL19875313; BDBM50459879	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCOCCNC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)C(C)(C)C)cc1	C51H64ClN9O9S2	BRD4	O60885	VHL	WO-2016146985-A1
TPD-EJFV56	WO2016146985A1_MZ3	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](NC(=O)[C@@H](Cc2ccccc2)NC(=O)COCCOCCOCCNC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)C(C)(C)C)cc1	C58H69ClN10O9S2	BRD4	O60885	VHL	WO-2016146985-A1
TPD-BYHRBF	SCHEMBL18090253	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[2-[2-[[2-[6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]acetyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL19875315	COc1ccc2c(c1)C(c1ccc(Cl)cc1)=NC(CC(=O)NCCOCCOCCOCCOCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(-c3scnc3C)cc1)C(C)(C)C)c1nnc(C)n1-2	C52H64ClN9O10S	BRD4	O60885	VHL	WO-2016146985-A1
TPD-M1TPPK	WO2016146985A1_MZP-12	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCNNN)C(C)(C)C)cc1	C30H47N7O7S	BRD4	O60885	VHL	WO-2016146985-A1
TPD-FTW6RV	SCHEMBL18090233	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[2-[[2-[6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]acetyl]amino]ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL19875317	COc1ccc2c(c1)C(c1ccc(Cl)cc1)=NC(CC(=O)NCCOCCOCCOCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(-c3scnc3C)cc1)C(C)(C)C)c1nnc(C)n1-2	C50H60ClN9O9S	BRD4	O60885	VHL	WO-2016146985-A1
TPD-KDQMPA	WO2016146985A1_MZP-20	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)[C@H](Cc2ccccc2)NC(=O)COCCOCCOCCNNN)C(C)(C)C)cc1	C39H56N8O8S	BRD4	O60885	VHL	WO-2016146985-A1
TPD-5877XG	SCHEMBL18090234	(2S,4R)-1-[(2S)-2-[[(2S)-2-[[2-[2-[2-[2-[[2-[6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]acetyl]amino]ethoxy]ethoxy]ethoxy]acetyl]amino]-3-phenylpropanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL19875326	COc1ccc2c(c1)C(c1ccc(Cl)cc1)=NC(CC(=O)NCCOCCOCCOCC(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(-c3scnc3C)cc1)C(C)(C)C)c1nnc(C)n1-2	C59H69ClN10O10S	BRD4	O60885	VHL	WO-2016146985-A1
TPD-D1XW93	WO2016146985A1_MZP-39	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCNNN)C(C)(C)C)cc1	C30H47N7O7S	BRD4	O60885	VHL	WO-2016146985-A1
TPD-KFXN97	MZP-54	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[2-[[4-[(2S,4R)-1-acetyl-4-(4-chloroanilino)-2-methyl-3,4-dihydro-2H-quinolin-6-yl]benzoyl]amino]ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; 2010159-47-2; CHEMBL4229193; (2S,4R)-1-[(2S)-2-[[2-[2-[2-[2-[[4-[(2S,4R)-1-acetyl-4-(4-chloroanilino)-2-methyl-3,4-dihydro-2H-quinolin-6-yl]benzoyl]amino]ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; (2S,4R)-1-((S)-1-(4-((2S,4R)-1-Acetyl-4-((4-chlorophenyl)amino)-2-methyl-1,2,3,4-tetrahydroquinolin-6-yl)phenyl)-15-(tert-butyl)-1,13-dioxo-5,8,11-trioxa-2,14-diazahexadecan-16-oyl)-4-hydroxy-N-(4-(4-methylthiazol-5-yl)benzyl)pyrrolidine-2-carboxamide; orb1707894; SCHEMBL18090252; SCHEMBL29597119; GLXC-25635; EX-A8737; KFD15947; BDBM50459876; AKOS037653371; BP-40149; DA-75838; HY-112376; CS-0045307; G16491; EN300-22955193; (2S,4R)-1-[(2S)-2-[2-(2-{2-[2-({4-[(2S,4R)-1-acetyl-4-[(4-chlorophenyl)amino]-2-methyl-1,2,3,4-tetrahydroquinolin-6-yl]phenyl}formamido)ethoxy]ethoxy}ethoxy)acetamido]-3,3-dimethylbutanoyl]-4-hydroxy-N-{[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl}pyrrolidine-2-carboxamide	CC(=O)N1c2ccc(-c3ccc(C(=O)NCCOCCOCCOCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)NCc4ccc(-c5scnc5C)cc4)C(C)(C)C)cc3)cc2[C@H](Nc2ccc(Cl)cc2)C[C@@H]1C	C55H66ClN7O9S	BRD4	O60885	VHL	WO-2016146985-A1
TPD-G7P393	MZP-55	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[2-[2-[[4-[(2S,4R)-1-acetyl-4-(4-chloroanilino)-2-methyl-3,4-dihydro-2H-quinolin-6-yl]benzoyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; 2010159-48-3; CHEMBL4226376; (2S,4R)-1-[(2S)-2-[[2-[2-[2-[2-[2-[[4-[(2S,4R)-1-acetyl-4-(4-chloroanilino)-2-methyl-3,4-dihydro-2H-quinolin-6-yl]benzoyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; orb1707893; SCHEMBL18076334; SCHEMBL29597868; EX-A8738; KFD15948; BDBM50459881; AKOS037653403; BP-40147; DA-75839; HY-112377; CS-0045308; G16492; (2S,4R)-1-((S)-1-(4-((2S,4R)-1-acetyl-4-((4-chlorophenyl)amino)-2-methyl-1,2,3,4-tetrahydroquinolin-6-yl)phenyl)-18-(tert-butyl)-1,16-dioxo-5,8,11,14-tetraoxa-2,17-diazanonadecan-19-oyl)-4-hydroxy-N-(4-(4-methylthiazol-5-yl)benzyl)pyrrolidine-2-carboxamide	CC(=O)N1c2ccc(-c3ccc(C(=O)NCCOCCOCCOCCOCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)NCc4ccc(-c5scnc5C)cc4)C(C)(C)C)cc3)cc2[C@H](Nc2ccc(Cl)cc2)C[C@@H]1C	C57H70ClN7O10S	BRD4	O60885	VHL	WO-2016146985-A1
TPD-QO3U4Z	WO2016146985A1_MZP-59	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCNNN)C(C)(C)C)cc1	C28H43N7O6S	BRD4	O60885	VHL	WO-2016146985-A1
TPD-XH80Q5	WO2016146985A1_MZP-60	.	Cc1ccc(C2=N[C@@H](CC(=O)NCCOCCOCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCc3ccc(-c4scnc4C)cc3)C(C)(C)C)c3nnc(C)n3-c3sc(C)c(C)c32)cc1	C48H59N9O7S2	BRD4	O60885	VHL	WO-2016146985-A1
TPD-7RK4T1	CHEMBL4227834	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[[4-[(2S,4R)-1-acetyl-4-(4-chloroanilino)-2-methyl-3,4-dihydro-2H-quinolin-6-yl]benzoyl]amino]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; MZP-61; SCHEMBL18090246; SCHEMBL29597479; BDBM50459878	CC(=O)N1c2ccc(-c3ccc(C(=O)NCCOCCOCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)NCc4ccc(-c5scnc5C)cc4)C(C)(C)C)cc3)cc2[C@H](Nc2ccc(Cl)cc2)C[C@@H]1C	C53H62ClN7O8S	BRD4	O60885	VHL	WO-2016146985-A1
TPD-9P7IM0	WO2016146985A1_MZP-9	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCOCCNNN)C(C)(C)C)cc1	C32H51N7O8S	BRD4	O60885	VHL	WO-2016146985-A1
TPD-GL0J9V	SCHEMBL18063870	US10730870, Example 1; US10730870, Example 1; BDBM454838	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=C(Br)N=CS2)C=C1)N1CC2=C(C=CC=C2)C1=O	C28H29BrN4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-G2K3NS	SCHEMBL18063896	US10730870, Example 10; BDBM454847; US10730870, Example 10	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C(C)C)N3CC4=C(C=C(F)C=C4)C3=O)C=C2)SC=N1	C29H31FN4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-QZKOD1	SCHEMBL18074873	(2S,4R)-4-hydroxy-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]-N-[[4-(2H-triazol-4-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=CN=NN2)C=C1)N1CC2=C(C=CC=C2)C1=O	C27H30N6O4	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-JWQJ5K	SCHEMBL18063979	US10730870, Example 101; BDBM454934; US10730870, Example 101	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=NOC=N2)C=C1)N1CC2=C(C=CC=C2)C1=O	C27H29N5O5	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-3IFK6W	SCHEMBL18063692	US10730870, Example 102; US10730870, Example 102; FEQYFWWATDFOMX-PUHATCMVSA-N; BDBM454935	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=C(C(F)(F)F)N=CS2)C=C1)N1CC2=C(C=CC=C2)C1=O	C29H29F3N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-6G8IXF	SCHEMBL18063688	US10730870, Example 103; BDBM454936; US10730870, Example 103	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C=C2)N(C)C=N1	C30H35N5O4	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-8L5C12	SCHEMBL18063731	US10730870, Example 104; BDBM454937; US10730870, Example 104	CC[C@H](C)[C@H](NCCC1=CC=CC=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=C(C)N=CS2)C=C1	C30H38N4O3S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-HUVEZU	SCHEMBL18063679	US10730870, Example 105; BDBM454938; US10730870, Example 105	CC[C@H](C)[C@H](NC(C)C1=CC=CC=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=C(C)N=CS2)C=C1	C30H38N4O3S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-JLV0I9	SCHEMBL18063882	US10730870, Example 106; BDBM454939; US10730870, Example 106	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C=C2)N=CN1C	C30H35N5O4	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-ZMU14B	SCHEMBL16267129	US10730870, Example 107; BDBM454940; US10730870, Example 107	CC[C@H](NC(C)=O)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=C(C)N=CS2)C=C1	C22H28N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-332FG2	CHEMBL4226127	(2S,4R)-1-[(2S)-2-[acetyl(methyl)amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL18063690; BDBM50459952	CC(=O)N(C)[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=C(C)N=CS2)C=C1)C(C)(C)C	C25H34N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-7NFXOD	SCHEMBL18063714	US10730870, Example 109; BDBM454942; US10730870, Example 109	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C3=CC(OC4=CC=CC=C4)=CC=C3)C=C2)SC=N1	C28H27N3O3S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-3V206A	SCHEMBL18063910	US10730870, Example 11; BDBM454848; US10730870, Example 11	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=C(Br)C=C4)C3=O)C=C2)SC=N1	C29H31BrN4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-18397P	SCHEMBL18063930	US11512083, Example 110; BDBM581946; US11512083, Example 110	CC1=C(C2=CC=C(CNC(=S)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C=C2)SC=N1	C29H32N4O3S2	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-TCH9RY	SCHEMBL18063869	US10730870, Example 111; BDBM454944; US10730870, Example 111	COC1=CC(=O)N([C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(C3=C(C)N=CS3)C=C2)C(C)C)C1	C26H32N4O5S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-I6QXD6	SCHEMBL18063838	US10730870, Example 112; SCHEMBL18063843; BDBM454945; US10730870, Example 112	CC1=C(C2=CC=C(CN/C(=N/C#N)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C=C2)SC=N1	C30H32N6O3S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-T35YH7	SCHEMBL18063819	US10730870, Example 113; BDBM454946; US10730870, Example 113	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2CC2)C=C1)N1CC2=C(C=CC=C2)C1=O	C28H33N3O4	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-F6FF1S	SCHEMBL18063969	US10730870, Example 114; BDBM454947; US10730870, Example 114	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2CCC2)C=C1)N1CC2=C(C=CC=C2)C1=O	C29H35N3O4	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-M4EYW4	SCHEMBL18063818	US10730870, Example 115; BDBM454948; US10730870, Example 115	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2CCCC2)C=C1)N1CC2=C(C=CC=C2)C1=O	C30H37N3O4	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-SHL16A	SCHEMBL18063755	US10730870, Example 116; BDBM454949; US10730870, Example 116	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=CCCC2)C=C1)N1CC2=C(C=CC=C2)C1=O	C30H35N3O4	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-YE3MBL	SCHEMBL18063779	US10730870, Example 117; BDBM454950; US10730870, Example 117	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2CCCCC2)C=C1)N1CC2=C(C=CC=C2)C1=O	C31H39N3O4	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-8I3YI8	SCHEMBL18063719	US10730870, Example 118; BDBM454951; US10730870, Example 118	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2CCOCC2)C=C1)N1CC2=C(C=CC=C2)C1=O	C30H37N3O5	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-GRVJS3	SCHEMBL18063920	(2S,4R)-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-4-sulfanylpyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](S)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C=C2)SC=N1	C29H32N4O3S2	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-REM5P4	SCHEMBL27116200	(2S,4R)-4-hydroxy-1-[(2S)-3-methyl-2-(propanoylamino)butanoyl]-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=C(C)N=CS2)C=C1)C(C)C	C24H32N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-BY619D	SCHEMBL18063883	US10730870, Example 120; SCHEMBL18063888; BDBM454952; US10730870, Example 120	CO/N=C(/NCC1=CC=C(C2=C(C)N=CS2)C=C1)[C@@H]1C[C@@H](O)CN1C(=O)[C@H](C(C)C)N1CC2=C(C=CC=C2)C1=O	C30H35N5O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-A538D5	SCHEMBL18063840	US10730870, Example 121; BDBM454953; US10730870, Example 121	CC1=C(C2=CC=C(CNC[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C=C2)SC=N1	C29H34N4O3S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-75X63V	SCHEMBL18088944	US10730870, Example 122; BDBM454954; US10730870, Example 122	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)[C@H](C)NC(=O)OC(C)(C)C)C(C)(C)C)C=C2)SC=N1	C30H43N5O6S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-EWZO4Y	SCHEMBL18063863	US10730870, Example 123; BDBM454955; US10730870, Example 123	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)[C@H](C)N)C(C)(C)C)C=C2)SC=N1	C25H35N5O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-QWF6BG	VH032-NH-CO-CH2-NHBoc	VH032-NH-CO-CH2-NHBoc; 2010986-19-1; tert-Butyl (2-(((S)-1-((2S,4R)-4-hydroxy-2-((4-(4-methylthiazol-5-yl)benzyl)carbamoyl)pyrrolidin-1-yl)-3,3-dimethyl-1-oxobutan-2-yl)amino)-2-oxoethyl)carbamate; SCHEMBL18063871; BDBM454956; US10730870, Example 124; HY-W584525; DA-58999; tert-butyl N-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethyl]carbamate; CS-0637365	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CNC(=O)OC(C)(C)C)C(C)(C)C)C=C2)SC=N1	C29H41N5O6S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-HIHTFE	(S,R,S)-AHPC-C1-NH2	(S,R,S)-Ahpc-C1-NH2; 2010986-20-4; (2S,4R)-1-((S)-2-(2-Aminoacetamido)-3,3-dimethylbutanoyl)-4-hydroxy-N-(4-(4-methylthiazol-5-yl)benzyl)pyrrolidine-2-carboxamide; orb1691323; SCHEMBL18064008; BDBM454957; US10730870, Example 125; AKOS040757201; (2S,4R)-1-[(2S)-2-[(2-aminoacetyl)amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; DA-59699; HY-138861; CS-0169553	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN)C(C)(C)C)C=C2)SC=N1	C24H33N5O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-JB7AB7	SCHEMBL18063864	US10730870, Example 126; BDBM454958; US10730870, Example 126	CC1=C(C2=CC=C(CNC(=N)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C=C2)SC=N1	C29H33N5O3S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-Y9RXX6	SCHEMBL18063942	US10730870, Example 127; BDBM454959; US10730870, Example 127	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2(O)COC2)C=C1)N1CC2=C(C=CC=C2)C1=O	C28H33N3O6	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-Z38WKM	SCHEMBL20325614	(2S,4R)-4-hydroxy-2-methyl-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@]3(C)C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C=C2)SC=N1	C30H34N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-CWKH5M	WO2016149668A1_13	.	CCCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=C(C)N=CS2)C=C1)C(C)C	C25H34N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-37CHUS	SCHEMBL18063814	US10730870, Example 130; BDBM454962; US10730870, Example 130	CC(=O)N[C@H](C(=S)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=C(C)N=CS2)C=C1)C(C)C	C23H30N4O3S2	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-CQWP6T	SCHEMBL18063830	US10730870, Example 133; BDBM454964; US10730870, Example 133	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C=C2)OC=N1	C29H32N4O5	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-ZXISXO	SCHEMBL18063955	US10730870, Example 134; BDBM454965; US10730870, Example 134	CC(=O)N(C)[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=C(C)N=CS2)C=C1)C(C)C	C24H32N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-Z5L7F1	CHEMBL3108882	(2S,4R)-4-hydroxy-1-(2-(3-methylisoxazol-5-yl)acetyl)-N-(4-(4-methylthiazol-5-yl)benzyl)pyrrolidine-2-carboxamide; SCHEMBL15111829; FEFYMYQFVDBQAU-MJGOQNOKSA-N; BDBM50446139; (2S,4R)-4-hydroxy-1-(2-(3-methylisoxazol-5-yl)acetyl)-N-(4-(4-methylthiazol-5-yl)benzyl)pyrrolidine-2-carboxamide	CC1=NOC(CC(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(C3=C(C)N=CS3)C=C2)=C1	C22H24N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-KHFMOG	WO2016149668A1_136	.	CC(C)[C@@H](C(=O)N1C[C@H](O)CC1C(=O)NCC1=CC=C(C2=CC=NO2)C=C1)N1CC2=C(C=CC=C2)C1=O	C28H30N4O5	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-2CRZXN	WO2016149668A1_137	(4R)-4-hydroxy-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]-N-[[4-(1,2-oxazol-4-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC(C)[C@@H](C(=O)N1C[C@H](O)CC1C(=O)NCC1=CC=C(C2=CON=C2)C=C1)N1CC2=C(C=CC=C2)C1=O	C28H30N4O5	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-S0CNEV	SCHEMBL18063801	US11512083, Example 138; BDBM581972; US11512083, Example 138	CC1=NOC([C@@H](C)C(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(C3=C(C)N=CS3)C=C2)=C1	C23H26N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-81M92R	SCHEMBL18063926	US10730870, Example 139; BDBM454970; US10730870, Example 139	CC1=NOC([C@H](C)C(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(C3=C(C)N=CS3)C=C2)=C1	C23H26N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-XXEYF0	WO2016149668A1_14	(2S,4R)-1-[(2S)-2-(2,2-dimethylpropanoylamino)-3-methylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C(C)(C)C)C(C)C)C=C2)SC=N1	C26H36N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-TWFMIO	SCHEMBL18063867	US10730870, Example 140; BDBM454971; US10730870, Example 140	CC1=NOC(C(C)(C)C(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(C3=C(C)N=CS3)C=C2)=C1	C24H28N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-SEMS2L	SCHEMBL18063740	US10730870, Example 141; BDBM454972; US10730870, Example 141	CC1=NOC(C(C(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(C3=C(C)N=CS3)C=C2)C(C)C)=C1	C25H30N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-P8CU1G	SCHEMBL18063834	US10730870, Example 142; BDBM454973; US10730870, Example 142	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@](C)(O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C=C2)SC=N1	C30H34N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-6A3UF0	SCHEMBL18063687	US10730870, Example 143; BDBM454974; US10730870, Example 143	CCC(C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=C(C)N=CS2)C=C1)C1=CC(C)=NO1	C24H28N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-M7FPFK	SCHEMBL18063812	(2S,4S)-4-hydroxy-4-(hydroxymethyl)-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@](O)(CO)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C=C2)SC=N1	C30H34N4O5S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-XXXZF1	SCHEMBL18063891	US10730870, Example 138; BDBM454969; US10730870, Example 138; US10730870, Example 145	CC1=NOC([C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(C3=C(C)N=CS3)C=C2)C(C)C)=C1	C25H30N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-588J8K	SCHEMBL18063917	US10730870, Example 146; BDBM454976; US10730870, Example 146	CC1=NOC([C@@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(C3=C(C)N=CS3)C=C2)C(C)C)=C1	C25H30N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-MW0A09	SCHEMBL18063973	US10730870, Example 147; BDBM454977; US10730870, Example 147	CC1=C(C2=CC=C(CNC(=O)[C@@H]3[C@@H](O)[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C=C2)SC=N1	C29H32N4O5S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-NBXJ2J	SCHEMBL18064010	US10730870, Example 148; BDBM454978; US10730870, Example 148	CCC[C@H](NC(C)=O)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=C(C)N=CS2)C=C1	C23H30N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-B4SRZ7	SCHEMBL18063686	(2S,4R)-4-hydroxy-1-[(2R)-2-(3-methyl-1,2-oxazol-5-yl)butanoyl]-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=C(C)N=CS2)C=C1)C1=CC(C)=NO1	C24H28N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-9XTZF4	SCHEMBL18063978	US10730870, Example 15; BDBM454852; US10730870, Example 15	COC1=CC=CC2=C1C(=O)N([C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C3=C(C)N=CS3)C=C1)C(C)C)C2	C30H34N4O5S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-0XAHMI	SCHEMBL18063983	(2S,4R)-1-[(2R)-3,3-dimethyl-2-(3-methyl-1,2-oxazol-5-yl)butanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=NOC([C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)=C1	C26H32N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-6BAUVT	SCHEMBL18063858	(2S,4R)-1-[(2R)-3,3-dimethyl-2-(3-methyl-1,2-oxazol-5-yl)butanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-oxazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=NOC([C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(C3=C(C)N=CO3)C=C2)C(C)(C)C)=C1	C26H32N4O5	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-6RVVP6	SCHEMBL18063990	(2S,4R)-4-hydroxy-1-[(2R)-3-methyl-2-(3-methyl-1,2-oxazol-5-yl)butanoyl]-N-[[4-(4-methyl-1,3-oxazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=NOC([C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(C3=C(C)N=CO3)C=C2)C(C)C)=C1	C25H30N4O5	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-4R8523	SCHEMBL18063901	(2S,4R)-4-hydroxy-1-[(2R)-2-(3-methyl-1,2-oxazol-5-yl)butanoyl]-N-[[4-(4-methyl-1,3-oxazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=C(C)N=CO2)C=C1)C1=CC(C)=NO1	C24H28N4O5	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-X32SUF	SCHEMBL18063831	(2S,4R)-4-hydroxy-1-[(2R)-2-(3-methyl-1,2-oxazol-5-yl)butanoyl]-N-[[4-(1,3-oxazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=CN=CO2)C=C1)C1=CC(C)=NO1	C23H26N4O5	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-OL3VZS	SCHEMBL18063703	(2S,4R)-4-hydroxy-1-[(2R)-2-(3-methyl-1,2-oxazol-5-yl)butanoyl]-N-[[4-(1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=CN=CS2)C=C1)C1=CC(C)=NO1	C23H26N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-GHJ0C5	SCHEMBL18063786	(2S,4R)-1-[(2R)-3,3-dimethyl-2-(3-methyl-1,2-oxazol-5-yl)butanoyl]-4-hydroxy-N-[[4-(1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=NOC([C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(C3=CN=CS3)C=C2)C(C)(C)C)=C1	C25H30N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-0XQDIJ	SCHEMBL18063846	(2S,4R)-4-hydroxy-1-[(2R)-3-methyl-2-(3-methyl-1,2-oxazol-5-yl)butanoyl]-N-[[4-(1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=NOC([C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(C3=CN=CS3)C=C2)C(C)C)=C1	C24H28N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-SN97I7	SCHEMBL18063825	(2S,4R)-4-hydroxy-1-[(2R)-3-methyl-2-(3-methyl-1,2-oxazol-5-yl)butanoyl]-N-[(1S)-1-[4-(1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=NOC([C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=CN=CS3)C=C2)C(C)C)=C1	C25H30N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-FKHXNO	SCHEMBL18063764	(2S,4R)-4-hydroxy-1-[(2R)-2-(3-methyl-1,2-oxazol-5-yl)butanoyl]-N-[(1S)-1-[4-(1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CN=CS2)C=C1)C1=CC(C)=NO1	C24H28N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-7EPGH3	SCHEMBL18064018	US10730870, Example 16; SCHEMBL31058425; BDBM454853; US10730870, Example 16	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC(F)=C4)C3=O)C=C2)SC=N1	C29H31FN4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-U3KASY	SCHEMBL18063808	(2S,4R)-1-[(2R)-3,3-dimethyl-2-(3-methyl-1,2-oxazol-5-yl)butanoyl]-4-hydroxy-N-[(1S)-1-[4-(1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=NOC([C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=CN=CS3)C=C2)C(C)(C)C)=C1	C26H32N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-A3VSMZ	SCHEMBL18063933	(2S,4R)-1-[(2R)-3,3-dimethyl-2-(3-methyl-1,2-oxazol-5-yl)butanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=NOC([C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)=C1	C27H34N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-3BZSS2	SCHEMBL18063710	(2S,4R)-4-hydroxy-1-[(2R)-2-(3-methyl-1,2-oxazol-5-yl)butanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=C(C)N=CS2)C=C1)C1=CC(C)=NO1	C25H30N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-WDQ229	SCHEMBL18063981	US10730870, Example 205; BDBM454979; US10730870, Example 205	CC1=NOC([C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=C(C)N=CS3)C=C2)C(C)C)=C1	C26H32N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-XQB79V	SCHEMBL18063742	(2S,4R)-4-hydroxy-1-[(2R)-3-methyl-2-(3-methyl-1,2-oxazol-5-yl)butanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-oxazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=NOC([C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=C(C)N=CO3)C=C2)C(C)C)=C1	C26H32N4O5	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-MFK5EE	SCHEMBL18064015	(2S,4R)-1-[(2R)-3,3-dimethyl-2-(3-methyl-1,2-oxazol-5-yl)butanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-oxazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=NOC([C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=C(C)N=CO3)C=C2)C(C)(C)C)=C1	C27H34N4O5	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-R7BEE4	SCHEMBL18063876	(2S,4R)-4-hydroxy-1-[(2R)-2-(3-methyl-1,2-oxazol-5-yl)butanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-oxazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=C(C)N=CO2)C=C1)C1=CC(C)=NO1	C25H30N4O5	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-1NEPUE	SCHEMBL18063806	(2S,4R)-4-hydroxy-1-[(2R)-2-(3-methyl-1,2-oxazol-5-yl)butanoyl]-N-[(1S)-1-[4-(1,3-oxazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CN=CO2)C=C1)C1=CC(C)=NO1	C24H28N4O5	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-IPGUHF	SCHEMBL18063715	(2S,4R)-1-[(2R)-3,3-dimethyl-2-(3-methyl-1,2-oxazol-5-yl)butanoyl]-4-hydroxy-N-[(1S)-1-[4-(1,3-oxazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=NOC([C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=CN=CO3)C=C2)C(C)(C)C)=C1	C26H32N4O5	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-D8QQ23	SCHEMBL18063712	(2S,4R)-4-hydroxy-1-[(2R)-3-methyl-2-(3-methyl-1,2-oxazol-5-yl)butanoyl]-N-[(1S)-1-[4-(1,3-oxazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=NOC([C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=CN=CO3)C=C2)C(C)C)=C1	C25H30N4O5	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-M76LLA	SCHEMBL18063705	US10730870, Example 17; BDBM454854; US10730870, Example 17	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=C(C#N)C=C4)C3=O)C=C2)SC=N1	C30H31N5O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-W3G4BP	SCHEMBL18063943	(2S,4R)-4-hydroxy-1-[(2S)-3-methyl-2-(3-methyl-1,2-thiazol-5-yl)butanoyl]-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=NSC([C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(C3=C(C)N=CS3)C=C2)C(C)C)=C1	C25H30N4O3S2	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-L9YINB	SCHEMBL18063758	(2S,4R)-4-hydroxy-1-[(2S)-3-methyl-2-(3-methyl-1,2,4-thiadiazol-5-yl)butanoyl]-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=NSC([C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(C3=C(C)N=CS3)C=C2)C(C)C)=N1	C24H29N5O3S2	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-SXHJTV	SCHEMBL18063928	(2S,4R)-4-hydroxy-1-[(2R)-3-methyl-2-(3-methyl-1,2,4-oxadiazol-5-yl)butanoyl]-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=NOC([C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(C3=C(C)N=CS3)C=C2)C(C)C)=N1	C24H29N5O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-PS36IY	SCHEMBL18063829	(2S,4R)-4-hydroxy-1-[(2R)-3-methyl-2-(5-methyl-1H-1,2,4-triazol-3-yl)butanoyl]-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL20330118; SCHEMBL21472204	CC1=NN=C([C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(C3=C(C)N=CS3)C=C2)C(C)C)N1	C24H30N6O3S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-NSYPLO	SCHEMBL18063699	(2S,4R)-4-hydroxy-1-[(2R)-3-methyl-2-(5-methyl-1,3,4-oxadiazol-2-yl)butanoyl]-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=NN=C([C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(C3=C(C)N=CS3)C=C2)C(C)C)O1	C24H29N5O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-VUDL0N	SCHEMBL18063972	(2S,4R)-4-hydroxy-1-[(2S)-3-methyl-2-(5-methyl-1,3,4-thiadiazol-2-yl)butanoyl]-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=NN=C([C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(C3=C(C)N=CS3)C=C2)C(C)C)S1	C24H29N5O3S2	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-LUT3X4	SCHEMBL18063790	(2S,4R)-4-hydroxy-1-[(2R)-3-methyl-2-(5-methyl-1,2-oxazol-3-yl)butanoyl]-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=CC([C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(C3=C(C)N=CS3)C=C2)C(C)C)=NO1	C25H30N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-VSM61E	SCHEMBL18063697	(2S,4R)-4-hydroxy-1-[(2R)-3-methyl-2-(5-methyl-1,2-thiazol-3-yl)butanoyl]-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=CC([C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(C3=C(C)N=CS3)C=C2)C(C)C)=NS1	C25H30N4O3S2	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-CEFCXZ	SCHEMBL18063918	(2S,4R)-4-hydroxy-1-[(2R)-3-methyl-2-(5-methyl-1,2,4-thiadiazol-3-yl)butanoyl]-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=NC([C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(C3=C(C)N=CS3)C=C2)C(C)C)=NS1	C24H29N5O3S2	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-9S01G1	SCHEMBL18063716	(2S,4R)-4-hydroxy-1-[(2R)-3-methyl-2-(5-methyl-1,2,4-oxadiazol-3-yl)butanoyl]-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=NC([C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(C3=C(C)N=CS3)C=C2)C(C)C)=NO1	C24H29N5O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-1F0L1G	SCHEMBL18063802	US10730870, Example 18; BDBM454855; US10730870, Example 18	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CC(C)C)C(C)(C)C)C=C2)SC=N1	C27H38N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-3IOBSZ	SCHEMBL18063743	(2S,4R)-4-hydroxy-1-[(2R)-3-methyl-2-(5-methyl-1H-pyrazol-3-yl)butanoyl]-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=CC([C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(C3=C(C)N=CS3)C=C2)C(C)C)=NN1	C25H31N5O3S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-INQ358	SCHEMBL18063775	(2S,4R)-4-hydroxy-1-[(2R)-3-methyl-2-(5-methyl-1H-imidazol-2-yl)butanoyl]-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL21025628	CC1=CN=C([C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(C3=C(C)N=CS3)C=C2)C(C)C)N1	C25H31N5O3S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-D6Y390	SCHEMBL18063899	(2S,4R)-4-hydroxy-1-[(2R)-3-methyl-2-(5-methyl-1,3-oxazol-2-yl)butanoyl]-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=CN=C([C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(C3=C(C)N=CS3)C=C2)C(C)C)O1	C25H30N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-4L1IV4	SCHEMBL18063694	(2S,4R)-4-hydroxy-1-[(2S)-3-methyl-2-(5-methyl-1,3-thiazol-2-yl)butanoyl]-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=CN=C([C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(C3=C(C)N=CS3)C=C2)C(C)C)S1	C25H30N4O3S2	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-17OVZ7	SCHEMBL18063938	(2S,4R)-4-hydroxy-1-[(2R)-3-methyl-2-(4-methyl-1,3-oxazol-2-yl)butanoyl]-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=COC([C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(C3=C(C)N=CS3)C=C2)C(C)C)=N1	C25H30N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-OWJ1KR	SCHEMBL18063720	(2S,4R)-4-hydroxy-1-[(2S)-3-methyl-2-(4-methyl-1,3-thiazol-2-yl)butanoyl]-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=CSC([C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(C3=C(C)N=CS3)C=C2)C(C)C)=N1	C25H30N4O3S2	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-SN76RZ	SCHEMBL18063997	(2S,4R)-4-hydroxy-1-[(2R)-3-methyl-2-(2-methyl-1,3-oxazol-4-yl)butanoyl]-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=NC([C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(C3=C(C)N=CS3)C=C2)C(C)C)=CO1	C25H30N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-S02DAF	SCHEMBL18063807	(2S,4R)-4-hydroxy-1-[(2R)-3-methyl-2-(2-methyl-1,3-thiazol-4-yl)butanoyl]-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=NC([C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(C3=C(C)N=CS3)C=C2)C(C)C)=CS1	C25H30N4O3S2	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-LX2HGI	SCHEMBL18063946	(2S,4R)-4-hydroxy-1-[(2R)-3-methyl-2-(2-methyl-1H-imidazol-5-yl)butanoyl]-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL23350147	CC1=NC=C([C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(C3=C(C)N=CS3)C=C2)C(C)C)N1	C25H31N5O3S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-MIR7HQ	SCHEMBL18064012	(2S,4R)-4-hydroxy-1-[(2R)-3-methyl-2-phenylbutanoyl]-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC=CC=C3)C(C)C)C=C2)SC=N1	C27H31N3O3S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-YRM9AF	(S,R,S)-AHPC-CO-C-cyclohexane	(S,R,S)-AHPC-CO-C-cyclohexane; 2010985-17-6; orb2665414; SCHEMBL18063877; BDBM454856; US10730870, Example 19; EX-A13164; HY-163933	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CC3CCCCC3)C(C)(C)C)C=C2)SC=N1	C30H42N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-UAV8KE	SCHEMBL18063922	(2S,4R)-4-hydroxy-1-[(2R)-3-methyl-2-pyridin-2-ylbutanoyl]-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC=CC=N3)C(C)C)C=C2)SC=N1	C26H30N4O3S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-O8QKVH	SCHEMBL18063769	(2S,4R)-4-hydroxy-1-[(2R)-3-methyl-2-pyridazin-3-ylbutanoyl]-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC=CN=N3)C(C)C)C=C2)SC=N1	C25H29N5O3S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-X1R4KO	SCHEMBL18063824	(2S,4R)-4-hydroxy-1-[(2R)-3-methyl-2-pyridin-3-ylbutanoyl]-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC=CN=C3)C(C)C)C=C2)SC=N1	C26H30N4O3S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-X5EMDN	SCHEMBL18063732	(2S,4R)-4-hydroxy-1-[(2R)-3-methyl-2-pyrazin-2-ylbutanoyl]-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=NC=CN=C3)C(C)C)C=C2)SC=N1	C25H29N5O3S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-KFYASG	SCHEMBL18088945	(2S,4R)-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-1-[(2R)-3-methyl-2-(1,2,4-triazin-3-yl)butanoyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=NC=CN=N3)C(C)C)C=C2)SC=N1	C24H28N6O3S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-4X8YVT	SCHEMBL18063707	(2S,4R)-1-[(2S)-2-acetamido-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-[4-(hydroxymethyl)-1,3-thiazol-5-yl]phenyl]methyl]pyrrolidine-2-carboxamide	CC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=C(CO)N=CS2)C=C1)C(C)(C)C	C24H32N4O5S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-RBF930	SCHEMBL18063889	(2S,4R)-1-[(2S)-2-acetamido-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methylthiadiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=C(C)N=NS2)C=C1)C(C)(C)C	C24H33N5O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-JO8QJG	SCHEMBL18063894	(2S,4R)-4-hydroxy-N-[(1S)-1-[4-[4-(hydroxymethyl)thiadiazol-5-yl]phenyl]ethyl]-1-[(2S)-3-methyl-2-(4-methylimidazol-1-yl)butanoyl]pyrrolidine-2-carboxamide	CC1=CN([C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=C(CO)N=NS3)C=C2)C(C)C)C=N1	C25H32N6O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-FVCYG4	SCHEMBL18063734	(2S,4R)-4-hydroxy-1-[(2S)-3-methyl-2-(4-methylpyrazol-1-yl)butanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=CN([C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=C(C)N=CS3)C=C2)C(C)C)N=C1	C26H33N5O3S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-WVT195	SCHEMBL18063895	US10730870, Example 2; US10730870, Example 2; BDBM454839	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=C(C3CC3)N=CS2)C=C1)N1CC2=C(C=CC=C2)C1=O	C31H34N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-EP0TTX	SCHEMBL18063681	US10730870, Example 20; BDBM454857; US10730870, Example 20	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCC3CCCCC3)C(C)(C)C)C=C2)SC=N1	C31H44N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-SOVMV9	SCHEMBL18063961	(2S,4R)-4-hydroxy-1-[(2S)-3-methyl-2-(4-phenylpyrazol-1-yl)butanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C(C4=CC=CC=C4)C=N3)C=C2)SC=N1	C31H35N5O3S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-E07TEN	SCHEMBL18063762	(2S,4R)-4-hydroxy-1-[(2S)-3-methyl-2-(4-pyridin-3-ylpyrazol-1-yl)butanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL31058426	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C(C4=CC=CN=C4)C=N3)C=C2)SC=N1	C30H34N6O3S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-2FVGNO	SCHEMBL18088946	(2S,4R)-4-hydroxy-1-[(2S)-3-methyl-2-(4-pyridin-4-ylpyrazol-1-yl)butanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C(C4=CC=NC=C4)C=N3)C=C2)SC=N1	C30H34N6O3S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-WPQDQW	SCHEMBL18063892	(2S,4R)-4-hydroxy-1-[(2S)-2-(4-methoxypyrazol-1-yl)-3-methylbutanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	COC1=CN([C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=C(C)N=CS3)C=C2)C(C)C)N=C1	C26H33N5O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-L4WJGJ	SCHEMBL18063696	(2S,4R)-4-hydroxy-1-[(2S)-3-methyl-2-(4-pyridin-2-ylpyrazol-1-yl)butanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C(C4=CC=CC=N4)C=N3)C=C2)SC=N1	C30H34N6O3S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-XN5DKG	SCHEMBL18063741	(2S,4R)-4-hydroxy-1-[(2S)-3-methyl-2-(4-phenoxypyrazol-1-yl)butanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C(OC4=CC=CC=C4)C=N3)C=C2)SC=N1	C31H35N5O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-KKIZBP	SCHEMBL18063736	US10730870, Example 207; BDBM454980; US10730870, Example 207	CC[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](C1=CC(C)=NO1)C(C)C)C1=CC=C(C2=C(C)N=CS2)C=C1	C27H34N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-3JT656	SCHEMBL18063739	US10730870, Example 208; BDBM454981; US10730870, Example 208	COC1=NOC([C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(C3=C(C)N=CS3)C=C2)C(C)C)=C1	C25H30N4O5S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-KH88T0	orb2665282	(S,R,S)-AHPC-phenylacetic acid; CHEMBL4783485; SCHEMBL18063879; (S,R,S)-AHPC-phenylacetic acid; BDBM454858; 2010985-19-8; US10730870, Example 21; HY-163934	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CC3=CC=CC=C3)C(C)(C)C)C=C2)SC=N1	C30H36N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-W1VW5Z	SCHEMBL18063773	US10730870, Example 22; BDBM454859; US10730870, Example 22	CSC[C@H](NC(=O)CCC(C)C)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=C(C)N=CS2)C=C1	C26H36N4O4S2	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-199ARY	SCHEMBL18064002	US10730870, Example 23; BDBM454860; US10730870, Example 23	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(Br)C=C1)N1CC2=C(C=CC=C2)C1=O	C25H28BrN3O4	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-L7XLL1	SCHEMBL18064001	US10730870, Example 24; BDBM454861; US10730870, Example 24	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(Br)C=C1)N1CC2=C(C=CC=C2)C1=O	C26H30BrN3O4	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-G9BQFK	SCHEMBL18063947	US10730870, Example 25; SCHEMBL31058434; BDBM454862; US10730870, Example 25	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC(Br)=C4)C3=O)C=C2)SC=N1	C29H31BrN4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-GWLH1N	SCHEMBL18063911	US10730870, Example 26; BDBM454863; US10730870, Example 26	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4Br)C3=O)C=C2)SC=N1	C29H31BrN4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-4VC35V	SCHEMBL18063792	US10730870, Example 27; BDBM454864; US10730870, Example 27	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C(C)C)C(C)(C)C)C=C2)SC=N1	C26H36N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-EKPCW6	SCHEMBL18063909	US10730870, Example 28; BDBM454865; US10730870, Example 28	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCC(C)C)C(C)(C)C)C=C2)SC=N1	C28H40N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-F9IV11	SCHEMBL18063765	US10730870, Example 29; BDBM454866; US10730870, Example 29	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3=CC=CC=C3)C(C)(C)C)C=C2)SC=N1	C29H34N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-Q5SR88	SCHEMBL18063701	US10730870, Example 30; BDBM454867; US10730870, Example 30	CC[C@H](C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=C(C)N=CS2)C=C1)N1CC2=C(C=CC=C2)C1=O	C30H34N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-6XUP10	SCHEMBL18063799	US10730870, Example 31; BDBM454868; US10730870, Example 31	CC[C@H](C)[C@H](NC(=O)CCC(C)C)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=C(C)N=CS2)C=C1	C28H40N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-CIFXEX	SCHEMBL18063751	US10730870, Example 32; BDBM454869; US10730870, Example 32	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NCCC(C)C)C3CCCC3)C=C2)SC=N1	C28H40N4O3S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-9ZFKGJ	SCHEMBL18063783	US10730870, Example 33; BDBM454870; US10730870, Example 33	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4F)C3=O)C=C2)SC=N1	C29H31FN4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-31UGXO	SCHEMBL18063995	US10730870, Example 34; BDBM454871; US10730870, Example 34	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC(C#N)=C4)C3=O)C=C2)SC=N1	C30H31N5O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-5P5X4L	SCHEMBL18063750	US10730870, Example 35; BDBM454872; US10730870, Example 35	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4C#N)C3=O)C=C2)SC=N1	C30H31N5O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-TDOVTL	SCHEMBL18063850	US10730870, Example 36; BDBM454873; US10730870, Example 36	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3CCCCC3)C(C)(C)C)C=C2)SC=N1	C29H40N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-1RGBNM	SCHEMBL18063777	US10730870, Example 37; BDBM454874; US10730870, Example 37	CSC[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=C(C)N=CS2)C=C1)N1CC2=C(C=CC=C2)C1=O	C28H30N4O4S2	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-O7NESS	SCHEMBL18063900	US10730870, Example 38; BDBM454875; US10730870, Example 38	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3CCCC3)N3CC4=C(C=CC=C4)C3=O)C=C2)SC=N1	C31H34N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-O6F7LD	SCHEMBL18063771	US10730870, Example 39; SCHEMBL31058432; BDBM454876; US10730870, Example 39	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C=C2)SC=N1	C30H34N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-MED3V7	SCHEMBL18063965	US10730870, Example 4; US10730870, Example 4; BDBM454841	C=CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C=C2)SC=N1	C30H32N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-XY0Q5J	SCHEMBL18063953	US10730870, Example 40; BDBM454877; US10730870, Example 40	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=CC=CC=C2)C=C1)N1CC2=C(C=CC=C2)C1=O	C31H33N3O4	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-OIEO1B	SCHEMBL18063851	(2S,4R)-4-hydroxy-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]-N-[[4-(1H-pyrazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=CC=NN2)C=C1)N1CC2=C(C=CC=C2)C1=O	C28H31N5O4	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-42LS93	SCHEMBL18063996	US10730870, Example 42; SCHEMBL31058435; BDBM454879; US10730870, Example 42	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C3=O)C(Br)=CC=C4)C=C2)SC=N1	C29H31BrN4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-KSP62N	SCHEMBL18064014	US10730870, Example 43; BDBM454880; US10730870, Example 43	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3=CC=C(C#N)C=C3)C(C)(C)C)C=C2)SC=N1	C30H33N5O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-IZ70ES	SCHEMBL18063852	US10730870, Example 44; BDBM454881; US10730870, Example 44	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCC3=CC=CC=C3)C(C)(C)C)C=C2)SC=N1	C31H38N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-FMFHTW	SCHEMBL18063875	US10730870, Example 45; BDBM454882; US10730870, Example 45	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H]([C@H](C)O)N3CC4=C(C=CC=C4)C3=O)C=C2)SC=N1	C28H30N4O5S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-UC20QZ	SCHEMBL18063685	US10730870, Example 46; BDBM454883; US10730870, Example 46	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C)(C)N3CC4=C(C=CC=C4)C3=O)C=C2)SC=N1	C28H30N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-UZE4RS	SCHEMBL18063963	US10730870, Example 47; BDBM454884; US10730870, Example 47	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C3=O)C(C#N)=CC=C4)C=C2)SC=N1	C30H31N5O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-5LUQ1L	SCHEMBL18063756	US10730870, Example 48; BDBM454885; US10730870, Example 48	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](CS)N3CC4=C(C=CC=C4)C3=O)C=C2)SC=N1	C27H28N4O4S2	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-IMVDYY	SCHEMBL18063988	US10730870, Example 49; BDBM454886; US10730870, Example 49	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C3(N4CC5=C(C=CC=C5)C4=O)CC3)C=C2)SC=N1	C28H28N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-1IBFBC	SCHEMBL18063823	US10730870, Example 5; US10730870, Example 5; BDBM454842	CCC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C=C2)SC=N1	C30H34N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-O4MIX3	SCHEMBL18063735	US10730870, Example 50; BDBM454887; US10730870, Example 50	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C3(N4CC5=C(C=CC=C5)C4=O)CCCC3)C=C2)SC=N1	C30H32N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-JNX8EA	SCHEMBL18063678	US10730870, Example 51; BDBM454888; US10730870, Example 51	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCC(C)C)[C@H](C)O)C=C2)SC=N1	C26H36N4O5S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-KGX0YV	SCHEMBL18063728	US10730870, Example 52; BDBM454889; US10730870, Example 52	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCC(C)C)C3=CC=CS3)C=C2)SC=N1	C28H34N4O4S2	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-P8O2C2	SCHEMBL18063959	US10730870, Example 53; BDBM454890; US10730870, Example 53	COCC#CC1=CC2=C(C=C1)C(=O)N([C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C3=C(C)N=CS3)C=C1)C(C)C)C2	C33H36N4O5S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-EFJHA1	SCHEMBL18063968	US10730870, Example 54; BDBM454891; US10730870, Example 54	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C3(N4CC5=C(C=CC=C5)C4=O)CCCCC3)C=C2)SC=N1	C31H34N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-Y20IKT	SCHEMBL18063737	US10730870, Example 55; BDBM454892; US10730870, Example 55	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C3(N4CC5=C(C=CC=C5)C4=O)CCC3)C=C2)SC=N1	C29H30N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-0JT744	SCHEMBL18063915	US10730870, Example 56; BDBM454893; US10730870, Example 56	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCC(C)C)C3CCCCC3)C=C2)SC=N1	C30H42N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-NZDN0I	SCHEMBL18063813	US10730870, Example 57; BDBM454894; US10730870, Example 57	COCCCC1=CC2=C(C=C1)C(=O)N([C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C3=C(C)N=CS3)C=C1)C(C)C)C2	C33H40N4O5S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-V238OX	SCHEMBL18063857	US10730870, Example 58; BDBM454895; US10730870, Example 58	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3=CC=CS3)N3CC4=C(C=CC=C4)C3=O)C=C2)SC=N1	C30H28N4O4S2	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-34N50C	SCHEMBL18063884	US10730870, Example 59; BDBM454896; US10730870, Example 59	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](CS)NC(=O)CCC(C)C)C=C2)SC=N1	C25H34N4O4S2	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-I5CY1J	VL285	(2S,4R)-4-hydroxy-1-((S)-3-methyl-2-(1-oxoisoindolin-2-yl)butanoyl)-N-(4-(4-methylthiazol-5-yl)benzyl)pyrrolidine-2-carboxamide; 1448188-57-5; (2S,4R)-4-hydroxy-1-((S)-3-methyl-2-(1-oxoisoindolin-2-yl)butanoyl)-N-(4-(4-methylthiazol-5-yl)benzyl)pyrrolidine-2-carboxamide; (2S,4R)-4-hydroxy-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; VL-285; orb1301878; SCHEMBL15126222; C29H32N4O4S; US10730870, Example 6; BDBM454843; (2S,4R)-4-Hydroxy-1-((S)-3-methyl-2-(1-oxoisoindolin-2- yl)butanoyl)-N-(4-(4-methylthiazol-5- yl)benzyl)pyrrolidine-2-carboxamide; (2S,4R)-4-hydroxy-N-{[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl}-1-[(2S)-3-methyl-2-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)butanoyl]pyrrolidine-2-carboxamide; BCP30479; EX-A2978; YHC18857; ZB1525; US10730870, Example 110; AKOS037653339; AT11305; VL-285; VL 285; VL-285?; AC-36306; BP-42122; HY-111663; CS-0089450; Z4119391197; (2S,4R)-4-hydroxy-1-[(2S)-3-methyl-2-(1-oxoisoindolin-2-yl)butanoyl]-N-[[4-(4-methylthiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C=C2)SC=N1	C29H32N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-UDTMUI	SCHEMBL18063986	US10730870, Example 60; BDBM454897; US10730870, Example 60	CC1=C(C2=CC=C(CNC(=O)[C@H]3C[C@H](O)CN3C(=O)[C@@H](CSSC[C@H](NC(=O)CCC(C)C)C(=O)N3C[C@H](O)C[C@H]3C(=O)NCC3=CC=C(C4=C(C)N=CS4)C=C3)NC(=O)CCC(C)C)C=C2)SC=N1	C50H66N8O8S4	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-83WDO6	SCHEMBL18063890	(2S)-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-4-oxopyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3CC(=O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C=C2)SC=N1	C29H30N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-YXD0ZD	SCHEMBL18063939	(2S,4S)-4-hydroxy-4-methyl-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@](C)(O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C=C2)SC=N1	C30H34N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-FMFU0G	SCHEMBL16267232	US10730870, Example 63; BDBM454898; US10730870, Example 63	COC1=CC=CC(C(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(C3=C(C)N=CS3)C=C2)=C1	C24H25N3O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-OGHWA4	SCHEMBL15126237	US10730870, Example 64; BDBM454899; US10730870, Example 64	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C3=CC=CC=C3)C=C2)SC=N1	C23H23N3O3S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-4NUR3H	SCHEMBL15126266	US10730870, Example 65; BDBM454900; US10730870, Example 65; PD128259; 1448188-03-1	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3CC4=C(C=CC=C4)C3=O)C(C)(C)C)C=C2)SC=N1	C30H34N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-2J3OTS	SCHEMBL18064007	(4R)-4-hydroxy-1-(3-methoxybenzoyl)-2-methyl-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	COC1=CC=CC(C(=O)N2C[C@H](O)CC2(C)C(=O)NCC2=CC=C(C3=C(C)N=CS3)C=C2)=C1	C25H27N3O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-QV4IKD	SCHEMBL18063970	(4R)-2-ethyl-4-hydroxy-1-(3-methoxybenzoyl)-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CCC1(C(=O)NCC2=CC=C(C3=C(C)N=CS3)C=C2)C[C@@H](O)CN1C(=O)C1=CC(OC)=CC=C1	C26H29N3O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-HEMUZ4	SCHEMBL18063763	US10730870, Example 68; BDBM454901; US10730870, Example 68	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4Cl)C3=O)C=C2)SC=N1	C29H31ClN4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-0UJ67G	SCHEMBL18063797	US10730870, Example 7; US10730870, Example 7; BDBM454844	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C3=O)C(Cl)=CC=C4)C=C2)SC=N1	C29H31ClN4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-HX13V9	SCHEMBL18063842	US11512083, Example 70; BDBM581891; US11512083, Example 70	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3=C(C#N)C=CC=C3)C(C)(C)C)C=C2)SC=N1	C30H33N5O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-PKTS4M	SCHEMBL18063727	US10730870, Example 71; BDBM454904; US10730870, Example 71	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3=CC(C#N)=CC=C3)C(C)(C)C)C=C2)SC=N1	C30H33N5O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-KRICFB	SCHEMBL18063906	US10730870, Example 72; BDBM454905; US10730870, Example 72	COC1=CC2=C(C=C1)C(=O)N([C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C3=C(C)N=CS3)C=C1)C(C)C)C2	C30H34N4O5S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-8PNZUH	SCHEMBL18063905	US10730870, Example 73; BDBM454906; US10730870, Example 73	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC(Cl)=C4)C3=O)C=C2)SC=N1	C29H31ClN4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-GR1ZAD	SCHEMBL18063932	US10730870, Example 74; BDBM454907; US10730870, Example 74	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=C(Cl)C=C4)C3=O)C=C2)SC=N1	C29H31ClN4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-DDUWNZ	SCHEMBL18063796	US11512083, Example 75; BDBM581896; US11512083, Example 75	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3CCN(C)CC3)C(C)(C)C)C=C2)SC=N1	C29H41N5O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-EJMQB7	SCHEMBL18063782	US10730870, Example 76; BDBM454909; US10730870, Example 76	COC1=CC=C(CCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)C=C1	C32H40N4O5S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-DO53D2	SCHEMBL18063708	US10730870, Example 77; BDBM454910; US10730870, Example 77	COC1=CC=CC(CCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)=C1	C32H40N4O5S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-UJ2AB4	SCHEMBL18063683	US10730870, Example 78; BDBM454911; US10730870, Example 78	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3=NC=CC=C3)C(C)(C)C)C=C2)SC=N1	C28H33N5O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-G9WKBK	SCHEMBL18063702	US10730870, Example 79; BDBM454912; US10730870, Example 79	CC(C)[C@@H](C(=O)N1C[C@](C)(O)C[C@H]1C(=O)O)N1CC2=C(C=CC=C2)C1=O	C19H24N2O5	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-59MBYI	SCHEMBL18063847	US10730870, Example 8; US10730870, Example 8; BDBM454845	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C3=O)C(F)=CC=C4)C=C2)SC=N1	C29H31FN4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-J1NF6G	SCHEMBL18063992	US10730870, Example 80; BDBM454913; US10730870, Example 80	CC1=CN=CC=C1C1=CC=C(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](C(C)C)N2CC3=C(C=CC=C3)C2=O)C=C1	C31H34N4O4	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-7SAOSL	SCHEMBL18063746	US10730870, Example 81; BDBM454914; US10730870, Example 81	COC1=CC=C(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](C(C)C)N2CC3=C(C=CC=C3)C2=O)C=C1	C26H31N3O5	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-S2X3JZ	SCHEMBL18063957	US10730870, Example 82; BDBM454915; US10730870, Example 82	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C(F)=C2)SC=N1	C29H31FN4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-HAKD3K	SCHEMBL18064003	US10730870, Example 83; BDBM454916; US10730870, Example 83	COC1=C(CCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)C=CC=C1	C32H40N4O5S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-DSP6PR	SCHEMBL18063800	US10730870, Example 84; BDBM454917; US10730870, Example 84	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3=CN=CC=C3)C(C)(C)C)C=C2)SC=N1	C28H33N5O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-BN026Z	CHEMBL4227864	(2~{s},4~{r})-1-[(2~{s})-2-Acetamidopropanoyl]-~{n}-[[4-(4-Methyl-1,3-Thiazol-5-Yl)phenyl]methyl]-4-Oxidanyl-Pyrrolidine-2-Carboxamide; (2~{s},4~{r})-1-[(2~{s})-2-Acetamidopropanoyl]-~{n}-[[4-(4-Methyl-1,3-Thiazol-5-Yl)phenyl]methyl]-4-Oxidanyl-Pyrrolidine-2-Carboxamide; SCHEMBL15126262; BDBM50459942; EN300-44822863; (2S,4R)-1-[(2S)-2-acetamidopropanoyl]-4-hydroxy-N-{[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl}pyrrolidine-2-carboxamide; 9B5	CC(=O)N[C@@H](C)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=C(C)N=CS2)C=C1	C21H26N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-VIJO87	SCHEMBL18063987	US10730870, Example 86; BDBM454919; US10730870, Example 86	CC(=O)NCC(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=C(C)N=CS2)C=C1	C20H24N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-C86JGL	SCHEMBL15111598	US10730870, Example 87; KBZQCHCLOJYNTO-VHSSKADRSA-N; BDBM454920; US10730870, Example 87; (S)-1-((2S,4R)-4-hydroxy-2-((4-(4-methylthiazol-5-yl)benzyl)carbamoyl)pyrrolidin-1-yl)-1-oxopropan-2-yl acetate	CC(=O)O[C@@H](C)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=C(C)N=CS2)C=C1	C21H25N3O5S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-SZ495Z	SCHEMBL18063680	US10730870, Example 88; BDBM454921; US10730870, Example 88	COC1=CC(C)=C(C(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(C3=C(C)N=CS3)C=C2)C=C1	C25H27N3O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-14Y1Y2	SCHEMBL18063784	US10730870, Example 89; US10730870, Example 89; FNBHJRUQIBKBLR-CNYCQXTOSA-N; BDBM454922	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(N)C(F)(F)F)C=C2)SC=N1	C19H21F3N4O3S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-ENT54R	SCHEMBL18063723	US10730870, Example 9; US10730870, Example 9; BDBM454846	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=C(F)C=C4)C3=O)C=C2)SC=N1	C29H31FN4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-G2B6EJ	SCHEMBL18063991	US10730870, Example 90; US10730870, Example 90; QFIBPTJZUZOBKU-LNKXUWQBSA-N; BDBM454923	CC(=O)NC(C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=C(C)N=CS2)C=C1)C(F)(F)F	C21H23F3N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-WPUNP3	SCHEMBL18063974	US10730870, Example 91; BDBM454924; US10730870, Example 91	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(N2CCOCC2)C=C1)N1CC2=C(C=CC=C2)C1=O	C29H36N4O5	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-CV8UL0	SCHEMBL18063770	US10730870, Example 96; BDBM454929; US10730870, Example 96	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=CN=CN2C)C=C1)N1CC2=C(C=CC=C2)C1=O	C29H33N5O4	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-SFCTVC	SCHEMBL18063921	US10730870, Example 93; BDBM454926; US10730870, Example 93	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C=C2F)SC=N1	C29H31FN4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-OB8VFT	SCHEMBL18063964	US10730870, Example 94; BDBM454927; US10730870, Example 94	CC[C@H](C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=C(C)N=CS2)C=C1)N1CC2=C(C=C(F)C=C2)C1=O	C30H33FN4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-8U7RA4	SCHEMBL18063738	US10730870, Example 95; BDBM454928; US10730870, Example 95	COC1=CC(C(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(C3=C(C)N=CS3)C=C2)=C(C)C=C1	C25H27N3O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-G821J4	SCHEMBL18063788	US10730870, Example 97; BDBM454930; US10730870, Example 97	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=CN=CS2)C=C1)N1CC2=C(C=CC=C2)C1=O	C28H30N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-RDDRNL	SCHEMBL18063791	US10730870, Example 98; BDBM454931; US10730870, Example 98	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CCCC3=O)C=C2)SC=N1	C25H32N4O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-09XTU3	SCHEMBL18063866	US10730870, Example 99; BDBM454932; US10730870, Example 99	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=N4)C3=O)C=C2)SC=N1	C28H31N5O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-OWKURW	SCHEMBL15111968	(2S,4R)-N-(4-(1H-pyrrol-3-yl)benzyl)-4-hydroxy-1-(2-(3-methylisoxazol-5-yl)acetyl)pyrrolidine-2-carboxamide; BUJBYIOVYQJWHD-QUCCMNQESA-N; (2S,4R)-N-(4-(1H-pyrrol-3-yl)benzyl)-4-hydroxy-1-(2-(3-methylisoxazol-5-yl)acetyl)pyrrolidine-2-carboxamide	CC1=NOC(CC(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(C3=CNC=C3)C=C2)=C1	C22H24N4O4	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-39Z28Z	SCHEMBL15125935	(2S,4R)-N-[(4-chlorophenyl)methyl]-4-hydroxy-1-(2-imidazol-1-ylacetyl)pyrrolidine-2-carboxamide	O=C(NCC1=CC=C(Cl)C=C1)[C@@H]1C[C@@H](O)CN1C(=O)CN1C=CN=C1	C17H19ClN4O3	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-2YGVXB	SCHEMBL15126271	(2S,4R)-1-(3-ethoxybenzoyl)-4-hydroxy-N-[[4-(1,3-oxazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL31253506	CCOC1=CC=CC(C(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(C3=CN=CO3)C=C2)=C1	C24H25N3O5	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-6TIH3N	SCHEMBL15126029	(2S,4R)-1-(3-ethoxybenzoyl)-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL30856526	CCOC1=CC=CC(C(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(C3=C(C)N=CS3)C=C2)=C1	C25H27N3O4S	HIF1A	Q16665	VHL	WO-2016149668-A1
TPD-ZZ3LYN	Bos-6-2-2-2-2-2-2-crbn	CHEMBL4742867; SCHEMBL18788276; BOS-6-2-2-2-2-2-2-CRBN	COc1cc(Nc2c(C#N)cnc3cc(OCCCN4CCN(CCCCCCOCCOCCOCCOCCOCCOCC(=O)Nc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)c(OC)cc23)c(Cl)cc1Cl	C56H70Cl2N8O14	BCR-ABL	Q16189	CRBN	WO-2017079267-A1
TPD-UJE0JT	Bos-6-2-2-2-2-2-2-vhl	BOS-6-2-2-2-2-2-2-VHL; CHEMBL4796635; SCHEMBL18788299	COc1cc(Nc2c(C#N)cnc3cc(OCCCN4CCN(CCCCCCOCCOCCOCCOCCOCCOCC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)NCc5ccc(-c6scnc6C)cc5)C(C)(C)C)CC4)c(OC)cc23)c(Cl)cc1Cl	C65H89Cl2N9O13S	BCR-ABL	Q16189	VHL	WO-2017079267-A1
TPD-N60RYU	CHEMBL4742759	6-[2-[2-[6-[4-[3-[3-cyano-4-(2,4-dichloro-5-methoxyanilino)-6-methoxyquinolin-7-yl]oxypropyl]piperazin-1-yl]hexoxy]ethoxy]ethoxy]-N-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]hexanamide; SCHEMBL18788262	COc1cc(Nc2c(C#N)cnc3cc(OCCCN4CCN(CCCCCCOCCOCCOCCCCCC(=O)Nc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)c(OC)cc23)c(Cl)cc1Cl	C54H66Cl2N8O11	BCR-ABL	Q16189	CRBN	WO-2017079267-A1
TPD-E58V7Q	Bos-6-2-2-6-vhl	BOS-6-2-2-6-VHL; SCHEMBL18788288	COc1cc(Nc2c(C#N)cnc3cc(OCCCN4CCN(CCCCCCOCCOCCOCCCCCC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)NCc5ccc(-c6scnc6C)cc5)C(C)(C)C)CC4)c(OC)cc23)c(Cl)cc1Cl	C63H85Cl2N9O10S	BCR-ABL	Q16189	VHL	WO-2017079267-A1
TPD-SSN8ZR	Bos-6-2-2-crbn	BOS-6-2-2-CRBN; CHEMBL4748640; SCHEMBL18788284	COc1cc(Nc2c(C#N)cnc3cc(OCCCN4CCN(CCCCCCOCCOCC(=O)Nc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)c(OC)cc23)c(Cl)cc1Cl	C48H54Cl2N8O10	BCR-ABL	Q16189	CRBN	WO-2017079267-A1
TPD-TO5Z99	Bos-6-2-2-vhl	BOS-6-2-2-VHL; CHEMBL4797656; SCHEMBL18788305	COc1cc(Nc2c(C#N)cnc3cc(OCCCN4CCN(CCCCCCOCCOCC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)NCc5ccc(-c6scnc6C)cc5)C(C)(C)C)CC4)c(OC)cc23)c(Cl)cc1Cl	C57H73Cl2N9O9S	BCR-ABL	Q16189	VHL	WO-2017079267-A1
TPD-RIE5ON	WO2017079267A1_BOS-6-5-6-CRBN	.	CCN(CCCOc1cc2ncc(C#N)c(Nc3cc(OC)c(Cl)cc3Cl)c2cc1OC)CCN(C)CCCCCCOCCCCCOCCCCCC(=O)Nc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O	C56H72Cl2N8O10	BCR-ABL	Q16189	CRBN	WO-2017079267-A1
TPD-FUF1KP	WO2017079267A1_BOS-6-5-6-VHL	.	COc1cc(Nc2c(C#N)cnc3cc(OCCCN4CCN(CCCCCCOCCCCCOCCCCCC(=O)N[C@H](C(=O)N5C[C@H](O)CC5C(=O)NCc5ccc(-c6scnc6C)cc5)C(C)(C)C)CC4)c(OC)cc23)c(Cl)cc1Cl	C64H87Cl2N9O9S	BCR-ABL	Q16189	VHL	WO-2017079267-A1
TPD-0PQ9E8	WO2017079267A1_DAS-6-2-2-2-2-2-2-CRBN	.	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCCCCOCCOCCOCCOCCOCCOCC(=O)N=Nc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)n1	C51H64ClN11O12S	BCR-ABL	Q16189	CRBN	WO-2017079267-A1
TPD-X7NNNM	Das-6-2-2-2-2-2-2-vhl	DAS-6-2-2-2-2-2-2-VHL; CHEMBL4746371; SCHEMBL18788341	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCCCCOCCOCCOCCOCCOCCOCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCc3ccc(-c4scnc4C)cc3)C(C)(C)C)CC2)n1	C60H84ClN11O11S2	BCR-ABL	Q16189	VHL	WO-2017079267-A1
TPD-9DQTV5	WO2017079267A1_DAS-6-2-2-6-CRBN	.	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCCCCOCCOCCOCCCCCC(=O)Nc3cccc(C(=O)NC4CCC(=O)NC4=O)c3C=O)CC2)n1	C49H63ClN10O9S	BCR-ABL	Q16189	CRBN	WO-2017079267-A1
TPD-Z9XYB1	WO2017079267A1_DAS-6-2-2-6-VHL	.	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCCCCOCCOCCOCCCCCC(=O)N[C@H](C(=O)N3C[C@H](O)CC3C(=O)NCc3ccc(-c4scnc4C)cc3)C(C)(C)C)CC2)n1	C58H80ClN11O8S2	BCR-ABL	Q16189	VHL	WO-2017079267-A1
TPD-XMBX66	Das-6-2-2-crbn	DAS-6-2-2-CRBN; SCHEMBL18788313	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCCCCOCCOCC(=O)Nc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)n1	C43H49ClN10O8S	BCR-ABL	Q16189	CRBN	WO-2017079267-A1
TPD-1NSWHL	Das-6-2-2-vhl	DAS-6-2-2-VHL; CHEMBL4761731; SCHEMBL18788339	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCCCCOCCOCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCc3ccc(-c4scnc4C)cc3)C(C)(C)C)CC2)n1	C52H68ClN11O7S2	BCR-ABL	Q16189	VHL	WO-2017079267-A1
TPD-2NBCDN	Das-6-5-6-crbn	DAS-6-5-6-CRBN; SCHEMBL18788298	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCCCCOCCCCCOCCCCCC(=O)Nc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)n1	C50H63ClN10O8S	BCR-ABL	Q16189	CRBN	WO-2017079267-A1
TPD-X0Z7PG	Das-6-5-6-vhl	DAS-6-5-6-VHL; SCHEMBL18788268	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCCCCOCCCCCOCCCCCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCc3ccc(-c4scnc4C)cc3)C(C)(C)C)CC2)n1	C59H82ClN11O7S2	BCR-ABL	Q16189	VHL	WO-2017079267-A1
TPD-6ZSNQW	Ima-6-2-2-2-2-2-2-crbn	SCHEMBL18788304; IMA-6-2-2-2-2-2-2-CRBN	Cc1ccc(NC(=O)c2ccc(CN3CCN(CCCCCCOCCOCCOCCOCCOCCOCC(=O)Nc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)cc2)cc1Nc1nccc(-c2cccnc2)n1	C59H72N10O12	BCR-ABL	Q16189	CRBN	WO-2017079267-A1
TPD-SGM4I7	WO2017079267A1_IMA-6-2-2-2-2-2-2-VHL	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCOCCOCCOCCCCCCN2CCN(Cc3ccc(C(=O)Nc4cccc(Nc5nccc(-c6cccnc6)n5)c4)cc3)CC2)C(C)(C)C)cc1	C67H89N11O11S	BCR-ABL	Q16189	VHL	WO-2017079267-A1
TPD-U7BS7C	WO2017079267A1_IMA-6-2-2-6-CRBN	.	Cc1ccc(NC(=O)c2ccc(CN3CCN(CCCCCCOCCOCCOCCCCCC(=O)Nc4cccc5c4C(=O)N(C(CCC=O)C(N)=O)C5=O)CC3)cc2)cc1Nc1nccc(-c2cccnc2)n1	C57H70N10O9	BCR-ABL	Q16189	CRBN	WO-2017079267-A1
TPD-MG3D9E	Ima-6-2-2-6-vhl	IMA-6-2-2-6-VHL; SCHEMBL18788312	Cc1ccc(NC(=O)c2ccc(CN3CCN(CCCCCCOCCOCCOCCCCCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)NCc4ccc(-c5scnc5C)cc4)C(C)(C)C)CC3)cc2)cc1Nc1nccc(-c2cccnc2)n1	C66H87N11O8S	BCR-ABL	Q16189	VHL	WO-2017079267-A1
TPD-S76OIL	Ima-6-2-2-crbn	IMA-6-2-2-CRBN; SCHEMBL18788267	Cc1ccc(NC(=O)c2ccc(CN3CCN(CCCCCCOCCOCC(=O)Nc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)cc2)cc1Nc1nccc(-c2cccnc2)n1	C51H56N10O8	BCR-ABL	Q16189	CRBN	WO-2017079267-A1
TPD-3NHIRQ	Ima-6-2-2-vhl	IMA-6-2-2-VHL; SCHEMBL18788291	Cc1ccc(NC(=O)c2ccc(CN3CCN(CCCCCCOCCOCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)NCc4ccc(-c5scnc5C)cc4)C(C)(C)C)CC3)cc2)cc1Nc1nccc(-c2cccnc2)n1	C60H75N11O7S	BCR-ABL	Q16189	VHL	WO-2017079267-A1
TPD-CL9RCF	Ima-6-5-6-crbn	IMA-6-5-6-CRBN; SCHEMBL18788321	Cc1ccc(NC(=O)c2ccc(CN3CCN(CCCCCCOCCCCCOCCCCCC(=O)Nc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)cc2)cc1Nc1nccc(-c2cccnc2)n1	C58H70N10O8	BCR-ABL	Q16189	CRBN	WO-2017079267-A1
TPD-M8IJ69	WO2017079267A1_IMA-6-5-6-VHL	.	Cc1ccc(NC(=O)c2ccc(CN3CCN(CCCCCCOCCCCCOCCCCCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)N(N)Cc4ccc(-c5scnc5C)cc4)C(C)(C)C)CC3)cc2)cc1Nc1nccc(-c2cccnc2)n1	C67H90N12O7S	BCR-ABL	Q16189	VHL	WO-2017079267-A1
TPD-QNQSMN	SCHEMBL20655231	2-[4-[3-[3-cyano-4-(2,4-dichloro-5-methoxyanilino)-6-methoxyquinolin-7-yl]oxypropyl]piperazin-1-yl]-N-[2-[2-[2-[2-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyacetyl]amino]ethoxy]ethoxy]ethoxy]ethyl]acetamide	COC1=CC(NC2=C3C=C(OC)C(OCCCN4CCN(CC(=O)NCCOCCOCCOCCNC(=O)COC5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)CC4)=CC3=NC=C2C#N)=C(Cl)C=C1Cl	C50H57Cl2N9O13	HER3	P21860	CRBN	WO-2017117474-A1
TPD-9QQ3JF	SCHEMBL20655217	2-[4-[4-(3-chloro-2-fluoroanilino)-7-methoxyquinazolin-6-yl]oxypiperidin-1-yl]-N-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethyl]acetamide	COC1=CC2=NC=NC(NC3=C(F)C(Cl)=CC=C3)=C2C=C1OC1CCN(CC(=O)NCCOCCOCCNC2=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=CC=C2)CC1	C41H44ClFN8O9	HER3	P21860	CRBN	WO-2017117474-A1
TPD-5IHA99	SCHEMBL20655218	2-[4-[4-(3-chloro-2-fluoroanilino)-7-methoxyquinazolin-6-yl]oxypiperidin-1-yl]-N-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethyl]acetamide	COC1=CC2=NC=NC(NC3=C(F)C(Cl)=CC=C3)=C2C=C1OC1CCN(CC(=O)NCCOCCOCCOCCNC2=CC=CC3=C2C(=O)N(C2CCC(=O)NC2=O)C3=O)CC1	C43H48ClFN8O10	HER3	P21860	CRBN	WO-2017117474-A1
TPD-NLCEQ9	SCHEMBL20655492	N-[4-[4-[3-[3-cyano-4-(2,4-dichloro-5-methoxyanilino)-6-methoxyquinolin-7-yl]oxypropyl]piperazin-1-yl]-4-oxobutyl]-2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyacetamide	COC1=CC(NC2=C3C=C(OC)C(OCCCN4CCN(C(=O)CCCNC(=O)COC5=CC=CC6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)=CC3=NC=C2C#N)=C(Cl)C=C1Cl	C44H44Cl2N8O10	HER3	P21860	CRBN	WO-2017117474-A1
TPD-L64VXA	SCHEMBL20655326	N-[4-[3-chloro-4-(pyridin-2-ylmethoxy)anilino]-3-cyano-7-ethoxyquinolin-6-yl]-3-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]propanamide	CCOC1=CC2=NC=C(C#N)C(NC3=CC=C(OCC4=CC=CC=N4)C(Cl)=C3)=C2C=C1NC(=O)CCOCCOCCNC1=CC=CC2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O	C44H41ClN8O9	HER3	P21860	CRBN	WO-2017117474-A1
TPD-X5ZBM3	SCHEMBL20655493	N-[4-[3-chloro-4-(pyridin-2-ylmethoxy)anilino]-3-cyano-7-ethoxyquinolin-6-yl]-3-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]propanamide	CCOC1=CC2=NC=C(C#N)C(NC3=CC=C(OCC4=CC=CC=N4)C(Cl)=C3)=C2C=C1NC(=O)CCOCCOCCOCCNC1=C2C(=O)N(C3CCC(=O)NC3=O)C(=O)C2=CC=C1	C46H45ClN8O10	HER3	P21860	CRBN	WO-2017117474-A1
TPD-SQUEGP	SCHEMBL20655344	N-[4-[3-chloro-4-(pyridin-2-ylmethoxy)anilino]-3-cyano-7-ethoxyquinolin-6-yl]-3-[2-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]propanamide	CCOC1=CC2=NC=C(C#N)C(NC3=CC=C(OCC4=CC=CC=N4)C(Cl)=C3)=C2C=C1NC(=O)CCOCCOCCOCCOCCOCCNC1=C2C(=O)N(C3CCC(=O)NC3=O)C(=O)C2=CC=C1	C50H53ClN8O12	HER3	P21860	CRBN	WO-2017117474-A1
TPD-QFVZJ0	CHEMBL5198264	4-(2,4-Dichloro-5-methoxyanilino)-7-[3-[4-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethyl]piperazin-1-yl]propoxy]-6-methoxyquinoline-3-carbonitrile; SCHEMBL20655333; PD141210	COC1=CC2=C(NC3=CC(OC)=C(Cl)C=C3Cl)C(C#N)=CN=C2C=C1OCCCN1CCN(CCOCCOCCNC2=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=CC=C2)CC1	C44H48Cl2N8O9	HER3	P21860	CRBN	WO-2017117474-A1
TPD-P3FBP5	SCHEMBL20655334	4-(2,4-Dichloro-5-methoxyanilino)-7-[3-[4-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethyl]piperazin-1-yl]propoxy]-6-methoxyquinoline-3-carbonitrile	COC1=CC2=C(NC3=CC(OC)=C(Cl)C=C3Cl)C(C#N)=CN=C2C=C1OCCCN1CCN(CCOCCOCCOCCNC2=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=CC=C2)CC1	C46H52Cl2N8O10	HER3	P21860	CRBN	WO-2017117474-A1
TPD-ETQ1SW	SCHEMBL20655332	4-(2,4-Dichloro-5-methoxyanilino)-7-[3-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]propoxy]-6-methoxyquinoline-3-carbonitrile	COC1=CC2=C(NC3=CC(OC)=C(Cl)C=C3Cl)C(C#N)=CN=C2C=C1OCCCOCCOCCOCCNC1=CC=CC2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O	C40H40Cl2N6O10	HER3	P21860	CRBN	WO-2017117474-A1
TPD-91J599	SCHEMBL20655216	4-(2,4-Dichloro-5-methoxyanilino)-7-[3-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethoxy]propoxy]-6-methoxyquinoline-3-carbonitrile	COC1=CC2=C(NC3=CC(OC)=C(Cl)C=C3Cl)C(C#N)=CN=C2C=C1OCCCOCCOCCOCCOCCNC1=C2C(=O)N(C3CCC(=O)NC3=O)C(=O)C2=CC=C1	C42H44Cl2N6O11	HER3	P21860	CRBN	WO-2017117474-A1
TPD-V60JN3	WO2017185036A1_I-10	.	O=C1CCC(N2C(=O)C3=C(C2=O)C(NCOCCOCCOCCN2CCN(C4=CC=C(C5=CC6=C(C=C5)CN(C(C(=O)NC5=NC=CS5)C5=C(O)C=CC(F)=C5)C6=O)C=C4)CC2)=CC=C3)C(=O)N1	C49H49FN8O10S	EGFR	P00533	CRBN	WO-2017185036-A1
TPD-GTQARS	SCHEMBL19475576	2-[5-[4-[4-[6-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]hexyl]piperazin-1-yl]phenyl]-3-oxo-1H-isoindol-2-yl]-2-(5-fluoro-2-hydroxyphenyl)-N-(1,3-thiazol-2-yl)acetamide	O=C1CCC(N2C(=O)C3=C(C2=O)C(NCCCCCCN2CCN(C4=CC=C(C5=CC6=C(C=C5)CN(C(C(=O)NC5=NC=CS5)C5=CC(F)=CC=C5O)C6=O)C=C4)CC2)=CC=C3)C(=O)N1	C48H47FN8O7S	EGFR	P00533	CRBN	WO-2017185036-A1
TPD-LH8TIQ	SCHEMBL19475612	2-[5-[4-[4-[8-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]octyl]piperazin-1-yl]phenyl]-3-oxo-1H-isoindol-2-yl]-2-(5-fluoro-2-hydroxyphenyl)-N-(1,3-thiazol-2-yl)acetamide	O=C1CCC(N2C(=O)C3=C(C2=O)C(NCCCCCCCCN2CCN(C4=CC=C(C5=CC6=C(C=C5)CN(C(C(=O)NC5=NC=CS5)C5=CC(F)=CC=C5O)C6=O)C=C4)CC2)=CC=C3)C(=O)N1	C50H51FN8O7S	EGFR	P00533	CRBN	WO-2017185036-A1
TPD-IJ7NBT	WO2017185036A1_I-13	.	O=C1CCC(N2C(=O)C3=C(C2=O)C(NCOCCOCCOCCOCCN2CCN(C4=CC=C(C5=CC6=C(C=C5)CN(C(C(=O)NC5=NC=CS5)C5=C(O)C=CC(F)=C5)C6=O)C=C4)CC2)=CC=C3)C(=O)N1	C51H53FN8O11S	EGFR	P00533	CRBN	WO-2017185036-A1
TPD-TVUQJO	SCHEMBL19475613	2-[5-[4-[4-[2-[2-[2-[3-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]azetidin-1-yl]ethoxy]ethoxy]ethyl]piperazin-1-yl]phenyl]-3-oxo-1H-isoindol-2-yl]-2-phenyl-N-(1,3-thiazol-2-yl)acetamide	O=C1CCC(N2C(=O)C3=CC=CC(NC4CN(CCOCCOCCN5CCN(C6=CC=C(C7=CC8=C(C=C7)CN(C(C(=O)NC7=NC=CS7)C7=CC=CC=C7)C8=O)C=C6)CC5)C4)=C3C2=O)C(=O)N1	C51H53N9O8S	EGFR	P00533	CRBN	WO-2017185036-A1
TPD-V7MCX7	SCHEMBL19475657	2-[5-[4-[4-[2-[2-[2-[2-[3-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]azetidin-1-yl]ethoxy]ethoxy]ethoxy]ethyl]piperazin-1-yl]phenyl]-3-oxo-1H-isoindol-2-yl]-2-phenyl-N-(1,3-thiazol-2-yl)acetamide	O=C1CCC(N2C(=O)C3=CC=CC(NC4CN(CCOCCOCCOCCN5CCN(C6=CC=C(C7=CC8=C(C=C7)CN(C(C(=O)NC7=NC=CS7)C7=CC=CC=C7)C8=O)C=C6)CC5)C4)=C3C2=O)C(=O)N1	C53H57N9O9S	EGFR	P00533	CRBN	WO-2017185036-A1
TPD-X34BCR	CHEMBL4449910	2-[5-[4-[4-[2-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethyl]piperazin-1-yl]phenyl]-3-oxo-1H-isoindol-2-yl]-2-phenyl-N-(1,3-thiazol-2-yl)acetamide; SCHEMBL19475628; PD140854	O=C1CCC(N2C(=O)C3=CC=CC(NCCOCCOCCOCCOCCN4CCN(C5=CC=C(C6=CC7=C(C=C6)CN(C(C(=O)NC6=NC=CS6)C6=CC=CC=C6)C7=O)C=C5)CC4)=C3C2=O)C(=O)N1	C52H56N8O10S	EGFR	P00533	CRBN	WO-2017185036-A1
TPD-QTTJTN	SCHEMBL19475759	(2S,4R)-1-[(2S)-3,3-dimethyl-2-[3-[2-[2-[2-[4-[5-[3-oxo-2-[2-oxo-1-phenyl-2-(1,3-thiazol-2-ylamino)ethyl]-1H-isoindol-5-yl]pyridin-2-yl]piperazin-1-yl]ethoxy]ethoxy]ethoxy]propanoylamino]butanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL31028398	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCOCCOCCOCCN3CCN(C4=NC=C(C5=CC6=C(C=C5)CN(C(C(=O)NC5=NC=CS5)C5=CC=CC=C5)C6=O)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C60H72N10O9S2	EGFR	P00533	VHL	WO-2017185036-A1
TPD-HUUTSU	SCHEMBL19475630	(2S,4R)-1-[(2S)-3,3-dimethyl-2-[3-[2-[2-[4-[5-[3-oxo-2-[2-oxo-1-phenyl-2-(1,3-thiazol-2-ylamino)ethyl]-1H-isoindol-5-yl]pyridin-2-yl]piperazin-1-yl]ethoxy]ethoxy]propanoylamino]butanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCOCCOCCN3CCN(C4=NC=C(C5=CC6=C(C=C5)CN(C(C(=O)NC5=NC=CS5)C5=CC=CC=C5)C6=O)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C58H68N10O8S2	EGFR	P00533	VHL	WO-2017185036-A1
TPD-7TO1HV	SCHEMBL23393944	(2S,4R)-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-1-[(2S)-2-[3-[2-[2-[3-oxo-3-[4-[4-[3-oxo-2-[2-oxo-1-phenyl-2-(1,3-thiazol-2-ylamino)ethyl]-1H-isoindol-5-yl]phenyl]piperazin-1-yl]propoxy]ethoxy]ethoxy]propanoylamino]propanoyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C)NC(=O)CCOCCOCCOCCC(=O)N3CCN(C4=CC=C(C5=CC6=C(C=C5)CN(C(C(=O)NC5=NC=CS5)C5=CC=CC=C5)C6=O)C=C4)CC3)C=C2)SC=N1	C58H65N9O10S2	EGFR	P00533	VHL	WO-2017185036-A1
TPD-OKZHOL	SCHEMBL19475779	(2S,4R)-1-[(2S)-2-[3-[2-[2-[3-[4-[4-[2-[1-(5-fluoro-2-hydroxyphenyl)-2-oxo-2-(1,3-thiazol-2-ylamino)ethyl]-3-oxo-1H-isoindol-5-yl]phenyl]piperazin-1-yl]-3-oxopropoxy]ethoxy]ethoxy]propanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCOCCOCCOCCC(=O)N3CCN(C4=CC=C(C5=CC6=C(C=C5)CN(C(C(=O)NC5=NC=CS5)C5=CC(F)=CC=C5O)C6=O)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C61H70FN9O11S2	EGFR	P00533	VHL	WO-2017185036-A1
TPD-FGBVEA	SCHEMBL19475658	2-[5-[4-[4-[3-[2-[2-[2-[[2-(3-methyl-2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]propanoyl]piperazin-1-yl]phenyl]-3-oxo-1H-isoindol-2-yl]-2-phenyl-N-(1,3-thiazol-2-yl)acetamide	CC1(N2C(=O)C3=CC=CC(NCCOCCOCCOCCC(=O)N4CCN(C5=CC=C(C6=CC7=C(C=C6)CN(C(C(=O)NC6=NC=CS6)C6=CC=CC=C6)C7=O)C=C5)CC4)=C3C2=O)CCC(=O)NC1=O	C52H54N8O10S	EGFR	P00533	CRBN	WO-2017185036-A1
TPD-5OC8E1	SCHEMBL19475707	2-[5-[4-[4-[3-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]propanoyl]piperazin-1-yl]phenyl]-3-oxo-1H-isoindol-2-yl]-2-(5-fluoro-2-hydroxyphenyl)-N-(1,3-thiazol-2-yl)acetamide	O=C1CCC(N2C(=O)C3=C(C2=O)C(NCCOCCOCCC(=O)N2CCN(C4=CC=C(C5=CC6=C(C=C5)CN(C(C(=O)NC5=NC=CS5)C5=C(O)C=CC(F)=C5)C6=O)C=C4)CC2)=CC=C3)C(=O)N1	C49H47FN8O10S	EGFR	P00533	CRBN	WO-2017185036-A1
TPD-MA2EN6	SCHEMBL19475650	2-[5-[4-[4-[3-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]propanoyl]piperazin-1-yl]phenyl]-3-oxo-1H-isoindol-2-yl]-2-(5-fluoro-2-hydroxyphenyl)-N-(1,3-thiazol-2-yl)acetamide	O=C1CCC(N2C(=O)C3=C(C2=O)C(NCCOCCC(=O)N2CCN(C4=CC=C(C5=CC6=C(C=C5)CN(C(C(=O)NC5=NC=CS5)C5=C(O)C=CC(F)=C5)C6=O)C=C4)CC2)=CC=C3)C(=O)N1	C47H43FN8O9S	EGFR	P00533	CRBN	WO-2017185036-A1
TPD-4QVRFK	WO2017185036A1_I-3	.	O=C1CCC(N2C(=O)C3=CC=CC(NCCOCCOCCOCCC(=O)N4CCN(C5=CC=C(C6=CC7=C(C=C6)CN(C(C(=O)NC6=NC=CC6)C6=CC(F)=CC=C6O)C7=O)C=C5)CC4)=C3C2=O)C(=O)N1	C52H53FN8O11	EGFR	P00533	CRBN	WO-2017185036-A1
TPD-RFZC2V	SCHEMBL19475778	2-[5-[4-[4-[3-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethoxy]propanoyl]piperazin-1-yl]phenyl]-3-oxo-1H-isoindol-2-yl]-2-(5-fluoro-2-hydroxyphenyl)-N-(1,3-thiazol-2-yl)acetamide	O=C1CCC(N2C(=O)C3=CC=CC(NCCOCCOCCOCCOCCC(=O)N4CCN(C5=CC=C(C6=CC7=C(C=C6)CN(C(C(=O)NC6=NC=CS6)C6=C(O)C=CC(F)=C6)C7=O)C=C5)CC4)=C3C2=O)C(=O)N1	C53H55FN8O12S	EGFR	P00533	CRBN	WO-2017185036-A1
TPD-0Z8Q8Y	SCHEMBL19475770	2-[5-[4-[4-[2-[2-[2-[2-[[2-(3-methyl-2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethyl]piperazin-1-yl]phenyl]-3-oxo-1H-isoindol-2-yl]-2-phenyl-N-(1,3-thiazol-2-yl)acetamide	CC1(N2C(=O)C3=CC=CC(NCCOCCOCCOCCN4CCN(C5=CC=C(C6=CC7=C(C=C6)CN(C(C(=O)NC6=NC=CS6)C6=CC=CC=C6)C7=O)C=C5)CC4)=C3C2=O)CCC(=O)NC1=O	C51H54N8O9S	EGFR	P00533	CRBN	WO-2017185036-A1
TPD-5EIPYE	SCHEMBL19475655	2-[5-[6-[4-[2-[2-[2-[2-[[2-(3-methyl-2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethyl]piperazin-1-yl]pyridin-3-yl]-3-oxo-1H-isoindol-2-yl]-2-phenyl-N-(1,3-thiazol-2-yl)acetamide	CC1(N2C(=O)C3=C(C2=O)C(NCCOCCOCCOCCN2CCN(C4=CC=C(C5=CC6=C(C=C5)CN(C(C(=O)NC5=NC=CS5)C5=CC=CC=C5)C6=O)C=N4)CC2)=CC=C3)CCC(=O)NC1=O	C50H53N9O9S	EGFR	P00533	CRBN	WO-2017185036-A1
TPD-WPDVXI	SCHEMBL20887896	2-[5-[4-[4-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethyl]piperazin-1-yl]phenyl]-3-oxo-1H-isoindol-2-yl]-2-(5-fluoro-2-hydroxyphenyl)-N-(1,3-thiazol-2-yl)acetamide	O=C1CCC(N2C(=O)C3=C(C2=O)C(NCCOCCOCCN2CCN(C4=CC=C(C5=CC6=C(C=C5)CN(C(C(=O)NC5=NC=CS5)C5=CC(F)=CC=C5O)C6=O)C=C4)CC2)=CC=C3)C(=O)N1	C48H47FN8O9S	EGFR	P00533	CRBN	WO-2017185036-A1
TPD-TZCE0Z	SCHEMBL20887921	2-[5-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperazin-1-yl]phenyl]-3-oxo-1H-isoindol-2-yl]-2-phenyl-N-(1,3-thiazol-2-yl)acetamide	O=C1CCC(N2C(=O)C3=C(C2=O)C(N2CCN(C4=CC=C(C5=CC6=C(C=C5)CN(C(C(=O)NC5=NC=CS5)C5=CC=CC=C5)C6=O)C=C4)CC2)=CC=C3)C(=O)N1	C42H35N7O6S	EGFR	P00533	CRBN	WO-2017185036-A1
TPD-UIVNHA	SCHEMBL20887819	(2R,4S)-1-[(2R)-3,3-dimethyl-2-[[2-[4-[4-[3-oxo-2-[2-oxo-1-phenyl-2-(1,3-thiazol-2-ylamino)ethyl]-1H-isoindol-5-yl]phenyl]piperazin-1-yl]acetyl]amino]butanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@H]3C[C@H](O)CN3C(=O)[C@H](NC(=O)CN3CCN(C4=CC=C(C5=CC6=C(C=C5)CN(C(C(=O)NC5=NC=CS5)C5=CC=CC=C5)C6=O)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C53H57N9O6S2	EGFR	P00533	VHL	WO-2017185036-A1
TPD-JS5QK6	WO2017204445A2_1	5-[4-[4-[[5-chloro-4-(2-propan-2-ylsulfonylanilino)pyrimidin-2-yl]amino]-2-methyl-5-propan-2-yloxyphenyl]piperidin-1-yl]-N-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]butyl]-5-oxopentanamide	CC1=CC(NC2=NC=C(Cl)C(NC3=CC=CC=C3S(=O)(=O)C(C)C)=N2)=C(OC(C)C)C=C1C1CCN(C(=O)CCCC(=O)NCCCCNC2=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=CC=C2)CC1	C50H60ClN9O9S	ALK	Q9UM73	CRBN	WO-2017204445-A2
TPD-NC9TZJ	WO2017204445A2_2	.	CCN(CCCC1=C(C)C=C(NC2=NC(NC3=CC=CC=C3S(=O)(=O)C(C)C)=C(Cl)C=N2)C(OC(C)C)=C1)C(=O)CCCC(=O)NCCOCCOCC(=O)NC(C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=C(C)N=CS2)C=C1)C(C)(C)C	C61H83ClN10O11S2	ALK	Q9UM73	VHL	WO-2017204445-A2
TPD-4PD5I1	SCHEMBL19662348	(2S,4R)-1-[(2R)-2-[[5-[4-[4-[[5-chloro-4-(2-propan-2-ylsulfonylanilino)pyrimidin-2-yl]amino]-2-methyl-5-propan-2-yloxyphenyl]piperidin-1-yl]-5-oxopentanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2CCN(C(=O)CCCC(=O)N[C@@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCC3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)CC2)C=C(OC(C)C)C(NC2=NC(NC3=CC=CC=C3S(=O)(=O)C(C)C)=C(Cl)C=N2)=C1	C55H70ClN9O8S2	ALK	Q9UM73	VHL	WO-2017204445-A2
TPD-A0LG6H	SCHEMBL22155714	5-[4-[4-[[5-chloro-4-(2-propan-2-ylsulfonylanilino)pyrimidin-2-yl]amino]-2-methyl-5-propan-2-yloxyphenyl]piperidin-1-yl]-N-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]pentanamide	CC1=CC(NC2=NC=C(Cl)C(NC3=CC=CC=C3S(=O)(=O)C(C)C)=N2)=C(OC(C)C)C=C1C1CCN(CCCCC(=O)NC2=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=CC=C2)CC1	C46H53ClN8O8S	ALK	Q9UM73	CRBN	WO-2017204445-A2
TPD-6FMKJ1	WO2017204445A2_5	.	CC1=CC(NC2=NC=C(Cl)C(NC3=CC=CC=C3S(=O)(=O)C(C)C)=N2)=C(OC(C)C)C=C1C1CCN(C(=O)CCCC(=O)NC2=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=CC=C2)CC1	C46H51ClN8O9S	ALK	Q9UM73	CRBN	WO-2017204445-A2
TPD-5YG312	WO2017204445A2_6	2-[2-[4-[4-[[5-chloro-4-(2-propan-2-ylsulfonylanilino)pyrimidin-2-yl]amino]-2-methyl-5-propan-2-yloxyphenyl]piperidin-1-yl]-2-oxoethoxy]-N-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]acetamide	CC1=CC(NC2=NC=C(Cl)C(NC3=CC=CC=C3S(=O)(=O)C(C)C)=N2)=C(OC(C)C)C=C1C1CCN(C(=O)COCC(=O)NC2=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=CC=C2)CC1	C45H49ClN8O10S	ALK	Q9UM73	CRBN	WO-2017204445-A2
TPD-JIZDQ2	WO2017204445A2_7	.	CC1=CC(NC2=NC=C(Cl)C(NC3=CC=CC=C3S(=O)(=O)C(C)C)=N2)=C(OC(C)C)C=C1C1CCN(CCCCC(=O)N[C@@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)CC1	C55H72ClN9O7S2	ALK	Q9UM73	VHL	WO-2017204445-A2
TPD-H0BIAF	WO2017204445A2_8	.	CC1=CC(NC2=NC=C(Cl)C(NC3=CC=CC=C3S(=O)(=O)C(C)C)=N2)=C(OC(C)C)C=C1C1CCN(C(=O)CCCCCC(=O)NC2=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=CC=C2)CC1	C48H55ClN8O9S	ALK	Q9UM73	CRBN	WO-2017204445-A2
TPD-NB73B7	WO2017204445A2_9	(2S,4R)-1-[2-[[2-[2-[4-[4-[[5-chloro-4-(2-propan-2-ylsulfonylanilino)pyrimidin-2-yl]amino]-2-methyl-5-propan-2-yloxyphenyl]piperidin-1-yl]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2CCN(CCOCC(=O)NC(C(=O)N3C[C@H](O)C[C@H]3C(=O)NCC3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)CC2)C=C(OC(C)C)C(NC2=NC(NC3=CC=CC=C3S(=O)(=O)C(C)C)=C(Cl)C=N2)=C1	C54H70ClN9O8S2	ALK	Q9UM73	VHL	WO-2017204445-A2
TPD-52444Q	WO2017204445A2_10	(2S,4R)-1-[(2R)-2-[[2-[4-[4-[4-[[5-chloro-4-(2-propan-2-ylsulfonylanilino)pyrimidin-2-yl]amino]-2-methyl-5-propan-2-yloxyphenyl]piperidin-1-yl]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=CC(NC2=NC=C(Cl)C(NC3=CC=CC=C3S(=O)(=O)C(C)C)=N2)=C(OC(C)C)C=C1C1CCN(CCCCOCC(=O)N[C@@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)CC1	C56H74ClN9O8S2	ALK	Q9UM73	VHL	WO-2017204445-A2
TPD-XT4QZJ	WO2017204445A2_11	(2S,4R)-1-[(2R)-2-[[7-[4-[4-[[5-chloro-4-(2-propan-2-ylsulfonylanilino)pyrimidin-2-yl]amino]-2-methyl-5-propan-2-yloxyphenyl]piperidin-1-yl]-7-oxoheptanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=CC(NC2=NC=C(Cl)C(NC3=CC=CC=C3S(=O)(=O)C(C)C)=N2)=C(OC(C)C)C=C1C1CCN(C(=O)CCCCCC(=O)N[C@@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)CC1	C57H74ClN9O8S2	ALK	Q9UM73	VHL	WO-2017204445-A2
TPD-SH7MM3	WO2017204445A2_12	2-[2-[2-[2-[4-[4-[[5-chloro-4-(2-propan-2-ylsulfonylanilino)pyrimidin-2-yl]amino]-2-methyl-5-propan-2-yloxyphenyl]piperidin-1-yl]ethoxy]ethoxy]ethoxy]-N-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]acetamide	CC1=C(C2CCN(CCOCCOCCOCC(=O)NC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)CC2)C=C(OC(C)C)C(NC2=NC(NC3=CC=CC=C3S(=O)(=O)C(C)C)=C(Cl)C=N2)=C1	C49H59ClN8O11S	ALK	Q9UM73	VHL	WO-2017204445-A2
TPD-E2B5WP	WO2017204445A2_13	2-[4-[4-[4-[[5-chloro-4-(2-propan-2-ylsulfonylanilino)pyrimidin-2-yl]amino]-2-methyl-5-propan-2-yloxyphenyl]piperidin-1-yl]butoxy]-N-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]acetamide	CC1=CC(NC2=NC=C(Cl)C(NC3=CC=CC=C3S(=O)(=O)C(C)C)=N2)=C(OC(C)C)C=C1C1CCN(CCCCOCC(=O)NC2=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=CC=C2)CC1	C47H55ClN8O9S	ALK	Q9UM73	CRBN	WO-2017204445-A2
TPD-FCFX7J	WO2017204445A2_14	2-[2-[2-[4-[4-[[5-chloro-4-(2-propan-2-ylsulfonylanilino)pyrimidin-2-yl]amino]-2-methyl-5-propan-2-yloxyphenyl]piperidin-1-yl]ethoxy]ethoxy]-N-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]acetamide	CC1=CC(NC2=NC(NC3=C(S(=O)(=O)C(C)C)C=CC=C3)=C(Cl)C=N2)=C(OC(C)C)C=C1C1CCN(CCOCCOCC(=O)NC2=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=CC=C2)CC1	C47H55ClN8O10S	ALK	Q9UM73	CRBN	WO-2017204445-A2
TPD-1IAILF	WO2017204445A2_15	2-[2-[4-[4-[[5-chloro-4-(2-propan-2-ylsulfonylanilino)pyrimidin-2-yl]amino]-2-methyl-5-propan-2-yloxyphenyl]piperidin-1-yl]ethoxy]-N-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]acetamide	CC1=CC(NC2=NC(NC3=C(S(=O)(=O)C(C)C)C=CC=C3)=C(Cl)C=N2)=C(OC(C)C)C=C1C1CCN(CCOCC(=O)NC2=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=CC=C2)CC1	C45H51ClN8O9S	ALK	Q9UM73	CRBN	WO-2017204445-A2
TPD-NODJ2H	WO2017204445A2_16	(2S,4R)-1-[2-[[2-[2-[2-[2-[4-[4-[[5-chloro-4-(2-propan-2-ylsulfonylanilino)pyrimidin-2-yl]amino]-2-methyl-5-propan-2-yloxyphenyl]piperidin-1-yl]ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2CCN(CCOCCOCCOCC(=O)NC(C(=O)N3C[C@H](O)C[C@H]3C(=O)NCC3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)CC2)C=C(OC(C)C)C(NC2=NC(NC3=CC=CC=C3S(=O)(=O)C(C)C)=C(Cl)C=N2)=C1	C58H78ClN9O10S2	ALK	Q9UM73	VHL	WO-2017204445-A2
TPD-XNRP3H	SCHEMBL22155197	6-[4-[4-[[5-chloro-4-(2-propan-2-ylsulfonylanilino)pyrimidin-2-yl]amino]-2-methyl-5-propan-2-yloxyphenyl]piperidin-1-yl]-N-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]hexanamide	CC1=C(C2CCN(CCCCCC(=O)NC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)CC2)C=C(OC(C)C)C(NC2=NC(NC3=CC=CC=C3S(=O)(=O)C(C)C)=C(Cl)C=N2)=C1	C47H55ClN8O8S	ALK	Q9UM73	CRBN	WO-2017204445-A2
TPD-39E7TI	WO2017204445A2_18	(2R,4S)-1-[(2S)-2-[[6-[4-[4-[[5-chloro-4-(2-propan-2-ylsulfonylanilino)pyrimidin-2-yl]amino]-2-methyl-5-propan-2-yloxyphenyl]piperidin-1-yl]-6-oxohexanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=CC(NC2=NC=C(Cl)C(NC3=CC=CC=C3S(=O)(=O)C(C)C)=N2)=C(OC(C)C)C=C1C1CCN(C(=O)CCCCC(=O)N[C@H](C(=O)N2C[C@@H](O)C[C@@H]2C(=O)NCC2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)CC1	C56H72ClN9O8S2	ALK	Q9UM73	VHL	WO-2017204445-A2
TPD-MZWOZQ	WO2017204445A2_19	(2R,4S)-1-[(2S)-2-[[2-[3-[4-[4-[[5-chloro-4-(2-propan-2-ylsulfonylanilino)pyrimidin-2-yl]amino]-2-methyl-5-propan-2-yloxyphenyl]piperidin-1-yl]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=CC(NC2=NC=C(Cl)C(NC3=CC=CC=C3S(=O)(=O)C(C)C)=N2)=C(OC(C)C)C=C1C1CCN(CCCOCC(=O)N[C@H](C(=O)N2C[C@@H](O)C[C@@H]2C(=O)NCC2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)CC1	C55H72ClN9O8S2	ALK	Q9UM73	VHL	WO-2017204445-A2
TPD-WROKPE	WO2017204445A2_20	2-[3-[4-[4-[[5-chloro-4-(2-propan-2-ylsulfonylanilino)pyrimidin-2-yl]amino]-2-methyl-5-propan-2-yloxyphenyl]piperidin-1-yl]propoxy]-N-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]acetamide	CC1=CC(NC2=NC=C(Cl)C(NC3=CC=CC=C3S(=O)(=O)C(C)C)=N2)=C(OC(C)C)C=C1C1CCN(CCCOCC(=O)NC2=CC=CC3=C2C(=O)N(C2CCC(=O)NC2=O)C3=O)CC1	C46H53ClN8O9S	ALK	Q9UM73	CRBN	WO-2017204445-A2
TPD-U9EJ0F	WO2018051107A1_18a	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2[C@H](F)[C@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCNC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)C(C)(C)C)cc1	C49H59ClFN9O8S2	BRD4	O60885	VHL	WO-2018051107-A1
TPD-4UVWQR	CHEMBL4443814	(2R,3R,4S)-1-[(2S)-2-[[2-[2-[2-[2-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-3-fluoro-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL19975561; PD142801	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2[C@@H](F)[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCNC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)C(C)(C)C)cc1	C49H59ClFN9O8S2	BRD4	O60885	VHL	WO-2018051107-A1
TPD-CYBHZY	WO2018051107A1_18c	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2[C@@H](F)[C@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCNC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)C(C)(C)C)cc1	C49H59ClFN9O8S2	BRD4	O60885	VHL	WO-2018051107-A1
TPD-H4TWW1	CHEMBL5176799	(2R,3S,4S)-1-[(2S)-2-[[2-[2-[2-[2-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-3-fluoro-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL19974507; BDBM50590277; PD142799	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2[C@H](F)[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCNC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)C(C)(C)C)cc1	C49H59ClFN9O8S2	BRD4	O60885	VHL	WO-2018051107-A1
TPD-MXQ3NE	SCHEMBL19985697	(2R,3S,4S)-1-[(2S)-2-[[2-[2-[2-[[4-[(2S,4R)-1-acetyl-4-(4-chloroanilino)-2-methyl-3,4-dihydro-2H-quinolin-6-yl]benzoyl]amino]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-3-fluoro-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC(=O)N1c2ccc(-c3ccc(C(=O)NCCOCCOCC(=O)N[C@H](C(=O)N4C[C@H](O)[C@@H](F)[C@H]4C(=O)NCc4ccc(-c5scnc5C)cc4)C(C)(C)C)cc3)cc2[C@H](Nc2ccc(Cl)cc2)C[C@@H]1C	C53H61ClFN7O8S	BRD4	O60885	VHL	WO-2018051107-A1
TPD-JP0V89	SCHEMBL19985692	(2R,3R,4S)-1-[(2R)-3-[6-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]hexylsulfanyl]-2-[(1-fluorocyclopropanecarbonyl)amino]-3-methylbutanoyl]-3-fluoro-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2[C@@H](F)[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)SCCCCCCNC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)cc1	C50H58ClF2N9O5S3	BRD4	O60885	VHL	WO-2018051107-A1
TPD-XCJA0D	BRD4 degrader AT1	BRD4 degrader AT1; 2098836-45-2; AT 1; (2S,4R)-1-((R)-2-acetamido-3-((6-(2-((S)-4-(4-chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl)acetamido)hexyl)thio)-3-methylbutanoyl)-4-hydroxy-N-(4-(4-methylthiazol-5-yl)benzyl)pyrrolidine-2-carboxamide; (2S,4R)-1-(2R)-2-Acetamido-3-[[6-[2-[(6S)-4-(4-chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl]acetamido]hexyl]thio]-3-methylbutanoyl]-4-hydroxy-N-[4-(4-methylthiazol-5-yl)benzyl)pyrrolidinine-2-carboxamide; (2S,4R)-1-[(2R)-2-acetamido-3-[6-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]hexylsulfanyl]-3-methylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; orb1689886; CHEMBL4455124; SCHEMBL19985702; AT1; EX-A3221; YID83645; s8766; AKOS034834076; AC-36715; BP-40142; DA-71091; HY-111433; CS-0040740; G16274; EN300-22885103; Z3417458822; (2S,4R)-1-[(2R)-3-[(6-{2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetraazatricyclo[8.3.0.0,2,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetamido}hexyl)sulfanyl]-2-acetamido-3-methylbutanoyl]-4-hydroxy-N-{[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl}pyrrolidine-2-carboxamide	CC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(-c2scnc2C)cc1)C(C)(C)SCCCCCCNC(=O)C[C@@H]1N=C(c2ccc(Cl)cc2)c2c(sc(C)c2C)-n2c(C)nnc21	C48H58ClN9O5S3	BRD4	O60885	VHL	WO-2018051107-A1
TPD-53JFN0	SCHEMBL20129304	(2S,4R)-1-[(2S)-3,3-dimethyl-2-[[2-[2-[2-[2-[5-(5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxyethoxy]ethoxy]ethoxy]acetyl]amino]butanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOC3=NC=C(C4=CC5=C(C=C4)C4=C(C=CN=C4)N5)C=C3)C(C)(C)C)C=C2)SC=N1	C46H53N7O8S	Tau	P10636	VHL	WO-2018102067-A2
TPD-5LO5GV	SCHEMBL20120573	2-(2,6-dioxopiperidin-3-yl)-4-[2-[2-[2-[2-[5-(5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxyethoxy]ethoxy]ethoxy]ethylamino]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=C(C2=O)C(NCCOCCOCCOCCOC2=NC=C(C4=CC5=C(C=C4)C4=C(C=CN=C4)N5)C=C2)=CC=C3)C(=O)N1	C37H36N6O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-PG1TBF	SCHEMBL20120282	2-(2,6-dioxopiperidin-3-yl)-4-[2-[2-[2-[5-(5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxyethoxy]ethoxy]ethylamino]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=C(C2=O)C(NCCOCCOCCOC2=NC=C(C4=CC5=C(C=C4)C4=C(C=CN=C4)N5)C=C2)=CC=C3)C(=O)N1	C35H32N6O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-JX7FW5	SCHEMBL20120558	2-(2,6-dioxopiperidin-3-yl)-4-[2-[2-[2-[2-[2-[5-(5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]ethylamino]isoindole-1,3-dione; SCHEMBL29548103	O=C1CCC(N2C(=O)C3=CC=CC(NCCOCCOCCOCCOCCOC4=CC=C(C5=CC6=C(C=C5)C5=CN=CC=C5N6)C=N4)=C3C2=O)C(=O)N1	C39H40N6O9	Tau	P10636	CRBN	WO-2018102067-A2
TPD-TM9LYG	SCHEMBL20120508	(2S,4R)-1-[(2S)-3,3-dimethyl-2-[[2-[2-[2-[5-(5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxyethoxy]ethoxy]acetyl]amino]butanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOC3=NC=C(C4=CC5=C(C=C4)C4=C(C=CN=C4)N5)C=C3)C(C)(C)C)C=C2)SC=N1	C44H49N7O7S	Tau	P10636	VHL	WO-2018102067-A2
TPD-N89R4E	SCHEMBL20129305	(2S,4R)-1-[(2S)-3,3-dimethyl-2-[[2-[2-[2-[2-[2-[5-(5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]butanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOCCOC3=NC=C(C4=CC5=C(C=C4)C4=C(C=CN=C4)N5)C=C3)C(C)(C)C)C=C2)SC=N1	C48H57N7O9S	Tau	P10636	VHL	WO-2018102067-A2
TPD-JR375V	SCHEMBL20120477	(2S,4R)-1-[(2S)-3,3-dimethyl-2-[[2-[2-[2-[2-(4-pyrimido[1,2-a]benzimidazol-2-ylpiperazin-1-yl)ethoxy]ethoxy]ethoxy]acetyl]amino]butanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCN3CCN(C4=NC5=NC6=CC=CC=C6N5C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C44H57N9O7S	Tau	P10636	VHL	WO-2018102067-A2
TPD-1PPZ8B	SCHEMBL20120855	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[3-[2-[4-(dimethylamino)phenyl]quinolin-6-yl]oxypropoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCCOC3=CC=C4N=C(C5=CC=C(N(C)C)C=C5)C=CC4=C3)C(C)(C)C)C=C2)SC=N1	C48H60N6O8S	Tau	P10636	VHL	WO-2018102067-A2
TPD-RWNHP5	SCHEMBL20129306	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[2-[3-[2-[4-(dimethylamino)phenyl]quinolin-6-yl]oxypropoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOCCCOC3=CC=C4N=C(C5=CC=C(N(C)C)C=C5)C=CC4=C3)C(C)(C)C)C=C2)SC=N1	C50H64N6O9S	Tau	P10636	VHL	WO-2018102067-A2
TPD-LDGXUA	SCHEMBL20120953	(2S,4R)-1-[(2S)-3,3-dimethyl-2-[[2-[2-[2-[2-oxo-2-(4-pyrimido[1,2-a]benzimidazol-2-ylpiperazin-1-yl)ethoxy]ethoxy]ethoxy]acetyl]amino]butanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCC(=O)N3CCN(C4=NC5=NC6=CC=CC=C6N5C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C44H55N9O8S	Tau	P10636	VHL	WO-2018102067-A2
TPD-FRXDD2	SCHEMBL20120716	(2S,4R)-1-[(2S)-3,3-dimethyl-2-[[2-[2-[2-[2-(4-pyrimido[1,2-a]benzimidazol-2-ylpiperazin-1-yl)ethoxy]ethoxy]ethoxy]acetyl]amino]butanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-oxazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCN3CCN(C4=NC5=NC6=CC=CC=C6N5C=C4)CC3)C(C)(C)C)C=C2)OC=N1	C44H57N9O8	Tau	P10636	VHL	WO-2018102067-A2
TPD-CT4E9I	SCHEMBL20120668	(2S,4R)-1-[(2S)-3,3-dimethyl-2-[[2-[2-[2-[2-[2-(4-pyrimido[1,2-a]benzimidazol-2-ylpiperazin-1-yl)ethoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]butanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-oxazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOCCN3CCN(C4=NC5=NC6=CC=CC=C6N5C=C4)CC3)C(C)(C)C)C=C2)OC=N1	C46H61N9O9	Tau	P10636	VHL	WO-2018102067-A2
TPD-4V4IK1	SCHEMBL20120896	(2S,4R)-1-[(2S)-3,3-dimethyl-2-[[2-[2-[2-[2-oxo-2-(4-pyrimido[1,2-a]benzimidazol-2-ylpiperazin-1-yl)ethoxy]ethoxy]ethoxy]acetyl]amino]butanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-oxazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCC(=O)N3CCN(C4=NC5=NC6=CC=CC=C6N5C=C4)CC3)C(C)(C)C)C=C2)OC=N1	C44H55N9O9	Tau	P10636	VHL	WO-2018102067-A2
TPD-M9N91P	SCHEMBL20120616	(2S,4R)-1-[(2S)-3,3-dimethyl-2-[[2-[2-[2-[2-[2-oxo-2-(4-pyrimido[1,2-a]benzimidazol-2-ylpiperazin-1-yl)ethoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]butanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-oxazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOCC(=O)N3CCN(C4=NC5=NC6=CC=CC=C6N5C=C4)CC3)C(C)(C)C)C=C2)OC=N1	C46H59N9O10	Tau	P10636	VHL	WO-2018102067-A2
TPD-PFX2B7	SCHEMBL20120505	(2S,4R)-1-[(2S)-3,3-dimethyl-2-[[2-[2-[2-[2-(4-pyrimido[1,2-a]benzimidazol-2-ylpiperazin-1-yl)ethoxy]ethoxy]ethoxy]acetyl]amino]butanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCN3CCN(C4=NC5=NC6=CC=CC=C6N5C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C45H59N9O7S	Tau	P10636	VHL	WO-2018102067-A2
TPD-MQ578F	SCHEMBL20120842	(2S,4R)-1-[(2S)-3,3-dimethyl-2-[[2-[2-[2-[2-[2-(4-pyrimido[1,2-a]benzimidazol-2-ylpiperazin-1-yl)ethoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]butanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOCCN3CCN(C4=NC5=NC6=CC=CC=C6N5C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C47H63N9O8S	Tau	P10636	VHL	WO-2018102067-A2
TPD-OVL24J	SCHEMBL20120840	(2S,4R)-1-[(2S)-3,3-dimethyl-2-[[2-[2-[2-[2-oxo-2-(4-pyrimido[1,2-a]benzimidazol-2-ylpiperazin-1-yl)ethoxy]ethoxy]ethoxy]acetyl]amino]butanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCC(=O)N3CCN(C4=NC5=NC6=CC=CC=C6N5C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C45H57N9O8S	Tau	P10636	VHL	WO-2018102067-A2
TPD-3NP4NB	SCHEMBL20120978	(2S,4R)-1-[(2S)-3,3-dimethyl-2-[[2-[2-[2-[2-[2-oxo-2-(4-pyrimido[1,2-a]benzimidazol-2-ylpiperazin-1-yl)ethoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]butanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOCC(=O)N3CCN(C4=NC5=NC6=CC=CC=C6N5C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C47H61N9O9S	Tau	P10636	VHL	WO-2018102067-A2
TPD-CWZGI7	SCHEMBL20120393	(2S,4R)-1-[(2S)-3,3-dimethyl-2-[[2-[2-[2-[2-(4-pyrimido[1,2-a]benzimidazol-2-ylpiperazin-1-yl)ethoxy]ethoxy]ethoxy]acetyl]amino]butanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-oxazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCN3CCN(C4=NC5=NC6=CC=CC=C6N5C=C4)CC3)C(C)(C)C)C=C2)OC=N1	C45H59N9O8	Tau	P10636	VHL	WO-2018102067-A2
TPD-90E30F	SCHEMBL20120823	(2S,4R)-1-[(2S)-3,3-dimethyl-2-[[2-[2-[2-[2-[2-(4-pyrimido[1,2-a]benzimidazol-2-ylpiperazin-1-yl)ethoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]butanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-oxazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOCCN3CCN(C4=NC5=NC6=CC=CC=C6N5C=C4)CC3)C(C)(C)C)C=C2)OC=N1	C47H63N9O9	Tau	P10636	VHL	WO-2018102067-A2
TPD-V8I7QG	SCHEMBL20129307	(2S,4R)-1-[(2S)-3,3-dimethyl-2-[[2-[2-[2-[2-oxo-2-(4-pyrimido[1,2-a]benzimidazol-2-ylpiperazin-1-yl)ethoxy]ethoxy]ethoxy]acetyl]amino]butanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-oxazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCC(=O)N3CCN(C4=NC5=NC6=CC=CC=C6N5C=C4)CC3)C(C)(C)C)C=C2)OC=N1	C45H57N9O9	Tau	P10636	VHL	WO-2018102067-A2
TPD-U46WTX	SCHEMBL20120534	(2S,4R)-1-[(2S)-3,3-dimethyl-2-[[2-[2-[2-[2-[2-oxo-2-(4-pyrimido[1,2-a]benzimidazol-2-ylpiperazin-1-yl)ethoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]butanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-oxazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOCC(=O)N3CCN(C4=NC5=NC6=CC=CC=C6N5C=C4)CC3)C(C)(C)C)C=C2)OC=N1	C47H61N9O10	Tau	P10636	VHL	WO-2018102067-A2
TPD-8IRFVT	SCHEMBL20129309	(2S,4R)-1-[(2S)-3,3-dimethyl-2-[[2-[2-[2-[2-[2-(4-pyrimido[1,2-a]benzimidazol-2-ylpiperazin-1-yl)ethoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]butanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOCCN3CCN(C4=NC5=NC6=CC=CC=C6N5C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C46H61N9O8S	Tau	P10636	VHL	WO-2018102067-A2
TPD-8RWIZJ	SCHEMBL20129308	(2S,4R)-1-[(2S)-3,3-dimethyl-2-[[2-[2-[2-[2-[2-oxo-2-(4-pyrimido[1,2-a]benzimidazol-2-ylpiperazin-1-yl)ethoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]butanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOCC(=O)N3CCN(C4=NC5=NC6=CC=CC=C6N5C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C46H59N9O9S	Tau	P10636	VHL	WO-2018102067-A2
TPD-36470U	SCHEMBL20120563	2-(2,6-Dioxopiperidin-3-yl)-4-[2-[2-[2-[2-(4-pyrimido[1,2-a]benzimidazol-2-ylpiperazin-1-yl)ethoxy]ethoxy]ethoxy]ethylamino]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC=CC(NCCOCCOCCOCCN4CCN(C5=NC6=NC7=CC=CC=C7N6C=C5)CC4)=C3C2=O)C(=O)N1	C35H40N8O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-98O5NW	SCHEMBL20120423	2-(2,6-Dioxopiperidin-3-yl)-4-[2-[2-[2-[2-[2-(4-pyrimido[1,2-a]benzimidazol-2-ylpiperazin-1-yl)ethoxy]ethoxy]ethoxy]ethoxy]ethylamino]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=C(C2=O)C(NCCOCCOCCOCCOCCN2CCN(C4=NC5=NC6=CC=CC=C6N5C=C4)CC2)=CC=C3)C(=O)N1	C37H44N8O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-QP31M3	SCHEMBL20120696	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[2-[4-(dimethylamino)phenyl]quinolin-6-yl]oxyethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOC3=CC=C4N=C(C5=CC=C(N(C)C)C=C5)C=CC4=C3)C(C)(C)C)C=C2)SC=N1	C45H54N6O7S	Tau	P10636	VHL	WO-2018102067-A2
TPD-HVG1X3	SCHEMBL20121032	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[2-[4-(dimethylamino)phenyl]quinolin-6-yl]oxyethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOC3=CC=C4N=C(C5=CC=C(N(C)C)C=C5)C=CC4=C3)C(C)(C)C)C=C2)SC=N1	C46H56N6O7S	Tau	P10636	VHL	WO-2018102067-A2
TPD-3Y0ZTH	WO2018102067A2_29	.	CC1=C(C2=CC=C(CNC(=O)C3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOC3=CC=C4N=C(C5=CC=C(N(C)C)C=C5)C=CC4=C3)C(C)(C)C)C=C2)SC=N1	C47H58N6O8S	Tau	P10636	VHL	WO-2018102067-A2
TPD-EZP0E6	SCHEMBL20129311	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[2-[2-[4-(dimethylamino)phenyl]quinolin-6-yl]oxyethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOC3=CC=C4N=C(C5=CC=C(N(C)C)C=C5)C=CC4=C3)C(C)(C)C)C=C2)SC=N1	C48H60N6O8S	Tau	P10636	VHL	WO-2018102067-A2
TPD-K0K3AH	SCHEMBL20129312	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[2-[2-[2-[4-(dimethylamino)phenyl]quinolin-6-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOCCOC3=CC=C4N=C(C5=CC=C(N(C)C)C=C5)C=CC4=C3)C(C)(C)C)C=C2)SC=N1	C49H62N6O9S	Tau	P10636	VHL	WO-2018102067-A2
TPD-DSVPLC	SCHEMBL20129313	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[2-[2-[2-[4-(dimethylamino)phenyl]quinolin-6-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOCCOC3=CC=C4N=C(C5=CC=C(N(C)C)C=C5)C=CC4=C3)C(C)(C)C)C=C2)SC=N1	C50H64N6O9S	Tau	P10636	VHL	WO-2018102067-A2
TPD-QQBHHM	SCHEMBL20120850	(2S,4R)-1-[(2S)-2-[[2-[4-[2-[4-(dimethylamino)phenyl]quinolin-6-yl]oxybutoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCOC3=CC=C4N=C(C5=CC=C(N(C)C)C=C5)C=CC4=C3)C(C)(C)C)C=C2)SC=N1	C45H54N6O6S	Tau	P10636	VHL	WO-2018102067-A2
TPD-V2A7TY	SCHEMBL20120917	(2S,4R)-1-[(2S)-2-[[2-[4-[2-[4-(dimethylamino)phenyl]quinolin-6-yl]oxybutoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCOC3=CC=C4N=C(C5=CC=C(N(C)C)C=C5)C=CC4=C3)C(C)(C)C)C=C2)SC=N1	C46H56N6O6S	Tau	P10636	VHL	WO-2018102067-A2
TPD-BC1R84	SCHEMBL20120530	(2S,4R)-1-[(2S)-2-[[2-[3-[3-[2-[4-(dimethylamino)phenyl]quinolin-6-yl]oxypropoxy]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCOCCCOC3=CC=C4N=C(C5=CC=C(N(C)C)C=C5)C=CC4=C3)C(C)(C)C)C=C2)SC=N1	C47H58N6O7S	Tau	P10636	VHL	WO-2018102067-A2
TPD-NPSE62	SCHEMBL20120745	(2S,4R)-1-[(2S)-2-[[2-[3-[3-[2-[4-(dimethylamino)phenyl]quinolin-6-yl]oxypropoxy]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCOCCCOC3=CC=C4N=C(C5=CC=C(N(C)C)C=C5)C=CC4=C3)C(C)(C)C)C=C2)SC=N1	C48H60N6O7S	Tau	P10636	VHL	WO-2018102067-A2
TPD-ZOWC9O	SCHEMBL20120630	(2S,4R)-1-[(2S)-2-[[2-[5-[2-[4-(dimethylamino)phenyl]quinolin-6-yl]oxypentoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCCOC3=CC=C4N=C(C5=CC=C(N(C)C)C=C5)C=CC4=C3)C(C)(C)C)C=C2)SC=N1	C46H56N6O6S	Tau	P10636	VHL	WO-2018102067-A2
TPD-TPEJ6Q	SCHEMBL20120522	(2S,4R)-1-[(2S)-2-[[2-[5-[2-[4-(dimethylamino)phenyl]quinolin-6-yl]oxypentoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCCOC3=CC=C4N=C(C5=CC=C(N(C)C)C=C5)C=CC4=C3)C(C)(C)C)C=C2)SC=N1	C47H58N6O6S	Tau	P10636	VHL	WO-2018102067-A2
TPD-GUB688	SCHEMBL20129314	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[2-[3-[2-[4-(dimethylamino)phenyl]quinolin-6-yl]oxypropoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOCCCOC3=CC=C4N=C(C5=CC=C(N(C)C)C=C5)C=CC4=C3)C(C)(C)C)C=C2)SC=N1	C51H66N6O9S	Tau	P10636	VHL	WO-2018102067-A2
TPD-2HD0Q5	SCHEMBL20120380	4-[2-[2-[2-[2-[3-[2-[4-(Dimethylamino)phenyl]quinolin-6-yl]oxypropoxy]ethoxy]ethoxy]ethoxy]ethylamino]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN(C)C1=CC=C(C2=NC3=CC=C(OCCCOCCOCCOCCOCCNC4=CC=CC5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)C=C3C=C2)C=C1	C41H47N5O9	Tau	P10636	CRBN	WO-2018102067-A2
TPD-8RZJ2C	SCHEMBL20120915	2-(2,6-Dioxopiperidin-3-yl)-4-[2-[2-[2-[2-oxo-2-(4-pyrimido[1,2-a]benzimidazol-2-ylpiperazin-1-yl)ethoxy]ethoxy]ethoxy]ethylamino]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC=CC(NCCOCCOCCOCC(=O)N4CCN(C5=NC6=NC7=CC=CC=C7N6C=C5)CC4)=C3C2=O)C(=O)N1	C35H38N8O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-KACMP0	SCHEMBL20120942	2-(2,6-Dioxopiperidin-3-yl)-4-[2-[2-[2-[2-[2-oxo-2-(4-pyrimido[1,2-a]benzimidazol-2-ylpiperazin-1-yl)ethoxy]ethoxy]ethoxy]ethoxy]ethylamino]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=C(C2=O)C(NCCOCCOCCOCCOCC(=O)N2CCN(C4=NC5=NC6=CC=CC=C6N5C=C4)CC2)=CC=C3)C(=O)N1	C37H42N8O9	Tau	P10636	CRBN	WO-2018102067-A2
TPD-7XFJ90	SCHEMBL20120986	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[3-[2-[4-(dimethylamino)phenyl]quinolin-6-yl]oxy-2-hydroxypropoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCC(O)COC3=CC=C4N=C(C5=CC=C(N(C)C)C=C5)C=CC4=C3)C(C)(C)C)C=C2)SC=N1	C48H60N6O9S	Tau	P10636	VHL	WO-2018102067-A2
TPD-UOTT6F	SCHEMBL20120428	4-[2-[2-[2-[3-[2-[4-(Dimethylamino)phenyl]quinolin-6-yl]oxypropoxy]ethoxy]ethoxy]ethylamino]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN(C)C1=CC=C(C2=NC3=CC=C(OCCCOCCOCCOCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C3C=C2)C=C1	C39H43N5O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-BDM0CF	SCHEMBL20120740	4-[2-[2-[2-[2-[3-[2-[4-(Dimethylamino)phenyl]quinolin-6-yl]oxy-2-hydroxypropoxy]ethoxy]ethoxy]ethoxy]ethylamino]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN(C)C1=CC=C(C2=NC3=CC=C(OCC(O)COCCOCCOCCOCCNC4=CC=CC5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)C=C3C=C2)C=C1	C41H47N5O10	Tau	P10636	CRBN	WO-2018102067-A2
TPD-5YKTS2	SCHEMBL20129315	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[2-[3-[2-[4-(dimethylamino)phenyl]quinolin-6-yl]oxy-2-hydroxypropoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOCC(O)COC3=CC=C4N=C(C5=CC=C(N(C)C)C=C5)C=CC4=C3)C(C)(C)C)C=C2)SC=N1	C50H64N6O10S	Tau	P10636	VHL	WO-2018102067-A2
TPD-3ZX3AI	SCHEMBL20129316	4-[2-[2-[2-[3-[2-[4-(Dimethylamino)phenyl]quinolin-6-yl]oxy-2-hydroxypropoxy]ethoxy]ethoxy]ethylamino]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN(C)C1=CC=C(C2=NC3=CC=C(OCC(O)COCCOCCOCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C3C=C2)C=C1	C39H43N5O9	Tau	P10636	CRBN	WO-2018102067-A2
TPD-XEMLYI	SCHEMBL20120403	2-(2,6-Dioxopiperidin-3-yl)-4-[2-[2-[2-[2-[2-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]ethylamino]isoindole-1,3-dione	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(OCCOCCOCCOCCOCCNC3=CC=CC4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)C=C1)C=C2	C40H42N6O9	Tau	P10636	CRBN	WO-2018102067-A2
TPD-0O4YO9	SCHEMBL20120521	3-[3-oxo-7-[2-[2-[2-[2-[2-[5-(5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]ethylamino]-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL29547399	O=C1CCC(N2CC3=C(C=CC=C3NCCOCCOCCOCCOCCOC3=NC=C(C4=CC5=C(C=C4)C4=C(C=CN=C4)N5)C=C3)C2=O)C(=O)N1	C39H42N6O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-VWOKOL	SCHEMBL20120703	3-[3-oxo-7-[2-[2-[2-[2-[2-[5-(5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]ethoxy]-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC=C3OCCOCCOCCOCCOCCOC3=NC=C(C4=CC5=C(C=C4)C4=C(C=CN=C4)N5)C=C3)C2=O)C(=O)N1	C39H41N5O9	Tau	P10636	CRBN	WO-2018102067-A2
TPD-AEMMRJ	SCHEMBL20120834	2-(2,6-dioxopiperidin-3-yl)-5-[2-[2-[2-[2-[2-[5-(5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]ethoxy]isoindole-1,3-dione; SCHEMBL29547543	O=C1CCC(N2C(=O)C3=C(C=C(OCCOCCOCCOCCOCCOC4=NC=C(C5=CC6=C(C=C5)C5=CN=CC=C5N6)C=C4)C=C3)C2=O)C(=O)N1	C39H39N5O10	Tau	P10636	CRBN	WO-2018102067-A2
TPD-5XIOIA	SCHEMBL20120867	2-(2,6-dioxopiperidin-3-yl)-5-[5-[4-[2-[3-[5-(5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]propoxy]ethyl]piperazin-1-yl]pentoxy]isoindole-1,3-dione; SCHEMBL29547499	O=C1CCC(N2C(=O)C3=C(C=C(OCCCCCN4CCN(CCOCCCC5=NC=C(C6=CC7=C(C=C6)C6=CN=CC=C6N7)C=C5)CC4)C=C3)C2=O)C(=O)N1	C43H47N7O6	Tau	P10636	CRBN	WO-2018102067-A2
TPD-CARXFF	SCHEMBL20120454	2-(2,6-dioxopiperidin-3-yl)-5-[4-[3-[3-[5-(5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypropyl]piperazin-1-yl]isoindole-1,3-dione; SCHEMBL20120456; SCHEMBL20120483; SCHEMBL29547546	O=C1CCC(N2C(=O)C3=C(C=C(N4CCN(CCCO[C@H]5C[C@@H](OC6=NC=C(C7=CC8=C(C=C7)C7=CN=CC=C7N8)C=C6)C5)CC4)C=C3)C2=O)C(=O)N1	C40H39N7O6	Tau	P10636	CRBN	WO-2018102067-A2
TPD-JCE33C	SCHEMBL20120641	2-(2,6-dioxopiperidin-3-yl)-5-[5-[4-[3-[5-(5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]propyl]piperazin-1-yl]pentoxy]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=C(C=C(OCCCCCN4CCN(CCCC5=NC=C(C6=CC7=C(C=C6)C6=CN=CC=C6N7)C=C5)CC4)C=C3)C2=O)C(=O)N1	C41H43N7O5	Tau	P10636	CRBN	WO-2018102067-A2
TPD-BRLPXI	SCHEMBL20120243	2-(2,6-dioxopiperidin-3-yl)-5-[3-[6-[4-[3-[5-(5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]propyl]piperazin-1-yl]pyridin-3-yl]propoxy]isoindole-1,3-dione; SCHEMBL29547699	O=C1CCC(N2C(=O)C3=C(C=C(OCCCC4=CN=C(N5CCN(CCCC6=NC=C(C7=CC8=C(C=C7)C7=CN=CC=C7N8)C=C6)CC5)C=C4)C=C3)C2=O)C(=O)N1	C44H42N8O5	Tau	P10636	CRBN	WO-2018102067-A2
TPD-29B0WK	WO2018102067A2_56	.	O=C1CCC(N2C(=O)C3=C(C=C(OCCCCCN4CCN(CCO[C@H]5C[C@@H](OC6=NC=C(C7=CC8=C(C=C7)C7=CN=CC=C7N8)C=C6)C5)CC4)C=C3)C2=O)C(=O)N1	C44H47N7O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-AS0FI1	SCHEMBL20120938	2-(2,6-dioxopiperidin-3-yl)-5-[2-[2-[2-[2-[2-[4-(5H-pyrido[4,3-b]indol-7-yl)piperidin-1-yl]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]isoindole-1,3-dione; SCHEMBL29547968	O=C1CCC(N2C(=O)C3=C(C=C(OCCOCCOCCOCCOCCN4CCC(C5=CC6=C(C=C5)C5=CN=CC=C5N6)CC4)C=C3)C2=O)C(=O)N1	C39H45N5O9	Tau	P10636	CRBN	WO-2018102067-A2
TPD-PZ2SI9	SCHEMBL20120473	2-(2,6-dioxopiperidin-3-yl)-5-[5-[2-[4-[3-[5-(5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]propyl]piperazin-1-yl]ethoxy]pentoxy]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=C(C=C(OCCCCCOCCN4CCN(CCCC5=NC=C(C6=CC7=C(C=C6)C6=CN=CC=C6N7)C=C5)CC4)C=C3)C2=O)C(=O)N1	C43H47N7O6	Tau	P10636	CRBN	WO-2018102067-A2
TPD-9H1S6Q	WO2018102067A2_59	.	O=C1CCC(N2C(=O)C3=C(C=C(OCCCCCN4CCN(CCO[C@H]5C[C@H](OC6=NC=C(C7=CC8=C(C=C7)C7=CN=CC=C7N8)C=C6)C5)CC4)C=C3)C2=O)C(=O)N1	C44H47N7O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-OH6PMT	WO2018102067A2_60	.	O=C1CCC(N2C(=O)C3=C(C=C(N4CCN(CCCO[C@H]5C[C@H](OC6=NC=C(C7=CC8=C(C=C7)C7=CN=CC=C7O8)C=C6)C5)CC4)C=C3)C2=O)C(=O)N1	C40H38N6O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-OS61A3	SCHEMBL20120857	2-(2,6-Dioxopiperidin-3-yl)-5-[5-[4-[3-[5-[5-(2,2,2-trifluoroethyl)pyrido[4,3-b]indol-7-yl]pyridin-2-yl]propyl]piperazin-1-yl]pentoxy]isoindole-1,3-dione; SCHEMBL29547558; KKEJTBILIMLIMX-UHFFFAOYSA-N; 2-(2,6-Dioxopiperidin-3-yl)-5-[5-[4-[3-[5-[5-(2,2,2-trifluoroethyl)pyrido[4,3-b]indol-7-yl]pyridin-2-yl]propyl]piperazin-1-yl]pentoxy]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=C(C=C(OCCCCCN4CCN(CCCC5=NC=C(C6=CC7=C(C=C6)C6=CN=CC=C6N7CC(F)(F)F)C=C5)CC4)C=C3)C2=O)C(=O)N1	C43H44F3N7O5	Tau	P10636	CRBN	WO-2018102067-A2
TPD-K5Y3NP	SCHEMBL20120746	3-[6-[5-[4-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]propyl]piperazin-1-yl]pentoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL29547578	CN1C2=CC=NC=C2C2=C1C=C(C1=CN=C(CCCN3CCN(CCCCCOC4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5)CC3)C=C1)C=C2	C42H47N7O4	Tau	P10636	CRBN	WO-2018102067-A2
TPD-FKHNKF	SCHEMBL20120541	2-(2,6-Dioxopiperidin-3-yl)-5-[5-[4-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)-3-(trifluoromethyl)pyridin-2-yl]propyl]piperazin-1-yl]pentoxy]isoindole-1,3-dione; SCHEMBL29547700; NAXVDGXEPMYEMD-UHFFFAOYSA-N; 2-(2,6-Dioxopiperidin-3-yl)-5-[5-[4-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)-3-(trifluoromethyl)pyridin-2-yl]propyl]piperazin-1-yl]pentoxy]isoindole-1,3-dione	CN1C2=CC=NC=C2C2=C1C=C(C1=CN=C(CCCN3CCN(CCCCCOC4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)C(C(F)(F)F)=C1)C=C2	C43H44F3N7O5	Tau	P10636	CRBN	WO-2018102067-A2
TPD-6937SP	WO2018102067A2_64	.	CN1C2=CC=NC=C2C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4=CN=C(CCCN5CCN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C=C4)C3)C=C1)C=C2	C46H44N8O6	Tau	P10636	CRBN	WO-2018102067-A2
TPD-CXHLAN	SCHEMBL20120801	2-(2,6-dioxopiperidin-3-yl)-5-[5-[4-[3-[5-(5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]pentoxy]isoindole-1,3-dione; SCHEMBL20120898; SCHEMBL29547241; SCHEMBL29773830	O=C1CCC(N2C(=O)C3=C(C=C(OCCCCCN4CCC(O[C@H]5C[C@H](OC6=NC=C(C7=CC8=C(C=C7)C7=CN=CC=C7N8)C=C6)C5)CC4)C=C3)C2=O)C(=O)N1	C43H44N6O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-RATL65	SCHEMBL20120290	2-(2,6-dioxopiperidin-3-yl)-5-[4-[2-[4-[3-[5-(5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]ethyl]piperazin-1-yl]isoindole-1,3-dione; SCHEMBL20120292; SCHEMBL30302301	O=C1CCC(N2C(=O)C3=C(C=C(N4CCN(CCN5CCC(O[C@H]6C[C@H](OC7=NC=C(C8=CC9=C(C=C8)C8=CN=CC=C8N9)C=C7)C6)CC5)CC4)C=C3)C2=O)C(=O)N1	C44H46N8O6	Tau	P10636	CRBN	WO-2018102067-A2
TPD-KN6N0K	SCHEMBL20120593	2-(2,6-Dioxopiperidin-3-yl)-5-[2-[2-[2-[2-[2-[5-(5-methylpyrido[4,3-b]indol-7-yl)-3-(trifluoromethyl)pyridin-2-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]ethoxy]isoindole-1,3-dione; GKMLGWJWJMAWKR-UHFFFAOYSA-N; 2-(2,6-Dioxopiperidin-3-yl)-5-[2-[2-[2-[2-[2-[5-(5-methylpyrido[4,3-b]indol-7-yl)-3-(trifluoromethyl)pyridin-2-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]ethoxy]isoindole-1,3-dione	CN1C2=CC=NC=C2C2=C1C=C(C1=CN=C(OCCOCCOCCOCCOCCOC3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C(C(F)(F)F)=C1)C=C2	C41H40F3N5O10	Tau	P10636	CRBN	WO-2018102067-A2
TPD-DO0K7F	SCHEMBL20120556	2-(2,6-Dioxopiperidin-3-yl)-5-[4-[5-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypentyl]piperazin-1-yl]isoindole-1,3-dione; SCHEMBL20120557; SCHEMBL29547561	CN1C2=CC=NC=C2C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OCCCCCN4CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C3)C=C1)C=C2	C43H45N7O6	Tau	P10636	CRBN	WO-2018102067-A2
TPD-2JFBDJ	SCHEMBL20120510	2-(2,6-Dioxopiperidin-3-yl)-5-[2-[2-[2-[2-[2-[5-(5-methylpyrido[4,3-b]indol-7-yl)-4-(trifluoromethyl)pyridin-2-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]ethoxy]isoindole-1,3-dione; NOERFWBWTYPCRB-UHFFFAOYSA-N; 2-(2,6-Dioxopiperidin-3-yl)-5-[2-[2-[2-[2-[2-[5-(5-methylpyrido[4,3-b]indol-7-yl)-4-(trifluoromethyl)pyridin-2-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]ethoxy]isoindole-1,3-dione	CN1C2=CC=NC=C2C2=C1C=C(C1=CN=C(OCCOCCOCCOCCOCCOC3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C=C1C(F)(F)F)C=C2	C41H40F3N5O10	Tau	P10636	CRBN	WO-2018102067-A2
TPD-FA59K3	SCHEMBL20120452	2-(2,6-Dioxopiperidin-3-yl)-5-[2-[2-[2-[2-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxyethoxy]ethoxy]ethoxy]ethoxy]isoindole-1,3-dione; SCHEMBL20120453; SCHEMBL29547345	CN1C2=CC=NC=C2C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OCCOCCOCCOCCOC4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)C=C1)C=C2	C42H43N5O10	Tau	P10636	CRBN	WO-2018102067-A2
TPD-ETC4Y1	SCHEMBL20120708	2-(2,6-Dioxopiperidin-3-yl)-5-[2-[2-[2-[2-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]prop-2-ynoxy]ethoxy]ethoxy]ethoxy]ethoxy]isoindole-1,3-dione; SCHEMBL29547567	CN1C2=CC=NC=C2C2=C1C=C(C1=CN=C(C#CCOCCOCCOCCOCCOC3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C=C1)C=C2	C41H39N5O9	Tau	P10636	CRBN	WO-2018102067-A2
TPD-6M2DZ4	SCHEMBL20120952	2-(2,6-dioxopiperidin-3-yl)-4,5,7-trifluoro-6-[2-[2-[2-[2-[2-[5-(5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]ethoxy]isoindole-1,3-dione; SCHEMBL29547461	O=C1CCC(N2C(=O)C3=C(F)C(F)=C(OCCOCCOCCOCCOCCOC4=CC=C(C5=CC6=C(C=C5)C5=CN=CC=C5N6)C=N4)C(F)=C3C2=O)C(=O)N1	C39H36F3N5O10	Tau	P10636	CRBN	WO-2018102067-A2
TPD-I04YY1	WO2018102067A2_73	.	O=C1CCC(N2C(=O)C3=C(C=C(OCC#CC4=NC=C(O[C@H]5C[C@H](OC6=NC=C(C7=CC8=C(C=C7)C7=CN=CC=C7N8)C=C6)C5)C=C4)C=C3)C2=O)C(=O)N1	C41H30N6O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-9ICHIR	WO2018102067A2_74	.	O=C1CCC(N2C(=O)C3=C(C=C(OCCOCCOCCOCCOCCCC4=NC=C(C5=CC6=C(C=C5)C5=CN=CC=C5N6)C=C4)C=C3)C2=O)C(=O)N1	C40H41N5O9	Tau	P10636	CRBN	WO-2018102067-A2
TPD-MLC3L1	SCHEMBL20120798	2-(2,6-Dioxopiperidin-3-yl)-5-[4-[5-[5-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxypentoxy]pentyl]piperidin-1-yl]isoindole-1,3-dione; SCHEMBL29547818	CN1C2=CC=NC=C2C2=C1C=C(C1=CN=C(OCCCCCOCCCCCC3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)C=C1)C=C2	C45H50N6O6	Tau	P10636	CRBN	WO-2018102067-A2
TPD-ZPK6HC	SCHEMBL20120698	2-(2,6-Dioxopiperidin-3-yl)-5-[3-[3-[4-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]prop-2-ynyl]piperazin-1-yl]propoxy]azetidin-1-yl]isoindole-1,3-dione; SCHEMBL29548182	CN1C2=CC=NC=C2C2=C1C=C(C1=CN=C(C#CCN3CCN(CCCOC4CN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)CC3)C=C1)C=C2	C43H42N8O5	Tau	P10636	CRBN	WO-2018102067-A2
TPD-H62EE7	SCHEMBL20120519	2-(2,6-dioxopiperidin-3-yl)-5-[3-[5-[3-[5-(5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]propoxy]isoindole-1,3-dione; SCHEMBL20120520; SCHEMBL29547859	O=C1CCC(N2C(=O)C3=C(C=C(OCCCC4=NC=C(O[C@H]5C[C@H](OC6=NC=C(C7=CC8=C(C=C7)C7=CN=CC=C7N8)C=C6)C5)C=C4)C=C3)C2=O)C(=O)N1	C41H34N6O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-LFJBFH	SCHEMBL20120482	2-(2,6-Dioxopiperidin-3-yl)-5-[4-[6-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxyhexyl]piperazin-1-yl]isoindole-1,3-dione; SCHEMBL20128949; SCHEMBL29548345	CN1C2=CC=NC=C2C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OCCCCCCN4CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C3)C=C1)C=C2	C44H47N7O6	Tau	P10636	CRBN	WO-2018102067-A2
TPD-PF7G5K	SCHEMBL20120621	2-(2,6-Dioxopiperidin-3-yl)-5-[3-[5-[5-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxypentoxy]pentoxy]azetidin-1-yl]isoindole-1,3-dione; SCHEMBL29547622	CN1C2=CC=NC=C2C2=C1C=C(C1=CN=C(OCCCCCOCCCCCOC3CN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)C=C1)C=C2	C43H46N6O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-NUPMD7	SCHEMBL20120365	2-(2,6-Dioxopiperidin-3-yl)-5-[1-[5-[5-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxypentoxy]pentyl]azetidin-3-yl]oxyisoindole-1,3-dione; SCHEMBL29547474	CN1C2=CC=NC=C2C2=C1C=C(C1=CN=C(OCCCCCOCCCCCN3CC(OC4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)C=C1)C=C2	C43H46N6O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-WOIW1B	SCHEMBL20121003	2-(2,6-dioxopiperidin-3-yl)-5-fluoro-6-[2-[2-[2-[2-[2-[5-(5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]ethoxy]isoindole-1,3-dione; SCHEMBL29547332	O=C1CCC(N2C(=O)C3=CC(F)=C(OCCOCCOCCOCCOCCOC4=CC=C(C5=CC6=C(C=C5)C5=CN=CC=C5N6)C=N4)C=C3C2=O)C(=O)N1	C39H38FN5O10	Tau	P10636	CRBN	WO-2018102067-A2
TPD-VU3VON	SCHEMBL20120709	2-(2,6-Dioxopiperidin-3-yl)-5-[5-[4-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]pentoxy]isoindole-1,3-dione; SCHEMBL20120711; SCHEMBL30302314	CN1C2=CC=NC=C2C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4CCN(CCCCCOC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C3)C=C1)C=C2	C44H46N6O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-WBHZXM	SCHEMBL20120318	2-(2,6-dioxopiperidin-3-yl)-5-[5-[5-[3-[5-(5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]pentoxy]isoindole-1,3-dione; SCHEMBL20120319; SCHEMBL30302385	O=C1CCC(N2C(=O)C3=C(C=C(OCCCCCC4=NC=C(O[C@H]5C[C@H](OC6=NC=C(C7=CC8=C(C=C7)C7=CN=CC=C7N8)C=C6)C5)C=C4)C=C3)C2=O)C(=O)N1	C43H38N6O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-QSJ610	SCHEMBL20120412	2-(2,6-Dioxopiperidin-3-yl)-5-[6-[3-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxyphenoxy]hexoxy]isoindole-1,3-dione; SCHEMBL20120644; SCHEMBL29547312	CN1C2=CC=NC=C2C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4=CC=CC(OCCCCCCOC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)=C4)C3)C=C1)C=C2	C46H43N5O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-WEM6UF	SCHEMBL20120959	2-(2,6-Dioxopiperidin-3-yl)-5-[3-[5-[5-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxypentoxy]pentoxy]cyclobutyl]oxyisoindole-1,3-dione; SCHEMBL20120960; SCHEMBL29547695	CN1C2=CC=NC=C2C2=C1C=C(C1=CN=C(OCCCCCOCCCCCO[C@H]3C[C@H](OC4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)C=C1)C=C2	C44H47N5O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-7GVA2K	SCHEMBL20120827	2-(2,6-dioxopiperidin-3-yl)-4-[2-[2-[2-[2-[2-[4-(5H-pyrido[4,3-b]indol-7-yl)phenoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethylamino]isoindole-1,3-dione; SCHEMBL29773874	O=C1CCC(N2C(=O)C3=C(C2=O)C(NCCOCCOCCOCCOCCOC2=CC=C(C4=CC5=C(C=C4)C4=CN=CC=C4N5)C=C2)=CC=C3)C(=O)N1	C40H41N5O9	Tau	P10636	CRBN	WO-2018102067-A2
TPD-A2C12A	SCHEMBL20120540	2-(2,6-dioxopiperidin-3-yl)-6-[2-[2-[2-[2-[2-[5-(5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]ethoxy]pyrrolo[3,4-c]pyridine-1,3-dione; SCHEMBL29548268	O=C1CCC(N2C(=O)C3=CN=C(OCCOCCOCCOCCOCCOC4=CC=C(C5=CC6=C(C=C5)C5=CN=CC=C5N6)C=N4)C=C3C2=O)C(=O)N1	C38H38N6O10	Tau	P10636	CRBN	WO-2018102067-A2
TPD-57BJ4E	SCHEMBL20120302	2-(2,6-Dioxopiperidin-3-yl)-5-[2-[2-[2-[2-[2-[5-[5-(2,2,2-trifluoroethyl)pyrido[4,3-b]indol-7-yl]pyridin-2-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]ethoxy]isoindole-1,3-dione; YXCXUCXJAZIZTH-UHFFFAOYSA-N; 2-(2,6-Dioxopiperidin-3-yl)-5-[2-[2-[2-[2-[2-[5-[5-(2,2,2-trifluoroethyl)pyrido[4,3-b]indol-7-yl]pyridin-2-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]ethoxy]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=C(C=C(OCCOCCOCCOCCOCCOC4=NC=C(C5=CC6=C(C=C5)C5=CN=CC=C5N6CC(F)(F)F)C=C4)C=C3)C2=O)C(=O)N1	C41H40F3N5O10	Tau	P10636	CRBN	WO-2018102067-A2
TPD-U5OTJE	WO2018102067A2_89	.	CN1C2=CC=NC=C2C2=C1C=C(C1=CN=C(OCCCCCOCCOC(CF)CC3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)C=C1)C=C2	C45H49FN6O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-0A989U	SCHEMBL20120756	5-[2-[2-[2-[2-[2-[3-Chloro-5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]ethoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione; SCHEMBL29548070	CN1C2=CC(C3=CN=C(OCCOCCOCCOCCOCCOC4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)C(Cl)=C3)=CC=C2C2=C1C=CN=C2	C40H40ClN5O10	Tau	P10636	CRBN	WO-2018102067-A2
TPD-N8ET7K	SCHEMBL20120462	2-(2,6-Dioxopiperidin-3-yl)-5-[5-[5-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]pent-4-ynoxy]isoindole-1,3-dione; SCHEMBL20120463; SCHEMBL29547130	CN1C2=CC=NC=C2C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4=CN=C(C#CCCCOC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C=C4)C3)C=C1)C=C2	C44H36N6O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-YKIZ6D	SCHEMBL20120806	2-(2,6-Dioxopiperidin-3-yl)-5-[5-[5-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]pentoxy]isoindole-1,3-dione; SCHEMBL20120808; SCHEMBL30302332	CN1C2=CC=NC=C2C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4=CN=C(CCCCCOC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C=C4)C3)C=C1)C=C2	C44H40N6O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-ZZQTPF	SCHEMBL20120227	2-(2,6-Dioxopiperidin-3-yl)-5-[4-[6-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxyhexyl]-3-(trifluoromethyl)piperazin-1-yl]isoindole-1,3-dione; SCHEMBL20129010; SCHEMBL29547580; WKHLDDPTXOBVSQ-LPOBGEIXSA-N; 2-(2,6-Dioxopiperidin-3-yl)-5-[4-[6-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxyhexyl]-3-(trifluoromethyl)piperazin-1-yl]isoindole-1,3-dione	CN1C2=CC=NC=C2C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OCCCCCCN4CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4C(F)(F)F)C3)C=C1)C=C2	C45H46F3N7O6	Tau	P10636	CRBN	WO-2018102067-A2
TPD-O85Z6A	SCHEMBL20120569	2-(2,6-Dioxopiperidin-3-yl)-5-[6-[5-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]hex-5-ynoxy]isoindole-1,3-dione; SCHEMBL20120570; SCHEMBL30302393	CN1C2=CC=NC=C2C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4=CN=C(C#CCCCCOC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C=C4)C3)C=C1)C=C2	C45H38N6O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-PUGLQT	SCHEMBL20120592	2-(2,6-Dioxopiperidin-3-yl)-5-[6-[5-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]hexoxy]isoindole-1,3-dione; SCHEMBL20129319; SCHEMBL29947972	CN1C2=CC=NC=C2C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4=CN=C(CCCCCCOC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C=C4)C3)C=C1)C=C2	C45H42N6O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-F6ER55	WO2018102067A2_99	.	O=C1CCC(N2C(=O)C3=C(C=C(OC4CN(CCCOCCCO[C@H]5C[C@H](OC6=NC=C(C7=CC8=C(C=C7)C7=C(C=CN=C7)N8)C=C6)C5)C4)C=C3)C2=O)C(=O)N1	C42H42N6O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-3ZCK2H	SCHEMBL20120316	2-(2,6-Dioxopiperidin-3-yl)-5-[6-[4-[4-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxybutoxy]butoxy]-2-azaspiro[3.3]heptan-2-yl]isoindole-1,3-dione; SCHEMBL29547916	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(OCCCCOCCCCOC3CC4(C3)CN(C3=CC5=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C5=O)C4)C=C1)C=C2	C44H46N6O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-0UILNJ	SCHEMBL20120797	2-(2,6-dioxopiperidin-3-yl)-5-[1-[3-[3-[3-[5-(5H-pyrido[4,3-b]indol-7-yl)-3-(trifluoromethyl)pyridin-2-yl]oxycyclobutyl]oxypropoxy]propyl]azetidin-3-yl]oxyisoindole-1,3-dione; SCHEMBL20120799; SCHEMBL29548032; PRODWFFGBOKDFC-LLQXBQLESA-N; 2-(2,6-dioxopiperidin-3-yl)-5-[1-[3-[3-[3-[5-(5H-pyrido[4,3-b]indol-7-yl)-3-(trifluoromethyl)pyridin-2-yl]oxycyclobutyl]oxypropoxy]propyl]azetidin-3-yl]oxyisoindole-1,3-dione	O=C1CCC(N2C(=O)C3=C(C=C(OC4CN(CCCOCCCO[C@H]5C[C@H](OC6=NC=C(C7=CC8=C(C=C7)C7=C(C=CN=C7)N8)C=C6C(F)(F)F)C5)C4)C=C3)C2=O)C(=O)N1	C43H41F3N6O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-3TAPDS	SCHEMBL20120244	2-(2,6-Dioxopiperidin-3-yl)-5-[6-[6-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridin-3-yl]hex-5-ynoxy]isoindole-1,3-dione; SCHEMBL20120246; SCHEMBL20120536; SCHEMBL29547416	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4=NC=C(C#CCCCCOC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C=C4)C3)C=C1)C=C2	C45H38N6O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-ZPE2M7	SCHEMBL20120253	5-[2-[2-[2-[2-[2-[5-(8,9-difluoro-5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]ethoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione; SCHEMBL29547626	O=C1CCC(N2C(=O)C3=C(C=C(OCCOCCOCCOCCOCCOC4=NC=C(C5=CC6=C(C7=CN=CC=C7N6)C(F)=C5F)C=C4)C=C3)C2=O)C(=O)N1	C39H37F2N5O10	Tau	P10636	CRBN	WO-2018102067-A2
TPD-OAUYSH	WO2018102067A2_104	.	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OCCCOCCCOC4CN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)C3)C=C1)C=C2	C43H44N6O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-PKQPVU	SCHEMBL20120446	2-(2,6-Dioxopiperidin-3-yl)-5-[1-[3-[3-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)-3-(trifluoromethyl)pyridin-2-yl]oxycyclobutyl]oxypropoxy]propyl]azetidin-3-yl]oxyisoindole-1,3-dione; SCHEMBL20120448; SCHEMBL30302320; LIFHTJVKOPKOBO-QZHRDHLUSA-N; 2-(2,6-Dioxopiperidin-3-yl)-5-[1-[3-[3-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)-3-(trifluoromethyl)pyridin-2-yl]oxycyclobutyl]oxypropoxy]propyl]azetidin-3-yl]oxyisoindole-1,3-dione	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OCCCOCCCN4CC(OC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)C3)C(C(F)(F)F)=C1)C=C2	C44H43F3N6O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-NVFIPD	SCHEMBL20120811	2-(2,6-Dioxopiperidin-3-yl)-5-[5-[5-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxyazetidin-1-yl]pentoxy]pentoxy]isoindole-1,3-dione	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(OC3CN(CCCCCOCCCCCOC4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)C=C1)C=C2	C43H46N6O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-VSDA0K	SCHEMBL20120281	2-(2,6-Dioxopiperidin-3-yl)-5-[4-[4-[6-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxy-2-azaspiro[3.3]heptan-2-yl]butoxy]butoxy]isoindole-1,3-dione; SCHEMBL29547791	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(OC3CC4(C3)CN(CCCCOCCCCOC3=CC5=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C5=O)C4)C=C1)C=C2	C44H46N6O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-DDRHHF	SCHEMBL20120595	2-(2,6-Dioxopiperidin-3-yl)-5-[6-[6-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]oxyhexoxy]isoindole-1,3-dione; SCHEMBL20120829; SCHEMBL20133147; SCHEMBL29547559	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4=CC=CC(OCCCCCCOC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)=N4)C3)C=C1)C=C2	C45H42N6O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-C3W7J8	WO2018102067A2_109	.	O=C1CCC(N2C(=O)C3=C(C=C(OCCCCCCOC4=CC(O[C@H]5C[C@H](OC6=NC=C(C7=CC8=C(C=C7)C7=C(C=CN=C7)N8)C=C6)C5)=CC=N4)C=C3)C2=O)C(=O)N1	C44H40N6O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-9HCWC3	WO2018102067A2_110	.	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4=NC=C(CCCCCCOC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C=C4)C3)C=C1)C=C2	C45H42N6O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-FG4SA5	WO2018102067A2_111	.	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4=CN=C(C#CCOC5CN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)C=C4)C3)C=C1)C=C2	C45H37N7O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-4WH6AR	SCHEMBL20120335	5-[2-[2-[2-[2-[2-[5-(8,9-Difluoro-5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]ethoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione; SCHEMBL29548478	CN1C2=CC=NC=C2C2=C1C=C(C1=CN=C(OCCOCCOCCOCCOCCOC3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C=C1)C(F)=C2F	C40H39F2N5O10	Tau	P10636	CRBN	WO-2018102067-A2
TPD-PPV1UY	SCHEMBL20120996	5-[2-[2-[2-[2-[2-[4-Chloro-5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]ethoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN1C2=CC(C3=CN=C(OCCOCCOCCOCCOCCOC4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)C=C3Cl)=CC=C2C2=C1C=CN=C2	C40H40ClN5O10	Tau	P10636	CRBN	WO-2018102067-A2
TPD-NNMGTN	SCHEMBL20120678	2-(2,6-Dioxopiperidin-3-yl)-5-[5-[4-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxybutoxy]pentoxy]isoindole-1,3-dione; SCHEMBL20120800; SCHEMBL29547702	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OCCCCOCCCCCOC4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)C=C1)C=C2	C43H45N5O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-JR6OD0	SCHEMBL20120368	2-(2,6-Dioxopiperidin-3-yl)-5-[5-[5-[1-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]azetidin-3-yl]oxypentoxy]pentoxy]isoindole-1,3-dione	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(N3CC(OCCCCCOCCCCCOC4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)C=C1)C=C2	C43H46N6O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-MWGE2M	SCHEMBL20120899	2-(2,6-Dioxopiperidin-3-yl)-5-[[2-[4-[4-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxybutoxy]butyl]-2-azaspiro[3.3]heptan-6-yl]oxy]isoindole-1,3-dione; SCHEMBL29548114	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(OCCCCOCCCCN3CC4(CC(OC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)C3)C=C1)C=C2	C44H46N6O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-SQRRAU	SCHEMBL20120276	2-(2,6-Dioxopiperidin-3-yl)-5-[3-[5-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]prop-2-ynoxy]isoindole-1,3-dione; SCHEMBL20120278; SCHEMBL29547875	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4=CN=C(C#CCOC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C=C4)C3)C=C1)C=C2	C42H32N6O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-4MK0OZ	SCHEMBL20120283	2-(2,6-Dioxopiperidin-3-yl)-5-[3-[3-[5-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)-3-(trifluoromethyl)pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]prop-2-ynoxy]azetidin-1-yl]isoindole-1,3-dione; SCHEMBL20120676; SCHEMBL30302403; UYSXLKVRGNQMCH-ZLAYGOEJSA-N; 2-(2,6-Dioxopiperidin-3-yl)-5-[3-[3-[5-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)-3-(trifluoromethyl)pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]prop-2-ynoxy]azetidin-1-yl]isoindole-1,3-dione	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4=CN=C(C#CCOC5CN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)C=C4)C3)C(C(F)(F)F)=C1)C=C2	C46H36F3N7O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-3IF61P	SCHEMBL20120475	(2S,4R)-1-[(2S)-3,3-dimethyl-2-[[2-[2-[2-[2-[2-[5-(5H-pyrido[4,3-b]indol-7-yl)-3-(trifluoromethyl)pyridin-2-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]butanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL29547623; XTNPWCQVYXFDQZ-XBUVSGBXSA-N; (2S,4R)-1-[(2S)-3,3-dimethyl-2-[[2-[2-[2-[2-[2-[5-(5H-pyrido[4,3-b]indol-7-yl)-3-(trifluoromethyl)pyridin-2-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]butanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOCCOC3=C(C(F)(F)F)C=C(C4=CC5=C(C=C4)C4=C(C=CN=C4)N5)C=N3)C(C)(C)C)C=C2)SC=N1	C50H58F3N7O9S	Tau	P10636	VHL	WO-2018102067-A2
TPD-FNLK21	WO2018102067A2_120	.	CC1=C(C2=CC=C([C@H](C)NC(=O)C3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOC3=CC=C(C4=CC5=C(C=C4)C4=C(C=CN=C4)N5)C=N3)C(C)(C)C)C=C2)SC=N1	C43H47N7O6S	Tau	P10636	VHL	WO-2018102067-A2
TPD-P3NRYY	SCHEMBL20120352	(2S,4R)-1-[(2S)-3,3-dimethyl-2-[[2-[2-[2-[2-[2-[2-[5-(5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]butanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL29547326	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOCCOCCOC3=CC=C(C4=CC5=C(C=C4)C4=C(C=CN=C4)N5)C=N3)C(C)(C)C)C=C2)SC=N1	C51H63N7O10S	Tau	P10636	VHL	WO-2018102067-A2
TPD-D1CR94	SCHEMBL20120464	(2S,4R)-1-[(2S)-3,3-dimethyl-2-[[2-[2-[2-[2-[2-[2-[2-[5-(5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]butanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOCCOCCOCCOC3=CC=C(C4=CC5=C(C=C4)C4=C(C=CN=C4)N5)C=N3)C(C)(C)C)C=C2)SC=N1	C53H67N7O11S	Tau	P10636	VHL	WO-2018102067-A2
TPD-XBD7ME	SCHEMBL20120551	2-(2,6-Dioxopiperidin-3-yl)-5-[5-[4-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)-3-(trifluoromethyl)pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]pentoxy]isoindole-1,3-dione; SCHEMBL20120553; SCHEMBL30302421; ORJNCUXRGKWLBW-LYTIDBDVSA-N; 2-(2,6-Dioxopiperidin-3-yl)-5-[5-[4-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)-3-(trifluoromethyl)pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]pentoxy]isoindole-1,3-dione	CN1C2=CC=NC=C2C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4CCN(CCCCCOC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C3)C(C(F)(F)F)=C1)C=C2	C45H45F3N6O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-A6PARC	WO2018102067A2_124	.	CN1C2=CC=NC=C2C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4=CC=C(C#CCCCCOC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C=C4)C3)C(C(F)(F)F)=C1)C=C2	C47H38F3N5O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-MGPBBL	SCHEMBL20120606	2-(2,6-Dioxopiperidin-3-yl)-5-[3-[3-[3-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)-3-(trifluoromethyl)pyridin-2-yl]oxycyclobutyl]oxypropoxy]propoxy]azetidin-1-yl]isoindole-1,3-dione; SCHEMBL20120614; SCHEMBL30302311; ZQBPRKYUJWSJTN-QZHRDHLUSA-N; 2-(2,6-Dioxopiperidin-3-yl)-5-[3-[3-[3-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)-3-(trifluoromethyl)pyridin-2-yl]oxycyclobutyl]oxypropoxy]propoxy]azetidin-1-yl]isoindole-1,3-dione	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OCCCOCCCOC4CN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)C3)C(C(F)(F)F)=C1)C=C2	C44H43F3N6O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-S30715	SCHEMBL20120341	2-(2,6-Dioxopiperidin-3-yl)-5-[5-[6-[methyl-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]amino]-2-azaspiro[3.3]heptan-2-yl]pentoxy]isoindole-1,3-dione; SCHEMBL20120344; SCHEMBL29547677	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](N(C)C4CC5(C4)CN(CCCCCOC4=CC6=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)C5)C3)C=C1)C=C2	C46H49N7O6	Tau	P10636	CRBN	WO-2018102067-A2
TPD-M7OYXZ	SCHEMBL20120761	3-[6-[4-[[1-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL29547589	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(N3CCC(CN4CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6)CC4)CC3)C=C1)C=C2	C40H42N8O3	Tau	P10636	CRBN	WO-2018102067-A2
TPD-W3KE5F	SCHEMBL20121031	3-[6-[4-[2-[1-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]piperidin-4-yl]ethyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL29548020	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(N3CCC(CCN4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)CC6=C5)CC4)CC3)C=C1)C=C2	C41H44N8O3	Tau	P10636	CRBN	WO-2018102067-A2
TPD-4T4OY4	SCHEMBL20120620	2-(2,6-Dioxopiperidin-3-yl)-5-[1,1,1-trifluoro-6-[2-[2-[2-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxyethoxy]ethoxy]ethoxy]hexan-2-yl]oxyisoindole-1,3-dione; SCHEMBL29547796; GMYLDLZGPLXPDB-UHFFFAOYSA-N; 2-(2,6-Dioxopiperidin-3-yl)-5-[1,1,1-trifluoro-6-[2-[2-[2-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxyethoxy]ethoxy]ethoxy]hexan-2-yl]oxyisoindole-1,3-dione	CN1C2=CC=NC=C2C2=C1C=C(C1=CN=C(OCCOCCOCCOCCCCC(OC3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C(F)(F)F)C=C1)C=C2	C42H42F3N5O9	Tau	P10636	CRBN	WO-2018102067-A2
TPD-0TMDLB	WO2018102067A2_130	.	O=C1CCC(N2C(=O)C3=C(C=C(N4CC(OCCCOCCCN5CCC(OC6=NC=C(C7=CC8=C(C=C7)C7=C(C=CN=C7)N8)C=C6CF)CC5)C4)C=C3)C2=O)C(=O)N1	C44H46FN7O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-8H18F2	SCHEMBL20120846	2-(2,6-Dioxopiperidin-3-yl)-5-[2-[2-[2-[2-[2-[2-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]isoindole-1,3-dione; SCHEMBL29547458	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CC=C(OCCOCCOCCOCCOCCOCCOC3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4=O)N=C1)C=C2	C42H45N5O11	Tau	P10636	CRBN	WO-2018102067-A2
TPD-CJ5N5B	WO2018102067A2_132	.	O=C1CCC(N2C(=O)C3=C(C=C(OCCOCCOCCOCCOCCOCCOCCOC4=CC=C(C5=CC6=C(C=C5)C5=C(C=CN=C5)N6)C=N4)C=C3)C2=O)C(=O)N1	C43H47N5O12	Tau	P10636	CRBN	WO-2018102067-A2
TPD-ZUEZIE	SCHEMBL20120780	2-(2,6-Dioxopiperidin-3-yl)-5-[3-[6-[5-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxypentoxy]hexyl]azetidin-1-yl]isoindole-1,3-dione; SCHEMBL29547692	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(OCCCCCOCCCCCCC3CN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)C=C1)C=C2	C44H48N6O6	Tau	P10636	CRBN	WO-2018102067-A2
TPD-9PEZZ2	SCHEMBL20120265	2-(2,6-Dioxopiperidin-3-yl)-5-[6-[6-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridazin-3-yl]hex-5-ynoxy]isoindole-1,3-dione; SCHEMBL20120268; SCHEMBL29547286	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4=NN=C(C#CCCCCOC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C=C4)C3)C=C1)C=C2	C44H37N7O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-DYD6RB	SCHEMBL20120305	2-(2,6-Dioxopiperidin-3-yl)-5-[4-[[2-[[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]methyl]-2-azaspiro[3.3]heptan-6-yl]oxy]butoxy]isoindole-1,3-dione; SCHEMBL20121016; SCHEMBL29547688	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](CN4CC5(CC(OCCCCOC6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)C4)C3)C=C1)C=C2	C45H46N6O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-WRITSA	SCHEMBL20120346	2-(2,6-Dioxopiperidin-3-yl)-5-[4-[[2-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutanecarbonyl]-2-azaspiro[3.3]heptan-6-yl]oxy]butoxy]isoindole-1,3-dione; SCHEMBL20120417; SCHEMBL20120674; SCHEMBL29547711	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@@H](C(=O)N4CC5(CC(OCCCCOC6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)C4)C3)C=C1)C=C2	C45H44N6O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-F1PCHV	SCHEMBL20120370	2-(2,6-Dioxopiperidin-3-yl)-5-[5-[6-[methyl-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]amino]-2-azaspiro[3.3]heptan-2-yl]-5-oxopentoxy]isoindole-1,3-dione; SCHEMBL20120372; SCHEMBL29547902	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](N(C)C4CC5(C4)CN(C(=O)CCCCOC4=CC6=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)C5)C3)C=C1)C=C2	C46H47N7O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-00OJ37	SCHEMBL20120345	5-[2-[2-[2-[2-[2-[5-[5-(Difluoromethyl)pyrido[4,3-b]indol-7-yl]pyridin-2-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]ethoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione; SCHEMBL29547618; OEKOSNJRSUQVFE-UHFFFAOYSA-N; 5-[2-[2-[2-[2-[2-[5-[5-(Difluoromethyl)pyrido[4,3-b]indol-7-yl]pyridin-2-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]ethoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=C(C=C(OCCOCCOCCOCCOCCOC4=CC=C(C5=CC6=C(C=C5)C5=C(C=CN=C5)N6C(F)F)C=N4)C=C3)C2=O)C(=O)N1	C40H39F2N5O10	Tau	P10636	CRBN	WO-2018102067-A2
TPD-H17ZE0	SCHEMBL20120250	2-(2,6-Dioxopiperidin-3-yl)-5-[2-[2-[2-[2-[2-[3-fluoro-5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]ethoxy]isoindole-1,3-dione; SCHEMBL29548055	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CC(F)=C(OCCOCCOCCOCCOCCOC3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4=O)N=C1)C=C2	C40H40FN5O10	Tau	P10636	CRBN	WO-2018102067-A2
TPD-9FCDF5	SCHEMBL20120964	2-(2,6-Dioxopiperidin-3-yl)-5-[2-[2-[2-[2-[2-[3-methyl-5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]ethoxy]isoindole-1,3-dione; SCHEMBL29547165	CC1=C(OCCOCCOCCOCCOCCOC2=CC3=C(C=C2)C(=O)N(C2CCC(=O)NC2=O)C3=O)N=CC(C2=CC3=C(C=C2)C2=C(C=CN=C2)N3C)=C1	C41H43N5O10	Tau	P10636	CRBN	WO-2018102067-A2
TPD-UDHPNB	SCHEMBL20120457	2-(2,6-Dioxopiperidin-3-yl)-5-[6-[5-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyrimidin-2-yl]hex-5-ynoxy]isoindole-1,3-dione; SCHEMBL20120974; SCHEMBL29547806	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4=CN=C(C#CCCCCOC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)N=C4)C3)C=C1)C=C2	C44H37N7O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-YNHJGS	SCHEMBL20120458	2-(2,6-Dioxopiperidin-3-yl)-5-[1-[3-[5-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)-3-(trifluoromethyl)pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]prop-2-ynyl]azetidin-3-yl]oxyisoindole-1,3-dione; SCHEMBL20120460; SCHEMBL30302391; STZPPLPCCRXOSE-ZLAYGOEJSA-N; 2-(2,6-Dioxopiperidin-3-yl)-5-[1-[3-[5-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)-3-(trifluoromethyl)pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]prop-2-ynyl]azetidin-3-yl]oxyisoindole-1,3-dione	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4=CN=C(C#CCN5CC(OC6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)C=C4)C3)C(C(F)(F)F)=C1)C=C2	C46H36F3N7O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-PMDZQR	SCHEMBL20120271	2-(2,6-Dioxopiperidin-3-yl)-5-[2-[2-[2-[2-[2-[5-(5-methylpyrido[4,3-b]indol-7-yl)-6-(trifluoromethyl)pyridin-2-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]ethoxy]isoindole-1,3-dione; SCHEMBL29547663; WHAYHTAQIWTMSP-UHFFFAOYSA-N; 2-(2,6-Dioxopiperidin-3-yl)-5-[2-[2-[2-[2-[2-[5-(5-methylpyrido[4,3-b]indol-7-yl)-6-(trifluoromethyl)pyridin-2-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]ethoxy]isoindole-1,3-dione	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CC=C(OCCOCCOCCOCCOCCOC3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4=O)N=C1C(F)(F)F)C=C2	C41H40F3N5O10	Tau	P10636	CRBN	WO-2018102067-A2
TPD-SP195U	WO2018102067A2_144	.	O=C1CCC(N2C(=O)C3=C(C=C(OCCCCC#CC4=CN=C(O[C@H]5C[C@@H](OC6=NC=C(C7=CC8=C(C=C7)C7=C(C=CN=C7)N8)C=C6)C5)C=C4)C=C3)C2=O)C(=O)N1	C44H36N6O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-EVH84I	WO2018102067A2_145	.	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@@H](OC4=NC=C(CCCCCCOC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C=C4)C3)C=C1)C=C2	C45H42N6O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-2UTCTU	SCHEMBL20120885	2-(2,6-Dioxopiperidin-3-yl)-5-[6-[6-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxypropoxy]pyridin-3-yl]hex-5-ynoxy]isoindole-1,3-dione; SCHEMBL29547871	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CC=C(OCCCOC3=NC=C(C#CCCCCOC4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C=C3)N=C1)C=C2	C44H38N6O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-V966KP	WO2018102067A2_147	.	O=C1CCC(N2C(=O)C3=C(C=C(OCCCCCCC4=CC=C(O[C@H]5C[C@H](OC6=NC=C(C7=CC8=C(C=C7)C7=CN=CC=C7N8)C=C6)C5)C=C4)C=C3)C2=O)C(=O)N1	C45H41N5O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-55AB1F	SCHEMBL20120691	2-(2,6-dioxopiperidin-3-yl)-5-[3-[3-[3-[3-[5-(5H-pyrido[4,3-b]indol-7-yl)-3-(trifluoromethyl)pyridin-2-yl]oxycyclobutyl]oxypropoxy]propoxy]azetidin-1-yl]isoindole-1,3-dione; SCHEMBL20120693; SCHEMBL29547610	O=C1CCC(N2C(=O)C3=C(C=C(N4CC(OCCCOCCCO[C@H]5C[C@H](OC6=NC=C(C7=CC8=C(C=C7)C7=C(C=CN=C7)N8)C=C6C(F)(F)F)C5)C4)C=C3)C2=O)C(=O)N1	C43H41F3N6O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-9AOOO4	WO2018102067A2_149	.	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4=NN=C(CCCCCCOC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6O)C=C4)C3)C=C1)C=C2	C44H43N7O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-P4B9EN	SCHEMBL20120331	5-[6-[2,2-Difluoro-5-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypentyl]-2,6-diazaspiro[3.3]heptan-2-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione; SCHEMBL20120333; SCHEMBL29548033; IUTLZLUVOPGGIP-UHFFFAOYSA-N; 5-[6-[2,2-Difluoro-5-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypentyl]-2,6-diazaspiro[3.3]heptan-2-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN1C2=CC=NC=C2C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OCCCC(F)(F)CN4CC5(C4)CN(C4=CC6=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)C5)C3)C=C1)C=C2	C44H43F2N7O6	Tau	P10636	CRBN	WO-2018102067-A2
TPD-T8NJ8F	SCHEMBL20120413	2-(2,6-Dioxopiperidin-3-yl)-5-[6-[5-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyrimidin-2-yl]hexoxy]isoindole-1,3-dione; SCHEMBL20120415; SCHEMBL30302404	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4=CN=C(CCCCCCOC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)N=C4)C3)C=C1)C=C2	C44H41N7O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-13LFPZ	SCHEMBL20121037	2-(2,6-Dioxopiperidin-3-yl)-5-[1-[3-[5-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]prop-2-ynyl]azetidin-3-yl]oxyisoindole-1,3-dione; SCHEMBL20121038; SCHEMBL30302354	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4=CN=C(C#CCN5CC(OC6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)C=C4)C3)C=C1)C=C2	C45H37N7O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-VEOHZH	SCHEMBL20120759	2-(2,6-Dioxopiperidin-3-yl)-5-[3-[3,3,3-trifluoro-2-[5-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypentoxy]propyl]azetidin-1-yl]isoindole-1,3-dione; SCHEMBL20120760; SCHEMBL29547680; NQLCEHYWANNIKZ-LPOBGEIXSA-N; 2-(2,6-Dioxopiperidin-3-yl)-5-[3-[3,3,3-trifluoro-2-[5-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypentoxy]propyl]azetidin-1-yl]isoindole-1,3-dione	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OCCCCCOC(CC4CN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)C(F)(F)F)C3)C=C1)C=C2	C45H45F3N6O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-HLX1H6	SCHEMBL20120905	2-(2,6-Dioxopiperidin-3-yl)-5-[3-[2,2,2-trifluoro-1-[6-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxyhexoxy]ethyl]azetidin-1-yl]isoindole-1,3-dione; SCHEMBL20120908; SCHEMBL30302306	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OCCCCCCOC(C4CN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)C(F)(F)F)C3)C=C1)C=C2	C45H45F3N6O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-X7ZBMW	SCHEMBL20120248	2-(2,6-Dioxopiperidin-3-yl)-5-[3-[5-[2-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxyethoxy]pyridin-2-yl]oxyazetidin-1-yl]isoindole-1,3-dione; SCHEMBL20120249; SCHEMBL30302362	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OCCOC4=CN=C(OC5CN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)C=C4)C3)C=C1)C=C2	C44H39N7O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-4892BO	WO2018102067A2_156	.	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4=CN=C(CCCOC5CN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)C=C4)C3)C=C1)C=C2	C45H41N7O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-OVOQM5	WO2018102067A2_157	.	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](C(=O)C4CC5(CC(OCCCCOC6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)C4)C3)C=C1)C=C2	C46H45N5O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-ZNZB31	SCHEMBL20120401	2-(2,6-Dioxopiperidin-3-yl)-5-[2-[6-[4-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]pyridazin-4-yl]oxyethoxy]isoindole-1,3-dione; SCHEMBL20120402; SCHEMBL29547271	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4CCN(C5=NN=CC(OCCOC6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)=C5)CC4)C3)C=C1)C=C2	C45H42N8O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-0YD1GV	WO2018102067A2_159	.	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@@H](OC4=CN=C(C#CCOC5CN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)C=C4)C3)C=C1)C=C2	C45H37N7O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-I6VTPA	WO2018102067A2_160	.	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@@H](OC4=CN=C(CCCOC5CN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)C=C4)C3)C=C1)C=C2	C45H41N7O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-V4BYKO	SCHEMBL20120284	2-(2,6-Dioxopiperidin-3-yl)-5-[3-[2-[2-[2-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxyethoxy]ethoxy]ethoxy]azetidin-1-yl]isoindole-1,3-dione; SCHEMBL20120285; SCHEMBL29547151	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OCCOCCOCCOC4CN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)C3)C=C1)C=C2	C43H44N6O9	Tau	P10636	CRBN	WO-2018102067-A2
TPD-0A7OPZ	SCHEMBL20120750	2-(2,6-Dioxopiperidin-3-yl)-5-[3-[4-[4-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxybutoxy]butoxy]azetidin-1-yl]isoindole-1,3-dione; SCHEMBL20120752; SCHEMBL30302299	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OCCCCOCCCCOC4CN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)C3)C=C1)C=C2	C45H48N6O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-ZLGVSF	SCHEMBL20120889	2-(2,6-Dioxopiperidin-3-yl)-5-[3-[2-[2-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxyethoxy]ethoxy]azetidin-1-yl]isoindole-1,3-dione; SCHEMBL20120891; SCHEMBL30302376	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OCCOCCOC4CN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)C3)C=C1)C=C2	C41H40N6O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-80P4XB	SCHEMBL20120538	2-(2,6-dioxopiperidin-3-yl)-5-[6-oxo-6-[4-[3-[5-(5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]hexoxy]isoindole-1,3-dione; SCHEMBL20120539; SCHEMBL29547780	O=C1CCC(N2C(=O)C3=C(C=C(OCCCCCC(=O)N4CCC(O[C@H]5C[C@H](OC6=NC=C(C7=CC8=C(C=C7)C7=C(C=CN=C7)N8)C=C6)C5)CC4)C=C3)C2=O)C(=O)N1	C44H44N6O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-5TYPZD	WO2018102067A2_165	.	O=C1CCC(N2C(=O)C3=C(C=C(OCCCCCOC4CCN(C(=O)[C@H]5C[C@H](OC6=NC=C(C7=CC8=C(C=C7)C7=C(C=CN=C7)N8)C=C6)C5)CC4)C=C3)C2=O)C(=O)N1	C44H44N6O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-L6TM0O	WO2018102067A2_166	.	O=C1CCC(N2C(=O)C3=C(C=C(OCCCCCOC4CCN(C(=O)[C@H]5C[C@@H](OC6=NC=C(C7=CC8=C(C=C7)C7=C(C=CN=C7)N8)C=C6)C5)CC4)C=C3)C2=O)C(=O)N1	C44H44N6O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-GP8W5I	SCHEMBL20120650	2-(2,6-Dioxopiperidin-3-yl)-5-[3-[3-[5-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxypropoxy]pyridin-2-yl]prop-2-ynoxy]azetidin-1-yl]isoindole-1,3-dione; SCHEMBL29547685	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(OCCCOC3=CN=C(C#CCOC4CN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)C=C3)C=C1)C=C2	C44H37N7O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-KGTEQY	SCHEMBL20120478	2-(2,6-Dioxopiperidin-3-yl)-5-[3-[3-[5-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxypropoxy]pyridin-2-yl]propoxy]azetidin-1-yl]isoindole-1,3-dione; SCHEMBL29548193	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(OCCCOC3=CN=C(CCCOC4CN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)C=C3)C=C1)C=C2	C44H41N7O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-IUC7PT	SCHEMBL20120356	2-(2,6-Dioxopiperidin-3-yl)-5-[3-[3-[[3-[[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxymethyl]oxetan-3-yl]methoxy]propoxy]azetidin-1-yl]isoindole-1,3-dione; SCHEMBL20120357; SCHEMBL29547344	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OCC4(COCCCOC5CN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)COC4)C3)C=C1)C=C2	C45H46N6O9	Tau	P10636	CRBN	WO-2018102067-A2
TPD-QWO9W8	WO2018102067A2_170	.	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@@H](OCCCOCCCOC4CN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)C3)C=C1)C=C2	C43H44N6O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-ZI4GRV	SCHEMBL20120375	5-[4,4-Difluoro-5-[4-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]pentoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione; 5-[4,4-Difluoro-5-[4-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]pentoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione; SCHEMBL20120377; SCHEMBL29547283; WDTQFLYQEJTPKI-JZSUORBJSA-N; WDTQFLYQEJTPKI-UHFFFAOYSA-N	CN1C2=CC=NC=C2C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4CCN(CC(F)(F)CCCOC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C3)C=C1)C=C2	C44H44F2N6O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-CT769C	SCHEMBL20120860	2-(2,6-dioxopiperidin-3-yl)-5-[6-[5-[3-[5-(5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]hex-5-ynoxy]isoindole-1,3-dione; SCHEMBL20120861; SCHEMBL30302345	O=C1CCC(N2C(=O)C3=C(C=C(OCCCCC#CC4=NC=C(O[C@H]5C[C@H](OC6=NC=C(C7=CC8=C(C=C7)C7=C(C=CN=C7)N8)C=C6)C5)C=C4)C=C3)C2=O)C(=O)N1	C44H36N6O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-8SX701	SCHEMBL20120665	2-(2,6-dioxopiperidin-3-yl)-5-[2-[3-[5-[3-[5-(5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]prop-2-ynoxy]ethoxy]isoindole-1,3-dione; SCHEMBL20120666; SCHEMBL29547643	O=C1CCC(N2C(=O)C3=C(C=C(OCCOCC#CC4=NC=C(O[C@H]5C[C@H](OC6=NC=C(C7=CC8=C(C=C7)C7=C(C=CN=C7)N8)C=C6)C5)C=C4)C=C3)C2=O)C(=O)N1	C43H34N6O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-POE8XA	WO2018102067A2_174	.	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OCC4(CCOCCCCOC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CCC4)C3)C=C1)C=C2	C45H47N5O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-PRHP0S	WO2018102067A2_175	.	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(OC3CN(C(=O)C4(CCOCCCCCOC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CCC4)C3)C=C1)C=C2	C45H46N6O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-BWE32T	SCHEMBL20120273	5-[3-[3-[3-[3-[5-(8,9-Difluoro-5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypropoxy]propoxy]azetidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione; SCHEMBL20120274; SCHEMBL29547238	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OCCCOCCCOC4CN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)C3)C=C1)C(F)=C2F	C43H42F2N6O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-CJSFK7	SCHEMBL20120932	3-[6-[3-[3-[3-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypropoxy]propoxy]azetidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL20120934; SCHEMBL29547361	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OCCCOCCCOC4CN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6)C4)C3)C=C1)C=C2	C43H46N6O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-BPXQHS	SCHEMBL20120484	2-(2,6-Dioxopiperidin-3-yl)-5-[3-[6-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxyhexoxymethyl]azetidin-1-yl]isoindole-1,3-dione; SCHEMBL20120488; SCHEMBL30302408	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OCCCCCCOCC4CN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)C3)C=C1)C=C2	C44H46N6O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-NVOQL2	SCHEMBL20120495	2-(2,6-Dioxopiperidin-3-yl)-5-[2-[3-[5-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]prop-2-ynoxy]ethoxy]isoindole-1,3-dione; SCHEMBL20120496; SCHEMBL30302305	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4=CN=C(C#CCOCCOC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C=C4)C3)C=C1)C=C2	C44H36N6O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-0YL3QV	SCHEMBL20120969	3-[3-oxo-6-[3-[5-[3-[5-(5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]prop-2-ynoxy]-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL20120971; SCHEMBL29547727	O=C1CCC(N2CC3=C(C=CC(OCC#CC4=NC=C(O[C@H]5C[C@H](OC6=NC=C(C7=CC8=C(C=C7)C7=C(C=CN=C7)N8)C=C6)C5)C=C4)=C3)C2=O)C(=O)N1	C41H32N6O6	Tau	P10636	CRBN	WO-2018102067-A2
TPD-LXQ3YW	SCHEMBL20120604	2-(2,6-Dioxopiperidin-3-yl)-5-[3-[2-[5-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypentoxy]ethyl]azetidin-1-yl]isoindole-1,3-dione; SCHEMBL20120605; SCHEMBL30302377	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OCCCCCOCCC4CN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)C3)C=C1)C=C2	C44H46N6O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-W25SLS	SCHEMBL20120625	2-(2,6-dioxopiperidin-3-yl)-5-[3-[3-[3-[3-[5-(5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypropoxy]propoxy]azetidin-1-yl]isoindole-1,3-dione; SCHEMBL20120626; SCHEMBL30302396	O=C1CCC(N2C(=O)C3=C(C=C(N4CC(OCCCOCCCO[C@H]5C[C@H](OC6=NC=C(C7=CC8=C(C=C7)C7=C(C=CN=C7)N8)C=C6)C5)C4)C=C3)C2=O)C(=O)N1	C42H42N6O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-QTW6ST	WO2018102067A2_183	.	O=C1CCC(N2C(=O)C3=C(C=C(OCC#CC4=NC=C(O[C@H]5C[C@@H](OC6=NC=C(C7=CC8=C(C=C7)C7=C(C=CN=C7)N8)C=C6)C5)C=C4)C=C3)C2=O)C(=O)N1	C41H30N6O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-9ET03F	WO2018102067A2_184	.	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(OC3CN(C(=O)C4(CCCCCCCCOC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CCC4)C3)C=C1)C=C2	C46H48N6O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-TEB6YD	SCHEMBL20120576	(2S,4R)-4-hydroxy-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]-N-[[4-(4-methyl-1,3-thiazol-5-yl)-2-[2-[5-(5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxyethoxy]phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL29547696	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C(OCCOC3=NC=C(C4=CC5=C(C=C4)C4=C(C=CN=C4)N5)C=C3)=C2)SC=N1	C47H45N7O6S	Tau	P10636	VHL	WO-2018102067-A2
TPD-1Z45DE	SCHEMBL20120937	(2S,4R)-4-hydroxy-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]-N-[[4-(4-methyl-1,3-thiazol-5-yl)-2-[2-[2-[5-(5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxyethoxy]ethoxy]phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C(OCCOCCOC3=NC=C(C4=CC5=C(C=C4)C4=C(C=CN=C4)N5)C=C3)=C2)SC=N1	C49H49N7O7S	Tau	P10636	VHL	WO-2018102067-A2
TPD-FASD1Z	SCHEMBL20120378	(2S,4R)-4-hydroxy-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]-N-[[4-(4-methyl-1,3-thiazol-5-yl)-2-[2-[2-[2-[5-(5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxyethoxy]ethoxy]ethoxy]phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C(OCCOCCOCCOC3=NC=C(C4=CC5=C(C=C4)C4=C(C=CN=C4)N5)C=C3)=C2)SC=N1	C51H53N7O8S	Tau	P10636	VHL	WO-2018102067-A2
TPD-QPLIC5	SCHEMBL20120254	2-(2,6-dioxopiperidin-3-yl)-5-[2-[3-[4-[3-[5-(5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxyphenyl]prop-2-ynoxy]ethoxy]isoindole-1,3-dione; SCHEMBL20129322; SCHEMBL29947991	O=C1CCC(N2C(=O)C3=C(C=C(OCCOCC#CC4=CC=C(O[C@H]5C[C@H](OC6=NC=C(C7=CC8=C(C=C7)C7=C(C=CN=C7)N8)C=C6)C5)C=C4)C=C3)C2=O)C(=O)N1	C44H35N5O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-ICY4Y4	SCHEMBL20120768	2-(2,6-dioxopiperidin-3-yl)-5-[3-[4-[3-[5-(5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxyphenyl]prop-2-ynoxy]isoindole-1,3-dione; SCHEMBL20120770; SCHEMBL30302416	O=C1CCC(N2C(=O)C3=C(C=C(OCC#CC4=CC=C(O[C@H]5C[C@H](OC6=NC=C(C7=CC8=C(C=C7)C7=C(C=CN=C7)N8)C=C6)C5)C=C4)C=C3)C2=O)C(=O)N1	C42H31N5O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-PNW0RK	SCHEMBL20121018	2-(2,6-Dioxopiperidin-3-yl)-5-[3-[2-[2-[2-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxyethoxy]ethoxy]ethyl]azetidin-1-yl]isoindole-1,3-dione; SCHEMBL20121020; SCHEMBL30302295	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OCCOCCOCCC4CN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)C3)C=C1)C=C2	C43H44N6O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-NUNW60	SCHEMBL20120742	2-(2,6-Dioxopiperidin-3-yl)-5-[3-[3-[2-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxyethoxy]propoxymethyl]azetidin-1-yl]isoindole-1,3-dione; SCHEMBL20120743; SCHEMBL30302406	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OCCOCCCOCC4CN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)C3)C=C1)C=C2	C43H44N6O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-WTR0CK	SCHEMBL20120868	2-(2,6-Dioxopiperidin-3-yl)-5-[3-[2-[2-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxyethoxy]ethoxymethyl]azetidin-1-yl]isoindole-1,3-dione; SCHEMBL20120870; SCHEMBL30302381	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OCCOCCOCC4CN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)C3)C=C1)C=C2	C42H42N6O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-9RSZ0K	SCHEMBL20120694	2-(2,6-Dioxopiperidin-3-yl)-5-[3-[3-[2-[6-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxy-2-azaspiro[3.3]heptan-2-yl]-2-oxoethoxy]propoxy]azetidin-1-yl]isoindole-1,3-dione	CN1C2=CC=NC=C2C2=C1C=C(C1=CN=C(OC3CC4(C3)CN(C(=O)COCCCOC3CN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C3)C4)C=C1)C=C2	C44H43N7O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-5O9UE5	SCHEMBL20120710	2-(2,6-dioxopiperidin-3-yl)-5-[3-[3-[5-[3-[5-(5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]prop-2-ynoxy]azetidin-1-yl]isoindole-1,3-dione; SCHEMBL20120712; SCHEMBL30302327	O=C1CCC(N2C(=O)C3=C(C=C(N4CC(OCC#CC5=NC=C(O[C@H]6C[C@H](OC7=NC=C(C8=CC9=C(C=C8)C8=C(C=CN=C8)N9)C=C7)C6)C=C5)C4)C=C3)C2=O)C(=O)N1	C44H35N7O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-02NQT0	SCHEMBL20120824	5-[2-[2-[2-[2-[2-[5-(4-Chloro-5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]ethoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione; SCHEMBL29547914	CN1C2=C(C=CC(C3=CC=C(OCCOCCOCCOCCOCCOC4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)N=C3)=C2)C2=C1C(Cl)=CN=C2	C40H40ClN5O10	Tau	P10636	CRBN	WO-2018102067-A2
TPD-KE5UHS	SCHEMBL20120726	(2S,4R)-4-hydroxy-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]-N-[[4-(4-methyl-1,3-thiazol-5-yl)-2-[2-[2-[2-[2-[5-(5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C(OCCOCCOCCOCCOC3=NC=C(C4=CC5=C(C=C4)C4=C(C=CN=C4)N5)C=C3)=C2)SC=N1	C53H57N7O9S	Tau	P10636	VHL	WO-2018102067-A2
TPD-NTJ7LX	SCHEMBL20120236	5-[6-[2,2-Difluoro-5-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypentoxy]-2-azaspiro[3.3]heptan-2-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione; SCHEMBL20120238; SCHEMBL29547535	CN1C2=CC=NC=C2C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OCCCC(F)(F)COC4CC5(C4)CN(C4=CC6=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)C5)C3)C=C1)C=C2	C45H44F2N6O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-FA6MM1	SCHEMBL20120426	2-(2,6-Dioxopiperidin-3-yl)-5-[3-[3-[4-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]phenyl]prop-2-ynoxy]isoindole-1,3-dione; SCHEMBL20120427; SCHEMBL30302325	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4CCN(C5=CC=CC(C#CCOC6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)=C5)CC4)C3)C=C1)C=C2	C48H42N6O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-X4OAQT	WO2018102067A2_199	.	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](N(C)C(=O)C4(CCOCCCCOC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CCC4)C3)C=C1)C=C2	C46H48N6O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-4CENZA	SCHEMBL20120790	2-(2,6-Dioxopiperidin-3-yl)-5-[3-[7-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxyheptoxy]azetidin-1-yl]isoindole-1,3-dione; SCHEMBL20120792; SCHEMBL30302414	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OCCCCCCCOC4CN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)C3)C=C1)C=C2	C44H46N6O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-S3JG04	SCHEMBL20120598	(2S,4R)-4-hydroxy-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]-N-[[4-(4-methyl-1,3-thiazol-5-yl)-2-[2-[2-[2-[2-[2-[5-(5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]ethoxy]phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C(OCCOCCOCCOCCOCCOC3=NC=C(C4=CC5=C(C=C4)C4=C(C=CN=C4)N5)C=C3)=C2)SC=N1	C55H61N7O10S	Tau	P10636	VHL	WO-2018102067-A2
TPD-EMB6FF	SCHEMBL20120695	2-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]methoxy]-N-methyl-N-[3-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypropyl]acetamide; SCHEMBL20120697; SCHEMBL29547774	CN(CCCO[C@H]1C[C@H](OC2=NC=C(C3=CC4=C(C=C3)C3=C(C=CN=C3)N4C)C=C2)C1)C(=O)COCC1CN(C2=CC3=C(C=C2)C(=O)N(C2CCC(=O)NC2=O)C3=O)C1	C44H45N7O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-TQ4781	SCHEMBL20120226	2-[2-[2-[2-[2-[2-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]ethoxy]-5-(5-methylpyrido[4,3-b]indol-7-yl)pyridine-3-carbonitrile; SCHEMBL29547289	CN1C2=CC=NC=C2C2=C1C=C(C1=CC(C#N)=C(OCCOCCOCCOCCOCCOC3=CC=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)N=C1)C=C2	C41H40N6O10	Tau	P10636	CRBN	WO-2018102067-A2
TPD-GNMH2Z	SCHEMBL20120526	5-[3-[5-[3-[5-(8,9-difluoro-5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]prop-2-ynoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione; SCHEMBL20120529; SCHEMBL30302321	O=C1CCC(N2C(=O)C3=C(C=C(OCC#CC4=NC=C(O[C@H]5C[C@H](OC6=NC=C(C7=CC8=C(C(F)=C7F)C7=C(C=CN=C7)N8)C=C6)C5)C=C4)C=C3)C2=O)C(=O)N1	C41H28F2N6O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-VWGQZN	SCHEMBL20120527	2-(2,6-Dioxopiperidin-3-yl)-5-[3-[3-[4-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]phenyl]propoxy]isoindole-1,3-dione; SCHEMBL20120828; SCHEMBL30302330	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4CCN(C5=CC=CC(CCCOC6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)=C5)CC4)C3)C=C1)C=C2	C48H46N6O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-8EDU9U	SCHEMBL20120559	2-(2,6-Dioxopiperidin-3-yl)-5-[3-[2-[2-[2-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxyethoxy]ethoxy]ethoxymethyl]azetidin-1-yl]isoindole-1,3-dione; SCHEMBL20120560; SCHEMBL30302380	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OCCOCCOCCOCC4CN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)C3)C=C1)C=C2	C44H46N6O9	Tau	P10636	CRBN	WO-2018102067-A2
TPD-4ASKD0	SCHEMBL20120892	2-(2,6-Dioxopiperidin-3-yl)-5-[2-[2-[2-[2-[2-(5-pyrimido[1,2-a]benzimidazol-2-ylpyridin-2-yl)oxyethoxy]ethoxy]ethoxy]ethoxy]ethoxy]isoindole-1,3-dione; SCHEMBL29547682	O=C1CCC(N2C(=O)C3=CC=C(OCCOCCOCCOCCOCCOC4=NC=C(C5=NC6=NC7=CC=CC=C7N6C=C5)C=C4)C=C3C2=O)C(=O)N1	C38H38N6O10	Tau	P10636	CRBN	WO-2018102067-A2
TPD-QVYZLS	SCHEMBL20120414	2-(2,6-Dioxopiperidin-3-yl)-5-[2-[2-[2-[2-[1-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]azetidin-3-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]isoindole-1,3-dione; SCHEMBL29548052	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(N3CC(OCCOCCOCCOCCOC4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)C=C1)C=C2	C41H42N6O9	Tau	P10636	CRBN	WO-2018102067-A2
TPD-2XUHH2	SCHEMBL20120386	2-(2,6-Dioxopiperidin-3-yl)-5-[2-[2-[[3-[[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxymethyl]-1-bicyclo[1.1.1]pentanyl]methoxy]ethoxy]ethoxy]isoindole-1,3-dione; SCHEMBL20120387; SCHEMBL29547601	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OCC45CC(COCCOCCOC6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)(C4)C5)C3)C=C1)C=C2	C45H45N5O9	Tau	P10636	CRBN	WO-2018102067-A2
TPD-MBYBZ8	SCHEMBL20120874	2-(2,6-Dioxopiperidin-3-yl)-5-[2-[2-[2-[2-[3-[4-(5-methylpyrido[4,3-b]indol-7-yl)piperazin-1-yl]propoxy]ethoxy]ethoxy]ethoxy]ethoxy]isoindole-1,3-dione; SCHEMBL29547434	CN1C2=CC=NC=C2C2=C1C=C(N1CCN(CCCOCCOCCOCCOCCOC3=CC=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)CC1)C=C2	C40H48N6O9	Tau	P10636	CRBN	WO-2018102067-A2
TPD-EQM8VL	SCHEMBL20120256	2-(2,6-Dioxopiperidin-3-yl)-5-[3-[3-[2-[6-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxy-2-azaspiro[3.3]heptan-2-yl]ethoxy]propoxy]azetidin-1-yl]isoindole-1,3-dione; SCHEMBL29547494	CN1C2=CC=NC=C2C2=C1C=C(C1=CN=C(OC3CC4(C3)CN(CCOCCCOC3CN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C3)C4)C=C1)C=C2	C44H45N7O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-M1JCZW	SCHEMBL20120405	2-(2,6-Dioxopiperidin-3-yl)-5-[3-[2-[4-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxybut-2-ynoxy]ethoxy]azetidin-1-yl]isoindole-1,3-dione; SCHEMBL20120406; SCHEMBL29547733	CN1C2=CC=NC=C2C2=C1C=C(C1=CC=C(O[C@H]3C[C@H](OCC#CCOCCOC4CN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)C3)N=C1)C=C2	C43H40N6O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-V920PF	SCHEMBL20120544	2-(2,6-Dioxopiperidin-3-yl)-5-[6-[2-[2-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxyethoxy]ethoxy]-2-azaspiro[3.3]heptan-2-yl]isoindole-1,3-dione; SCHEMBL20120548; SCHEMBL30302341	CN1C2=CC=NC=C2C2=C1C=C(C1=CC=C(O[C@H]3C[C@H](OCCOCCOC4CC5(C4)CN(C4=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C4)C5)C3)N=C1)C=C2	C44H44N6O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-11WEZG	SCHEMBL20120803	2-(2,6-Dioxopiperidin-3-yl)-5-[4-[3-[3-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypropoxy]propyl]piperazin-1-yl]isoindole-1,3-dione; SCHEMBL20120805; SCHEMBL30302411	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OCCCOCCCN4CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C3)C=C1)C=C2	C44H47N7O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-7K4NCB	SCHEMBL20120572	2-(2,6-Dioxopiperidin-3-yl)-5-[3-[2-[3-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypropoxy]ethyl-propan-2-ylamino]cyclobutyl]oxyisoindole-1,3-dione; SCHEMBL20129324	CC(C)N(CCOCCCO[C@H]1C[C@H](OC2=NC=C(C3=CC4=C(C=C3)C3=C(C=CN=C3)N4C)C=C2)C1)[C@H]1C[C@H](OC2=CC3=C(C=C2)C(=O)N(C2CCC(=O)NC2=O)C3=O)C1	C46H50N6O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-MYBO7Z	SCHEMBL20120735	2-(2,6-Dioxopiperidin-3-yl)-5-[4-[2-[3-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypropoxy]ethoxy]piperidin-1-yl]isoindole-1,3-dione; SCHEMBL20129277; SCHEMBL29547350	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OCCCOCCOC4CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C3)C=C1)C=C2	C44H46N6O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-5EETQK	SCHEMBL20121023	2-(2,6-Dioxopiperidin-3-yl)-5-[3-[2-[3-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypropoxy]ethylamino]cyclobutyl]oxyisoindole-1,3-dione; SCHEMBL20233872; SCHEMBL29547731	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OCCCOCCN[C@H]4C[C@H](OC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)C3)C=C1)C=C2	C43H44N6O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-CH0WZI	SCHEMBL20120502	2-(2,6-Dioxopiperidin-3-yl)-5-[2-[2-[2-[2-[2-[5-(4-fluoro-5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]ethoxy]isoindole-1,3-dione	CN1C2=C(C=CC(C3=CN=C(OCCOCCOCCOCCOCCOC4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C=C3)=C2)C2=C1C(F)=CN=C2	C40H40FN5O10	Tau	P10636	CRBN	WO-2018102067-A2
TPD-66N4BU	SCHEMBL20120773	3-[6-[3-[5-[3-[5-(8,9-difluoro-5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]prop-2-ynoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL20120775; SCHEMBL30302364	O=C1CCC(N2CC3=C(C=CC(OCC#CC4=NC=C(O[C@H]5C[C@H](OC6=NC=C(C7=CC8=C(C(F)=C7F)C7=C(C=CN=C7)N8)C=C6)C5)C=C4)=C3)C2=O)C(=O)N1	C41H30F2N6O6	Tau	P10636	CRBN	WO-2018102067-A2
TPD-OLZSLM	SCHEMBL20120267	3-[3-oxo-6-[2-[3-[5-[3-[5-(5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]prop-2-ynoxy]ethoxy]-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL20120270; SCHEMBL30302398	O=C1CCC(N2CC3=C(C=CC(OCCOCC#CC4=NC=C(O[C@H]5C[C@H](OC6=NC=C(C7=CC8=C(C=C7)C7=C(C=CN=C7)N8)C=C6)C5)C=C4)=C3)C2=O)C(=O)N1	C43H36N6O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-IRX5OU	SCHEMBL20120979	3-[3-oxo-6-[3-[3-[5-[3-[5-(5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]prop-2-ynoxy]azetidin-1-yl]-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL20120984; SCHEMBL30302350	O=C1CCC(N2CC3=C(C=CC(N4CC(OCC#CC5=NC=C(O[C@H]6C[C@H](OC7=NC=C(C8=CC9=C(C=C8)C8=C(C=CN=C8)N9)C=C7)C6)C=C5)C4)=C3)C2=O)C(=O)N1	C44H37N7O6	Tau	P10636	CRBN	WO-2018102067-A2
TPD-Q0O8LE	SCHEMBL20121000	3-[3-oxo-6-[3-[5-[3-[5-(5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyrimidin-2-yl]prop-2-ynoxy]-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL20121002; SCHEMBL30302313	O=C1CCC(N2CC3=C(C=CC(OCC#CC4=NC=C(O[C@H]5C[C@H](OC6=NC=C(C7=CC8=C(C=C7)C7=C(C=CN=C7)N8)C=C6)C5)C=N4)=C3)C2=O)C(=O)N1	C40H31N7O6	Tau	P10636	CRBN	WO-2018102067-A2
TPD-UJNX2M	SCHEMBL20121024	3-[3-oxo-6-[3-[6-[3-[5-(5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridin-3-yl]prop-2-ynoxy]-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL20121026; SCHEMBL30302382	O=C1CCC(N2CC3=C(C=CC(OCC#CC4=CN=C(O[C@H]5C[C@H](OC6=NC=C(C7=CC8=C(C=C7)C7=C(C=CN=C7)N8)C=C6)C5)C=C4)=C3)C2=O)C(=O)N1	C41H32N6O6	Tau	P10636	CRBN	WO-2018102067-A2
TPD-A0B4PW	SCHEMBL20120784	3-[3-oxo-6-[3-[3-[5-[3-[5-(5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]propoxy]prop-1-ynyl]-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL20120786; SCHEMBL30302339	O=C1CCC(N2CC3=C(C=CC(C#CCOCCCC4=NC=C(O[C@H]5C[C@H](OC6=NC=C(C7=CC8=C(C=C7)C7=C(C=CN=C7)N8)C=C6)C5)C=C4)=C3)C2=O)C(=O)N1	C44H38N6O6	Tau	P10636	CRBN	WO-2018102067-A2
TPD-CWVACN	SCHEMBL20120777	3-[3-oxo-6-[3-[3-[5-[3-[5-(5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]prop-2-ynoxy]propyl]-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL20120782; SCHEMBL30302331	O=C1CCC(N2CC3=C(C=CC(CCCOCC#CC4=NC=C(O[C@H]5C[C@H](OC6=NC=C(C7=CC8=C(C=C7)C7=C(C=CN=C7)N8)C=C6)C5)C=C4)=C3)C2=O)C(=O)N1	C44H38N6O6	Tau	P10636	CRBN	WO-2018102067-A2
TPD-VWM2WM	SCHEMBL20120552	3-[5,7-difluoro-3-oxo-6-[3-[5-[3-[5-(5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]prop-2-ynoxy]-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL20120554; SCHEMBL30302300	O=C1CCC(N2CC3=C(C=C(F)C(OCC#CC4=NC=C(O[C@H]5C[C@H](OC6=NC=C(C7=CC8=C(C=C7)C7=C(C=CN=C7)N8)C=C6)C5)C=C4)=C3F)C2=O)C(=O)N1	C41H30F2N6O6	Tau	P10636	CRBN	WO-2018102067-A2
TPD-E5RLZW	SCHEMBL20120849	3-[3-oxo-6-[3-[3-[5-[3-[5-(5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]prop-2-ynoxy]cyclobutyl]oxy-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL20129326	O=C1CCC(N2CC3=C(C=CC(O[C@H]4C[C@H](OCC#CC5=NC=C(O[C@H]6C[C@H](OC7=NC=C(C8=CC9=C(C=C8)C8=C(C=CN=C8)N9)C=C7)C6)C=C5)C4)=C3)C2=O)C(=O)N1	C45H38N6O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-YLFNFJ	SCHEMBL20120684	3-[3-oxo-6-[4-[3-[5-[3-[5-(5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]prop-2-ynyl]piperazin-1-yl]-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL20120687; SCHEMBL30302316	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC#CC5=NC=C(O[C@H]6C[C@H](OC7=NC=C(C8=CC9=C(C=C8)C8=C(C=CN=C8)N9)C=C7)C6)C=C5)CC4)=C3)C2=O)C(=O)N1	C45H40N8O5	Tau	P10636	CRBN	WO-2018102067-A2
TPD-5EW3KF	SCHEMBL20120608	N-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-N-methyl-2-[3-[5-[3-[5-(5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]prop-2-ynoxy]acetamide; SCHEMBL20120610; SCHEMBL30302386	CN(C(=O)COCC#CC1=NC=C(O[C@H]2C[C@H](OC3=NC=C(C4=CC5=C(C=C4)C4=C(C=CN=C4)N5)C=C3)C2)C=C1)C1=CC2=C(C=C1)C(=O)N(C1CCC(=O)NC1=O)C2	C44H37N7O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-Q0TFJZ	SCHEMBL20120928	3-[3-oxo-6-[3-[3-[5-[3-[5-(5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]prop-2-ynoxy]cyclobutyl]-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL20129327	O=C1CCC(N2CC3=C(C=CC([C@H]4C[C@H](OCC#CC5=NC=C(O[C@H]6C[C@H](OC7=NC=C(C8=CC9=C(C=C8)C8=C(C=CN=C8)N9)C=C7)C6)C=C5)C4)=C3)C2=O)C(=O)N1	C45H38N6O6	Tau	P10636	CRBN	WO-2018102067-A2
TPD-EH6NKA	SCHEMBL20120636	3-[3-oxo-6-[3-[6-[3-[5-(5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridazin-3-yl]prop-2-ynoxy]-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL20120637; SCHEMBL30302412	O=C1CCC(N2CC3=C(C=CC(OCC#CC4=NN=C(O[C@H]5C[C@H](OC6=NC=C(C7=CC8=C(C=C7)C7=C(C=CN=C7)N8)C=C6)C5)C=C4)=C3)C2=O)C(=O)N1	C40H31N7O6	Tau	P10636	CRBN	WO-2018102067-A2
TPD-1MU00J	SCHEMBL20120966	3-[3-oxo-6-[3-[5-[3-[5-(5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyrazin-2-yl]prop-2-ynoxy]-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL20120967; SCHEMBL30302355	O=C1CCC(N2CC3=C(C=CC(OCC#CC4=NC=C(O[C@H]5C[C@H](OC6=NC=C(C7=CC8=C(C=C7)C7=C(C=CN=C7)N8)C=C6)C5)N=C4)=C3)C2=O)C(=O)N1	C40H31N7O6	Tau	P10636	CRBN	WO-2018102067-A2
TPD-HFZPDG	SCHEMBL20120911	3-[6-[2-[3-[5-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]prop-2-ynoxy]ethoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL20120914; SCHEMBL30302352	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4=CN=C(C#CCOCCOC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6)C=C4)C3)C=C1)C=C2	C44H38N6O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-GMQNYF	SCHEMBL20120700	3-[6-[3-[5-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]prop-2-ynoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL20120701; SCHEMBL30302439	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4=CN=C(C#CCOC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6)C=C4)C3)C=C1)C=C2	C42H34N6O6	Tau	P10636	CRBN	WO-2018102067-A2
TPD-98GCGP	SCHEMBL20121025	2-[3-[6-[3-[2-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxyethoxy]prop-1-ynyl]pyridin-3-yl]oxycyclobutyl]oxy-5-(5-methylpyrido[4,3-b]indol-7-yl)pyridine-3-carbonitrile; SCHEMBL20121027	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4=CN=C(C#CCOCCOC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C=C4)C3)C(C#N)=C1)C=C2	C45H35N7O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-Y0XFJC	SCHEMBL20120339	5-[2-[3-[5-[3-[5-[5-(Difluoromethyl)pyrido[4,3-b]indol-7-yl]pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]prop-2-ynoxy]ethoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione; SCHEMBL20120340; SCHEMBL30302395; OJGDGSGMUIYINX-JZSUORBJSA-N; 5-[2-[3-[5-[3-[5-[5-(Difluoromethyl)pyrido[4,3-b]indol-7-yl]pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]prop-2-ynoxy]ethoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=C(C=C(OCCOCC#CC4=NC=C(O[C@H]5C[C@H](OC6=NC=C(C7=CC8=C(C=C7)C7=C(C=CN=C7)N8C(F)F)C=C6)C5)C=C4)C=C3)C2=O)C(=O)N1	C44H34F2N6O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-GPN6CB	SCHEMBL20120418	2-(2,6-Dioxopiperidin-3-yl)-5-[2-[3-[5-[3-[3-methyl-5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]prop-2-ynoxy]ethoxy]isoindole-1,3-dione; SCHEMBL20120420; SCHEMBL30302389	CC1=CC(C2=CC3=C(C=C2)C2=C(C=CN=C2)N3C)=CN=C1O[C@H]1C[C@H](OC2=CN=C(C#CCOCCOC3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C=C2)C1	C45H38N6O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-J0KJDJ	SCHEMBL20120920	2-[3-[6-[3-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]oxy]ethoxy]prop-1-ynyl]pyridin-3-yl]oxycyclobutyl]oxy-5-(5-methylpyrido[4,3-b]indol-7-yl)pyridine-3-carbonitrile; SCHEMBL20120922	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4=CN=C(C#CCOCCOC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6)C=C4)C3)C(C#N)=C1)C=C2	C45H37N7O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-PHGEQS	SCHEMBL20120725	3-[6-[2-[3-[5-[3-[5-[5-(difluoromethyl)pyrido[4,3-b]indol-7-yl]pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]prop-2-ynoxy]ethoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL20120727; SCHEMBL30302372; SHPSCWSBIDLSJW-PLNJQJAISA-N; 3-[6-[2-[3-[5-[3-[5-[5-(difluoromethyl)pyrido[4,3-b]indol-7-yl]pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]prop-2-ynoxy]ethoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(OCCOCC#CC4=NC=C(O[C@H]5C[C@H](OC6=NC=C(C7=CC8=C(C=C7)C7=C(C=CN=C7)N8C(F)F)C=C6)C5)C=C4)=C3)C2=O)C(=O)N1	C44H36F2N6O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-45FXZZ	SCHEMBL20121019	3-[6-[2-[3-[5-[3-[3-methyl-5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]prop-2-ynoxy]ethoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL20121021; SCHEMBL30302465	CC1=CC(C2=CC3=C(C=C2)C2=C(C=CN=C2)N3C)=CN=C1O[C@H]1C[C@H](OC2=CN=C(C#CCOCCOC3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4)C=C2)C1	C45H40N6O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-J4LAQ2	SCHEMBL20121009	3-[6-[3-[3-[4-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]phenyl]prop-2-ynoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL20121010; SCHEMBL30302440	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4CCN(C5=CC=CC(C#CCOC6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)=C5)CC4)C3)C=C1)C=C2	C48H44N6O6	Tau	P10636	CRBN	WO-2018102067-A2
TPD-GQ6PJV	SCHEMBL20120583	2-(2,6-Dioxopiperidin-3-yl)-5-[3-[4-[4-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]pyridin-2-yl]prop-2-ynoxy]isoindole-1,3-dione; SCHEMBL20120585; SCHEMBL30302365	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4CCN(C5=CC=NC(C#CCOC6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)=C5)CC4)C3)C=C1)C=C2	C47H41N7O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-W6KU3J	SCHEMBL20120499	3-[6-[3-[4-[4-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]pyridin-2-yl]prop-2-ynoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL20120500; SCHEMBL30302297	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4CCN(C5=CC=NC(C#CCOC6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)=C5)CC4)C3)C=C1)C=C2	C47H43N7O6	Tau	P10636	CRBN	WO-2018102067-A2
TPD-3OF8C1	SCHEMBL20120680	2-(2,6-Dioxopiperidin-3-yl)-5-[3-[4-[4-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]pyrimidin-2-yl]prop-2-ynoxy]isoindole-1,3-dione; SCHEMBL20120682; SCHEMBL30302336	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4CCN(C5=CC=NC(C#CCOC6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)=N5)CC4)C3)C=C1)C=C2	C46H40N8O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-HYHFAY	SCHEMBL20120486	3-[6-[3-[4-[4-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]pyrimidin-2-yl]prop-2-ynoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL20120489; SCHEMBL30302343	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4CCN(C5=CC=NC(C#CCOC6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)=N5)CC4)C3)C=C1)C=C2	C46H42N8O6	Tau	P10636	CRBN	WO-2018102067-A2
TPD-PQS4LR	SCHEMBL20120566	2-(2,6-Dioxopiperidin-3-yl)-5-[3-[2-[4-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]prop-2-ynoxy]isoindole-1,3-dione; SCHEMBL20120568; SCHEMBL30302368	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4CCN(C5=NC=CC(C#CCOC6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)=N5)CC4)C3)C=C1)C=C2	C46H40N8O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-WCY6CA	SCHEMBL20120762	3-[6-[3-[2-[4-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]prop-2-ynoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL20120766; SCHEMBL30302317	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4CCN(C5=NC=CC(C#CCOC6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)=N5)CC4)C3)C=C1)C=C2	C46H42N8O6	Tau	P10636	CRBN	WO-2018102067-A2
TPD-DZIR08	SCHEMBL20120802	2-(2,6-Dioxopiperidin-3-yl)-5-[2-[3-[4-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]propoxy]ethoxy]isoindole-1,3-dione; SCHEMBL20120804; SCHEMBL30302349	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4CCN(CCCOCCOC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C3)C=C1)C=C2	C44H46N6O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-Q6ITDE	SCHEMBL20120442	3-[6-[2-[3-[4-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]propoxy]ethoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL20120444; SCHEMBL30302302	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4CCN(CCCOCCOC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6)CC4)C3)C=C1)C=C2	C44H48N6O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-Q9XNBX	SCHEMBL20120622	2-(2,6-Dioxopiperidin-3-yl)-5-[6-[4-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]hex-2-ynoxy]isoindole-1,3-dione; SCHEMBL20120623; SCHEMBL30302426	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4CCN(CCCC#CCOC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C3)C=C1)C=C2	C45H44N6O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-EZVJR3	SCHEMBL20120926	3-[6-[6-[4-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]hex-2-ynoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL20120927; SCHEMBL30302369	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4CCN(CCCC#CCOC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6)CC4)C3)C=C1)C=C2	C45H46N6O6	Tau	P10636	CRBN	WO-2018102067-A2
TPD-IMO47R	SCHEMBL20120941	2-(2,6-Dioxopiperidin-3-yl)-5-[2-[2-[2-[2-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxyazetidin-1-yl]ethoxy]ethoxy]ethoxy]ethoxy]isoindole-1,3-dione	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(OC3CN(CCOCCOCCOCCOC4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)C=C1)C=C2	C41H42N6O9	Tau	P10636	CRBN	WO-2018102067-A2
TPD-3Z4SSM	SCHEMBL20121028	N-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]oxyethyl]-N-methyl-4-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxybutanamide; SCHEMBL20121030; SCHEMBL30302452	CN(CCOC1CN(C2=CC3=C(C=C2)C(=O)N(C2CCC(=O)NC2=O)C3=O)C1)C(=O)CCCO[C@H]1C[C@H](OC2=NC=C(C3=CC4=C(C=C3)C3=C(C=CN=C3)N4C)C=C2)C1	C44H45N7O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-9NFIP9	SCHEMBL20120948	2-(2,6-Dioxopiperidin-3-yl)-5-[1-[2-[4-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]-2-oxoethyl]azetidin-3-yl]oxyisoindole-1,3-dione; SCHEMBL20120949; SCHEMBL30302407	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4CCN(C(=O)CN5CC(OC6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)C3)C=C1)C=C2	C44H43N7O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-T690A0	SCHEMBL20120383	2-(2,6-Dioxopiperidin-3-yl)-5-[3-[2-[4-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]-2-oxoethoxy]azetidin-1-yl]isoindole-1,3-dione; SCHEMBL20120385; SCHEMBL30302388	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(OC3CC(OC4CCN(C(=O)COC5CN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)C3)C=C1)C=C2	C44H43N7O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-E9SFU9	SCHEMBL20120647	2-(2,6-Dioxopiperidin-3-yl)-5-[3-[3-[4-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]phenoxy]azetidin-1-yl]isoindole-1,3-dione; SCHEMBL20120649; SCHEMBL30302318	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4CCN(C5=CC=CC(OC6CN(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8=O)C6)=C5)CC4)C3)C=C1)C=C2	C48H45N7O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-N0SSAS	SCHEMBL20120506	2-(2,6-Dioxopiperidin-3-yl)-5-[3-[3-[3-[[1-hydroxy-3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]methoxy]propoxy]propoxy]azetidin-1-yl]isoindole-1,3-dione; SCHEMBL30302348	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@](O)(COCCCOCCCOC4CN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)C3)C=C1)C=C2	C44H46N6O9	Tau	P10636	CRBN	WO-2018102067-A2
TPD-AQZCM3	SCHEMBL20120821	2-(2,6-Dioxopiperidin-3-yl)-5-[2-[9-[2-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxyethyl]-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl]ethoxy]isoindole-1,3-dione; SCHEMBL20120822; SCHEMBL30302294	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OCCN4CCC5(CC4)CN(CCOC4=CC6=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CCO5)C3)C=C1)C=C2	C46H49N7O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-SSDGCA	SCHEMBL20120744	2-(2,6-Dioxopiperidin-3-yl)-5-[4-[9-[[1-hydroxy-3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]methyl]-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl]but-2-ynoxy]isoindole-1,3-dione; SCHEMBL20120747; SCHEMBL30302357	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@](O)(CN4CCC5(CC4)CN(CC#CCOC4=CC6=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CCO5)C3)C=C1)C=C2	C47H47N7O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-JQD1T6	SCHEMBL20120465	2-(2,6-Dioxopiperidin-3-yl)-5-[3-[3-[4-[[1-hydroxy-3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]methyl]piperazin-1-yl]phenyl]prop-2-ynoxy]isoindole-1,3-dione; SCHEMBL30302378	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@](O)(CN4CCN(C5=CC=CC(C#CCOC6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)=C5)CC4)C3)C=C1)C=C2	C48H43N7O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-F16ZS4	SCHEMBL20120355	2-(2,6-Dioxopiperidin-3-yl)-5-[3-[3-[4-[[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]methyl]piperazin-1-yl]phenyl]prop-2-ynoxy]isoindole-1,3-dione; SCHEMBL20129328; SCHEMBL29948153	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](CN4CCN(C5=CC=CC(C#CCOC6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)=C5)CC4)C3)C=C1)C=C2	C48H43N7O6	Tau	P10636	CRBN	WO-2018102067-A2
TPD-RIO87T	SCHEMBL20120677	2-(2,6-Dioxopiperidin-3-yl)-5-[2-[3-[3-[[1-hydroxy-3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]methoxy]propoxy]propoxy]ethoxy]isoindole-1,3-dione; SCHEMBL20120679; SCHEMBL30302340	CN1C2=CC=NC=C2C2=C1C=C(C1=CN=C(O[C@H]3C[C@](O)(COCCCOCCCOCCOC4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)C=C1)C=C2	C43H45N5O10	Tau	P10636	CRBN	WO-2018102067-A2
TPD-LOKBUL	SCHEMBL20120546	2-(2,6-Dioxopiperidin-3-yl)-5-[2-[3-[3-[[3-hydroxy-1-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]azetidin-3-yl]methoxy]propoxy]propoxy]ethoxy]isoindole-1,3-dione	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(N3CC(O)(COCCCOCCCOCCOC4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)C=C1)C=C2	C42H44N6O9	Tau	P10636	CRBN	WO-2018102067-A2
TPD-5UM3IA	WO2018102067A2_264	.	CN1C2=CC=NC=C2C2=C1C=C(C1=CN=C3OC4(CC3=C1)CC(OCCCCOCCCOC1CN(C3=CC5=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C5=O)C1)C4)C=C2	C45H46N6O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-2U0MQB	SCHEMBL20121043	5-[2-[2-[2-[2-[2-[5-(6,8-Difluoro-5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]ethoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN1C2=CC=NC=C2C2=C1C(F)=C(C1=CC=C(OCCOCCOCCOCCOCCOC3=CC=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)N=C1)C(F)=C2	C40H39F2N5O10	Tau	P10636	CRBN	WO-2018102067-A2
TPD-FC9NKO	SCHEMBL20120778	2-(2,6-Dioxopiperidin-3-yl)-5-[2-[2-[2-[2-[2-[1-(5-methylpyrido[4,3-b]indol-7-yl)piperidin-4-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]ethoxy]isoindole-1,3-dione	CN1C2=CC=NC=C2C2=C1C=C(N1CCC(OCCOCCOCCOCCOCCOC3=CC=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)CC1)C=C2	C40H47N5O10	Tau	P10636	CRBN	WO-2018102067-A2
TPD-Y0QV45	SCHEMBL20120685	2-(2,6-Dioxopiperidin-3-yl)-5-[3-[2-[3-[2-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxyethyl]cyclobutyl]ethoxy]azetidin-1-yl]isoindole-1,3-dione; SCHEMBL20129330; SCHEMBL22906781; SCHEMBL29547521	CN1C2=CC=NC=C2C2=C1C=C(C1=CC=C(O[C@H]3C[C@H](OCC[C@H]4C[C@H](CCOC5CN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)C4)C3)N=C1)C=C2	C45H46N6O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-ISYIVU	SCHEMBL20120632	2-(2,6-dioxopiperidin-3-yl)-5-[3-[(1S,2R)-2-[4-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxybutoxymethyl]cyclopropyl]azetidin-1-yl]isoindole-1,3-dione; SCHEMBL20129329	CN1C2=CC=NC=C2C2=C1C=C(C1=CC=C(OC3CC(OCCCCOC[C@@H]4C[C@H]4C4CN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)C3)N=C1)C=C2	C45H46N6O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-WTIQP0	SCHEMBL20129331	2-(2,6-dioxopiperidin-3-yl)-5-[3-[4-[[(1R)-2-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]cyclopropyl]methoxy]butoxy]azetidin-1-yl]isoindole-1,3-dione	CN1C2=CC=NC=C2C2=C1C=C(C1=CC=C(O[C@H]3C[C@H](C4C[C@H]4COCCCCOC4CN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)C3)N=C1)C=C2	C45H46N6O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-WX1LNB	WO2018102067A2_270	.	CN1C2=CC=NC=C2C2=C1C=C(C1=CN=C(OC3CC([C@@H]4C[C@H]4COCCOCCOC4CN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)C3)C=C1)C=C2	C45H46N6O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-UM9D8G	SCHEMBL20120947	2-(2,6-Dioxopiperidin-3-yl)-5-[3-[2-[3-[[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxymethyl]cyclobutyl]oxyethoxy]azetidin-1-yl]isoindole-1,3-dione; SCHEMBL20129333; SCHEMBL20233825	CN1C2=CC=NC=C2C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC[C@H]4C[C@H](OCCOC5CN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)C4)C3)C=C1)C=C2	C44H44N6O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-DBSJB1	SCHEMBL20120714	5-[3-[3-[2,2-Difluoro-3-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypropoxy]propoxy]azetidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione; SCHEMBL20120715; SCHEMBL30302322; SIHYDQJIUGTMPB-ARBFJVLTSA-N; 5-[3-[3-[2,2-Difluoro-3-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypropoxy]propoxy]azetidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN1C2=CC=NC=C2C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OCC(F)(F)COCCCOC4CN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)C3)C=C1)C=C2	C43H42F2N6O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-7W6DHJ	SCHEMBL20120262	5-[3-[2,2-Difluoro-3-[3-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypropoxy]propoxy]azetidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione; SCHEMBL20120264; SCHEMBL30302296; USPHFVLALAGYBH-ARBFJVLTSA-N; 5-[3-[2,2-Difluoro-3-[3-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypropoxy]propoxy]azetidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN1C2=CC=NC=C2C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OCCCOCC(F)(F)COC4CN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)C3)C=C1)C=C2	C43H42F2N6O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-GJJ2G1	SCHEMBL20120596	2-(2,6-Dioxopiperidin-3-yl)-5-[2-[3-[5-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]prop-2-ynoxy]propoxy]isoindole-1,3-dione; SCHEMBL20120597; SCHEMBL30302443	CC(COC1=CC=C2C(=O)N(C3CCC(=O)NC3=O)C(=O)C2=C1)OCC#CC1=NC=C(O[C@H]2C[C@H](OC3=NC=C(C4=CC5=C(C=C4)C4=CN=CC=C4N5C)C=C3)C2)C=C1	C45H38N6O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-PAUUFJ	SCHEMBL20120893	2-(2,6-Dioxopiperidin-3-yl)-5-[2-[4-[5-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]but-3-yn-2-yloxy]ethoxy]isoindole-1,3-dione; SCHEMBL20120894; SCHEMBL30302319	CC(C#CC1=NC=C(O[C@H]2C[C@H](OC3=NC=C(C4=CC5=C(C=C4)C4=CN=CC=C4N5C)C=C3)C2)C=C1)OCCOC1=CC=C2C(=O)N(C3CCC(=O)NC3=O)C(=O)C2=C1	C45H38N6O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-93803S	SCHEMBL20120432	5-[2-[1,1-Difluoro-3-[5-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]prop-2-ynoxy]ethoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione; SCHEMBL20120434; SCHEMBL30302405; VQSGEZBIGCWBDO-JZSUORBJSA-N; 5-[2-[1,1-Difluoro-3-[5-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]prop-2-ynoxy]ethoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN1C2=CC=NC=C2C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4=CN=C(C#CC(F)(F)OCCOC5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C=C4)C3)C=C1)C=C2	C44H34F2N6O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-ESYK84	SCHEMBL20120296	3-[3-oxo-6-[4-[5-[3-[5-(5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]but-3-ynoxy]-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL20120299; SCHEMBL30302356	O=C1CCC(N2CC3=C(C=CC(OCCC#CC4=NC=C(O[C@H]5C[C@H](OC6=NC=C(C7=CC8=C(C=C7)C7=C(C=CN=C7)N8)C=C6)C5)C=C4)=C3)C2=O)C(=O)N1	C42H34N6O6	Tau	P10636	CRBN	WO-2018102067-A2
TPD-SQGK9M	SCHEMBL20120877	3-[3-oxo-6-[3-[5-[3-[5-(5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]prop-2-ynoxymethyl]-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL20120878; SCHEMBL30302370	O=C1CCC(N2CC3=C(C=CC(COCC#CC4=NC=C(O[C@H]5C[C@H](OC6=NC=C(C7=CC8=C(C=C7)C7=C(C=CN=C7)N8)C=C6)C5)C=C4)=C3)C2=O)C(=O)N1	C42H34N6O6	Tau	P10636	CRBN	WO-2018102067-A2
TPD-0T9XFS	SCHEMBL20120816	3-[3-oxo-6-[3-[4-[5-[3-[5-(5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]but-3-ynoxy]azetidin-1-yl]-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL20120819; SCHEMBL30302312	O=C1CCC(N2CC3=C(C=CC(N4CC(OCCC#CC5=NC=C(O[C@H]6C[C@H](OC7=NC=C(C8=CC9=C(C=C8)C8=C(C=CN=C8)N9)C=C7)C6)C=C5)C4)=C3)C2=O)C(=O)N1	C45H39N7O6	Tau	P10636	CRBN	WO-2018102067-A2
TPD-T9ICKZ	SCHEMBL20120329	2-(2,6-dioxopiperidin-3-yl)-5-[3-[4-[5-[3-[5-(5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]but-3-ynoxy]azetidin-1-yl]isoindole-1,3-dione; SCHEMBL20120330; SCHEMBL30302402	O=C1CCC(N2C(=O)C3=C(C=C(N4CC(OCCC#CC5=NC=C(O[C@H]6C[C@H](OC7=NC=C(C8=CC9=C(C=C8)C8=C(C=CN=C8)N9)C=C7)C6)C=C5)C4)C=C3)C2=O)C(=O)N1	C45H37N7O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-U8Y26T	SCHEMBL20120430	2-(2,6-dioxopiperidin-3-yl)-5-[3-[5-[5-[3-[5-(5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]pent-4-ynoxy]azetidin-1-yl]isoindole-1,3-dione; SCHEMBL20120431; SCHEMBL30302315	O=C1CCC(N2C(=O)C3=C(C=C(N4CC(OCCCC#CC5=NC=C(O[C@H]6C[C@H](OC7=NC=C(C8=CC9=C(C=C8)C8=C(C=CN=C8)N9)C=C7)C6)C=C5)C4)C=C3)C2=O)C(=O)N1	C46H39N7O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-N9JNF4	SCHEMBL20120640	3-[3-oxo-6-[3-[5-[5-[3-[5-(5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]pent-4-ynoxy]azetidin-1-yl]-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL20120642; SCHEMBL30302358	O=C1CCC(N2CC3=C(C=CC(N4CC(OCCCC#CC5=NC=C(O[C@H]6C[C@H](OC7=NC=C(C8=CC9=C(C=C8)C8=C(C=CN=C8)N9)C=C7)C6)C=C5)C4)=C3)C2=O)C(=O)N1	C46H41N7O6	Tau	P10636	CRBN	WO-2018102067-A2
TPD-ZF7EJH	SCHEMBL20120863	2-(2,6-Dioxopiperidin-3-yl)-5-[1-[4-[5-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]but-3-ynyl]azetidin-3-yl]oxyisoindole-1,3-dione; SCHEMBL20120864; SCHEMBL30302334	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4=CN=C(C#CCCN5CC(OC6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)C=C4)C3)C=C1)C=C2	C46H39N7O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-R2QQZI	SCHEMBL20120612	3-[6-[1-[4-[5-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]but-3-ynyl]azetidin-3-yl]oxy-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL20120613; SCHEMBL30302363	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4=CN=C(C#CCCN5CC(OC6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)C5)C=C4)C3)C=C1)C=C2	C46H41N7O6	Tau	P10636	CRBN	WO-2018102067-A2
TPD-V7VDH6	SCHEMBL20120258	5-[2-[2,2-Difluoro-3-[4-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]propoxy]ethoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione; SCHEMBL20120260; SCHEMBL30302424; QQKQXNAKLSQLCU-JZSUORBJSA-N; 5-[2-[2,2-Difluoro-3-[4-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]propoxy]ethoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN1C2=CC=NC=C2C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4CCN(CC(F)(F)COCCOC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C3)C=C1)C=C2	C44H44F2N6O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-767WOI	SCHEMBL20120294	2-[3-[6-[3-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]oxy]prop-1-ynyl]pyridin-3-yl]oxycyclobutyl]oxy-5-(5H-pyrido[4,3-b]indol-7-yl)pyridine-3-carbonitrile; SCHEMBL20120295	N#CC1=CC(C2=CC3=C(C=C2)C2=C(C=CN=C2)N3)=CN=C1O[C@H]1C[C@H](OC2=CN=C(C#CCOC3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4)C=C2)C1	C42H31N7O6	Tau	P10636	CRBN	WO-2018102067-A2
TPD-HJBPQE	SCHEMBL20120323	3-[6-[3-[5-[3-[3-methyl-5-(5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]prop-2-ynoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL20120326; SCHEMBL30302418	CC1=CC(C2=CC3=C(C=C2)C2=C(C=CN=C2)N3)=CN=C1O[C@H]1C[C@H](OC2=CN=C(C#CCOC3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4)C=C2)C1	C42H34N6O6	Tau	P10636	CRBN	WO-2018102067-A2
TPD-839SBI	SCHEMBL20120836	3-[6-[3-[5-[3-[5-(4-chloro-5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]prop-2-ynoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL20120837; SCHEMBL30302384	O=C1CCC(N2CC3=C(C=CC(OCC#CC4=NC=C(O[C@H]5C[C@H](OC6=NC=C(C7=CC8=C(C=C7)C7=C(N8)C(Cl)=CN=C7)C=C6)C5)C=C4)=C3)C2=O)C(=O)N1	C41H31ClN6O6	Tau	P10636	CRBN	WO-2018102067-A2
TPD-L676L6	SCHEMBL20120307	3-[6-[3-[5-[3-[5-(4-fluoro-5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]prop-2-ynoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL20120309; SCHEMBL30302308	O=C1CCC(N2CC3=C(C=CC(OCC#CC4=NC=C(O[C@H]5C[C@H](OC6=NC=C(C7=CC8=C(C=C7)C7=C(N8)C(F)=CN=C7)C=C6)C5)C=C4)=C3)C2=O)C(=O)N1	C41H31FN6O6	Tau	P10636	CRBN	WO-2018102067-A2
TPD-RBNIFQ	SCHEMBL20120655	3-[6-[3-[5-[3-[5-[5-(difluoromethyl)pyrido[4,3-b]indol-7-yl]pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]prop-2-ynoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL20120656; SCHEMBL30302361; QUKUQYQWDZZUQZ-BVOFGUPTSA-N; 3-[6-[3-[5-[3-[5-[5-(difluoromethyl)pyrido[4,3-b]indol-7-yl]pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]prop-2-ynoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(OCC#CC4=NC=C(O[C@H]5C[C@H](OC6=NC=C(C7=CC8=C(C=C7)C7=C(C=CN=C7)N8C(F)F)C=C6)C5)C=C4)=C3)C2=O)C(=O)N1	C42H32F2N6O6	Tau	P10636	CRBN	WO-2018102067-A2
TPD-88TKTP	SCHEMBL20120241	2-(2,6-Dioxopiperidin-3-yl)-5-[2-[3-[3-[[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxymethyl]-1-bicyclo[1.1.1]pentanyl]prop-2-ynoxy]ethoxy]isoindole-1,3-dione; SCHEMBL20120242; SCHEMBL30302353	CN1C2=CC=NC=C2C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OCC45CC(C#CCOCCOC6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)(C4)C5)C3)C=C1)C=C2	C45H41N5O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-IZFCS1	SCHEMBL20120872	2-(2,6-Dioxopiperidin-3-yl)-5-[2-[3-[3-[[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxymethyl]cyclobutyl]prop-2-ynoxy]ethoxy]isoindole-1,3-dione; SCHEMBL20129334	CN1C2=CC=NC=C2C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC[C@H]4C[C@H](C#CCOCCOC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)C3)C=C1)C=C2	C44H41N5O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-30EXIJ	SCHEMBL20120358	3-[3-oxo-6-[4-[3-[5-[3-[5-(5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]prop-2-ynoxy]piperidin-1-yl]-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL20120361; SCHEMBL30302307	O=C1CCC(N2CC3=C(C=CC(N4CCC(OCC#CC5=NC=C(O[C@H]6C[C@H](OC7=NC=C(C8=CC9=C(C=C8)C8=C(C=CN=C8)N9)C=C7)C6)C=C5)CC4)=C3)C2=O)C(=O)N1	C46H41N7O6	Tau	P10636	CRBN	WO-2018102067-A2
TPD-9W4NAP	SCHEMBL20120255	2-(2,6-dioxopiperidin-3-yl)-6-[2-[3-[5-[3-[5-(5H-pyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]prop-2-ynoxy]ethoxy]pyrrolo[3,4-c]pyridine-1,3-dione; SCHEMBL20120257; SCHEMBL29948013	O=C1CCC(N2C(=O)C3=C(C=C(OCCOCC#CC4=NC=C(O[C@H]5C[C@H](OC6=NC=C(C7=CC8=C(C=C7)C7=C(C=CN=C7)N8)C=C6)C5)C=C4)N=C3)C2=O)C(=O)N1	C42H33N7O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-W6SYBU	SCHEMBL20120924	2-(2,6-Dioxopiperidin-3-yl)-5-[3-[2-[[3-[[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxymethyl]-1-bicyclo[1.1.1]pentanyl]methoxy]ethoxy]azetidin-1-yl]isoindole-1,3-dione; SCHEMBL20120925; SCHEMBL30302328	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OCC45CC(COCCOC6CN(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8=O)C6)(C4)C5)C3)C=C1)C=C2	C46H46N6O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-PZSU3S	SCHEMBL20132983	2-[3-[2-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxyethoxy]prop-1-ynyl]-5-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridine-4-carbonitrile; SCHEMBL30302359	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4=CN=C(C#CCOCCOC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C=C4C#N)C3)C=C1)C=C2	C45H35N7O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-WCZ54Z	SCHEMBL20133334	2-[3-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]oxy]ethoxy]prop-1-ynyl]-5-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridine-4-carbonitrile; SCHEMBL30302304	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4=CN=C(C#CCOCCOC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6)C=C4C#N)C3)C=C1)C=C2	C45H37N7O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-ELSDXS	SCHEMBL20120997	2-(2,6-Dioxopiperidin-3-yl)-5-[2-[3-[4-methyl-5-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]prop-2-ynoxy]ethoxy]isoindole-1,3-dione; SCHEMBL20120998; SCHEMBL30302323	CC1=CC(C#CCOCCOC2=CC3=C(C=C2)C(=O)N(C2CCC(=O)NC2=O)C3=O)=NC=C1O[C@H]1C[C@H](OC2=NC=C(C3=CC4=C(C=C3)C3=C(C=CN=C3)N4C)C=C2)C1	C45H38N6O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-85FJML	SCHEMBL20120599	3-[6-[2-[3-[4-methyl-5-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]prop-2-ynoxy]ethoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL20120603; SCHEMBL30302438	CC1=CC(C#CCOCCOC2=CC3=C(C=C2)C(=O)N(C2CCC(=O)NC2=O)C3)=NC=C1O[C@H]1C[C@H](OC2=NC=C(C3=CC4=C(C=C3)C3=C(C=CN=C3)N4C)C=C2)C1	C45H40N6O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-EXD7VH	SCHEMBL20120724	3-[6-[2-[3-[5-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxy-4-(trifluoromethyl)pyridin-2-yl]prop-2-ynoxy]ethoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL20120728; SCHEMBL30302413; YUUZQWVFZDNJIB-UDFALXFKSA-N; 3-[6-[2-[3-[5-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxy-4-(trifluoromethyl)pyridin-2-yl]prop-2-ynoxy]ethoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4=CN=C(C#CCOCCOC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6)C=C4C(F)(F)F)C3)C=C1)C=C2	C45H37F3N6O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-H7F05V	SCHEMBL20120424	2-(2,6-Dioxopiperidin-3-yl)-5-[2-[3-[5-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxy-4-(trifluoromethyl)pyridin-2-yl]prop-2-ynoxy]ethoxy]isoindole-1,3-dione; SCHEMBL20120425; SCHEMBL30302351; FJUDEABXUANZON-VZASAIHWSA-N; 2-(2,6-Dioxopiperidin-3-yl)-5-[2-[3-[5-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxy-4-(trifluoromethyl)pyridin-2-yl]prop-2-ynoxy]ethoxy]isoindole-1,3-dione	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4=CN=C(C#CCOCCOC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C=C4C(F)(F)F)C3)C=C1)C=C2	C45H35F3N6O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-CT4EZ9	SCHEMBL20129335	6-[3-[2-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxyethoxy]prop-1-ynyl]-3-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridine-2-carbonitrile; SCHEMBL30302399	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4=C(C#N)N=C(C#CCOCCOC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C=C4)C3)C=C1)C=C2	C45H35N7O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-P9LADU	SCHEMBL20120856	6-[3-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]oxy]ethoxy]prop-1-ynyl]-3-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridine-2-carbonitrile; SCHEMBL20129336; SCHEMBL30302374	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4=C(C#N)N=C(C#CCOCCOC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6)C=C4)C3)C=C1)C=C2	C45H37N7O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-FZGEH6	SCHEMBL20120809	2-(2,6-Dioxopiperidin-3-yl)-5-[2-[3-[6-methyl-5-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]prop-2-ynoxy]ethoxy]isoindole-1,3-dione; SCHEMBL20120810; SCHEMBL30302342	CC1=C(O[C@H]2C[C@H](OC3=NC=C(C4=CC5=C(C=C4)C4=C(C=CN=C4)N5C)C=C3)C2)C=CC(C#CCOCCOC2=CC3=C(C=C2)C(=O)N(C2CCC(=O)NC2=O)C3=O)=N1	C45H38N6O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-N5AX3D	SCHEMBL20120815	3-[6-[2-[3-[6-methyl-5-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]prop-2-ynoxy]ethoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL20120818; SCHEMBL30302333	CC1=C(O[C@H]2C[C@H](OC3=NC=C(C4=CC5=C(C=C4)C4=C(C=CN=C4)N5C)C=C3)C2)C=CC(C#CCOCCOC2=CC3=C(C=C2)C(=O)N(C2CCC(=O)NC2=O)C3)=N1	C45H40N6O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-GOAQRZ	SCHEMBL20120564	2-(2,6-Dioxopiperidin-3-yl)-5-[2-[3-[5-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxy-6-(trifluoromethyl)pyridin-2-yl]prop-2-ynoxy]ethoxy]isoindole-1,3-dione; SCHEMBL20120565; SCHEMBL30302400; VQBMJWZMIMWFPD-DJYSDWLISA-N; 2-(2,6-Dioxopiperidin-3-yl)-5-[2-[3-[5-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxy-6-(trifluoromethyl)pyridin-2-yl]prop-2-ynoxy]ethoxy]isoindole-1,3-dione	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4=C(C(F)(F)F)N=C(C#CCOCCOC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C=C4)C3)C=C1)C=C2	C45H35F3N6O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-DAEH6U	SCHEMBL20120989	3-[6-[2-[3-[5-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxy-6-(trifluoromethyl)pyridin-2-yl]prop-2-ynoxy]ethoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL20120991; SCHEMBL30302367; BYSGTYYBCLKBPI-NNMFAMJJSA-N; 3-[6-[2-[3-[5-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxy-6-(trifluoromethyl)pyridin-2-yl]prop-2-ynoxy]ethoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4=C(C(F)(F)F)N=C(C#CCOCCOC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6)C=C4)C3)C=C1)C=C2	C45H37F3N6O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-GIRZ2M	SCHEMBL20120999	2-(2,6-Dioxopiperidin-3-yl)-5-[2-[2-methyl-4-[5-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]but-3-yn-2-yl]oxyethoxy]isoindole-1,3-dione; SCHEMBL20121001; SCHEMBL30302366	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4=CN=C(C#CC(C)(C)OCCOC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C=C4)C3)C=C1)C=C2	C46H40N6O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-DZ72HH	SCHEMBL20120438	3-[6-[2-[2-methyl-4-[5-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]but-3-yn-2-yl]oxyethoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL20120439; SCHEMBL30302458	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4=CN=C(C#CC(C)(C)OCCOC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6)C=C4)C3)C=C1)C=C2	C46H42N6O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-RIF7MC	SCHEMBL20120232	3-[6-[2-[1-[2-[5-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]ethynyl]cyclopropyl]oxyethoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL20120234; SCHEMBL30302409	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4=CN=C(C#CC5(OCCOC6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)CC5)C=C4)C3)C=C1)C=C2	C46H40N6O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-SC5D89	SCHEMBL20120266	2-(2,6-Dioxopiperidin-3-yl)-5-[2-[1-[2-[5-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridin-2-yl]ethynyl]cyclopropyl]oxyethoxy]isoindole-1,3-dione; SCHEMBL20120269; SCHEMBL30302347	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4=CN=C(C#CC5(OCCOC6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C=C4)C3)C=C1)C=C2	C46H38N6O8	Tau	P10636	CRBN	WO-2018102067-A2
TPD-7IKKUW	SCHEMBL20120858	4-[3-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxyprop-1-ynyl]-2-[4-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]benzonitrile; SCHEMBL20120859; SCHEMBL30302310	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4CCN(C5=C(C#N)C=CC(C#CCOC6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)=C5)CC4)C3)C=C1)C=C2	C49H41N7O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-S8GPQO	SCHEMBL20120943	4-[3-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]oxy]prop-1-ynyl]-2-[4-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]benzonitrile; SCHEMBL20120944; SCHEMBL30302375	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4CCN(C5=C(C#N)C=CC(C#CCOC6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)=C5)CC4)C3)C=C1)C=C2	C49H43N7O6	Tau	P10636	CRBN	WO-2018102067-A2
TPD-N4OZB2	SCHEMBL20120751	3-[6-[3-[4-methyl-3-[4-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]phenyl]prop-2-ynoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL20120753; SCHEMBL30302442	CC1=C(N2CCC(O[C@H]3C[C@H](OC4=NC=C(C5=CC6=C(C=C5)C5=C(C=CN=C5)N6C)C=C4)C3)CC2)C=C(C#CCOC2=CC3=C(C=C2)C(=O)N(C2CCC(=O)NC2=O)C3)C=C1	C49H46N6O6	Tau	P10636	CRBN	WO-2018102067-A2
TPD-DHR8CZ	SCHEMBL20120479	3-[6-[3-[3-[4-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]-4-(trifluoromethyl)phenyl]prop-2-ynoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL20120480; SCHEMBL30302337; NKOJXKSPFAIWRT-GRVYEOBCSA-N; 3-[6-[3-[3-[4-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]-4-(trifluoromethyl)phenyl]prop-2-ynoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4CCN(C5=C(C(F)(F)F)C=CC(C#CCOC6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)=C5)CC4)C3)C=C1)C=C2	C49H43F3N6O6	Tau	P10636	CRBN	WO-2018102067-A2
TPD-KD0BQN	SCHEMBL20120888	3-[6-[3-[4-[4-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]-5-(trifluoromethyl)pyridin-2-yl]prop-2-ynoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL20120890; SCHEMBL30302432; VKMWSZRVOWZLKL-XXVNREIUSA-N; 3-[6-[3-[4-[4-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]-5-(trifluoromethyl)pyridin-2-yl]prop-2-ynoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4CCN(C5=C(C(F)(F)F)C=NC(C#CCOC6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)=C5)CC4)C3)C=C1)C=C2	C48H42F3N7O6	Tau	P10636	CRBN	WO-2018102067-A2
TPD-4G3LR8	SCHEMBL20120779	6-[3-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]oxy]prop-1-ynyl]-4-[4-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]pyridine-3-carbonitrile; SCHEMBL20120781; SCHEMBL30302390	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4CCN(C5=C(C#N)C=NC(C#CCOC6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)=C5)CC4)C3)C=C1)C=C2	C48H42N8O6	Tau	P10636	CRBN	WO-2018102067-A2
TPD-7RQOTO	SCHEMBL20120689	3-[3-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxyprop-1-ynyl]-5-[4-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]benzonitrile; SCHEMBL20120690; SCHEMBL30302360	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4CCN(C5=CC(C#N)=CC(C#CCOC6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)=C5)CC4)C3)C=C1)C=C2	C49H41N7O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-W5MHMW	SCHEMBL20120847	3-[3-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]oxy]prop-1-ynyl]-5-[4-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]benzonitrile; SCHEMBL20120848; SCHEMBL30302344	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4CCN(C5=CC(C#N)=CC(C#CCOC6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)=C5)CC4)C3)C=C1)C=C2	C49H43N7O6	Tau	P10636	CRBN	WO-2018102067-A2
TPD-7RSIMZ	SCHEMBL20120259	3-[6-[3-[3-methyl-5-[4-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]phenyl]prop-2-ynoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL20120261; SCHEMBL30302298	CC1=CC(C#CCOC2=CC3=C(C=C2)C(=O)N(C2CCC(=O)NC2=O)C3)=CC(N2CCC(O[C@H]3C[C@H](OC4=NC=C(C5=CC6=C(C=C5)C5=C(C=CN=C5)N6C)C=C4)C3)CC2)=C1	C49H46N6O6	Tau	P10636	CRBN	WO-2018102067-A2
TPD-HY4WMH	SCHEMBL20120970	3-[6-[3-[3-[4-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]-5-(trifluoromethyl)phenyl]prop-2-ynoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL20120972; SCHEMBL30302335; GDTZFTCSRQFCLM-HMRDGLPVSA-N; 3-[6-[3-[3-[4-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]-5-(trifluoromethyl)phenyl]prop-2-ynoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4CCN(C5=CC(C(F)(F)F)=CC(C#CCOC6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)=C5)CC4)C3)C=C1)C=C2	C49H43F3N6O6	Tau	P10636	CRBN	WO-2018102067-A2
TPD-KWCTAP	SCHEMBL20120657	3-[6-[3-[4-[4-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]-6-(trifluoromethyl)pyridin-2-yl]prop-2-ynoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL20120658; SCHEMBL30302457; XKJJYTKYAJJTHB-BHSYBDTKSA-N; 3-[6-[3-[4-[4-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]-6-(trifluoromethyl)pyridin-2-yl]prop-2-ynoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4CCN(C5=CC(C(F)(F)F)=NC(C#CCOC6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)=C5)CC4)C3)C=C1)C=C2	C48H42F3N7O6	Tau	P10636	CRBN	WO-2018102067-A2
TPD-FCJEEQ	SCHEMBL20120364	3-[6-[3-[2-[4-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]-6-(trifluoromethyl)pyridin-4-yl]prop-2-ynoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL20120366; SCHEMBL30302338; JIBWYSQTVFCOIX-XWCQTXCCSA-N; 3-[6-[3-[2-[4-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]-6-(trifluoromethyl)pyridin-4-yl]prop-2-ynoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4CCN(C5=NC(C(F)(F)F)=CC(C#CCOC6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)=C5)CC4)C3)C=C1)C=C2	C48H42F3N7O6	Tau	P10636	CRBN	WO-2018102067-A2
TPD-4YNUFT	SCHEMBL20120869	2-(2,6-Dioxopiperidin-3-yl)-5-[2-methyl-4-[3-[4-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]phenyl]but-3-yn-2-yl]oxyisoindole-1,3-dione; SCHEMBL20120871; SCHEMBL30302371	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4CCN(C5=CC=CC(C#CC(C)(C)OC6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)=C5)CC4)C3)C=C1)C=C2	C50H46N6O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-1J7NNI	SCHEMBL20120853	3-[6-[2-methyl-4-[3-[4-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]phenyl]but-3-yn-2-yl]oxy-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL20120854; SCHEMBL30302449	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4CCN(C5=CC=CC(C#CC(C)(C)OC6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)=C5)CC4)C3)C=C1)C=C2	C50H48N6O6	Tau	P10636	CRBN	WO-2018102067-A2
TPD-7LZBDK	SCHEMBL20120930	3-[6-[2-methyl-4-[4-[4-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]pyridin-2-yl]but-3-yn-2-yl]oxy-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL20129343; SCHEMBL29948095	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4CCN(C5=CC=NC(C#CC(C)(C)OC6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)=C5)CC4)C3)C=C1)C=C2	C49H47N7O6	Tau	P10636	CRBN	WO-2018102067-A2
TPD-P9MF7L	SCHEMBL20120721	3-[6-[1,1-difluoro-3-[4-[4-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]pyridin-2-yl]prop-2-ynoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL20120722; SCHEMBL30302326; XCKRVYCLMYMKEG-BHSYBDTKSA-N; 3-[6-[1,1-difluoro-3-[4-[4-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]pyridin-2-yl]prop-2-ynoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4CCN(C5=CC=NC(C#CC(F)(F)OC6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)=C5)CC4)C3)C=C1)C=C2	C47H41F2N7O6	Tau	P10636	CRBN	WO-2018102067-A2
TPD-OK6FFN	SCHEMBL20120767	3-[6-[2-methyl-4-[4-[4-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]pyrimidin-2-yl]but-3-yn-2-yl]oxy-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL20120771; SCHEMBL30302430	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4CCN(C5=CC=NC(C#CC(C)(C)OC6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)=N5)CC4)C3)C=C1)C=C2	C48H46N8O6	Tau	P10636	CRBN	WO-2018102067-A2
TPD-6TVTRD	SCHEMBL20120445	6-[3-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]oxy]-3-methylbut-1-ynyl]-4-[4-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]pyridine-3-carbonitrile; SCHEMBL20120447; SCHEMBL30302419	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4CCN(C5=C(C#N)C=NC(C#CC(C)(C)OC6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)=C5)CC4)C3)C=C1)C=C2	C50H46N8O6	Tau	P10636	CRBN	WO-2018102067-A2
TPD-IAPB2Q	SCHEMBL20120584	2-[3-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]oxy]ethoxy]-3-methylbut-1-ynyl]-5-[3-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]oxycyclobutyl]oxypyridine-4-carbonitrile; SCHEMBL20120589; SCHEMBL30302373	CN1C2=C(C=NC=C2)C2=C1C=C(C1=CN=C(O[C@H]3C[C@H](OC4=CN=C(C#CC(C)(C)OCCOC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6)C=C4C#N)C3)C=C1)C=C2	C47H41N7O7	Tau	P10636	CRBN	WO-2018102067-A2
TPD-ZVL961	SCHEMBL20211857	(2S,4R)-4-hydroxy-1-[(2S)-2-[[2-[2-[4-[2-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]ethyl]piperazin-1-yl]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCN3CCN(CCOC4=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=CC=C5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C54H66N6O7S	ERα;ERβ	P03372/Q92731	VHL	WO-2018102725-A1
TPD-AUWDCY	SCHEMBL20234860	(2S,4R)-4-hydroxy-1-[(2S)-2-[[2-[2-[4-[2-[4-[(1S,2R)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]ethyl]piperazin-1-yl]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCN3CCN(CCOC4=CC=C([C@H]5C6=CC=C(O)C=C6CC[C@H]5C5=CC=CC=C5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C54H66N6O7S	ERα;ERβ	P03372/Q92731	VHL	WO-2018102725-A1
TPD-I9340T	WO2018102725A1_3	.	O=C1CC[C@H](N2CC3=C(OCCCN4CCN(CCOC5=CC=C(C6C7=CC=C(O)C=C7CCN6C6=CC=CC=C6)C=C5)CC4)C=CC=C3C2=O)C(=O)N1	C43H47N5O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-Q1FUBU	WO2018102725A1_4	3-[7-[2-[4-[2-[4-(6-hydroxy-2-phenyl-3,4-dihydro-1H-isoquinolin-1-yl)phenoxy]ethyl]piperazin-1-yl]ethoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(OCCN4CCN(CCOC5=CC=C(C6C7=CC=C(O)C=C7CCN6C6=CC=CC=C6)C=C5)CC4)C=CC=C3C2=O)C(=O)N1	C42H45N5O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-26E6ST	WO2018102725A1_5	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCN3CCN(CCOC4=CC=C(C5C6=CC=C(O)C=C6CCN5C5=CC=CC=C5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C53H65N7O7S	ERα;ERβ	P03372/Q92731	VHL	WO-2018102725-A1
TPD-69FUS0	WO2018102725A1_6	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCN3CCN(CCOC4=CC=C([C@H]5C6=CC=C(O)C=C6C=C[C@H]5C5=CC=CC=C5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C55H66N6O7S	ERα;ERβ	P03372/Q92731	VHL	WO-2018102725-A1
TPD-ZEB4HO	WO2018102725A1_7	.	O=C1CC[C@H](N2CC3=C(C=CC(OCCN4CCN(CCOC5=CC=C(C6C7=CC=C(O)C=C7CC[C@H]6C6=CC=CC=C6)C=C5)CC4)=C3)C2=O)C(=O)N1	C43H46N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-KE275T	SCHEMBL20234461	(3S)-3-[6-[2-[4-[2-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]ethyl]piperazin-1-yl]ethoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CC[C@H](N2CC3=C(C=CC(OCCN4CCN(CCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)=C3)C2=O)C(=O)N1	C43H46N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-3DKFS6	SCHEMBL20234976	(3S)-3-[6-[2-[(1R,4R)-5-[2-[4-[2-(4-fluorophenyl)-6-hydroxy-3,4-dihydro-1H-isoquinolin-1-yl]phenoxy]ethyl]-2,5-diazabicyclo[2.2.1]heptan-2-yl]ethoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CC[C@H](N2CC3=C(C=CC(OCCN4C[C@H]5C[C@@H]4CN5CCOC4=CC=C(C5C6=CC=C(O)C=C6CCN5C5=CC=C(F)C=C5)C=C4)=C3)C2=O)C(=O)N1	C43H44FN5O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-YM3LZU	WO2018102725A1_10	.	O=C1CCC(N2CC3=C(C=CC(NCCN4CCN(CCOC5=CC=C([C@H]6C7=CC=C(O)C=C7CC[C@H]6C6=CC=CC=C6)C=C5)CC4)=C3)C2=O)C(=O)N1	C43H47N5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-QUMN6O	SCHEMBL20231773	3-[6-[2-[4-[2-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]ethyl]piperazin-1-yl]ethylamino]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(NCCN4CCN(CCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)=C3)C2=O)C(=O)N1	C43H47N5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-D4UHO1	WO2018102725A1_12	.	O=C1CCC(N2CC3=CC(NCCCN4CCN(CCOC5=CC=C([C@H]6C7=CC=C(O)C=C7CC[C@H]6C6=CC=CC=C6)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C44H49N5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-I1QE0G	WO2018102725A1_13	.	O=C1CCC(N2CC3=CC(NCCCN4CCN(CCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C44H49N5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-LP87G8	WO2018102725A1_14	.	O=C1CC[C@H](N2CC3=C(C=CC(OCCN4C[C@H]5C[C@@H]4CN5CCOC4=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=CC=C5)C=C4)=C3)C2=O)C(=O)N1	C44H46N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-YUW156	SCHEMBL21982878	(3S)-3-[6-[3-[2-[2-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]ethoxy]ethoxy]propylamino]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CC[C@H](N2CC3=C(C=CC(NCCCOCCOCCOC4=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=CC=C5)C=C4)=C3)C2=O)C(=O)N1	C42H45N3O7	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-D6QAH6	WO2018102725A1_16	.	O=C1CCC(N2CC3=C(C=CC=C3OCCN3CC4(CN(CCOC5=CC=C([C@H]6C7=CC=C(O)C=C7CC[C@H]6C6=CC=CC=C6)C=C5)C4)C3)C2=O)C(=O)N1	C44H46N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-G13744	WO2018102725A1_17	.	O=C1CCC(N2CC3=C(C=CC=C3OCCN3CC4(CN(CCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)C4)C3)C2=O)C(=O)N1	C44H46N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-U9TE5R	WO2018102725A1_18	.	O=C1CC[C@H](N2CC3=C(C=CC(OCCN4CC5(CN(CCOC6=CC=C([C@H]7C8=CC=C(O)C=C8CC[C@H]7C7=CC=CC=C7)C=C6)C5)C4)=C3)C2=O)C(=O)N1	C44H46N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-SJZTMO	SCHEMBL20234962	(3S)-3-[6-[2-[6-[2-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]ethyl]-2,6-diazaspiro[3.3]heptan-2-yl]ethoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CC[C@H](N2CC3=C(C=CC(OCCN4CC5(CN(CCOC6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=CC=C7)C=C6)C5)C4)=C3)C2=O)C(=O)N1	C44H46N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-R0OU89	WO2018102725A1_20	.	O=C1CC[C@H](N2CC3=C(C=CC(OCCN4C[C@H]5C[C@@H]4CN5CCOC4=CC=C([C@H]5C6=CC=C(O)C=C6CC[C@H]5C5=CC=CC=C5)C=C4)=C3)C2=O)C(=O)N1	C44H46N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-XJZ0A3	WO2018102725A1_21	.	O=C1CCC(N2CC3=CC(CCCCC(=O)N4CCN(CCOC5=CC=C(C6C7=CC=C(O)C=C7CC[C@H]6C6=CC=CC=C6)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C46H50N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-9HJ9DU	WO2018102725A1_22	.	O=C1CC[C@H](N2CC3=C(C=CC(OCCN4C[C@@H]5C[C@H]4CN5CCOC4=CC=C(C5C6=CC=C(O)C=C6CCN5C5=CC=C(F)C=C5)C=C4)=C3)C2=O)C(=O)N1	C43H44FN5O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-YJANWL	WO2018102725A1_23	.	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCOC5=CC=C([C@H]6C7=CC=C(O)C=C7CC[C@H]6C6=CC=CC=C6)C=C5)CC4)C=C3C2=O)C(=O)N1	C41H40N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-9JSNF4	WO2018102725A1_24	.	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)C=C3C2=O)C(=O)N1	C41H40N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-3FRJLE	WO2018102725A1_25	.	O=C1CCC(N2CC3=CC(NCCCCN4CCN(CCOC5=CC=C([C@H]6C7=CC=C(O)C=C7CC[C@H]6C6=CC=CC=C6)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C45H51N5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-ZPCV3N	SCHEMBL20234689	3-[6-[4-[4-[2-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]ethyl]piperazin-1-yl]butylamino]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(NCCCCN4CCN(CCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C45H51N5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-O034XS	WO2018102725A1_27	.	O=C1CCC(N2CC3=CC(CCC(=O)N4CCN(CCOC5=CC=C([C@H]6C7=CC=C(O)C=C7CC[C@H]6C6=CC=CC=C6)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C44H46N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-SNRLIM	WO2018102725A1_28	.	O=C1CCC(N2CC3=CC(CCC(=O)N4CCN(CCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C44H46N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-RICQG7	SCHEMBL21982912	3-[6-[5-[4-[2-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]ethyl]piperazin-1-yl]-5-oxopentyl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(CCCCC(=O)N4CCN(CCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C46H50N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-0D7HA6	WO2018102725A1_30	.	O=C1CC[C@H](N2CC3=C(C=CC(NCCCOCCCOC4=CC=C([C@H]5C6=CC=C(O)C=C6CC[C@H]5C5=CC=CC=C5)C=C4)=C3)C2=O)C(=O)N1	C41H43N3O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-LQCN5P	WO2018102725A1_31	.	O=C1CC[C@H](N2CC3=C(C=CC(NCCCOCCCOC4=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=CC=C5)C=C4)=C3)C2=O)C(=O)N1	C41H43N3O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-RPJO2Q	WO2018102725A1_32	.	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCCCOC5=CC=C([C@H]6C7=CC=C(O)C=C7CC[C@H]6C6=CC=CC=C6)C=C5)CC4)C=C3C2=O)C(=O)N1	C43H44N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-DKF9CD	WO2018102725A1_33	.	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCCCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)C=C3C2=O)C(=O)N1	C43H44N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-1EA7I4	WO2018102725A1_34	.	O=C1CCC(N2CC3=CC(N4CCN(CCCCOC5=CC=C([C@H]6C7=CC=C(O)C=C7CC[C@H]6C6=CC=CC=C6)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C43H46N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-Y6Y6LY	WO2018102725A1_35	.	O=C1CCC(N2CC3=CC(N4CCN(CCCCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C43H46N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-GN8Q57	WO2018102725A1_36	.	O=C1CCC(N2CC3=CC(N4CCN(CCOC5=CC=C([C@H]6C7=CC=C(O)C=C7CC[C@H]6C6=CC=CC=C6)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C41H42N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-FGNFJE	WO2018102725A1_37	.	O=C1CCC(N2CC3=CC(N4CCN(CCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C41H42N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-MWBNWL	WO2018102725A1_38	.	O=C1CCC(N2C(=O)C3=CC=C(NCCC4CCN(CCOC5=CC=C([C@H]6C7=CC=C(O)C=C7CC[C@H]6C6=CC=CC=C6)C=C5)CC4)C=C3C2=O)C(=O)N1	C44H46N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-W7NU71	SCHEMBL20234425	2-(2,6-dioxopiperidin-3-yl)-5-[2-[1-[2-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]ethyl]piperidin-4-yl]ethylamino]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC=C(NCCC4CCN(CCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)C=C3C2=O)C(=O)N1	C44H46N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-LZLTCM	WO2018102725A1_40	.	O=C1CCC(N2CC3=CC(NCCC4CCN(CCOC5=CC=C([C@H]6C7=CC=C(O)C=C7CC[C@H]6C6=CC=CC=C6)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C44H48N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-MHG1M6	SCHEMBL20234408	3-[6-[2-[1-[2-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]ethyl]piperidin-4-yl]ethylamino]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(NCCC4CCN(CCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C44H48N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-RLR8JN	WO2018102725A1_42	.	O=C1CCC(N2C(=O)C3=CC=C(NCCCC4CCN(CCOC5=CC=C([C@H]6C7=CC=C(O)C=C7CC[C@H]6C6=CC=CC=C6)C=C5)CC4)C=C3C2=O)C(=O)N1	C45H48N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-233AVI	WO2018102725A1_43	.	O=C1CCC(N2C(=O)C3=CC=C(NCCCC4CCN(CCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)C=C3C2=O)C(=O)N1	C45H48N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-I98LU2	WO2018102725A1_44	.	O=C1CCC(N2CC3=CC(NCCCC4CCN(CCOC5=CC=C([C@H]6C7=CC=C(O)C=C7CCC6C6=CC=CC=C6)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C45H50N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-KDTK7J	WO2018102725A1_45	.	O=C1CCC(N2CC3=CC(NCCCC4CCN(CCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C45H50N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-G3RAJA	WO2018102725A1_46	.	O=C1CCC(N2C(=O)C3=CC=C(NCC4CCN(CCOC5=CC=C([C@H]6C7=CC=C(O)C=C7CC[C@H]6C6=CC=CC=C6)C=C5)CC4)C=C3C2=O)C(=O)N1	C43H44N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-MA9RFQ	WO2018102725A1_47	.	O=C1CCC(N2C(=O)C3=CC=C(NCC4CCN(CCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)C=C3C2=O)C(=O)N1	C43H44N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-T91S51	SCHEMBL20231776	3-[6-[[1-[2-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]ethyl]piperidin-4-yl]amino]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(NC4CCN(CCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C42H44N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-EVPIUI	WO2018102725A1_49	.	O=C1CCC(N2C(=O)C3=CC=C(NC4CCN(CCOC5=CC=C([C@H]6C7=CC=C(O)C=C7CC[C@H]6C6=CC=CC=C6)C=C5)CC4)C=C3C2=O)C(=O)N1	C42H42N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-MUTYBF	WO2018102725A1_50	.	O=C1CCC(N2C(=O)C3=CC=C(NC4CCN(CCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)C=C3C2=O)C(=O)N1	C42H42N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-EVIPTH	WO2018102725A1_51	.	O=C1CC[C@H](N2CC3=C(C=CC(OCCN4C[C@@H]5C[C@H]4CN5CCOC4=CC=C([C@H]5C6=CC=C(O)C=C6CC[C@H]5C5=CC=CC=C5)C=C4)=C3)C2=O)C(=O)N1	C44H46N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-0I6DE8	WO2018102725A1_52	.	O=C1CC[C@H](N2CC3=C(C=CC(OCCN4C[C@@H]5C[C@H]4CN5CCOC4=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=CC=C5)C=C4)=C3)C2=O)C(=O)N1	C44H46N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-T3WS99	WO2018102725A1_53	.	O=C1CCC(N2CC3=CC(CCCOC4CCN(CCOC5=CC=C([C@H]6C7=CC=C(O)C=C7CC[C@H]6C6=CC=CC=C6)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C45H49N3O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-8BM51G	SCHEMBL21982882	3-[6-[3-[1-[2-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]ethyl]piperidin-4-yl]oxypropyl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(CCCOC4CCN(CCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C45H49N3O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-6UXYRY	WO2018102725A1_55	.	O=C1CCC(N2C(=O)C3=CC=C(CCCOC4CCN(CCOC5=CC=C([C@H]6C7=CC=C(O)C=C7CC[C@H]6C6=CC=CC=C6)C=C5)CC4)C=C3C2=O)C(=O)N1	C45H47N3O7	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-TJA1EE	WO2018102725A1_56	.	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCCCCOC5=CC=C(C6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)C=C3C2=O)C(=O)N1	C44H46N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-GZ5YAD	WO2018102725A1_57	.	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCCCCCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)C=C3C2=O)C(=O)N1	C45H48N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-0RHO40	WO2018102725A1_58	.	O=C1CCC(N2CC3=CC(NC4CCN(CCOC5=CC=C([C@H]6C7=CC=C(O)C=C7CCC6C6=CC=CC=C6)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C42H44N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-17PDWZ	WO2018102725A1_59	.	O=C1CCC(N2CC3=CC(OCCCOCCCOC4=CC=C([C@H]5C6=CC=C(O)C=C6CC[C@H]5C5=CC=CC=C5)C=C4)=CC=C3C2=O)C(=O)N1	C41H42N2O7	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-UEGE2H	SCHEMBL20231626	3-[6-[3-[3-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]propoxy]propoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(OCCCOCCCOC4=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=CC=C5)C=C4)=CC=C3C2=O)C(=O)N1	C41H42N2O7	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-FGH1BT	WO2018102725A1_61	.	O=C1CCC(N2CC3=CC(N4CCN(CCCCCOC5=CC=C([C@H]6C7=CC=C(O)C=C7CC[C@H]6C6=CC=CC=C6)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C44H48N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-PIRS8N	SCHEMBL20211908	3-[6-[4-[5-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]pentyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(N4CCN(CCCCCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C44H48N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-KMHXV5	WO2018102725A1_63	.	O=C1CCC(N2C(=O)C3=CC=C(CCCOC4CCN(CCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)C=C3C2=O)C(=O)N1	C45H47N3O7	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-0Q7VRZ	WO2018102725A1_64	.	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCCCCCOC5=CC=C([C@H]6C7=CC=C(O)C=C7CC[C@H]6C6=CC=CC=C6)C=C5)CC4)C=C3C2=O)C(=O)N1	C45H48N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-C16ZT9	WO2018102725A1_66	.	O=C1CCC(N2CC3=CC(N4CCN(CCCCCCOC5=CC=C([C@H]6C7=CC=C(O)C=C7CC[C@H]6C6=CC=CC=C6)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C45H50N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-62QN8U	WO2018102725A1_67	.	O=C1CCC(N2CC3=CC(N4CCN(CCCCCCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C45H50N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-CWWC5B	WO2018102725A1_68	.	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCCCCOC5=CC=C([C@H]6C7=CC=C(O)C=C7CC[C@H]6C6=CC=CC=C6)C=C5)CC4)C=C3C2=O)C(=O)N1	C44H46N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-S60OUY	SCHEMBL20211897	2-(2,6-dioxopiperidin-3-yl)-5-[4-[5-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]pentyl]piperazin-1-yl]isoindole-1,3-dione; SCHEMBL30591782	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCCCCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)C=C3C2=O)C(=O)N1	C44H46N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-Z5MVUZ	WO2018102725A1_70	.	O=C1CC[C@@H](N2CC3=CC(OCCCCOCCCOC4=CC=C([C@H]5C6=CC=C(O)C=C6CC[C@H]5C5=CC=CC=C5)C=C4)=CC=C3C2=O)C(=O)N1	C42H44N2O7	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-V8MZIO	WO2018102725A1_71	.	O=C1CC[C@@H](N2CC3=CC(OCCCCOCCCOC4=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=CC=C5)C=C4)=CC=C3C2=O)C(=O)N1	C42H44N2O7	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-DED6WQ	WO2018102725A1_72	(3S)-3-[6-[6-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]hexa-2,4-diynoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CC[C@H](N2CC3=C(C=CC(OCC#CC#CCOC4=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=CC=C5)C=C4)=C3)C2=O)C(=O)N1	C41H34N2O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-HTUHQU	WO2018102725A1_73	.	O=C1CCC(N2CC3=CC(N4CCN(CCCOC5=CC=C([C@H]6C7=CC=C(O)C=C7CC[C@H]6C6=CC=CC=C6)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C42H44N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-8DWL4C	WO2018102725A1_74	.	O=C1CCC(N2CC3=CC(N4CCN(CCCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C42H44N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-DC21MU	WO2018102725A1_75	.	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCCOC5=CC=C([C@H]6C7=CC=C(O)C=C7CC[C@H]6C6=CC=CC=C6)C=C5)CC4)C=C3C2=O)C(=O)N1	C42H42N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-OSMM8E	WO2018102725A1_76	.	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)C=C3C2=O)C(=O)N1	C42H42N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-XK0AMS	WO2018102725A1_77	.	O=C1CC[C@H](N2CC3=C(C=CC(OCCN4CCCN(CCOC5=CC=C([C@H]6C7=CC=C(O)C=C7CC[C@H]6C6=CC=CC=C6)C=C5)CC4)=C3)C2=O)C(=O)N1	C44H48N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-5QCKLN	WO2018102725A1_78	.	O=C1CC[C@H](N2CC3=C(C=CC(OCCN4CCCN(CCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)=C3)C2=O)C(=O)N1	C44H48N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-SNF2EZ	WO2018102725A1_79	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(OCCCN4CCN(CCOC5=CC=C([C@H]6C7=CC=C(O)C=C7CC[C@H]6C6=CC=CC=C6)C=C5)CC4)=NO3)C(C)C)C=C2)SC=N1	C55H64N6O7S	ERα;ERβ	P03372/Q92731	VHL	WO-2018102725-A1
TPD-61JYM8	SCHEMBL20234713	(2S,4R)-4-hydroxy-1-[2-[3-[3-[4-[2-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]ethyl]piperazin-1-yl]propoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(OCCCN4CCN(CCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)=NO3)C(C)C)C=C2)SC=N1	C55H64N6O7S	ERα;ERβ	P03372/Q92731	VHL	WO-2018102725-A1
TPD-PKV8DW	WO2018102725A1_81	.	O=C1CCC(N2C(=O)C3=CC=C(OCCCCCN4CCN(C5=CC=C([C@H]6C7=CC=C(O)C=C7CC[C@H]6C6=CC=CC=C6)C=C5)CC4)C=C3C2=O)C(=O)N1	C44H46N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-XTL94C	WO2018102725A1_82	.	O=C1CCC(N2C(=O)C3=CC=C(OCCCCCN4CCN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)C=C3C2=O)C(=O)N1	C44H46N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-4MFXFS	WO2018102725A1_83	.	O=C1CCC(N2CC3=CC(OCCCCCN4CCN(C5=CC=C([C@H]6C7=CC=C(O)C=C7CC[C@H]6C6=CC=CC=C6)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C44H48N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-FEJSIX	SCHEMBL20234387	3-[6-[5-[4-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperazin-1-yl]pentoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(OCCCCCN4CCN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C44H48N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-5GOYF5	WO2018102725A1_85	.	O=C1CCC(N2C(=O)C3=CC=C(OCCCCN4CCN(C5=CC=C([C@H]6C7=CC=C(O)C=C7CC[C@H]6C6=CC=CC=C6)C=C5)CC4)C=C3C2=O)C(=O)N1	C43H44N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-K1HHXQ	SCHEMBL20234950	2-(2,6-dioxopiperidin-3-yl)-5-[4-[4-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperazin-1-yl]butoxy]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC=C(OCCCCN4CCN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)C=C3C2=O)C(=O)N1	C43H44N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-33WLNQ	WO2018102725A1_87	.	O=C1CCC(N2CC3=CC(OCCCCN4CCN(C5=CC=C([C@H]6C7=CC=C(O)C=C7CC[C@H]6C6=CC=CC=C6)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C43H46N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-82TSZH	WO2018102725A1_88	.	O=C1CCC(N2CC3=CC(OCCCCN4CCN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C43H46N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-Z9P0W1	WO2018102725A1_89	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(OCCCN4CCN(CCOC5=CC=C([C@H]6C7=CC=C(O)C=C7CC[C@H]6C6=CC=CC=C6)C=C5)CC4)=NO3)C(C)C)C=C2)SC=N1	C55H64N6O7S	ERα;ERβ	P03372/Q92731	VHL	WO-2018102725-A1
TPD-YJJ99X	WO2018102725A1_90	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(OCCCN4CCN(CCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)=NO3)C(C)C)C=C2)SC=N1	C55H64N6O7S	ERα;ERβ	P03372/Q92731	VHL	WO-2018102725-A1
TPD-61RMU5	WO2018102725A1_91	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3=CC(OCCCN4CCN(CCOC5=CC=C([C@H]6C7=CC=C(O)C=C7CC[C@H]6C6=CC=CC=C6)C=C5)CC4)=NO3)C(C)C)C=C2)SC=N1	C55H64N6O7S	ERα;ERβ	P03372/Q92731	VHL	WO-2018102725-A1
TPD-HPV8AU	WO2018102725A1_92	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3=CC(OCCCN4CCN(CCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)=NO3)C(C)C)C=C2)SC=N1	C55H64N6O7S	ERα;ERβ	P03372/Q92731	VHL	WO-2018102725-A1
TPD-FE8BB1	WO2018102725A1_93	.	O=C1CCC(N2C(=O)C3=CC=C(NCCCCCN4CCN(C5=CC=C([C@H]6C7=CC=C(O)C=C7CC[C@H]6C6=CC=CC=C6)C=C5)CC4)C=C3C2=O)C(=O)N1	C44H47N5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-7LV4R0	WO2018102725A1_94	.	O=C1CCC(N2C(=O)C3=CC=C(NCCCCCN4CCN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)C=C3C2=O)C(=O)N1	C44H47N5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-3XS9YX	WO2018102725A1_95	.	O=C1CCC(N2C(=O)C3=CC=C(NCCCCN4CCN(C5=CC=C([C@H]6C7=CC=C(O)C=C7CC[C@H]6C6=CC=CC=C6)C=C5)CC4)C=C3C2=O)C(=O)N1	C43H45N5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-ENI833	WO2018102725A1_96	.	O=C1CC[C@H](N2C(=O)C3=CC=C(NCCCCN4CCN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)C=C3C2=O)C(=O)N1	C43H45N5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-9EZ7S3	WO2018102725A1_97	.	O=C(CN1CCN(CCOC2=CC=C([C@H]3C4=C(C=C(O)C=C4)CC[C@H]3C3=CC=CC=C3)C=C2)CC1)NCC1=CC=C2C(=O)N(C3CCC(=O)NC3=O)CC2=C1	C44H47N5O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-P0SUC7	SCHEMBL20234927	N-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]methyl]-2-[4-[2-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]ethyl]piperazin-1-yl]acetamide	O=C(CN1CCN(CCOC2=CC=C([C@@H]3C4=C(C=C(O)C=C4)CC[C@@H]3C3=CC=CC=C3)C=C2)CC1)NCC1=CC=C2C(=O)N(C3CCC(=O)NC3=O)CC2=C1	C44H47N5O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-ADLPNZ	WO2018102725A1_99	.	O=C1CC[C@H](N2CC3=C(C=CC(OCCCOCCCOCCCOC4=CC=C([C@H]5C6=CC=C(O)C=C6CC[C@H]5C5=CC=CC=C5)C=C4)=C3)C2=O)C(=O)N1	C44H48N2O8	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-HOWZ9N	WO2018102725A1_100	.	O=C1CC[C@H](N2CC3=C(C=CC(OCCCOCCCOCCCOC4=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=CC=C5)C=C4)=C3)C2=O)C(=O)N1	C44H48N2O8	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-6HJXBA	WO2018102725A1_101	.	O=C1CC[C@H](N2CC3=C(C=CC(OCCOCCOCCOC4=CC=C([C@H]5C6=CC=C(O)C=C6CC[C@H]5C5=CC=CC=C5)C=C4)=C3)C2=O)C(=O)N1	C41H42N2O8	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-AM37AF	WO2018102725A1_102	.	O=C1CC[C@H](N2CC3=C(C=CC(OCCOCCOCCOC4=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=CC=C5)C=C4)=C3)C2=O)C(=O)N1	C41H42N2O8	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-MM5LR1	WO2018102725A1_103	.	O=C1CC[C@H](N2CC3=C(C=CC(OCCCOCCOCCOC4=CC=C([C@H]5C6=CC=C(O)C=C6CC[C@H]5C5=CC=CC=C5)C=C4)=C3)C2=O)C(=O)N1	C42H44N2O8	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-5IQ3W5	WO2018102725A1_104	.	O=C1CC[C@H](N2CC3=C(C=CC(OCCCOCCOCCOC4=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=CC=C5)C=C4)=C3)C2=O)C(=O)N1	C42H44N2O8	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-FHH3TU	SCHEMBL20231329	(3S)-3-[6-[2-[(3S)-1-[2-[4-[(1S,2R)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]ethyl]piperidin-3-yl]ethoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CC[C@H](N2CC3=CC(OCC[C@@H]4CCCN(CCOC5=CC=C([C@H]6C7=CC=C(O)C=C7CC[C@H]6C6=CC=CC=C6)C=C5)C4)=CC=C3C2=O)C(=O)N1	C44H47N3O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-1PKMU8	SCHEMBL20234693	(3S)-3-[6-[2-[(3R)-1-[2-[4-[(1S,2R)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]ethyl]piperidin-3-yl]ethoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CC[C@H](N2CC3=CC(OCC[C@H]4CCCN(CCOC5=CC=C([C@H]6C7=CC=C(O)C=C7CC[C@H]6C6=CC=CC=C6)C=C5)C4)=CC=C3C2=O)C(=O)N1	C44H47N3O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-R7ULCX	WO2018102725A1_107	.	O=C1CC[C@H](N2CC3=CC(C4=CC=C(NCCCCOC5=CC=C([C@H]6C7=CC=C(O)C=C7CC[C@H]6C6=CC=CC=C6)C=C5)C=C4)=CC=C3C2=O)C(=O)N1	C45H43N3O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-29E6C9	SCHEMBL20234973	(3S)-3-[6-[4-[4-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]butylamino]phenyl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CC[C@H](N2CC3=CC(C4=CC=C(NCCCCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)C=C4)=CC=C3C2=O)C(=O)N1	C45H43N3O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-S3HH0Q	WO2018102725A1_109	.	O=C1CC[C@H](N2CC3=CC(OCCOCCOC4=CC=C([C@H]5C6=CC=C(O)C=C6CC[C@H]5C5=CC=CC=C5)C=C4)=CC=C3C2=O)C(=O)N1	C39H38N2O7	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-SX78TO	WO2018102725A1_110	.	O=C1CC[C@H](N2CC3=CC(OCCOCCOC4=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=CC=C5)C=C4)=CC=C3C2=O)C(=O)N1	C39H38N2O7	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-0Q5KJT	WO2018102725A1_111	.	O=C1CCC(N2C(=O)C3=CC=C(OCCOCCOC4=CC=C([C@H]5C6=CC=C(O)C=C6CC[C@H]5C5=CC=CC=C5)C=C4)C=C3C2=O)C(=O)N1	C39H36N2O8	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-GOH8E5	SCHEMBL20234469	2-(2,6-dioxopiperidin-3-yl)-5-[2-[2-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]ethoxy]ethoxy]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC=C(OCCOCCOC4=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=CC=C5)C=C4)C=C3C2=O)C(=O)N1	C39H36N2O8	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-X0SHUH	WO2018102725A1_113	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCN3CCN(CCOC4=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=C(F)C=C5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C54H65FN6O7S	ERα;ERβ	P03372/Q92731	VHL	WO-2018102725-A1
TPD-GR6VJG	WO2018102725A1_114	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCN3CCN(CCOC4=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=C(C(F)(F)F)C=C5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C55H65F3N6O7S	ERα;ERβ	P03372/Q92731	VHL	WO-2018102725-A1
TPD-U8FJRY	WO2018102725A1_115	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCN3C[C@H](C)N(CCOC4=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=C(F)C=C5)C=C4)C[C@H]3C)C(C)(C)C)C=C2)SC=N1	C56H69FN6O7S	ERα;ERβ	P03372/Q92731	VHL	WO-2018102725-A1
TPD-3CFZOH	WO2018102725A1_116	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCN3[C@H](C)CN(CCOC4=CC=C(C5C6=CC=C(O)C=C6CCN5C5=CC=C(F)C=C5)C=C4)C[C@@H]3C)C(C)(C)C)C=C2)SC=N1	C55H68FN7O7S	ERα;ERβ	P03372/Q92731	VHL	WO-2018102725-A1
TPD-LWCPWP	WO2018102725A1_117	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCN3CCN(CCOC4=CC=C(C5C6=CC=C(O)C=C6CCN5C5=C(F)C=C(F)C=C5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C53H63F2N7O7S	ERα;ERβ	P03372/Q92731	VHL	WO-2018102725-A1
TPD-FL383T	WO2018102725A1_118	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCN3CCN(CCOC4=CC=C(C5C6=CC=C(O)C=C6CCN5C5=CC=C(C(F)(F)F)C=C5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C54H64F3N7O7S	ERα;ERβ	P03372/Q92731	VHL	WO-2018102725-A1
TPD-CVI64G	WO2018102725A1_119	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCN3CC4(C3)CN(CCOC3=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=C(C(F)(F)F)C=C5)C=C3)C4)C(C)(C)C)C=C2)SC=N1	C56H65F3N6O7S	ERα;ERβ	P03372/Q92731	VHL	WO-2018102725-A1
TPD-NEN2O5	WO2018102725A1_120	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCN3CC4(C3)CN(CCOC3=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=C(F)C=C5)C=C3)C4)C(C)(C)C)C=C2)SC=N1	C55H65FN6O7S	ERα;ERβ	P03372/Q92731	VHL	WO-2018102725-A1
TPD-AFKFV9	WO2018102725A1_121	.	C[C@@H]1CN(CCCCCOC2=CC=C([C@@H]3C4=CC=C(O)C=C4CC[C@@H]3C3=CC=CC=C3)C=C2)[C@@H](C)CN1C1=CC=C2C(=O)N(C3CCC(=O)NC3=O)CC2=C1	C46H52N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-70KJJ4	WO2018102725A1_122	.	O=C1CCC(N2CC3=CC(N4CCN(CCCCCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=C(Br)C=C6)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C44H47BrN4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-P4POM3	WO2018102725A1_123	.	O=C1CCC(N2CC3=CC(N4CCN(CCCCCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=C(C(F)(F)F)C=C6)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C45H47F3N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-HZLUXG	WO2018102725A1_124	.	O=C1CCC(N2CC3=CC(N4CCN(CCCCCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=C(F)C=C(F)C=C6)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C44H46F2N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-5GAP5P	WO2018102725A1_125	.	O=C1CCC(N2CC3=CC(N4CCN(CCCCCOC5=CC=CC([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)=C5)CC4)=CC=C3C2=O)C(=O)N1	C44H48N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-8A3TXO	WO2018102725A1_126	.	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCCCCOC5=CC([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)=CC=C5)CC4)C=C3C2=O)C(=O)N1	C44H46N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-XCR4Y5	SCHEMBL20234935	2-(2,6-dioxopiperidin-3-yl)-5-[4-[5-[3-[(1R,2S)-2-(4-fluorophenyl)-6-hydroxy-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]pentyl]piperazin-1-yl]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCCCCOC5=CC([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=C(F)C=C6)=CC=C5)CC4)C=C3C2=O)C(=O)N1	C44H45FN4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-AESTJ6	SCHEMBL21982917	3-[6-[4-[5-[3-[(1R,2S)-2-(4-fluorophenyl)-6-hydroxy-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]pentyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(N4CCN(CCCCCOC5=CC=CC([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=C(F)C=C6)=C5)CC4)=CC=C3C2=O)C(=O)N1	C44H47FN4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-K5X2WT	WO2018102725A1_129	.	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCCCCOC5=CC([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=C(C(F)(F)F)C=C6)=CC=C5)CC4)C=C3C2=O)C(=O)N1	C45H45F3N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-SNIT29	WO2018102725A1_130	.	O=C1CCC(N2CC3=CC(N4CCN(CCCCCOC5=CC=CC([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=C(C(F)(F)F)C=C6)=C5)CC4)=CC=C3C2=O)C(=O)N1	C45H47F3N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-A8OE38	WO2018102725A1_131	.	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCCCCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=C(F)C=C(F)C=C6)C=C5)CC4)C=C3C2=O)C(=O)N1	C44H44F2N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-J0SMPG	WO2018102725A1_132	.	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCCCCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=C(C(F)(F)F)C=C6)C=C5)CC4)C=C3C2=O)C(=O)N1	C45H45F3N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-Q97FQE	WO2018102725A1_133	.	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(C[C@H]5CC[C@H](OC6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=C(F)C=C7)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C46H47FN4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-X0P7GE	WO2018102725A1_134	.	O=C1CCC(N2CC3=CC(N4CCN(C[C@H]5CC[C@H](OC6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=C(F)C=C7)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C46H49FN4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-NHAWBD	WO2018102725A1_135	.	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(C[C@H]5CC[C@H](OC6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=C(C(F)(F)F)C=C7)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C47H47F3N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-DBHJ9E	WO2018102725A1_136	.	O=C1CCC(N2CC3=CC(N4CCN(C[C@H]5CC[C@H](OC6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=C(C(F)(F)F)C=C7)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C47H49F3N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-6GXGWM	WO2018102725A1_137	.	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCO[C@H]5CC[C@H](OC6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=C(F)C=C7)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C47H49FN4O7	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-3C8CI0	WO2018102725A1_138	.	O=C1CCC(N2CC3=CC(N4CCN(CCO[C@H]5CC[C@H](OC6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=C(F)C=C7)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C47H51FN4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-XNF1KP	WO2018102725A1_139	.	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCO[C@H]5CC[C@H](OC6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=C(C(F)(F)F)C=C7)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C48H49F3N4O7	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-UUQZNS	WO2018102725A1_140	.	O=C1CCC(N2CC3=CC(N4CCN(CCO[C@H]5CC[C@H](OC6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=C(C(F)(F)F)C=C7)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C48H51F3N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-5ULVAY	WO2018102725A1_141	(3S)-3-[6-[2-[[2-[2-[4-[(1S,2R)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]ethyl]-2-azaspiro[3.3]heptan-6-yl]oxy]ethoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CC[C@H](N2CC3=C(C=CC(OCCOC4CC5(C4)CN(CCOC4=CC=C([C@H]6C7=CC=C(O)C=C7CC[C@H]6C6=CC=CC=C6)C=C4)C5)=C3)C2=O)C(=O)N1	C45H47N3O7	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-KJQIFQ	WO2018102725A1_142	.	O=C1CCC(N2CC3=CC(NCCCCN4CCN(C5=CC=C([C@H]6C7=CC=C(O)C=C7CC[C@H]6C6=CC=CC=C6)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C43H47N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-G9II0W	WO2018102725A1_143	.	O=C1CCC(N2CC3=CC(NCCCCN4CCN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C43H47N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-IWXSAN	WO2018102725A1_144	.	O=C1CC[C@H](N2CC3=CC(OCCC4CCCN(CCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)C4)=CC=C3C2=O)C(=O)N1	C44H47N3O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-IJZLI8	WO2018102725A1_145	.	O=C1CC[C@H](N2CC3=CC(NCCOCCOC4=CC=C([C@H]5C6=CC=C(O)C=C6CC[C@H]5C5=CC=CC=C5)C=C4)=CC=C3C2=O)C(=O)N1	C39H39N3O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-694Z42	WO2018102725A1_146	.	O=C1CC[C@H](N2CC3=CC(NCCOCCOC4=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=CC=C5)C=C4)=CC=C3C2=O)C(=O)N1	C39H39N3O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-C5EEED	WO2018102725A1_147	.	O=C1CCC(N2C(=O)C3=CC=C(NCCOCCOC4=CC=C([C@H]5C6=CC=C(O)C=C6CC[C@H]5C5=CC=CC=C5)C=C4)C=C3C2=O)C(=O)N1	C39H37N3O7	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-321JYB	SCHEMBL20234468	2-(2,6-dioxopiperidin-3-yl)-5-[2-[2-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]ethoxy]ethylamino]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC=C(NCCOCCOC4=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=CC=C5)C=C4)C=C3C2=O)C(=O)N1	C39H37N3O7	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-25N404	WO2018102725A1_149	.	C[C@H](COC1=CC=C([C@H]2C3=CC=C(O)C=C3CC[C@H]2C2=CC=CC=C2)C=C1)N1CCN(CC(=O)NCC2=CC=C3C(=O)N(C4CCC(=O)NC4=O)CC3=C2)CC1	C45H49N5O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-ODX3PN	SCHEMBL20232005	N-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]methyl]-2-[4-[(2R)-1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]propan-2-yl]piperazin-1-yl]acetamide	C[C@H](COC1=CC=C([C@@H]2C3=CC=C(O)C=C3CC[C@@H]2C2=CC=CC=C2)C=C1)N1CCN(CC(=O)NCC2=CC=C3C(=O)N(C4CCC(=O)NC4=O)CC3=C2)CC1	C45H49N5O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-DDLO3O	WO2018102725A1_151	.	C[C@@H](COC1=CC=C([C@H]2C3=CC=C(O)C=C3CC[C@H]2C2=CC=CC=C2)C=C1)N1CCN(CC(=O)NCC2=CC=C3C(=O)N(C4CCC(=O)NC4=O)CC3=C2)CC1	C45H49N5O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-9HLXMV	WO2018102725A1_152	.	C[C@@H](COC1=CC=C([C@@H]2C3=CC=C(O)C=C3CC[C@@H]2C2=CC=CC=C2)C=C1)N1CCN(CC(=O)NCC2=CC=C3C(=O)N(C4CCC(=O)NC4=O)CC3=C2)CC1	C45H49N5O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-R5R1WM	WO2018102725A1_153	.	O=C1CCC(N2CC3=C(C=CC(CCCN4CCCN(CCCOC5=CC=C([C@H]6C7=CC=C(O)C=C7CC[C@H]6C6=CC=CC=C6)C=C5)CC4)=C3)C2=O)C(=O)N1	C46H52N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-QB5KEI	WO2018102725A1_154	.	O=C1CCC(N2CC3=C(C=CC(CCCN4CCCN(CCCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)=C3)C2=O)C(=O)N1	C46H52N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-4ZVJBG	WO2018102725A1_155	.	O=C1CCC(N2CC3=CC(NCCCCCN4CCN(C5=CC=C([C@H]6C7=CC=C(O)C=C7CC[C@H]6C6=CC=CC=C6)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C44H49N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-94ICBI	WO2018102725A1_156	.	O=C1CCC(N2CC3=CC(NCCCCCN4CCN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C44H49N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-4SQHTH	WO2018102725A1_157	.	O=C1CC[C@H](N2CC3=C(C=CC(OCCCOCCOC4=CC=C([C@H]5C6=CC=C(O)C=C6CC[C@H]5C5=CC=CC=C5)C=C4)=C3)C2=O)C(=O)N1	C40H40N2O7	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-2XX431	WO2018102725A1_158	.	O=C1CC[C@H](N2CC3=C(C=CC(OCCCOCCOC4=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=CC=C5)C=C4)=C3)C2=O)C(=O)N1	C40H40N2O7	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-ZZ18MF	WO2018102725A1_159	.	O=C1CCC(N2C(=O)C3=C(C=C(OCCCOCCOC4=CC=C([C@H]5C6=CC=C(O)C=C6CC[C@H]5C5=CC=CC=C5)C=C4)C=C3)C2=O)C(=O)N1	C40H38N2O8	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-MEYHJR	WO2018102725A1_160	.	O=C1CC[C@H](N2C(=O)C3=C(C=C(OCCCOCCOC4=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=CC=C5)C=C4)C=C3)C2=O)C(=O)N1	C40H38N2O8	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-9NB1V8	WO2018102725A1_161	.	O=C1CCC(N2CC3=C(C=CC(OCCCOCCCOCCOC4=CC=C([C@H]5C6=CC=C(O)C=C6CC[C@H]5C5=CC=CC=C5)C=C4)=C3)C2=O)C(=O)N1	C43H46N2O8	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-FH408O	WO2018102725A1_162	.	O=C1CCC(N2CC3=C(C=CC(OCCCOCCCOCCOC4=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=CC=C5)C=C4)=C3)C2=O)C(=O)N1	C43H46N2O8	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-IGNMJL	WO2018102725A1_163	.	O=C1CCC(N2CC3=C(C=CC(CCN4CCCN(CCCCOC5=CC=C([C@H]6C7=CC=C(O)C=C7CC[C@H]6C6=CC=CC=C6)C=C5)CC4)=C3)C2=O)C(=O)N1	C46H52N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-RVS501	SCHEMBL22006007	3-[6-[2-[4-[4-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]butyl]-1,4-diazepan-1-yl]ethyl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(CCN4CCCN(CCCCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)=C3)C2=O)C(=O)N1	C46H52N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-Q071TY	SCHEMBL20235049	(3S)-3-[6-[4-amino-3-[5-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]pentoxy]phenyl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	NC1=C(OCCCCCOC2=CC=C([C@@H]3C4=CC=C(O)C=C4CC[C@@H]3C3=CC=CC=C3)C=C2)C=C(C2=CC=C3C(=O)N([C@H]4CCC(=O)NC4=O)CC3=C2)C=C1	C46H45N3O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-KX5SJ3	WO2018102725A1_166	.	NC1=C(OCCCCOC2=CC=C([C@@H]3C4=CC=C(O)C=C4CC[C@@H]3C3=CC=CC=C3)C=C2)C=C(C2=CC=C3C(=O)N([C@H]4CCC(=O)NC4=O)CC3=C2)C=C1	C45H43N3O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-YILHH8	WO2018102725A1_167	.	O=C1CC[C@H](N2CC3=C(C=CC(NCCCOCCOC4=CC=C([C@H]5C6=CC=C(O)C=C6CC[C@H]5C5=CC=CC=C5)C=C4)=C3)C2=O)C(=O)N1	C40H41N3O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-CJO7YG	WO2018102725A1_168	.	O=C1CC[C@H](N2C(=O)C3=C(C=C(NCCCOCCOC4=CC=C([C@H]5C6=CC=C(O)C=C6CC[C@H]5C5=CC=CC=C5)C=C4)C=C3)C2=O)C(=O)N1	C40H39N3O7	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-BFA1BI	WO2018102725A1_169	.	O=C1CC[C@H](N2C(=O)C3=C(C=C(NCCCOCCOC4=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=CC=C5)C=C4)C=C3)C2=O)C(=O)N1	C40H39N3O7	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-KX36M0	WO2018102725A1_170	.	O=C1CC[C@H](N2CC3=C(C=CC(OCCCOCCCOCCCCOC4=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=CC=C5)C=C4)=C3)C2=O)C(=O)N1	C45H50N2O8	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-69R49M	SCHEMBL20231354	(3S)-3-[6-[3-[(3R)-1-[2-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]ethyl]piperidin-3-yl]propyl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CC[C@H](N2CC3=CC(CCC[C@@H]4CCCN(CCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)C4)=CC=C3C2=O)C(=O)N1	C45H49N3O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-BR9FK5	WO2018102725A1_172	.	O=C1CC[C@H](N2CC3=CC(CCC[C@H]4CCCN(CCOC5=CC=C([C@H]6C7=CC=C(O)C=C7CC[C@H]6C6=CC=CC=C6)C=C5)C4)=CC=C3C2=O)C(=O)N1	C45H49N3O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-Y9CDFN	SCHEMBL20235022	(3S)-3-[6-[3-[(3S)-1-[2-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]ethyl]piperidin-3-yl]propyl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CC[C@H](N2CC3=CC(CCC[C@H]4CCCN(CCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)C4)=CC=C3C2=O)C(=O)N1	C45H49N3O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-XSQOTI	WO2018102725A1_174	.	O=C1CC[C@H](N2CC3=CC(CCN4CCCN(CCOC5=CC=C([C@H]6C7=CC=C(O)C=C7CC[C@H]6C6=CC=CC=C6)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C44H48N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-GPTZER	WO2018102725A1_175	(3S)-3-[6-[2-[4-[2-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]ethyl]-1,4-diazepan-1-yl]ethyl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CC[C@H](N2CC3=CC(CCN4CCCN(CCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C44H48N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-1JR1NR	WO2018102725A1_176	.	O=C1CC[C@H](N2CC3=CC(C4=CC5=C(C=C4)NC(CCCOC4=CC=C([C@H]6C7=CC=C(O)C=C7CC[C@H]6C6=CC=CC=C6)C=C4)=C5)=CC=C3C2=O)C(=O)N1	C46H41N3O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-ZNVFZS	SCHEMBL20231544	(3S)-3-[6-[2-[3-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]propyl]-1H-indol-5-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CC[C@H](N2CC3=CC(C4=CC5=C(C=C4)NC(CCCOC4=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C4)=C5)=CC=C3C2=O)C(=O)N1	C46H41N3O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-0JRVAI	WO2018102725A1_178	.	O=C1CC[C@H](N2CC3=CC(C4=CC5=C(C=C4)NC(CCCCOC4=CC=C([C@H]6C7=CC=C(O)C=C7CC[C@H]6C6=CC=CC=C6)C=C4)=C5)=CC=C3C2=O)C(=O)N1	C47H43N3O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-BF4ZVA	WO2018102725A1_179	.	O=C1CC[C@H](N2CC3=CC(C4=CC5=C(C=C4)NC(CCCCOC4=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C4)=C5)=CC=C3C2=O)C(=O)N1	C47H43N3O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-PRG6CB	WO2018102725A1_180	.	O=C1CC[C@H](N2CC3=CC(C4=CC5=C(C=C4)NC=C5CCCCCOC4=CC=C([C@H]5C6=CC=C(O)C=C6CC[C@H]5C5=CC=CC=C5)C=C4)=CC=C3C2=O)C(=O)N1	C48H45N3O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-0ZP30J	SCHEMBL20234987	(3S)-3-[6-[3-[5-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]pentyl]-1H-indol-5-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CC[C@H](N2CC3=CC(C4=CC5=C(C=C4)NC=C5CCCCCOC4=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=CC=C5)C=C4)=CC=C3C2=O)C(=O)N1	C48H45N3O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-I3UH4M	WO2018102725A1_182	.	O=C1CC[C@H](N2CC3=C(C=CC(NCCCOCCOC4=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=CC=C5)C=C4)=C3)C2=O)C(=O)N1	C40H41N3O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-EEFMKX	WO2018102725A1_183	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCCCCOC5=CC=C([C@H]6C7=C(C=C(O)C=C7)CC[C@H]6C6=CC=C(F)C=C6)C=C5)CC4)=C3)C2=O)C(=O)N1	C44H47FN4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-WPO527	WO2018102725A1_184	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCCCCOC5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=C(F)C=C6)C=C5)CC4)=C3)C2=O)C(=O)N1	C44H47FN4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-294AAJ	WO2018102725A1_185	.	O=C1CCC(N2C(=O)C3=C(C=C(N4CCN(CCCCCOC5=CC=C([C@H]6C7=C(C=C(O)C=C7)CC[C@H]6C6=CC=C(F)C=C6)C=C5)CC4)C=C3)C2=O)C(=O)N1	C44H45FN4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-TYZP2O	WO2018102725A1_186	.	O=C1CCC(N2C(=O)C3=C(C=C(N4CCN(CCCCCOC5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=C(F)C=C6)C=C5)CC4)C=C3)C2=O)C(=O)N1	C44H45FN4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-6AN6RR	SCHEMBL20231318	(3S)-3-[6-[2-[1-[3-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]propyl]piperidin-3-yl]oxyethyl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CC[C@H](N2CC3=CC(CCOC4CCCN(CCCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)C4)=CC=C3C2=O)C(=O)N1	C45H49N3O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-M7W2EB	WO2018102725A1_188	.	O=C1CC[C@H](N2CC3=CC(CCOC4CCCN(CCCOC5=CC=C([C@H]6C7=CC=C(O)C=C7CC[C@H]6C6=CC=CC=C6)C=C5)C4)=CC=C3C2=O)C(=O)N1	C45H49N3O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-91HC5X	WO2018102725A1_189	.	O=C1CC[C@H](N2CC3=CC(CCOC4CCCN(CCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)C4)=CC=C3C2=O)C(=O)N1	C44H47N3O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-Z8K8Z7	WO2018102725A1_190	.	CN(CCOCC1=CC=C([C@H]2C3=CC=C(O)C=C3CC[C@H]2C2=CC=CC=C2)C=C1)[C@H]1CC[C@H](C2=CC=C3C(=O)N([C@H]4CCC(=O)NC4=O)CC3=C2)CC1	C45H49N3O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-DRV2KB	SCHEMBL20231323	(3S)-3-[6-[4-[2-[[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]methoxy]ethyl-methylamino]cyclohexyl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CN(CCOCC1=CC=C([C@@H]2C3=CC=C(O)C=C3CC[C@@H]2C2=CC=CC=C2)C=C1)[C@H]1CC[C@H](C2=CC=C3C(=O)N([C@H]4CCC(=O)NC4=O)CC3=C2)CC1	C45H49N3O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-517O2K	WO2018102725A1_192	.	O=C1CCC(N2CC3=CC(N4CCCN(CCCCCOC5=CC=C([C@H]6C7=CC=C(O)C=C7CC[C@H]6C6=CC=CC=C6)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C45H50N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-EKXDS4	WO2018102725A1_193	.	O=C1CCC(N2CC3=CC(N4CCCN(CCCCCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C45H50N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-HW75UE	WO2018102725A1_194	.	O=C1CCC(N2C(=O)C3=CC=C(N4CCCN(CCCCCOC5=CC=C([C@H]6C7=CC=C(O)C=C7CC[C@H]6C6=CC=CC=C6)C=C5)CC4)C=C3C2=O)C(=O)N1	C45H48N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-33AALU	WO2018102725A1_195	.	O=C1CCC(N2C(=O)C3=CC=C(N4CCCN(CCCCCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)C=C3C2=O)C(=O)N1	C45H48N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-XJMX02	WO2018102725A1_196	.	O=C1CCC(N2CC3=CC(N4CCCN(CCCCOC5=CC=C([C@H]6C7=CC=C(O)C=C7CC[C@H]6C6=CC=CC=C6)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C44H48N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-E3208Z	WO2018102725A1_197	.	O=C1CCC(N2CC3=CC(N4CCCN(CCCCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C44H48N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-MH3BO1	WO2018102725A1_198	.	O=C1CCC(N2C(=O)C3=CC=C(N4CCCN(CCCCOC5=CC=C([C@H]6C7=CC=C(O)C=C7CC[C@H]6C6=CC=CC=C6)C=C5)CC4)C=C3C2=O)C(=O)N1	C44H46N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-7V5LV7	WO2018102725A1_199	.	O=C1CCC(N2C(=O)C3=CC=C(N4CCCN(CCCCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)C=C3C2=O)C(=O)N1	C44H46N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-MVAOMO	SCHEMBL20231981	3-[6-[4-[2-[(1S,2R)-2-[[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]methyl]cyclopropyl]ethyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC[C@@H]5C[C@H]5COC5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)=C3)C2=O)C(=O)N1	C45H48N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-F6PH2K	WO2018102725A1_201	.	O=C1CCC(N2C(=O)C3=C(C=C(N4CCN(CC[C@H]5C[C@@H]5COC5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)C=C3)C2=O)C(=O)N1	C45H46N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-GFT7II	WO2018102725A1_202	.	O=C1CCC(N2C(=O)C3=C(C=C(N4CCN(CC[C@@H]5C[C@H]5COC5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)C=C3)C2=O)C(=O)N1	C45H46N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-F4KF61	WO2018102725A1_203	.	O=C1CCC(N2C(=O)C3=CC=C(N4CCC(CN5CCC(OC6=CC=C([C@H]7C8=C(C=C(O)C=C8)CC[C@H]7C7=CC=CC=C7)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C46H48N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-2326Z1	SCHEMBL20234719	2-(2,6-dioxopiperidin-3-yl)-5-[4-[[4-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]piperidin-1-yl]methyl]piperidin-1-yl]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC=C(N4CCC(CN5CCC(OC6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C46H48N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-AZFR9H	WO2018102725A1_205	.	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(C5CCN(CCOC6=CC=C([C@H]7C8=CC=C(O)C=C8CC[C@H]7C7=CC=CC=C7)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C46H49N5O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-CS2H1X	SCHEMBL21982884	2-(2,6-dioxopiperidin-3-yl)-5-[4-[1-[2-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]ethyl]piperidin-4-yl]piperazin-1-yl]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(C5CCN(CCOC6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C46H49N5O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-ZFJPM2	WO2018102725A1_207	.	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CC5CCN(CCOC6=CC=C([C@H]7C8=CC=C(O)C=C8CC[C@H]7C7=CC=CC=C7)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C47H51N5O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-JHWX8J	WO2018102725A1_208	.	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CC5CCN(CCOC6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C47H51N5O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-H5S9C8	WO2018102725A1_209	.	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CC5CN(CCOC6=CC=C([C@H]7C8=CC=C(O)C=C8CC[C@H]7C7=CC=CC=C7)C=C6)C5)CC4)C=C3C2=O)C(=O)N1	C45H47N5O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-6L1OCN	SCHEMBL20231273	2-(2,6-dioxopiperidin-3-yl)-5-[4-[[1-[2-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]ethyl]azetidin-3-yl]methyl]piperazin-1-yl]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CC5CN(CCOC6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=CC=C7)C=C6)C5)CC4)C=C3C2=O)C(=O)N1	C45H47N5O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-X3DCAA	WO2018102725A1_211	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC[C@H]5C[C@H]5COC5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=C(F)C=C6)C=C5)CC4)=C3)C2=O)C(=O)N1	C45H47FN4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-PXSMUR	WO2018102725A1_212	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC[C@@H]5C[C@@H]5COC5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=C(F)C=C6)C=C5)CC4)=C3)C2=O)C(=O)N1	C45H47FN4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-MCDFQT	WO2018102725A1_213	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCCC(F)(F)COC5=CC=C([C@H]6C7=C(C=C(O)C=C7)CC[C@H]6C6=CC=CC=C6)C=C5)CC4)=C3)C2=O)C(=O)N1	C44H46F2N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-QUX91G	SCHEMBL20231267	3-[6-[4-[4,4-difluoro-5-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]pentyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; DLOJSADPWFQRKI-CONNHYNKSA-N; 3-[6-[4-[4,4-difluoro-5-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]pentyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCCC(F)(F)COC5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)=C3)C2=O)C(=O)N1	C44H46F2N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-5E2J68	WO2018102725A1_215	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC[C@H]5C[C@@H]5COC5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)=C3)C2=O)C(=O)N1	C45H48N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-62UOK7	WO2018102725A1_216	.	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCC5CN(CCOC6=CC=C([C@H]7C8=CC=C(O)C=C8CC[C@H]7C7=CC=CC=C7)C=C6)C5)CC4)C=C3C2=O)C(=O)N1	C46H49N5O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-7D9GV1	WO2018102725A1_217	.	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCC5CN(CCOC6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=CC=C7)C=C6)C5)CC4)C=C3C2=O)C(=O)N1	C46H49N5O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-CMSEZ0	SCHEMBL20231781	2-(2,6-dioxopiperidin-3-yl)-5-[4-[5-[4-[(1R,2S)-2-(4-fluorophenyl)-6-hydroxy-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]-1,2,3,3a,4,5,6,6a-octahydropentalen-2-yl]piperazin-1-yl]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=C(C=C(N4CCN(C5CC6CC(OC7=CC=C([C@@H]8C9=CC=C(O)C=C9CC[C@@H]8C8=CC=C(F)C=C8)C=C7)CC6C5)CC4)C=C3)C2=O)C(=O)N1	C47H47FN4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-YL10PI	WO2018102725A1_219	.	CN1C(=O)CCC(N2CC3=C(C=CC(N4CCN(CCCCCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)=C3)C2=O)C1=O	C45H50N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-TV078A	WO2018102725A1_220	.	CN1C(=O)CCC(N2CC3=C(C=CC(N4CCN(CCCCCOC5=CC=C([C@H]6C7=CC=C(O)C=C7CC[C@H]6C6=CC=CC=C6)C=C5)CC4)=C3)C2=O)C1=O	C45H50N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-YAPZB1	WO2018102725A1_221	.	O=C1CCC(N2CC3=C(C=CC(C4=CN=C(O[C@H]5CCN(CCOC6=CC=C([C@H]7C8=CC=C(O)C=C8CC[C@H]7C7=CC=CC=C7)C=C6)C5)C=C4)=C3)C2=O)C(=O)N1	C46H44N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-OB154R	WO2018102725A1_222	.	O=C1CCC(N2CC3=C(C=CC(C4=CN=C(O[C@@H]5CCN(CCOC6=CC=C([C@H]7C8=CC=C(O)C=C8CC[C@H]7C7=CC=CC=C7)C=C6)C5)C=C4)=C3)C2=O)C(=O)N1	C46H44N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-3ISWAD	SCHEMBL20234478	3-[6-[6-[(3R)-1-[2-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]ethyl]pyrrolidin-3-yl]oxypyridin-3-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(C4=CN=C(O[C@@H]5CCN(CCOC6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=CC=C7)C=C6)C5)C=C4)=C3)C2=O)C(=O)N1	C46H44N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-OSR0HP	WO2018102725A1_224	.	COC1=CC=C2C(=C1)CC[C@H](C1=CC=CC=C1)[C@@H]2C1=CC=C(OCCCCCN2CCN(C3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4)CC2)C=C1	C45H50N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-WPV1LT	WO2018102725A1_225	.	COC1=CC=C2C(=C1)CC[C@H](C1=CC=CC=C1)[C@@H]2C1=CC=C(OCCCCCN2CCN(C3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)C=C1	C45H48N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-XT1Y55	WO2018102725A1_226	.	O=C1CCC(N2C(=O)C3=C(C=C(N4CCN(C[C@H]5CCN(CCOC6=CC=C([C@H]7C8=CC=C(O)C=C8CC[C@H]7C7=CC=C(F)C=C7)C=C6)C5)CC4)C=C3)C2=O)C(=O)N1	C46H48FN5O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-T7AXM4	WO2018102725A1_227	.	O=C1CCC(N2C(=O)C3=C(C=C(N4CCN(C[C@@H]5CCN(CCOC6=CC=C([C@H]7C8=CC=C(O)C=C8CC[C@H]7C7=CC=C(F)C=C7)C=C6)C5)CC4)C=C3)C2=O)C(=O)N1	C46H48FN5O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-3AOF8A	SCHEMBL20234537	2-(2,6-dioxopiperidin-3-yl)-5-[4-[[(3S)-1-[2-[4-[(1R,2S)-2-(4-fluorophenyl)-6-hydroxy-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]ethyl]pyrrolidin-3-yl]methyl]piperazin-1-yl]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=C(C=C(N4CCN(C[C@@H]5CCN(CCOC6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=C(F)C=C7)C=C6)C5)CC4)C=C3)C2=O)C(=O)N1	C46H48FN5O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-PT6Q56	WO2018102725A1_229	.	O=C1CCC(N2C(=O)C3=C(C=C(N4CCC(CN5CCN(CCOC6=CC=C([C@H]7C8=CC=C(O)C=C8CC[C@H]7C7=CC=C(F)C=C7)C=C6)CC5)CC4)C=C3)C2=O)C(=O)N1	C47H50FN5O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-TQJTBQ	WO2018102725A1_230	.	O=C1CCC(N2C(=O)C3=C(C=C(N4CCC(CN5CCN(CCOC6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=C(F)C=C7)C=C6)CC5)CC4)C=C3)C2=O)C(=O)N1	C47H50FN5O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-R963A0	WO2018102725A1_231	.	O=C1CCC(N2C(=O)C3=CC=C(N4C[C@@H]5C[C@H]4CN5C4CCN(CCOC5=CC=C([C@H]6C7=CC=C(O)C=C7CC[C@H]6C6=CC=CC=C6)C=C5)CC4)C=C3C2=O)C(=O)N1	C47H49N5O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-CLCQSZ	WO2018102725A1_232	.	O=C1CCC(N2C(=O)C3=CC=C(N4C[C@@H]5C[C@H]4CN5C4CCN(CCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)C=C3C2=O)C(=O)N1	C47H49N5O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-1LQTYU	WO2018102725A1_233	.	O=C1CCC(N2C(=O)C3=CC=C(N4C[C@H]5C[C@@H]4CN5C4CCN(CCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)C=C3C2=O)C(=O)N1	C47H49N5O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-TMJ655	WO2018102725A1_234	.	O=C1CCC(N2C(=O)C3=CC=C(N4C[C@@H]5C[C@H]4CN5CC4CCN(CCOC5=CC=C([C@H]6C7=CC=C(O)C=C7CC[C@H]6C6=CC=CC=C6)C=C5)CC4)C=C3C2=O)C(=O)N1	C48H51N5O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-ZN3CXG	WO2018102725A1_235	.	O=C1CCC(N2C(=O)C3=CC=C(N4C[C@@H]5C[C@H]4CN5CC4CCN(CCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)C=C3C2=O)C(=O)N1	C48H51N5O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-0WPCNK	WO2018102725A1_236	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC[C@@H]5C[C@@H]5COC5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)=C3)C2=O)C(=O)N1	C45H48N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-06VM69	WO2018102725A1_237	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC[C@H]5C[C@H]5COC5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)=C3)C2=O)C(=O)N1	C45H48N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-D180UH	SCHEMBL20231501	3-[6-[(3R,5S)-4-[5-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]pentyl]-3,5-dimethylpiperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C[C@@H]1CN(C2=CC3=C(C=C2)C(=O)N(C2CCC(=O)NC2=O)C3)C[C@H](C)N1CCCCCOC1=CC=C([C@@H]2C3=C(C=C(O)C=C3)CC[C@@H]2C2=CC=CC=C2)C=C1	C46H52N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-WVDAGX	WO2018102725A1_239	.	C[C@@H]1CN(C2=CC3=C(C=C2)C(=O)N(C2CCC(=O)NC2=O)C3)C[C@H](C)N1CCCCCOC1=CC=C([C@H]2C3=C(C=C(O)C=C3)CC[C@H]2C2=CC=CC=C2)C=C1	C46H52N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-D5EE4F	WO2018102725A1_240	.	O=C1CCC(N2CC3=CC(N4CCC(CN5CCC(OC6=CC=C([C@H]7C8=C(C=C(O)C=C8)CC[C@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C46H50N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-IES75Z	SCHEMBL22297637	3-[6-[4-[[4-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]piperidin-1-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(N4CCC(CN5CCC(OC6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C46H50N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-T27CRP	WO2018102725A1_242	.	O=C1CCC(N2CC3=C(C=CC(C4=CN=C(O[C@H]5CCN(CCOC6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=CC=C7)C=C6)C5)C=C4)=C3)C2=O)C(=O)N1	C46H44N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-HVD13O	WO2018102725A1_243	.	O=C1CCC(N2C(=O)C3=C(C=C(N4CC5(CCN(CCCCOC6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=C(F)C=C7)C=C6)CC5)C4)C=C3)C2=O)C(=O)N1	C46H47FN4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-XKOEJO	WO2018102725A1_244	.	O=C1CCC(N2C(=O)C3=C(C=C(N4CC5(CCN(CCCCOC6=CC=C([C@H]7C8=CC=C(O)C=C8CC[C@H]7C7=CC=C(F)C=C7)C=C6)CC5)C4)C=C3)C2=O)C(=O)N1	C46H47FN4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-VNMCYN	WO2018102725A1_245	.	O=C1CCC(N2C(=O)C3=C(C=C(N4CCN(C[C@H]5CCN(CCOC6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=C(F)C=C7)C=C6)C5)CC4)C=C3)C2=O)C(=O)N1	C46H48FN5O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-6PDP1K	WO2018102725A1_246	.	O=C1CCC(N2C(=O)C3=CC=C(N4C[C@H]5C[C@@H]4CN5CC4CCN(CCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)C=C3C2=O)C(=O)N1	C48H51N5O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-O5UMUE	WO2018102725A1_247	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCCCCOC5=CC=C(C6C7=C(C=C(O)C=C7)CCN6C6=CC=C(F)C=C6)C=C5)CC4)=C3)C2=O)C(=O)N1	C43H46FN5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-VPKM4W	WO2018102725A1_248	.	O=C1CCC(N2C(=O)C3=C(C=C(N4CCN(CCCCCOC5=CC=C([C@H]6C7=CC=C(O)C=C7CC[C@H]6C6=CC=C(F)C=C6)C=C5)CC4)N=C3)C2=O)C(=O)N1	C43H44FN5O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-0HNU3L	WO2018102725A1_249	.	O=C1CCC(N2C(=O)C3=C(C=C(N4CCN(CCCCCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=C(F)C=C6)C=C5)CC4)N=C3)C2=O)C(=O)N1	C43H44FN5O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-GVHIPN	WO2018102725A1_250	.	O=C1CCC(N2CC3=C(C=CC(N4CC5(CCN(CCCCOC6=CC=C([C@H]7C8=CC=C(O)C=C8CC[C@H]7C7=CC=C(F)C=C7)C=C6)CC5)C4)=C3)C2=O)C(=O)N1	C46H49FN4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-MMMA0Q	WO2018102725A1_251	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(C[C@H]5CCN(CCOC6=CC=C([C@H]7C8=CC=C(O)C=C8CC[C@H]7C7=CC=C(F)C=C7)C=C6)C5)CC4)=C3)C2=O)C(=O)N1	C46H50FN5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-MTV03W	WO2018102725A1_252	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(C[C@H]5CCN(CCOC6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=C(F)C=C7)C=C6)C5)CC4)=C3)C2=O)C(=O)N1	C46H50FN5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-ZYSR1W	WO2018102725A1_253	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(C[C@@H]5CCN(CCOC6=CC=C([C@H]7C8=CC=C(O)C=C8CC[C@H]7C7=CC=C(F)C=C7)C=C6)C5)CC4)=C3)C2=O)C(=O)N1	C46H50FN5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-7NWKDG	WO2018102725A1_254	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(C[C@@H]5CCN(CCOC6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=C(F)C=C7)C=C6)C5)CC4)=C3)C2=O)C(=O)N1	C46H50FN5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-NAT7V2	WO2018102725A1_255	.	O=C1CCC(N2C(=O)C3=C(C=C(N4CC5(CN(CCCCOC6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=C(F)C=C7)C=C6)C5)C4)C=C3)C2=O)C(=O)N1	C44H43FN4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-LZDYM6	WO2018102725A1_256	.	O=C1CCC(N2C(=O)C3=C(C=C(N4CC5(CN(CCCCOC6=CC=C([C@H]7C8=CC=C(O)C=C8CC[C@H]7C7=CC=C(F)C=C7)C=C6)C5)C4)C=C3)C2=O)C(=O)N1	C44H43FN4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-V152NC	WO2018102725A1_257	.	O=C1CC[C@H](N2CC3=C(C=CC(OCCN4CCN(C5=CC=C(OC6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)N=C5)CC4)=C3)C2=O)C(=O)N1	C46H45N5O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-6VHGA9	WO2018102725A1_258	2-(2,6-dioxopiperidin-3-yl)-5-[2-[4-[6-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]pyridin-3-yl]piperazin-1-yl]ethoxy]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=C(C=C(OCCN4CCN(C5=CC=C(OC6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)N=C5)CC4)C=C3)C2=O)C(=O)N1	C46H43N5O7	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-GRYFLT	WO2018102725A1_259	.	O=C1CCC(N2C(=O)C3=C(C=C(OCCCN4CCN(C5=CC=C(OC6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)N=C5)CC4)C=C3)C2=O)C(=O)N1	C47H45N5O7	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-PQ6LID	WO2018102725A1_260	.	O=C1CCC(N2CC3=C(C=CC(OCCCN4CCN(C5=CC=C(OC6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)N=C5)CC4)=C3)C2=O)C(=O)N1	C47H47N5O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-SCNZVG	SCHEMBL20234708	2-(2,6-dioxopiperidin-3-yl)-5-[4-[3-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]propyl]-1-oxa-4,9-diazaspiro[5.5]undecan-9-yl]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC=C(N4CCC5(CC4)CN(CCCOC4=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C4)CCO5)C=C3C2=O)C(=O)N1	C46H48N4O7	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-GL06L5	WO2018102725A1_262	.	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCOC5CCC(OC6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=C(C(F)(F)F)C=C7)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C48H49F3N4O7	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-N5F4TI	WO2018102725A1_263	.	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCOC5CCC(OC6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=C(F)C=C7)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C47H49FN4O7	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-DUK14W	WO2018102725A1_264	.	C[C@@H]1CN(CCCCCOC2=CC=C([C@@H]3C4=C(C=C(O)C=C4)CC[C@@H]3C3=CC=C(F)C=C3)C=C2)[C@@H](C)CN1C1=CC2=C(C=C1)C(=O)N(C1CCC(=O)NC1=O)C2	C46H51FN4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-6SH68A	WO2018102725A1_265	.	C[C@@H]1CN(CCCCCOC2=CC=C([C@H]3C4=C(C=C(O)C=C4)CC[C@H]3C3=CC=C(F)C=C3)C=C2)[C@@H](C)CN1C1=CC2=C(C=C1)C(=O)N(C1CCC(=O)NC1=O)C2	C46H51FN4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-27OWZV	WO2018102725A1_266	.	O=C1CCC(N2CC3=C(C=CC(N4CC5(CCN(CCCCOC6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=C(F)C=C7)C=C6)CC5)C4)=C3)C2=O)C(=O)N1	C46H49FN4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-JFX72R	WO2018102725A1_267	.	O=C1CCC(N2C(=O)C3=C(C=C(C4=NC=C(O[C@H]5CCN(CCOC6=CC=C([C@H]7C8=CC=C(O)C=C8CC[C@H]7C7=CC=C(F)C=C7)C=C6)C5)N=C4)C=C3)C2=O)C(=O)N1	C45H40FN5O7	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-BJKFWC	WO2018102725A1_268	.	O=C1CCC(N2C(=O)C3=C(C=C(C4=NC=C(O[C@H]5CCN(CCOC6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=C(F)C=C7)C=C6)C5)N=C4)C=C3)C2=O)C(=O)N1	C45H40FN5O7	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-3UXH3G	WO2018102725A1_269	.	O=C1CCC(N2C(=O)C3=C(C=C(C4=NC=C(O[C@@H]5CCN(CCOC6=CC=C([C@H]7C8=CC=C(O)C=C8CC[C@H]7C7=CC=C(F)C=C7)C=C6)C5)N=C4)C=C3)C2=O)C(=O)N1	C45H40FN5O7	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-AFRAGX	SCHEMBL20234439	2-(2,6-dioxopiperidin-3-yl)-5-[5-[(3R)-1-[2-[4-[(1R,2S)-2-(4-fluorophenyl)-6-hydroxy-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]ethyl]pyrrolidin-3-yl]oxypyrazin-2-yl]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=C(C=C(C4=NC=C(O[C@@H]5CCN(CCOC6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=C(F)C=C7)C=C6)C5)N=C4)C=C3)C2=O)C(=O)N1	C45H40FN5O7	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-YUHWK7	WO2018102725A1_271	.	O=C1CCC(N2C(=O)C3=C(C=C(C4=NC=C(N5CCN(CCOC6=CC=C([C@H]7C8=CC=C(O)C=C8CC[C@H]7C7=CC=C(F)C=C7)C=C6)CC5)N=C4)C=C3)C2=O)C(=O)N1	C45H41FN6O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-JN5QZ9	WO2018102725A1_272	.	O=C1CCC(N2C(=O)C3=C(C=C(C4=NC=C(N5CCN(CCOC6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=C(F)C=C7)C=C6)CC5)N=C4)C=C3)C2=O)C(=O)N1	C45H41FN6O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-RKV9WS	WO2018102725A1_273	.	O=C1CCC(N2C(=O)C3=C(C=C(C4=NC=C(OCC5CN(CCOC6=CC=C([C@H]7C8=CC=C(O)C=C8CC[C@H]7C7=CC=C(F)C=C7)C=C6)C5)N=C4)C=C3)C2=O)C(=O)N1	C45H40FN5O7	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-X4R7D8	WO2018102725A1_274	.	O=C1CCC(N2C(=O)C3=C(C=C(C4=NC=C(OCC5CN(CCOC6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=C(F)C=C7)C=C6)C5)N=C4)C=C3)C2=O)C(=O)N1	C45H40FN5O7	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-HM6T0E	WO2018102725A1_275	2-(2,6-dioxopiperidin-3-yl)-5-[2-[4-[2-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]ethyl]piperazin-1-yl]pyrimidin-5-yl]oxyisoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC=C(OC4=CN=C(N5CCN(CCOC6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)N=C4)C=C3C2=O)C(=O)N1	C45H42N6O7	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-XV6NTW	WO2018102725A1_276	.	O=C1CCC(N2CC3=CC(N4CCN(CCOC5CCC(OC6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=C(C(F)(F)F)C=C7)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C48H51F3N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-6MZ8JS	WO2018102725A1_277	.	O=C1CCC(N2CC3=CC(N4CCN(CCOC5CCC(OC6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=C(F)C=C7)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C47H51FN4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-QY5Q1B	WO2018102725A1_278	.	O=C1CCC(N2C(=O)C3=C(N=C(N4CCN(CCCCCOC5=CC=C([C@H]6C7=CC=C(O)C=C7CC[C@H]6C6=CC=C(F)C=C6)C=C5)CC4)C=N3)C2=O)C(=O)N1	C42H43FN6O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-9BRQVG	WO2018102725A1_279	.	O=C1CCC(N2C(=O)C3=C(N=C(N4CCN(CCCCCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=C(F)C=C6)C=C5)CC4)C=N3)C2=O)C(=O)N1	C42H43FN6O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-YKVB7I	WO2018102725A1_280	.	O=C1CCC(N2C(=O)C3=C(C=C(C4CCN(C5CCN(CCOC6=CC=C([C@H]7C8=CC=C(O)C=C8CC[C@H]7C7=CC=C(F)C=C7)C=C6)CC5)CC4)C=C3)C2=O)C(=O)N1	C47H49FN4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-OK1J70	SCHEMBL20231949	2-(2,6-dioxopiperidin-3-yl)-5-[1-[1-[2-[4-[(1R,2S)-2-(4-fluorophenyl)-6-hydroxy-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]ethyl]piperidin-4-yl]piperidin-4-yl]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=C(C=C(C4CCN(C5CCN(CCOC6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=C(F)C=C7)C=C6)CC5)CC4)C=C3)C2=O)C(=O)N1	C47H49FN4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-48ILJZ	WO2018102725A1_282	.	O=C1CCC(N2C(=O)C3=CC=C(OC4=CC=C(N5CCN(CCOC6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)N=C4)C=C3C2=O)C(=O)N1	C46H43N5O7	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-II4LMW	WO2018102725A1_283	.	O=C1CCC(N2CC3=CC(N4CCN(CCCN5C=C(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)C=N5)CC4)=CC=C3C2=O)C(=O)N1	C45H46N6O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-FRF58D	WO2018102725A1_284	.	O=C1CCC(N2CC3=CC(N4CCN(CCCCCOC5=CC=C(C6C7=CC=C(O)C=C7CCN6C6=C(F)C=C(C(F)(F)F)C=C6)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C44H45F4N5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-99C2QX	WO2018102725A1_285	.	O=C1CCC(N2C(=O)C3=C(N=C(N4CCN(CCCCCOC5=CC=C([C@H]6C7=CC=C(O)C=C7CC[C@H]6C6=CC=C(F)C=C6)C=C5)CC4)N=C3)C2=O)C(=O)N1	C42H43FN6O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-R82EML	WO2018102725A1_286	.	O=C1CCC(N2C(=O)C3=C(N=C(N4CCN(CCCCCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=C(F)C=C6)C=C5)CC4)N=C3)C2=O)C(=O)N1	C42H43FN6O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-O85564	WO2018102725A1_287	.	O=C1CCC(N2CC3=C(C=CC(C4CCN(C5CCN(CCOC6=CC=C([C@H]7C8=CC=C(O)C=C8CC[C@H]7C7=CC=C(F)C=C7)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C47H51FN4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-61DABQ	WO2018102725A1_288	.	O=C1CCC(N2CC3=C(C=CC(C4CCN(C5CCN(CCOC6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=C(F)C=C7)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C47H51FN4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-P7UO5O	WO2018102725A1_289	2-(2,6-dioxopiperidin-3-yl)-5-[4-[2-[4-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]piperidin-1-yl]ethyl]piperazin-1-yl]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCN5CCC(OC6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C46H49N5O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-U03ED7	WO2018102725A1_290	.	O=C1CCC(N2CC3=CC(N4CCN(C5CCN(CCCC6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)C5)CC4)=CC=C3C2=O)C(=O)N1	C46H51N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-X1U5GP	WO2018102725A1_291	.	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(C5CCN(CCCC6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)C5)CC4)C=C3C2=O)C(=O)N1	C46H49N5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-5DDS3Q	WO2018102725A1_292	.	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CC5CN(CCCC6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)C5)CC4)C=C3C2=O)C(=O)N1	C46H49N5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-IX44SP	WO2018102725A1_293	.	O=C1CCC(N2CC3=CC(N4CCN(CC5CN(CCCC6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)C5)CC4)=CC=C3C2=O)C(=O)N1	C46H51N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-GQYCUO	WO2018102725A1_294	.	O=C1CC[C@@H](N2CC3=CC(OC4=CC=C(N5CCN(CCOC6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)N=C4)=CC=C3C2=O)C(=O)N1	C46H45N5O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-SA5JWC	WO2018102725A1_295	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCN5CCN(C6=CC=C([C@H]7C8=C(C=C(O)C=C8)CC[C@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C45H50N6O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-TSUPGY	WO2018102725A1_296	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCN5CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C45H50N6O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-UOJ4ZC	WO2018102725A1_297	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCN5CCC(C6=CC=C([C@H]7C8=CC=C(O)C=C8CC[C@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C46H51N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-PFG5FV	SCHEMBL20234960	3-[6-[4-[2-[4-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-1-yl]ethyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCN5CCC(C6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C46H51N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-UP3O8V	WO2018102725A1_299	.	O=C1CCC(N2C(=O)C3=C(C=C(N4CCN(CCN5CCC(C6=CC=C([C@H]7C8=CC=C(O)C=C8CC[C@H]7C7=CC=CC=C7)C=C6)CC5)CC4)C=C3)C2=O)C(=O)N1	C46H49N5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-3V9LTW	WO2018102725A1_300	.	O=C1CCC(N2C(=O)C3=C(C=C(N4CCN(CCN5CCC(C6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)C=C3)C2=O)C(=O)N1	C46H49N5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-L1XRR1	WO2018102725A1_301	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(C5CC6(C5)CN(CCOC5=CC=C([C@H]7C8=C(C=C(O)C=C8)CC[C@H]7C7=CC=CC=C7)C=C5)C6)CC4)=C3)C2=O)C(=O)N1	C47H51N5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-C1WJ8K	WO2018102725A1_302	.	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCCCCOC5=CC=C(C6C7=CC=C(O)C=C7CCN6C6=C(F)C=C(C(F)(F)F)C=C6)C=C5)CC4)C=C3C2=O)C(=O)N1	C44H43F4N5O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-0AY0I6	WO2018102725A1_303	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC5CN(CCCC6=CC=C([C@H]7C8=CC=C(O)C=C8CC[C@H]7C7=CC=CC=C7)C=C6)C5)CC4)=C3)C2=O)C(=O)N1	C46H51N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-Q9EAGB	WO2018102725A1_305	.	O=C1CCC(N2C(=O)C3=C(C=C(N4CCN(CC5CN(CCCC6=CC=C([C@H]7C8=CC=C(O)C=C8CC[C@H]7C7=CC=CC=C7)C=C6)C5)CC4)C=C3)C2=O)C(=O)N1	C46H49N5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-BN625B	SCHEMBL20234698	2-(2,6-dioxopiperidin-3-yl)-5-[4-[3-[4-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]pyrazol-1-yl]propyl]piperazin-1-yl]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCCN5C=C(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)C=N5)CC4)C=C3C2=O)C(=O)N1	C45H44N6O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-1GA5CJ	WO2018102725A1_307	.	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCCN5N=NC(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)=N5)CC4)C=C3C2=O)C(=O)N1	C43H42N8O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-CD5L4Q	WO2018102725A1_308	3-[6-[4-[3-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]propyl]-1-oxa-4,9-diazaspiro[5.5]undecan-9-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(N4CCC5(CC4)CN(CCCOC4=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C4)CCO5)=CC=C3C2=O)C(=O)N1	C46H50N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-XTLV6O	WO2018102725A1_310	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC5CCN(CCCC6=CC=C([C@H]7C8=CC=C(O)C=C8CC[C@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C48H55N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-KJL9O2	WO2018102725A1_311	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC5CCN(CCCC6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C48H55N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-H31F3F	WO2018102725A1_312	.	O=C1CCC(N2C(=O)C3=C(C=C(N4CCN(CC5CCN(CCCC6=CC=C([C@H]7C8=CC=C(O)C=C8CC[C@H]7C7=CC=CC=C7)C=C6)CC5)CC4)C=C3)C2=O)C(=O)N1	C48H53N5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-59CZ66	WO2018102725A1_313	.	O=C1CCC(N2C(=O)C3=C(C=C(N4CCN(CC5CCN(CCCC6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)C=C3)C2=O)C(=O)N1	C48H53N5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-72PVIH	WO2018102725A1_314	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(C5CCN(CCCC6=CC=C([C@H]7C8=CC=C(O)C=C8CC[C@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C47H53N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-4BY2WL	WO2018102725A1_315	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(C5CCN(CCCC6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C47H53N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-0PDE4D	WO2018102725A1_316	.	O=C1CCC(N2C(=O)C3=C(C=C(N4CCN(C5CCN(CCCC6=CC=C([C@H]7C8=CC=C(O)C=C8CC[C@H]7C7=CC=CC=C7)C=C6)CC5)CC4)C=C3)C2=O)C(=O)N1	C47H51N5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-0WADC4	WO2018102725A1_317	.	O=C1CCC(N2C(=O)C3=C(C=C(N4CCN(C5CCN(CCCC6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)C=C3)C2=O)C(=O)N1	C47H51N5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-V1UQF9	WO2018102725A1_318	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCCN5CCC(C6=CC=C([C@H]7C8=CC=C(O)C=C8CC[C@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C47H53N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-6WIT7A	WO2018102725A1_319	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCCN5CCC(C6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C47H53N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-Z90RG9	WO2018102725A1_320	.	O=C1CCC(N2C(=O)C3=C(C=C(N4CCN(CCCN5CCC(C6=CC=C([C@H]7C8=CC=C(O)C=C8CC[C@H]7C7=CC=CC=C7)C=C6)CC5)CC4)C=C3)C2=O)C(=O)N1	C47H51N5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-20AQ9V	WO2018102725A1_321	.	O=C1CCC(N2C(=O)C3=C(C=C(N4CCN(CCCN5CCC(C6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)C=C3)C2=O)C(=O)N1	C47H51N5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-IA5MAQ	WO2018102725A1_322	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(C5CC6CC(OC7=CC=C([C@@H]8C9=C(C=C(O)C=C9)CC[C@@H]8C8=CC=C(F)C=C8)C=C7)CC6C5)CC4)=C3)C2=O)C(=O)N1	C47H49FN4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-BI7K6O	WO2018102725A1_323	.	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCCCCCC5=CC=C([C@H]6C7=C(C=C(O)C=C7)CC[C@H]6C6=CC=CC=C6)C=C5)CC4)C=C3C2=O)C(=O)N1	C45H48N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-NHRLXC	WO2018102725A1_324	.	O=C1CCC(N2C(=O)C3=CC=C(N4C[C@@H]5C[C@H]4CN5CCCCCCC4=CC=C([C@H]5C6=C(C=C(O)C=C6)CC[C@H]5C5=CC=CC=C5)C=C4)C=C3C2=O)C(=O)N1	C46H48N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-QDZKW8	WO2018102725A1_325	.	O=C1CCC(N2C(=O)C3=CC=C(N4C[C@H]5C[C@@H]4CN5CCCCCCC4=CC=C([C@H]5C6=C(C=C(O)C=C6)CC[C@H]5C5=CC=CC=C5)C=C4)C=C3C2=O)C(=O)N1	C46H48N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-34TXOP	WO2018102725A1_326	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCCCCOC5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)=C3Cl)C2=O)C(=O)N1	C44H47ClN4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-ZVKGWI	WO2018102725A1_327	.	O=C1CCC(N2CC3=C(C=C(F)C(N4CCN(CCCCCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)=C3)C2=O)C(=O)N1	C44H47FN4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-AXR1K7	WO2018102725A1_328	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(C5CC6(C5)CN(CCOC5=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C5)C6)CC4)=C3)C2=O)C(=O)N1	C47H51N5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-94RRGV	WO2018102725A1_329	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(C5CC6(C5)CN(CCOC5=CC=C([C@H]7C8=C(C=C(O)C=C8)CC[C@H]7C7=CC=CC=C7)C=C5)C6)CC4)=C3F)C2=O)C(=O)N1	C47H50FN5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-F0X0XS	WO2018102725A1_330	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(C5CC6(C5)CN(CCOC5=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C5)C6)CC4)=C3F)C2=O)C(=O)N1	C47H50FN5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-EKCEIL	WO2018102725A1_331	.	O=C1CCC(N2CC3=C(C=C(F)C(N4CCN(C5CC6(C5)CN(CCOC5=CC=C([C@H]7C8=C(C=C(O)C=C8)CC[C@H]7C7=CC=CC=C7)C=C5)C6)CC4)=C3F)C2=O)C(=O)N1	C47H49F2N5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-39FWU1	WO2018102725A1_332	.	O=C1CCC(N2CC3=C(C=C(F)C(N4CCN(C5CC6(C5)CN(CCOC5=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C5)C6)CC4)=C3F)C2=O)C(=O)N1	C47H49F2N5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-SC11NY	WO2018102725A1_333	.	O=C1CCC(N2CC3=C(C=C(F)C(N4CCN(CCCCCOC5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)=C3F)C2=O)C(=O)N1	C44H46F2N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-30OYE9	WO2018102725A1_334	.	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCCCCCC5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)C=C3C2=O)C(=O)N1	C45H48N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-G2LHZD	WO2018102725A1_335	.	O=C1CCC(N2CC3=CC(N4CCN(CCN5CCC(OC6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C46H51N5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-VTK8RW	WO2018102725A1_336	2-(2,6-dioxopiperidin-3-yl)-5-[4-[3-[3-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]azetidin-1-yl]propyl]piperazin-1-yl]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCCN5CC(OC6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)C5)CC4)C=C3C2=O)C(=O)N1	C45H47N5O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-49GJFX	WO2018102725A1_337	.	O=C1CCC(N2CC3=CC(OC4=CN=C(N5CCN(CCOC6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)N=C4)=CC=C3C2=O)C(=O)N1	C45H44N6O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-MQONB9	WO2018102725A1_338	.	O=C1CCC(N2CC3=C(C2=O)C(Cl)=CC(N2CCN(CCCCCOC4=CC=C([C@H]5C6=C(C=C(O)C=C6)CC[C@H]5C5=CC=CC=C5)C=C4)CC2)=C3)C(=O)N1	C44H47ClN4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-P93B6S	WO2018102725A1_339	.	O=C1CCC(N2CC3=C(C2=O)C(Cl)=CC(N2CCN(CCCCCOC4=CC=C([C@@H]5C6=C(C=C(O)C=C6)CC[C@@H]5C5=CC=CC=C5)C=C4)CC2)=C3)C(=O)N1	C44H47ClN4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-8DOI13	WO2018102725A1_340	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC5CCN(C6=CC=C([C@H]7C8=C(C=C(O)C=C8)CC[C@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C45H49N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-NZ5HR7	(Rac)-Vepdegestrant	(Rac)-Vepdegestrant; vepdegrestrant; 2229711-08-2; 3-(5-(4-((1-(4-((1R,2S)-6-Hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl)phenyl)piperidin-4-yl)methyl)piperazin-1-yl)-1-oxoisoindolin-2-yl)piperidine-2,6-dione; 3-[6-[4-[[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; EX-A5021; starbld0007729; CHEMBL5434043; SCHEMBL20231167; SCHEMBL29632151; GTPL11511; HY-138642A; 3-[1,3-Dihydro-1-oxo-5-[4-[[1-[4-[(1R,2S)-1,2,3,4-tetrahydro-6-hydroxy-2-phenyl-1-naphthalenyl]phenyl]-4-piperidinyl]methyl]-1-piperazinyl]-2H-isoindol-2-yl]-2,6-piperidinedione; compound 341 [WO2018102725A1]; DB-136101; CS-0198428	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC5CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C45H49N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-OPIF2K	WO2018102725A1_342	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCC5CCN(C6=CC=C([C@H]7C8=C(C=C(O)C=C8)CC[C@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C46H51N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-EHQNHT	SCHEMBL20211901	3-[6-[4-[2-[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]ethyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL29683535	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCC5CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C46H51N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-G2SMTN	WO2018102725A1_344	.	O=C1CCC(N2CC3=C(C=C(N4CCN(CCCCCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)C(F)=C3)C2=O)C(=O)N1	C44H47FN4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-43KLRO	WO2018102725A1_345	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCCCCOC5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)=C3F)C2=O)C(=O)N1	C44H47FN4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-H86KFT	WO2018102725A1_346	.	O=C1CCC(N2CC3=CC(N4CCN(CCCCCOC5=CC=C([C@@H]6C7=CC(F)=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C44H47FN4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-DK9RO1	WO2018102725A1_347	.	O=C1CCC(N2CC3=CC(N4CCN(CCCCCOC5=CC=C([C@H]6C7=CC(F)=C(O)C=C7CC[C@H]6C6=CC=CC=C6)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C44H47FN4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-JS9IN4	WO2018102725A1_348	.	O=C1CCC(N2C(=O)C3=C(C=C(N4CCN(CCCCCOC5=CC=C([C@@H]6C7=CC(F)=C(O)C(F)=C7CC[C@@H]6C6=CC=C(F)C=C6)C=C5)CC4)C=C3)C2=O)C(=O)N1	C44H43F3N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-S25OK6	WO2018102725A1_349	.	O=C1CCC(N2C(=O)C3=C(C=C(N4CCN(CCCCCOC5=CC=C([C@H]6C7=CC(F)=C(O)C(F)=C7CC[C@H]6C6=CC=C(F)C=C6)C=C5)CC4)C=C3)C2=O)C(=O)N1	C44H43F3N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-A290F6	WO2018102725A1_350	.	O=C1CCC(N2C(=O)C3=C(C=C(N4CCN(CCCCCOC5=CC=C([C@H]6C7=CC=C(O)C(F)=C7CC[C@H]6C6=CC=C(F)C=C6)C=C5)CC4)C=C3)C2=O)C(=O)N1	C44H44F2N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-IV1YRF	WO2018102725A1_351	.	O=C1CCC(N2C(=O)C3=C(C=C(N4CCN(CCCCCOC5=CC=C([C@@H]6C7=CC=C(O)C(F)=C7CC[C@@H]6C6=CC=C(F)C=C6)C=C5)CC4)C=C3)C2=O)C(=O)N1	C44H44F2N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-CIIFRC	WO2018102725A1_352	.	O=C1CC[C@H](N2CC3=C(C=CC(CCN4CCCN(CC5CCN(C6=CC=C([C@H]7C8=C(C=C(O)C=C8)CC[C@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C48H55N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-JICBL2	WO2018102725A1_353	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(C5CC6CC(COC7=CC=C([C@@H]8C9=C(C=C(O)C=C9)CC[C@@H]8C8=CC=C(F)C=C8)C=C7)CC6C5)CC4)=C3)C2=O)C(=O)N1	C48H51FN4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-B42X4T	WO2018102725A1_354	.	O=C1CCC(N2C(=O)C3=CC=C(N4C[C@@H]5C[C@H]4CN5CCCCCCC4=CC=C([C@@H]5C6=C(C=C(O)C=C6)CC[C@@H]5C5=CC=CC=C5)C=C4)C=C3C2=O)C(=O)N1	C46H48N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-78XGWR	WO2018102725A1_355	.	O=C1CCC(N2C(=O)C3=CC=C(N4C[C@H]5C[C@@H]4CN5CCCCCCC4=CC=C([C@@H]5C6=C(C=C(O)C=C6)CC[C@@H]5C5=CC=CC=C5)C=C4)C=C3C2=O)C(=O)N1	C46H48N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-XIH6LZ	WO2018102725A1_356	.	O=C1CCC(N2CC3=C(C=CC(N4CC5(CN(CCCCOC6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=C(F)C=C7)C=C6)C5)C4)=C3)C2=O)C(=O)N1	C44H45FN4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-LPHLK4	WO2018102725A1_357	.	O=C1CCC(N2CC3=C(C=CC(N4CC5(CN(CCCCOC6=CC=C([C@H]7C8=CC=C(O)C=C8CC[C@H]7C7=CC=C(F)C=C7)C=C6)C5)C4)=C3)C2=O)C(=O)N1	C44H45FN4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-S4ROO7	WO2018102725A1_358	.	O=C1CCC(N2CC3=C(C=CC(N4CCN5CCN(CCCCOC6=CC=C([C@H]7C8=C(C=C(O)C=C8)CC[C@H]7C7=CC=CC=C7)C=C6)CC5C4)=C3)C2=O)C(=O)N1	C46H51N5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-1E5A3R	WO2018102725A1_359	.	O=C1CCC(N2CC3=C(C=CC(N4CCN5CCN(CCCCOC6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)CC5C4)=C3)C2=O)C(=O)N1	C46H51N5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-3YLQ8G	SCHEMBL20231091	3-[6-[4-[2-hydroxy-5-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]pentyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC(O)CCCOC5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)=C3)C2=O)C(=O)N1	C44H48N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-QQYN43	WO2018102725A1_361	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(C5CC(CCCOC6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)C5)CC4)=C3)C2=O)C(=O)N1	C46H50N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-HBLRS5	WO2018102725A1_362	.	O=C1CCC(N2CC3=C(C2=O)C(F)=CC(N2CCN(CCCCCOC4=CC=C([C@@H]5C6=C(C=C(O)C=C6)CC[C@@H]5C5=CC=CC=C5)C=C4)CC2)=C3)C(=O)N1	C44H47FN4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-81NW2Q	SCHEMBL21983065	3-[6-[4-[3-hydroxy-5-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]-3-methylpentyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CC(O)(CCOC1=CC=C([C@@H]2C3=CC=C(O)C=C3CC[C@@H]2C2=CC=CC=C2)C=C1)CCN1CCN(C2=CC=C3C(=O)N(C4CCC(=O)NC4=O)CC3=C2)CC1	C45H50N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-1V691G	WO2018102725A1_364	.	O=C1CC[C@H](N2CC3=C(C=CC(CCN4CCCN(CC5CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C48H55N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-PYVCO0	SCHEMBL20235015	3-[6-[4-[5-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]-2-oxopentyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C(CCCOC1=CC=C([C@@H]2C3=C(C=C(O)C=C3)CC[C@@H]2C2=CC=CC=C2)C=C1)CN1CCN(C2=CC3=C(C=C2)C(=O)N(C2CCC(=O)NC2=O)C3)CC1	C44H46N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-OUD2F7	WO2018102725A1_366	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC(O)CCCOC5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)=C3F)C2=O)C(=O)N1	C44H47FN4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-Y9J4R5	WO2018102725A1_367	.	O=C1CCC(N2CC3=C(C=C(F)C(N4CCN(CC(O)CCCOC5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)=C3F)C2=O)C(=O)N1	C44H46F2N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-5JHTYI	WO2018102725A1_368	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(C5CC(CCOC6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)C5)CC4)=C3)C2=O)C(=O)N1	C45H48N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-O1UINP	WO2018102725A1_369	.	[H][C@@]12CN(CCCCOC3=CC=C([C@H]4C5=C(C=C(O)C=C5)CC[C@H]4C4=CC=CC=C4)C=C3)C[C@]1([H])CN(C1=CC3=C(C=C1)C(=O)N(C1CCC(=O)NC1=O)C3=O)C2	C45H46N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-B754VH	WO2018102725A1_370	.	[H][C@@]12CN(CCCCOC3=CC=C([C@@H]4C5=C(C=C(O)C=C5)CC[C@@H]4C4=CC=CC=C4)C=C3)C[C@]1([H])CN(C1=CC3=C(C=C1)C(=O)N(C1CCC(=O)NC1=O)C3=O)C2	C45H46N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-UME1HT	WO2018102725A1_371	.	[H][C@@]12CN(CCCOC3=CC=C([C@H]4C5=C(C=C(O)C=C5)CC[C@H]4C4=CC=CC=C4)C=C3)C[C@]1([H])CN(C1=CC3=C(C=C1)C(=O)N(C1CCC(=O)NC1=O)C3=O)C2	C44H44N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-AIR7BI	WO2018102725A1_372	.	[H][C@@]12CN(CCCOC3=CC=C([C@@H]4C5=C(C=C(O)C=C5)CC[C@@H]4C4=CC=CC=C4)C=C3)C[C@]1([H])CN(C1=CC3=C(C=C1)C(=O)N(C1CCC(=O)NC1=O)C3=O)C2	C44H44N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-CW6L6F	WO2018102725A1_373	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCOCCOC5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)=C3)C2=O)C(=O)N1	C43H46N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-5O1PWA	WO2018102725A1_374	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCO[C@H]5C[C@H](OC6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)C5)CC4)=C3)C2=O)C(=O)N1	C45H48N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-HJJNJ0	WO2018102725A1_375	.	O=C1CCC(N2C(=O)C3=C(C=C(N4CCN(CCCC(F)(F)COC5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)C=C3)C2=O)C(=O)N1	C44H44F2N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-VP87QO	WO2018102725A1_376	.	O=C1CCC(N2C(=O)C3=C(C=C(N4CCN(C5CCC6CCC(OC7=CC=C([C@@H]8C9=CC=C(O)C=C9CC[C@@H]8C8=CC=C(F)C=C8)C=C7)CC6C5)CC4)C=C3)C2=O)C(=O)N1	C49H51FN4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-NAFP38	SCHEMBL21982923	3-[6-[4-[3-hydroxy-5-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]pentyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCC(O)CCOC5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)=C3)C2=O)C(=O)N1	C44H48N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-KK5DQT	WO2018102725A1_378	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC5CC6CC(OC7=CC=C([C@@H]8C9=C(C=C(O)C=C9)CC[C@@H]8C8=CC=C(F)C=C8)C=C7)CC6C5)CC4)=C3)C2=O)C(=O)N1	C48H51FN4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-SIHQP5	WO2018102725A1_379	.	O=C1CCC(N2CC3=C(C=C(F)C(N4CCN(CC5CC6CC(OC7=CC=C([C@@H]8C9=C(C=C(O)C=C9)CC[C@@H]8C8=CC=C(F)C=C8)C=C7)CC6C5)CC4)=C3F)C2=O)C(=O)N1	C48H49F3N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-3IA2VN	WO2018102725A1_380	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(C5CCC(CCOC6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)C5)CC4)=C3)C2=O)C(=O)N1	C46H50N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-BLQSSQ	WO2018102725A1_381	.	[H][C@@]12CN(CCCCOC3=CC=C([C@H]4C5=C(C=C(O)C=C5)CC[C@H]4C4=CC=CC=C4)C=C3)C[C@]1([H])CN(C1=CC3=C(C=C1)C(=O)N(C1CCC(=O)NC1=O)C3)C2	C45H48N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-M503EE	WO2018102725A1_382	.	[H][C@@]12CN(CCCCOC3=CC=C([C@@H]4C5=C(C=C(O)C=C5)CC[C@@H]4C4=CC=CC=C4)C=C3)C[C@]1([H])CN(C1=CC3=C(C=C1)C(=O)N(C1CCC(=O)NC1=O)C3)C2	C45H48N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-T1LA3Y	WO2018102725A1_383	.	[H][C@@]12CN(CCCOC3=CC=C([C@H]4C5=C(C=C(O)C=C5)CC[C@H]4C4=CC=CC=C4)C=C3)C[C@]1([H])CN(C1=CC3=C(C=C1)C(=O)N(C1CCC(=O)NC1=O)C3)C2	C44H46N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-25EMG6	WO2018102725A1_384	.	[H][C@@]12CN(CCCOC3=CC=C([C@@H]4C5=C(C=C(O)C=C5)CC[C@@H]4C4=CC=CC=C4)C=C3)C[C@]1([H])CN(C1=CC3=C(C=C1)C(=O)N(C1CCC(=O)NC1=O)C3)C2	C44H46N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-3FR75E	WO2018102725A1_385	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCCCCS(=O)(=O)C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)=C3)C2=O)C(=O)N1	C44H48N4O6S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-PN97KF	WO2018102725A1_386	.	O=C1CC[C@H](N2CC3=C(C=CC(CCN4CCCN(CC5CN(C6=CC=C([C@H]7C8=C(C=C(O)C=C8)CC[C@H]7C7=CC=CC=C7)C=C6)C5)CC4)=C3)C2=O)C(=O)N1	C46H51N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-JR1PXI	SCHEMBL20234472	(3S)-3-[6-[2-[4-[[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]azetidin-3-yl]methyl]-1,4-diazepan-1-yl]ethyl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CC[C@H](N2CC3=C(C=CC(CCN4CCCN(CC5CN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)C5)CC4)=C3)C2=O)C(=O)N1	C46H51N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-TYBSAG	WO2018102725A1_388	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCCCCOC5=C(F)C=C([C@H]6C7=C(C=C(O)C=C7)CC[C@H]6C6=CC=CC=C6)C=C5F)CC4)=C3)C2=O)C(=O)N1	C44H46F2N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-OF8JPD	WO2018102725A1_389	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCCCCOC5=C(F)C=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5F)CC4)=C3)C2=O)C(=O)N1	C44H46F2N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-IKYFWV	WO2018102725A1_390	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCO[C@H]5C[C@@H](OC6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)C5)CC4)=C3)C2=O)C(=O)N1	C45H48N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-7PAI7H	WO2018102725A1_391	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCNCCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)=C3)C2=O)C(=O)N1	C43H47N5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-UKNHMK	WO2018102725A1_392	.	O=C1CCC(N2C(=O)C3=C(C=C(N4CCN(CC5CCN(C6=CC=C([C@H]7C8=C(C=C(O)C=C8)CC[C@H]7C7=CC=CC=C7)C=C6)CC5)CC4)C=C3)C2=O)C(=O)N1	C45H47N5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-XKQMS5	SCHEMBL20211886	2-(2,6-dioxopiperidin-3-yl)-5-[4-[[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]isoindole-1,3-dione; SCHEMBL29882897	O=C1CCC(N2C(=O)C3=C(C=C(N4CCN(CC5CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)C=C3)C2=O)C(=O)N1	C45H47N5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-FLR1VB	WO2018102725A1_394	.	O=C1CCC(N2C(=O)C3=C(C=C(N4CCN(CCC5CCN(C6=CC=C([C@H]7C8=C(C=C(O)C=C8)CC[C@H]7C7=CC=CC=C7)C=C6)CC5)CC4)C=C3)C2=O)C(=O)N1	C46H49N5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-JAH3CR	SCHEMBL20211893	2-(2,6-dioxopiperidin-3-yl)-5-[4-[2-[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]ethyl]piperazin-1-yl]isoindole-1,3-dione; SCHEMBL29683711	O=C1CCC(N2C(=O)C3=C(C=C(N4CCN(CCC5CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)C=C3)C2=O)C(=O)N1	C46H49N5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-BMT4NS	WO2018102725A1_396	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCCCCSC5=CC=C([C@H]6C7=CC=C(O)C=C7CC[C@H]6C6=CC=CC=C6)C=C5)CC4)=C3)C2=O)C(=O)N1	C44H48N4O4S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-H324MG	WO2018102725A1_397	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(C[C@H]5CC[C@H](COC6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)O5)CC4)=C3)C2=O)C(=O)N1	C45H48N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-9JQN02	WO2018102725A1_398	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC[C@H]5C[C@@H](OC6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=CC=C7)C=C6)C5)CC4)=C3)C2=O)C(=O)N1	C45H48N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-G39VHL	WO2018102725A1_399	.	CC1(C2=CC=C(OCCCCCN3CCN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5)CC3)C=C2)C2=CC=C(O)C=C2CCN1C1=CC=C(F)C=C1	C44H48FN5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-CR7ZJ1	WO2018102725A1_400	.	CC1(C2=CC=C(OCCCCCN3CCN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)C=C2)C2=CC=C(O)C=C2CCN1C1=CC=C(F)C=C1	C44H46FN5O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-EEU9H4	WO2018102725A1_401	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCCCCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)=N3)C2=O)C(=O)N1	C43H47N5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-W7AG76	WO2018102725A1_402	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCCC(F)(F)COC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)=N3)C2=O)C(=O)N1	C43H45F2N5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-URMMZT	WO2018102725A1_403	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCCCCSC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)=C3)C2=O)C(=O)N1	C44H48N4O4S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-161JWY	SCHEMBL20235072	3-[6-[4-[5-fluoro-5-[[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]methyl]-2,3,3a,4,6,6a-hexahydro-1H-pentalen-2-yl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(N4CCN(C5CC6CC(F)(COC7=CC=C([C@@H]8C9=C(C=C(O)C=C9)CC[C@@H]8C8=CC=CC=C8)C=C7)CC6C5)CC4)=C3)C2=O)C(=O)N1	C48H51FN4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-0YBFDG	WO2018102725A1_405	.	O=C1CCC(N2CC3=C(C=NC(N4CCN(CCCCCOC5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)=C3)C2=O)C(=O)N1	C43H47N5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-ZHMFYH	WO2018102725A1_406	.	CC(C)C1=CC=C(N2CCC3=CC(O)=CC=C3C2(C)C2=CC=C(OCCCCCN3CCN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5)CC3)C=C2)C=C1	C47H55N5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-2BG8FA	WO2018102725A1_407	.	O=C1CC[C@@H](N2CC3=C(C=CC(N4CCN(C5CC6CC(OC7=CC=C([C@@H]8C9=CC=C(O)C=C9CC[C@@H]8C8=CC=C(F)C=C8)C=C7)CC6C5)CC4)=C3)C2=O)C(=O)N1	C47H49FN4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-UGTRIS	WO2018102725A1_408	.	O=C1CC[C@H](N2CC3=C(C=CC(N4CCN(C5CC6CC(OC7=CC=C([C@@H]8C9=CC=C(O)C=C9CC[C@@H]8C8=CC=C(F)C=C8)C=C7)CC6C5)CC4)=C3)C2=O)C(=O)N1	C47H49FN4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-8UM9FE	WO2018102725A1_409	.	O=C1CCC(N2C(=O)C3=C(C=C(CCCCC4CCN(CCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)C4)C=C3)C2=O)C(=O)N1	C45H47N3O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-XJ6J54	WO2018102725A1_410	(3S)-3-[6-[4-[[1-[4-[(1S,2R)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CC[C@H](N2CC3=C(C=CC(N4CCN(CC5CCN(C6=CC=C([C@H]7C8=C(C=C(O)C=C8)CC[C@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C45H49N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-YIITA5	Arv-471	ARV-471; Vepdegestrant; ARV471; ARV-471 (protac); Arv 471; PF-07850327; PF07850327; PROTAC Protein Degrader ARV-471; ER alpha PROTAC Protein Degrader ARV-471; PF 07850327; Estrogen Receptor alpha PROTAC Protein Degrader ARV-471; ER alpha Proteolysis-targeting Chimera Protein Degrader ARV-471; 2229711-68-4; WC1U3R1YMI; (S)-3-(5-(4-((1-(4-((1R,2S)-6-Hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl)phenyl)piperidin-4-yl)methyl)piperazin-1-yl)-1-oxoisoindolin-2-yl)piperidine-2,6-dione; (3S)-3-[6-[4-[[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; (S)-3-(5-(4-((1-(4-(rel-(1R,2S)-6-Hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl)phenyl)piperidin-4-yl)methyl)piperazin-1-yl)-1-oxoisoindolin-2-yl)piperidine-2,6-dione; 2614417-52-4; EX-A5021; vepdegestrant [INN]; starbld0006985; UNII-WC1U3R1YMI; Vepdegestrant [WHO-DD]; VEPDEGESTRANT [USAN]; orb1303493; CHEMBL5095210; SCHEMBL20211870; SCHEMBL29390872; SCHEMBL29631983; SCHEMBL30712284; Vepdegestrant (JAN/USAN/INN); ARV-471?; BDBM50623923; AKOS040757430; AT25218; BP-41005; MS-31245; HY-138642; CS-0159885; D12628; EN300-37105519; (2(1)R,2(2)S,8(3)S)-2-hydroxy-2(1),2(2),2(3),2-tetrahydro-7(5,2)-isoindola-6(1,4)-piperazina-4(1,4),8(3)-dipiperidina-2(2,1)-naphthalena-1(1),3(1,4)-dibenzenaoctaphane-7(1),8(2),8(7(3)H)-trione; (3S)-3-(5-{4-[(1-{4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl}piperidin-4-yl)methyl]piperazin-1-yl}-1-oxo-2,3-dihydro-1H-isoindol-2-yl)piperidine-2,6-dione; (3S)-3-[5-[4-[[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-tetralin-1-yl]phenyl]-4-piperidyl]methyl]piperazin-1-yl]-1-oxo-isoindolin-2-yl]piperidine-2,6-dione; 2,6-Piperidinedione, 3-(1,3-dihydro-1-oxo-5-(4-((1-(4-((1R,2S)-1,2,3,4-tetrahydro-6-hydroxy-2-phenyl-1-naphthalenyl)phenyl)-4-piperidinyl)methyl)-1-piperazinyl)-2H-isoindol-2-yl)-, (3S)-; 2,6-Piperidinedione, 3-[1,3-dihydro-1-oxo-5-[4-[[1-[4-[(1R,2S)-1,2,3,4-tetrahydro-6-hydroxy-2-phenyl-1-naphthalenyl]phenyl]-4-piperidinyl]methyl]-	O=C1CC[C@H](N2CC3=C(C=CC(N4CCN(CC5CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C45H49N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-I1Z9DW	WO2018102725A1_412	.	O=C1CC[C@@H](N2CC3=C(C=CC(N4CCN(CC5CCN(C6=CC=C([C@H]7C8=C(C=C(O)C=C8)CC[C@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C45H49N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-DEZWUQ	SCHEMBL20234509	(3R)-3-[6-[4-[[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CC[C@@H](N2CC3=C(C=CC(N4CCN(CC5CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C45H49N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-A9P88G	WO2018102725A1_414	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(C[C@H]5C[C@@H](COC6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)C5)CC4)=C3)C2=O)C(=O)N1	C45H48N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-ABOA6W	WO2018102725A1_415	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(C[C@H]5C[C@H](COC6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)C5)CC4)=C3)C2=O)C(=O)N1	C45H48N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-C8X74K	WO2018102725A1_416	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCC5CCC(OC6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)C5)CC4)=C3)C2=O)C(=O)N1	C46H50N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-1D1VRO	WO2018102725A1_417	.	O=C1CCC(N2CC3=C(C=CC(CCCCC4CCN(CCOC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)C4)=N3)C2=O)C(=O)N1	C44H48N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-LO3LVS	WO2018102725A1_418	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC5CCN(C6=CC=C([C@H]7C8=C(C=C(O)C=C8)CC[C@H]7C7=CC=CC=C7)C=C6F)CC5)CC4)=C3)C2=O)C(=O)N1	C45H48FN5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-VR81ZP	SCHEMBL20211921	3-[6-[4-[[1-[2-fluoro-4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC5CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6F)CC5)CC4)=C3)C2=O)C(=O)N1	C45H48FN5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-NLVPWS	WO2018102725A1_420	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC5CCN(C6=NC=C([C@H]7C8=C(C=C(O)C=C8)CC[C@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C44H48N6O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-52WNFN	WO2018102725A1_421	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC5CCN(C6=NC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C44H48N6O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-K04O2S	WO2018102725A1_422	.	O=C1CC[C@@H](N2CC3=C(C=CC(N4CCN(CCC5CCN(C6=CC=C([C@H]7C8=C(C=C(O)C=C8)CC[C@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C46H51N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-Z5WG9D	WO2018102725A1_423	.	O=C1CC[C@@H](N2CC3=C(C=CC(N4CCN(CCC5CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C46H51N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-PWC16X	WO2018102725A1_424	.	O=C1CC[C@H](N2CC3=C(C=CC(N4CCN(CCC5CCN(C6=CC=C([C@H]7C8=C(C=C(O)C=C8)CC[C@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C46H51N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-PZNIZ6	WO2018102725A1_425	.	O=C1CC[C@H](N2CC3=C(C=CC(N4CCN(CCC5CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C46H51N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-T56LHN	WO2018102725A1_426	.	O=C1CCC(N2CC3=C(C=CC(OCC4CCN(CC5CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C47H52N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-6FZ0NA	WO2018102725A1_427	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC[C@H]5C[C@H](OC6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=CC=C7)C=C6)C5)CC4)=C3)C2=O)C(=O)N1	C45H48N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-V7TYZH	WO2018102725A1_428	.	O=C1CCC(N2C(=O)C3=C(C2=O)C(CCCCC2CCN(CCOC4=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=CC=C5)C=C4)C2)=CC=C3)C(=O)N1	C45H47N3O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-FL0WCS	WO2018102725A1_429	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC5CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=N3)C2=O)C(=O)N1	C44H48N6O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-37DSFB	WO2018102725A1_430	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCC5CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=N3)C2=O)C(=O)N1	C45H50N6O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-VIK2GT	WO2018102725A1_431	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCC5CCN(C6=NC=C([C@H]7C8=C(C=C(O)C=C8)CC[C@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C45H50N6O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-U06AUI	WO2018102725A1_432	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCC5CCN(C6=NC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C45H50N6O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-5QLO5P	WO2018102725A1_433	.	O=C1CCC(N2C(=O)C3=C(C=C(N4CCN(CCC5CCN(C6=NC=C([C@H]7C8=C(C=C(O)C=C8)CC[C@H]7C7=CC=CC=C7)C=C6)CC5)CC4)C=C3)C2=O)C(=O)N1	C45H48N6O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-7LSTHX	WO2018102725A1_434	.	O=C1CCC(N2C(=O)C3=C(C=C(N4CCN(CCC5CCN(C6=NC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)C=C3)C2=O)C(=O)N1	C45H48N6O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-OAA5DN	WO2018102725A1_435	.	O=C1CCC(N2CC3=C(C=CC(CCC4CCN(CC5CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C48H54N4O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-CPPCYR	WO2018102725A1_436	.	O=C1CCC(N2C(=O)C3=C(C=C(OCC4CCN(CC5CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)C=C3)C2=O)C(=O)N1	C47H50N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-EUUIBA	WO2018102725A1_437	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(C[C@H]5CC[C@@H](COC6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)O5)CC4)=C3)C2=O)C(=O)N1	C45H48N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-HOM9OU	WO2018102725A1_438	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(C[C@@H]5CC[C@H](COC6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)O5)CC4)=C3)C2=O)C(=O)N1	C45H48N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-2LJEQ7	WO2018102725A1_439	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(C[C@@H]5CC[C@@H](COC6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)O5)CC4)=C3)C2=O)C(=O)N1	C45H48N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-J7L01Q	SCHEMBL20234737	3-[6-[4-[[6-[[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]methyl]pyridazin-3-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC5=CC=C(COC6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=CC=C7)C=C6)N=N5)CC4)=C3)C2=O)C(=O)N1	C45H44N6O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-QRDDPT	WO2018102725A1_441	.	O=C1CCC(N2C(=O)C3=C(C=C(N4CCN(CC5CCN(C6=NC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)C=C3)C2=O)C(=O)N1	C44H46N6O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-RJX2FC	WO2018102725A1_442	.	C[C@@]1(N2CC3=C(C=CC(N4CCN(CC5CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=C3)C2=O)CCC(=O)NC1=O	C46H51N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-ABPIYS	WO2018102725A1_443	.	C[C@]1(N2CC3=C(C=CC(N4CCN(CC5CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=C3)C2=O)CCC(=O)NC1=O	C46H51N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-0RTQUU	WO2018102725A1_444	.	O=C1CCC(N2CC3=C(C=CC(N4CC5(CCN(CC6CCN(C7=CC=C([C@@H]8C9=C(C=C(O)C=C9)CC[C@@H]8C8=CC=CC=C8)C=C7)CC6)CC5)C4)=C3)C2=O)C(=O)N1	C48H53N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-Z11TTM	SCHEMBL20231397	3-[5-[2-[4-[3-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]cyclobutyl]oxypiperidin-1-yl]ethoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=C(OCCN4CCC(O[C@H]5C[C@H](OC6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)C5)CC4)C=C3)C2=O)C(=O)N1	C46H49N3O7	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-CCKAPO	WO2018102725A1_446	.	O=C1CCC(N2C(=O)C3=C(C=C(N4CCN(CCCCC(OC5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)C(F)(F)F)CC4)C=C3)C2=O)C(=O)N1	C45H45F3N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-1ZQQM3	SCHEMBL23350090	3-[3-oxo-6-[4-[6,6,6-trifluoro-5-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]hexyl]piperazin-1-yl]-1H-isoindol-2-yl]piperidine-2,6-dione; YOCNBWNIGFMELA-FDCUJMSUSA-N; 3-[3-oxo-6-[4-[6,6,6-trifluoro-5-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]hexyl]piperazin-1-yl]-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCCCC(OC5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)C(F)(F)F)CC4)=C3)C2=O)C(=O)N1	C45H47F3N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-XUWYPA	SCHEMBL20232039	3-[6-[4-[[5-[[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]methyl]pyridin-2-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC5=CC=C(COC6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=CC=C7)C=C6)C=N5)CC4)=C3)C2=O)C(=O)N1	C46H45N5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-OTR932	WO2018102725A1_449	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC5CCN(C6=CC=C([C@H]7C8=C(C=C(O)C=C8)CC[C@H]7C7=CC=C(F)C=C7)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C45H48FN5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-V6PLWP	WO2018102725A1_450	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC5CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=C(F)C=C7)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C45H48FN5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-AL503U	WO2018102725A1_451	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC5CCN(C6=CC=CC([C@H]7C8=C(C=C(O)C=C8)CC[C@H]7C7=CC=CC=C7)=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C45H49N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-KPSXKY	WO2018102725A1_452	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC5CCN(C6=CC=CC([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C45H49N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-RW1AEN	WO2018102725A1_453	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCC5CCN(C6=CC=CC([C@H]7C8=C(C=C(O)C=C8)CC[C@H]7C7=CC=CC=C7)=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C46H51N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-RM5J4Y	WO2018102725A1_454	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCC5CCN(C6=CC=CC([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C46H51N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-H6IV9V	WO2018102725A1_455	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC5CCN(C6=C(F)C=C([C@H]7C8=C(C=C(O)C=C8)CC[C@H]7C7=CC=CC=C7)C=C6F)CC5)CC4)=C3)C2=O)C(=O)N1	C45H47F2N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-8MPDI5	WO2018102725A1_456	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC5CCN(C6=C(F)C=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6F)CC5)CC4)=C3)C2=O)C(=O)N1	C45H47F2N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-L50P84	WO2018102725A1_457	.	O=C1CCC(N2C(=O)C3=C(C=C(N4CCN(CC5CCN(C6=C(F)C=C([C@H]7C8=C(C=C(O)C=C8)CC[C@H]7C7=CC=CC=C7)C=C6F)CC5)CC4)C=C3)C2=O)C(=O)N1	C45H45F2N5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-16SIKY	WO2018102725A1_458	.	O=C1CCC(N2C(=O)C3=C(C=C(N4CCN(CC5CCN(C6=C(F)C=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6F)CC5)CC4)C=C3)C2=O)C(=O)N1	C45H45F2N5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-05JIT8	WO2018102725A1_459	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC5CCN(C6=C(F)C=C([C@H]7C8=C(C=C(O)C=C8)CC[C@H]7C7=CC=CC=C7)C=C6F)CC5)CC4)=N3)C2=O)C(=O)N1	C44H46F2N6O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-POG3L1	WO2018102725A1_460	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC5CCN(C6=C(F)C=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6F)CC5)CC4)=N3)C2=O)C(=O)N1	C44H46F2N6O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-CUIXNR	WO2018102725A1_461	.	O=C1CCC(N2CC3=C(C=NC(N4CCN(CC5CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C44H48N6O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-9SMP5V	WO2018102725A1_462	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC5CCN(C6=NC=C([C@H]7C8=C(C=C(O)C=C8)CC[C@H]7C7=CC=CC=C7)C=N6)CC5)CC4)=C3)C2=O)C(=O)N1	C43H47N7O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-EXDB9F	WO2018102725A1_463	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC5CCN(C6=NC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=N6)CC5)CC4)=C3)C2=O)C(=O)N1	C43H47N7O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-UECBLN	WO2018102725A1_464	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(C5CC6(CCN(C7=CC=C([C@H]8C9=C(C=C(O)C=C9)CC[C@H]8C8=CC=CC=C8)C=C7)CC6)C5)CC4)=C3)C2=O)C(=O)N1	C47H51N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-0NSBRA	SCHEMBL23350031	3-[6-[4-[7-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-7-azaspiro[3.5]nonan-2-yl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(N4CCN(C5CC6(CCN(C7=CC=C([C@@H]8C9=C(C=C(O)C=C9)CC[C@@H]8C8=CC=CC=C8)C=C7)CC6)C5)CC4)=C3)C2=O)C(=O)N1	C47H51N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-AO7Z6P	WO2018102725A1_466	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(C5CC6(CCN(C7=CC=C([C@H]8C9=C(C=C(O)C=C9)CC[C@H]8C8=CC=CC=C8)C=C7)CC6)C5)CC4)=N3)C2=O)C(=O)N1	C46H50N6O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-HR6SQX	WO2018102725A1_467	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(C5CC6(CCN(C7=CC=C([C@@H]8C9=C(C=C(O)C=C9)CC[C@@H]8C8=CC=CC=C8)C=C7)CC6)C5)CC4)=N3)C2=O)C(=O)N1	C46H50N6O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-92ILM9	WO2018102725A1_468	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCC5CCN(C6=C(F)C=C([C@H]7C8=C(C=C(O)C=C8)CC[C@H]7C7=CC=CC=C7)C=C6F)CC5)CC4)=C3)C2=O)C(=O)N1	C46H49F2N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-23CYQH	WO2018102725A1_469	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCC5CCN(C6=C(F)C=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6F)CC5)CC4)=C3)C2=O)C(=O)N1	C46H49F2N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-YQOLGW	WO2018102725A1_470	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCC5CCN(C6=CC=C([C@H]7C8=C(C=C(O)C=C8)CC[C@H]7C7=CC=CC=C7)C=C6F)CC5)CC4)=C3)C2=O)C(=O)N1	C46H50FN5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-OZ7BL3	WO2018102725A1_471	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCC5CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6F)CC5)CC4)=C3)C2=O)C(=O)N1	C46H50FN5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-RI3DDA	WO2018102725A1_472	.	O=C1CCC(N2CC3=C(C=NC(N4CCN(CCC5CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C45H50N6O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-TEY6AU	WO2018102725A1_473	.	CC1(CN2CCN(C3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4)CC2)CCN(C2=CC=C([C@H]3C4=C(C=C(O)C=C4)CC[C@H]3C3=CC=CC=C3)C=C2)CC1	C46H51N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-H9TNOG	WO2018102725A1_474	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC5CCN(C6=C(F)C=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=N3)C2=O)C(=O)N1	C44H47FN6O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-VN6JZ3	WO2018102725A1_475	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC5CCN(C6=CC=C([C@H]7C8=C(C=C(O)C=C8)CC[C@H]7C7=CC=C(F)C=C7)C=C6)CC5)CC4)=N3)C2=O)C(=O)N1	C44H47FN6O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-NR5TN7	WO2018102725A1_476	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC5CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=C(F)C=C7)C=C6)CC5)CC4)=N3)C2=O)C(=O)N1	C44H47FN6O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-3O9Y8X	WO2018102725A1_477	.	O=C1CCC(N2CC3=C(C=C(F)C(N4CCN(CC5CCN(C6=CC=C([C@H]7C8=C(C=C(O)C=C8)CC[C@H]7C7=CC=C(F)C=C7)C=C6)CC5)CC4)=C3F)C2=O)C(=O)N1	C45H46F3N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-XB4HD6	WO2018102725A1_478	.	O=C1CCC(N2CC3=C(C=C(F)C(N4CCN(CC5CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=C(F)C=C7)C=C6)CC5)CC4)=C3F)C2=O)C(=O)N1	C45H46F3N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-2TK7O6	WO2018102725A1_479	.	O=C1CC[C@H](N2CC3=C(C=CC(OC4CCN(CC5CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C46H50N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-TQU5NB	WO2018102725A1_480	.	O=C1CCC(N2CC3=C(C=CC(N4CCC(NCC5CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)C4)=N3)C2=O)C(=O)N1	C44H48N6O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-FU5GX8	WO2018102725A1_481	.	COC1=CC=C([C@@H]2CCC3=C(C=CC(O)=C3)[C@@H]2C2=CC=C(N3CCC(CN4CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6)CC4)CC3)C=C2)C=C1	C46H51N5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-04E2CM	SCHEMBL21982925	3-[6-[4-[[1-[4-[(1R,2S)-6-hydroxy-2-(4-methoxyphenyl)-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	COC1=CC=C([C@H]2CCC3=C(C=CC(O)=C3)[C@H]2C2=CC=C(N3CCC(CN4CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6)CC4)CC3)C=C2)C=C1	C46H51N5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-KECYM9	WO2018102725A1_483	3-[7-fluoro-6-[4-[[1-[4-[(1S,2R)-2-(4-fluorophenyl)-6-hydroxy-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC5CCN(C6=CC=C([C@H]7C8=C(C=C(O)C=C8)CC[C@H]7C7=CC=C(F)C=C7)C=C6)CC5)CC4)=C3F)C2=O)C(=O)N1	C45H47F2N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-42FBXW	WO2018102725A1_484	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC5CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=C(F)C=C7)C=C6)CC5)CC4)=C3F)C2=O)C(=O)N1	C45H47F2N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-7AF0QN	WO2018102725A1_485	.	O=C1CCC(N2CC3=C(C=C(N4CCN(CC5CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)C=C3)C2=O)C(=O)N1	C45H49N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-IUTY8J	WO2018102725A1_486	.	O=C1CCC(N2CC3=C(C=CC(N4CC[C@H](NCC5CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)C4)=C3)C2=O)C(=O)N1	C45H49N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-5DJS2Q	WO2018102725A1_487	.	O=C1CCC(N2CC3=C(C=CC(N4CC[C@@H](NCC5CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)C4)=C3)C2=O)C(=O)N1	C45H49N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-S6PTYR	WO2018102725A1_488	3-[6-[4-[[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]-1-methylpiperidine-2,6-dione	CN1C(=O)CCC(N2CC3=C(C=CC(N4CCN(CC5CCN(C6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=C3)C2=O)C1=O	C46H51N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-SD06T0	WO2018102725A1_489	3-[6-[4-[[1-[2-fluoro-4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]-1-methylpiperidine-2,6-dione	CN1C(=O)CCC(N2CC3=C(C=CC(N4CCN(CC5CCN(C6=C(F)C=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=C3)C2=O)C1=O	C46H50FN5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-SVZV4S	WO2018102725A1_490	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC5(O)CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C45H49N5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-RKRPV2	SCHEMBL20231813	3-[6-[4-[[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-4-methylpiperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CC1(CN2CCN(C3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4)CC2)CCN(C2=CC=C([C@@H]3C4=C(C=C(O)C=C4)CC[C@@H]3C3=CC=CC=C3)C=C2)CC1	C46H51N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-Y240KH	WO2018102725A1_492	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC5CC6(CCN(C7=CC=C([C@@H]8C9=C(C=C(O)C=C9)CC[C@@H]8C8=CC=CC=C8)C=C7)C6)C5)CC4)=C3)C2=O)C(=O)N1	C47H51N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-9NYN3I	WO2018102725A1_493	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC5CC6(CCN(C7=CC=C([C@@H]8C9=C(C=C(O)C=C9)CC[C@@H]8C8=CC=CC=C8)C=C7)C6)C5)CC4)=N3)C2=O)C(=O)N1	C46H50N6O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-DE2CZH	SCHEMBL20234560	3-[6-[4-[[1-[4-[(1R,2S)-2-(4-fluorophenyl)-6-hydroxy-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-4-hydroxypiperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC5(O)CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=C(F)C=C7)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C45H48FN5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-06KROW	WO2018102725A1_495	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC5CCN(C6=CC=C([C@H]7C8=C(C=C(O)C=C8)CC[C@H]7C7=CC=CC=C7)C(F)=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C45H48FN5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-9IFP6U	SCHEMBL20211903	3-[6-[4-[[1-[3-fluoro-4-[(1S,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL29683774	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC5CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C(F)=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C45H48FN5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-V2WG6Q	WO2018102725A1_497	.	O=C1CCC(N2CC3=C(C=CC(N4CCC(NCC5CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C46H51N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-FSFTJU	WO2018102725A1_498	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC5CCN(C6=CC=C([C@H]7C8=C(C=C(O)C=C8)CC[C@H]7C7=CC=CC=C7)C(F)=C6)CC5)CC4)=N3)C2=O)C(=O)N1	C44H47FN6O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-42QQ0D	WO2018102725A1_499	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC5CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C(F)=C6)CC5)CC4)=N3)C2=O)C(=O)N1	C44H47FN6O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-8MP5NN	SCHEMBL20231560	3-[6-[4-[[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]amino]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(N4CCC(NC5CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C45H49N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-3OES5D	WO2018102725A1_501	3-[6-[4-[[4-fluoro-1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC5(F)CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C45H48FN5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-HX2G28	WO2018102725A1_502	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC5(F)CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=N3)C2=O)C(=O)N1	C44H47FN6O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-ITRZSQ	WO2018102725A1_503	.	CC1C2=C(C=CC(N3CCN(CC4CCN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)CC3)=C2)C(=O)N1C1CCC(=O)NC1=O	C46H51N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-JGUI7N	WO2018102725A1_504	.	O=C1CCC(N2CC3=CC=C(N4CCN(CCC5CCN(C6=CC=C([C@H]7C8=C(C=C(O)C=C8)CC[C@H]7C7=CC=CC=C7)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C46H51N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-2HS95D	WO2018102725A1_505	.	O=C1CCC(N2CC3=CC=C(N4CCN(CCC5CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C46H51N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-MVPF5U	WO2018102725A1_506	.	O=C1CCC(N2CC3=CC(N4CCN(CC5CCN(C6=CC=C([C@H]7C8=C(C=C(O)C=C8)CC[C@H]7C7=CC=C(O)C=C7)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C45H49N5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-FGP8LY	SCHEMBL23051715	3-[6-[4-[[1-[4-[(1R,2S)-6-hydroxy-2-(4-hydroxyphenyl)-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(N4CCN(CC5CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=C(O)C=C7)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C45H49N5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-OWVGGV	WO2018102725A1_508	.	O=C1CCC(N2CC3=NC(N4CCN(CCC5CCN(C6=CC=C([C@H]7C8=C(C=C(O)C=C8)CC[C@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C45H50N6O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-Q3K2HN	WO2018102725A1_509	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCC5CCN(C6=CC=C([C@H]7C8=C(C=C(O)C=C8)CC[C@H]7C7=CC=CC=C7)C=C6)C5)CC4)=N3)C2=O)C(=O)N1	C44H48N6O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-P3OLZY	WO2018102725A1_510	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCC5CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)C5)CC4)=N3)C2=O)C(=O)N1	C44H48N6O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-DJVS8U	WO2018102725A1_511	.	CC1C2=C(C=CC(N3CCN(CC4CCN(C5=C(F)C=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)CC3)=C2)C(=O)N1C1CCC(=O)NC1=O	C46H50FN5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-AIIKFT	WO2018102725A1_512	.	O=C1CCC(N2CC3=CC(N4CCN(CCC5CCN(C6=CC=C([C@H]7C8=C(C=C(O)C=C8)CC[C@H]7C7=CC=C(O)C=C7)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C46H51N5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-MRBKKK	SCHEMBL22297079	2-(2,6-dioxopiperidin-3-yl)-5-[3-[[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl-propan-2-ylamino]cyclobutyl]oxyisoindole-1,3-dione	CC(C)N(CC1CCN(C2=CC=C([C@@H]3C4=C(C=C(O)C=C4)CC[C@@H]3C3=CC=CC=C3)C=C2)CC1)[C@H]1C[C@H](OC2=CC3=C(C=C2)C(=O)N(C2CCC(=O)NC2=O)C3=O)C1	C48H52N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-XADWDG	WO2018102725A1_514	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCC5CCN(C6=NC=C([C@H]7C8=C(C=C(O)C=C8)CC[C@H]7C7=CC=CC=C7)C=N6)CC5)CC4)=C3)C2=O)C(=O)N1	C44H49N7O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-OVQVQJ	WO2018102725A1_515	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCC5CCN(C6=NC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=N6)CC5)CC4)=C3)C2=O)C(=O)N1	C44H49N7O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-25Q7M3	WO2018102725A1_516	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCC5CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)C5)CC4)=C3)C2=O)C(=O)N1	C45H49N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-EUU3FP	WO2018102725A1_517	.	COC1=CC=C([C@@H]2CCC3=C(C=CC(O)=C3)[C@@H]2C2=CC=C(N3CCC(CCN4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)CC6=C5)CC4)CC3)C=C2)C=C1	C47H53N5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-NIK3TL	WO2018102725A1_518	.	COC1=CC=C([C@H]2CCC3=C(C=CC(O)=C3)[C@H]2C2=CC=C(N3CCC(CCN4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)CC6=C5)CC4)CC3)C=C2)C=C1	C47H53N5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-ZR803V	WO2018102725A1_519	.	O=C1CCC(N2CC3=CC(N4CCN(CCC5CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=C(O)C=C7)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C46H51N5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-0R9J1D	SCHEMBL20231437	3-[6-[3-[[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl-propan-2-ylamino]cyclobutyl]oxy-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CC(C)N(CC1CCN(C2=CC=C([C@@H]3C4=C(C=C(O)C=C4)CC[C@@H]3C3=CC=CC=C3)C=C2)CC1)[C@H]1C[C@H](OC2=CC3=C(C=C2)C(=O)N(C2CCC(=O)NC2=O)C3)C1	C48H54N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-OQP1S6	SCHEMBL20235039	3-[2-[4-[[4-hydroxy-1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-5-oxo-7H-pyrrolo[3,4-b]pyridin-6-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC5(O)CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=N3)C2=O)C(=O)N1	C44H48N6O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-DNBQM5	WO2018102725A1_522	3-[6-[4-hydroxy-4-[[4-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperazin-1-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(N4CCC(O)(CN5CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C45H49N5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-K4Y01K	SCHEMBL20231947	3-[6-[4-[3-[2-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]ethyl]azetidin-1-yl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(N4CCC(N5CC(CCOC6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)C5)CC4)=CC=C3C2=O)C(=O)N1	C45H48N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-0KK29Q	SCHEMBL20211934	(3S)-3-[6-[4-[[1-[2-fluoro-4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CC[C@H](N2CC3=C(C=CC(N4CCN(CC5CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6F)CC5)CC4)=C3)C2=O)C(=O)N1	C45H48FN5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-2Z1T3V	SCHEMBL20232063	(3R)-3-[6-[4-[[1-[2-fluoro-4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL29683643	O=C1CC[C@@H](N2CC3=C(C=CC(N4CCN(CC5CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6F)CC5)CC4)=C3)C2=O)C(=O)N1	C45H48FN5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-X09P6O	SCHEMBL21982924	3-[6-[3-[4-[2-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]ethyl]piperidin-1-yl]cyclobutyl]oxy-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(O[C@H]4C[C@@H](N5CCC(CCOC6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)C4)=C3)C2=O)C(=O)N1	C46H49N3O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-IKL6TD	WO2018102725A1_527	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCO[C@H]5CCN(C6=CC=C([C@H]7C8=C(C=C(O)C=C8)CC[C@H]7C7=CC=CC=C7)C=C6)C5)CC4)=C3)C2=O)C(=O)N1	C45H49N5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-Y7NOCC	WO2018102725A1_528	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCO[C@H]5CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)C5)CC4)=C3)C2=O)C(=O)N1	C45H49N5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-ULPLW2	WO2018102725A1_529	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCO[C@@H]5CCN(C6=CC=C([C@H]7C8=C(C=C(O)C=C8)CC[C@H]7C7=CC=CC=C7)C=C6)C5)CC4)=C3)C2=O)C(=O)N1	C45H49N5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-A6LX5V	WO2018102725A1_530	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCO[C@@H]5CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)C5)CC4)=C3)C2=O)C(=O)N1	C45H49N5O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-QSRGDE	WO2018102725A1_531	.	O=C1CCC(N2CC3=C(C=CC(O[C@H]4C[C@@H](N5CCC(COC6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)C4)=C3)C2=O)C(=O)N1	C45H47N3O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-4FA5DQ	WO2018102725A1_532	3-[6-[3-[4-[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]ethyl]piperidin-1-yl]cyclobutyl]oxy-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CC(OC1=CC=C([C@@H]2C3=C(C=C(O)C=C3)CC[C@@H]2C2=CC=CC=C2)C=C1)C1CCN([C@H]2C[C@@H](OC3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4)C2)CC1	C46H49N3O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-1816HA	WO2018102725A1_533	.	O=C1CCC(N2CC3=C(C=CC(O[C@H]4CCN(CC5CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)C4)=C3)C2=O)C(=O)N1	C45H48N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-5GCS8E	WO2018102725A1_534	.	O=C1CCC(N2CC3=CC(N4CCC(C5CN(CCOC6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)C5)CC4)=CC=C3C2=O)C(=O)N1	C45H48N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-L6XAFJ	WO2018102725A1_535	.	O=C1CCC(N2CC3=C(C=CC(O[C@H]4C[C@@H](N5CCN(CCOC6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)C4)=C3)C2=O)C(=O)N1	C45H48N4O6	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-CREMPE	WO2018102725A1_536	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC5CCN(C6=CC=C([C@H]7C8=C(C=C(O)C=C8)CC[C@H]7C7=CC=CC=C7)N=N6)CC5)CC4)=C3)C2=O)C(=O)N1	C43H47N7O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-1CAHL3	WO2018102725A1_537	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC5CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)N=N6)CC5)CC4)=C3)C2=O)C(=O)N1	C43H47N7O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-PB3195	WO2018102725A1_538	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCC5CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)N=N6)CC5)CC4)=C3)C2=O)C(=O)N1	C44H49N7O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-R2WZ0C	WO2018102725A1_539	.	O=C1CCC(N2CC3=C(C=CC(C4=CN(C5CN(CC6CCN(C7=CC=C([C@@H]8C9=C(C=C(O)C=C9)CC[C@@H]8C8=CC=CC=C8)C=C7)CC6)C5)N=C4)=C3)C2=O)C(=O)N1	C47H48N6O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-4N68ZT	WO2018102725A1_540	.	O=C1CC[C@H](N2CC3=C(C=CC(O[C@@H]4CCN(CC5CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)C4)=C3)C2=O)C(=O)N1	C45H48N4O5	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-IJHVMM	SCHEMBL20235048	3-[6-[1-[2-[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]ethyl]pyrazol-4-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(C4=CN(CCC5CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)N=C4)=C3)C2=O)C(=O)N1	C45H45N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-N0DRXB	WO2018102725A1_542	.	O=C1CCC(N2CC3=C(C=CC(C4=CN(C5CN(C[C@@H]6CCN(C7=CC=C([C@@H]8C9=C(C=C(O)C=C9)CC[C@@H]8C8=CC=CC=C8)C=C7)C6)C5)N=C4)=C3)C2=O)C(=O)N1	C46H46N6O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-AFNC5V	WO2018102725A1_543	.	O=C1CCC(N2CC3=C(C=CC(C4=CN(C5CN(C[C@@H]6CCN(C7=CC=C([C@H]8C9=C(C=C(O)C=C9)CC[C@H]8C8=CC=CC=C8)C=C7)C6)C5)N=C4)=C3)C2=O)C(=O)N1	C46H46N6O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-SFRMUL	WO2018102725A1_544	.	O=C1CCC(N2CC3=C(C=CC(C4=CN(C5CN(C[C@H]6CCN(C7=CC=C([C@@H]8C9=C(C=C(O)C=C9)CC[C@@H]8C8=CC=CC=C8)C=C7)C6)C5)N=C4)=C3)C2=O)C(=O)N1	C46H46N6O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-SMGP7M	WO2018102725A1_545	.	O=C1CCC(N2CC3=C(C=CC(C4=CN(C5CN(C[C@H]6CCN(C7=CC=C([C@H]8C9=C(C=C(O)C=C9)CC[C@H]8C8=CC=CC=C8)C=C7)C6)C5)N=C4)=C3)C2=O)C(=O)N1	C46H46N6O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-W78TD9	WO2018102725A1_546	.	O=C1CC[C@@H](N2CC3=C(C=CC(N4CCN(CC5CCN(C6=CC(F)=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C(F)=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C45H47F2N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-PR3R7W	WO2018102725A1_547	.	O=C1CC[C@H](N2CC3=C(C=CC(N4CCN(CC5CCN(C6=CC(F)=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C(F)=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C45H47F2N5O4	ERα;ERβ	P03372/Q92731	CRBN	WO-2018102725-A1
TPD-6VMZRD	SCHEMBL24079446	1-cyclopentyl-N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-6-[4-[[4-[2-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]ethyl]piperazin-1-yl]methyl]phenyl]indole-4-carboxamide	CC1=CC(C)=C(CNC(=O)C2=C3C=CN(C4CCCC4)C3=CC(C3=CC=C(CN4CCN(CCOCC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)NCC5=CC=C(C6=C(C)N=CS6)C=C5)C(C)(C)C)CC4)C=C3)=C2)C(=O)N1	C59H73N9O7S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-WRS8VZ	WO2018119357A1_2	.	CC1=CC(C)=C(CCC(=O)C2=C3C=CN(C4CCCC4)C3=CC(C3=CC=C(CN4CCN(CCOCCOCC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)NCC5=CC=C(C6=C(C)N=CS6)C=C5)C(C)(C)C)CC4)C=C3)=C2)C(=O)N1	C62H78N8O8S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-YPTE64	SCHEMBL24079444	1-cyclopentyl-N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-6-[4-[[4-[2-[4-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]butoxy]ethyl]piperazin-1-yl]methyl]phenyl]indole-4-carboxamide	CC1=CC(C)=C(CNC(=O)C2=C3C=CN(C4CCCC4)C3=CC(C3=CC=C(CN4CCN(CCOCCCCOCC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)NCC5=CC=C(C6=C(C)N=CS6)C=C5)C(C)(C)C)CC4)C=C3)=C2)C(=O)N1	C63H81N9O8S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-8Q7RWY	SCHEMBL20294981	1-cyclopentyl-N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-6-[4-[[4-[2-[3-[3-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]propoxy]propoxy]ethyl]piperazin-1-yl]methyl]phenyl]indole-4-carboxamide	CC1=CC(C)=C(CNC(=O)C2=C3C=CN(C4CCCC4)C3=CC(C3=CC=C(CN4CCN(CCOCCCOCCCOCC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)NCC5=CC=C(C6=C(C)N=CS6)C=C5)C(C)(C)C)CC4)C=C3)=C2)C(=O)N1	C65H85N9O9S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-3VB0BW	SCHEMBL20317468	1-cyclopentyl-N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-6-[4-[[4-[2-[4-[4-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]butoxy]butoxy]ethyl]piperazin-1-yl]methyl]phenyl]indole-4-carboxamide	CC1=CC(C)=C(CNC(=O)C2=C3C=CN(C4CCCC4)C3=CC(C3=CC=C(CN4CCN(CCOCCCCOCCCCOCC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)NCC5=CC=C(C6=C(C)N=CS6)C=C5)C(C)(C)C)CC4)C=C3)=C2)C(=O)N1	C67H89N9O9S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-GFYJDZ	SCHEMBL26973852	1-cyclopentyl-N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-6-[4-[[4-[2-[5-[5-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]pentoxy]pentoxy]ethyl]piperazin-1-yl]methyl]phenyl]indole-4-carboxamide	CC1=CC(C)=C(CNC(=O)C2=C3C=CN(C4CCCC4)C3=CC(C3=CC=C(CN4CCN(CCOCCCCCOCCCCCOCC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)NCC5=CC=C(C6=C(C)N=CS6)C=C5)C(C)(C)C)CC4)C=C3)=C2)C(=O)N1	C69H93N9O9S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-4ESIRA	SCHEMBL20294903	N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-1-[1-[1-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]acetyl]piperidin-4-yl]ethyl]-2-methylindole-3-carboxamide	CC1=CC(C)=C(CNC(=O)C2=C(C)N(C(C)C3CCN(C(=O)COCCOCCOCCNC4=CC=CC5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)C3=C2C=CC=C3)C(=O)N1	C46H55N7O10	EZH2	Q15910	CRBN	WO-2018119357-A1
TPD-0U5Y7I	SCHEMBL20331294	N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-1-[1-[1-[2-[2-[2-[2-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]ethoxy]ethoxy]ethoxy]acetyl]piperidin-4-yl]ethyl]-2-methylindole-3-carboxamide	CC1=CC(C)=C(CNC(=O)C2=C(C)N(C(C)C3CCN(C(=O)COCCOCCOCCOCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)NCC4=CC=C(C5=C(C)N=CS5)C=C4)C(C)(C)C)CC3)C3=C2C=CC=C3)C(=O)N1	C57H76N8O11S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-2VIMGK	SCHEMBL20294867	N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-1-[1-[1-[2-[2-[2-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]ethoxy]ethoxy]acetyl]piperidin-4-yl]ethyl]-2-methylindole-3-carboxamide	CC1=CC(C)=C(CNC(=O)C2=C(C)N(C(C)C3CCN(C(=O)COCCOCCOCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)NCC4=CC=C(C5=C(C)N=CS5)C=C4)C(C)(C)C)CC3)C3=C2C=CC=C3)C(=O)N1	C55H72N8O10S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-BUG8WV	WO2018119357A1_10	.	CC1=CC(C)=C(CNC(=O)C2=C(C)N(C(C)C3CCN(C(=O)COCCOCCOCCOCCC(=O)C4=CC=CC5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)C3=C2C=CC=C3)C(=O)N1	C49H58N6O12	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-72057P	WO2018119357A1_11	.	CC1=CC(C)=C(CNC(=O)C2C3=C(C=CC=C3)N(C(C)C3CCN(C(=O)COCCOCCOCCOCCOCC(=O)N[C@H](C(=O)N4C[C@H](O)CC4C(=O)NCC4=CC=C(C5=C(C)N=CS5)C=C4)C(C)(C)C)CC3)C2C)C(=O)N1	C59H82N8O12S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-19IDFY	WO2018119357A1_12	.	CC1=CC(C)=C(CNC(O)C2C3=C(C=CC=C3)N(C(C)C3CCN(C(=O)COCCOCCOCCOCCOCCNC4=CC=CC5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)C2C)C(=O)N1	C50H67N7O12	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-LJ5WOO	SCHEMBL20295019	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[2-[4-[3-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methylcarbamoyl]-5-[ethyl(oxan-4-yl)amino]-4-methylphenyl]phenoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL30098672; PD172380	CCN(C1=CC(C2=CC=C(OCCOCCOCCOCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCC3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C59H77N7O11S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-8NNVVG	SCHEMBL20294902	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[2-[2-[4-[3-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methylcarbamoyl]-5-[ethyl(oxan-4-yl)amino]-4-methylphenyl]phenoxy]ethoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL30098680	CCN(C1=CC(C2=CC=C(OCCOCCOCCOCCOCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCC3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C61H81N7O12S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-WR4JYM	SCHEMBL20295023	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[2-[2-[2-[4-[3-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methylcarbamoyl]-5-[ethyl(oxan-4-yl)amino]-4-methylphenyl]phenoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL30098778	CCN(C1=CC(C2=CC=C(OCCOCCOCCOCCOCCOCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCC3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C63H85N7O13S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-XU8APD	SCHEMBL20295017	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[2-[2-[2-[2-[4-[3-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methylcarbamoyl]-5-[ethyl(oxan-4-yl)amino]-4-methylphenyl]phenoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL30098698	CCN(C1=CC(C2=CC=C(OCCOCCOCCOCCOCCOCCOCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCC3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C65H89N7O14S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-SPS2A3	SCHEMBL20294931	N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-5-[4-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethoxy]phenyl]-3-[ethyl(oxan-4-yl)amino]-2-methylbenzamide; SCHEMBL30098708	CCN(C1=CC(C2=CC=C(OCCOCCOCCOCCNC3=CC=CC4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C50H60N6O11	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-68FO0Q	SCHEMBL20294888	N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-5-[4-[2-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]phenyl]-3-[ethyl(oxan-4-yl)amino]-2-methylbenzamide; SCHEMBL30098697	CCN(C1=CC(C2=CC=C(OCCOCCOCCOCCOCCNC3=CC=CC4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C52H64N6O12	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-3037X8	SCHEMBL20294922	N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-5-[4-[2-[2-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]phenyl]-3-[ethyl(oxan-4-yl)amino]-2-methylbenzamide	CCN(C1=CC(C2=CC=C(OCCOCCOCCOCCOCCOCCNC3=CC=CC4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C54H68N6O13	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-IXTYN8	SCHEMBL20295014	N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-5-[4-[2-[2-[2-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]phenyl]-3-[ethyl(oxan-4-yl)amino]-2-methylbenzamide	CCN(C1=CC(C2=CC=C(OCCOCCOCCOCCOCCOCCOCCNC3=CC=CC4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C56H72N6O14	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-PVDDQG	SCHEMBL20295043	N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-5-[3-[2-[2-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]phenyl]-3-[ethyl(oxan-4-yl)amino]-2-methylbenzamide	CCN(C1=CC(C2=CC=CC(OCCOCCOCCOCCOCCOCCNC3=CC=CC4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C54H68N6O13	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-TU6DA8	SCHEMBL20294929	N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-5-[4-[2-[2-[2-[2-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]phenyl]-3-[ethyl(oxan-4-yl)amino]-2-methylbenzamide; SCHEMBL30098705	CCN(C1=CC(C2=CC=C(OCCOCCOCCOCCOCCOCCOCCOCCNC3=CC=CC4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C58H76N6O15	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-MN4SLV	SCHEMBL20295049	N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-5-[4-[2-[2-[2-[2-[2-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]phenyl]-3-[ethyl(oxan-4-yl)amino]-2-methylbenzamide	CCN(C1=CC(C2=CC=C(OCCOCCOCCOCCOCCOCCOCCOCCOCCNC3=CC=CC4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C60H80N6O16	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-Y582QR	SCHEMBL20294986	N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-5-[2-[2-[2-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]phenyl]-3-[ethyl(oxan-4-yl)amino]-2-methylbenzamide; SCHEMBL30098740	CCN(C1=CC(C2=CC=CC=C2OCCOCCOCCOCCOCCOCCNC2=CC=CC3=C2C(=O)N(C2CCC(=O)NC2=O)C3=O)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C54H68N6O13	EZH2	Q15910	CRBN	WO-2018119357-A1
TPD-2UBU1P	SCHEMBL27127786	5-[4-[2-[2-[2-[4-[2-[(3aR,7aS)-1-[2-cyclohexyl-2-[2-(methylamino)propanoylamino]acetyl]-3,3a,4,5,7,7a-hexahydro-2H-pyrrolo[2,3-c]pyridin-6-yl]ethyl]phenoxy]ethoxy]ethoxy]ethoxy]phenyl]-N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-3-[ethyl(oxan-4-yl)amino]-2-methylbenzamide	[H][C@]12CCN(CCC3=CC=C(OCCOCCOCCOC4=CC=C(C5=CC(C(=O)NCC6=C(C)C=C(C)NC6=O)=C(C)C(N(CC)C6CCOCC6)=C5)C=C4)C=C3)C[C@@]1([H])N(C(=O)C(NC(=O)C(C)NC)C1CCCCC1)CC2	C62H87N7O9	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-YPILVW	WO2018119357A1_28	.	CCN(C1=CC(C2=CC=C(OCCOCCOCCOC3=C4C=CC=CC4=C(C4=COC([C@@H]5CCCN5C(=O)[C@@H](NC(=O)[C@H](C)NC)C5CCCCC5)=N4)C=C3)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C64H81N7O10	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-1AO5O4	SCHEMBL20294964	5-[4-[2-[2-[2-[2-[2-[4-[2-[(3aR,7aS)-1-[(2S)-2-cyclohexyl-2-[[(2S)-2-(methylamino)propanoyl]amino]acetyl]-3,3a,4,5,7,7a-hexahydro-2H-pyrrolo[2,3-c]pyridin-6-yl]ethyl]phenoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]phenyl]-N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-3-[ethyl(oxan-4-yl)amino]-2-methylbenzamide; SCHEMBL30098684	[H][C@]12CCN(CCC3=CC=C(OCCOCCOCCOCCOCCOC4=CC=C(C5=CC(C(=O)NCC6=C(C)C=C(C)NC6=O)=C(C)C(N(CC)C6CCOCC6)=C5)C=C4)C=C3)C[C@@]1([H])N(C(=O)[C@@H](NC(=O)[C@H](C)NC)C1CCCCC1)CC2	C66H95N7O11	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-LY70KV	WO2018119357A1_30	.	CCN(C1=CC(C2=CC=C(OCCOCCOCCOCCOCCOC3=C4C=CC=CC4=C(C4=COC([C@@H]5CCCN5C(=O)[C@@H](NC(=O)[C@H](C)NC)C5CCCCC5)=N4)C=C3)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C68H89N7O12	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-Z0AO4R	WO2018119357A1_31	.	CCN(C1=CC(C2=CC=C(OCCOCCOCCN[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCC3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C57H75N7O9S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-E9XXGH	SCHEMBL20330431	(2S,4R)-1-[(2S)-2-[[2-[2-[4-[3-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methylcarbamoyl]-5-[ethyl(oxan-4-yl)amino]-4-methylphenyl]phenoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL30098658; PD172372	CCN(C1=CC(C2=CC=C(OCCOCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCC3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C55H69N7O9S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-PE186U	WO2018119357A1_33	.	CNC(C1=CC(C2=CC=C(OCCOCCOCCNC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C48H56N6O10	EZH2	Q15910	CRBN	WO-2018119357-A1
TPD-5Z60A6	WO2018119357A1_34	.	CNC(C1=CC(C2=CC=C(OCCOCCNC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C46H52N6O9	EZH2	Q15910	CRBN	WO-2018119357-A1
TPD-0PCBE2	WO2018119357A1_35	.	CNC(C1=CC(C2=CC=C(OCCOCCOCCOCCOCCOC3=CC(C4=C(C)N=CS4)=CC=C3CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C68H85N7O13S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-JZYZDM	WO2018119357A1_36	.	CNC(C1=CC(C2=CC=C(OCCOCCOCCOCCOC3=CC(C4=C(C)N=CS4)=CC=C3CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C66H81N7O12S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-LUQE9D	WO2018119357A1_37	.	CNC(C1=CC(C2=CC=C(OCCOCCOCCOC3=CC(C4=C(C)N=CS4)=CC=C3CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C64H77N7O11S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-GCER6Q	WO2018119357A1_38	.	CNC(C1=CC(C2=CC=C(OCCOCCOC3=CC(C4=C(C)N=CS4)=CC=C3CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C62H73N7O10S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-P76MFC	WO2018119357A1_39	.	CNC(C1=CC(C2=CC=C(OCCCOCCCOCCCOC3=CC(C4=C(C)N=CS4)=CC=C3CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C67H83N7O11S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-4UY5W0	WO2018119357A1_40	.	CNC(C1=CC(C2=CC=C(OCCCCOCCOC3=CC(C4=C(C)N=CS4)=CC=C3CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C64H77N7O10S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-1FVWDB	YM281	CID 135147352; 2230914-84-6; orb1982938; CHEMBL5094323; SCHEMBL20294957; SCHEMBL30098660; DA-79045; PD172374; HY-145762; CS-0432576; (2S,4R)-1-[(2S)-2-[[2-[3-[4-[3-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methylcarbamoyl]-5-[ethyl(oxan-4-yl)amino]-4-methylphenyl]phenoxy]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CCN(C1=CC(C2=CC=C(OCCCOCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCC3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C56H71N7O9S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-U5PEO8	SCHEMBL24079480	(2S,4R)-1-[(2S)-2-[[2-[4-[4-[3-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methylcarbamoyl]-5-[ethyl(oxan-4-yl)amino]-4-methylphenyl]phenoxy]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL30098715	CCN(C1=CC(C2=CC=C(OCCCCOCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCC3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C57H73N7O9S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-IFY78A	SCHEMBL20294967	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[4-[3-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methylcarbamoyl]-5-[ethyl(oxan-4-yl)amino]-4-methylphenyl]phenoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL30098728	CCN(C1=CC(C2=CC=C(OCCOCCOCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](C)C3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C58H75N7O10S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-AA9FCS	SCHEMBL20317449	(2S,4R)-1-[(2S)-2-[5-[3-[4-[3-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methylcarbamoyl]-5-[ethyl(oxan-4-yl)amino]-4-methylphenyl]phenyl]propoxy]pentanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL30098704	CCN(C1=CC(C2=CC=C(CCCOCCCCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCC3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C59H77N7O8S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-W9RSBE	SCHEMBL20294886	(2S,4R)-1-[(2S)-2-[[2-[2-[3-[4-[3-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methylcarbamoyl]-5-[ethyl(oxan-4-yl)amino]-4-methylphenyl]phenoxy]propoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL30098687	CCN(C1=CC(C2=CC=C(OCCCOCCOCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCC3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C58H75N7O10S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-42LEKZ	SCHEMBL20294966	(2S,4R)-1-[(2S)-2-[[2-[5-[4-[3-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methylcarbamoyl]-5-[ethyl(oxan-4-yl)amino]-4-methylphenyl]phenoxy]pentoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL30098750	CCN(C1=CC(C2=CC=C(OCCCCCOCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCC3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C58H75N7O9S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-Q2T40C	SCHEMBL20317491	(2S,4R)-1-[(2S)-2-[[2-[2-[3-[4-[3-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methylcarbamoyl]-5-[ethyl(oxan-4-yl)amino]-4-methylphenyl]phenyl]propoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL30098667	CCN(C1=CC(C2=CC=C(CCCOCCOCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCC3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C58H75N7O9S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-CNZX68	SCHEMBL20317495	(2S,4R)-1-[(2S)-2-[[2-[3-[3-[4-[3-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methylcarbamoyl]-5-[ethyl(oxan-4-yl)amino]-4-methylphenyl]phenoxy]propoxy]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL30098718	CCN(C1=CC(C2=CC=C(OCCCOCCCOCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCC3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C59H77N7O10S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-PKRTMJ	SCHEMBL20317492	(4R)-N-[[2-[5-[2-[4-[3-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methylcarbamoyl]-5-[ethyl(oxan-4-yl)amino]-4-methylphenyl]phenoxy]ethoxy]pentoxy]-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-4-hydroxy-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]pyrrolidine-2-carboxamide	CCN(C1=CC(C2=CC=C(OCCOCCCCCOC3=C(CNC(=O)C4C[C@@H](O)CN4C(=O)[C@H](C(C)C)N4CC5=C(C=CC=C5)C4=O)C=CC(C4=C(C)N=CS4)=C3)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C65H79N7O10S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-L2UFYU	WO2018119357A1_50	.	CCN(C1=CC(C2=CC=C(OCCCCCCCCOC3=C(CNC(=O)C4C[C@@H](O)CN4C(=O)[C@H](C(C)C)N4CC5=C(C=CC=C5)C4=O)C=CC(C4=C(C)N=CS4)=C3)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C66H81N7O9S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-RLS0YU	SCHEMBL20317494	(4R)-N-[[2-[4-[3-[4-[3-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methylcarbamoyl]-5-[ethyl(oxan-4-yl)amino]-4-methylphenyl]phenoxy]propoxy]butoxy]-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-4-hydroxy-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]pyrrolidine-2-carboxamide	CCN(C1=CC(C2=CC=C(OCCCOCCCCOC3=C(CNC(=O)C4C[C@@H](O)CN4C(=O)[C@H](C(C)C)N4CC5=C(C=CC=C5)C4=O)C=CC(C4=C(C)N=CS4)=C3)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C65H79N7O10S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-F0587S	SCHEMBL20317497	(4R)-N-[[2-[3-[4-[4-[3-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methylcarbamoyl]-5-[ethyl(oxan-4-yl)amino]-4-methylphenyl]phenoxy]butoxy]propoxy]-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-4-hydroxy-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]pyrrolidine-2-carboxamide	CCN(C1=CC(C2=CC=C(OCCCCOCCCOC3=C(CNC(=O)C4C[C@@H](O)CN4C(=O)[C@H](C(C)C)N4CC5=C(C=CC=C5)C4=O)C=CC(C4=C(C)N=CS4)=C3)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C65H79N7O10S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-KCYCGN	SCHEMBL20317498	(4R)-N-[[2-[2-[4-[4-[3-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methylcarbamoyl]-5-[ethyl(oxan-4-yl)amino]-4-methylphenyl]phenoxy]butoxy]ethoxy]-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-4-hydroxy-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]pyrrolidine-2-carboxamide	CCN(C1=CC(C2=CC=C(OCCCCOCCOC3=C(CNC(=O)C4C[C@@H](O)CN4C(=O)[C@H](C(C)C)N4CC5=C(C=CC=C5)C4=O)C=CC(C4=C(C)N=CS4)=C3)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C64H77N7O10S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-C6XWTD	SCHEMBL24079424	(4R)-N-[[2-[2-[2-[3-[4-[3-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methylcarbamoyl]-5-[ethyl(oxan-4-yl)amino]-4-methylphenyl]phenoxy]propoxy]ethoxy]ethoxy]-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-4-hydroxy-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]pyrrolidine-2-carboxamide	CCN(C1=CC(C2=CC=C(OCCCOCCOCCOC3=C(CNC(=O)C4C[C@@H](O)CN4C(=O)[C@H](C(C)C)N4CC5=C(C=CC=C5)C4=O)C=CC(C4=C(C)N=CS4)=C3)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C65H79N7O11S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-P6BVC0	WO2018119357A1_55	(4R)-N-[[2-[2-[2-[4-[4-[3-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methylcarbamoyl]-5-[ethyl(oxan-4-yl)amino]-4-methylphenyl]phenoxy]butoxy]ethoxy]ethoxy]-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-4-hydroxy-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]pyrrolidine-2-carboxamide	CCN(C1=CC(C2=CC=C(OCCCCOCCOCCOC3=C(CNC(=O)C4C[C@@H](O)CN4C(=O)[C@H](C(C)C)N4CC5=C(C=CC=C5)C4=O)C=CC(C4=C(C)N=CS4)=C3)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C66H81N7O11S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-D5STU7	SCHEMBL20317496	(4R)-N-[[2-[2-[3-[4-[3-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methylcarbamoyl]-5-[ethyl(oxan-4-yl)amino]-4-methylphenyl]phenoxy]propoxy]ethoxy]-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-4-hydroxy-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]pyrrolidine-2-carboxamide	CCN(C1=CC(C2=CC=C(OCCCOCCOC3=C(CNC(=O)C4C[C@@H](O)CN4C(=O)[C@H](C(C)C)N4CC5=C(C=CC=C5)C4=O)C=CC(C4=C(C)N=CS4)=C3)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C63H75N7O10S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-FUA2GW	SCHEMBL20294907	N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-5-[4-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxyethoxy]ethoxy]phenyl]-3-[ethyl(oxan-4-yl)amino]-2-methylbenzamide; SCHEMBL30098764	CCN(C1=CC(C2=CC=C(OCCOCCOC3=CC=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C46H51N5O10	EZH2	Q15910	CRBN	WO-2018119357-A1
TPD-X2DY75	SCHEMBL20294865	N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-5-[4-[2-[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxypropoxy]ethoxy]phenyl]-3-[ethyl(oxan-4-yl)amino]-2-methylbenzamide; SCHEMBL30098664	CCN(C1=CC(C2=CC=C(OCCOCCCOC3=CC=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C47H53N5O10	EZH2	Q15910	CRBN	WO-2018119357-A1
TPD-D0B2MH	SCHEMBL20294925	(2S,4R)-1-[(2S)-2-[[2-[4-[4-[4-[3-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methylcarbamoyl]-5-[ethyl(oxan-4-yl)amino]-4-methylphenyl]phenyl]piperazin-1-yl]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL30098651	CCN(C1=C(C)C(C(=O)NCC2=C(C)C=C(C)NC2=O)=CC(C2=CC=C(N3CCN(CCCCOCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)N[C@@H](C)C4=CC=C(C5=C(C)N=CS5)C=C4)C(C)(C)C)CC3)C=C2)=C1)C1CCOCC1	C62H83N9O8S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-DO829B	SCHEMBL20295062	N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-5-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxybutoxy]phenyl]-3-[ethyl(oxan-4-yl)amino]-2-methylbenzamide; SCHEMBL30098721	CCN(C1=CC(C2=CC=C(OCCCCOC3=CC=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C46H51N5O9	EZH2	Q15910	CRBN	WO-2018119357-A1
TPD-98WXEQ	SCHEMBL20295045	N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-5-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]propoxy]phenyl]-3-[ethyl(oxan-4-yl)amino]-2-methylbenzamide	CCN(C1=CC(C2=CC=C(OCCCN3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C49H57N7O8	EZH2	Q15910	CRBN	WO-2018119357-A1
TPD-1XVHGY	SCHEMBL20317504	N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-3-[4-[3-[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxypropoxy]propoxy]phenyl]-5-[ethyl(oxan-4-yl)amino]benzamide	CCN(C1=CC(C2=CC=C(OCCCOCCCOC3=CC=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1)C1CCOCC1	C47H53N5O10	EZH2	Q15910	CRBN	WO-2018119357-A1
TPD-MU9855	WO2018119357A1_63	.	CCN(C1=CC(C2=CC=C(OCCCCOC3=CC(C4=C(C)N=CS4)=CC=C3CNC(=O)C3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C62H73N7O9S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-A7MV6F	SCHEMBL24079463	(4R)-N-[[2-[2-[4-[3-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methylcarbamoyl]-5-[ethyl(oxan-4-yl)amino]-4-methylphenyl]phenoxy]ethoxy]-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-4-hydroxy-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]pyrrolidine-2-carboxamide	CCN(C1=CC(C2=CC=C(OCCOC3=CC(C4=C(C)N=CS4)=CC=C3CNC(=O)C3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C60H69N7O9S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-OIZYYX	SCHEMBL20295038	N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-5-[2-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]propoxy]pyrimidin-5-yl]-3-[ethyl(oxan-4-yl)amino]-2-methylbenzamide; SCHEMBL30098692	CCN(C1=C(C)C(C(=O)NCC2=C(C)C=C(C)NC2=O)=CC(C2=CN=C(OCCCN3CCN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)N=C2)=C1)C1CCOCC1	C47H55N9O8	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-JNRAEL	SCHEMBL20295005	(2S,4R)-1-[(2S)-2-[5-[3-[6-[3-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methylcarbamoyl]-5-[ethyl(oxan-4-yl)amino]-4-methylphenyl]pyridin-3-yl]propoxy]pentanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL30098743	CCN(C1=CC(C2=NC=C(CCCOCCCCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCC3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C58H76N8O8S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-O99O9Z	SCHEMBL20295057	N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-5-[4-[4-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxyethoxy]ethyl]piperazin-1-yl]phenyl]-3-[ethyl(oxan-4-yl)amino]-2-methylbenzamide; SCHEMBL30098683	CCN(C1=C(C)C(C(=O)NCC2=C(C)C=C(C)NC2=O)=CC(C2=CC=C(N3CCN(CCOCCOC4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)C=C2)=C1)C1CCOCC1	C50H59N7O9	EZH2	Q15910	CRBN	WO-2018119357-A1
TPD-N844QP	SCHEMBL20294898	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[5-[3-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methylcarbamoyl]-5-[ethyl(oxan-4-yl)amino]-4-methylphenyl]pyridin-2-yl]oxyethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL30098714	CCN(C1=CC(C2=CN=C(OCCOCCOCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](C)C3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C57H74N8O10S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-DKNBED	SCHEMBL20294848	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[4-[6-[3-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methylcarbamoyl]-5-[ethyl(oxan-4-yl)amino]-4-methylphenyl]pyridin-3-yl]piperazin-1-yl]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL30098686	CCN(C1=CC(C2=NC=C(N3CCN(CCOCCOCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)NCC4=CC=C(C5=C(C)N=CS5)C=C4)C(C)(C)C)CC3)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C60H80N10O9S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-NR3WJG	WO2018119357A1_70	.	CCN(C1=CC(C2=CN=C(NCCOCCOCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCC3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C56H73N9O9S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-FDFPPM	SCHEMBL20295046	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[4-[4-[3-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methylcarbamoyl]-5-[ethyl(oxan-4-yl)amino]-4-methylphenyl]phenyl]piperazin-1-yl]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL30098716	CCN(C1=CC(C2=CC=C(N3CCN(CCOCCOCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)NCC4=CC=C(C5=C(C)N=CS5)C=C4)C(C)(C)C)CC3)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C61H81N9O9S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-SEYGB8	SCHEMBL20294976	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[4-[4-[3-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methylcarbamoyl]-5-[ethyl(oxan-4-yl)amino]-4-methylphenyl]phenyl]piperazin-1-yl]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL30098739	CCN(C1=CC(C2=CC=C(N3CCN(CCOCCOCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)N[C@@H](C)C4=CC=C(C5=C(C)N=CS5)C=C4)C(C)(C)C)CC3)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C62H83N9O9S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-14DIFA	SCHEMBL20295041	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[[5-[3-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methylcarbamoyl]-5-[ethyl(oxan-4-yl)amino]-4-methylphenyl]pyridin-2-yl]amino]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL30098713	CCN(C1=CC(C2=CN=C(NCCOCCOCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](C)C3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C57H75N9O9S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-Q2QY0Z	WO2018119357A1_74	.	CCN(C1=CC(C2=CN=C(NCCOCCOCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](C)C3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)C=C2)=CC(C(=O)NCC2=C(OC)C=C(C)NC2=O)=C1C)C1CCOCC1	C57H75N9O10S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-JDYGC0	SCHEMBL20294877	N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-5-[4-[4-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]oxy]ethoxy]ethyl]piperazin-1-yl]phenyl]-3-[ethyl(oxan-4-yl)amino]-2-methylbenzamide; SCHEMBL30098646	CCN(C1=C(C)C(C(=O)NCC2=C(C)C=C(C)NC2=O)=CC(C2=CC=C(N3CCN(CCOCCOC4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5)CC3)C=C2)=C1)C1CCOCC1	C50H61N7O8	EZH2	Q15910	CRBN	WO-2018119357-A1
TPD-QSAPXP	SCHEMBL20294921	N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-5-[4-[4-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-3-oxo-1H-isoindol-5-yl]oxy]ethoxy]ethyl]piperazin-1-yl]phenyl]-3-[ethyl(oxan-4-yl)amino]-2-methylbenzamide; SCHEMBL30098652	CCN(C1=C(C)C(C(=O)NCC2=C(C)C=C(C)NC2=O)=CC(C2=CC=C(N3CCN(CCOCCOC4=CC5=C(C=C4)CN(C4CCC(=O)NC4=O)C5=O)CC3)C=C2)=C1)C1CCOCC1	C50H61N7O8	EZH2	Q15910	CRBN	WO-2018119357-A1
TPD-169M2W	SCHEMBL20317508	(2S,4R)-1-[(2S)-2-[[2-[2-[3-[4-[3-[ethyl(oxan-4-yl)amino]-5-[(4-methoxy-6-methyl-2-oxo-1H-pyridin-3-yl)methylcarbamoyl]-4-methylphenyl]phenyl]prop-2-ynoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CCN(C1=CC(C2=CC=C(C#CCOCCOCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](C)C3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)C=C2)=CC(C(=O)NCC2=C(OC)C=C(C)NC2=O)=C1C)C1CCOCC1	C59H73N7O10S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-BGKQGL	SCHEMBL20294977	(2S,4R)-1-[(2S)-2-[[2-[2-[3-[4-[3-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methylcarbamoyl]-5-[ethyl(oxan-4-yl)amino]-4-methylphenyl]phenyl]prop-2-ynoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL30098654	CCN(C1=CC(C2=CC=C(C#CCOCCOCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](C)C3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C59H73N7O9S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-S204LM	SCHEMBL20294961	(2S,4R)-1-[(2S)-2-[[2-[2-[4-[4-[3-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methylcarbamoyl]-5-[ethyl(oxan-4-yl)amino]-4-methylphenyl]phenyl]triazol-1-yl]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL30098734	CCN(C1=CC(C2=CC=C(C3=CN(CCOCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)N[C@@H](C)C4=CC=C(C5=C(C)N=CS5)C=C4)C(C)(C)C)N=N3)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C58H72N10O8S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-188W6P	SCHEMBL20294881	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[4-[4-[3-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methylcarbamoyl]-5-[ethyl(oxan-4-yl)amino]-4-methylphenyl]phenyl]triazol-1-yl]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL30098730	CCN(C1=CC(C2=CC=C(C3=CN(CCOCCOCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)N[C@@H](C)C4=CC=C(C5=C(C)N=CS5)C=C4)C(C)(C)C)N=N3)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C60H76N10O9S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-K1MDQ0	SCHEMBL20294946	6-[2-[2-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]ethoxy]ethoxy]-N-[(4-methoxy-6-methyl-2-oxo-1H-pyridin-3-yl)methyl]-2-methyl-1-[(1S)-1-(oxan-4-yl)ethyl]indole-3-carboxamide	COC1=C(CNC(=O)C2=C(C)N([C@@H](C)C3CCOCC3)C3=CC(OCCOCCOCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)N[C@@H](C)C4=CC=C(C5=C(C)N=CS5)C=C4)C(C)(C)C)=CC=C32)C(=O)NC(C)=C1	C54H71N7O11S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-281J3Z	WO2018119357A1_82	.	COC1=C(CNC(=O)C2=CN([C@@H](C)C3CCOCC3)C3=CC(OCCOCCOCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)N[C@@H](C)C4=CC=C(C5=C(C)N=CS5)C=C4)C(C)(C)C)=CC=C23)C(=O)NC(C)=C1	C53H69N7O11S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-XJVTWR	SCHEMBL20294870	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[2-[4-[[3-chloro-4-(2-cyano-3-pyridazin-4-ylphenoxy)benzoyl]amino]-2,2,6,6-tetramethylpiperidin-1-yl]ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCN3C(C)(C)CC(NC(=O)C4=CC(Cl)=C(OC5=C(C#N)C(C6=CN=NC=C6)=CC=C5)C=C4)CC3(C)C)C(C)(C)C)C=C2)SC=N1	C58H72ClN9O9S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-EDG2KS	WO2018119357A1_84	.	CCC1=C(CNC(=O)C2=NN(C(C)C)C3=CC(C4=CC=C(N5CCN(CCOCCOCCOCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)(C)C)CC5)N=C4)=CC=C32)C(=O)NC(C)=C1	C60H79N11O9S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-DQUNFF	WO2018119357A1_85	.	CC[C@H](C)N1N=C(C(=O)NCC2=C(C)C=C(C)NC2=O)C2=CC=C(C3=CC=C(N4CCN(CCOCCOCCOCC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=C(C)N=CS6)C=C5)C(C)(C)C)CC4)N=C3)C=C21	C60H79N11O9S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-2CHPC0	SCHEMBL20294993	6-[2-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]ethoxy]ethoxy]-N-[(4-methoxy-6-methyl-2-oxo-1H-pyridin-3-yl)methyl]-2-methyl-1-[(1S)-1-(oxan-4-yl)ethyl]indole-3-carboxamide; SCHEMBL30098774	COC1=C(CNC(=O)C2=C(C)N([C@@H](C)C3CCOCC3)C3=CC(OCCOCCN4CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)=CC=C32)C(=O)NC(C)=C1	C46H55N7O10	EZH2	Q15910	CRBN	WO-2018119357-A1
TPD-V8UCER	WO2018119357A1_87	.	COC1=C(CNC(=O)C2=C(C)N([C@@H](C)C3CCOCC3)C3=CC(CCOCCOC4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)=CC=C32)C(=O)NC(C)=C1	C42H47N5O10	EZH2	Q15910	CRBN	WO-2018119357-A1
TPD-0676SU	SCHEMBL20294988	(2S,4R)-1-[(2S)-2-[5-[3-[4-[3-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methylcarbamoyl]-5-[ethyl(oxan-4-yl)amino]-4-methylphenyl]phenyl]propoxy]pentanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CCN(C1=CC(C2=CC=C(CCCOCCCCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](C)C3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C60H79N7O8S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-PV3Z7W	SCHEMBL20294932	(2S,4R)-1-[(2S)-2-[[2-[2-[3-[4-[3-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methylcarbamoyl]-5-[ethyl(oxan-4-yl)amino]-4-methylphenyl]phenyl]propoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CCN(C1=CC(C2=CC=C(CCCOCCOCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](C)C3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C59H77N7O9S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-Z27SFH	WO2018119357A1_90	.	CCN(C1=CC(C2=CC=C(OCCCOC3=CC(C4=C(C)N=CS4)=CC=C3CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4C=CC=CC4C3=O)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C61H73N7O9S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-EJ6D6H	SCHEMBL20294924	N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-5-[4-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]ethoxy]phenyl]-3-[ethyl(oxan-4-yl)amino]-2-methylbenzamide; SCHEMBL30098744	CCN(C1=CC(C2=CC=C(OCCN3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C48H55N7O8	EZH2	Q15910	CRBN	WO-2018119357-A1
TPD-YGCVVZ	WO2018119357A1_92	.	CCN(C1=CC(C2=CC=C(OCCCCN3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)C=C2)=CC(C(=O)NCC2C(=O)NC(C)=CC2C)=C1C)C1CCOCC1	C50H61N7O8	EZH2	Q15910	CRBN	WO-2018119357-A1
TPD-47VSV6	SCHEMBL20294904	(2S,4R)-1-[(2S)-2-[[2-[4-[4-[3-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methylcarbamoyl]-5-[ethyl(oxan-4-yl)amino]-4-methylphenyl]phenoxy]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CCN(C1=CC(C2=CC=C(OCCCCOCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](C)C3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C58H75N7O9S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-ZZZVZR	SCHEMBL20294845	(2S,4R)-1-[(2S)-2-[[2-[5-[4-[3-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methylcarbamoyl]-5-[ethyl(oxan-4-yl)amino]-4-methylphenyl]phenoxy]pentoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL30098678	CCN(C1=CC(C2=CC=C(OCCCCCOCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](C)C3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C59H77N7O9S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-8I5CTA	WO2018119357A1_95	.	CCN(C1=CC(C2=CC=C(OCCCOCC(=O)N[C@H](C(=O)N3CC(=O)C[C@H]3C(=O)N[C@@H](C)C3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C57H71N7O9S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-JJXSVI	SCHEMBL20294939	(2R,4S)-1-[(2S)-2-[[2-[2-[2-[4-[3-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methylcarbamoyl]-5-[ethyl(oxan-4-yl)amino]-4-methylphenyl]phenoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL30098670	CCN(C1=CC(C2=CC=C(OCCOCCOCC(=O)N[C@H](C(=O)N3C[C@@H](O)C[C@@H]3C(=O)N[C@@H](C)C3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C58H75N7O10S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-RZM4T4	SCHEMBL20294954	(2S,4R)-1-[(2R)-2-[5-[3-[4-[3-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methylcarbamoyl]-5-[ethyl(oxan-4-yl)amino]-4-methylphenyl]phenoxy]propoxy]-3-oxo-1H-isoindol-2-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL30098666	CCN(C1=C(C)C(C(=O)NCC2=C(C)C=C(C)NC2=O)=CC(C2=CC=C(OCCCOC3=CC=C4CN([C@@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=C(C)N=CS6)C=C5)C(C)C)C(=O)C4=C3)C=C2)=C1)C1CCOCC1	C62H73N7O9S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-67N5XN	SCHEMBL20294926	(2S,4R)-1-[(2S)-2-[5-[3-[4-[3-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methylcarbamoyl]-5-[ethyl(oxan-4-yl)amino]-4-methylphenyl]phenoxy]propoxy]-3-oxo-1H-isoindol-2-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL30098677	CCN(C1=C(C)C(C(=O)NCC2=C(C)C=C(C)NC2=O)=CC(C2=CC=C(OCCCOC3=CC=C4CN([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=C(C)N=CS6)C=C5)C(C)C)C(=O)C4=C3)C=C2)=C1)C1CCOCC1	C62H73N7O9S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-MWZ2L6	SCHEMBL20294894	(2S,4R)-1-[(2S)-2-[5-[2-[[4-[3-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methylcarbamoyl]-5-[ethyl(oxan-4-yl)amino]-4-methylphenyl]phenyl]methoxy]ethoxy]-3-oxo-1H-isoindol-2-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL30098735	CCN(C1=C(C)C(C(=O)NCC2=C(C)C=C(C)NC2=O)=CC(C2=CC=C(COCCOC3=CC=C4CN([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=C(C)N=CS6)C=C5)C(C)C)C(=O)C4=C3)C=C2)=C1)C1CCOCC1	C62H73N7O9S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-7FU38Z	SCHEMBL20294858	(2S,4R)-1-[(2S)-2-[5-[2-[4-[3-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methylcarbamoyl]-5-[ethyl(oxan-4-yl)amino]-4-methylphenyl]phenoxy]ethoxy]-3-oxo-1H-isoindol-2-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CCN(C1=C(C)C(C(=O)NCC2=C(C)C=C(C)NC2=O)=CC(C2=CC=C(OCCOC3=CC=C4CN([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=C(C)N=CS6)C=C5)C(C)C)C(=O)C4=C3)C=C2)=C1)C1CCOCC1	C61H71N7O9S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-IE89BZ	WO2018119357A1_101	.	CCN(C1=C(C)C(C(=O)NCC2=C(C)C=C(C)NC2=O)=CC(C2=CC=C(OCCCCOC3C=C4C(=O)N([C@@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=C(C)N=CS6)C=C5)C(C)C)CC4=CC3)C=C2)=C1)C1CCOCC1	C63H77N7O9S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-6L3YR9	WO2018119357A1_102	.	CCN(C1=C(C)C(C(=O)NCC2=C(C)C=C(C)NC2=O)=CC(C2=CC=C(OCCCCOC3C=C4C(=O)N([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=C(C)N=CS6)C=C5)C(C)C)CC4=CC3)C=C2)=C1)C1CCOCC1	C63H77N7O9S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-85BEQ2	WO2018119357A1_103	.	CCN(C1=C(C)C(C(=O)NCC2=C(C)C=C(C)NC2=O)=CC(C2=CC=C(OCCCCOC3C=C4C(=O)N(C(C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=C(C)N=CS6)C=C5)C(C)C)CC4=CC3)C=C2)=C1)C1CCOCC1	C63H77N7O9S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-T260NU	SCHEMBL20294854	(2S,4R)-1-[2-[3-[5-[4-[3-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methylcarbamoyl]-5-[ethyl(oxan-4-yl)amino]-4-methylphenyl]phenoxy]pentoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL30098763	CCN(C1=C(C)C(C(=O)NCC2=C(C)C=C(C)NC2=O)=CC(C2=CC=C(OCCCCCOC3=NOC(C(C(=O)N4C[C@H](O)C[C@H]4C(=O)N[C@@H](C)C4=CC=C(C5=C(C)N=CS5)C=C4)C(C)C)=C3)C=C2)=C1)C1CCOCC1	C59H73N7O9S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-INBR8D	SCHEMBL20295004	(2S,4R)-1-[2-[3-[2-[2-[4-[3-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methylcarbamoyl]-5-[ethyl(oxan-4-yl)amino]-4-methylphenyl]phenoxy]ethoxy]ethoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CCN(C1=C(C)C(C(=O)NCC2=C(C)C=C(C)NC2=O)=CC(C2=CC=C(OCCOCCOC3=NOC(C(C(=O)N4C[C@H](O)C[C@H]4C(=O)N[C@@H](C)C4=CC=C(C5=C(C)N=CS5)C=C4)C(C)C)=C3)C=C2)=C1)C1CCOCC1	C58H71N7O10S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-WC2T7H	SCHEMBL20294887	(2S,4R)-1-[2-[3-[6-[4-[3-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methylcarbamoyl]-5-[ethyl(oxan-4-yl)amino]-4-methylphenyl]phenoxy]hexoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL30098648	CCN(C1=C(C)C(C(=O)NCC2=C(C)C=C(C)NC2=O)=CC(C2=CC=C(OCCCCCCOC3=NOC(C(C(=O)N4C[C@H](O)C[C@H]4C(=O)N[C@@H](C)C4=CC=C(C5=C(C)N=CS5)C=C4)C(C)C)=C3)C=C2)=C1)C1CCOCC1	C60H75N7O9S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-GVG58P	SCHEMBL20295050	(2S,4R)-1-[2-[3-[4-[4-[3-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methylcarbamoyl]-5-[ethyl(oxan-4-yl)amino]-4-methylphenyl]phenoxy]butoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL30098709	CCN(C1=C(C)C(C(=O)NCC2=C(C)C=C(C)NC2=O)=CC(C2=CC=C(OCCCCOC3=NOC(C(C(=O)N4C[C@H](O)C[C@H]4C(=O)N[C@@H](C)C4=CC=C(C5=C(C)N=CS5)C=C4)C(C)C)=C3)C=C2)=C1)C1CCOCC1	C58H71N7O9S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-1BSXY0	SCHEMBL20317518	(2S,4R)-1-[(2S)-2-[5-[2-[4-[3-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methylcarbamoyl]-5-[ethyl(oxan-4-yl)amino]-4-methylphenyl]phenoxy]ethoxymethyl]-3-oxo-1H-isoindol-2-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CCN(C1=C(C)C(C(=O)NCC2=C(C)C=C(C)NC2=O)=CC(C2=CC=C(OCCOCC3=CC=C4CN([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=C(C)N=CS6)C=C5)C(C)C)C(=O)C4=C3)C=C2)=C1)C1CCOCC1	C62H73N7O9S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-7425QN	SCHEMBL20295037	(2S,4R)-1-[2-[3-[3-[2-[4-[3-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methylcarbamoyl]-5-[ethyl(oxan-4-yl)amino]-4-methylphenyl]phenoxy]ethoxy]propoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CCN(C1=C(C)C(C(=O)NCC2=C(C)C=C(C)NC2=O)=CC(C2=CC=C(OCCOCCCOC3=NOC(C(C(=O)N4C[C@H](O)C[C@H]4C(=O)N[C@@H](C)C4=CC=C(C5=C(C)N=CS5)C=C4)C(C)C)=C3)C=C2)=C1)C1CCOCC1	C59H73N7O10S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-2U0GZD	SCHEMBL20294893	(2S,4R)-1-[2-[3-[2-[2-[4-[3-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methylcarbamoyl]-5-[ethyl(oxan-4-yl)amino]-4-methylphenyl]phenyl]ethoxy]ethoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CCN(C1=C(C)C(C(=O)NCC2=C(C)C=C(C)NC2=O)=CC(C2=CC=C(CCOCCOC3=NOC(C(C(=O)N4C[C@H](O)C[C@H]4C(=O)N[C@@H](C)C4=CC=C(C5=C(C)N=CS5)C=C4)C(C)C)=C3)C=C2)=C1)C1CCOCC1	C58H71N7O9S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-BZHXQ1	SCHEMBL20295008	(2S,4R)-1-[2-[3-[2-[3-[4-[3-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methylcarbamoyl]-5-[ethyl(oxan-4-yl)amino]-4-methylphenyl]phenyl]propoxy]ethoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL30098770	CCN(C1=C(C)C(C(=O)NCC2=C(C)C=C(C)NC2=O)=CC(C2=CC=C(CCCOCCOC3=NOC(C(C(=O)N4C[C@H](O)C[C@H]4C(=O)N[C@@H](C)C4=CC=C(C5=C(C)N=CS5)C=C4)C(C)C)=C3)C=C2)=C1)C1CCOCC1	C59H73N7O9S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-2UV6UF	WO2018119357A1_112	.	CCN(C1=C(C)C(C(=O)NCC2=C(C)C=C(C)NC2=O)=CC(C2=CC=C(OCCCOCCOC3=NOC(C(C(=O)N4C[C@H](O)C[C@H]4C(O)N[C@@H](C)C4=CC=C(C5=C(C)N=CS5)C=C4)C(C)C)=C3)C=C2)=C1)C1CCOCC1	C59H75N7O10S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-WHCCDI	SCHEMBL20317463	N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-5-[4-[[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]methyl]phenyl]-3-[ethyl(oxan-4-yl)amino]-2-methylbenzamide; SCHEMBL30098676	CCN(C1=C(C)C(C(=O)NCC2=C(C)C=C(C)NC2=O)=CC(C2=CC=C(CN3CCN(CC4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)C=C2)=C1)C1CCOCC1	C53H64N8O7	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-0T44J4	SCHEMBL20294940	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[4-[[4-[3-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methylcarbamoyl]-5-[ethyl(oxan-4-yl)amino]-4-methylphenyl]phenyl]methyl]piperazin-1-yl]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL30098702	CCN(C1=C(C)C(C(=O)NCC2=C(C)C=C(C)NC2=O)=CC(C2=CC=C(CN3CCN(CCOCCOCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)N[C@@H](C)C4=CC=C(C5=C(C)N=CS5)C=C4)C(C)(C)C)CC3)C=C2)=C1)C1CCOCC1	C63H85N9O9S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-7PL83Y	SCHEMBL20295003	N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-5-[4-[[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]methyl]phenyl]-3-[ethyl(oxan-4-yl)amino]-2-methylbenzamide; SCHEMBL30098673	CCN(C1=C(C)C(C(=O)NCC2=C(C)C=C(C)NC2=O)=CC(C2=CC=C(CN3CCC(CN4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)C=C2)=C1)C1CCOCC1	C53H64N8O7	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-TLKSZW	SCHEMBL20294912	(2S,4R)-1-[(2S)-2-[[2-[2-[4-[[4-[3-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methylcarbamoyl]-5-[ethyl(oxan-4-yl)amino]-4-methylphenyl]phenyl]methyl]piperazin-1-yl]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL30098691	CCN(C1=C(C)C(C(=O)NCC2=C(C)C=C(C)NC2=O)=CC(C2=CC=C(CN3CCN(CCOCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)N[C@@H](C)C4=CC=C(C5=C(C)N=CS5)C=C4)C(C)(C)C)CC3)C=C2)=C1)C1CCOCC1	C61H81N9O8S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-2FCBYI	SCHEMBL20295026	(2S,4R)-1-[(2S)-2-[[2-[4-[4-[[4-[3-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methylcarbamoyl]-5-[ethyl(oxan-4-yl)amino]-4-methylphenyl]phenyl]methyl]piperazin-1-yl]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL30098724	CCN(C1=C(C)C(C(=O)NCC2=C(C)C=C(C)NC2=O)=CC(C2=CC=C(CN3CCN(CCCCOCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)N[C@@H](C)C4=CC=C(C5=C(C)N=CS5)C=C4)C(C)(C)C)CC3)C=C2)=C1)C1CCOCC1	C63H85N9O8S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-DFP7LI	SCHEMBL20295058	(2S,4R)-1-[(2S)-2-[[2-[3-[4-[[4-[3-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methylcarbamoyl]-5-[ethyl(oxan-4-yl)amino]-4-methylphenyl]phenyl]methyl]piperazin-1-yl]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL30098720	CCN(C1=C(C)C(C(=O)NCC2=C(C)C=C(C)NC2=O)=CC(C2=CC=C(CN3CCN(CCCOCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)N[C@@H](C)C4=CC=C(C5=C(C)N=CS5)C=C4)C(C)(C)C)CC3)C=C2)=C1)C1CCOCC1	C62H83N9O8S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-HXZ0L5	SCHEMBL20294936	(2S,4R)-1-[(2S)-2-[[2-[2-[3-[4-[4-[3-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methylcarbamoyl]-5-[ethyl(oxan-4-yl)amino]-4-methylphenyl]phenyl]piperazin-1-yl]propoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL30098675	CCN(C1=C(C)C(C(=O)NCC2=C(C)C=C(C)NC2=O)=CC(C2=CC=C(N3CCN(CCCOCCOCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)N[C@@H](C)C4=CC=C(C5=C(C)N=CS5)C=C4)C(C)(C)C)CC3)C=C2)=C1)C1CCOCC1	C63H85N9O9S	EZH2	Q15910	VHL	WO-2018119357-A1
TPD-60EULJ	WO2018119441A1_1	.	CC1=C(c2ccc(CNC(=O)C3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCN3CCN(Cc4ccc(-c5cc6c(NCc7ccccc7C)ncnc6[nH]5)cc4)CC3)C(C)(C)C)cc2)CC=N1	C56H72N10O7	EGFR	P00533	VHL	WO-2018119441-A1
TPD-LC3RYT	US10994015, Example 2	US10994015, Example 2; BDBM494868	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCOCCN2CCN(Cc3ccc(-c4cc5c(NCc6ccccc6Cl)ncnc5[nH]4)cc3)CC2)C(C)(C)C)cc1	C56H71ClN10O8S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-LSQM1D	WO2018119441A1_3	.	Cc1ccccc1CNc1ncnc2[nH]c(-c3ccc(CN4CCN(CCOCCOCCOCCOCCOCC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)NCc5ccc(-c6scnc6C)cc5)C(C)(C)C)CC4)cc3)cc12	C59H78N10O9S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-SJYHQU	US10994015, Example 4	US10994015, Example 4; BDBM494870	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCN2CCN(Cc3ccc(-c4cc5c(NCc6ccccc6Cl)ncnc5[nH]4)cc3)CC2)C(C)(C)C)cc1	C52H63ClN10O6S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-EY2KKO	US10994015, Example 5	US10994015, Example 5; BDBM494871	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCN2CCN(Cc3ccc(-c4cc5c(NCc6ccccc6Cl)ncnc5[nH]4)cc3)CC2)C(C)(C)C)cc1	C50H59ClN10O5S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-5IZT0I	US10994015, Example 6	US10994015, Example 6; BDBM494872	O=C1CCC(N2C(=O)c3cccc(NCCOCCOCCOCCN4CCN(Cc5ccc(-c6cc7c(NCc8ccccc8Cl)ncnc7[nH]6)cc5)CC4)c3C2=O)C(=O)N1	C45H50ClN9O7	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-TPQPY9	US10994015, Example 7	US10994015, Example 7; BDBM494873	O=C1CCC(N2C(=O)c3cccc(NCCOCCOCCOCCOCCN4CCN(Cc5ccc(-c6cc7c(NCc8ccccc8Cl)ncnc7[nH]6)cc5)CC4)c3C2=O)C(=O)N1	C47H54ClN9O8	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-9BUNRP	SCHEMBL20305649	US10994015, Example 8; US10994015, Example 8; BDBM494874; 4-((17-(4-(4-(4-((2-chlorobenzyl)amino)-7H-pyrrolo[2,3-d]pyrimidin-6-yl)benzyl)piperazin-1-yl)-3,6,9,12,15-pentaoxaheptadecyl)amino)-2-(2,6-dioxopiperidin-3-yl)isoindoline-1,3-dione	O=C1CCC(N2C(=O)c3cccc(NCCOCCOCCOCCOCCOCCN4CCN(Cc5ccc(-c6cc7c(NCc8ccccc8Cl)ncnc7[nH]6)cc5)CC4)c3C2=O)C(=O)N1	C49H58ClN9O9	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-HOUJS5	US10994015, Example 9	US10994015, Example 9; BDBM494875	O=C1CCC(N2C(=O)c3cccc(NCCOCCOCCN4CCN(Cc5ccc(-c6cc7c(NCc8ccccc8Cl)ncnc7[nH]6)cc5)CC4)c3C2=O)C(=O)N1	C43H46ClN9O6	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-9ZV7W6	WO2018119441A1_10	.	Cc1ccccc1CNc1ncnc2[nH]c(-c3ccc(OCCOCCOCCOCCNc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)cc3)cc12	C41H43N7O8	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-5U1K05	WO2018119441A1_11	.	O=C1CCC(N2C(=O)c3cccc(NCCOCCN4CCN(Cc5ccc(-c6cc7c(NCc8ccccc8Cl)ncnc7[nH]6)cc5)CC4)c3C2=O)C(=O)N1	C41H42ClN9O5	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-DTNEP2	BDBM494879	US10994015, Example 12; US10994015, Example 12	O=C1CCC(N2C(=O)c3cccc(NCCOCCOCCOc4ccc(-c5cc6c(NCc7ccccc7Cl)ncnc6[nH]5)cc4)c3C2=O)C(=O)N1	C38H36ClN7O7	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-HK1YIS	BDBM494922	US10994015, Example 13; US10994015, Example 13	O=C1CCC(N2C(=O)c3cccc(NCCOCCOc4ccc(-c5cc6c(NCc7ccccc7Cl)ncnc6[nH]5)cc4)c3C2=O)C(=O)N1	C36H32ClN7O6	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-WYZHP9	SCHEMBL20305784	US10994015, Example 14; BDBM494923; US10994015, Example 14; (2S,4R)-1-((S)-2-(tert-butyl)-14-(4-(4-((2-chlorobenzyl)amino)-7H-pyrrolo[2,3-d]pyrimidin-6-yl)phenoxy)-4-oxo-6,9,12-trioxa-3-azatetradecanoyl)-4-hydroxy-N-(4-(4-methylthiazol-5-yl)benzyl)pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCOc2ccc(-c3cc4c(NCc5ccccc5Cl)ncnc4[nH]3)cc2)C(C)(C)C)cc1	C49H57ClN8O8S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-TWCTX0	BDBM494924	US10994015, Example 15; US10994015, Example 15	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOc2ccc(-c3cc4c(NCc5ccccc5Cl)ncnc4[nH]3)cc2)C(C)(C)C)cc1	C47H53ClN8O7S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-Z0B2TM	WO2018119441A1_16	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)C(NC(=O)COCCOc2ccc(-c3cc4c(NCc5ccccc5O)ncnc4[nH]3)cc2)C(C)(C)C)cc1	C45H50N8O7S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-HW3HP4	SCHEMBL20305646	US10994015, Example 17; BDBM494925; US10994015, Example 17; 5-(2-(2-(2-(4-(4-(4-((2-chlorobenzyl)amino)-7H-pyrrolo[2,3-d]pyrimidin-6-yl)benzyl)piperazin-1-yl)ethoxy)ethoxy)ethoxy)-2-(2,6-dioxopiperidin-3-yl)isoindoline-1,3-dione	O=C1CCC(N2C(=O)c3ccc(OCCOCCOCCN4CCN(Cc5ccc(-c6cc7c(NCc8ccccc8Cl)ncnc7[nH]6)cc5)CC4)cc3C2=O)C(=O)N1	C43H45ClN8O7	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-YR9V06	SCHEMBL20305500	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[2-[2-[2-[4-(3-chloro-4-fluoroanilino)-7-methoxyquinazolin-6-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1OCCOCCOCCOCCOCCOCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(-c2scnc2C)cc1)C(C)(C)C	C49H61ClFN7O11S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-TWBTJ6	WO2018119441A1_19	.	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1OCCOCCOCCOCCOCCOCCOCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(-c2scnc2C)cc1)C(C)(C)C	C51H65ClFN7O12S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-A7Q4IB	WO2018119441A1_20	.	COc1cc2ncnc(Nc3ccc(F)c(CI)c3)c2cc1OCCOCCOCCOCCOc1cc(-c2scnc2C)ccc1CNC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@H](C(C)C)N1Cc2ccccc2C1=O	C53H59FIN7O10S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-ZEVZQ0	WO2018119441A1_21	(2S,4R)-N-[[2-[2-[2-[2-[2-[2-[4-(3-chloro-4-fluoroanilino)-7-methoxyquinazolin-6-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]ethoxy]-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-4-hydroxy-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]pyrrolidine-2-carboxamide	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1OCCOCCOCCOCCOCCOc1cc(-c2scnc2C)ccc1CNC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@H](C(C)C)N1Cc2ccccc2C1=O	C54H61ClFN7O11S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-8LFSJE	WO2018119441A1_22	(2S,4R)-N-[[2-[2-[2-[2-[2-[2-[2-[4-(3-chloro-4-fluoroanilino)-7-methoxyquinazolin-6-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-4-hydroxy-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]pyrrolidine-2-carboxamide	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1OCCOCCOCCOCCOCCOCCOc1cc(-c2scnc2C)ccc1CNC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@H](C(C)C)N1Cc2ccccc2C1=O	C56H65ClFN7O12S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-NLFD5C	WO2018119441A1_23	(2S,4R)-N-[[2-[2-[2-[3-[2-[2-[4-(3-chloro-4-fluoroanilino)-7-methoxyquinazolin-6-yl]oxyethoxy]ethoxy]propoxy]ethoxy]ethoxy]-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-4-hydroxy-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]pyrrolidine-2-carboxamide	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1OCCOCCOCCCOCCOCCOc1cc(-c2scnc2C)ccc1CNC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@H](C(C)C)N1Cc2ccccc2C1=O	C55H63ClFN7O11S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-XAQVD5	WO2018119441A1_24	(2S,4R)-N-[[2-[2-[2-[4-[2-[2-[4-(3-chloro-4-fluoroanilino)-7-methoxyquinazolin-6-yl]oxyethoxy]ethoxy]butoxy]ethoxy]ethoxy]-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-4-hydroxy-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]pyrrolidine-2-carboxamide	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1OCCOCCOCCCCOCCOCCOc1cc(-c2scnc2C)ccc1CNC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@H](C(C)C)N1Cc2ccccc2C1=O	C56H65ClFN7O11S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-4AWSM7	WO2018119441A1_25	(2S,4R)-N-[[2-[2-[2-[4-[4-[2-[2-[4-(3-chloro-4-fluoroanilino)-7-methoxyquinazolin-6-yl]oxyethoxy]ethoxy]butoxy]butoxy]ethoxy]ethoxy]-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-4-hydroxy-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]pyrrolidine-2-carboxamide	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1OCCOCCOCCCCOCCCCOCCOCCOc1cc(-c2scnc2C)ccc1CNC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@H](C(C)C)N1Cc2ccccc2C1=O	C60H73ClFN7O12S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-LY903Z	WO2018119441A1_26	.	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1OCCOCCOCCCCCOCCCCCOCCOCCOc1cc(-c2scnc2C)ccc1CNC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@H](C(C)C)N1Cc2ccccc2C1O	C62H79ClFN7O12S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-RGLAGR	WO2018119441A1_27	.	COc1cc2ncnc(Nc3ccc(F)c(C)c3)c2cc1OCCOCCOCCCOCCOCCOCC(=O)N[C@H](C(=O)N1C[C@@H](O)C[C@H]1C(=O)NCc1ccc(-c2scnc2C)cc1)C(C)(C)C	C51H66FN7O11S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-DQRME7	WO2018119441A1_28	.	C=C(COCCOCCOCCCCOCCOCCOc1cc2c(Nc3ccc(F)c(Cl)c3)ncnc2cc1OC)N[C@H](C(=O)N1C[C@@H](O)C[C@H]1C(=O)NCc1ccc(-c2scnc2C)cc1)C(C)(C)C	C52H67ClFN7O10S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-OXOAVO	WO2018119441A1_29	.	COc1cc2ncnc(Nc3ccc(F)c(C)c3)c2cc1OCCOCCOCCCOc1cc(-c2scnc2C)ccc1CNC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@H](C(C)C)N1Cc2ccccc2[C@@H]1O	C52H60FN7O9S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-X9SGD1	WO2018119441A1_30	.	COc1cc2nccc(Nc3ccc(F)c(Cl)c3)c2cc1OCCOCCOCCCOCCCCOCCOCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(C2=C(C)NCS2)cc1)C(C)(C)C	C53H70ClFN6O11S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-5WIHMN	WO2018119441A1_31	.	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1OCCOCCOCCCCCOCCOCCOc1cc(-c2scnc2C)ccc1CNC(=O)C1C[C@@H](O)CN1C(=O)[C@H](C(C)C)N1Cc2ccccc2C1=O	C57H67ClFN7O11S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-AR9QTW	WO2018119441A1_32	(2S,4R)-N-[[2-[4-[4-[4-[4-(3-chloro-4-fluoroanilino)-7-methoxyquinazolin-6-yl]oxybutoxy]butoxy]butoxy]-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-4-hydroxy-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]pyrrolidine-2-carboxamide	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1OCCCCOCCCCOCCCCOc1cc(-c2scnc2C)ccc1CNC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@H](C(C)C)N1Cc2ccccc2C1=O	C56H65ClFN7O9S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-M8T7KA	WO2018119441A1_33	.	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1OCCOCCOCCCCCCCCCOCCOCC(O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(-c2scnc2C)cc1)C(C)(C)C	C54H73ClFN7O10S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-RGXUKW	WO2018119441A1_34	.	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1OCCOCCNCCCCCOCCCCCOCCOCC(=O)N[C@H](C(O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(C2=C(C)NCS2)cc1)C(C)(C)C	C55H78ClFN8O10S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-HCWOST	WO2018119441A1_35	.	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1OCCOCCCOCCCOc1cc(-c2scnc2C)ccc1CNC(=O)[C@@H]1C[C@H](O)CN1C(=O)[C@H](C(C)C)N1Cc2ccccc2C1=O	C52H57ClFN7O9S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-H87ABN	WO2018119441A1_36	.	COc1cc2c(cc1OCCCCOCCCCOCCCCCCC(=O)N[C@H](C(=O)N1C[C@@H](O)CC1[C@H](O)NCc1ccc(-c3scnc3C)cc1)C(C)(C)C)=C(Nc1ccc(F)c(Cl)c1)N=C[Ni]=2	C52H69ClFN6NiO8S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-RAE7TB	WO2018119441A1_37	.	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1OCCCCOCCCCOCCCCCC(=O)N[C@H](C(=O)N1C[C@@H](O)C[C@H]1C(=O)NCc1ccc(-c2scnc2C)cc1)C(C)(C)C	C51H65ClFN7O8S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-WTXIJP	WO2018119441A1_38	.	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1OCCCCCOCCCOCC(=O)N[C@H](C(=O)N1C[C@@H](O)C[C@H]1C(=O)NCC1=CC=C(c2scnc2C)CC1)C(C)(C)C	C47H59ClFN7O8S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-N5NJP1	WO2018119441A1_39	.	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1OCCCCCOCCOCCC(=O)N[C@H](C(=O)N1C[C@@H](O)C[C@H]1C(=O)NCc1ccc(-c2scnc2C)cc1)C(C)(C)C	C47H57ClFN7O8S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-GDUHUT	WO2018119441A1_40	.	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1OCCCCCOCCOCCOCC(=O)N[C@H](C(O)N1C[C@@H](O)C[C@H]1C(=O)NCc1ccc(-c2scnc2C)cc1)C(C)(C)C	C48H61ClFN7O9S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-OFVV6M	WO2018119441A1_41	.	COc1cc2ncnc(NC3=CC=C(F)C(C)C3)c2cc1NC(=O)/C=C/CN(C)CCOCCOCC(=O)N[C@H](C(=O)N1C[C@@H](O)C[C@H]1CNCc1ccc(-c2scnc2C)cc1)C(C)(C)C	C49H64FN9O7S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-F7ZZC4	WO2018119441A1_42	.	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1NC(=O)/C=C/CN(C)CCOCCOCCOCCOCC(=O)N[C@H](C(=O)N1C[C@@H](O)C[C@H]1C(=O)NCc1ccc(-c2scnc2C)cc1)C(C)(C)C	C52H65ClFN9O10S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-JLK30Y	WO2018119441A1_43	.	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1NC(=O)/C=C/CN(C)CCOCCOCCOCCOCCOCC(=O)N[C@H](C(=O)N1C[C@@H](O)C[C@H]1C(=O)NCc1ccc(-c2scnc2C)cc1)C(C)(C)C	C54H69ClFN9O11S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-UHFMX3	WO2018119441A1_44	.	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1NC(=O)/C=C/CN(C)CCOCCOCCOCC(=O)N[C@H](C(=O)N1C[C@@H](O)C[C@H]1C(=O)NCc1ccc(-c2scnc2C)cc1)C(C)(C)C	C50H61ClFN9O9S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-3JFF84	WO2018119441A1_45	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOc2cc3ncnc(Nc4ccc(F)c(Cl)c4)c3cc2NC(=O)/C=C/CN(C)C)C(C)(C)C)cc1	C48H57ClFN9O8S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-L3LLMB	WO2018119441A1_46	.	COc1cc2ncnc(NC3C=C(Cl)C(F)=CC3)c2cc1NC(=O)/C=C/CN(C)CCOCCOCCOCCOCCOCCOCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(-c2scnc2C)cc1)C(C)(C)C	C56H75ClFN9O12S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-ARM34A	WO2018119441A1_47	.	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1NC(=O)/C=C/CN(C)CCCOCCCCOCCCOCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N=NCc1ccc(-c2scnc2C)cc1)C(C)(C)C	C54H68ClFN10O9S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-W3P3PO	WO2018119441A1_48	.	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1NC(=O)/C=C/CNCCCOCCCOCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(-c2scnc2C)cc1)C(C)(C)C	C49H59ClFN9O8S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-A0VB0C	WO2018119441A1_49	.	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1NC(=O)/C=C/CN(C)CCCCOCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(-c2scnc2C)cc1)C(C)(C)C	C48H57ClFN9O7S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-8GXBKK	WO2018119441A1_50	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCOCCOc2cc3ncnc(Nc4ccc(F)c(Cl)c4)c3cc2NC(=O)/C=C/CN(C)C)C(C)(C)C)cc1	C52H65ClFN9O10S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-X7ZMTU	WO2018119441A1_51	.	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1NC(=O)/C=C/CN(C)CCOCCCCCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(-c2scnc2C)cc1)C(C)(C)C	C50H61ClFN9O7S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-23O6A3	WO2018119441A1_52	.	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1NC(=O)CCCN(C)CCCCOCCOCCOCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(-c2scnc2C)cc1)C(C)(C)C	C52H67ClFN9O9S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-NGH715	WO2018119441A1_53	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCOCCOCCOc2cc3ncnc(Nc4ccc(F)c(Cl)c4)c3cc2NC(=O)/C=C/CN(C)C)C(C)(C)C)cc1	C54H69ClFN9O11S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-29LMYS	WO2018119441A1_54	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCCCOc2cc3ncnc(Nc4ccc(F)c(Cl)c4)c3cc2NC(=O)/C=C/CN(C)C)C(C)(C)C)cc1	C52H65ClFN9O9S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-QNL7VK	WO2018119441A1_55	.	Cc1ncsc1-c1ccc(CNC(=O)C2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCOc2cc3ncnc(Nc4ccc(F)c(Cl)c4)c3cc2NC(=O)/C=C/CN(C)C)C(C)(C)C)cc1	C50H61ClFN9O9S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-F0TXED	WO2018119441A1_56	.	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1NC(=O)/C=C/CN(C)CCCCCOCCCOCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(-c2scnc2C)cc1)C(C)(C)C	C52H65ClFN9O8S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-7YJQT6	WO2018119441A1_57	.	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1NC(=O)/C=C/CN(C)CCCCOCCCCOCCCCCC(=O)N[C@H](C(=O)N1C[C@@H](O)CC1C(=O)NCc1ccc(-c2scnc2C)cc1)C(C)(C)C	C56H73ClFN9O8S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-XDIMEP	WO2018119441A1_58	.	COc1cc2ncnc(Nc3ccc(F)c(C)c3)c2cc1NC(=O)/C=C/CNCCOCCCCOCCCCOCCOCC(=O)N[C@H](C(=O)N1C[C@@H](O)CC1C(=O)NCc1ccc(-c2scnc2C)cc1)C(C)(C)C	C56H74FN9O10S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-Y9HLXN	WO2018119441A1_59	.	Cc1ncsc1-c1ccc(CNC(=O)C2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCOCCOc2cc3ncnc(Nc4ccc(F)c(Cl)c4)c3cc2NC(=O)/C=C/CN(C)C)C(C)(C)C)cc1	C50H61ClFN9O7S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-OEFZN6	WO2018119441A1_60	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCOCCOCCOCCOc2cc3ncnc(Nc4ccc(F)c(Cl)c4)c3cc2NC(=O)/C=C/CN(C)C)C(C)(C)C)cc1	C56H73ClFN9O12S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-U12O8K	WO2018119441A1_61	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCCOCCCCOCCCOc2cc3ncnc(Nc4ccc(F)c(Cl)c4)c3cc2NC(=O)/C=C/CN(C)C)C(C)(C)C)cc1	C54H69ClFN9O9S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-4FWQX9	WO2018119441A1_62	.	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1NC(=O)/C=C/CN(C)CCCOCCCOCCCOCCCOCCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(-c2scnc2C)cc1)C(C)(C)C	C57H75ClFN9O10S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-2YK4E3	WO2018119441A1_63	.	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1NC(=O)/C=C/CN(C)CCOCCOCCCCOCCCCOCCOCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(-c2scnc2C)cc1)C(C)(C)C	C58H77ClFN9O11S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-481WMS	WO2018119441A1_64	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCCOCCCCCOc2cc3ncnc(Nc4ccc(F)c(Cl)c4)c3cc2NC(=O)/C=C/CN(C)C)C(C)(C)C)cc1	C52H65ClFN9O8S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-UJSX9W	WO2018119441A1_65	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCCOCCCOc2cc3ncnc(Nc4ccc(F)c(Cl)c4)c3cc2NC(=O)/C=C/CN(C)C)C(C)(C)C)cc1	C50H61ClFN9O8S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-66WCDG	CHEMBL5199166	US10994015, Example 66; SCHEMBL20305804; BDBM494927; US10994015, Example 66; PD142723; (2S,4R)-1-((S)-2-(6-(4-(4-((4-((3-chloro-4-fluorophenyl)amino)-6-((E)-4-(dimethylamino)but-2-enamido)quinazolin-7-yl)oxy)butoxy)butoxy)hexanamido)-3,3-dimethylbutanoyl)-4-hydroxy-N-(4-(4-methylthiazol-5-yl)benzyl)pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCOCCCCOCCCCOc2cc3ncnc(Nc4ccc(F)c(Cl)c4)c3cc2NC(=O)/C=C/CN(C)C)C(C)(C)C)cc1	C56H73ClFN9O8S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-6IQZTK	WO2018119441A1_67	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(O)COCCOCCCCOCCCCOCCOc2cc3ncnc(Nc4ccc(F)c(Cl)c4)c3cc2NC(=O)/C=C/CN(C)C)C(C)(C)C)cc1	C56H75ClFN9O10S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-SEW76J	WO2018119441A1_68	.	Cc1ncsc1-c1ccc(CNC(=O)C2C[C@H](O)CN2C(=O)[C@@H](NC(=O)CCOCCCOCCCOCCCOCCCOc2cc3ncnc(Nc4ccc(F)c(Cl)c4)c3cc2NC(=O)CCCN(C)C)C(C)(C)C)cc1	C57H77ClFN9O10S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-I2NT9K	WO2018119441A1_69	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCCCOCCCCOCCOCCOc2cc3ccnc(Nc4ccc(F)c(Cl)c4)c3cc2NC(=O)/C=C/CN(C)C)C(C)(C)C)cc1	C59H78ClFN8O11S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-L6A4SG	SCHEMBL20305570	US10994015, Example 70; BDBM494928; US10994015, Example 70; 2-(2,6-dioxopiperidin-3-yl)-5-(2-(2-(2-((1-isopropyl-6-((2-(4-methoxypiperidin-1-yl)pyrimidin-4-yl)amino)-1H-imidazo[4,5-c]pyridin-2-yl)methoxy)ethoxy)ethoxy)ethoxy)isoindoline-1,3-dione	COC1CCN(c2nccc(Nc3cc4c(cn3)nc(COCCOCCOCCOc3ccc5c(c3)C(=O)N(C3CCC(=O)NC3=O)C5=O)n4C(C)C)n2)CC1	C39H47N9O9	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-PR9LDV	SCHEMBL20305695	US10994015, Example 71; BDBM494929; US10994015, Example 71; 2-(2,6-dioxopiperidin-3-yl)-5-(4-(2-((1-isopropyl-6-((2-(4-methoxypiperidin-1-yl)pyrimidin-4-yl)amino)-1H-imidazo[4,5-c]pyridin-2-yl)methoxy)ethyl)piperazin-1-yl)isoindoline-1,3-dione	COC1CCN(c2nccc(Nc3cc4c(cn3)nc(COCCN3CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC3)n4C(C)C)n2)CC1	C39H47N11O6	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-MGZI1L	SCHEMBL23314155	2-(2,6-Dioxopiperidin-3-yl)-5-[2-[[6-[[2-(4-methoxypiperidin-1-yl)pyrimidin-4-yl]amino]-1-propan-2-ylimidazo[4,5-c]pyridin-2-yl]methoxy]ethoxy]isoindole-1,3-dione	COC1CCN(c2nccc(Nc3cc4c(cn3)nc(COCCOc3ccc5c(c3)C(=O)N(C3CCC(=O)NC3=O)C5=O)n4C(C)C)n2)CC1	C35H39N9O7	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-XGRNM9	WO2018119441A1_73	.	COC1CCN(c2nccc(Nc3cc4c(cn3)nc(COCCOCCOCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](C)c3ccc(-c5scnc5C)cc3)C(C)(C)C)n4C(C)C)n2)CC1	C49H67N11O8S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-84C5DC	WO2018119441A1_74	.	COC1CCN(c2nccc(Nc3cc4c(cn3)nc(COCCOCCOc3ccc5c(c3)C(=O)N(C3CCC(=O)NC3=O)C5=O)n4C(C)C)n2)CC1	C37H43N9O8	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-923A35	SCHEMBL23314156	2-(2,6-Dioxopiperidin-3-yl)-5-[2-[2-[2-[2-[[6-[[2-(4-methoxypiperidin-1-yl)pyrimidin-4-yl]amino]-1-propan-2-ylimidazo[4,5-c]pyridin-2-yl]methoxy]ethoxy]ethoxy]ethoxy]ethoxy]isoindole-1,3-dione	COC1CCN(c2nccc(Nc3cc4c(cn3)nc(COCCOCCOCCOCCOc3ccc5c(c3)C(=O)N(C3CCC(=O)NC3=O)C5=O)n4C(C)C)n2)CC1	C41H51N9O10	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-D4EEH2	SCHEMBL20305768	US10994015, Example 76; BDBM494934; US10994015, Example 76; 2-(2,6-dioxopiperidin-3-yl)-5-(2-(4-(2-((1-isopropyl-6-((2-(4-methoxypiperidin-1-yl)pyrimidin-4-yl)amino)-1H-imidazo[4,5-c]pyridin-2-yl)methoxy)ethyl)piperazin-1-yl)ethoxy)isoindoline-1,3-dione	COC1CCN(c2nccc(Nc3cc4c(cn3)nc(COCCN3CCN(CCOc5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC3)n4C(C)C)n2)CC1	C41H51N11O7	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-T34KUY	WO2018119441A1_77	.	COC1CCN(c2nccc(Nc3cc4c(cn3)nc(COCCOCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](C)c3ccc(-c5scnc5C)cc3)C(C)(C)C)n4C(C)C)n2)CC1	C47H63N11O7S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-ES46S8	SCHEMBL20305763	US10994015, Example 78; BDBM494936; US10994015, Example 78; 2-(2,6-dioxopiperidin-3-yl)-5-(4-(2-(1-(4-((1-isopropyl-2-methyl-1H-imidazo[4,5-c]pyridin-6-yl)amino)pyrimidin-2-yl)-4-methoxypiperidin-4-yl)ethyl)piperazin-1-yl)isoindoline-1,3-dione	COC1(CCN2CCN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)CCN(c2nccc(Nc3cc4c(cn3)nc(C)n4C(C)C)n2)CC1	C39H47N11O5	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-9DZLN0	WO2018119441A1_79	.	COC1CCN(c2nccc(Nc3cc4c(cn3)nc(COCCOCCOCCOCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](C)c3ccc(-c5scnc5C)cc3)C(C)(C)C)n4C(C)C)n2)CC1	C51H71N11O9S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-SH7N7I	SCHEMBL20305785	US10994015, Example 80; BDBM494938; US10994015, Example 80	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CN2CCN(CCCC#Cc3cccc4c3C(=O)N(C(C(=O)Nc3nccs3)c3cc(F)ccc3O)C4)CC2)C(C)(C)C)cc1	C53H60FN9O7S2	EGFR	P00533	VHL	WO-2018119441-A1
TPD-NMWNMT	SCHEMBL20305636	US10994015, Example 81; BDBM494939; US10994015, Example 81; (2S,4R)-1-((S)-18-(tert-butyl)-1-(1-isopropyl-6-((2-(4-methoxypiperidin-1-yl)pyrimidin-4-yl)amino)-1H-imidazo[4,5-c]pyridin-2-yl)-16-oxo-2,5,8,11,14-pentaoxa-17-azanonadecan-19-oyl)-4-hydroxy-N-((S)-1-(4-(4-methylthiazol-5-yl)phenyl)ethyl)pyrrolidine-2-carboxamide	COC1CCN(c2nccc(Nc3cc4c(cn3)nc(COCCOCCOCCOCCOCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](C)c3ccc(-c5scnc5C)cc3)C(C)(C)C)n4C(C)C)n2)CC1	C53H75N11O10S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-MY6WOE	SCHEMBL20305811	US10994015, Example 82; BDBM494940; US10994015, Example 82; 2-(7-(3-(2-(2-(2-((2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindolin-5-yl)amino)ethoxy)ethoxy)ethoxy)prop-1-yn-1-yl)-1-oxoisoindolin-2-yl)-2-(5-fluoro-2-hydroxyphenyl)-N-(thiazol-2-yl)acetamide	O=C1CCC(N2C(=O)c3ccc(NCCOCCOCCOCC#Cc4cccc5c4C(=O)N(C(C(=O)Nc4nccs4)c4cc(F)ccc4O)C5)cc3C2=O)C(=O)N1	C41H37FN6O10S	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-BRIL6M	BDBM494941	US10994015, Example 83; US10994015, Example 83	O=C1CCC(N2C(=O)c3ccc(NCCOCCOCC#Cc4cccc5c4C(=O)N(C(C(=O)Nc4nccs4)c4cc(F)ccc4O)C5)cc3C2=O)C(=O)N1	C39H33FN6O9S	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-2U1FE9	WO2018119441A1_84	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCC#Cc2cccc3c2C(=O)N(C(C(=O)Nc2nccs2)c2cc(F)ccc2O)C3)C(C)(C)C)cc1	C51H56FN7O10S2	EGFR	P00533	VHL	WO-2018119441-A1
TPD-A5QA1O	SCHEMBL20305527	US10994015, Example 85; BDBM494943; US10994015, Example 85; (2S,4R)-4-hydroxy-1-((S)-2-(2-(3-(4-(3-((1-isopropyl-6-((2-(4-methoxypiperidin-1-yl)pyrimidin-4-yl)amino)-1H-imidazo[4,5-c]pyridin-2-yl)methoxy)propyl)piperazin-1-yl)propoxy)acetamido)-3,3-dimethylbutanoyl)-N-((S)-1-(4-(4-methylthiazol-5-yl)phenyl)ethyl)pyrrolidine-2-carboxamide	COC1CCN(c2nccc(Nc3cc4c(cn3)nc(COCCCN3CCN(CCCOCC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)c5ccc(-c6scnc6C)cc5)C(C)(C)C)CC3)n4C(C)C)n2)CC1	C55H79N13O7S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-IL7DHQ	BDBM494944	US10994015, Example 86; US10994015, Example 86	COC1CCN(c2nccc(Nc3cc4c(cn3)nc(COCCN3CCN(CCOCC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)c5ccc(-c6scnc6C)cc5)C(C)(C)C)CC3)n4C(C)C)n2)CC1	C53H75N13O7S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-D26E41	WO2018119441A1_87	.	COC1CCN(c2nccc(Nc3cc4c(cn3)nc(COCCN3CCN(CC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)c5ccc(-c6scnc6C)cc5)C(C)(C)C)CC3)n4C(C)C)n2)CC1	C51H71N13O6S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-DJXHD3	BDBM494946	US10994015, Example 88; US10994015, Example 88	COC1CCN(c2nccc(Nc3cc4c(cn3)nc(COCCOCCN3CCN(CCOc5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC3)n4C(C)C)n2)CC1	C43H55N11O8	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-3KV5FZ	BDBM494947	US10994015, Example 89; US10994015, Example 89	COC1CCN(c2nccc(Nc3cc4c(cn3)nc(COCCCN3CCN(CCCOc5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC3)n4C(C)C)n2)CC1	C43H55N11O7	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-RBAMLZ	WO2018119441A1_90	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CN2CCN(CCCOCC#Cc3cccc4c3C(=O)N(C(C(=O)Nc3nccs3)c3cc(F)ccc3O)C4)CC2)C(C)(C)C)cc1	C54H62FN9O8S2	EGFR	P00533	VHL	WO-2018119441-A1
TPD-5I1LUF	WO2018119441A1_91	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCN2CCN(CCCC#Cc3cccc4c3C(=O)N(C(C(=O)Nc3nccs3)c3cc(F)ccc3O)C4)CC2)C(C)(C)C)cc1	C55H64FN9O8S2	EGFR	P00533	VHL	WO-2018119441-A1
TPD-I49WG1	WO2018119441A1_92	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCCC#Cc2cccc3c2C(=O)N(C(C(=O)Nc2nccs2)c2cc(F)ccc2O)C3)C(C)(C)C)cc1	C49H52FN7O8S2	EGFR	P00533	VHL	WO-2018119441-A1
TPD-4A9401	WO2018119441A1_93	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCCOCCCC#Cc2cccc3c2C(=O)N(C(C(=O)Nc2nccs2)c2cc(F)ccc2O)C3)C(C)(C)C)cc1	C52H58FN7O9S2	EGFR	P00533	VHL	WO-2018119441-A1
TPD-WFUSPW	BDBM494952	US10994015, Example 94; US10994015, Example 94	O=C1CCC(N2C(=O)c3ccc(OCCN4CCN(CCCC#Cc5cccc6c5C(=O)N(C(C(=O)Nc5nccs5)c5cc(F)ccc5O)C6)CC4)cc3C2=O)C(=O)N1	C43H40FN7O8S	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-4CZ1HM	BDBM494953	US10994015, Example 95; US10994015, Example 95	O=C1CCC(N2C(=O)c3ccc(N4CCN(CCCOCCCC#Cc5cccc6c5C(=O)N(C(C(=O)Nc5nccs5)c5cc(F)ccc5O)C6)CC4)cc3C2=O)C(=O)N1	C44H42FN7O8S	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-10S7GO	BDBM494954	US10994015, Example 96; US10994015, Example 96	O=C1CCC(N2C(=O)c3ccc(N4CCN(CCCC#Cc5cccc6c5C(=O)N(C(C(=O)Nc5nccs5)c5cc(F)ccc5O)C6)CC4)cc3C2=O)C(=O)N1	C41H36FN7O7S	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-GMVM72	SCHEMBL20305622	(2R,4S)-1-[(2S)-2-[[2-[2-[2-[4-[4-[3-chloro-4-[(3-fluorophenyl)methoxy]anilino]quinazolin-6-yl]phenoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@H]2C[C@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOc2ccc(-c3ccc4ncnc(Nc5ccc(OCc6cccc(F)c6)c(Cl)c5)c4c3)cc2)C(C)(C)C)cc1	C55H57ClFN7O8S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-EG49CU	SCHEMBL20305697	(2S,4S)-1-[(2S)-2-[[2-[2-[2-[2-[4-[4-[3-chloro-4-[(3-fluorophenyl)methoxy]anilino]quinazolin-6-yl]phenoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCOc2ccc(-c3ccc4ncnc(Nc5ccc(OCc6cccc(F)c6)c(Cl)c5)c4c3)cc2)C(C)(C)C)cc1	C57H61ClFN7O9S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-FTMYD2	WO2018119441A1_101	.	O=C1CCC(N2C(=O)c3ccc(OCCN4CCN(Cc5ccc(-c6cc7c(NCc8ccccc8Cl)ncnc7[nH]6)cc5)CC4)cc3C2=O)C(=O)N1	C39H37ClN8O5	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-D59NAK	SCHEMBL20305680	5-[2-[2-[4-[[4-[4-[(2-chlorophenyl)methylamino]-7H-pyrrolo[2,3-d]pyrimidin-6-yl]phenyl]methyl]piperazin-1-yl]ethoxy]ethoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	O=C1CCC(N2C(=O)c3ccc(OCCOCCN4CCN(Cc5ccc(-c6cc7c(NCc8ccccc8Cl)ncnc7[nH]6)cc5)CC4)cc3C2=O)C(=O)N1	C41H41ClN8O6	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-LHT4VG	WO2018119441A1_103	.	O=C1CCC(N2C(=O)c3ccc(OCCOCCOCCOCCN4CCN(Cc5ccc(-c6cc7c(NCc8ccccc8Cl)ncnc7[nH]6)cc5)CC4)cc3C2=O)C(=O)N1	C45H49ClN8O8	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-BJXWKB	WO2018119441A1_104	.	O=C1CCC(N2C(=O)c3ccc(OCCOCCOCCOCCOCCN4CCN(Cc5ccc(-c6cc7c(NCc8ccccc8Cl)ncnc7[nH]6)cc5)CC4)cc3C2=O)C(=O)N1	C47H53ClN8O9	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-V0DT1U	WO2018119441A1_105	.	Cc1ccccc1CNc1ncnc2[nH]c(-c3ccc(CN4CCN(CCOCCOCCOCCOCCOCCOc5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)cc3)cc12	C50H60N8O10	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-DODFLM	SCHEMBL20305515	US10994015, Example 106; BDBM494960; US10994015, Example 106; (2S,4R)-N-(2-(2-(4-(4-(4-((2-chlorobenzyl)amino)-7H-pyrrolo[2,3-d]pyrimidin-6-yl)benzyl)piperazin-1-yl)ethoxy)-4-(4-methylthiazol-5-yl)benzyl)-4-hydroxy-1-((S)-3-methyl-2-(1-oxoisoindolin-2-yl)butanoyl)pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](C(C)C)N2Cc3ccccc3C2=O)c(OCCN2CCN(Cc3ccc(-c4cc5c(NCc6ccccc6Cl)ncnc5[nH]4)cc3)CC2)c1	C55H59ClN10O5S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-4UVJ31	BDBM494961	US10994015, Example 107; US10994015, Example 107	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](C(C)C)N2Cc3ccccc3C2=O)c(OCCOCCN2CCN(Cc3ccc(-c4cc5c(NCc6ccccc6Cl)ncnc5[nH]4)cc3)CC2)c1	C57H63ClN10O6S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-TLH756	SCHEMBL20305702	US10994015, Example 108; BDBM494962; US10994015, Example 108	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](C(C)C)N2Cc3ccccc3C2=O)c(OCCOCCOCCN2CCN(Cc3ccc(-c4cc5c(NCc6ccccc6Cl)ncnc5[nH]4)cc3)CC2)c1	C59H67ClN10O7S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-RC8AA8	WO2018119441A1_109	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)C(C(C)C)N2Cc3ccccc3C2=O)c(OCCOCCOCCOCCN2CCN(Cc3ccc(-c4cc5c(NCc6ccccc6Cl)ncnc5[nH]4)cc3)CC2)c1	C61H71ClN10O8S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-QZSCTF	WO2018119441A1_110	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](C(C)C)N2Cc3ccccc3C2=O)c(OCCOCCOCCOCCOCCN2CCN(Cc3ccc(-c4cc5c(NCC6=C(Cl)C=CCC6)ncnc5[nH]4)cc3)CC2)c1	C63H77ClN10O9S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-PW0U7U	WO2018119441A1_111	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCN2CCN(Cc3ccc(-c4cc5c(NCc6ccccc6Cl)ncnc5[nH]4)cc3)CC2)C(C)(C)C)cc1	C55H69ClN10O7S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-0IREKU	WO2018119441A1_112	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCN2CCN(Cc3ccc(-c4cc5c(N[C@H](C)c6ccccc6)ncnc5[nH]4)cc3)CC2)C(C)(C)C)cc1	C56H72N10O7S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-QXFZVM	WO2018119441A1_113	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](c2cc(OCCOCCOCCN3CCN(Cc4ccc(-c5cc6c(N[C@H](C)c7ccccc7)ncnc6[nH]5)cc4)CC3)no2)C(C)(C)C)cc1	C57H70N10O7S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-1S61M9	WO2018119441A1_114	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](c2cc(CCCOCCOCCN3CCN(Cc4ccc(-c5cc6c(N[C@H](C)c7ccccc7)ncnc6[nH]5)cc4)CC3)no2)C(C)C)cc1	C57H70N10O6S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-34JM84	WO2018119441A1_115	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCCN2CCN(CCCc3ccc(-c4cc5c(NCc6ccccc6Cl)ncnc5[nH]4)cc3)CC2)C(C)(C)C)cc1	C56H71ClN10O6S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-YXACC3	WO2018119441A1_116	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCN2CCC(Cc3ccc(-c4cc5c(NCc6ccccc6Cl)ncnc5[nH]4)cc3)CC2)C(C)(C)C)cc1	C56H70ClN9O7S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-WF8SJJ	WO2018119441A1_117	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCC2CCN(Cc3ccc(-c4cc5c(NCc6ccccc6Cl)ncnc5[nH]4)cc3)CC2)C(C)(C)C)cc1	C56H70ClN9O7S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-IU1F0O	WO2018119441A1_118	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCCC2CCN(CCCc3ccc(-c4cc5c(NCc6ccccc6Cl)ncnc5[nH]4)cc3)CC2)C(C)(C)C)cc1	C57H72ClN9O6S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-180R4X	WO2018119441A1_119	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCCN2CCC(CCCc3ccc(-c4cc5c(NCc6ccccc6Cl)ncnc5[nH]4)cc3)CC2)C(C)(C)C)cc1	C57H72ClN9O6S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-EG6VIA	WO2018119441A1_120	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CN2CCC(CCOCCN3CCN(Cc4ccc(-c5cc6c(NCc7ccccc7CI)ncnc6[nH]5)cc4)CC3)CC2)C(C)(C)C)cc1	C59H76IN11O5S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-Y03666	WO2018119441A1_122	.	O=C1CCC(N2Cc3cc(OCCOCCOCCOCCN4CCN(Cc5ccc(-c6cc7c(NCc8ccccc8Cl)ncnc7[nH]6)cc5)CC4)ccc3C2=O)C(=O)N1	C45H51ClN8O7	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-7ENRIT	WO2018119441A1_123	.	C[C@@H](Nc1ncnc2[nH]c(-c3ccc(CN4CCN(CCOCCOCCOCCOc5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)cc3)cc12)c1ccccc1	C46H52N8O8	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-OZX0XI	WO2018119441A1_124	.	O=C1CCC(N2C(=O)c3ccc(OCCOCCOCCCC4CCN(CCCc5ccc(-c6cc7c(NCc8ccccc8Cl)ncnc7[nH]6)cc5)CC4)cc3C2=O)C(=O)N1	C47H52ClN7O7	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-NIXJCT	WO2018119441A1_125	.	O=C1CCC(N2C(=O)c3ccc(OCCOCCOCCCN4CCC(CCCc5ccc(-c6cc7c(NCc8ccccc8Cl)ncnc7[nH]6)cc5)CC4)cc3C2=O)C(=O)N1	C47H52ClN7O7	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-SMVQ1L	WO2018119441A1_127	.	O=C1CCC(N2C(=O)c3ccc(N4CCN(CCOCCCN5CCN(CCCc6ccc(-c7cc8c(NCc9ccccc9Cl)ncnc8[nH]7)cc6)CC5)CC4)cc3C2=O)C(=O)N1	C48H55ClN10O5	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-HAW2C4	WO2018119441A1_128	.	O=C1CCC(N2C(=O)c3ccc(N4CCN(CCOCCCN5CCN(CCOc6ccc(-c7cc8c(NCc9ccccc9Cl)ncnc8[nH]7)cc6)CC5)CC4)cc3C2=O)C(=O)N1	C47H53ClN10O6	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-V1LNQW	WO2018119441A1_129	.	O=C1CCC(N2C(=O)c3ccc(OCCOCCOCCCN4CCN(CCOc5ccc(-c6cc7c(NCc8ccccc8Cl)ncnc7[nH]6)cc5)CC4)cc3C2=O)C(=O)N1	C45H49ClN8O8	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-Y7VG5S	WO2018119441A1_130	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCCN2CCN(CCOc3ccc(-c4cc5c(NCc6ccccc6Cl)ncnc5[nH]4)cc3)CC2)C(C)(C)C)cc1	C55H69ClN10O7S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-1OJK9Y	WO2018119441A1_131	.	COc1cc(N(C)CCN(C)C)c(NC(=O)/C=C/CNCCOCCOCCOCCOCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)c2ccc(-c3scnc3C)cc2)C(C)(C)C)cc1Nc1ncc(-c2cnn(C)c2)c(-c2cn3c4c(cccc24)CCC3)n1	C68H90N14O10S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-AGZ7T7	WO2018119441A1_132	.	COc1cc(N(C)CCN(C)C)c(NC(=O)/C=C/CNCCOCCOCCOCCOc2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)cc1Nc1ncc(-c2cnn(C)c2)c(-c2cn3c4c(cccc24)CCC3)n1	C56H66N12O10	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-RA3AXM	WO2018119441A1_133	.	COc1cc(N(C)CCN(C)C)c(NC(=O)/C=C/CNCCOCCOCCOCCNc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)cc1Nc1ncc(-c2cnn(C)c2)c(-c2cn3c4c(cccc24)CCC3)n1	C56H67N13O9	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-NQ4X6A	WO2018119441A1_134	.	COc1cc(N(C)CCN(C)C)c(NC(=O)/C=C/CNCCOCCOCCOCCOc2ccc3c(c2)CN(C2CCC(=O)NC2=O)C3=O)cc1Nc1ncc(-c2cnn(C)c2)c(-c2cn3c4c(cccc24)CCC3)n1	C56H68N12O9	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-0LQEPD	WO2018119441A1_135	.	COc1cc(N(C)CCN(C)C)c(NC(=O)/C=C/CNCCOCCOCCOCCCc2cc([C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](C)c3ccc(-c4scnc4C)cc3)C(C)C)on2)cc1Nc1ncc(-c2cnn(C)c2)c(-c2cn3c4c(cccc24)CCC3)n1	C69H88N14O9S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-AVNNS1	WO2018119441A1_136	.	COc1cc(N(C)CCN(C)C)c(NC(=O)/C=C/CNCCOCCOCCOCCOc2cc([C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](C)c3ccc(-c4scnc4C)cc3)C(C)C)on2)cc1Nc1ncc(-c2cnn(C)c2)c(-c2cn3c4c(cccc24)CCC3)n1	C68H86N14O10S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-NIAG0I	WO2018119441A1_137	.	COc1cc(N(C)CCN(C)C)c(NC(=O)/C=C/COCCOCCOCCOCCOc2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)cc1Nc1ncc(-c2cnn(C)c2)c(-c2cn3c4c(cccc24)CCC3)n1	C56H65N11O11	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-LY1YMZ	WO2018119441A1_138	.	COc1cc(N(C)CCN(C)C)c(NC(=O)/C=C/COCCOCCOCCOCCOCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)c2ccc(-c3scnc3C)cc2)C(C)(C)C)cc1Nc1ncc(-c2cnn(C)c2)c(-c2cn3c4c(cccc24)CCC3)n1	C68H89N13O11S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-0LCSIA	WO2018119441A1_139	.	COc1cc(N(C)CCN(C)C)c(NC(=O)/C=C/COCCOCCOCCOCCOc2cc([C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCc3ccc(-c4scnc4C)cc3)C(C)C)on2)cc1Nc1ncc(-c2cnn(C)c2)c(-c2cn3c4c(cccc24)CCC3)n1	C67H83N13O11S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-F9OBWF	WO2018119441A1_140	.	COc1cc(N2CCN(C)CC2)c(NC(=O)/C=C/CNCCOCCOCCOCCOCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)c2ccc(-c3scnc3C)cc2)C(C)(C)C)cc1Nc1ncc(-c2cnn(C)c2)c(-c2cn3c4c(cccc24)CCC3)n1	C68H88N14O10S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-N6S5WU	WO2018119441A1_141	.	COc1cc(N2CCN(C)CC2)c(NC(=O)/C=C/CNCCOCCOCCOCCOc2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)cc1Nc1ncc(-c2cnn(C)c2)c(-c2cn3c4c(cccc24)CCC3)n1	C56H64N12O10	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-EEH3FT	WO2018119441A1_142	.	COc1cc(N2CCN(C)CC2)c(NC(=O)/C=C/CNCCOCCOCCOCCOc2cc([C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCc3ccc(-c4scnc4C)cc3)C(C)C)on2)cc1Nc1ncc(-c2cnn(C)c2)c(-c2cn3c4c(cccc24)CCC3)n1	C67H82N14O10S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-4S5NH9	WO2018119441A1_143	.	COc1cc(N2CCN(C(C)=O)CC2)c(NC(=O)/C=C/CNCCOCCOCCOCCOCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)c2ccc(-c3scnc3C)cc2)C(C)(C)C)cc1Nc1ncc(-c2cnn(C)c2)c(-c2cn3c4c(cccc24)CCC3)n1	C69H88N14O11S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-7AKWWE	WO2018119441A1_144	.	COc1cc(N2CCN(C(C)=O)CC2)c(NC(=O)/C=C/CNCCOCCOCCOCCOc2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)cc1Nc1ncc(-c2cnn(C)c2)c(-c2cn3c4c(cccc24)CCC3)n1	C57H64N12O11	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-O7S1FO	WO2018119441A1_145	.	COc1cc(N2CCN(C(C)=O)CC2)c(NC(=O)/C=C/CNCCOCCOCCOCCOc2cc([C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCc3ccc(-c4scnc4C)cc3)C(C)C)on2)cc1Nc1ncc(-c2cnn(C)c2)c(-c2cn3c4c(cccc24)CCC3)n1	C68H82N14O11S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-RK77F3	WO2018119441A1_146	.	COc1cc(N2CCN(C(=O)CN(C)C)CC2)c(NC(=O)/C=C/CNCCOCCOCCOCCOCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)c2ccc(-c3scnc3C)cc2)C(C)(C)C)cc1Nc1ncc(-c2cnn(C)c2)c(-c2cn3c4c(cccc24)CCC3)n1	C71H93N15O11S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-T5DG8V	WO2018119441A1_147	.	CN(C)CC(=O)N1CCN(c2cc(O)c(Nc3ncc(-c4cnn(C)c4)c(-c4cn5c6c(cccc46)CCC5)n3)cc2NC(=O)/C=C/CNCCOCCOCCOCCOc2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)CC1	C58H67N13O11	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-X57C4W	WO2018119441A1_148	.	COc1cc(N2CCN(C(=O)CN(C)C)CC2)c(NC(=O)/C=C/CNCCOCCOCCOCCOc2cc([C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCc3ccc(-c4scnc4C)cc3)C(C)C)on2)cc1Nc1ncc(-c2cnn(C)c2)c(-c2cn3c4c(cccc24)CCC3)n1	C70H87N15O11S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-XI2OCA	WO2018119441A1_149	.	COc1cc(N2CCN(C(=O)C3CCCCN3)CC2)c(NC(=O)/C=C/CNCCOCCOCCOCCOCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)c2ccc(-c3scnc3C)cc2)C(C)(C)C)cc1Nc1ncc(-c2cnn(C)c2)c(-c2cn3c4c(cccc24)CCC3)n1	C73H95N15O11S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-XYPB6V	WO2018119441A1_150	.	COc1cc(N2CCN(C(=O)C3CCCCN3)CC2)c(NC(=O)/C=C/CNCCOCCOCCOCCOc2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)cc1Nc1ncc(-c2cnn(C)c2)c(-c2cn3c4c(cccc24)CCC3)n1	C61H71N13O11	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-6O65LT	WO2018119441A1_151	.	COc1cc(N2CCN(C(=O)C3CCCCN3)CC2)c(NC(=O)/C=C/CNCCOCCOCCOCCOc2cc(C(C(=O)N3C[C@H](O)C[C@H]3C(=O)NCc3ccc(-c4scnc4C)cc3)C(C)C)on2)cc1Nc1ncc(-c2cnn(C)c2)c(-c2cn3c4c(cccc24)CCC3)n1	C72H89N15O11S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-YYUZ8P	WO2018119441A1_152	.	COc1cc(N2CC(N(C)C)C2)c(NC(=O)/C=C/CNCCOCCOCCOCCOCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)c2ccc(-c3scnc3C)cc2)C(C)(C)C)cc1Nc1ncc(-c2cnn(C)c2)c(-c2cn3c4c(cccc24)CCC3)n1	C68H88N14O10S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-7YGFZT	WO2018119441A1_153	.	COc1cc(N2CC(N(C)C)C2)c(NC(=O)/C=C/CNCCOCCOCCOCCOc2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)cc1Nc1ncc(-c2cnn(C)c2)c(-c2cn3c4c(cccc24)CCC3)n1	C56H64N12O10	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-6SIWNK	WO2018119441A1_154	.	COc1cc(N2CC(N(C)C)C2)c(NC(=O)/C=C/CNCCOCCOCCOCCOc2cc([C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCc3ccc(-c4scnc4C)cc3)C(C)C)on2)cc1Nc1ncc(-c2cnn(C)c2)c(-c2cn3c4c(cccc24)CCC3)n1	C67H82N14O10S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-C3UCW8	WO2018119441A1_155	.	COc1cc(N(C)CCCOCCOCCOCCOCCOCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)c2ccc(-c3scnc3C)cc2)C(C)(C)C)c(N)cc1Nc1ncc(-c2cnn(C)c2)c(-c2cn3c4c(cccc24)CCC3)n1	C63H82N12O10S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-KM8ZOE	WO2018119441A1_156	.	COc1cc(N(C)CCCOCCOCCOCCOCCOc2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)c(N)cc1Nc1ncc(-c2cnn(C)c2)c(-c2cn3c4c(cccc24)CCC3)n1	C51H58N10O10	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-TUPB6L	WO2018119441A1_157	.	COc1cc(N(C)CCCOCCOCCOCCOCCOc2cc([C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCc3ccc(-c4scnc4C)cc3)C(C)C)on2)c(N)cc1Nc1ncc(-c2cnn(C)c2)c(-c2cn3c4c(cccc24)CCC3)n1	C62H76N12O10S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-8X9BVP	WO2018119441A1_158	.	COc1cc(N(C)CCCOCCOCCOCCOCCOCC(=O)N[C@H](C(=O)N2C[C@H](O)CC2C(=O)N[C@@H](C)c2ccc(-c3scnc3C)cc2)C(C)(C)C)ccc1Nc1ncc(-c2cnn(C)c2)c(-c2cn3c4c(cccc24)CCC3)n1	C63H81N11O10S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-LG3EVR	WO2018119441A1_159	.	COc1cc(N(C)CCCOCCOCCOCCOCCOc2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)ccc1Nc1ncc(-c2cnn(C)c2)c(-c2cn3c4c(cccc24)CCC3)n1	C51H57N9O10	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-CIU56W	WO2018119441A1_160	.	COc1cc(NCCCOCCOCCOCCOCCOc2cc([C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCc3ccc(-c4scnc4C)cc3)C(C)C)on2)ccc1Nc1ncc(-c2cnn(C)c2)c(-c2cn3c4c(cccc24)CCC3)n1	C61H73N11O10S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-NK62RO	WO2018119441A1_161	.	COc1cc(N2CCN(CCOCCOCCOCCOCCOCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](C)c3ccc(-c4scnc4C)cc3)C(C)(C)C)CC2)ccc1Nc1ncc(-c2cnn(C)c2)c(-c2cn3c4c(cccc24)CCC3)n1	C65H84N12O10S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-WMN0Q9	WO2018119441A1_162	.	COc1cc(N2CCN(C(=O)COCCOCCOCCOCCOCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](C)c3ccc(-c4scnc4C)cc3)C(C)(C)C)CC2)ccc1Nc1ncc(-c2cnn(C)c2)c(-c2cn3c4c(cccc24)CCC3)n1	C65H82N12O11S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-JQZ5F6	WO2018119441A1_163	.	COc1cc(N2CCN(CCOCCOCCOCCOCCOc3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)ccc1Nc1ncc(-c2cnn(C)c2)c(-c2cn3c4c(cccc24)CCC3)n1	C53H60N10O10	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-MCKVNF	WO2018119441A1_164	.	COc1cc(N2CCN(C(=O)COCCOCCOCCOCCOc3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)ccc1Nc1ncc(-c2cnn(C)c2)c(-c2cn3c4c(cccc24)CCC3)n1	C53H58N10O11	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-DISA93	WO2018119441A1_165	.	COc1cc(N2CCN(CCOCCOCCOCCOCCOc3cc([C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)NCc4ccc(-c5scnc5C)cc4)C(C)C)on3)CC2)ccc1Nc1ncc(-c2cn[nH]c2)c(-c2cn3c4c(cccc24)CCC3)n1	C63H76N12O10S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-LKXYNR	WO2018119441A1_166	.	COc1cc(N2CCN(C(=O)COCCOCCOCCOCCOc3cc([C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)NCc4ccc(-c5scnc5C)cc4)C(C)C)on3)CC2)ccc1Nc1ncc(-c2cnn(C)c2)c(-c2cn3c4c(cccc24)CCC3)n1	C64H76N12O11S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-XI8FN7	WO2018119441A1_167	.	COc1cc(N2CCNCC2)c(OCCOCCOCCOCCOCCOCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)c2ccc(-c3scnc3C)cc2)C(C)(C)C)cc1Nc1ncc(-c2cnn(C)c2)c(-c2cn3c4c(cccc24)CCC3)n1	C65H84N12O11S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-N01ST4	WO2018119441A1_168	.	COc1cc(N2CCN(C)CC2)c(OCCOCCOCCOCCOCCOc2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)cc1Nc1ncc(-c2cnn(C)c2)c(-c2cn3c4c(cccc24)CCC3)n1	C54H62N10O11	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-GV0MJO	WO2018119441A1_169	.	COc1cc(N2CCN(C)CC2)c(OCCOCCOCCOCCOCCOc2cc([C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCc3ccc(-c4scnc4C)cc3)C(C)C)on2)cc1Nc1ncc(-c2cnn(C)c2)c(-c2cn3c4c(cccc24)CCC3)n1	C65H80N12O11S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-DDTOKZ	WO2018119441A1_170	.	COc1cc(N2CCN(C)CC2)c(C#CCOCCOCCOCCOCCOCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)c2ccc(-c3scnc3C)cc2)C(C)(C)C)cc1Nc1ncc(-c2cnn(C)c2)c(-c2cn3c4c(cccc24)CCC3)n1	C67H84N12O10S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-6L05SP	WO2018119441A1_171	.	COc1cc(N2CCN(C)CC2)c(C#CCOCCOCCOCCOCCOc2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)cc1Nc1ncc(-c2cnn(C)c2)c(-c2cn3c4c(cccc24)CCC3)n1	C55H60N10O10	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-UR2XTV	WO2018119441A1_172	.	COc1cc(N2CCN(C)CC2)c(C#CCOCCOCCOCCOCCOc2cc([C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCc3ccc(-c4scnc4C)cc3)C(C)C)on2)cc1Nc1ncc(-c2cnn(C)c2)c(-c2cn3c4c(cccc24)CCC3)n1	C66H78N12O10S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-V91Z90	WO2018119441A1_173	.	COc1cc(N2CCN(C)CC2)c(C#CCOCCOCCOCCOCCOCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)c2ccc(-c3scnc3C)cc2)C(C)(C)C)cc1Nc1ncc(C(F)(F)F)c(-c2cn3c4c(cccc24)CCC3)n1	C64H79F3N10O10S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-X8IK1E	WO2018119441A1_174	.	COc1cc(N2CCN(C)CC2)c(C#CCOCCOCCOCCOCCOc2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)cc1Nc1ncc(C(F)(F)F)c(-c2cn3c4c(cccc24)CCC3)n1	C52H55F3N8O10	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-5OQJZH	WO2018119441A1_175	.	COc1cc(N2CCN(C)CC2)c(C#CCOCCOCCOCCOCCOc2cc([C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCc3ccc(-c4scnc4C)cc3)C(C)C)on2)cc1Nc1ncc(C(F)(F)F)c(-c2cn3c4c(cccc24)CCC3)n1	C63H73F3N10O10S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-PBPUON	WO2018119441A1_176	.	COc1cc(N2CCN(C)CC2)c(C#CCOCCCCCN2CCN(CCOCC(=O)N[C@H](C(=O)N3C[C@H](O)CC3C(=O)N[C@@H](C)c3ccc(-c4scnc4C)cc3)C(C)(C)C)CC2)cc1Nc1cc(-c2cn3c4c(cccc24)CCC3)c(-c2cnn(C)c2)cn1	C71H91N13O7S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-NWY6FA	WO2018119441A1_177	.	COc1cc(N2CCNCC2)c(C#CCOCCCCCN2CCN(CCOc3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)cc1Nc1ncc(-c2cnn(C)c2)c(-c2cn3c4c(cccc24)CCC3)n1	C57H64N12O7	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-3QSMFZ	WO2018119441A1_178	.	COc1cc(N2CCN(C)CC2)c(C#CCOCCCCCN2CCN(CCOc3cc([C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)NCc4ccc(-c5scnc5C)cc4)C(C)C)on3)CC2)cc1Nc1ncc(-c2cnn(C)c2)c(-c2cn3c4c(cccc24)CCC3)n1	C69H84N14O7S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-BFYX9U	WO2018119441A1_179	.	COc1cc(N2CCN(C)CC2)c(C#CCOCCCCCN2CCN(CCOCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](C)c3ccc(-c4scnc4C)cc3)C(C)(C)C)CC2)cc1Nc1ncc(C(F)(F)F)c(-c2cn3c4c(cccc24)CCC3)n1	C67H85F3N12O7S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-FKVRPO	WO2018119441A1_180	.	COc1cc(N2CCN(C)CC2)c(C#CCOCCCCCN2CCN(CCOc3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)cc1Nc1ncc(C(F)(F)F)c(-c2cn3c4c(cccc24)CCC3)n1	C55H61F3N10O7	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-B2AG2D	WO2018119441A1_181	.	COc1cc(N2CCN(C)CC2)c(C#CCOCCCCCN2CCN(CCOc3cc([C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)NCc4ccc(-c5scnc5C)cc4)C(C)C)on3)CC2)cc1Nc1ncc(C(F)(F)F)c(-c2cn3c4c(cccc24)CCC3)n1	C66H79F3N12O7S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-AEUU2L	WO2018119441A1_182	.	C=CC(=O)Nc1cccc(Oc2nc(Nc3ccc(N4CCN(C(=O)COCCOCCOCCOCCOCC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)c5ccc(-c6scnc6C)cc5)C(C)(C)C)CC4)cc3OC)ncc2Cl)c1	C59H75ClN10O13S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-HMSCZZ	WO2018119441A1_183	.	C=CC(=O)Nc1cccc(Oc2nc(Nc3ccc(N4CCN(C(=O)COCCOCCOCCOCCOc5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)cc3OC)ncc2Cl)c1	C47H51ClN8O13	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-M3FYRC	WO2018119441A1_184	.	C=CC(=O)Nc1cccc(Oc2nc(Nc3ccc(N4CCN(C(=O)COCCOCCOCCOCCOc5cc([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)Nc6ccc(-c7scnc7C)cc6)C(C)C)on5)CC4)cc3OC)ncc2Cl)c1	C57H67ClN10O13S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-Q2BC9N	WO2018119441A1_185	.	C=CC(=O)Nc1cccc(Oc2nc(Nc3ccc(N4CCN(CCOCCOCCOCCOCCOCC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)c5ccc(-c6scnc6C)cc5)C(C)(C)C)CC4)cc3OC)ncc2Cl)c1	C59H77ClN10O12S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-K4M5EW	WO2018119441A1_186	.	C=CC(=O)Nc1cccc(Oc2nc(Nc3ccc(N4CCN(CCOCCOCCOCCOCCOc5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)cc3OC)ncc2Cl)c1	C47H53ClN8O12	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-GGN30V	WO2018119441A1_187	.	C=CC(=O)Nc1cccc(Oc2nc(Nc3ccc(N4CCN(CCOCCOCCOCCOCCOc5cc([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)NCc6ccc(-c7scnc7C)cc6)C(C)C)on5)CC4)cc3OC)ncc2Cl)c1	C58H71ClN10O12S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-R77UYC	WO2018119441A1_188	.	COc1cc(N2CCN(C)CC2)ccc1Nc1cc(Oc2cccc(NC(=O)/C=C/CNCCOCCOCCOCCOCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](C)c3ccc(-c4scnc4C)cc3)C(C)(C)C)c2)c(Cl)cn1	C60H79ClN10O11S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-B3BTLS	WO2018119441A1_189	.	COc1cc(N2CCN(C)CC2)ccc1Nc1ncc(Cl)c(Oc2cccc(NC(=O)/C=C/CNCCOCCOCCOCCOc3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)c2)n1	C47H54ClN9O11	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-KZ9BZG	WO2018119441A1_190	.	COc1cc(N2CCN(C)CC2)ccc1Nc1ncc(Cl)c(Oc2cccc(NC(=O)/C=C/CNCCOCCOCCOCCOc3cc([C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)NCc4ccc(-c5scnc5C)cc4)C(C)C)on3)c2)n1	C58H72ClN11O11S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-88I54O	WO2018119441A1_191	.	COc1cc(N2CCN(C)CC2)ccc1Nc1ncc(Cl)c(Oc2cccc(NC(=O)/C=C/CCCCOCCOCCOCCOCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](C)c3ccc(-c4scnc4C)cc3)C(C)(C)C)c2)n1	C60H79ClN10O11S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-RON2FC	WO2018119441A1_192	.	COc1cc(N2CCN(C)CC2)ccc1Nc1ncc(C)c(Oc2cccc(NC(=O)/C=C/CCCCOCCOCCOCCOc3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)c2)n1	C49H58N8O11	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-XRW2KP	WO2018119441A1_193	.	COc1cc(N2CCN(C)CC2)ccc1Nc1ncc(O)c(Oc2cccc(NC(=O)/C=C/CCCCOCCOCCOCCOc3cc([C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)NCc4ccc(-c5scnc5C)cc4)C(C)C)on3)c2)n1	C59H74N10O12S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-2H7EVG	WO2018119441A1_194	.	COc1cc(N2CCN(C)CC2)ccc1Nc1ncc(Cl)c(Oc2cccc(OCCOCCOCCOCCOCCOCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(O)N[C@@H](C)c3ccc(-c4scnc4C)cc3)C(C)(C)C)c2)n1	C57H78ClN9O12S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-OLNPHN	WO2018119441A1_195	.	COc1cc(N2CCN(C)CC2)ccc1Nc1ncc(Cl)c(Oc2cccc(OCCOCCOCCOCCOCCOc3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)c2)n1	C45H52ClN7O12	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-QN5LYR	WO2018119441A1_196	.	COc1cc(N2CCN(C)CC2)ccc1Nc1ncc(Cl)c(Oc2cccc(OCCOCCOCCOCCOCCOc3cc([C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)NCc4ccc(-c5scnc5C)cc4)C(C)C)on3)c2)n1	C56H70ClN9O12S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-KPCJ5U	WO2018119441A1_197	.	COc1cc(N2CCN(C)CC2)ccc1Nc1ncc(Cl)c(Oc2cccc(OCCCCCN3CCN(CCCCCOCC(=O)NC(C(=O)N4C[C@H](O)C[C@H]4C(=O)N[C@@H](C)c4ccc(-c5scnc5C)cc4)C(C)(C)C)CC3)c2)n1	C61H84ClN11O8S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-CQ68PN	WO2018119441A1_198	.	COc1cc(N2CCN(C)CC2)ccc1Nc1ncc(Cl)c(Oc2cccc(OCCCCCN3CCN(CCCCCOc4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)c2)n1	C49H60ClN9O8	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-KXTU8P	WO2018119441A1_199	.	COc1cc(N2CCN(C)CC2)ccc1Nc1ncc(Cl)c(Oc2cccc(OCCCCCN3CCN(CCCCCOc4cc([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)NCc5ccc(-c6scnc6C)cc5)C(C)C)on4)CC3)c2)n1	C60H78ClN11O8S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-RB4F4F	WO2018119441A1_200	.	COc1nn(C)cc1Nc1nc(N2C[C@@H](F)[C@H](NC(=O)/C=C/CNCCN3CCN(CCCCCOCC(=O)NC(C(=O)N4C[C@H](O)C[C@H]4C(=O)N[C@@H](C)c4ccc(-c5scnc5C)cc4)C(C)(C)C)CC3)C2)nc2c1ncn2C	C55H79FN16O7S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-QOG29J	WO2018119441A1_201	.	COc1nn(C)cc1Nc1nc(N2C[C@@H](F)[C@H](NC(=O)/C=C/CNCCN3CCN(CCCCCOc4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)C2)nc2c1ncn2C	C43H55FN14O7	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-F94EFJ	WO2018119441A1_202	.	COc1nn(C)cc1Nc1nc(N2C[C@@H](F)[C@H](NC(=O)/C=C/CNCCN3CCN(CCCCCOc4cc([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)NCc5ccc(-c6scnc6C)cc5)C(C)C)on4)CC3)C2)nc2c1ncn2C	C54H73FN16O7S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-XD4M9Q	WO2018119441A1_203	.	COc1nn(C)cc1Nc1nc(N2C[C@@H](F)[C@H](NC(=O)/C=C/CCCCN3CCN(CCCCCOCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)N[C@@H](C)c4ccc(-c5scnc5C)cc4)C(C)(C)C)CC3)C2)nc2c1ncn2C	C56H80FN15O7S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-AAT3D3	WO2018119441A1_204	.	COc1nn(C)cc1Nc1nc(N2C[C@@H](F)[C@H](NC(=O)/C=C/CCCCN3CCN(CCCCCOc4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)C2)nc2c1ncn2C	C44H56FN13O7	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-G2JWOS	WO2018119441A1_205	.	COc1nn(C)cc1Nc1nc(N2C[C@@H](F)[C@H](NC(=O)/C=C/CCCCN3CCN(CCCCCOc4cc([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)NCc5ccc(-c6scnc6C)cc5)C(C)C)on4)CC3)C2)nc2c1ncn2C	C55H74FN15O7S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-GUTX3L	WO2018119441A1_206	.	COc1nn(C)cc1Nc1nc(N2C[C@@H](F)[C@H](NC(=O)/C=C/CNCCOCCOCCOCCOCC(O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](C)c3ccc(-c4scnc4C)cc3)C(C)(C)C)C2)nc2c1ncn2C	C52H75FN14O10S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-PD96NP	WO2018119441A1_207	.	COc1nn(C)cc1Nc1nc(N2C[C@@H](F)[C@H](NC(=O)/C=C/CNCCOCCOCCOCCOc3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)nc2c1ncn2C	C40H49FN12O10	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-6CN09D	WO2018119441A1_208	.	COc1nn(C)cc1Nc1nc(N2C[C@@H](F)[C@H](NC(=O)/C=C/CNCCOCCOCCOCCOc3cc([C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)NCc4ccc(-c5scnc5C)cc4)C(C)C)on3)C2)nc2c1ncn2C	C51H67FN14O10S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-D3X5R7	WO2018119441A1_209	.	C=CC(=O)N[C@@H]1CN(c2nc(Nc3cn(CCOCCOCCOCCOCCOCCOCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)N[C@@H](C)c4ccc(-c5scnc5C)cc4)C(C)(C)C)nc3OC)c3ncn(C)c3n2)C[C@H]1F	C54H76FN13O12S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-YP64V4	WO2018119441A1_210	.	C=CC(=O)N[C@@H]1CN(c2nc(Nc3cn(CCOCCOCCOCCOCCOCCOc4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)nc3OC)c3ncn(C)c3n2)C[C@H]1F	C42H52FN11O12	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-AQOEQX	WO2018119441A1_211	.	C=CC(=O)N[C@@H]1CN(c2cc(Nc3cn(CCOCCOCCOCCOCCOCCOc4cc([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)NCc5ccc(-c6scnc6C)cc5)C(C)C)on4)nc3OC)c3ncn(C)c3n2)C[C@H]1F	C54H71FN12O12S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-XTPFQQ	WO2018119441A1_212	.	C=CC(=O)N[C@@H]1CN(c2nc(Nc3cn(CCCCCCCOCCCCCOCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)N[C@@H](C)c4ccc(-c5scnc5C)cc4)C(C)(C)C)nc3OC)c3ncn(C)c3n2)C[C@H]1F	C54H76FN13O8S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-G0UJWX	WO2018119441A1_213	.	C=CC(=O)N[C@@H]1CN(c2nc(Nc3cn(CCCCOCCOCCCCCOc4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)nc3OC)c3ncn(C)c3n2)C[C@H]1F	C41H50FN11O9	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-9CAD06	WO2018119441A1_214	.	C=CC(=O)N[C@@H]1CN(c2nc(Nc3cn(CCCCOCCOCCCCCOc4cc([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)NCc5ccc(-c6scnc6C)cc5)C(C)C)on4)nc3OC)c3ncn(C)c3n2)C[C@H]1F	C52H68FN13O9S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-9GGV8E	WO2018119441A1_215	.	C=CC(=O)N[C@@H]1CN(c2nc(Nc3cn(CCCCCN4CCN(CCCCOCC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)c5ccc(-c6scnc6C)cc5)C(C)(C)C)CC4)nc3OC)c3ncn(C)c3n2)C[C@H]1N	C55H80N16O7S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-ORHN5M	WO2018119441A1_216	.	C=CC(=O)N[C@@H]1CN(c2nc(Nc3cn(CCCCCN4CCN(CCCCOc5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)nc3OC)c3ncn(C)c3n2)C[C@H]1F	C43H54FN13O7	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-VOQEW0	WO2018119441A1_217	.	C=CC(=O)N[C@@H]1CN(c2nc(Nc3cn(CCCCCN4CCN(CCCCOc5cc([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)NCc6ccc(-c7scnc7C)cc6)C(C)C)on5)CC4)nc3OC)c3ncn(C)c3n2)C[C@H]1F	C54H72FN15O7S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-JM1LAW	WO2018119441A1_218	.	COc1nn(C)cc1Nc1nc(N2C[C@@H](F)[C@H](NCCOCCOCCOCCOCCOCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](C)c3ccc(-c4scnc4C)cc3)C(C)(C)C)C2)nc2c1N=CC2C	C51H73FN12O10S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-OG36H5	WO2018119441A1_219	.	COc1nn(C)cc1Nc1nc(N2C[C@@H](F)[C@H](NCCOCCOCCOCCOCCOc3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)nc2c1ncn2C	C38H48FN11O10	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-TEA2BC	WO2018119441A1_220	.	COc1nn(C)cc1Nc1nc(N2C[C@@H](F)[C@H](NCCOCCOCCOCCOCCOc3cc([C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)NCc4ccc(-c5scnc5C)cc4)C(C)C)on3)C2)nc2c1ncn2C	C49H66FN13O10S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-1BT06C	WO2018119441A1_221	.	CO[C@@H]1CN(C(=O)/C=C/CNCCOCCOCCOCCOCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)c2ccc(-c3scnc3C)cc2)C(C)(C)C)C[C@H]1COc1nc(N/C(C=N)=C/N(C)C)nc2[nH]cc(Cl)c12	C54H77ClN12O11S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-09RQYH	WO2018119441A1_222	.	CO[C@@H]1CN(C(=O)/C=C/CNCCOCCOCCOCCOc2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)C[C@H]1COc1nc(Nc2cnn(C)c2)nc2[nH]cc(Cl)c12	C41H49ClN10O11	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-5ZMOAQ	WO2018119441A1_223	.	CO[C@@H]1CN(C(=O)/C=C/CNCCOCCOCCOCCOc2cc([C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCc3ccc(-c4scnc4C)cc3)C(C)C)on2)C[C@H]1COc1nc(Nc2cnn(C)c2)nc2[nH]cc(Cl)c12	C52H67ClN12O11S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-5UEQC1	WO2018119441A1_224	.	C=CC(=O)N1C[C@@H](COc2nc(Nc3ccn(CCOCCOCCOCCOCCOCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)N[C@@H](C)c4ccc(-c5scnc5C)cc4)C(C)(C)C)c3)nc3[nH]cc(Cl)c23)[C@H](O)C1	C53H71ClN10O12S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-MHVKU8	WO2018119441A1_225	.	C=CC(=O)N1C[C@@H](COc2nc(Nc3cnn(CCOCCOCCOCCOCCOc4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)c3)nc3[nH]cc(Cl)c23)[C@H](OC)C1	C41H48ClN9O12	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-BYLLD6	WO2018119441A1_226	.	C=CC(=O)N1C[C@@H](COc2nc(Nc3cnn(CCOCCOCCOCCOCCOc4cc([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)NCc5ccc(-c6scnc6C)cc5)C(C)C)on4)c3)nc3[nH]cc(Cl)c23)[C@H](OC)C1	C52H66ClN11O12S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-4OV8N8	WO2018119441A1_227	.	CO[C@@H]1CN(CCOCCOCCOCCOCCOCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)c2ccc(-c3scnc3C)cc2)C(C)(C)C)C[C@H]1COc1nc(Nc2cnn(C)c2)nc2[nH]cc(Cl)c12	C51H72ClN11O11S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-62E94F	WO2018119441A1_228	.	CO[C@@H]1CN(CCOCCOCCOCCOCCOc2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)C[C@H]1COc1nc(Nc2cnn(C)c2)nc2[nH]cc(Cl)c12	C39H48ClN9O11	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-66DCNL	WO2018119441A1_229	.	CO[C@@H]1CN(CCOCCOCCOCCCCCOc2cc([C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCc3ccc(-c4scnc4C)cc3)C(C)C)on2)C[C@H]1COc1nc(Nc2cnn(C)c2)nc2[nH]cc(Cl)c12	C51H68ClN11O10S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-JQXGCW	WO2018119441A1_230	.	Cc1cc(C(=O)Nc2nc3cccc(Cl)c3n2[C@@H]2CCCCN(C(=O)/C=C/CN(C)CCOCCOCCOCCOCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](C)c3ccc(-c4scnc4C)cc3)C(C)(C)C)C2)ccn1	C58H77ClN10O10S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-P9YVTF	WO2018119441A1_231	.	Cc1cc(C(=O)Nc2nc3cccc(Cl)c3n2[C@@H]2CCCCN(C(=O)/C=C/CN(C)CCOCCOCCOCCOc3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)ccn1	C46H53ClN8O10	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-507W4T	WO2018119441A1_232	.	Cc1cc(C(=O)Nc2nc3cccc(Cl)c3n2[C@@H]2CCCCN(C(=O)/C=C/CN(C)CCOCCOCCOCCOc3cc([C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)NCc4ccc(-c5scnc5C)cc4)C(C)C)on3)C2)ccn1	C57H71ClN10O10S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-NVD8XQ	WO2018119441A1_233	.	Cc1cc(C(=O)Nc2nc3cccc(Cl)c3n2[C@@H]2CCCCN(C(=O)/C=C/CCCCOCCOCCOCCOCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](C)c3ccc(-c4scnc4C)cc3)C(C)(C)C)C2)ccn1	C58H76ClN9O10S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-WUP51O	WO2018119441A1_234	.	Cc1cc(C(=O)Nc2nc3cccc(Cl)c3n2[C@@H]2CCCCN(C(=O)/C=C/CCCCOCCOCCOCCOc3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)ccn1	C46H52ClN7O10	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-ZJYNA3	WO2018119441A1_235	.	Cc1cc(C(=O)Nc2nc3cccc(Cl)c3n2[C@@H]2CCCCN(C(=O)/C=C/CCCCOCCOCCOCCOc3cc([C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)NCc4ccc(-c5scnc5C)cc4)C(C)C)on3)C2)ccn1	C57H70ClN9O10S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-UT7X8T	WO2018119441A1_236	.	C=CC(=O)N1CCCC[C@H](n2c(NC(=O)c3ccnc(C)c3)nc3ccc(OCCOCCOCCOCCOCCOCC(=O)N[C@H](C(=O)N4C[C@H](O)CC4C(=O)N[C@@H](C)c4ccc(-c5scnc5C)cc4)C(C)(C)C)c(Cl)c32)C1	C58H76ClN9O12S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-MEBAXC	WO2018119441A1_237	.	C=CC(=O)N1CCCC[C@H](n2c(NC(=O)c3ccnc(C)c3)nc3ccc(OCCOCCOCCOCCOCCOc4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)c(Cl)c32)C1	C46H52ClN7O12	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-6XPLSI	WO2018119441A1_238	.	C=CC(=O)N1CCCC[C@H](n2c(NC(=O)c3ccnc(C)c3)nc3ccc(OCCOCCOCCOCCOCCOc4cc([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)NCc5ccc(-c6scnc6C)cc5)C(C)C)on4)c(Cl)c32)C1	C57H70ClN9O12S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-TPL9DN	WO2018119441A1_239	.	C=CC(=O)N1CCCC[C@H](n2c(NC(=O)c3ccnc(C)c3)nc3ccc(OCCOCCN4CCN(CCOCCOCC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)c5ccc(-c6scnc6C)cc5)C(C)(C)C)CC4)c(Cl)c32)C1	C60H80ClN11O10S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-NGE18W	WO2018119441A1_240	.	C=CC(=O)N1CCCC[C@H](n2c(NC(=O)c3ccnc(C)c3)nc3ccc(OCCOCCN4CCN(CCOCCOc5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)c(Cl)c32)C1	C48H56ClN9O10	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-A4RGMS	WO2018119441A1_241	.	C=CC(=O)N1CCCC[C@H](n2c(NC(=O)c3ccnc(C)c3)nc3ccc(OCCOCCN4CCN(CCOCCOc5cc([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)NCc6ccc(-c7scnc7C)cc6)C(C)C)on5)CC4)c(Cl)c32)C1	C59H74ClN11O10S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-COM67X	WO2018119441A1_242	.	C=CC(=O)N1CCCC[C@H](n2c(NC(=O)c3ccnc(C)c3)nc3ccc(OCCCCCN4CCN(CCCCCOCC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)c5ccc(-c6scnc6C)cc5)C(C)(C)C)CC4)c(Cl)c32)C1	C62H84ClN11O8S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-J2TTWH	WO2018119441A1_243	.	C=CC(=O)N1CCCC[C@H](n2c(NC(=O)c3ccnc(C)c3)nc3ccc(OCCCCCN4CCN(CCCCCOc5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)c(Cl)c32)C1	C50H60ClN9O8	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-8UX2T2	WO2018119441A1_244	.	C=CC(=O)N1CCCC[C@H](n2c(NC(=O)c3ccnc(C)c3)nc3ccc(OCCCCCN4CCN(CCCCCOc5cc([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)NCc6ccc(-c7scnc7C)cc6)C(C)C)on5)CC4)c(Cl)c32)C1	C61H78ClN11O8S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-LIXMX6	WO2018119441A1_245	.	Cc1cc(C(=O)Nc2nc3cccc(Cl)c3n2[C@@H]2CCCCN(CCOCCOCCOCCOCCOCC(=O)N[C@H](C(=O)N3CC(O)C[C@H]3C(=O)N[C@@H](C)c3ccc(-c4scnc4C)cc3)C(C)(C)C)C2)ccn1	C55H74ClN9O10S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-CPFUTH	WO2018119441A1_246	.	Cc1cc(C(=O)Nc2nc3cccc(Cl)c3n2[C@@H]2CCCCN(CCOCCOCCOCCOCCOc3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)ccn1	C43H50ClN7O10	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-P7U7ID	WO2018119441A1_247	.	Cc1cc(C(=O)Nc2nc3cccc(Cl)c3n2[C@@H]2CCCCN(CCOCCOCCOCCOCCOc3cc([C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)NCc4ccc(-c5scnc5C)cc4)C(C)C)on3)C2)ccn1	C54H68ClN9O10S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-R861OJ	WO2018119441A1_248	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCN2CCN(Cc3ccc(-c4cc5c(Nc6ccc(OCc7cccc(F)c7)c(Cl)c6)ncnc5[nH]4)cc3)CC2)C(C)(C)C)cc1	C61H72ClFN10O8S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-TE9G1X	WO2018119441A1_249	.	O=C1CCC(N2C(=O)c3ccc(OCCOCCOCCOCCN4CCN(Cc5ccc(-c6cc7c(Nc8ccc(OCc9cccc(F)c9)c(Cl)c8)ncnc7[nH]6)cc5)CC4)cc3C2=O)C(=O)N1	C51H52ClFN8O9	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-WQ1SFI	WO2018119441A1_250	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](c2cc(OCCOCCOCCN3CCN(Cc4ccc(-c5cc6c(Nc7ccc(OCc8cccc(F)c8)c(Cl)c7)ncnc6[nH]5)cc4)CC3)no2)C(C)C)cc1	C60H66ClFN10O8S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-E9NO5N	WO2018119441A1_251	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCN2CCN(Cc3ccc(-c4cc5c(Nc6ccc(OCc7ccccn7)c(Cl)c6)c(C#N)cnc5[nH]4)cc3)CC2)C(C)(C)C)cc1	C62H72ClN11O8S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-474DQT	WO2018119441A1_252	.	N#Cc1cnc2[nH]c(-c3ccc(CN4CCN(CCOCCOCCOCCOc5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)cc3)cc2c1Nc1ccc(OCc2ccccn2)c(Cl)c1	C52H52ClN9O9	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-SANTJL	WO2018119441A1_253	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](c2cc(OCCOCCOCCN3CCN(Cc4ccc(-c5cc6c(Nc7ccc(OCc8ccccn8)c(Cl)c7)c(C#N)cnc6[nH]5)cc4)CC3)no2)C(C)C)cc1	C61H66ClN11O8S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-TCG04A	WO2018119441A1_254	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCOCC#Cc2cccc3c2C(=O)N(C(C(=O)Nc2nccs2)c2cc(F)ccc2O)C3)C(C)(C)C)cc1	C53H60FN7O11S2	EGFR	P00533	VHL	WO-2018119441-A1
TPD-Y5OPCP	WO2018119441A1_255	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCOCCOCC#Cc2cccc3c2C(=O)N(C(C(=O)Nc2nccs2)c2cc(F)ccc2O)C3)C(C)(C)C)cc1	C55H64FN7O12S2	EGFR	P00533	VHL	WO-2018119441-A1
TPD-UZDNZF	SCHEMBL20305708	(2S,4R)-N-[[2-[2-[2-[3-[2-[1-(5-fluoro-2-hydroxyphenyl)-2-oxo-2-(1,3-thiazol-2-ylamino)ethyl]-3-oxo-1H-isoindol-4-yl]prop-2-ynoxy]ethoxy]ethoxy]-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-4-hydroxy-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](C(C)C)N2Cc3ccccc3C2=O)c(OCCOCCOCC#Cc2cccc3c2C(=O)N(C(C(=O)Nc2nccs2)c2cc(F)ccc2O)C3)c1	C55H54FN7O10S2	EGFR	P00533	VHL	WO-2018119441-A1
TPD-7BCOID	WO2018119441A1_258	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](C(C)C)N2Cc3ccccc3C2=O)c(OCCOCCOCCOCC#Cc2cccc3c2C(=O)N(C(C(=O)Nc2nccs2)c2cc(F)ccc2O)C3)c1	C57H58FN7O11S2	EGFR	P00533	VHL	WO-2018119441-A1
TPD-YEM0YC	WO2018119441A1_259	.	Cc1ccc(O)c(C(C(=O)Nc2nccs2)N2Cc3cccc(C#CCOCCOCCOCCOCCOc4cc(-c5scnc5C)ccc4CNC(=O)[C@@H]4C[C@@H](O)CN4C(=O)[C@H](C(C)C)N4Cc5ccccc5C4=O)c3C2=O)c1	C60H65N7O12S2	EGFR	P00533	VHL	WO-2018119441-A1
TPD-C7FXAB	WO2018119441A1_260	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](C(C)C)N2Cc3ccccc3C2=O)c(OCCOCCOCCOCCOCCOCC#Cc2cccc3c2C(=O)N(C(C(=O)Nc2nccs2)c2cc(F)ccc2O)C3)c1	C61H66FN7O13S2	EGFR	P00533	VHL	WO-2018119441-A1
TPD-SAVNJG	WO2018119441A1_261	.	O=C1CCC(N2C(=O)c3ccc(OCCOCCOCCOCC#Cc4cccc5c4C(=O)N(C(C(=O)Nc4nccs4)c4cc(F)ccc4O)C5)cc3C2=O)C(=O)N1	C41H36FN5O11S	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-PN9NH4	WO2018119441A1_262	.	O=C1CCC(N2C(=O)c3ccc(OCCOCCOCCOCCOCC#Cc4cccc5c4C(=O)N(C(C(=O)Nc4nccs4)c4cc(F)ccc4O)C5)cc3C2=O)C(=O)N1	C43H40FN5O12S	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-X5T9EK	WO2018119441A1_263	.	O=C1CCC(N2C(=O)c3ccc(OCCOCCOCCOCCOCCOCC#Cc4cccc5c4C(=O)N(C(C(=O)Nc4nccs4)c4cc(F)ccc4O)C5)cc3C2=O)C(=O)N1	C45H44FN5O13S	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-AJY3AJ	WO2018119441A1_264	.	O=C1CCC(N2C(=O)c3cccc(NCCOCCOCC#Cc4cccc5c4C(=O)N(C(C(=O)Nc4nccs4)c4cc(F)ccc4O)C5)c3C2=O)C(=O)N1	C39H33FN6O9S	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-0R79Y4	WO2018119441A1_265	.	O=C1CCC(N2C(=O)c3cccc(NCCOCCOCCOCC#Cc4cccc5c4C(=O)N(C(C(=O)Nc4nccs4)c4cc(F)ccc4O)C5)c3C2=O)C(=O)N1	C41H37FN6O10S	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-4TPZF8	WO2018119441A1_266	.	O=C1CCC(N2C(=O)c3cccc(NCCOCCOCCOCCOCC#Cc4cccc5c4C(=O)N(C(C(=O)Nc4nccs4)c4cc(F)ccc4O)C5)c3C2=O)C(=O)N1	C43H41FN6O11S	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-QLYISC	WO2018119441A1_267	.	O=C1CCC(N2C(=O)c3cccc(NCCOCCOCCOCCOCCOCC#Cc4cccc5c4C(=O)N(C(C(=O)Nc4nccs4)c4cc(F)ccc4O)C5)c3C2=O)C(=O)N1	C45H45FN6O12S	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-12XSFK	WO2018119441A1_268	.	C=CC(=O)Nc1cc(Nc2nccc(-c3cn(C)c4ccccc34)n2)c(OC)cc1N(C)CCOCCOCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(-c2scnc2C)cc1)C(C)(C)C	C52H62N10O8S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-73BHEV	WO2018119441A1_269	.	C=CC(=O)Nc1cc(Nc2nccc(-c3cn(C)c4ccccc34)n2)c(OC)cc1N(C)CCN(C)CCCCOCCC(=O)N[C@@H](C(=O)N1C[C@@H](O)C[C@@H]1C(=O)NCc1ccc(-c2scnc2C)cc1)C(C)(C)C	C56H71N11O7S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-N9WNCX	WO2018119441A1_270	.	C=CC(=O)Nc1cc(Nc2nccc(-c3cn(C)c4ccccc34)n2)c(OC)cc1N(C)CCN(C)CCCOCCCCOCCCOCCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(-c2scnc2C)cc1)C(C)(C)C	C62H83N11O9S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-FIKJ15	WO2018119441A1_271	.	C=CC(O)Nc1cc(Nc2nccc(-c3cn(C)c4ccccc34)n2)c(OC)cc1N(C)CCN(C)CCCOCCCCOCCCOCCC(=O)NCCNc1ccc2c(c1)C(=O)N(C1CCC(=O)NC1=O)C2=C	C56H73N11O9	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-3SAKRS	WO2018119441A1_272	.	C=CC(=O)Nc1cc(Nc2nccc(-c3cn(C)c4ccccc34)n2)c(OC)cc1NCCN(C)CCCCOCCC(=O)NCCOc1ccc2c(c1)C(=O)N(C1CCC(=O)NC1=O)C2=O	C48H54N10O9	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-E1IB0C	WO2018119441A1_273	.	C=CC(=O)Nc1cc(Nc2nccc(-c3cn(C)c4ccccc34)n2)c(OC)cc1N(C)CCN(C)C(=O)COCCOCCOCCOCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(-c2scnc2C)cc1)C(C)(C)C	C59H75N11O11S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-O6RB60	WO2018119441A1_274	.	C=CC(=O)Nc1cc(Nc2nccc(-c3cn(C)c4ccccc34)n2)c(OC)cc1N(C)CCN(C)CCOCCOCCC(=O)NCCOc1ccc2c(c1)C(=O)N(C1CCC(=O)NC1=O)C2=O	C49H56N10O10	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-LHHJHV	WO2018119441A1_275	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCOCCOCCOCC#Cc2cccc3c2C(=O)N(C(C(=O)Nc2nccs2)c2cc(F)ccc2O)C3)C(C)(C)C)cc1	C57H68FN7O13S2	EGFR	P00533	VHL	WO-2018119441-A1
TPD-WXERTH	SCHEMBL20305573	US10994015, Example 276; BDBM494980; US10994015, Example 276	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@H]2C[C@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOc2ccc(-c3nccc(Nc4cc5c(cn4)nc(C)n5C(C)C)n3)cc2)C(C)(C)C)cc1	C49H60N10O7S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-6URQA4	WO2018119441A1_277	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](C(C)C)N2Cc3ccccc3C2=O)c(OCCCCOc2ccc(-c3nccc(Nc4cc5c(cn4)cc(C)n5C(C)C)n3)cc2)c1	C54H59N9O6S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-0PLKKF	WO2018119441A1_278	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCOc2ccc(-c3nccc(Nc4cc5c(cn4)nc(C)n5C(C)C)n3)cc2)C(C)(C)C)cc1	C50H62N10O8S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-S2SE3E	WO2018119441A1_279	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCOCCOc2ccc(-c3nccc(Nc4cc5c(cn4)nc(C)n5C(C)C)n3)cc2)C(C)(C)C)cc1	C52H66N10O9S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-PWJPIH	WO2018119441A1_280	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCOCCOCCOc2ccc(-c3nccc(Nc4cc5c(cn4)nc(C)n5C(C)C)n3)cc2)C(C)(C)C)cc1	C54H70N10O10S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-HA7HU7	WO2018119441A1_281	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](C(C)C)N2Cc3ccccc3C2=O)c(OCCOCCOCCOCCOc2ccc(-c3nccc(Nc4cc5c(cn4)nc(C)n5C(C)C)n3)cc2)c1	C57H66N10O9S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-WZSGH6	SCHEMBL20305663	US10994015, Example 282; BDBM494986; US10994015, Example 282; (2S,4R)-4-hydroxy-1-((S)-2-(2-(3-(3-(9-(4-((1-isopropyl-2-methyl-1H-imidazo[4,5-c]pyridin-6-yl)amino)pyrimidin-2-yl)-3,9-diazaspiro[5.5]undecan-3-yl)propoxy)propoxy)acetamido)-3,3-dimethylbutanoyl)-N-((S)-1-(4-(4-methylthiazol-5-yl)phenyl)ethyl)pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCCOCCCN2CCC3(CC2)CCN(c2nccc(Nc4cc5c(cn4)nc(C)n5C(C)C)n2)CC3)C(C)(C)C)cc1	C54H76N12O6S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-BCTELE	SCHEMBL20305728	US10994015, Example 283; SCHEMBL31218244; BDBM494987; US10994015, Example 283; 2-(7-(3-(2-(2-(2-((2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindolin-5-yl)oxy)ethoxy)ethoxy)ethoxy)propyl)-1-oxoisoindolin-2-yl)-2-(5-fluoro-2-hydroxyphenyl)-N-(thiazol-2-yl)acetamide	O=C1CCC(N2C(=O)c3ccc(OCCOCCOCCOCCCc4cccc5c4C(=O)N(C(C(=O)Nc4nccs4)c4cc(F)ccc4O)C5)cc3C2=O)C(=O)N1	C41H40FN5O11S	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-6TASA9	WO2018119441A1_284	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCOCCOC2CCN(c3nccc(Nc4cc5c(cn4)nc(C)n5C(C)C)n3)CC2)C(C)(C)C)cc1	C52H73N11O9S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-CYK84A	WO2018119441A1_285	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCCOCCCN2CCOC3(CCN(c4nccc(Nc5cc6c(cn5)nc(C)n6C(C)C)n4)CC3)C2)C(C)(C)C)cc1	C53H74N12O7S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-2BK59V	SCHEMBL20305608	US10994015, Example 286; SCHEMBL31218235; BDBM494990; US10994015, Example 286; 2-(2,6-dioxopiperidin-3-yl)-5-(2-(4-(4-(1-isopropyl-6-((2-(4-methoxypiperidin-1-yl)pyrimidin-4-yl)amino)-1H-imidazo[4,5-c]pyridin-2-yl)benzyl)piperazin-1-yl)ethoxy)isoindoline-1,3-dione	COC1CCN(c2nccc(Nc3cc4c(cn3)nc(-c3ccc(CN5CCN(CCOc6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)cc3)n4C(C)C)n2)CC1	C45H51N11O6	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-3ARBM2	SCHEMBL23314161	US10994015, Example 287; BDBM494991; US10994015, Example 287	COC1CCN(c2nccc(Nc3cc4c(cn3)nc(COCCN3CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC3)n4C(C)(C)C)n2)CC1	C40H49N11O6	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-DF21MT	WO2018119441A1_288	.	COC1CCN(c2nccc(Nc3cc4[nH]c(COCCN5C=CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)nc4cn3)n2)CC1	C36H39N11O6	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-63X1BY	BDBM494993	US10994015, Example 289; US10994015, Example 289	O=C1CCC(N2C(=O)c3ccc(N4CCN(CCCOCCCCNc5cccc6c5C(=O)N(C(C(=O)Nc5nccs5)c5cc(F)ccc5O)C6)CC4)cc3C2=O)C(=O)N1	C43H45FN8O8S	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-WJI9XF	BDBM494994	US10994015, Example 290; US10994015, Example 290	O=C1CCC(N2C(=O)c3ccc(N4CCC(CN5CCC(OCC#Cc6cccc7c6C(=O)N(C(C(=O)Nc6nccs6)c6cc(F)ccc6O)C7)CC5)CC4)cc3C2=O)C(=O)N1	C46H44FN7O8S	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-G6E4RV	SCHEMBL20325439	US10994015, Example 291; BDBM494995; US10994015, Example 291; (2S,4R)-1-((S)-2-(Tert-butyl)-14-(4-((1-(4-((1-isopropyl-2-methyl-1H-imidazo[4,5-c]pyridin-6-yl)amino)pyrimidin-2-yl)piperidin-4-yl)oxy)phenyl)-4-oxo-6,9,12-trioxa-3-azatetradecanoyl)-4-hydroxy-N-((S)-1-(4-(4-methylthiazol-5-yl)phenyl)ethyl)pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCc2ccc(OC3CCN(c4nccc(Nc5cc6c(cn5)nc(C)n6C(C)C)n4)CC3)cc2)C(C)(C)C)cc1	C56H73N11O8S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-SZ19TR	SCHEMBL20305654	US10994015, Example 292; BDBM494996; US10994015, Example 292; (2S,4R)-4-hydroxy-1-((S)-2-(2-(3-(3-(4-(2-(1-(4-((1-isopropyl-2-methyl-1H-imidazo[4,5-c]pyridin-6-yl)amino)pyrimidin-2-yl)-4-methoxypiperidin-4-yl)ethyl)piperazin-1-yl)propoxy)propoxy)acetamido)-3,3-dimethylbutanoyl)-N-((S)-1-(4-(4-methylthiazol-5-yl)phenyl)ethyl)pyrrolidine-2-carboxamide	COC1(CCN2CCN(CCCOCCCOCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](C)c3ccc(-c4scnc4C)cc3)C(C)(C)C)CC2)CCN(c2nccc(Nc3cc4c(cn3)nc(C)n4C(C)C)n2)CC1	C57H83N13O7S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-82ZJ8M	WO2018119441A1_293	.	O=C1CCC(N2C(=O)c3ccc(N4CCN(CC5CCN(CC#Cc6cccc7c6C(=O)N(C(C(=O)Nc6nccs6)C6CC(F)=CCC6O)C7)CC5)CC4)cc3C2=O)C(=O)N1	C45H47FN8O7S	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-RLQHR3	BDBM494998	US10994015, Example 294; US10994015, Example 294	O=C1CCC(N2C(=O)c3ccc(N4CCN(CC5CCN(CCCc6cccc7c6C(=O)N(C(C(=O)Nc6nccs6)c6cc(F)ccc6O)C7)CC5)CC4)cc3C2=O)C(=O)N1	C45H47FN8O7S	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-0WOX46	BDBM494999	US10994015, Example 295; US10994015, Example 295	O=C1CCC(N2C(=O)c3cccc(NCCOCCOCCOCCOCCOCCOCC#Cc4cccc5c4C(=O)N(C(C(=O)Nc4nccs4)c4cc(F)ccc4O)C5)c3C2=O)C(=O)N1	C47H49FN6O13S	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-BKSFTL	WO2018119441A1_296	.	O=C1CCC(N2C(=O)c3ccc(N4CCN(CCCOCCCCCc5cccc6c5C(=O)N(C(C(=O)Nc5nccs5)c5cc(F)ccc5O)C6)CC4)cc3C2=O)C(=O)N1	C44H46FN7O8S	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-NMT8CN	BDBM495001	US10994015, Example 297; US10994015, Example 297	O=C1CCC(N2C(=O)c3ccc(N4CCC(CN5CCC(OCCCc6cccc7c6C(=O)N(C(C(=O)Nc6nccs6)c6cc(F)ccc6O)C7)CC5)CC4)cc3C2=O)C(=O)N1	C46H48FN7O8S	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-KUN6LV	BDBM495003	US10994015, Example 299; US10994015, Example 299	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCOCCOCCOCCOCC#Cc2cccc3c2C(=O)N(C(C(=O)Nc2nccs2)c2cc(F)ccc2O)C3)C(C)(C)C)cc1	C59H72FN7O14S2	EGFR	P00533	VHL	WO-2018119441-A1
TPD-62IGGY	BDBM495004	US10994015, Example 300; US10994015, Example 300	O=C1CCC(N2C(=O)c3cccc(NCCOCCOCCOCCOCCOCCOCCCc4cccc5c4C(=O)N(C(C(=O)Nc4nccs4)c4cc(F)ccc4O)C5)c3C2=O)C(=O)N1	C47H53FN6O13S	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-AOIAWE	SCHEMBL20359612	US10994015, Example 301; BDBM495005; US10994015, Example 301; 2-(2,6-dioxopiperidin-3-yl)-5-(4-(3-(4-(4-(2-((1-isopropyl-6-((2-(4-methoxypiperidin-1-yl)pyrimidin-4-yl)amino)-1H-imidazo[4,5-c]pyridin-2-yl)methoxy)ethyl)piperazin-1-yl)phenoxy)propyl)piperazin-1-yl)isoindoline-1,3-dione	COC1CCN(c2nccc(Nc3cc4c(cn3)nc(COCCN3CCN(c5ccc(OCCCN6CCN(c7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)cc5)CC3)n4C(C)C)n2)CC1	C52H65N13O7	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-H12V5O	WO2018119441A1_302	.	COC1CCN(c2nccc(Nc3cc4c(cn3)nc(COCCN3CCN(c5ccc(C[C@H]6C[C@H](OCC(=O)C[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)NCc7ccc(-c8scnc8C)cc7)C(C)(C)C)C6)cc5)CC3)n4C(C)C)n2)CC1	C62H82N12O7S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-TXJUMH	BDBM495007	US10994015, Example 303; US10994015, Example 303	COC1CCN(c2nccc(Nc3cc4c(cn3)nc(COCCN3CCN(c5ccc(OCCCOCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)NCc6ccc(-c7scnc7C)cc6)C(C)(C)C)cc5)CC3)n4C(C)C)n2)CC1	C59H79N13O8S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-38LJLX	BDBM495008	US10994015, Example 304; US10994015, Example 304	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CO[C@H]2C[C@H](Oc3ccc(N4CCN(CCOCc5nc6cnc(Nc7ccnc(-c8cnn(S(=O)(=O)C9CC9)c8)n7)cc6n5C(C)C)CC4)cc3)C2)C(C)(C)C)cc1	C60H74N14O9S2	EGFR	P00533	VHL	WO-2018119441-A1
TPD-7CX93D	WO2018119441A1_306	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCCOc2ccc(N3CCN(CCOCc4nc5cnc(Nc6ccnc(-c7cnn(S(=O)(=O)C8CC8)c7)n6)cc5n4C(C)C)CC3)cc2)C(C)(C)C)cc1	C59H74N14O9S2	EGFR	P00533	VHL	WO-2018119441-A1
TPD-AC44QA	SCHEMBL20305656	US10994015, Example 307; BDBM495011; US10994015, Example 307; 2-(7-((4-(3-(4-(4-(2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindolin-5-yl)piperazin-1-yl)piperidin-1-yl)propoxy)butyl)amino)-1-oxoisoindolin-2-yl)-2-(5-fluoro-2-hydroxyphenyl)-N-(thiazol-2-yl)acetamide	O=C1CCC(N2C(=O)c3ccc(N4CCN(C5CCN(CCCOCCCCNc6cccc7c6C(=O)N(C(C(=O)Nc6nccs6)c6cc(F)ccc6O)C7)CC5)CC4)cc3C2=O)C(=O)N1	C48H54FN9O8S	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-MKCKZM	WO2018119441A1_308	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCCNCC2CN(c3nn(C(C)C)c4cc(Nc5ccnc(-c6cnn(S(=O)(=O)C7CC7)c6)n5)ncc34)C2)C(C)(C)C)cc1	C52H68N14O8S2	EGFR	P00533	VHL	WO-2018119441-A1
TPD-2MXH3D	BDBM495013	US10994015, Example 309; US10994015, Example 309	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CN2CCN(CCOCCOCCOCCOCC#Cc3cccc4c3C(=O)N(C(C(=O)Nc3nccs3)c3cc(F)ccc3O)C4)CC2)C(C)(C)C)cc1	C59H72FN9O11S2	EGFR	P00533	VHL	WO-2018119441-A1
TPD-2LCNG6	BDBM495014	US10994015, Example 310; US10994015, Example 310	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCN2CCN(CCOCC#Cc3cccc4c3C(=O)N(C(C(=O)Nc3nccs3)c3cc(F)ccc3O)C4)CC2)C(C)(C)C)cc1	C59H72FN9O11S2	EGFR	P00533	VHL	WO-2018119441-A1
TPD-PTF9Y0	BDBM495015	US10994015, Example 311; US10994015, Example 311	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCN2CCN(CCOCCOCCOCC#Cc3cccc4c3C(=O)N(C(C(=O)Nc3nccs3)c3cc(F)ccc3O)C4)CC2)C(C)(C)C)cc1	C59H72FN9O11S2	EGFR	P00533	VHL	WO-2018119441-A1
TPD-MGPFI1	WO2018119441A1_312	.	CC(C)N1NC(N2CCN(CC3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)c2cnc(Nc3ccnc(-c4cnn(S(=O)(=O)C5CC5)c4)n3)cc21	C42H49N13O6S	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-OS2K7L	SCHEMBL23314123	US10994015, Example 313; BDBM495017; US10994015, Example 313; US10994015, Example 314	CC(C)n1nc(N2CC(CN3CCN(CC4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)C2)c2cnc(Nc3ccnc(-c4cnn(S(=O)(=O)C5CC5)c4)n3)cc21	C46H54N14O6S	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-GHC1DZ	WO2018119441A1_315	.	CCC(C)S(=O)(=O)n1cc(-c2nccc(Nc3cc4c(cn3)c(N3CCC(O)(CN5CCN(CCCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)NCc6ccc(-c7scnc7C)cc6)C(C)(C)C)CC5)CC3)nn4C(C)C)n2)cn1	C56H77N15O7S2	EGFR	P00533	VHL	WO-2018119441-A1
TPD-Q6YW64	WO2018119441A1_316	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCN2CCC(O)(CN3CCN(c4nn(C(C)C)c5cc(Nc6ccnc(-c7cnn(S(=O)(=O)C8CC8)c7)n6)ncc45)CC3)CC2)C(C)(C)C)cc1	C55H73N15O7S2	EGFR	P00533	VHL	WO-2018119441-A1
TPD-17B9F9	WO2018119441A1_317	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCc2ccc(CCC3CCN(c4nn(C(C)C)c5cc(Nc6ccnc(-c7cnn(S(=O)(=O)C8C=C8)c7)n6)ncc45)CC3)cc2)C(C)(C)C)cc1	C57H67N13O7S2	EGFR	P00533	VHL	WO-2018119441-A1
TPD-WV6CJG	SCHEMBL23314125	5-[4-[2-[3-[[1-[6-[[2-(1-Cyclopropylsulfonylpyrazol-4-yl)pyrimidin-4-yl]amino]-1-propan-2-ylpyrazolo[4,3-c]pyridin-3-yl]azetidin-3-yl]methylamino]propoxy]ethyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CC(C)n1nc(N2CC(CNCCCOCCN3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)C2)c2cnc(Nc3ccnc(-c4cnn(S(=O)(=O)C5CC5)c4)n3)cc21	C45H54N14O7S	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-MYBKUH	SCHEMBL23314124	US10994015, Example 319; BDBM495019; US10994015, Example 319	CC(C)n1nc(N2CC(CN[C@H]3C[C@H](Oc4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)C2)c2cnc(Nc3ccnc(-c4cnn(S(=O)(=O)C5CC5)c4)n3)cc21	C40H42N12O7S	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-JRX8HA	SCHEMBL20305721	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[2-[2-[[5-[4-[3-chloro-4-[(3-fluorophenyl)methoxy]anilino]quinazolin-6-yl]furan-2-yl]methoxy]ethoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCOCCOCc2ccc(-c3ccc4ncnc(Nc5ccc(OCc6cccc(F)c6)c(Cl)c5)c4c3)o2)C(C)(C)C)cc1	C58H65ClFN7O11S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-U9ZA7C	WO2018119441A1_321	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCc2ccc(-c3ccc4ncnc(Nc5ccc(OCc6cccc(F)c6)c(Cl)c5)c4c3)o2)C(C)(C)C)cc1	C54H57ClFN7O9S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-3VRB14	WO2018119441A1_322	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCOCCOc2ccc(-c3ccc4ncnc(Nc5ccc(OCc6cccc(F)c6)c(Cl)c5)c4c3)cc2)C(C)(C)C)cc1	C59H65ClFN7O10S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-723H5B	WO2018119441A1_323	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOc2ccc(-c3ccc4ncnc(Nc5ccc(OCc6cccc(F)c6)c(Cl)c5)c4c3)cc2)C(C)(C)C)cc1	C53H53ClFN7O7S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-9AFD1M	WO2018119441A1_324	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCOCCCCCCOCc2ccc(-c3ccc4ncnc(Nc5ccc(OCc6cccc(F)c6)c(Cl)c5)c4c3)o2)C(C)(C)C)cc1	C62H73ClFN7O11S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-0BFMII	WO2018119441A1_325	.	Cc1ncsc1-c1ccc(CN=NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCOCCOCCCCCNCc2ccc(-c3ccc4ncnc(Nc5ccc(OCc6cccc(F)c6)c(Cl)c5)c4c3)o2)C(C)(C)C)cc1	C58H65ClFN9O8S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-EITYNI	WO2018119441A1_326	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCOCCNCc2ccc(-c3ccc4ncnc(Nc5ccc(OCc6cccc(F)c6)c(Cl)c5)c4c3)o2)C(C)(C)C)cc1	C58H66ClFN8O10S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-Y0K6IN	WO2018119441A1_328	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCCCCCNCc2ccc(-c3ccc4ncnc(Nc5ccc(OCc6cccc(F)c6)c(Cl)c5)c4c3)o2)C(C)(C)C)cc1	C60H70ClFN8O9S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-X3FAZV	WO2018119441A1_329	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCOCCCCCCNCc2ccc(-c3ccc4ncnc(N=Nc5ccc(OCc6cccc(F)c6)c(Cl)c5)c4c3)o2)C(C)(C)C)cc1	C62H73ClFN9O10S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-BN7R00	WO2018119441A1_330	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCOCCOCCOCCCCCCNCc2ccc(-c3ccc4ncnc(Nc5ccc(OCc6cccc(F)c6)c(Cl)c5)c4c3)o2)C(C)(C)C)cc1	C63H76ClFN8O9S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-PPQJ2R	WO2018119441A1_331	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCOCCOCCOCCCCCCNCc2ccc(-c3ccc4ncnc(Nc5ccc(OCc6cccc(F)c6)c(Cl)c5)c4c3)o2)C(C)(C)C)cc1	C64H78ClFN8O9S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-8FVTCB	WO2018119441A1_332	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCOCCOCCCCCCNCc2ccc(-c3ccc4ncnc(Nc5ccc(OCc6cccc(F)c6)c(Cl)c5)c4c3)o2)C(C)(C)C)cc1	C62H74ClFN8O8S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-KK9W61	WO2018119441A1_333	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCOCCOCCOCCOCCCCCCNCc2ccc(-c3ccc4ncnc(Nc5ccc(OCc6cccc(F)c6)c(Cl)c5)c4c3)o2)C(C)(C)C)cc1	C66H82ClFN8O10S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-R9ZP7Y	WO2018119441A1_334	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCOCCOCCCCCCNCc2ccc(-c3ccc4ncnc(Nc5ccc(OCc6cccc(F)c6)c(Cl)c5)c4c3)o2)C(C)(C)C)cc1	C64H78ClFN8O11S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-J3I2H5	WO2018119441A1_335	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCOCCOCCOCCOCCOCCCCCCNCc2ccc(-c3ccc4ncnc(Nc5ccc(OCc6cccc(F)c6)c(Cl)c5)c4c3)o2)C(C)(C)C)cc1	C68H86ClFN8O11S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-4HNZDV	WO2018119441A1_336	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCOCCCCCCNCc2ccc(-c3ccc4ncnc(Nc5ccc(OCc6cccc(F)c6)c(Cl)c5)c4c3)o2)C(C)(C)C)cc1	C60H70ClFN8O7S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-YFWVPC	WO2018119441A1_337	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCOCc2ccc(-c3ccc4ncnc(Nc5ccc(OCc6cccc(F)c6)c(Cl)c5)c4c3)o2)C(C)(C)C)cc1	C56H61ClFN7O10S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-999IXQ	WO2018119441A1_338	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)C(NC(=O)CCCCCOCCCOCCCCCCNCc2ccc(-c3ccc4ncnc(Nc5ccc(OCc6cccc(F)c6)c(CI)c5)c4c3)o2)C(C)(C)C)cc1	C64H78FIN8O8S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-DAF3PD	WO2018119441A1_339	.	Cc1ncsc1-c1ccc(CNC(O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCOCCCCCOCCCCCCNCc2ccc(-c3ccc4ncnc(Nc5ccc(OCc6cccc(F)c6)c(Cl)c5)c4c3)o2)C(C)(C)C)cc1	C65H82ClFN8O8S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-4D1B62	WO2018119441A1_340	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCOCCOc2ccc(-c3ccc4ncnc(Nc5ccc(OCc6cccc(F)c6)c(Cl)c5)c4c3)cc2)C(C)(C)C)cc1	C54H55ClFN7O7S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-W3EK16	WO2018119441A1_341	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCOCCOCCNCc2ccc(-c3ccc4ncnc(Nc5ccc(OCc6cccc(F)c6)c(Cl)c5)c4c3)o2)C(C)(C)C)cc1	C55H60ClFN8O8S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-WIMI4Z	WO2018119441A1_342	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCOCCCNCc2ccc(-c3ccc4ncnc(Nc5ccc(OCc6cccc(F)c6)c(Cl)c5)c4c3)o2)C(C)(C)C)cc1	C54H58ClFN8O7S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-BBQ458	WO2018119441A1_343	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCCCOCCCCNCc2ccc(-c3ccc4ncnc(Nc5ccc(OCc6cccc(F)c6)c(Cl)c5)c4c3)o2)C(C)(C)C)cc1	C58H66ClFN8O8S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-4A9FP0	WO2018119441A1_344	.	O=C(COCCCCOCCCCNCc1ccc(-c2ccc3ncnc(Nc4ccc(OCc5cccc(F)c5)c(Cl)c4)c3c2)o1)NCCOc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O	C51H51ClFN7O10	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-3MWAEB	WO2018119441A1_345	.	O=C(CCCCCOCCCCCCOCCCCCCNCc1ccc(-c2ccc3ncnc(Nc4ccc(OCc5cccc(F)c5)c(Cl)c4)c3c2)o1)NCCOc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O	C59H67ClFN7O10	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-FXUNWR	WO2018119441A1_346	.	O=C(CCCCCOCCOCCCCCCNCc1ccc(-c2ccc3ncnc(Nc4ccc(OCc5cccc(F)c5)c(Cl)c4)c3c2)o1)NCCOc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O	C55H59ClFN7O10	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-M854WR	WO2018119441A1_347	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCOCCCCCCOCCCCCCNCc2ccc(-c3ccc4ncnc(Nc5ccc(OCc6cccc(F)c6)c(Cl)c5)c4c3)o2)C(C)(C)C)cc1	C66H82ClFN8O8S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-0O0WHY	WO2018119441A1_348	.	O=C(COCCOCCOCCOCc1ccc(-c2ccc3ncnc(Nc4ccc(OCc5cccc(F)c5)c(Cl)c4)c3c2)o1)NCCOc1cccc2c1C(=O)C(C1CCC(=O)NC1=O)C2=O	C50H47ClFN5O12	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-AUV0X1	SCHEMBL20305536	2-[2-[2-[2-[2-[[5-[4-[3-chloro-4-[(3-fluorophenyl)methoxy]anilino]quinazolin-6-yl]furan-2-yl]methoxy]ethoxy]ethoxy]ethoxy]ethoxy]-N-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyethyl]acetamide	O=C(COCCOCCOCCOCCOCc1ccc(-c2ccc3ncnc(Nc4ccc(OCc5cccc(F)c5)c(Cl)c4)c3c2)o1)NCCOc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O	C51H50ClFN6O13	EGFR	P00533	CRBN	WO-2018119441-A1
TPD-GKTDG2	WO2018119441A1_350	.	COc1cc2c(Cc3ccc(NC(=O)C4(C(=O)Nc5ccc(F)cc5)CC4)cc3F)ccnc2cc1OCCCCCCCCCCC(=O)C[C@H](C(=O)C1C[C@@H](O)C[C@H]1C(=O)NCc1ccc(-c2ocnc2C)cc1)C(C)(C)C	C63H73F2N5O9	EGFR	P00533	VHL	WO-2018119441-A1
TPD-0DN9O5	WO2018119441A1_351	.	COC1=Cc2c(cccc2Oc2ccc(NC(=O)C3(C(=O)Nc4ccc(F)cc4)CC3)cc2F)CC1OCCCCCCCCCCC(=O)N[C@H](C(=O)C1C[C@H](O)C[C@H]1C(=O)NCc1ccc(-c2scnc2C)cc1)C(C)(C)C	C62H73F2N5O9S	EGFR	P00533	VHL	WO-2018119441-A1
TPD-C3UKFJ	SCHEMBL20323888	(2S,4R)-4-hydroxy-1-[(2S)-2-[[2-[2-[2-[2-[2-[4-[(1E)-1-hydroxyimino-2,3-dihydroinden-5-yl]-3-pyridin-4-ylpyrazol-1-yl]ethoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCOCCn2cc(-c3ccc4c(c3)CC/C4=N\O)c(-c3ccncc3)n2)C(C)(C)C)cc1	C49H60N8O9S	BRAF	P15056	VHL	WO-2018119448-A1
TPD-JLS9U5	SCHEMBL20325367	2-(2,6-dioxopiperidin-3-yl)-4-[2-[2-[2-[2-[4-[(1Z)-1-hydroxyimino-2,3-dihydroinden-5-yl]-3-pyridin-4-ylpyrazol-1-yl]ethoxy]ethoxy]ethoxy]ethylamino]isoindole-1,3-dione	O=C1CCC(N2C(=O)c3cccc(NCCOCCOCCOCCn4cc(-c5ccc6c(c5)CC/C6=N/O)c(-c5ccncc5)n4)c3C2=O)C(=O)N1	C38H39N7O8	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-B4792I	SCHEMBL20323741	(2S,4R)-1-[(2S)-3,3-dimethyl-2-[[2-[2-[2-[2-[2-[4-(1-oxo-2,3-dihydroinden-5-yl)-3-pyridin-4-ylpyrazol-1-yl]ethoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]butanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCOCCn2cc(-c3ccc4c(c3)CCC4=O)c(-c3ccncc3)n2)C(C)(C)C)cc1	C49H59N7O9S	BRAF	P15056	VHL	WO-2018119448-A1
TPD-ST72GV	SCHEMBL20323744	3-[7-[2-[2-[2-[2-[4-[(1E)-1-hydroxyimino-2,3-dihydroinden-5-yl]-3-pyridin-4-ylpyrazol-1-yl]ethoxy]ethoxy]ethoxy]ethylamino]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2Cc3c(NCCOCCOCCOCCn4cc(-c5ccc6c(c5)CC/C6=N\O)c(-c5ccncc5)n4)cccc3C2=O)C(=O)N1	C38H41N7O7	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-665RCW	SCHEMBL20325196	(2S,4R)-4-hydroxy-N-[[2-[2-[2-[3-[4-[(1E)-1-hydroxyimino-2,3-dihydroinden-5-yl]-3-pyridin-4-ylpyrazol-1-yl]propoxy]ethoxy]ethoxy]-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](C(C)C)N2Cc3ccccc3C2=O)c(OCCOCCOCCCn2cc(-c3ccc4c(c3)CC/C4=N\O)c(-c3ccncc3)n2)c1	C53H58N8O8S	BRAF	P15056	VHL	WO-2018119448-A1
TPD-ULUDJ9	SCHEMBL22266415	(2S,4R)-4-hydroxy-1-[(2S)-2-[[2-[2-[3-[4-[(1E)-1-hydroxyimino-2,3-dihydroinden-5-yl]-3-pyridin-4-ylpyrazol-1-yl]propoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCCn2cc(-c3ccc4c(c3)CC/C4=N\O)c(-c3ccncc3)n2)C(C)(C)C)cc1	C46H54N8O7S	BRAF	P15056	VHL	WO-2018119448-A1
TPD-YEADPE	SCHEMBL20324185	(2S,4R)-4-hydroxy-1-[(2S)-2-[[2-[2-[2-[3-[4-[(1E)-1-hydroxyimino-2,3-dihydroinden-5-yl]-3-pyridin-4-ylpyrazol-1-yl]propoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCCn2cc(-c3ccc4c(c3)CC/C4=N\O)c(-c3ccncc3)n2)C(C)(C)C)cc1	C48H58N8O8S	BRAF	P15056	VHL	WO-2018119448-A1
TPD-EVUJOH	SCHEMBL20324186	(2S,4R)-4-hydroxy-1-[(2S)-2-[[2-[2-[2-[2-[2-[3-[4-[(1E)-1-hydroxyimino-2,3-dihydroinden-5-yl]-3-pyridin-4-ylpyrazol-1-yl]propoxy]ethoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCOCCOCCCn2cc(-c3ccc4c(c3)CC/C4=N\O)c(-c3ccncc3)n2)C(C)(C)C)cc1	C52H66N8O10S	BRAF	P15056	VHL	WO-2018119448-A1
TPD-TM1ALQ	SCHEMBL20324180	(2S,4R)-4-hydroxy-1-[(2S)-2-[[2-[2-[2-[2-[2-[2-[3-[4-[(1E)-1-hydroxyimino-2,3-dihydroinden-5-yl]-3-pyridin-4-ylpyrazol-1-yl]propoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCOCCOCCOCCCn2cc(-c3ccc4c(c3)CC/C4=N\O)c(-c3ccncc3)n2)C(C)(C)C)cc1	C54H70N8O11S	BRAF	P15056	VHL	WO-2018119448-A1
TPD-MEF8UV	SCHEMBL20324181	(2S,4R)-4-hydroxy-1-[(2S)-2-[[2-[2-[2-[2-[2-[2-[3-[4-[(1E)-1-hydroxyimino-2,3-dihydroinden-5-yl]-5-pyridin-4-ylpyrazol-1-yl]propoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCOCCOCCOCCCn2ncc(-c3ccc4c(c3)CC/C4=N\O)c2-c2ccncc2)C(C)(C)C)cc1	C54H70N8O11S	BRAF	P15056	VHL	WO-2018119448-A1
TPD-22XHSM	SCHEMBL20326124	(2S,4R)-4-hydroxy-N-[[2-[2-[3-[4-[(1E)-1-hydroxyimino-2,3-dihydroinden-5-yl]-3-pyridin-4-ylpyrazol-1-yl]propoxy]ethoxy]-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](C(C)C)N2Cc3ccccc3C2=O)c(OCCOCCCn2cc(-c3ccc4c(c3)CC/C4=N\O)c(-c3ccncc3)n2)c1	C51H54N8O7S	BRAF	P15056	VHL	WO-2018119448-A1
TPD-NXULO4	SCHEMBL22266405	(2S,4R)-4-hydroxy-N-[[2-[2-[2-[2-[3-[4-[(1E)-1-hydroxyimino-2,3-dihydroinden-5-yl]-3-pyridin-4-ylpyrazol-1-yl]propoxy]ethoxy]ethoxy]ethoxy]-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](C(C)C)N2Cc3ccccc3C2=O)c(OCCOCCOCCOCCCn2cc(-c3ccc4c(c3)CC/C4=N\O)c(-c3ccncc3)n2)c1	C55H62N8O9S	BRAF	P15056	VHL	WO-2018119448-A1
TPD-CNZ049	SCHEMBL20323793	(2S,4R)-4-hydroxy-N-[[2-[2-[2-[2-[2-[3-[4-[(1E)-1-hydroxyimino-2,3-dihydroinden-5-yl]-3-pyridin-4-ylpyrazol-1-yl]propoxy]ethoxy]ethoxy]ethoxy]ethoxy]-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](C(C)C)N2Cc3ccccc3C2=O)c(OCCOCCOCCOCCOCCCn2cc(-c3ccc4c(c3)CC/C4=N\O)c(-c3ccncc3)n2)c1	C57H66N8O10S	BRAF	P15056	VHL	WO-2018119448-A1
TPD-6ZWXPH	SCHEMBL20323795	(2S,4R)-4-hydroxy-N-[[2-[2-[2-[2-[2-[2-[3-[4-[(1E)-1-hydroxyimino-2,3-dihydroinden-5-yl]-3-pyridin-4-ylpyrazol-1-yl]propoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](C(C)C)N2Cc3ccccc3C2=O)c(OCCOCCOCCOCCOCCOCCCn2cc(-c3ccc4c(c3)CC/C4=N\O)c(-c3ccncc3)n2)c1	C59H70N8O11S	BRAF	P15056	VHL	WO-2018119448-A1
TPD-ECUR0R	SCHEMBL20323792	2-(2,6-dioxopiperidin-3-yl)-4-[2-[2-[3-[4-[(1E)-1-hydroxyimino-2,3-dihydroinden-5-yl]-3-pyridin-4-ylpyrazol-1-yl]propoxy]ethoxy]ethylamino]isoindole-1,3-dione	O=C1CCC(N2C(=O)c3cccc(NCCOCCOCCCn4cc(-c5ccc6c(c5)CC/C6=N\O)c(-c5ccncc5)n4)c3C2=O)C(=O)N1	C37H37N7O7	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-KC27HA	SCHEMBL20323790	2-(2,6-dioxopiperidin-3-yl)-4-[2-[2-[2-[3-[4-[(1E)-1-hydroxyimino-2,3-dihydroinden-5-yl]-3-pyridin-4-ylpyrazol-1-yl]propoxy]ethoxy]ethoxy]ethylamino]isoindole-1,3-dione	O=C1CCC(N2C(=O)c3cccc(NCCOCCOCCOCCCn4cc(-c5ccc6c(c5)CC/C6=N\O)c(-c5ccncc5)n4)c3C2=O)C(=O)N1	C39H41N7O8	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-5B3DC6	WO2018119448A1_24	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCOCCCN2C=C(c3ccc4c(c3)CC/C4=N\O)C(c3ccncc3)N2)C(C)(C)C)cc1	C50H64N8O9S	BRAF	P15056	VHL	WO-2018119448-A1
TPD-1NR78L	SCHEMBL20323791	(2S,4R)-4-hydroxy-1-[(2S)-2-[[2-[2-[2-[2-[3-[4-[(1E)-1-hydroxyimino-2,3-dihydroinden-5-yl]-3-pyridin-4-ylpyrazol-1-yl]propoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCOCCCn2cc(-c3ccc4c(c3)CC/C4=N\O)c(-c3ccncc3)n2)C(C)(C)C)cc1	C50H62N8O9S	BRAF	P15056	VHL	WO-2018119448-A1
TPD-TUSSE0	WO2018119448A1_26	.	Cc1ncsc1-c1ccc(CNC(O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](C(C)C)N2Cc3ccccc3C2=O)c(OCCOCCOCCOCCCn2ncc(-c3ccc4c(c3)CC/C4=N\O)c2-c2ccncc2)c1	C55H64N8O9S	BRAF	P15056	VHL	WO-2018119448-A1
TPD-JKB843	SCHEMBL20323811	3-[7-[2-[2-[2-[2-[4-[(1E)-1-hydroxyimino-2,3-dihydroinden-5-yl]-3-pyridin-4-ylpyrazol-1-yl]ethoxy]ethoxy]ethoxy]ethoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2Cc3c(OCCOCCOCCOCCn4cc(-c5ccc6c(c5)CC/C6=N\O)c(-c5ccncc5)n4)cccc3C2=O)C(=O)N1	C38H40N6O8	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-C4UQE4	SCHEMBL20325376	2-(2,6-dioxopiperidin-3-yl)-4-[2-[3-[4-[(1E)-1-hydroxyimino-2,3-dihydroinden-5-yl]-3-pyridin-4-ylpyrazol-1-yl]propoxy]ethylamino]isoindole-1,3-dione	O=C1CCC(N2C(=O)c3cccc(NCCOCCCn4cc(-c5ccc6c(c5)CC/C6=N\O)c(-c5ccncc5)n4)c3C2=O)C(=O)N1	C35H33N7O6	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-3BO1B4	WO2018119448A1_31	.	O=C1CCC(N2C(=O)c3cccc(NCCOCCOCCOCCOCCCN4C=C(c5ccc6c(c5)CC/C6=N\O)C(c5ccncc5)N4)c3C2=O)C(=O)N1	C41H47N7O9	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-9140GC	SCHEMBL20324187	2-(2,6-dioxopiperidin-3-yl)-4-[2-[2-[2-[2-[3-[4-[(1E)-1-hydroxyimino-2,3-dihydroinden-5-yl]-3-pyridin-4-ylpyrazol-1-yl]propoxy]ethoxy]ethoxy]ethoxy]ethylamino]isoindole-1,3-dione	O=C1CCC(N2C(=O)c3cccc(NCCOCCOCCOCCOCCCn4cc(-c5ccc6c(c5)CC/C6=N\O)c(-c5ccncc5)n4)c3C2=O)C(=O)N1	C41H45N7O9	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-GNOCU0	SCHEMBL20324182	2-(2,6-dioxopiperidin-3-yl)-4-[2-[2-[2-[2-[2-[3-[4-[(1E)-1-hydroxyimino-2,3-dihydroinden-5-yl]-3-pyridin-4-ylpyrazol-1-yl]propoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethylamino]isoindole-1,3-dione	O=C1CCC(N2C(=O)c3cccc(NCCOCCOCCOCCOCCOCCCn4cc(-c5ccc6c(c5)CC/C6=N\O)c(-c5ccncc5)n4)c3C2=O)C(=O)N1	C43H49N7O10	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-IY2VY7	SCHEMBL20324183	2-(2,6-dioxopiperidin-3-yl)-4-[2-[2-[2-[4-[4-[(1E)-1-hydroxyimino-2,3-dihydroinden-5-yl]-3-pyridin-4-ylpyrazol-1-yl]phenoxy]ethoxy]ethoxy]ethoxy]isoindole-1,3-dione	O=C1CCC(N2C(=O)c3cccc(OCCOCCOCCOc4ccc(-n5cc(-c6ccc7c(c6)CC/C7=N\O)c(-c6ccncc6)n5)cc4)c3C2=O)C(=O)N1	C42H38N6O9	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-GOO7PT	SCHEMBL20323798	2-(2,6-dioxopiperidin-3-yl)-4-[2-[4-[4-[(1E)-1-hydroxyimino-2,3-dihydroinden-5-yl]-3-pyridin-4-ylpyrazol-1-yl]phenoxy]ethoxy]isoindole-1,3-dione	O=C1CCC(N2C(=O)c3cccc(OCCOc4ccc(-n5cc(-c6ccc7c(c6)CC/C7=N\O)c(-c6ccncc6)n5)cc4)c3C2=O)C(=O)N1	C38H30N6O7	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-4O0URX	WO2018119448A1_39	.	O=C1CCC(N2C(=O)c3cccc(OCCOCCOc4ccc(-n5cc(-c6ccc7c(c6)CC/C7=N\O)c(-c6ccncc6)n5)cc4)c3C2=O)C(=O)N1	C40H34N6O8	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-DTVDA8	SCHEMBL20323799	2-(2,6-dioxopiperidin-3-yl)-4-[2-[2-[2-[2-[2-[2-[3-[4-[(1E)-1-hydroxyimino-2,3-dihydroinden-5-yl]-3-pyridin-4-ylpyrazol-1-yl]propoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethylamino]isoindole-1,3-dione	O=C1CCC(N2C(=O)c3cccc(NCCOCCOCCOCCOCCOCCOCCCn4cc(-c5ccc6c(c5)CC/C6=N\O)c(-c5ccncc5)n4)c3C2=O)C(=O)N1	C45H53N7O11	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-VU4KYW	SCHEMBL22266397	(2S,4R)-N-[[2-[2-[2-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenoxy]ethoxy]ethoxy]-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-4-hydroxy-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](C(C)C)N2Cc3ccccc3C2=O)c(OCCOCCOc2ccc(-c3cnc4[nH]cc(C(=O)c5c(F)ccc(NS(=O)(=O)N6CC[C@@H](F)C6)c5F)c4c3)cc2)c1	C57H57F3N8O10S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-GNVDXL	SCHEMBL22266376	2-(2,6-dioxopiperidin-3-yl)-5-[2-[4-[4-[(1E)-1-hydroxyimino-2,3-dihydroinden-5-yl]-3-pyridin-4-ylpyrazol-1-yl]phenoxy]ethoxy]isoindole-1,3-dione	O=C1CCC(N2C(=O)c3ccc(OCCOc4ccc(-n5cc(-c6ccc7c(c6)CC/C7=N\O)c(-c6ccncc6)n5)cc4)cc3C2=O)C(=O)N1	C38H30N6O7	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-RCDKEH	SCHEMBL20323883	2-(2,6-dioxopiperidin-3-yl)-5-[2-[2-[2-[4-[4-[(1E)-1-hydroxyimino-2,3-dihydroinden-5-yl]-3-pyridin-4-ylpyrazol-1-yl]phenoxy]ethoxy]ethoxy]ethoxy]isoindole-1,3-dione	O=C1CCC(N2C(=O)c3ccc(OCCOCCOCCOc4ccc(-n5cc(-c6ccc7c(c6)CC/C7=N\O)c(-c6ccncc6)n5)cc4)cc3C2=O)C(=O)N1	C42H38N6O9	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-6IM03U	SCHEMBL20323885	2-(2,6-dioxopiperidin-3-yl)-4-[2-[2-[2-[2-[4-[4-[(1E)-1-hydroxyimino-2,3-dihydroinden-5-yl]-3-pyridin-4-ylpyrazol-1-yl]phenoxy]ethoxy]ethoxy]ethoxy]ethoxy]isoindole-1,3-dione	O=C1CCC(N2C(=O)c3cccc(OCCOCCOCCOCCOc4ccc(-n5cc(-c6ccc7c(c6)CC/C7=N\O)c(-c6ccncc6)n5)cc4)c3C2=O)C(=O)N1	C44H42N6O10	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-UDNOFS	SCHEMBL20323884	2-(2,6-dioxopiperidin-3-yl)-4-[2-[2-[2-[2-[2-[4-[4-[(1E)-1-hydroxyimino-2,3-dihydroinden-5-yl]-3-pyridin-4-ylpyrazol-1-yl]phenoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]isoindole-1,3-dione	O=C1CCC(N2C(=O)c3cccc(OCCOCCOCCOCCOCCOc4ccc(-n5cc(-c6ccc7c(c6)CC/C7=N\O)c(-c6ccncc6)n5)cc4)c3C2=O)C(=O)N1	C46H46N6O11	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-I8LKA4	SCHEMBL20323886	(2S,4R)-N-[[2-[2-[2-[2-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenoxy]ethoxy]ethoxy]ethoxy]-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-4-hydroxy-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](C(C)C)N2Cc3ccccc3C2=O)c(OCCOCCOCCOc2ccc(-c3cnc4[nH]cc(C(=O)c5c(F)ccc(NS(=O)(=O)N6CC[C@@H](F)C6)c5F)c4c3)cc2)c1	C59H61F3N8O11S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-QD1L2G	SCHEMBL22266414	(2S,4R)-N-[[2-[2-[2-[2-[2-[2-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-4-hydroxy-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](C(C)C)N2Cc3ccccc3C2=O)c(OCCOCCOCCOCCOCCOc2ccc(-c3cnc4[nH]cc(C(=O)c5c(F)ccc(NS(=O)(=O)N6CC[C@@H](F)C6)c5F)c4c3)cc2)c1	C63H69F3N8O13S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-4BRLNX	WO2018119448A1_49	.	Cc1ncsc1-c1ccc(CNC(=O)C2C[C@@H](O)CN2C(=O)[C@H](C(C)C)N2Cc3ccccc3C2=O)c(OCCOCCOCCOCCOCCOCCOc2ccc(-c3cnc4[nH]cc(C(=O)c5c(F)ccc(NS(=O)(=O)N6CC[C@@H](F)C6)c5F)c4c3)cc2)c1	C65H73F3N8O14S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-VH5AL2	SCHEMBL20323854	2-(2,6-dioxopiperidin-3-yl)-5-[2-[2-[4-[4-[(1E)-1-hydroxyimino-2,3-dihydroinden-5-yl]-3-pyridin-4-ylpyrazol-1-yl]phenoxy]ethoxy]ethoxy]isoindole-1,3-dione	O=C1CCC(N2C(=O)c3ccc(OCCOCCOc4ccc(-n5cc(-c6ccc7c(c6)CC/C7=N\O)c(-c6ccncc6)n5)cc4)cc3C2=O)C(=O)N1	C40H34N6O8	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-PP3VBR	WO2018119448A1_51	.	O=C1CCC(N2C(=O)c3cccc(OCCOCCOCCOCCOCCOc4ccc(-n5cc(-c6ccc7c(c6)CCC7NO)c(-c6ccncc6)n5)cc4)c3C2=O)C(=O)N1	C46H48N6O11	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-GTOSAN	SCHEMBL20323850	(3R)-N-[3-[5-[4-[2-[2-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2C(=O)c3cccc(OCCOCCOCCOCCOc4ccc(-c5cnc6[nH]cc(C(=O)c7c(F)ccc(NS(=O)(=O)N8CC[C@@H](F)C8)c7F)c6c5)cc4)c3C2=O)C(=O)N1	C45H43F3N6O12S	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-23NDHO	WO2018119448A1_53	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)C(C(C)C)N2Cc3ccccc3C2=O)c(OCCOCCOCCOCCOc2ccc(-c3cnc4[nH]cc(C(=O)c5c(F)ccc(NS(=O)(=O)N6CC[C@@H](F)C6)c5F)c4c3)cc2)c1	C61H65F3N8O12S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-698ULC	SCHEMBL20326106	2-(2,6-dioxopiperidin-3-yl)-5-[2-[2-[2-[2-[4-[4-[(1E)-1-hydroxyimino-2,3-dihydroinden-5-yl]-3-pyridin-4-ylpyrazol-1-yl]phenoxy]ethoxy]ethoxy]ethoxy]ethoxy]isoindole-1,3-dione	O=C1CCC(N2C(=O)c3ccc(OCCOCCOCCOCCOc4ccc(-n5cc(-c6ccc7c(c6)CC/C7=N\O)c(-c6ccncc6)n5)cc4)cc3C2=O)C(=O)N1	C44H42N6O10	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-0AX3HB	SCHEMBL20323876	2-(2,6-dioxopiperidin-3-yl)-5-[2-[2-[2-[2-[2-[4-[4-[(1E)-1-hydroxyimino-2,3-dihydroinden-5-yl]-3-pyridin-4-ylpyrazol-1-yl]phenoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]isoindole-1,3-dione	O=C1CCC(N2C(=O)c3ccc(OCCOCCOCCOCCOCCOc4ccc(-n5cc(-c6ccc7c(c6)CC/C7=N\O)c(-c6ccncc6)n5)cc4)cc3C2=O)C(=O)N1	C46H46N6O11	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-ZBKTXG	SCHEMBL20323877	(3R)-N-[3-[5-[4-[2-[2-[2-[2-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2C(=O)c3cccc(OCCOCCOCCOCCOCCOCCOc4ccc(-c5cnc6[nH]cc(C(=O)c7c(F)ccc(NS(=O)(=O)N8CC[C@@H](F)C8)c7F)c6c5)cc4)c3C2=O)C(=O)N1	C49H51F3N6O14S	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-SN3O1Y	SCHEMBL22266410	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOc2ccc(-c3cnc4[nH]cc(C(=O)c5c(F)ccc(NS(=O)(=O)N6CC[C@@H](F)C6)c5F)c4c3)cc2)C(C)(C)C)cc1	C52H57F3N8O10S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-EUC82K	SCHEMBL22266395	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[2-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCOc2ccc(-c3cnc4[nH]cc(C(=O)c5c(F)ccc(NS(=O)(=O)N6CC[C@@H](F)C6)c5F)c4c3)cc2)C(C)(C)C)cc1	C54H61F3N8O11S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-WIULG7	SCHEMBL20323875	2-(2,6-dioxopiperidin-3-yl)-5-[2-[2-[3-[4-[(1E)-1-hydroxyimino-2,3-dihydroinden-5-yl]-3-pyridin-4-ylpyrazol-1-yl]propoxy]ethoxy]ethoxy]isoindole-1,3-dione	O=C1CCC(N2C(=O)c3ccc(OCCOCCOCCCn4cc(-c5ccc6c(c5)CC/C6=N\O)c(-c5ccncc5)n4)cc3C2=O)C(=O)N1	C37H36N6O8	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-40NZEK	SCHEMBL20323868	2-(2,6-dioxopiperidin-3-yl)-5-[2-[2-[2-[2-[3-[4-[(1E)-1-hydroxyimino-2,3-dihydroinden-5-yl]-3-pyridin-4-ylpyrazol-1-yl]propoxy]ethoxy]ethoxy]ethoxy]ethoxy]isoindole-1,3-dione	O=C1CCC(N2C(=O)c3ccc(OCCOCCOCCOCCOCCCn4cc(-c5ccc6c(c5)CC/C6=N\O)c(-c5ccncc5)n4)cc3C2=O)C(=O)N1	C41H44N6O10	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-ZANHO1	SCHEMBL20323869	(3R)-N-[3-[5-[4-[2-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxyethoxy]ethoxy]ethoxy]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2C(=O)c3ccc(OCCOCCOCCOc4ccc(-c5cnc6[nH]cc(C(=O)c7c(F)ccc(NS(=O)(=O)N8CC[C@@H](F)C8)c7F)c6c5)cc4)cc3C2=O)C(=O)N1	C43H39F3N6O11S	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-IGDIXZ	SCHEMBL20323870	(3R)-N-[3-[5-[4-[2-[2-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2C(=O)c3ccc(OCCOCCOCCOCCOc4ccc(-c5cnc6[nH]cc(C(=O)c7c(F)ccc(NS(=O)(=O)N8CC[C@@H](F)C8)c7F)c6c5)cc4)cc3C2=O)C(=O)N1	C45H43F3N6O12S	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-H5WS51	SCHEMBL20323873	(3R)-N-[3-[5-[4-[2-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyethoxy]ethoxy]ethoxy]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2C(=O)c3cccc(OCCOCCOCCOc4ccc(-c5cnc6[nH]cc(C(=O)c7c(F)ccc(NS(=O)(=O)N8CC[C@@H](F)C8)c7F)c6c5)cc4)c3C2=O)C(=O)N1	C43H39F3N6O11S	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-5QJSE9	SCHEMBL20323871	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[2-[2-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenoxy]ethoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCOCCOc2ccc(-c3cnc4[nH]cc(C(=O)c5c(F)ccc(NS(=O)(=O)N6CC[C@@H](F)C6)c5F)c4c3)cc2)C(C)(C)C)cc1	C56H65F3N8O12S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-12WPAM	SCHEMBL20325220	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[2-[2-[2-[2-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCOCCOCCOCCOc2ccc(-c3cnc4[nH]cc(C(=O)c5c(F)ccc(NS(=O)(=O)N6CC[C@@H](F)C6)c5F)c4c3)cc2)C(C)(C)C)cc1	C60H73F3N8O14S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-15T28H	SCHEMBL20324171	2-(2,6-dioxopiperidin-3-yl)-5-[2-[2-[2-[2-[2-[3-[4-[(1E)-1-hydroxyimino-2,3-dihydroinden-5-yl]-3-pyridin-4-ylpyrazol-1-yl]propoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]isoindole-1,3-dione	O=C1CCC(N2C(=O)c3ccc(OCCOCCOCCOCCOCCOCCCn4cc(-c5ccc6c(c5)CC/C6=N\O)c(-c5ccncc5)n4)cc3C2=O)C(=O)N1	C43H48N6O11	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-Y1VE3N	SCHEMBL20324169	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[2-[2-[2-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCOCCOCCOc2ccc(-c3cnc4[nH]cc(C(=O)c5c(F)ccc(NS(=O)(=O)N6CC[C@@H](F)C6)c5F)c4c3)cc2)C(C)(C)C)cc1	C58H69F3N8O13S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-OHO0M8	SCHEMBL20324173	2-(2,6-dioxopiperidin-3-yl)-5-[2-[2-[2-[3-[4-[(1E)-1-hydroxyimino-2,3-dihydroinden-5-yl]-3-pyridin-4-ylpyrazol-1-yl]propoxy]ethoxy]ethoxy]ethoxy]isoindole-1,3-dione	O=C1CCC(N2C(=O)c3ccc(OCCOCCOCCOCCCn4cc(-c5ccc6c(c5)CC/C6=N\O)c(-c5ccncc5)n4)cc3C2=O)C(=O)N1	C39H40N6O9	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-DO7ZCP	SCHEMBL20324174	3-[6-[2-[4-[4-[(1E)-1-hydroxyimino-2,3-dihydroinden-5-yl]-3-pyridin-4-ylpyrazol-1-yl]phenoxy]ethoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2Cc3cc(OCCOc4ccc(-n5cc(-c6ccc7c(c6)CC/C7=N\O)c(-c6ccncc6)n5)cc4)ccc3C2=O)C(=O)N1	C38H32N6O6	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-QPYO5A	SCHEMBL22266471	(3R)-N-[3-[5-[4-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxyethoxy]ethoxy]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2C(=O)c3ccc(OCCOCCOc4ccc(-c5cnc6[nH]cc(C(=O)c7c(F)ccc(NS(=O)(=O)N8CC[C@@H](F)C8)c7F)c6c5)cc4)cc3C2=O)C(=O)N1	C41H35F3N6O10S	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-BJ4PGK	SCHEMBL20324170	(3R)-N-[3-[5-[4-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyethoxy]ethoxy]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2C(=O)c3cccc(OCCOCCOc4ccc(-c5cnc6[nH]cc(C(=O)c7c(F)ccc(NS(=O)(=O)N8CC[C@@H](F)C8)c7F)c6c5)cc4)c3C2=O)C(=O)N1	C41H35F3N6O10S	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-VUMD22	SCHEMBL20323931	3-[6-[2-[2-[4-[4-[(1E)-1-hydroxyimino-2,3-dihydroinden-5-yl]-3-pyridin-4-ylpyrazol-1-yl]phenoxy]ethoxy]ethoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2Cc3cc(OCCOCCOc4ccc(-n5cc(-c6ccc7c(c6)CC/C7=N\O)c(-c6ccncc6)n5)cc4)ccc3C2=O)C(=O)N1	C40H36N6O7	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-9YN2MS	WO2018119448A1_73	.	O=C1CCC(N2Cc3cc(OCCOCCOc4ccc(-n5cc(-c6ccc7c(c6)CCC7NO)c(-c6ccncc6)n5)cc4)ccc3C2=O)C(=O)N1	C40H38N6O7	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-RVHMUN	SCHEMBL20325251	(3R)-N-[3-[5-[4-[2-[2-[2-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]ethoxy]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2C(=O)c3ccc(OCCOCCOCCOCCOCCOc4ccc(-c5cnc6[nH]cc(C(=O)c7c(F)ccc(NS(=O)(=O)N8CC[C@@H](F)C8)c7F)c6c5)cc4)cc3C2=O)C(=O)N1	C47H47F3N6O13S	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-VB07S8	SCHEMBL20323934	3-[6-[2-[2-[2-[4-[4-[(1E)-1-hydroxyimino-2,3-dihydroinden-5-yl]-3-pyridin-4-ylpyrazol-1-yl]phenoxy]ethoxy]ethoxy]ethoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2Cc3cc(OCCOCCOCCOc4ccc(-n5cc(-c6ccc7c(c6)CC/C7=N\O)c(-c6ccncc6)n5)cc4)ccc3C2=O)C(=O)N1	C42H40N6O8	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-90N5R6	SCHEMBL20323936	3-[6-[2-[2-[2-[2-[4-[4-[(1E)-1-hydroxyimino-2,3-dihydroinden-5-yl]-3-pyridin-4-ylpyrazol-1-yl]phenoxy]ethoxy]ethoxy]ethoxy]ethoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2Cc3cc(OCCOCCOCCOCCOc4ccc(-n5cc(-c6ccc7c(c6)CC/C7=N\O)c(-c6ccncc6)n5)cc4)ccc3C2=O)C(=O)N1	C44H44N6O9	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-TZDFZU	SCHEMBL20323932	3-[6-[2-[2-[2-[2-[2-[4-[4-[(1E)-1-hydroxyimino-2,3-dihydroinden-5-yl]-3-pyridin-4-ylpyrazol-1-yl]phenoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2Cc3cc(OCCOCCOCCOCCOCCOc4ccc(-n5cc(-c6ccc7c(c6)CC/C7=N\O)c(-c6ccncc6)n5)cc4)ccc3C2=O)C(=O)N1	C46H48N6O10	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-JO2HSK	SCHEMBL20326165	(3R)-N-[3-[5-[4-[2-[2-[2-[2-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2C(=O)c3ccc(OCCOCCOCCOCCOCCOCCOc4ccc(-c5cnc6[nH]cc(C(=O)c7c(F)ccc(NS(=O)(=O)N8CC[C@@H](F)C8)c7F)c6c5)cc4)cc3C2=O)C(=O)N1	C49H51F3N6O14S	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-NU96TN	SCHEMBL20324204	(3R)-N-[3-[5-[4-[2-[2-[2-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]ethoxy]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2C(=O)c3cccc(OCCOCCOCCOCCOCCOc4ccc(-c5cnc6[nH]cc(C(=O)c7c(F)ccc(NS(=O)(=O)N8CC[C@@H](F)C8)c7F)c6c5)cc4)c3C2=O)C(=O)N1	C47H47F3N6O13S	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-7FCXRF	SCHEMBL20324205	(2S,4R)-1-[(2S)-2-[[2-[3-[3-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenoxy]propoxy]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCCOCCCOc2ccc(-c3cnc4[nH]cc(C(=O)c5c(F)ccc(NS(=O)(=O)N6CC[C@@H](F)C6)c5F)c4c3)cc2)C(C)(C)C)cc1	C54H61F3N8O10S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-BOMRZA	SCHEMBL20324207	2-(2,6-dioxopiperidin-3-yl)-5-[2-[3-[4-[(1E)-1-hydroxyimino-2,3-dihydroinden-5-yl]-3-pyridin-4-ylpyrazol-1-yl]propoxy]ethoxy]isoindole-1,3-dione	O=C1CCC(N2C(=O)c3ccc(OCCOCCCn4cc(-c5ccc6c(c5)CC/C6=N\O)c(-c5ccncc5)n4)cc3C2=O)C(=O)N1	C35H32N6O7	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-DIT1PR	WO2018119448A1_83	.	O=C1CCC(N2C(=O)c3ccc(OCCOCCCN4C=C(c5ccc6c(c5)CCC6NO)C(c5ccncc5)N4)cc3C2=O)C(=O)N1	C35H36N6O7	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-MZ80DS	WO2018119448A1_85	.	Cc1ncsc1-c1ccc(CNC(=O)[C@H]2C[C@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOc2ccc(-c3cnc4[nH]cc(C(=O)c5c(F)ccc(NS(=O)(=O)N6CC[C@@H](C)C6)c5F)c4c3)cc2)C(C)(C)C)cc1	C53H60F2N8O10S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-S42Y31	WO2018119448A1_86	.	O=C1CCC(N2C(=O)c3ccc(OCCOCCN4CCN(c5ccc(-c6cnc7c(c6)C(C(=O)c6c(F)ccc(NS(=O)(=O)N8CC[C@@H](F)C8)c6F)CN7)cc5)CC4)cc3C2=O)C(=O)N1	C45H45F3N8O9S	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-H4WN6T	SCHEMBL24021827	(3R)-N-[3-[5-[4-[4-[2-[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxypropoxy]ethyl]piperazin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2C(=O)c3ccc(OCCCOCCN4CCN(c5ccc(-c6cnc7[nH]cc(C(=O)c8c(F)ccc(NS(=O)(=O)N9CC[C@@H](F)C9)c8F)c7c6)cc5)CC4)cc3C2=O)C(=O)N1	C46H45F3N8O9S	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-H0V9UA	WO2018119448A1_88	.	N[C@@H]1CCN(S(=O)(=O)Nc2ccc(F)c(C(=O)c3c[nH]c4ncc(-c5ccc(N6CCC(CN7CCN(c8ccc9c(c8)C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)CC6)cc5)cc34)c2F)C1	C47H48F2N10O7S	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-MOZKO8	SCHEMBL24021832	(3R)-N-[3-[5-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxybutyl]piperazin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2C(=O)c3ccc(OCCCCN4CCN(c5ccc(-c6cnc7[nH]cc(C(=O)c8c(F)ccc(NS(=O)(=O)N9CC[C@@H](F)C9)c8F)c7c6)cc5)CC4)cc3C2=O)C(=O)N1	C45H43F3N8O8S	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-K6A2SP	SCHEMBL24021830	(3R)-N-[3-[5-[4-[4-[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxypropyl]piperazin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2C(=O)c3ccc(OCCCN4CCN(c5ccc(-c6cnc7[nH]cc(C(=O)c8c(F)ccc(NS(=O)(=O)N9CC[C@@H](F)C9)c8F)c7c6)cc5)CC4)cc3C2=O)C(=O)N1	C44H41F3N8O8S	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-M5RNR8	WO2018119448A1_91	.	O=C1CCC(N2C(=O)C3C=CC(N4CCN(CCOCCOc5ccc(-c6cnc7[nH]cc(C(=O)c8c(F)ccc(NS(=O)(=O)N9CC[C@@H](F)C9)c8F)c7c6)cc5)CC4)=CC3C2=O)C(=O)N1	C45H45F3N8O9S	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-AEFPIW	WO2018119448A1_92	.	O=C1CCC(N2C(=O)c3ccc(N4CCN(CCCCCOc5ccc(-c6cnc7[nH]cc(C(=O)c8c(F)ccc(NS(=O)(=O)N9CC[C@@H](F)C9)c8F)c7c6)cc5)CC4)cc3C2=O)C(=O)N1	C46H45F3N8O8S	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-SL3SNB	SCHEMBL24021870	(3R)-N-[3-[5-[4-[6-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]hexoxy]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2C(=O)c3ccc(N4CCN(CCCCCCOc5ccc(-c6cnc7[nH]cc(C(=O)c8c(F)ccc(NS(=O)(=O)N9CC[C@@H](F)C9)c8F)c7c6)cc5)CC4)cc3C2=O)C(=O)N1	C47H47F3N8O8S	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-C4LODP	WO2018119448A1_94	.	O=C1CCC(N2C(=O)C3C=CC(N4CCN(CCOCCCOc5ccc(-c6cnc7[nH]cc(C(=O)c8c(F)ccc(NS(=O)(=O)N9CC[C@@H](F)C9)c8F)c7c6)cc5)CC4)=CC3C2=O)C(=O)N1	C46H47F3N8O9S	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-P99MHO	SCHEMBL24021786	(3R)-N-[3-[5-[4-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]ethoxy]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2C(=O)c3ccc(N4CCN(CCOc5ccc(-c6cnc7[nH]cc(C(=O)c8c(F)ccc(NS(=O)(=O)N9CC[C@@H](F)C9)c8F)c7c6)cc5)CC4)cc3C2=O)C(=O)N1	C43H39F3N8O8S	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-6URM28	WO2018119448A1_96	.	O=C1CCC(N2C(=O)c3ccc(N4CCN(CCCCOc5ccc(C6=CC7C(C(=O)C8C(F)=CC=C(NS(=O)(=O)N9CC[C@@H](F)C9)C8F)=CNC7N=C6)cc5)CC4)cc3C2=O)C(=O)N1	C45H47F3N8O8S	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-H9PLSO	WO2018119448A1_97	.	O=C1CCC(N2C(=O)c3ccc(N4CCN(CCCOc5ccc(C6=CC7C(C(=O)c8c(F)ccc(NS(=O)(=O)N9CC[C@@H](F)C9)c8F)=CNC7N=C6)cc5)CC4)cc3C2=O)C(=O)N1	C44H43F3N8O8S	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-44A3MS	WO2018119448A1_98	.	CC1=C(c2ccc(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(O)CN3CCN(CCOc4ccc(-c5cnc6[nH]cc(C(=O)c7cc(NS(=O)(=O)N8CC[C@@H](F)C8)ccc7F)c6c5)cc4)CC3)C(C)(C)C)cc2)SCN1	C54H66F2N10O8S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-50E21H	SCHEMBL20294839	(2S,4R)-1-[(2S)-2-[[2-[2-[4-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]piperazin-1-yl]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCN2CCN(c3ccc(-c4cnc5[nH]cc(C(=O)c6c(F)ccc(NS(=O)(=O)N7CC[C@@H](F)C7)c6F)c5c4)cc3)CC2)C(C)(C)C)cc1	C54H61F3N10O8S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-UP2UAB	SCHEMBL20294580	(2S,4R)-1-[(2S)-2-[[2-[3-[4-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]piperazin-1-yl]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCCN2CCN(c3ccc(-c4cnc5[nH]cc(C(=O)c6c(F)ccc(NS(=O)(=O)N7CC[C@@H](F)C7)c6F)c5c4)cc3)CC2)C(C)(C)C)cc1	C55H63F3N10O8S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-D50L9U	SCHEMBL22266547	(2S,4R)-1-[(2S)-2-[[2-[4-[3-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenoxy]propyl]piperazin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CN2CCN(CCCOc3ccc(-c4cnc5[nH]cc(C(=O)c6c(F)ccc(NS(=O)(=O)N7CC[C@@H](F)C7)c6F)c5c4)cc3)CC2)C(C)(C)C)cc1	C55H63F3N10O8S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-GYK956	SCHEMBL22266422	(2S,4R)-1-[(2S)-2-[3-[3-[4-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]piperazin-1-yl]azetidin-1-yl]propanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCN2CC(N3CCN(c4ccc(-c5cnc6[nH]cc(C(=O)c7c(F)ccc(NS(=O)(=O)N8CC[C@@H](F)C8)c7F)c6c5)cc4)CC3)C2)C(C)(C)C)cc1	C56H64F3N11O7S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-R8496O	SCHEMBL22266426	(2S,4R)-1-[(2S)-2-[[2-[3-[[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]methyl]azetidin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CN2CC(Cc3ccc(-c4cnc5[nH]cc(C(=O)c6c(F)ccc(NS(=O)(=O)N7CC[C@@H](F)C7)c6F)c5c4)cc3)C2)C(C)(C)C)cc1	C52H56F3N9O7S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-0WJGQT	WO2018119448A1_104	.	CC(C)(C)[C@H](NC(=O)CN1CCN(CCc2ccc(-c3cnc4[nH]cc(C(=O)c5c(F)ccc(NS(=O)(=O)N6CC[C@@H](F)C6)c5F)c4c3)cc2)CC1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(-c2cncs2)cc1	C53H59F3N10O7S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-8L1QKD	SCHEMBL22266512	(2S,4R)-1-[(2S)-2-[[2-[3-[[4-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]piperazin-1-yl]methyl]azetidin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CN2CC(CN3CCN(c4ccc(-c5cnc6[nH]cc(C(=O)c7c(F)ccc(NS(=O)(=O)N8CC[C@@H](F)C8)c7F)c6c5)cc4)CC3)C2)C(C)(C)C)cc1	C56H64F3N11O7S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-CTDGGZ	SCHEMBL22266515	(2S,4R)-1-[(2S)-2-[[2-[3-[2-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]ethyl]azetidin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CN2CC(CCc3ccc(-c4cnc5[nH]cc(C(=O)c6c(F)ccc(NS(=O)(=O)N7CC[C@@H](F)C7)c6F)c5c4)cc3)C2)C(C)(C)C)cc1	C53H58F3N9O7S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-LR9JOO	SCHEMBL22266513	(2S,4R)-1-[(2S)-2-[[2-[2-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOc2ccc(-c3cnc4[nH]cc(C(=O)c5c(F)ccc(NS(=O)(=O)N6CC[C@@H](F)C6)c5F)c4c3)cc2)C(C)(C)C)cc1	C50H53F3N8O9S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-Y01MZI	SCHEMBL22266514	(2S,4R)-1-[(2S)-2-[[2-[3-[2-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenoxy]ethoxy]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCCOCCOc2ccc(-c3cnc4[nH]cc(C(=O)c5c(F)ccc(NS(=O)(=O)N6CC[C@@H](F)C6)c5F)c4c3)cc2)C(C)(C)C)cc1	C53H59F3N8O10S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-FDUYJI	SCHEMBL22266475	(2S,4R)-1-[(2S)-2-[5-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenoxy]pentanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCOc2ccc(-c3cnc4[nH]cc(C(=O)c5c(F)ccc(NS(=O)(=O)N6CC[C@@H](F)C6)c5F)c4c3)cc2)C(C)(C)C)cc1	C51H55F3N8O8S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-54BYA2	SCHEMBL22266474	(2S,4R)-1-[(2S)-2-[[2-[4-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]piperazin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CN2CCN(c3ccc(-c4cnc5[nH]cc(C(=O)c6c(F)ccc(NS(=O)(=O)N7CC[C@@H](F)C7)c6F)c5c4)cc3)CC2)C(C)(C)C)cc1	C52H57F3N10O7S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-CPR7GD	SCHEMBL22266476	(2S,4R)-1-[(2S)-2-[4-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenoxy]butanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCOc2ccc(-c3cnc4[nH]cc(C(=O)c5c(F)ccc(NS(=O)(=O)N6CC[C@@H](F)C6)c5F)c4c3)cc2)C(C)(C)C)cc1	C50H53F3N8O8S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-NA4W6T	SCHEMBL22266477	(2S,4R)-1-[(2S)-2-[5-[4-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]piperazin-1-yl]pentanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCN2CCN(c3ccc(-c4cnc5[nH]cc(C(=O)c6c(F)ccc(NS(=O)(=O)N7CC[C@@H](F)C7)c6F)c5c4)cc3)CC2)C(C)(C)C)cc1	C55H63F3N10O7S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-W6Q6Q4	SCHEMBL22266539	(2S,4R)-1-[(2S)-2-[6-[4-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]piperazin-1-yl]hexanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCN2CCN(c3ccc(-c4cnc5[nH]cc(C(=O)c6c(F)ccc(NS(=O)(=O)N7CC[C@@H](F)C7)c6F)c5c4)cc3)CC2)C(C)(C)C)cc1	C56H65F3N10O7S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-7D4V30	WO2018119448A1_114	.	Cc1ncsc1-c1ccc(CNC(=O)[C@H]2CCCN2C(=O)[C@H](NC(=O)CN2CC(N3CCN(c4ccc(-c5cnc6[nH]cc(C(=O)c7c(F)ccc(NS(=O)(=O)N8CC[C@@H](F)C8)c7F)c6c5)cc4)CC3)C2)C(C)(C)C)cc1	C55H62F3N11O6S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-PF4097	SCHEMBL22266540	(2S,4R)-1-[(2S)-2-[[2-[4-[[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenoxy]methyl]piperidin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CN2CCC(COc3ccc(-c4cnc5[nH]cc(C(=O)c6c(F)ccc(NS(=O)(=O)N7CC[C@@H](F)C7)c6F)c5c4)cc3)CC2)C(C)(C)C)cc1	C54H60F3N9O8S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-4AZZ9T	SCHEMBL22266545	(2S,4R)-1-[(2S)-2-[[2-[4-[3-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]azetidin-1-yl]piperidin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CN2CCC(N3CC(c4ccc(-c5cnc6[nH]cc(C(=O)c7c(F)ccc(NS(=O)(=O)N8CC[C@@H](F)C8)c7F)c6c5)cc4)C3)CC2)C(C)(C)C)cc1	C56H63F3N10O7S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-FAGXEM	SCHEMBL20294556	2-(2,6-dioxopiperidin-3-yl)-5-[4-[4-[4-[(1E)-1-hydroxyimino-2,3-dihydroinden-5-yl]-3-pyridin-4-ylpyrazol-1-yl]phenyl]piperazin-1-yl]isoindole-1,3-dione	O=C1CCC(N2C(=O)c3ccc(N4CCN(c5ccc(-n6cc(-c7ccc8c(c7)CC/C8=N\O)c(-c7ccncc7)n6)cc5)CC4)cc3C2=O)C(=O)N1	C40H34N8O5	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-D4OMKV	WO2018119448A1_118	.	O=C1CCC(N2C(=O)c3ccc(N4CC(Cc5ccc(-n6cc(-c7ccc8c(c7)CC/C8=N\O)c(-c7ccncc7)n6)cc5)C4)cc3C2=O)C(=O)N1	C40H33N7O5	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-3ILD8R	WO2018119448A1_119	.	O=C1CCC(N2C(=O)c3ccc(N4CC(Oc5ccc(-n6cc(-c7ccc8c(c7)CC/C8=N\O)c(-c7ccncc7)n6)cc5)C4)cc3C2=O)C(=O)N1	C39H31N7O6	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-YOEF7Y	WO2018119448A1_120	.	O=C1CCC(N2C(=O)c3ccc(N4CC[C@@H](Oc5ccc(-n6cc(-c7ccc8c(c7)CC/C8=N\O)c(-c7ccncc7)n6)cc5)C4)cc3C2=O)C(=O)N1	C40H33N7O6	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-YLZVOP	WO2018119448A1_121	.	O=C1CCC(N2C(=O)c3ccc(N4CCC(c5ccc(-n6cc(-c7ccc8c(c7)CC/C8=N\O)c(-c7ccncc7)n6)cc5)C4)cc3C2=O)C(=O)N1	C40H33N7O5	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-71T2E9	WO2018119448A1_122	.	O=C1CCC(N2C(=O)c3cccc(N4CCN(c5ccc(-n6cc(-c7ccc8c(c7)CC/C8=N\O)c(-c7ccncc7)n6)cc5)CC4)c3C2=O)C(=O)N1	C40H34N8O5	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-36IPH3	WO2018119448A1_123	.	O=C1CCC(N2C(=O)c3ccc(N4CCN(c5cccc(-n6cc(-c7ccc8c(c7)CC/C8=N\O)c(-c7ccncc7)n6)c5)CC4)cc3C2=O)C(=O)N1	C40H34N8O5	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-X742OQ	WO2018119448A1_124	.	O=C1CCC(N2C(=O)c3ccc(N4CCCN(c5ccc(-n6cc(-c7ccc8c(c7)CC/C8=N\O)c(-c7ccncc7)n6)cc5)CC4)cc3C2=O)C(=O)N1	C41H36N8O5	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-P8UEOR	WO2018119448A1_125	.	O=C1CCC(N2C(=O)c3ccc(N4CCN(CCc5ccc(-n6cc(-c7ccc8c(c7)CC/C8=N\O)c(-c7ccncc7)n6)cc5)CC4)cc3C2=O)C(=O)N1	C42H38N8O5	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-ADM9XG	WO2018119448A1_126	.	O=C1CCC(N2C(=O)c3ccc(N4CCN(Cc5ccc(-n6cc(-c7ccc8c(c7)CC/C8=N\O)c(-c7ccncc7)n6)cc5)CC4)cc3C2=O)C(=O)N1	C41H36N8O5	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-DZUWSI	WO2018119448A1_127	.	O=C1CCC(N2C(=O)c3ccc(N4CCC(c5ccc(-n6cc(-c7ccc8c(c7)CC/C8=N\O)c(-c7ccncc7)n6)cc5)CC4)cc3C2=O)C(=O)N1	C41H35N7O5	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-44BAGC	WO2018119448A1_128	.	O=C1CCC(N2C(=O)c3ccc(N4CCC[C@H](c5ccc(-n6cc(-c7ccc8c(c7)CC/C8=N\O)c(-c7ccncc7)n6)cc5)C4)cc3C2=O)C(=O)N1	C41H35N7O5	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-VOFDDM	WO2018119448A1_129	.	O=C1CCC(N2C(=O)c3ccc(N4CCN(C5CN(c6ccc(-n7cc(-c8ccc9c(c8)CC/C9=N\O)c(-c8ccncc8)n7)cc6)C5)CC4)cc3C2=O)C(=O)N1	C43H39N9O5	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-FRDOGJ	WO2018119448A1_130	.	O=C1CCC(N2C(=O)c3cccc(N4CC[C@H](N5CCN(c6ccc(-n7cc(-c8ccc9c(c8)CC/C9=N\O)c(-c8ccncc8)n7)cc6)CC5)C4)c3C2=O)C(=O)N1	C44H41N9O5	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-YE5YVD	WO2018119448A1_131	.	O=C1CCC(N2C(=O)c3cccc(N4CC[C@@H](N5CCN(c6ccc(-n7cc(-c8ccc9c(c8)CC/C9=N\O)c(-c8ccncc8)n7)cc6)CC5)C4)c3C2=O)C(=O)N1	C44H41N9O5	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-10V37Y	WO2018119448A1_132	.	O=C1CCC(N2C(=O)c3ccc(N4CCN(c5ccc(C6C=C(c7ccc8c(c7)CC/C8=N\O)C(c7ccncc7)=N6)cc5)CC4)c(Cl)c3C2=O)C(=O)N1	C41H34ClN7O5	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-FVNI4C	WO2018119448A1_133	.	C[C@H]1CN(c2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)C[C@H](C)N1c1ccc(-n2cc(-c3ccc4c(c3)CC/C4=N\O)c(C3=CC=NCC3)n2)cc1	C42H40N8O5	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-MP3X7Q	WO2018119448A1_134	.	O=C1CCC(N2C(=O)c3ccc(N4C[C@H]5C[C@@H]4CN5c4ccc(-n5cc(-c6ccc7c(c6)CC/C7=N\O)c(-c6ccncc6)n5)cc4)cc3C2=O)C(=O)N1	C41H34N8O5	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-718L73	WO2018119448A1_135	.	O=C1CCC(N2C(=O)c3ccc(N4C[C@@H]5C[C@H]4CN5c4ccc(-n5cc(-c6ccc7c(c6)CC/C7=N\O)c(-c6ccncc6)n5)cc4)cc3C2=O)C(=O)N1	C41H34N8O5	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-4FQT68	WO2018119448A1_136	.	C[C@@H]1CN(c2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)C[C@H](C)N1c1ccc(-n2cc(-c3ccc4c(c3)CC/C4=N\O)c(-c3ccncc3)n2)cc1	C42H38N8O5	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-44NMTD	WO2018119448A1_137	.	O=C1CCC(N2C(=O)c3ccc(NCCOc4ccc(-n5cc(-c6ccc7c(c6)CC/C7=N\O)c(-c6ccncc6)n5)cc4)cc3C2=O)C(=O)N1	C38H31N7O6	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-1MD3N7	WO2018119448A1_138	.	O=C1CCC(N2C(=O)c3cccc(N4CCN(CCc5ccc(-n6cc(-c7ccc8c(c7)CC/C8=N\O)c(-c7ccncc7)n6)cc5)CC4)c3C2=O)C(=O)N1	C42H38N8O5	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-NGP3EX	WO2018119448A1_139	.	CCCS(=O)(=O)Nc1ccnc2cc(-c3cn(-c4ccc(N5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)cc4)nc3-c3ccncc3)ccc12	C43H39N9O6S	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-FVTQFG	WO2018119448A1_140	.	CCCS(=O)(=O)Nc1cccc2cc(-c3cn(-c4ccc(N5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)cc4)nc3-c3ccncc3)cnc12	C43H39N9O6S	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-74GUTE	WO2018119448A1_141	.	O=C1CCC(N2C(=O)c3cccc(N4CCN(c5cccc(-n6cc(-c7ccc8c(c7)CC/C8=N\O)c(-c7ccncc7)n6)c5)CC4)c3C2=O)C(=O)N1	C40H34N8O5	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-HQ0ZX5	WO2018119448A1_142	.	O=C1CCC(N2C(=O)c3cccc(N4CCN(Cc5ccc(-n6cc(-c7ccc8c(c7)CC/C8=N\O)c(-c7ccncc7)n6)cc5)CC4)c3C2=O)C(=O)N1	C41H36N8O5	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-5AQKYN	WO2018119448A1_143	.	O=C1CCC(N2C(=O)c3cc(F)c(N4CCN(c5ccc(-n6cc(-c7ccc8c(c7)CC/C8=N\O)c(-c7ccncc7)n6)cc5)CC4)cc3C2=O)C(=O)N1	C40H33FN8O5	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-03KTQE	WO2018119448A1_144	.	O=C1CCC(N2C(=O)c3ccc(N4CC(CCOc5ccc(N6C=C(c7ccc8c(c7)CC/C8=N\O)C(c7ccncc7)N6)cc5)C4)cc3C2=O)C(=O)N1	C41H37N7O6	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-LW7PLC	WO2018119448A1_145	.	O=C1CCC(N2C(=O)c3ccc(N4CC(CCCOc5ccc(-n6cc(-c7ccc8c(c7)CC/C8=N\O)c(C7C=CN=CC7)n6)cc5)C4)cc3C2=O)C(=O)N1	C42H39N7O6	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-JMMW1J	WO2018119448A1_146	.	CN(c1ccc2c(c1)C(=O)N(C1CCC(=O)NC1=O)C2=O)[C@H]1C[C@@H](Oc2ccc(-n3cc(-c4ccc5c(c4)CC/C5=N\O)c(-c4ccncc4)n3)cc2)C1	C41H35N7O6	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-W60PIV	WO2018119448A1_147	.	CN(c1ccc2c(c1)C(=O)N(C1CCC(=O)NC1=O)C2=O)[C@H]1C[C@H](Oc2ccc(-n3cc(-c4ccc5c(c4)CC/C5=N\O)c(-c4ccncc4)n3)cc2)C1	C41H35N7O6	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-BJEZW1	WO2018119448A1_148	.	COc1cc(N2CCN(c3ccc(-n4cc(-c5ccc6c(c5)CC/C6=N\O)c(-c5ccncc5)n4)cc3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O	C41H36N8O6	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-9JWTV9	WO2018119448A1_149	.	COc1cc2c(cc1N1CCN(c3ccc(-n4cc(-c5ccc6c(c5)CC/C6=N\O)c(-c5ccncc5)n4)cc3)CC1)C(=O)N(C1CCC(=O)NC1=O)C2=O	C41H36N8O6	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-XNKBD8	SCHEMBL20294567	2-(2,6-dioxopiperidin-3-yl)-4-[4-[3-[2-[4-[4-[(1E)-1-hydroxyimino-2,3-dihydroinden-5-yl]-3-pyridin-4-ylpyrazol-1-yl]phenoxy]ethoxy]propyl]piperazin-1-yl]isoindole-1,3-dione	O=C1CCC(N2C(=O)c3cccc(N4CCN(CCCOCCOc5ccc(-n6cc(-c7ccc8c(c7)CC/C8=N\O)c(-c7ccncc7)n6)cc5)CC4)c3C2=O)C(=O)N1	C45H44N8O7	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-NH1J7H	WO2018119448A1_151	.	O=C1CCC(N2C(=O)c3cccc(N4CCN(CCOc5ccc(-n6cc(-c7ccc8c(c7)CC/C8=N\O)c(-c7ccncc7)n6)cc5)CC4)c3C2=O)C(=O)N1	C42H38N8O6	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-WKM9JE	SCHEMBL20294779	2-(2,6-dioxopiperidin-3-yl)-5-[4-[2-[4-[4-[(1E)-1-hydroxyimino-2,3-dihydroinden-5-yl]-3-pyridin-4-ylpyrazol-1-yl]phenoxy]ethyl]piperazin-1-yl]isoindole-1,3-dione	O=C1CCC(N2C(=O)c3ccc(N4CCN(CCOc5ccc(-n6cc(-c7ccc8c(c7)CC/C8=N\O)c(-c7ccncc7)n6)cc5)CC4)cc3C2=O)C(=O)N1	C42H38N8O6	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-2Q9ULI	WO2018119448A1_153	.	CN(CCOc1ccc(-n2cc(-c3ccc4c(c3)CC/C4=N\O)c(-c3ccncc3)n2)cc1)CCOc1ccc2c(c1)C(=O)N(C1CCC(=O)NC1=O)C2=O	C41H37N7O7	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-YNOXG4	WO2018119448A1_154	.	O=C1CCC(N2C(=O)C3=C(CCC(N4CCN(CCOc5cccc(-n6cc(-c7ccc8c(c7)CC/C8=N\O)c(-c7ccncc7)n6)c5)CC4)=C3)C2=O)C(=O)N1	C42H40N8O6	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-2HLI76	WO2018119448A1_155	.	CCCS(=O)(=O)Nc1cccc2cc(-c3cn(-c4ccc(OCCOCCOCCN5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)cc4)nc3-c3ccncc3)cnc12	C49H51N9O9S	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-SVAEGV	WO2018119448A1_156	.	CCCS(=O)(=O)Nc1ccnc2cc(-c3cn(-c4ccc(OCCN5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)cc4)nc3-c3ccncc3)ccc12	C45H43N9O7S	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-NPDIS7	WO2018119448A1_157	.	CCCS(=O)(=O)NC1=CCNc2cc(-c3cn(-c4ccc(OCCOCCN5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)cc4)nc3-c3ccncc3)ccc21	C47H49N9O8S	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-4STYZE	WO2018119448A1_158	N-[3-[1-[4-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]ethoxy]phenyl]-3-pyridin-4-ylpyrazol-4-yl]quinolin-8-yl]propane-1-sulfonamide	CCCS(=O)(=O)Nc1cccc2cc(-c3cn(-c4ccc(OCCN5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)cc4)nc3-c3ccncc3)cnc12	C45H43N9O7S	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-1ME5VI	WO2018119448A1_159	N-[3-[1-[4-[2-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]ethoxy]ethoxy]phenyl]-3-pyridin-4-ylpyrazol-4-yl]quinolin-8-yl]propane-1-sulfonamide	CCCS(=O)(=O)Nc1cccc2cc(-c3cn(-c4ccc(OCCOCCN5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)cc4)nc3-c3ccncc3)cnc12	C47H47N9O8S	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-9GXKML	WO2018119448A1_160	2-(2,6-dioxopiperidin-3-yl)-5-[4-[2-[2-[3-[4-[(1E)-1-hydroxyimino-2,3-dihydroinden-5-yl]-3-pyridin-4-ylpyrazol-1-yl]phenoxy]ethoxy]ethyl]piperazin-1-yl]isoindole-1,3-dione	O=C1CCC(N2C(=O)c3ccc(N4CCN(CCOCCOc5cccc(-n6cc(-c7ccc8c(c7)CC/C8=N\O)c(-c7ccncc7)n6)c5)CC4)cc3C2=O)C(=O)N1	C44H42N8O7	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-5FSZG4	WO2018119448A1_161	.	O=C1CCC(N2C(=O)c3ccc(N4CC5(CN(CCOc6ccc(-n7cc(-c8ccc9c(c8)CC/C9=N\O)c(-c8ccncc8)n7)cc6)C5)C4)cc3C2=O)C(=O)N1	C43H38N8O6	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-6WZLY4	WO2018119448A1_162	.	O=C1CCC(N2C(=O)c3cccc(N4CCN(CCCCOc5ccc(-n6cc(-c7ccc8c(c7)CC/C8=N\O)c(-c7ccncc7)n6)cc5)CC4)c3C2=O)C(=O)N1	C44H42N8O6	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-1INH4U	WO2018119448A1_163	.	O=C1CCC(N2C(=O)c3cccc(N4CCN(CCCOc5ccc(-n6cc(-c7ccc8c(c7)CC/C8=N\O)c(-c7ccncc7)n6)cc5)CC4)c3C2=O)C(=O)N1	C43H40N8O6	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-0EBXKY	WO2018119448A1_164	.	O=C1CCC(N2C(=O)c3ccc(N4CCN(CCCOc5ccc(-n6cc(-c7ccc8c(c7)CC/C8=N\O)c(-c7ccncc7)n6)cc5)CC4)cc3C2=O)C(=O)N1	C43H40N8O6	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-YWKIFH	WO2018119448A1_165	.	O=C1CCC(N2C(=O)c3ccc(N4CCN(CCCCOc5ccc(-n6cc(-c7ccc8c(c7)CC/C8=N\O)c(-c7ccncc7)n6)cc5)CC4)cc3C2=O)C(=O)N1	C44H42N8O6	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-9WCQYT	WO2018119448A1_166	.	O=C1CCC(N2C(=O)c3ccc(N4CCN(CC5CCN(c6ccc(-n7cc(-c8ccc9c(c8)CC/C9=N\O)c(-c8ccncc8)n7)cc6)CC5)CC4)cc3C2=O)C(=O)N1	C46H45N9O5	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-WC9LGM	WO2018119448A1_167	.	O=C1CCC(N2C(=O)c3ccc(N4CCC(C5CN(CCOc6ccc(-n7cc(-c8ccc9c(c8)CC/C9=N\O)c(-c8ccncc8)n7)cc6)C5)CC4)cc3C2=O)C(=O)N1	C46H44N8O6	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-QEZ671	WO2018119448A1_168	.	O=C1CCC(N2Cc3cc(N4CCN(CCOc5ccc(-n6cc(-c7ccc8c(c7)CC/C8=N\O)c(-c7ccncc7)n6)cc5)CC4)ccc3C2=O)C(=O)N1	C42H40N8O5	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-254LPH	WO2018119448A1_169	.	O=C1CCC(N2C(=O)c3ccc(N4CCN(CCC5CCN(c6ccc(-n7cc(-c8ccc9c(c8)CC/C9=N\O)c(-c8ccncc8)n7)cc6)CC5)CC4)cc3C2=O)C(=O)N1	C47H47N9O5	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-QR4JQS	WO2018119448A1_170	.	O=C1CCC(N2C(=O)c3ccc(OC4CCN(CCOc5ccc(-n6cc(-c7ccc8c(c7)CC/C8=N\O)c(-c7ccncc7)n6)cc5)CC4)cc3C2=O)C(=O)N1	C43H39N7O7	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-N6MENJ	WO2018119448A1_171	.	O=C1CCC(N2C(=O)c3ccc(OCC4CCN(CCOc5ccc(-n6cc(-c7ccc8c(c7)CC/C8=N\O)c(-c7ccncc7)n6)cc5)CC4)cc3C2=O)C(=O)N1	C44H41N7O7	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-HE2S58	WO2018119448A1_172	.	O=C1CCC(N2C(=O)c3ccc(OCCN4CCN(CCOc5ccc(-n6cc(-c7ccc8c(c7)CC/C8=N\O)c(-c7ccncc7)n6)cc5)CC4)cc3C2=O)C(=O)N1	C44H42N8O7	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-2LPC1K	WO2018119448A1_173	.	O=C1CCC(N2C(=O)c3cccc(OCCN4CCN(c5ccc(-n6cc(-c7ccc8c(c7)CC/C8=N\O)c(-c7ccncc7)n6)cc5)CC4)c3C2=O)C(=O)N1	C42H38N8O6	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-KHXTZP	WO2018119448A1_174	.	O=C1CCC(N2C(=O)c3cccc(OCCCCN4CCN(c5ccc(-n6cc(-c7ccc8c(c7)CC/C8=N\O)c(-c7ccncc7)n6)cc5)CC4)c3C2=O)C(=O)N1	C44H42N8O6	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-0D0Y8Z	WO2018119448A1_175	.	O=C1CCC(N2C(=O)c3cccc(N4CC(N5CCN(c6ccc(-n7cc(-c8ccc9c(c8)CC/C9=N\O)c(-c8ccncc8)n7)cc6)CC5)C4)c3C2=O)C(=O)N1	C43H39N9O5	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-B6TIYQ	WO2018119448A1_176	.	O=C1CCC(N2C(=O)c3cccc(N4CC(CC5CCN(c6ccc(-n7cc(-c8ccc9c(c8)CC/C9=N\O)c(-c8ccncc8)n7)cc6)CC5)C4)c3C2=O)C(=O)N1	C45H42N8O5	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-8R7W41	WO2018119448A1_177	.	O=C1CCC(N2C(=O)c3ccc(N4CC(N5CCC(c6ccc(-n7cc(-c8ccc9c(c8)CC/C9=N\O)c(-c8ccncc8)n7)cc6)CC5)C4)cc3C2=O)C(=O)N1	C44H40N8O5	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-Y0FBQR	WO2018119448A1_178	.	O=C1CCC(N2C(=O)c3cccc(N4CC(CN5CC(c6ccc(-n7cc(-c8ccc9c(c8)CC/C9=N\O)c(-c8ccncc8)n7)cc6)C5)C4)c3C2=O)C(=O)N1	C43H38N8O5	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-0X4J5M	WO2018119448A1_179	.	O=C1CCC(N2C(=O)c3ccc(N4CC(CN5CC(c6ccc(-n7cc(-c8ccc9c(c8)CC/C9=N\O)c(-c8ccncc8)n7)cc6)C5)C4)cc3C2=O)C(=O)N1	C43H38N8O5	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-S1L2VL	WO2018119448A1_180	.	O=C1CCC(N2C(=O)c3cccc(OCCCN4CC(c5ccc(-n6cc(-c7ccc8c(c7)CC/C8=N\O)c(-c7ccncc7)n6)cc5)C4)c3C2=O)C(=O)N1	C42H37N7O6	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-1SBDEB	WO2018119448A1_181	.	O=C1CCC(N2C(=O)c3cccc(OCCCCN4CC(c5ccc(-n6cc(-c7ccc8c(c7)CC/C8=N\O)c(-c7ccncc7)n6)cc5)C4)c3C2=O)C(=O)N1	C43H39N7O6	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-4CZLI4	SCHEMBL20294749	N-[3-[5-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperidin-4-yl]-methylamino]-3-pyrimidin-5-ylpyrrolo[3,2-b]pyridin-1-yl]-2,4-difluorophenyl]propane-1-sulfonamide	CCCS(=O)(=O)Nc1ccc(F)c(-n2cc(-c3cncnc3)c3nc(N(C)C4CCN(c5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)ccc32)c1F	C39H37F2N9O6S	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-NFEQ9Z	WO2018119448A1_183	.	CCCS(=O)(=O)Nc1ccc(F)c(-n2cc(-c3cncnc3)c3nc(N(C)C4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)ccc32)c1F	C39H37F2N9O6S	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-XCR6VL	SCHEMBL20294696	N-[3-[5-[[1-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyethyl]piperidin-4-yl]-methylamino]-3-pyrimidin-5-ylpyrrolo[3,2-b]pyridin-1-yl]-2,4-difluorophenyl]propane-1-sulfonamide	CCCS(=O)(=O)Nc1ccc(F)c(-n2cc(-c3cncnc3)c3nc(N(C)C4CCN(CCOc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)ccc32)c1F	C41H41F2N9O7S	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-0GMX0A	WO2018119448A1_185	.	CCCS(=O)(=O)Nc1ccc(F)c(-n2cc(-c3cncnc3)c3nc(N(C)C4CCN(CCOCCOc5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)ccc32)c1F	C43H45F2N9O8S	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-DMECA9	WO2018119448A1_186	.	CCCS(=O)(=O)Nc1ccc(F)c(-n2cc(-c3cncnc3)c3nc(NC4CCN(CCOc5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)ccc32)c1F	C40H39F2N9O7S	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-XX0WX5	WO2018119448A1_187	.	C=Nc1c(-c2cncnc2)cn(-c2c(F)ccc(NS(=O)(=O)CCC)c2F)c1/C=C\CN(C)C1CCN(CCOCCOc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)CC1	C44H49F2N9O8S	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-UWN4VA	WO2018119448A1_188	.	CCCS(=O)(=O)Nc1ccc(F)c(-n2cc(-c3cncnc3)c3nc(N(C)C4CCN(CCOCCOCCOc5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)ccc32)c1F	C45H49F2N9O9S	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-2RFYN8	WO2018119448A1_189	.	CCCS(=O)(=O)Nc1ccc(F)c(-n2cc(-c3cncnc3)c3nc(N(C)C4CCN(CCOCCOCCOc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)ccc32)c1F	C45H49F2N9O9S	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-UJ4TNP	WO2018119448A1_190	.	CCCS(=O)(=O)Nc1ccc(F)c(-n2cc(-c3cncnc3)c3nc(N(C)C4CCN(CC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)NCc5ccc(-c6scnc6C)cc5)C(C)(C)C)CC4)ccc32)c1F	C50H59F2N11O6S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-ZZPKX2	SCHEMBL20294688	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[4-[[1-[2,6-difluoro-3-(propylsulfonylamino)phenyl]-3-pyrimidin-5-ylpyrrolo[3,2-b]pyridin-5-yl]-methylamino]piperidin-1-yl]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CCCS(=O)(=O)Nc1ccc(F)c(-n2cc(-c3cncnc3)c3nc(N(C)C4CCN(CCOCCOCC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)NCc5ccc(-c6scnc6C)cc5)C(C)(C)C)CC4)ccc32)c1F	C54H67F2N11O8S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-30E7JR	WO2018119448A1_192	.	CCCS(=O)(=O)Nc1ccc(F)c(-n2cc(-c3cncnc3)c3nc(N(C)C4CCN(CCOCC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)NCc5ccc(-c6scnc6C)cc5)C(C)(C)C)CC4)ccc32)c1F	C52H63F2N11O7S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-9TBA9M	SCHEMBL22266419	(3R)-N-[3-[5-[4-[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxypropoxy]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2C(=O)c3ccc(OCCCOc4ccc(-c5cnc6[nH]cc(C(=O)c7c(F)ccc(NS(=O)(=O)N8CC[C@@H](F)C8)c7F)c6c5)cc4)cc3C2=O)C(=O)N1	C40H33F3N6O9S	BRAF	P15056	VHL	WO-2018119448-A1
TPD-0JGP26	SCHEMBL24021719	(3R)-N-[3-[5-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxybutoxy]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2C(=O)c3ccc(OCCCCOc4ccc(-c5cnc6[nH]cc(C(=O)c7c(F)ccc(NS(=O)(=O)N8CC[C@@H](F)C8)c7F)c6c5)cc4)cc3C2=O)C(=O)N1	C41H35F3N6O9S	BRAF	P15056	VHL	WO-2018119448-A1
TPD-I9S0SP	SCHEMBL20294731	(3R)-N-[3-[5-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxyethoxy]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2C(=O)c3ccc(OCCOc4ccc(-c5cnc6[nH]cc(C(=O)c7c(F)ccc(NS(=O)(=O)N8CC[C@@H](F)C8)c7F)c6c5)cc4)cc3C2=O)C(=O)N1	C39H31F3N6O9S	BRAF	P15056	VHL	WO-2018119448-A1
TPD-V5RXTA	SCHEMBL20323740	2-(2,6-dioxopiperidin-3-yl)-5-[3-[4-[4-[4-[(1E)-1-hydroxyimino-2,3-dihydroinden-5-yl]-3-pyridin-4-ylpyrazol-1-yl]phenoxy]butoxy]phenyl]isoindole-1,3-dione	O=C1CCC(N2C(=O)c3ccc(-c4cccc(OCCCCOc5ccc(-n6cc(-c7ccc8c(c7)CC/C8=N\O)c(-c7ccncc7)n6)cc5)c4)cc3C2=O)C(=O)N1	C46H38N6O7	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-DJSHL6	SCHEMBL20294836	2-(2,6-dioxopiperidin-3-yl)-5-[4-[2-[2-[4-[4-[(1E)-1-hydroxyimino-2,3-dihydroinden-5-yl]-3-pyridin-4-ylpyrazol-1-yl]phenoxy]ethoxy]ethyl]piperazin-1-yl]isoindole-1,3-dione	O=C1CCC(N2C(=O)c3ccc(N4CCN(CCOCCOc5ccc(-n6cc(-c7ccc8c(c7)CC/C8=N\O)c(-c7ccncc7)n6)cc5)CC4)cc3C2=O)C(=O)N1	C44H42N8O7	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-8Z0K57	SCHEMBL20294637	2-(2,6-dioxopiperidin-3-yl)-5-[2-[2-[4-[4-[4-[(1E)-1-hydroxyimino-2,3-dihydroinden-5-yl]-3-pyridin-4-ylpyrazol-1-yl]phenyl]piperazin-1-yl]ethoxy]ethoxy]isoindole-1,3-dione	O=C1CCC(N2C(=O)c3ccc(OCCOCCN4CCN(c5ccc(-n6cc(-c7ccc8c(c7)CC/C8=N\O)c(-c7ccncc7)n6)cc5)CC4)cc3C2=O)C(=O)N1	C44H42N8O7	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-W9XPSB	WO2018119448A1_199	.	N/N=C1\CCc2cc(-c3cn(-c4ccc(N5CCN(CCCOc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)cc4)nc3-c3ccncc3)ccc21	C43H41N9O5	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-MJQT7A	SCHEMBL20294530	2-(2,6-dioxopiperidin-3-yl)-4-[3-[3-[4-[4-[(1E)-1-hydroxyimino-2,3-dihydroinden-5-yl]-3-pyridin-4-ylpyrazol-1-yl]phenoxy]propoxy]phenyl]isoindole-1,3-dione	O=C1CCC(N2C(=O)c3cccc(-c4cccc(OCCCOc5ccc(-n6cc(-c7ccc8c(c7)CC/C8=N\O)c(-c7ccncc7)n6)cc5)c4)c3C2=O)C(=O)N1	C45H36N6O7	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-WFQQKS	SCHEMBL20323662	5-[4-[4-[4-[(1E)-1-hydroxyimino-2,3-dihydroinden-5-yl]-3-pyridin-4-ylpyrazol-1-yl]phenyl]piperazin-1-yl]-2-(1-methyl-2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN1C(=O)CCC(N2C(=O)c3ccc(N4CCN(c5ccc(-n6cc(-c7ccc8c(c7)CC/C8=N\O)c(-c7ccncc7)n6)cc5)CC4)cc3C2=O)C1=O	C41H36N8O5	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-AA9OXK	WO2018119448A1_202	.	O=C1CCC(N2C(=O)C3C=CC(N4CCN(CCN5CCN(c6ccc(-c7cnc8[nH]cc(C(=O)c9c(F)ccc(NS(=O)(=O)N%10CC[C@@H](F)C%10)c9F)c8c7)cc6)CC5)CC4)=CC3C2=O)C(=O)N1	C47H49F3N10O7S	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-MOJHD9	WO2018119448A1_203	.	O=C1CCC(N2C(=O)c3ccc(OCCOc4cccc(N5C=C(c6ccc7c(c6)CC/C7=N\O)C(c6ccncc6)N5)c4)cc3C2=O)C(=O)N1	C38H32N6O7	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-TOXK3I	WO2018119448A1_204	.	O=C1CCC(N2C(=O)c3ccc(OCCOCCOc4cccc(-n5cc(-c6ccc7c(c6)CCC7NO)c(-c6ccncc6)n5)c4)cc3C2=O)C(=O)N1	C40H36N6O8	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-98A4ZW	WO2018119448A1_205	.	O=C1CCC(N2C(=O)c3ccc(OCCOCCOCCOc4cccc(-n5cc(-c6ccc7c(c6)CCC7NO)c(-c6ccncc6)n5)c4)cc3C2=O)C(=O)N1	C42H40N6O9	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-WO29BV	SCHEMBL20294517	2-(2,6-dioxopiperidin-3-yl)-5-[2-[4-[4-[(1E)-1-hydroxyimino-2,3-dihydroinden-5-yl]-3-pyridin-4-ylpyrazol-1-yl]piperidin-1-yl]ethoxy]isoindole-1,3-dione	O=C1CCC(N2C(=O)c3ccc(OCCN4CCC(n5cc(-c6ccc7c(c6)CC/C7=N\O)c(-c6ccncc6)n5)CC4)cc3C2=O)C(=O)N1	C37H35N7O6	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-HJ3TBR	SCHEMBL20294681	2-(2,6-dioxopiperidin-3-yl)-5-[4-[4-[4-[(1E)-1-hydroxyimino-2,3-dihydroinden-5-yl]-3-pyridin-4-ylpyrazol-1-yl]piperidin-1-yl]piperidin-1-yl]isoindole-1,3-dione	O=C1CCC(N2C(=O)c3ccc(N4CCC(N5CCC(n6cc(-c7ccc8c(c7)CC/C8=N\O)c(-c7ccncc7)n6)CC5)CC4)cc3C2=O)C(=O)N1	C40H40N8O5	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-EB7TI5	SCHEMBL20294527	(3R)-N-[3-[5-[4-[2-[2-[2-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]ethoxy]ethoxy]ethoxy]ethoxy]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2C(=O)c3ccc(N4CCN(CCOCCOCCOCCOc5ccc(-c6cnc7[nH]cc(C(=O)c8c(F)ccc(NS(=O)(=O)N9CC[C@@H](F)C9)c8F)c7c6)cc5)CC4)cc3C2=O)C(=O)N1	C49H51F3N8O11S	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-95ME0I	SCHEMBL20294650	2-(2,6-dioxopiperidin-3-yl)-5-[4-[(1S,3R)-3-[4-[(1E)-1-hydroxyimino-2,3-dihydroinden-5-yl]-3-pyridin-4-ylpyrazol-1-yl]cyclohexyl]oxypiperidin-1-yl]isoindole-1,3-dione	O=C1CCC(N2C(=O)c3ccc(N4CCC(O[C@H]5CCC[C@@H](n6cc(-c7ccc8c(c7)CC/C8=N\O)c(-c7ccncc7)n6)C5)CC4)cc3C2=O)C(=O)N1	C41H41N7O6	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-JA5OZ7	WO2018119448A1_210	.	O=C1CCC(N2C(=O)c3ccc(N4CCC(O[C@@H]5CCC[C@@H](N6C=C(c7ccc8c(c7)CC/C8=N\O)C(c7ccncc7)N6)C5)CC4)cc3C2=O)C(=O)N1	C41H43N7O6	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-XHUIFZ	SCHEMBL20294721	2-(2,6-dioxopiperidin-3-yl)-5-[3-[1-[2-[4-[4-[(1E)-1-hydroxyimino-2,3-dihydroinden-5-yl]-3-pyridin-4-ylpyrazol-1-yl]phenoxy]ethyl]piperidin-4-yl]azetidin-1-yl]isoindole-1,3-dione	O=C1CCC(N2C(=O)c3ccc(N4CC(C5CCN(CCOc6ccc(-n7cc(-c8ccc9c(c8)CC/C9=N\O)c(-c8ccncc8)n7)cc6)CC5)C4)cc3C2=O)C(=O)N1	C46H44N8O6	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-EW81HV	WO2018119448A1_212	.	O=C1CCC(N2C(=O)c3cccc(OCCOCCOc4cccc(OCCOc5ccc(-n6cc(-c7ccc8c(c7)CC/C8=N\O)c(-c7ccncc7)n6)cc5)c4)c3C2=O)C(=O)N1	C48H42N6O10	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-GBDSL2	WO2018119448A1_213	.	O=C1CCC(N2C(=O)c3c(OCCCOCCOc4ccccc4COc4ccc(-n5cc(-c6ccc7c(c6)CCC7NO)c(-c6ccncc6)n5)cc4)cccc3C2O)C(=O)N1	C48H46N6O9	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-07HHDC	WO2018119448A1_214	.	O=C1CCC(N2C(=O)c3cccc(OCCCOc4cccc(-c5ccc(-n6cc(-c7ccc8c(c7)CC/C8=N\O)c(-c7ccncc7)n6)cc5)c4)c3C2=O)C(=O)N1	C45H36N6O7	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-83IYJW	SCHEMBL20294646	2-(2,6-dioxopiperidin-3-yl)-4-[3-[3-[4-[4-[4-[(1E)-1-hydroxyimino-2,3-dihydroinden-5-yl]-3-pyridin-4-ylpyrazol-1-yl]phenyl]phenoxy]propoxy]propoxy]isoindole-1,3-dione	O=C1CCC(N2C(=O)c3cccc(OCCCOCCCOc4ccc(-c5ccc(-n6cc(-c7ccc8c(c7)CC/C8=N\O)c(-c7ccncc7)n6)cc5)cc4)c3C2=O)C(=O)N1	C48H42N6O8	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-H3BH75	SCHEMBL20294660	(2S,4R)-1-[(2S)-2-[3-[2-[3-[3-[2,6-difluoro-3-(propylsulfonylamino)benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenoxy]ethoxy]propanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CCCS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(-c4cccc(OCCOCCC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)NCc5ccc(-c6scnc6C)cc5)C(C)(C)C)c4)cc23)c1F	C50H55F2N7O9S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-92307C	SCHEMBL20294521	N-[4-[3-[2,6-difluoro-3-(propylsulfonylamino)benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]-N'-[(2S)-1-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]pentanediamide	CCCS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(-c4ccc(NC(=O)CCCC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)NCc5ccc(-c6scnc6C)cc5)C(C)(C)C)cc4)cc23)c1F	C50H54F2N8O8S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-NW3Y91	SCHEMBL20294526	(2S,4R)-1-[(2S)-2-[[5-[4-[3-[2,6-difluoro-3-(propylsulfonylamino)benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]piperazin-1-yl]-5-oxopentanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CCCS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(N4CCN(C(=O)CCCC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)NCc5ccc(-c6scnc6C)cc5)C(C)(C)C)CC4)cc23)c1F	C48H57F2N9O8S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-W2E40D	SCHEMBL20294703	(2S,4R)-1-[(2S)-2-[[4-[4-[3-[2,6-difluoro-3-(propylsulfonylamino)benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]piperazin-1-yl]-4-oxobutanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CCCS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(N4CCN(C(=O)CCC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)NCc5ccc(-c6scnc6C)cc5)C(C)(C)C)CC4)cc23)c1F	C47H55F2N9O8S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-314NB7	SCHEMBL20294625	N-[4-[3-[2,6-difluoro-3-(propylsulfonylamino)benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]-N'-[(2S)-1-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]butanediamide; SCHEMBL30179122	CCCS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(-c4ccc(NC(=O)CCC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)NCc5ccc(-c6scnc6C)cc5)C(C)(C)C)cc4)cc23)c1F	C49H52F2N8O8S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-GP64UC	SCHEMBL20294599	N-[4-[3-[2,6-difluoro-3-(propylsulfonylamino)benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]-N'-[(2S)-1-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]propanediamide	CCCS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(-c4ccc(NC(=O)CC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)NCc5ccc(-c6scnc6C)cc5)C(C)(C)C)cc4)cc23)c1F	C48H50F2N8O8S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-Z266EJ	SCHEMBL20294750	(2S,4R)-1-[(2S)-2-[[3-[4-[3-[2,6-difluoro-3-(propylsulfonylamino)benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]piperazin-1-yl]-3-oxopropanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CCCS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(N4CCN(C(=O)CC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)NCc5ccc(-c6scnc6C)cc5)C(C)(C)C)CC4)cc23)c1F	C46H53F2N9O8S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-3UXZJD	SCHEMBL22266437	(2S,4R)-1-[(2S)-2-[[2-[2-[4-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]piperidin-1-yl]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCN2CCC(c3ccc(-c4cnc5[nH]cc(C(=O)c6c(F)ccc(NS(=O)(=O)N7CC[C@@H](F)C7)c6F)c5c4)cc3)CC2)C(C)(C)C)cc1	C55H62F3N9O8S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-1GOYGG	SCHEMBL22266436	(2S,4R)-1-[(2S)-2-[[2-[3-[4-[5-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]pyrimidin-2-yl]piperazin-1-yl]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCCN2CCN(c3ncc(-c4cnc5[nH]cc(C(=O)c6c(F)ccc(NS(=O)(=O)N7CC[C@@H](F)C7)c6F)c5c4)cn3)CC2)C(C)(C)C)cc1	C53H61F3N12O8S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-IP3DKO	SCHEMBL22266507	(2S,4R)-1-[(2S)-2-[[2-[3-[4-[5-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]pyrimidin-2-yl]piperazin-1-yl]azetidin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CN2CC(N3CCN(c4ncc(-c5cnc6[nH]cc(C(=O)c7c(F)ccc(NS(=O)(=O)N8CC[C@@H](F)C8)c7F)c6c5)cn4)CC3)C2)C(C)(C)C)cc1	C53H60F3N13O7S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-BQBGZM	CHEMBL4633881	(2S,4R)-1-[(2S)-2-[[2-[4-[[4-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]piperazin-1-yl]methyl]piperidin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL20294790	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CN2CCC(CN3CCN(c4ccc(-c5cnc6[nH]cc(C(=O)c7c(F)ccc(NS(=O)(=O)N8CC[C@@H](F)C8)c7F)c6c5)cc4)CC3)CC2)C(C)(C)C)cc1	C58H68F3N11O7S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-LQ8VN3	CHEMBL4644860	(2S,4R)-1-[(2S)-2-[[2-[4-[[1-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL20294695	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CN2CCN(CC3CCN(c4ccc(-c5cnc6[nH]cc(C(=O)c7c(F)ccc(NS(=O)(=O)N8CC[C@@H](F)C8)c7F)c6c5)cc4)CC3)CC2)C(C)(C)C)cc1	C58H68F3N11O7S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-71MH5O	SCHEMBL22266508	(2S,4R)-1-[(2S)-2-[[2-[4-[2-[4-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]piperazin-1-yl]ethyl]piperidin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CN2CCC(CCN3CCN(c4ccc(-c5cnc6[nH]cc(C(=O)c7c(F)ccc(NS(=O)(=O)N8CC[C@@H](F)C8)c7F)c6c5)cc4)CC3)CC2)C(C)(C)C)cc1	C59H70F3N11O7S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-DIU67Q	SCHEMBL22266481	(2S,4R)-1-[(2S)-2-[[2-[2-[4-[5-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]pyrimidin-2-yl]piperazin-1-yl]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCN2CCN(c3ncc(-c4cnc5[nH]cc(C(=O)c6c(F)ccc(NS(=O)(=O)N7CC[C@@H](F)C7)c6F)c5c4)cn3)CC2)C(C)(C)C)cc1	C52H59F3N12O8S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-J6VNAC	SCHEMBL22266484	(2S,4R)-1-[(2S)-2-[[2-[3-[4-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidine-1-carbonyl]amino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]piperazin-1-yl]azetidin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CN2CC(N3CCN(c4ccc(-c5cnc6[nH]cc(C(=O)c7c(F)ccc(NC(=O)N8CC[C@@H](F)C8)c7F)c6c5)cc4)CC3)C2)C(C)(C)C)cc1	C56H62F3N11O6S	BRAF	P15056	VHL	WO-2018119448-A1
TPD-EQ9JM9	WO2018119448A1_231	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CC2CC(OCCOc3ccc(-c4cnc5[nH]cc(C(=O)c6c(F)ccc(NS(=O)(=O)N7CC[C@@H](F)C7)c6F)c5c4)cc3)C2)C(C)(C)C)cc1	C54H59F3N8O9S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-1F59H5	WO2018119448A1_232	.	Cc1ncsc1-c1ccc(CNC(O)[C@@H]2C[C@@H](O)CC2C(=O)[C@@H](NC(=O)CN2CCN(CCC3CCN(c4ccc(-c5cnc6[nH]cc(C(=O)c7c(F)ccc(NS(=O)(=O)N8CC[C@@H](F)C8)c7F)c6c5)cc4)CC3)CC2)C(C)(C)C)cc1	C60H73F3N10O7S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-PNBI8G	SCHEMBL22266502	(2S,4R)-1-[(2S)-2-[[2-[3-[[4-[5-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]pyrimidin-2-yl]piperazin-1-yl]methyl]azetidin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CN2CC(CN3CCN(c4ncc(-c5cnc6[nH]cc(C(=O)c7c(F)ccc(NS(=O)(=O)N8CC[C@@H](F)C8)c7F)c6c5)cn4)CC3)C2)C(C)(C)C)cc1	C54H62F3N13O7S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-EVMIW2	SCHEMBL22266505	(2S,4R)-1-[(2S)-2-[[2-[4-[1-[[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]methyl]piperidin-4-yl]piperazin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CN2CCN(C3CCN(Cc4ccc(-c5cnc6[nH]cc(C(=O)c7c(F)ccc(NS(=O)(=O)N8CC[C@@H](F)C8)c7F)c6c5)cc4)CC3)CC2)C(C)(C)C)cc1	C58H68F3N11O7S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-G3JPF0	SCHEMBL22266506	(2S,4R)-1-[(2S)-2-[[2-[4-[4-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenoxy]butyl]piperazin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CN2CCN(CCCCOc3ccc(-c4cnc5[nH]cc(C(=O)c6c(F)ccc(NS(=O)(=O)N7CC[C@@H](F)C7)c6F)c5c4)cc3)CC2)C(C)(C)C)cc1	C56H65F3N10O8S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-VIFQV9	WO2018119448A1_236	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CN2CC3(CN(CCc4ccc(-c5cnc6[nH]cc(C(=O)c7c(F)ccc(NS(=O)(=O)N8CC[C@@H](F)C8)c7F)c6c5)cc4)C3)C2)C(C)(C)C)cc1	C55H61F3N10O7S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-Z8IFWG	SCHEMBL22266517	(2S,4R)-1-[(2S)-2-[[2-[4-[[4-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]piperidin-1-yl]methyl]piperidin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CN2CCC(CN3CCC(c4ccc(-c5cnc6[nH]cc(C(=O)c7c(F)ccc(NS(=O)(=O)N8CC[C@@H](F)C8)c7F)c6c5)cc4)CC3)CC2)C(C)(C)C)cc1	C59H69F3N10O7S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-QU13QO	SCHEMBL22266519	(2S,4R)-1-[(2S)-2-[[2-[2-[4-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]piperazin-1-yl]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCN2CCN(c3ccc(-c4cnc5[nH]cc(C(=O)c6c(F)ccc(NS(=O)(=O)N7CC[C@@H](F)C7)c6F)c5c4)cc3)CC2)C(C)(C)C)cc1	C55H63F3N10O8S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-AV118N	CHEMBL4635857	(2S,4R)-1-[(2S)-2-[[2-[4-[[4-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]piperazin-1-yl]methyl]piperidin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL22266518	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CN2CCC(CN3CCN(c4ccc(-c5cnc6[nH]cc(C(=O)c7c(F)ccc(NS(=O)(=O)N8CC[C@@H](F)C8)c7F)c6c5)cc4)CC3)CC2)C(C)(C)C)cc1	C59H70F3N11O7S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-OV3W5S	WO2018119448A1_240	.	Cc1ncsc1-c1ccc([C@H](C)N[C@H](O)C2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CN2CC(N3CCN(c4ccc(-c5cnc6[nH]cc(C(=O)c7c(F)ccc(NS(=O)(=O)N8CC[C@@H](F)C8)c7F)c6c5)cc4)CC3)C2)C(C)(C)C)cc1	C56H66F3N11O7S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-O546DR	SCHEMBL22266441	(2S,4R)-1-[(2S)-2-[[2-[4-[4-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]piperazin-1-yl]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCCCN2CCN(c3ccc(-c4cnc5[nH]cc(C(=O)c6c(F)ccc(NS(=O)(=O)N7CC[C@@H](F)C7)c6F)c5c4)cc3)CC2)C(C)(C)C)cc1	C56H65F3N10O8S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-K0TLE9	SCHEMBL22266440	(2S,4R)-1-[(2S)-2-[[2-[2-[4-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]piperazin-1-yl]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1R)-2-hydroxy-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](CO)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCN2CCN(c3ccc(-c4cnc5[nH]cc(C(=O)c6c(F)ccc(NS(=O)(=O)N7CC[C@@H](F)C7)c6F)c5c4)cc3)CC2)C(C)(C)C)cc1	C55H63F3N10O9S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-0HOWES	SCHEMBL22266438	(2S,4R)-1-[(2S)-2-[[2-[4-[[4-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]piperazin-1-yl]methyl]piperidin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1R)-2-hydroxy-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](CO)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CN2CCC(CN3CCN(c4ccc(-c5cnc6[nH]cc(C(=O)c7c(F)ccc(NS(=O)(=O)N8CC[C@@H](F)C8)c7F)c6c5)cc4)CC3)CC2)C(C)(C)C)cc1	C59H70F3N11O8S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-5XPIO9	SCHEMBL22266439	(2S,4R)-1-[(2S)-2-[[2-[3-[4-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]piperazin-1-yl]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCCN2CCN(c3ccc(-c4cnc5[nH]cc(C(=O)c6c(F)ccc(NS(=O)(=O)N7CC[C@@H](F)C7)c6F)c5c4)cc3)CC2)C(C)(C)C)cc1	C56H65F3N10O8S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-447DC3	SCHEMBL22266520	(2S,4R)-1-[(2S)-2-[[2-[3-[4-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]piperazin-1-yl]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1R)-2-hydroxy-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](CO)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCCN2CCN(c3ccc(-c4cnc5[nH]cc(C(=O)c6c(F)ccc(NS(=O)(=O)N7CC[C@@H](F)C7)c6F)c5c4)cc3)CC2)C(C)(C)C)cc1	C56H65F3N10O9S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-BCS9BK	WO2018119448A1_246	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CN2CCC(CN3CCN(c4ccc(-c5cnc6[nH]cc(C(=O)c7c(F)ccc(NS(=O)(=O)CCN(C)C)c7F)c6c5)cc4)CC3)CC2)C(C)(C)C)cc1	C58H71F2N11O7S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-RK9BGZ	WO2018119448A1_247	.	Cc1ncsc1-c1ccc([C@H](CO)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CN2CC(N3CCN(c4ccc(-c5cnc6[nH]cc(C(=O)c7c(F)ccc(NS(=O)(=O)N8CC[C@@H](F)C8)c7F)c6c5)cc4)CC3)C2)C(C)(C)C)cc1	C56H64F3N11O8S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-U5ZKD7	WO2018119448A1_248	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2CC(=O)CN2C(=O)[C@@H](NC(=O)CN2CCC(C(=O)N3CCN(c4ccc(-c5cnc6[nH]cc(C(=O)c7c(F)ccc(NS(=O)(=O)N8CC[C@@H](F)C8)c7F)c6c5)cc4)CC3)CC2)C(C)(C)C)cc1	C58H64F3N11O8S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-YD26HL	SCHEMBL22266402	(2S,4R)-1-[(2S)-2-[[2-[4-[[4-[4-[3-[3-(2,3-dihydroxypropylsulfonylamino)-2,6-difluorobenzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]piperazin-1-yl]methyl]piperidin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CN2CCC(CN3CCN(c4ccc(-c5cnc6[nH]cc(C(=O)c7c(F)ccc(NS(=O)(=O)CC(O)CO)c7F)c6c5)cc4)CC3)CC2)C(C)(C)C)cc1	C57H68F2N10O9S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-WINXTD	WO2018119448A1_250	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(O)CN2CCN(CC3CCN(c4ncc(-c5cnc6[nH]cc(C(=O)c7c(F)ccc(NS(=O)(=O)N8CC[C@@H](F)C8)c7F)c6c5)cn4)CC3)CC2)C(C)(C)C)cc1	C57H70F3N13O7S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-2PI1N0	SCHEMBL22266403	(2S,4R)-1-[(2S)-2-[[2-[4-[[4-[5-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]pyrimidin-2-yl]piperazin-1-yl]methyl]piperidin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CN2CCC(CN3CCN(c4ncc(-c5cnc6[nH]cc(C(=O)c7c(F)ccc(NS(=O)(=O)N8CC[C@@H](F)C8)c7F)c6c5)cn4)CC3)CC2)C(C)(C)C)cc1	C57H68F3N13O7S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-AZ44Z7	SCHEMBL22266399	(2S,4R)-1-[(2S)-2-[[2-[2-[4-[2-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenoxy]ethyl]piperazin-1-yl]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCN2CCN(CCOc3ccc(-c4cnc5[nH]cc(C(=O)c6c(F)ccc(NS(=O)(=O)N7CC[C@@H](F)C7)c6F)c5c4)cc3)CC2)C(C)(C)C)cc1	C56H65F3N10O9S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-7GD1BV	SCHEMBL22266446	(2S,4R)-1-[(2S)-2-[[2-[3-[2-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]ethyl-methylamino]cyclobutyl]oxyacetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CO[C@H]2C[C@H](N(C)CCc3ccc(-c4cnc5[nH]cc(C(=O)c6c(F)ccc(NS(=O)(=O)N7CC[C@@H](F)C7)c6F)c5c4)cc3)C2)C(C)(C)C)cc1	C55H62F3N9O8S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-B7U64L	WO2018119448A1_254	.	Cc1ncsc1-c1ccc(CNC(=O)C2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CN2CC(N3CCC(c4ccc(-c5cnc6[nH]cc(C(=O)c7c(F)ccc(NS(=O)(=O)N8CC[C@@H](F)C8)c7F)c6c5)cc4)CC3)C2)C(C)(C)C)cc1	C56H63F3N10O7S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-KD3DT4	SCHEMBL22266444	(2S,4R)-1-[(2S)-2-[[2-[3-[[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]methyl-methylamino]cyclobutyl]oxyacetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CO[C@H]2C[C@H](N(C)Cc3ccc(-c4cnc5[nH]cc(C(=O)c6c(F)ccc(NS(=O)(=O)N7CC[C@@H](F)C7)c6F)c5c4)cc3)C2)C(C)(C)C)cc1	C54H60F3N9O8S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-KPG7UV	SCHEMBL22266445	(2S,4R)-1-[(2S)-2-[[2-[4-[[4-[5-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]pyrimidin-2-yl]piperazin-1-yl]methyl]piperidin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CN2CCC(CN3CCN(c4ncc(-c5cnc6[nH]cc(C(=O)c7c(F)ccc(NS(=O)(=O)N8CC[C@@H](F)C8)c7F)c6c5)cn4)CC3)CC2)C(C)(C)C)cc1	C56H66F3N13O7S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-XX28I7	WO2018119448A1_257	.	Cc1ncsc1C1=CC=C(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CN2CC(OCCCOc3ccc(-c4cnc5[nH]cc(C(=O)c6c(F)ccc(NS(=O)(=O)N7CC[C@@H](F)C7)c6F)c5c4)cc3)C2)C(C)(C)C)CC1	C54H62F3N9O9S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-SYG6BZ	SCHEMBL22266488	(2S,4R)-1-[(2S)-2-[[2-[3-[3-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]propoxy]azetidin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CN2CC(OCCCc3ccc(-c4cnc5[nH]cc(C(=O)c6c(F)ccc(NS(=O)(=O)N7CC[C@@H](F)C7)c6F)c5c4)cc3)C2)C(C)(C)C)cc1	C54H60F3N9O8S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-9EYFWJ	SCHEMBL22266489	(2S,4R)-1-[(2S)-2-[[2-[4-[[1-[5-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]pyrimidin-2-yl]piperidin-4-yl]methyl]piperazin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CN2CCN(CC3CCN(c4ncc(-c5cnc6[nH]cc(C(=O)c7c(F)ccc(NS(=O)(=O)N8CC[C@@H](F)C8)c7F)c6c5)cn4)CC3)CC2)C(C)(C)C)cc1	C56H66F3N13O7S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-1G5JEE	SCHEMBL22266486	(2S,4R)-1-[(2S)-2-[[2-[3-[4-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]butoxy]azetidin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CN2CC(OCCCCc3ccc(-c4cnc5[nH]cc(C(=O)c6c(F)ccc(NS(=O)(=O)N7CC[C@@H](F)C7)c6F)c5c4)cc3)C2)C(C)(C)C)cc1	C55H62F3N9O8S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-HT4HJJ	SCHEMBL22266495	(2S,4R)-1-[(2S)-2-[[2-[3-[3-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]propyl-methylamino]cyclobutyl]oxyacetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CO[C@H]2C[C@H](N(C)CCCc3ccc(-c4cnc5[nH]cc(C(=O)c6c(F)ccc(NS(=O)(=O)N7CC[C@@H](F)C7)c6F)c5c4)cc3)C2)C(C)(C)C)cc1	C56H64F3N9O8S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-OTL7W9	WO2018119448A1_262	.	Cc1ncsc1C1C=CC(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CN2CC(CCN3CCN(c4ccc(-c5cnc6[nH]cc(C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)C7F)c6c5)cc4)CC3)C2)C(C)(C)C)=CC1	C57H70F3N11O7S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-CPHG73	SCHEMBL22266497	(2S,4R)-1-[(2S)-2-[[2-[4-[2-[1-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]azetidin-3-yl]ethyl]piperazin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CN2CCN(CCC3CN(c4ccc(-c5cnc6[nH]cc(C(=O)c7c(F)ccc(NS(=O)(=O)N8CC[C@@H](F)C8)c7F)c6c5)cc4)C3)CC2)C(C)(C)C)cc1	C57H66F3N11O7S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-7GCXBZ	SCHEMBL22266498	(2S,4R)-1-[(2S)-2-[[2-[4-[[4-[5-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]pyridin-2-yl]piperazin-1-yl]methyl]piperidin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CN2CCC(CN3CCN(c4ccc(-c5cnc6[nH]cc(C(=O)c7c(F)ccc(NS(=O)(=O)N8CC[C@@H](F)C8)c7F)c6c5)cn4)CC3)CC2)C(C)(C)C)cc1	C57H67F3N12O7S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-LN2ODP	SCHEMBL22266451	(2S,4R)-1-[(2S)-2-[[2-[4-[[4-[6-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]pyridazin-3-yl]piperazin-1-yl]methyl]piperidin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CN2CCC(CN3CCN(c4ccc(-c5cnc6[nH]cc(C(=O)c7c(F)ccc(NS(=O)(=O)N8CC[C@@H](F)C8)c7F)c6c5)nn4)CC3)CC2)C(C)(C)C)cc1	C56H66F3N13O7S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-JUJZVW	SCHEMBL22266450	(2S,4R)-1-[(2S)-2-[[2-[4-[[4-[6-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]pyridin-3-yl]piperazin-1-yl]methyl]piperidin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CN2CCC(CN3CCN(c4ccc(-c5cnc6[nH]cc(C(=O)c7c(F)ccc(NS(=O)(=O)N8CC[C@@H](F)C8)c7F)c6c5)nc4)CC3)CC2)C(C)(C)C)cc1	C57H67F3N12O7S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-HVZ27F	SCHEMBL22266454	(2S,4R)-1-[(2S)-2-[[2-[4-[[4-[5-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]pyrazin-2-yl]piperazin-1-yl]methyl]piperidin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CN2CCC(CN3CCN(c4cnc(-c5cnc6[nH]cc(C(=O)c7c(F)ccc(NS(=O)(=O)N8CC[C@@H](F)C8)c7F)c6c5)cn4)CC3)CC2)C(C)(C)C)cc1	C56H66F3N13O7S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-UXIG7E	SCHEMBL22266453	(2S,4R)-1-[(2S)-2-[[2-[3-[4-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenoxy]butoxy]azetidin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CN2CC(OCCCCOc3ccc(-c4cnc5[nH]cc(C(=O)c6c(F)ccc(NS(=O)(=O)N7CC[C@@H](F)C7)c6F)c5c4)cc3)C2)C(C)(C)C)cc1	C55H62F3N9O9S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-PJKJ1L	SCHEMBL22266533	(2S,4R)-1-[(2S)-2-[[2-[3-[2-[1-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]azetidin-3-yl]oxyethyl]azetidin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CN2CC(CCOC3CN(c4ccc(-c5cnc6[nH]cc(C(=O)c7c(F)ccc(NS(=O)(=O)N8CC[C@@H](F)C8)c7F)c6c5)cc4)C3)C2)C(C)(C)C)cc1	C56H63F3N10O8S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-HRRPUN	WO2018119448A1_271	.	O=C1CCC(N2C(=O)c3cc(N4CCN(c5ccc(-n6cc(-c7ccc8c(c7)CC/C8=N\O)c(-c7ccncc7)n6)cc5)CC4)cc(OCC4CCC4)c3C2=O)C(=O)N1	C45H42N8O6	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-N38DZ5	WO2018119448A1_273	.	O=C1CCC(N2C(=O)c3cc(OCF)c(N4CCN(c5ccc(-n6cc(-c7ccc8c(c7)CC/C8=N\O)c(-c7ccncc7)n6)cc5)CC4)cc3C2=O)C(=O)N1	C41H35FN8O6	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-7SBHSW	WO2018119448A1_274	.	CCOc1cc(N2CCN(c3ccc(-n4cc(-c5ccc6c(c5)CC/C6=N\O)c(-c5ccncc5)n4)cc3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O	C42H38N8O6	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-DIDCNN	WO2018119448A1_276	.	O=C1CCC(N2C(=O)c3cc(N4CCN(c5ccc(-n6cc(-c7ccc8c(c7)CC/C8=N\O)c(-c7ccncc7)n6)cc5)CC4)cc(OCc4ccccc4)c3C2=O)C(=O)N1	C47H40N8O6	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-Z7DUXU	WO2018119448A1_277	.	O=C1CCC(N2C(=O)c3cc(N4CCN(c5ccc(-n6cc(-c7ccc8c(c7)CC/C8=N\O)c(-c7ccncc7)n6)cc5)CC4)cc(OCC4CC4)c3C2=O)C(=O)N1	C44H40N8O6	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-1ZOVYG	WO2018119448A1_278	.	CC(C)COc1cc(N2CCN(c3ccc(-n4cc(-c5ccc6c(c5)CC/C6=N\O)c(-c5ccncc5)n4)cc3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O	C44H42N8O6	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-UXF2EB	WO2018119448A1_279	.	O=C1CCC(N2C(=O)c3cc(Cl)c(N4CCN(c5ccc(-n6cc(-c7ccc8c(c7)CC/C8=N\O)c(-c7ccncc7)n6)cc5)CC4)cc3C2=O)C(=O)N1	C40H33ClN8O5	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-9455K3	WO2018119448A1_280	.	O=C1CCC(N2C(=O)c3cc(N4CCN(c5ccc(-n6cc(-c7ccc8c(c7)CC/C8=N\O)c(-c7ccncc7)n6)cc5)CC4)cc(F)c3C2=O)C(=O)N1	C40H33FN8O5	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-PXDN9M	WO2018119448A1_281	.	O=C1CCC(N2C(=O)c3cc(F)cc(N4CCN(c5ccc(-n6cc(-c7ccc8c(c7)CC/C8=N\O)c(-c7ccncc7)n6)cc5)CC4)c3C2=O)C(=O)N1	C40H33FN8O5	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-ZQCG1I	WO2018119448A1_282	.	O=C1CCC(N2C(=O)c3ccc(N4CCN(CC5CN(c6ccc(N7C=C(c8ccc9c(c8)CC/C9=N\O)C(c8ccncc8)N7)cc6)C5)CC4)cc3C2=O)C(=O)N1	C44H43N9O5	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-W7L90I	WO2018119448A1_283	.	O=C1CCC(N2Cc3cc(N4CCN(CCc5ccc(-n6cc(-c7ccc8c(c7)CC/C8=N\O)c(-c7ccncc7)n6)cc5)CC4)ccc3C2=O)C(=O)N1	C42H40N8O4	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-NOI4I6	WO2018119448A1_284	.	O=C1CCC(N2C(=O)c3ccc(O[C@H]4C[C@H](NCCc5ccc(-n6cc(-c7ccc8c(c7)CC/C8=N\O)c(-c7ccncc7)n6)cc5)C4)cc3C2=O)C(=O)N1	C42H37N7O6	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-WVSYQF	SCHEMBL20294719	(2S,4R)-1-[(2S)-2-[3-[2-[4-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]piperazin-1-yl]ethoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](c2cc(OCCN3CCN(c4ccc(-c5cnc6[nH]cc(C(=O)c7c(F)ccc(NS(=O)(=O)N8CC[C@@H](F)C8)c7F)c6c5)cc4)CC3)no2)C(C)C)cc1	C54H57F3N10O8S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-A8YAN6	CHEMBL4643114	(2S,4R)-1-[(2R)-2-[3-[2-[4-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]piperazin-1-yl]ethoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL20294559	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](c2cc(OCCN3CCN(c4ccc(-c5cnc6[nH]cc(C(=O)c7c(F)ccc(NS(=O)(=O)N8CC[C@@H](F)C8)c7F)c6c5)cc4)CC3)no2)C(C)C)cc1	C54H57F3N10O8S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-VTY20K	SCHEMBL22266534	(2S,4R)-1-[(2S)-2-[3-[3-[4-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]piperazin-1-yl]propoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](c2cc(OCCCN3CCN(c4ccc(-c5cnc6[nH]cc(C(=O)c7c(F)ccc(NS(=O)(=O)N8CC[C@@H](F)C8)c7F)c6c5)cc4)CC3)no2)C(C)C)cc1	C55H59F3N10O8S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-2XMUPC	WO2018119448A1_288	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2CC(=O)CN2C(=O)[C@@H](c2cc(OCCCN3CCN(c4ccc(-c5cnc6[nH]cc(C(=O)c7c(F)ccc(NS(=O)(=O)N8CC[C@@H](F)C8)c7F)c6c5)cc4)CC3)no2)C(C)C)cc1	C55H57F3N10O8S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-QLWYI7	WO2018119448A1_289	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOc2ccc(-n3cc(-c4ccc5c(c4)CC/C5=N\O)c(-c4ccncc4)n3)cc2)C(C)(C)C)cc1	C51H56N8O8S	BRAF	P15056	VHL	WO-2018119448-A1
TPD-3I31EK	WO2018119448A1_290	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCOc2ccc(-n3cc(-c4ccc5c(c4)CC/C5=N\O)c(-c4ccncc4)n3)cc2)C(C)(C)C)cc1	C53H60N8O9S	BRAF	P15056	VHL	WO-2018119448-A1
TPD-H1YOZO	WO2018119448A1_291	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C[C@@H](NC(=O)COCCOc2ccc(-n3cc(-c4ccc5c(c4)CC/C5=N\O)c(-c4ccncc4)n3)cc2)C(C)(C)C)cc1	C49H54N8O6S	BRAF	P15056	VHL	WO-2018119448-A1
TPD-W6C1HC	WO2018119448A1_292	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCOCCOc2ccc(N3CC(c4ccc5c(c4)CC/C5=N\O)C(c4ccncc4)N3)cc2)C(C)(C)C)cc1	C55H68N8O10S	BRAF	P15056	VHL	WO-2018119448-A1
TPD-VCVZD7	WO2018119448A1_293	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(O)COCCOCCOCCOCCOCCOc2ccc(-n3cc(-c4ccc5c(c4)CC/C5=N\O)c(-c4ccncc4)n3)cc2)C(C)(C)C)cc1	C57H70N8O11S	BRAF	P15056	VHL	WO-2018119448-A1
TPD-F79MZZ	SCHEMBL20294838	2-(2,6-dioxopiperidin-3-yl)-5-[3-[3-[4-[4-[(1E)-1-hydroxyimino-2,3-dihydroinden-5-yl]-3-pyridin-4-ylpyrazol-1-yl]phenoxy]azetidin-1-yl]azetidin-1-yl]isoindole-1,3-dione	O=C1CCC(N2C(=O)c3ccc(N4CC(N5CC(Oc6ccc(-n7cc(-c8ccc9c(c8)CC/C9=N\O)c(-c8ccncc8)n7)cc6)C5)C4)cc3C2=O)C(=O)N1	C42H36N8O6	BRAF	P15056	CRBN	WO-2018119448-A1
TPD-0Z5XMO	SCHEMBL20294807	(2S,4R)-1-[(2S)-2-[[2-[4-[[4-[4-[3-[2,6-difluoro-3-[[(3S,4S)-3-fluoro-4-hydroxypyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]piperazin-1-yl]methyl]piperidin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CN2CCC(CN3CCN(c4ccc(-c5cnc6[nH]cc(C(=O)c7c(F)ccc(NS(=O)(=O)N8C[C@H](O)[C@@H](F)C8)c7F)c6c5)cc4)CC3)CC2)C(C)(C)C)cc1	C58H68F3N11O8S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-WBFQPQ	WO2018119448A1_298	.	CCCS(=O)(=O)Nc1ccc(F)c(C(=O)c2cnnc3ncc(-c4ccc(OCC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)NCc5ccc(-c6scnc6C)cc5)C(C)(C)C)cc4)cc23)c1F	C47H48F2N8O8S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-SFM75S	SCHEMBL20294817	(2S,4R)-1-[2-[4-[3-[3-[2,6-difluoro-3-(propylsulfonylamino)benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenoxy]butanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CCCS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(-c4cccc(OCCCC(=O)NC(C(=O)N5C[C@H](O)C[C@H]5C(=O)NCc5ccc(-c6scnc6C)cc5)C(C)(C)C)c4)cc23)c1F	C49H53F2N7O8S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-VQF6FP	SCHEMBL20294552	(2S,4R)-1-[(2S)-2-[[2-[2-[3-[3-[2,6-difluoro-3-(propylsulfonylamino)benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CCCS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(-c4cccc(OCCOCC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)NCc5ccc(-c6scnc6C)cc5)C(C)(C)C)c4)cc23)c1F	C49H53F2N7O9S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-9BUITD	SCHEMBL20294691	(2S,4R)-1-[2-[4-[4-[3-[3-(butanoylamino)-2,6-difluorobenzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenoxy]butanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CCCC(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(-c4ccc(OCCCC(=O)NC(C(=O)N5C[C@H](O)C[C@H]5C(=O)NCc5ccc(-c6scnc6C)cc5)C(C)(C)C)cc4)cc23)c1F	C50H53F2N7O7S	BRAF	P15056	VHL	WO-2018119448-A1
TPD-LEFVT3	WO2018119448A1_302	.	Cc1ncsc1C1C=CC(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCOc2ccc(-c3cnc4[nH]cc(C(=O)c5c(F)ccc(N)c5F)c4c3)cc2)C(C)(C)C)=CC1	C46H49F2N7O6S	BRAF	P15056	VHL	WO-2018119448-A1
TPD-IB39AN	SCHEMBL20294613	(2S,4R)-1-[(2S)-2-[4-[4-[3-(2,6-difluorobenzoyl)-1H-pyrrolo[2,3-b]pyridin-5-yl]phenoxy]butanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCOc2ccc(-c3cnc4[nH]cc(C(=O)c5c(F)cccc5F)c4c3)cc2)C(C)(C)C)cc1	C46H46F2N6O6S	BRAF	P15056	VHL	WO-2018119448-A1
TPD-35SKA0	SCHEMBL20294648	(2S,4R)-1-[2-[4-[4-[3-[2,6-difluoro-3-(propylsulfonylamino)benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]piperazin-1-yl]butanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CCCS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(N4CCN(CCCC(=O)NC(C(=O)N5C[C@H](O)C[C@H]5C(=O)NCc5ccc(-c6scnc6C)cc5)C(C)(C)C)CC4)cc23)c1F	C47H57F2N9O7S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-SLXLDI	WO2018119448A1_305	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCOc2ccc(-c3cnc4[nH]cc(C(=O)C5C=CC=CC5)c4c3)cc2)C(C)(C)C)cc1	C46H50N6O6S	BRAF	P15056	VHL	WO-2018119448-A1
TPD-3ELN8I	SCHEMBL20294819	(2S,4R)-1-[(2S)-2-[[2-[2-[4-[3-[2,6-difluoro-3-(propylsulfonylamino)benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]piperazin-1-yl]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CCCS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(N4CCN(CCOCC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)NCc5ccc(-c6scnc6C)cc5)C(C)(C)C)CC4)cc23)c1F	C47H57F2N9O8S2	BRAF	P15056	VHL	WO-2018119448-A1
TPD-QDSUIS	SCHEMBL21906723	2-[4-[2-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperazin-1-yl]-N-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]methyl]acetamide	O=C(CN1CCN(CCOC2=CC=C(OC3=C(C4=CC=C(Br)C=C4)SC4=C3C=CC(O)=C4)C=C2)CC1)NCC1=CC2=C(C=C1)C(=O)N(C1CCC(=O)NC1=O)C2	C42H40BrN5O7S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-MCPENM	SCHEMBL21907842	3-[7-[2-[4-[2-[4-[(6-hydroxy-2-phenyl-3a,7a-dihydro-1-benzothiophen-3-yl)oxy]phenoxy]ethyl]piperazin-1-yl]ethylamino]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC=C3NCCN3CCN(CCOC4=CC=C(OC5=C(C6=CC=CC=C6)SC6C=C(O)C=CC56)C=C4)CC3)C2=O)C(=O)N1	C41H43N5O6S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-FB01AJ	SCHEMBL21906854	2-(2,6-Dioxopiperidin-3-yl)-4-[2-[4-[2-[4-[[6-hydroxy-2-(4-hydroxyphenyl)-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperazin-1-yl]ethylamino]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=C(C2=O)C(NCCN2CCN(CCOC4=CC=C(OC5=C(C6=CC=C(O)C=C6)SC6=C5C=CC(O)=C6)C=C4)CC2)=CC=C3)C(=O)N1	C41H39N5O8S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-0MLT6L	SCHEMBL21906818	3-[7-[2-[4-[2-[4-[[6-hydroxy-2-(4-hydroxyphenyl)-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperazin-1-yl]ethylamino]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC=C3NCCN3CCN(CCOC4=CC=C(OC5=C(C6=CC=C(O)C=C6)SC6=C5C=CC(O)=C6)C=C4)CC3)C2=O)C(=O)N1	C41H41N5O7S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-YJIKK4	SCHEMBL21906713	3-[7-[2-[4-[2-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperazin-1-yl]ethylamino]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC=C3NCCN3CCN(CCOC4=CC=C(OC5=C(C6=CC=C(Br)C=C6)SC6=C5C=CC(O)=C6)C=C4)CC3)C2=O)C(=O)N1	C41H40BrN5O6S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-KQOIAH	SCHEMBL21906833	4-[2-[4-[2-[4-[[2-(4-Bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperazin-1-yl]ethylamino]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=C(C2=O)C(NCCN2CCN(CCOC4=CC=C(OC5=C(C6=CC=C(Br)C=C6)SC6=C5C=CC(O)=C6)C=C4)CC2)=CC=C3)C(=O)N1	C41H38BrN5O7S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-EKE08Y	SCHEMBL21906850	3-[7-[2-[4-[2-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperazin-1-yl]ethoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC=C3OCCN3CCN(CCOC4=CC=C(OC5=C(C6=CC=C(Br)C=C6)SC6=C5C=CC(O)=C6)C=C4)CC3)C2=O)C(=O)N1	C41H39BrN4O7S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-2SNXC4	WO2018140809A1_8	.	O=C1CCC(N2CC3=CC(OCC(=O)N4CCN(CCOC5=CC=C(OC6=C(C7=CC=C(Br)C=C7)SC7=C6C=CC(O)=C7)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C41H37BrN4O8S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-UH22ZN	WO2018140809A1_9	3-[7-[[6-[[4-[2-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperazin-1-yl]methyl]pyridin-3-yl]methoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(OCC4=CC=C(CN5CCN(CCOC6=CC=C(OC7=C(C8=CC=C(Br)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)N=C4)C=CC=C3C2=O)C(=O)N1	C46H42BrN5O7S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-8TMAFP	SCHEMBL21906852	2-(2,6-Dioxopiperidin-3-yl)-4-[2-[4-[2-[4-[(6-hydroxy-2-phenyl-1-benzothiophen-3-yl)oxy]phenoxy]ethyl]piperazin-1-yl]ethylamino]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=C(C2=O)C(NCCN2CCN(CCOC4=CC=C(OC5=C(C6=CC=CC=C6)SC6=C5C=CC(O)=C6)C=C4)CC2)=CC=C3)C(=O)N1	C41H39N5O7S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-N4U6TT	SCHEMBL20425591	2-[4-[(2R)-1-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]propan-2-yl]piperazin-1-yl]-N-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]methyl]acetamide	C[C@H](COC1=CC=C(OC2=C(C3=CC=C(Br)C=C3)SC3=C2C=CC(O)=C3)C=C1)N1CCN(CC(=O)NCC2=CC3=C(C=C2)C(=O)N(C2CCC(=O)NC2=O)C3)CC1	C43H42BrN5O7S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-96I27S	SCHEMBL21907845	2-[4-[(2S)-1-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]propan-2-yl]piperazin-1-yl]-N-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]methyl]acetamide	C[C@@H](COC1=CC=C(OC2=C(C3=CC=C(Br)C=C3)SC3=C2C=CC(O)=C3)C=C1)N1CCN(CC(=O)NCC2=CC3=C(C=C2)C(=O)N(C2CCC(=O)NC2=O)C3)CC1	C43H42BrN5O7S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-BF40HK	SCHEMBL21907082	3-[7-[2-[4-[(2S)-1-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]propan-2-yl]piperazin-1-yl]ethoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C[C@@H](COC1=CC=C(OC2=C(C3=CC=C(Br)C=C3)SC3=C2C=CC(O)=C3)C=C1)N1CCN(CCOC2=CC=CC3=C2CN(C2CCC(=O)NC2=O)C3=O)CC1	C42H41BrN4O7S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-CNAQU6	SCHEMBL20423557	3-[8-[2-[4-[2-[4-[[2-(4-Bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperazin-1-yl]ethylamino]-2-methyl-4-oxoquinazolin-3-yl]piperidine-2,6-dione; SCHEMBL30480009	CC1=NC2=C(C=CC=C2NCCN2CCN(CCOC3=CC=C(OC4=C(C5=CC=C(Br)C=C5)SC5=CC(O)=CC=C54)C=C3)CC2)C(=O)N1C1CCC(=O)NC1=O	C42H41BrN6O6S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-XFXYKJ	SCHEMBL21906726	3-[7-[2-[4-[(2R)-1-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]propan-2-yl]piperazin-1-yl]ethoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C[C@H](COC1=CC=C(OC2=C(C3=CC=C(Br)C=C3)SC3=C2C=CC(O)=C3)C=C1)N1CCN(CCOC2=CC=CC3=C2CN(C2CCC(=O)NC2=O)C3=O)CC1	C42H41BrN4O7S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-CNCMLX	SCHEMBL20423260	3-[8-[2-[4-[2-[4-[[2-(4-Bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperazin-1-yl]ethoxy]-2-methyl-4-oxoquinazolin-3-yl]piperidine-2,6-dione; SCHEMBL30479953	CC1=NC2=C(C=CC=C2OCCN2CCN(CCOC3=CC=C(OC4=C(C5=CC=C(Br)C=C5)SC5=CC(O)=CC=C54)C=C3)CC2)C(=O)N1C1CCC(=O)NC1=O	C42H40BrN5O7S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-6TX9FB	SCHEMBL21907844	3-[7-[2-[2-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethoxy]ethoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC=C3OCCOCCOC3=CC=C(OC4=C(C5=CC=C(Br)C=C5)SC5=C4C=CC(O)=C5)C=C3)C2=O)C(=O)N1	C37H31BrN2O8S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-LZKLDD	WO2018140809A1_18	3-[7-[2-[2-[2-[2-[2-[4-[[2-(4-Bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethylamino]-3-oxo-1,2-dihydroinden-2-yl]piperidine-2,6-dione	O=C1CCC(C2CC3=C(NCCOCCOCCOCCOCCOC4=CC=C(OC5=C(C6=CC=C(Br)C=C6)SC6=C5C=CC(O)=C6)C=C4)C=CC=C3C2=O)C(=O)N1	C44H45BrN2O10S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-DL1VIT	SCHEMBL21906729	3-[7-[2-[2-[2-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethoxy]ethoxy]ethoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC=C3OCCOCCOCCOC3=CC=C(OC4=C(C5=CC=C(Br)C=C5)SC5=C4C=CC(O)=C5)C=C3)C2=O)C(=O)N1	C39H35BrN2O9S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-PVU2SB	WO2018140809A1_20	.	COC1=CC2=C(C=C1)C(OC1=CC=C(OCCOCCOCCOCCOCCNC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)C=C1)=C(C1=CC=C(Br)C=C1)S2	C44H44BrN3O11S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-XK5AKM	WO2018140809A1_21	.	O=C1CCC(C2CC3=C(C=CC=C3OCCOCCOCCOCCOC3=CC=C(OC4=C(C5=CC=C(Br)C=C5)SC5=C4C=CC(O)=C5)C=C3)C2=O)C(=O)N1	C42H40BrNO10S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-NBY8JE	SCHEMBL21906724	3-[7-[2-[2-[2-[2-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethoxy]ethoxy]ethoxy]ethylamino]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC=C3NCCOCCOCCOCCOC3=CC=C(OC4=C(C5=CC=C(Br)C=C5)SC5=C4C=CC(O)=C5)C=C3)C2=O)C(=O)N1	C41H40BrN3O9S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-95799B	SCHEMBL21906728	4-[2-[2-[2-[2-[4-[[2-(4-Bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethoxy]ethoxy]ethoxy]ethylamino]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=C(C2=O)C(NCCOCCOCCOCCOC2=CC=C(OC4=C(C5=CC=C(Br)C=C5)SC5=C4C=CC(O)=C5)C=C2)=CC=C3)C(=O)N1	C41H38BrN3O10S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-0T2HRH	SCHEMBL21906721	3-[7-[2-[2-[2-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethoxy]ethoxy]ethylamino]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC=C3NCCOCCOCCOC3=CC=C(OC4=C(C5=CC=C(Br)C=C5)SC5=C4C=CC(O)=C5)C=C3)C2=O)C(=O)N1	C39H36BrN3O8S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-YMTA9F	SCHEMBL21907088	3-[7-[2-[2-[2-[2-[2-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC=C3OCCOCCOCCOCCOCCOC3=CC=C(OC4=C(C5=CC=C(Br)C=C5)SC5=C4C=CC(O)=C5)C=C3)C2=O)C(=O)N1	C43H43BrN2O11S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-QLUK3D	SCHEMBL21907091	4-[2-[2-[2-[4-[[2-(4-Bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethoxy]ethoxy]ethylamino]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=C(C2=O)C(NCCOCCOCCOC2=CC=C(OC4=C(C5=CC=C(Br)C=C5)SC5=C4C=CC(O)=C5)C=C2)=CC=C3)C(=O)N1	C39H34BrN3O9S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-AE7K3C	SCHEMBL21907854	3-[7-[2-[2-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethoxy]ethylamino]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC=C3NCCOCCOC3=CC=C(OC4=C(C5=CC=C(Br)C=C5)SC5=C4C=CC(O)=C5)C=C3)C2=O)C(=O)N1	C37H32BrN3O7S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-EALAOM	WO2018140809A1_28	.	O=C1CCC(N2CC3=C(C=CC=C3OCCOC3=CC=C(OC4C5=C(C=C(O)C=C5)SC4C4=CC=C(Br)C=C4)C=C3)C2=O)C(=O)N1	C35H29BrN2O7S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-YDII27	SCHEMBL21906837	4-[2-[2-[4-[[2-(4-Bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethoxy]ethylamino]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=C(C2=O)C(NCCOCCOC2=CC=C(OC4=C(C5=CC=C(Br)C=C5)SC5=C4C=CC(O)=C5)C=C2)=CC=C3)C(=O)N1	C37H30BrN3O8S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-894GEZ	SCHEMBL21906826	3-[6-[2-[4-[2-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperazin-1-yl]ethoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(OCCN4CCN(CCOC5=CC=C(OC6=C(C7=CC=C(Br)C=C7)SC7=C6C=CC(O)=C7)C=C5)CC4)=C3)C2=O)C(=O)N1	C41H39BrN4O7S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-0YC84Q	SCHEMBL21906838	3-[7-[2-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethylamino]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC=C3NCCOC3=CC=C(OC4=C(C5=CC=C(Br)C=C5)SC5=C4C=CC(O)=C5)C=C3)C2=O)C(=O)N1	C35H28BrN3O6S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-F9B834	SCHEMBL21906732	4-[2-[4-[[2-(4-Bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethylamino]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=C(C2=O)C(NCCOC2=CC=C(OC4=C(C5=CC=C(Br)C=C5)SC5=C4C=CC(O)=C5)C=C2)=CC=C3)C(=O)N1	C35H26BrN3O7S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-KFHXD8	SCHEMBL21906865	3-[6-[2-[2-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethoxy]ethoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(OCCOCCOC4=CC=C(OC5=C(C6=CC=C(Br)C=C6)SC6=C5C=CC(O)=C6)C=C4)=C3)C2=O)C(=O)N1	C37H31BrN2O8S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-0PXFUV	SCHEMBL21906844	3-[6-[3-[4-[2-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperazin-1-yl]propoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(OCCCN4CCN(CCOC5=CC=C(OC6=C(C7=CC=C(Br)C=C7)SC7=C6C=CC(O)=C7)C=C5)CC4)=C3)C2=O)C(=O)N1	C42H41BrN4O7S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-STQAN8	SCHEMBL21906840	3-[6-[3-[3-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]propoxy]propoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(OCCCOCCCOC4=CC=C(OC5=C(C6=CC=C(Br)C=C6)SC6=C5C=CC(O)=C6)C=C4)=CC=C3C2=O)C(=O)N1	C39H35BrN2O8S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-SFJ8FM	SCHEMBL21907090	3-[6-[3-[3-[3-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]propoxy]propoxy]propoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(OCCCOCCCOCCCOC4=CC=C(OC5=C(C6=CC=C(Br)C=C6)SC6=C5C=CC(O)=C6)C=C4)=C3)C2=O)C(=O)N1	C42H41BrN2O9S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-TVVNH0	SCHEMBL21906830	3-[7-[2-[6-[2-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]-2,6-diazaspiro[3.3]heptan-2-yl]ethoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC=C3OCCN3CC4(CN(CCOC5=CC=C(OC6=C(C7=CC=C(Br)C=C7)SC7=C6C=CC(O)=C7)C=C5)C4)C3)C2=O)C(=O)N1	C42H39BrN4O7S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-1YZ24I	SCHEMBL21907081	(3S)-3-[6-[2-[(1R,4R)-5-[2-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]-2,5-diazabicyclo[2.2.1]heptan-2-yl]ethoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CC[C@H](N2CC3=C(C=CC(OCCN4C[C@H]5C[C@@H]4CN5CCOC4=CC=C(OC5=C(C6=CC=C(Br)C=C6)SC6=C5C=CC(O)=C6)C=C4)=C3)C2=O)C(=O)N1	C42H39BrN4O7S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-1HZYBC	SCHEMBL24611040	3-[6-[2-[2-[2-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethoxy]ethoxy]ethoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(OCCOCCOCCOC4=CC=C(OC5=C(C6=CC=C(Br)C=C6)SC6=C5C=CC(O)=C6)C=C4)=C3)C2=O)C(=O)N1	C39H35BrN2O9S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-9P5LXL	SCHEMBL24611041	3-[6-[3-[2-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethoxy]propoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(OCCCOCCOC4=CC=C(OC5=C(C6=CC=C(Br)C=C6)SC6=C5C=CC(O)=C6)C=C4)=C3)C2=O)C(=O)N1	C38H33BrN2O8S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-5LJA8L	WO2018140809A1_41	.	O=C1CCC(N2CC3=C(C=CC(OCCN4CC5(CN(CCOC6=CC=C(OC7=C(C8=CC=C(Br)C=C8)SC8=C7C=CC(O)=C8)C=C6)C5)C4)=C3)C2=O)C(=O)N1	C42H39BrN4O7S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-YCMWU3	SCHEMBL21906842	(3S)-3-[6-[2-[(1S,4S)-5-[2-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]-2,5-diazabicyclo[2.2.1]heptan-2-yl]ethoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CC[C@H](N2CC3=C(C=CC(OCCN4C[C@@H]5C[C@H]4CN5CCOC4=CC=C(OC5=C(C6=CC=C(Br)C=C6)SC6=C5C=CC(O)=C6)C=C4)=C3)C2=O)C(=O)N1	C42H39BrN4O7S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-UHAWWZ	SCHEMBL21906725	3-[6-[3-[2-[2-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethoxy]ethoxy]propoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(OCCCOCCOCCOC4=CC=C(OC5=C(C6=CC=C(Br)C=C6)SC6=C5C=CC(O)=C6)C=C4)=C3)C2=O)C(=O)N1	C40H37BrN2O9S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-C1IERN	SCHEMBL21907851	(3S)-3-[6-[2-[1-[2-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperidin-4-yl]oxyethoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CC[C@H](N2CC3=C(C=CC(OCCOC4CCN(CCOC5=CC=C(OC6=C(C7=CC=C(Br)C=C7)SC7=C6C=CC(O)=C7)C=C5)CC4)=C3)C2=O)C(=O)N1	C42H40BrN3O8S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-QY04QH	SCHEMBL21907838	3-[6-[3-[3-[2-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethoxy]propoxy]propoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(OCCCOCCCOCCOC4=CC=C(OC5=C(C6=CC=C(Br)C=C6)SC6=C5C=CC(O)=C6)C=C4)=C3)C2=O)C(=O)N1	C41H39BrN2O9S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-570I5N	SCHEMBL21907856	3-[6-[3-[4-[2-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperazin-1-yl]-3-oxopropyl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(CCC(=O)N4CCN(CCOC5=CC=C(OC6=C(C7=CC=C(Br)C=C7)SC7=C6C=CC(O)=C7)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C42H39BrN4O7S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-RSCIHI	SCHEMBL21907093	3-[6-[5-[4-[2-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperazin-1-yl]-5-oxopentyl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(CCCCC(=O)N4CCN(CCOC5=CC=C(OC6=C(C7=CC=C(Br)C=C7)SC7=C6C=CC(O)=C7)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C44H43BrN4O7S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-UQ6AYR	SCHEMBL24611064	3-[6-[3-[3-[4-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]butoxy]propoxy]propoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(OCCCOCCCOCCCCOC4=CC=C(OC5=C(C6=CC=C(Br)C=C6)SC6=C5C=CC(O)=C6)C=C4)=C3)C2=O)C(=O)N1	C43H43BrN2O9S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-MWBSOZ	SCHEMBL21907097	5-[4-[3-[4-[[2-(4-Bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]propyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=C(C=C(N4CCN(CCCOC5=CC=C(OC6=C(C7=CC=C(Br)C=C7)SC7=C6C=CC(O)=C7)C=C5)CC4)C=C3)C2=O)C(=O)N1	C40H35BrN4O7S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-ZURIU4	SCHEMBL21906733	3-[6-[[7-[2-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]-7-azaspiro[3.5]nonan-2-yl]oxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(OC4CC5(CCN(CCOC6=CC=C(OC7=C(C8=CC=C(Br)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)C4)=C3)C2=O)C(=O)N1	C43H40BrN3O7S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-CLTDE2	SCHEMBL21906861	5-[4-[6-[4-[[2-(4-Bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]hexyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=C(C=C(N4CCN(CCCCCCOC5=CC=C(OC6=C(C7=CC=C(Br)C=C7)SC7=C6C=CC(O)=C7)C=C5)CC4)C=C3)C2=O)C(=O)N1	C43H41BrN4O7S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-S2GIYM	SCHEMBL21907099	3-[6-[4-[5-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]pentyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCCCCOC5=CC=C(OC6=C(C7=CC=C(Br)C=C7)SC7=C6C=CC(O)=C7)C=C5)CC4)=C3)C2=O)C(=O)N1	C42H41BrN4O6S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-AO0F5E	SCHEMBL24611058	3-[6-[4-[4-[1-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]propan-2-yl]piperazin-1-yl]butyl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CC(COC1=CC=C(OC2=C(C3=CC=C(Br)C=C3)SC3=C2C=CC(O)=C3)C=C1)N1CCN(CCCCC2=CC3=C(C=C2)C(=O)N(C2CCC(=O)NC2=O)C3)CC1	C44H45BrN4O6S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-XQG2NF	SCHEMBL21906856	3-[6-[4-[6-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]hexyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCCCCCOC5=CC=C(OC6=C(C7=CC=C(Br)C=C7)SC7=C6C=CC(O)=C7)C=C5)CC4)=C3)C2=O)C(=O)N1	C43H43BrN4O6S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-FS88J7	SCHEMBL20442634	3-[6-[4-[2-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCOC5=CC=C(OC6=C(C7=CC=C(Br)C=C7)SC7=C6C=CC(O)=C7)C=C5)CC4)=C3)C2=O)C(=O)N1	C39H35BrN4O6S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-T4EXHS	SCHEMBL21906835	5-[4-[2-[4-[[2-(4-Bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=C(C=C(N4CCN(CCOC5=CC=C(OC6=C(C7=CC=C(Br)C=C7)SC7=C6C=CC(O)=C7)C=C5)CC4)C=C3)C2=O)C(=O)N1	C39H33BrN4O7S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-9N60HD	SCHEMBL21907848	1-[2-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]-N-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]methyl]piperidine-4-carboxamide	O=C1CCC(N2CC3=C(C=CC(CNC(=O)C4CCN(CCOC5=CC=C(OC6=C(C7=CC=C(Br)C=C7)SC7=C6C=CC(O)=C7)C=C5)CC4)=C3)C2=O)C(=O)N1	C42H39BrN4O7S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-O4TSYS	WO2018140809A1_58	.	O=C1CCC(N2CC3=C(CCC(N4CCN(CCCCOC5=CC=C(OC6=C(C7=CC=C(Br)C=C7)SC7=C6C=CC(O)=C7)C=C5)CC4)=C3)C2=O)C(=O)N1	C41H41BrN4O6S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-EGEBVL	SCHEMBL21907096	3-[6-[4-[3-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]propyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCCOC5=CC=C(OC6=C(C7=CC=C(Br)C=C7)SC7=C6C=CC(O)=C7)C=C5)CC4)=C3)C2=O)C(=O)N1	C40H37BrN4O6S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-JHVDO7	SCHEMBL21906849	5-[4-[4-[4-[[2-(4-Bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]butyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=C(C=C(N4CCN(CCCCOC5=CC=C(OC6=C(C7=CC=C(Br)C=C7)SC7=C6C=CC(O)=C7)C=C5)CC4)C=C3)C2=O)C(=O)N1	C41H37BrN4O7S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-45VYEK	WO2018140809A1_61	.	COC1=CC2=C(C=C1)C(OC1=CC=C(OCCCCCN3CCN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)C=C1)=C(C1=CC=C(Br)C=C1)S2	C43H41BrN4O7S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-H476TB	SCHEMBL21906863	5-[2-[1-[2-[4-[[2-(4-Bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperidin-4-yl]ethylamino]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=C(C=C(NCCC4CCN(CCOC5=CC=C(OC6=C(C7=CC=C(Br)C=C7)SC7=C6C=CC(O)=C7)C=C5)CC4)C=C3)C2=O)C(=O)N1	C42H39BrN4O7S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-YWJMR8	SCHEMBL21907852	2-[1-[2-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperidin-4-yl]-N-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]methyl]acetamide	O=C(CC1CCN(CCOC2=CC=C(OC3=C(C4=CC=C(Br)C=C4)SC4=C3C=CC(O)=C4)C=C2)CC1)NCC1=CC2=C(C=C1)C(=O)N(C1CCC(=O)NC1=O)C2	C43H41BrN4O7S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-M5N0E6	SCHEMBL21907849	3-[6-[3-[1-[2-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperidin-4-yl]propylamino]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(NCCCC4CCN(CCOC5=CC=C(OC6=C(C7=CC=C(Br)C=C7)SC7=C6C=CC(O)=C7)C=C5)CC4)=C3)C2=O)C(=O)N1	C43H43BrN4O6S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-38RUGX	SCHEMBL21906839	3-[6-[2-[1-[2-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperidin-4-yl]ethylamino]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(NCCC4CCN(CCOC5=CC=C(OC6=C(C7=CC=C(Br)C=C7)SC7=C6C=CC(O)=C7)C=C5)CC4)=C3)C2=O)C(=O)N1	C42H41BrN4O6S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-PK8X21	SCHEMBL21907098	5-[2-[2-[4-[[2-(4-Bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethoxy]ethoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=C(C=C(OCCOCCOC4=CC=C(OC5=C(C6=CC=C(Br)C=C6)SC6=C5C=CC(O)=C6)C=C4)C=C3)C2=O)C(=O)N1	C37H29BrN2O9S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-MDVLC2	SCHEMBL21906857	5-[2-[2-[2-[4-[[2-(4-Bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethoxy]ethoxy]ethylamino]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=C(C=C(NCCOCCOCCOC4=CC=C(OC5=C(C6=CC=C(Br)C=C6)SC6=C5C=CC(O)=C6)C=C4)C=C3)C2=O)C(=O)N1	C39H34BrN3O9S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-I0RMNV	SCHEMBL21906735	5-[3-[1-[2-[4-[[2-(4-Bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperidin-4-yl]propylamino]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=C(C=C(NCCCC4CCN(CCOC5=CC=C(OC6=C(C7=CC=C(Br)C=C7)SC7=C6C=CC(O)=C7)C=C5)CC4)C=C3)C2=O)C(=O)N1	C43H41BrN4O7S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-R000O1	SCHEMBL21906858	5-[4-[7-[4-[[2-(4-Bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]heptyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=C(C=C(N4CCN(CCCCCCCOC5=CC=C(OC6=C(C7=CC=C(Br)C=C7)SC7=C6C=CC(O)=C7)C=C5)CC4)C=C3)C2=O)C(=O)N1	C44H43BrN4O7S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-R4YPMJ	SCHEMBL20442579	5-[3-[1-[2-[4-[[2-(4-Bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperidin-4-yl]oxypropyl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=C(C=C(CCCOC4CCN(CCOC5=CC=C(OC6=C(C7=CC=C(Br)C=C7)SC7=C6C=CC(O)=C7)C=C5)CC4)C=C3)C2=O)C(=O)N1	C43H40BrN3O8S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-8XCOSH	SCHEMBL21907101	3-[6-[2-[2-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethoxy]ethylamino]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(NCCOCCOC4=CC=C(OC5=C(C6=CC=C(Br)C=C6)SC6=C5C=CC(O)=C6)C=C4)=C3)C2=O)C(=O)N1	C37H32BrN3O7S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-9KK8VX	SCHEMBL21907102	3-[6-[3-[1-[2-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperidin-4-yl]oxypropyl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(CCCOC4CCN(CCOC5=CC=C(OC6=C(C7=CC=C(Br)C=C7)SC7=C6C=CC(O)=C7)C=C5)CC4)=C3)C2=O)C(=O)N1	C43H42BrN3O7S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-ZK20M9	SCHEMBL21907100	3-[6-[3-[4-[2-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]-1,4-diazepan-1-yl]propylamino]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(NCCCN4CCCN(CCOC5=CC=C(OC6=C(C7=CC=C(Br)C=C7)SC7=C6C=CC(O)=C7)C=C5)CC4)=C3)C2=O)C(=O)N1	C43H44BrN5O6S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-2JKSGQ	SCHEMBL21906737	5-[2-[2-[4-[[2-(4-Bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethoxy]ethylamino]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC=C(NCCOCCOC4=CC=C(OC5=C(C6=CC=C(Br)C=C6)SC6=C5C=CC(O)=C6)C=C4)C=C3C2=O)C(=O)N1	C37H30BrN3O8S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-IH96HJ	WO2018140809A1_76	.	O=C1CCC(N2C(=O)C3=C(C=C(OCCCOCCOC4=CC=C(OC5=C(C6=CC=C(Br)C=C6)SC6=C5C=CC(O)=C6)C=C4)N=C3)C2=O)C(=O)N1	C37H30BrN3O9S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-7Y7FK9	SCHEMBL21906859	5-[3-[3-[4-[[2-(4-Bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]propoxy]propoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=C(C=C(OCCCOCCCOC4=CC=C(OC5=C(C6=CC=C(Br)C=C6)SC6=C5C=CC(O)=C6)C=C4)C=C3)C2=O)C(=O)N1	C39H33BrN2O9S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-YZQT2S	SCHEMBL24654389	5-[2-[2-[2-[4-[[2-(4-Bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethoxy]ethoxy]ethoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC=C(OCCOCCOCCOC4=CC=C(OC5=C(C6=CC=C(Br)C=C6)SC6=C5C=CC(O)=C6)C=C4)C=C3C2=O)C(=O)N1	C39H33BrN2O10S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-NM316B	SCHEMBL21907092	5-[3-[2-[2-[4-[[2-(4-Bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethoxy]ethoxy]propoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=C(C=C(OCCCOCCOCCOC4=CC=C(OC5=C(C6=CC=C(Br)C=C6)SC6=C5C=CC(O)=C6)C=C4)C=C3)C2=O)C(=O)N1	C40H35BrN2O10S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-0BX4BQ	WO2018140809A1_80	.	O=C1CCC(C2C(=O)C3=CC=C(OCCCOCCCOCCCOC4=CC=C(OC5C6=C(C=C(O)C=C6)SC5C5=CC=C(Br)C=C5)C=C4)C=C3C2=O)C(=O)N1	C43H42BrNO10S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-7EDRMF	SCHEMBL21906871	5-[3-[2-[4-[[2-(4-Bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethoxy]propylamino]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=C(C=C(NCCCOCCOC4=CC=C(OC5=C(C6=CC=C(Br)C=C6)SC6=C5C=CC(O)=C6)C=C4)C=C3)C2=O)C(=O)N1	C38H32BrN3O8S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-RAJ0E0	SCHEMBL21906731	5-[3-[3-[4-[[2-(4-Bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]propoxy]propylamino]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC=C(NCCCOCCCOC4=CC=C(OC5=C(C6=CC=C(Br)C=C6)SC6=C5C=CC(O)=C6)C=C4)C=C3C2=O)C(=O)N1	C39H34BrN3O8S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-0VJSAA	SCHEMBL21907087	5-[3-[2-[2-[4-[[2-(4-Bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethoxy]ethoxy]propylamino]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC=C(NCCCOCCOCCOC4=CC=C(OC5=C(C6=CC=C(Br)C=C6)SC6=C5C=CC(O)=C6)C=C4)C=C3C2=O)C(=O)N1	C40H36BrN3O9S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-0XW9WT	SCHEMBL21906866	5-[3-[3-[3-[4-[[2-(4-Bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]propoxy]propoxy]propylamino]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC=C(NCCCOCCCOCCCOC4=CC=C(OC5=C(C6=CC=C(Br)C=C6)SC6=C5C=CC(O)=C6)C=C4)C=C3C2=O)C(=O)N1	C42H40BrN3O9S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-CZVO2E	SCHEMBL21907104	3-[6-[3-[2-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethoxy]propylamino]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(NCCCOCCOC4=CC=C(OC5=C(C6=CC=C(Br)C=C6)SC6=C5C=CC(O)=C6)C=C4)=C3)C2=O)C(=O)N1	C38H34BrN3O7S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-WR7NDP	SCHEMBL21906870	3-[6-[2-[2-[2-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethoxy]ethoxy]ethylamino]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(NCCOCCOCCOC4=CC=C(OC5=C(C6=CC=C(Br)C=C6)SC6=C5C=CC(O)=C6)C=C4)=CC=C3C2=O)C(=O)N1	C39H36BrN3O8S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-O3T5C8	SCHEMBL21906845	5-[3-[3-[2-[4-[[2-(4-Bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethoxy]propoxy]propoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC=C(OCCCOCCCOCCOC4=CC=C(OC5=C(C6=CC=C(Br)C=C6)SC6=C5C=CC(O)=C6)C=C4)C=C3C2=O)C(=O)N1	C41H37BrN2O10S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-T90AWW	SCHEMBL21907853	3-[6-[3-[3-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]propoxy]propylamino]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(NCCCOCCCOC4=CC=C(OC5=C(C6=CC=C(Br)C=C6)SC6=C5C=CC(O)=C6)C=C4)=CC=C3C2=O)C(=O)N1	C39H36BrN3O7S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-4SHHXD	SCHEMBL21906864	3-[6-[3-[3-[2-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethoxy]propoxy]propylamino]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(NCCCOCCCOCCOC4=CC=C(OC5=C(C6=CC=C(Br)C=C6)SC6=C5C=CC(O)=C6)C=C4)=CC=C3C2=O)C(=O)N1	C41H40BrN3O8S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-SLW21J	SCHEMBL20442652	5-[3-[3-[4-[4-[[2-(4-Bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]butoxy]propoxy]propoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC=C(OCCCOCCCOCCCCOC4=CC=C(OC5=C(C6=CC=C(Br)C=C6)SC6=C5C=CC(O)=C6)C=C4)C=C3C2=O)C(=O)N1	C43H41BrN2O10S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-BTMQTQ	SCHEMBL20442618	5-[3-[3-[2-[4-[[2-(4-Bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethoxy]propoxy]propylamino]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC=C(NCCCOCCCOCCOC4=CC=C(OC5=C(C6=CC=C(Br)C=C6)SC6=C5C=CC(O)=C6)C=C4)C=C3C2=O)C(=O)N1	C41H38BrN3O9S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-P398VP	SCHEMBL20442656	5-[3-[3-[4-[4-[[2-(4-Bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]butoxy]propoxy]propylamino]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC=C(NCCCOCCCOCCCCOC4=CC=C(OC5=C(C6=CC=C(Br)C=C6)SC6=C5C=CC(O)=C6)C=C4)C=C3C2=O)C(=O)N1	C43H42BrN3O9S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-R8X16T	SCHEMBL20442655	3-[6-[3-[3-[4-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]butoxy]propoxy]propylamino]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(NCCCOCCCOCCCCOC4=CC=C(OC5=C(C6=CC=C(Br)C=C6)SC6=C5C=CC(O)=C6)C=C4)=CC=C3C2=O)C(=O)N1	C43H44BrN3O8S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-CRPSX6	SCHEMBL20442622	3-[6-[3-[3-[3-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]propoxy]propoxy]propylamino]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(NCCCOCCCOCCCOC4=CC=C(OC5=C(C6=CC=C(Br)C=C6)SC6=C5C=CC(O)=C6)C=C4)=CC=C3C2=O)C(=O)N1	C42H42BrN3O8S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-GT89OF	SCHEMBL20442617	3-[6-[3-[2-[2-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethoxy]ethoxy]propylamino]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(NCCCOCCOCCOC4=CC=C(OC5=C(C6=CC=C(Br)C=C6)SC6=C5C=CC(O)=C6)C=C4)=CC=C3C2=O)C(=O)N1	C40H38BrN3O8S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-1LPD88	SCHEMBL20442653	5-[3-[4-[2-[4-[[2-(4-Bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperazin-1-yl]propylamino]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC=C(NCCCN4CCN(CCOC5=CC=C(OC6=C(C7=CC=C(Br)C=C7)SC7=C6C=CC(O)=C7)C=C5)CC4)C=C3C2=O)C(=O)N1	C42H40BrN5O7S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-75IJL3	SCHEMBL20442771	5-[3-[4-[2-[4-[[2-(4-Bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]-1,4-diazepan-1-yl]propylamino]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC=C(NCCCN4CCCN(CCOC5=CC=C(OC6=C(C7=CC=C(Br)C=C7)SC7=C6C=CC(O)=C7)C=C5)CC4)C=C3C2=O)C(=O)N1	C43H42BrN5O7S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-1IMV9C	SCHEMBL20442657	3-[6-[3-[4-[2-[4-[[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperazin-1-yl]propylamino]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(NCCCN4CCN(CCOC5=CC=C(OC6=C(C7=CC=C(F)C=C7)SC7=C6C=CC(O)=C7)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C42H42FN5O6S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-PXORJN	SCHEMBL20442747	3-[6-[3-[4-[2-[4-[[6-hydroxy-2-[4-(trifluoromethyl)phenyl]-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperazin-1-yl]propylamino]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; LUFHLYAAJHDSPC-UHFFFAOYSA-N; 3-[6-[3-[4-[2-[4-[[6-hydroxy-2-[4-(trifluoromethyl)phenyl]-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperazin-1-yl]propylamino]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(NCCCN4CCN(CCOC5=CC=C(OC6=C(C7=CC=C(C(F)(F)F)C=C7)SC7=C6C=CC(O)=C7)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C43H42F3N5O6S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-13VO8W	SCHEMBL21906742	3-[6-[3-[4-[2-[4-[[6-hydroxy-2-(4-methoxyphenyl)-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperazin-1-yl]propylamino]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	COC1=CC=C(C2=C(OC3=CC=C(OCCN4CCN(CCCNC5=CC=C6C(=O)N(C7CCC(=O)NC7=O)CC6=C5)CC4)C=C3)C3=C(C=C(O)C=C3)S2)C=C1	C43H45N5O7S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-PF9VHP	SCHEMBL21906743	5-[3-[4-[3-[4-[[2-(4-Bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenyl]propyl]piperazin-1-yl]propylamino]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC=C(NCCCN4CCN(CCCC5=CC=C(OC6=C(C7=CC=C(Br)C=C7)SC7=C6C=CC(O)=C7)C=C5)CC4)C=C3C2=O)C(=O)N1	C43H42BrN5O6S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-MCDDBC	SCHEMBL21906875	5-[3-[4-[3-[4-[[2-(4-Bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenyl]propyl]-1,4-diazepan-1-yl]propylamino]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC=C(NCCCN4CCCN(CCCC5=CC=C(OC6=C(C7=CC=C(Br)C=C7)SC7=C6C=CC(O)=C7)C=C5)CC4)C=C3C2=O)C(=O)N1	C44H44BrN5O6S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-64PM2V	SCHEMBL21906874	5-[3-[4-[4-[[2-(4-Bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenyl]piperidin-1-yl]propylamino]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC=C(NCCCN4CCC(C5=CC=C(OC6=C(C7=CC=C(Br)C=C7)SC7=C6C=CC(O)=C7)C=C5)CC4)C=C3C2=O)C(=O)N1	C41H37BrN4O6S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-P4XU04	SCHEMBL21907855	5-[4-[4-[4-[[2-(4-Bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenyl]piperidin-1-yl]butylamino]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC=C(NCCCCN4CCC(C5=CC=C(OC6=C(C7=CC=C(Br)C=C7)SC7=C6C=CC(O)=C7)C=C5)CC4)C=C3C2=O)C(=O)N1	C42H39BrN4O6S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-OE0LA4	SCHEMBL21906877	3-[6-[3-[4-[3-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenyl]propyl]piperazin-1-yl]propylamino]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(NCCCN4CCN(CCCC5=CC=C(OC6=C(C7=CC=C(Br)C=C7)SC7=C6C=CC(O)=C7)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C43H44BrN5O5S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-12HLN7	SCHEMBL21907861	3-[6-[3-[4-[3-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenyl]propyl]-1,4-diazepan-1-yl]propylamino]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(NCCCN4CCCN(CCCC5=CC=C(OC6=C(C7=CC=C(Br)C=C7)SC7=C6C=CC(O)=C7)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C44H46BrN5O5S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-BXJMP4	SCHEMBL21906876	3-[6-[3-[4-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenyl]piperidin-1-yl]propylamino]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(NCCCN4CCC(C5=CC=C(OC6=C(C7=CC=C(Br)C=C7)SC7=C6C=CC(O)=C7)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C41H39BrN4O5S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-NGYTR6	SCHEMBL21906741	3-[6-[5-[4-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenyl]piperidin-1-yl]pentylamino]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(NCCCCCN4CCC(C5=CC=C(OC6=C(C7=CC=C(Br)C=C7)SC7=C6C=CC(O)=C7)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C43H43BrN4O5S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-A341VQ	SCHEMBL21906879	3-[6-[2-[4-[4-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]butyl]-1,4-diazepan-1-yl]ethyl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(CCN4CCCN(CCCCOC5=CC=C(OC6=C(C7=CC=C(Br)C=C7)SC7=C6C=CC(O)=C7)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C44H45BrN4O6S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-AJ4J6F	SCHEMBL21907103	3-[6-[2-[4-[5-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenyl]pentyl]-1,4-diazepan-1-yl]ethyl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(CCN4CCCN(CCCCCC5=CC=C(OC6=C(C7=CC=C(Br)C=C7)SC7=C6C=CC(O)=C7)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C45H47BrN4O5S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-JDHOBJ	SCHEMBL20442627	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[2-[4-[[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOC3=CC=C(OC4=C(C5=CC=C(F)C=C5)SC5=C4C=CC(O)=C5)C=C3)C(C)(C)C)C=C2)SC=N1	C51H57FN4O10S2	ERα;ERβ	P03372/Q92731	VHL	WO-2018140809-A1
TPD-OT3D8O	SCHEMBL20442628	(2S,4R)-1-[(2S)-2-[[2-[3-[3-[4-[[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]propoxy]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCOCCCOC3=CC=C(OC4=C(C5=CC=C(F)C=C5)SC5=C4C=CC(O)=C5)C=C3)C(C)(C)C)C=C2)SC=N1	C51H57FN4O9S2	ERα;ERβ	P03372/Q92731	VHL	WO-2018140809-A1
TPD-5UALFP	SCHEMBL20442626	(2S,4R)-1-[(2S)-2-[[2-[2-[3-[4-[[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]propoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCCOC3=CC=C(OC4=C(C5=CC=C(F)C=C5)SC5=C4C=CC(O)=C5)C=C3)C(C)(C)C)C=C2)SC=N1	C50H55FN4O9S2	ERα;ERβ	P03372/Q92731	VHL	WO-2018140809-A1
TPD-4MIDRN	WO2018140809A1_114	.	CC1=C(C2=CC=C(CNC(=O)C3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCC(=O)N3CCN(CCOC4=CC=C(OC5=C(C6=CC=C(F)C=C6)SC6=C5C=CC(O)=C6)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C53H59FN6O8S2	ERα;ERβ	P03372/Q92731	VHL	WO-2018140809-A1
TPD-204GEE	SCHEMBL20442548	(2S,4R)-1-[(2S)-2-[[4-[2-[2-[4-[[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-5-yl]-4-oxobutanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCC(=O)N3CC4CN(CCOC5=CC=C(OC6=C(C7=CC=C(F)C=C7)SC7=C6C=CC(O)=C7)C=C5)CC4C3)C(C)(C)C)C=C2)SC=N1	C54H59FN6O8S2	ERα;ERβ	P03372/Q92731	VHL	WO-2018140809-A1
TPD-8B0F7P	SCHEMBL20442546	(2S,4R)-1-[(2S)-2-[[2-[2-[(3R)-1-[2-[4-[[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]pyrrolidin-3-yl]oxyethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCO[C@@H]3CCN(CCOC4=CC=C(OC5=C(C6=CC=C(F)C=C6)SC6=C5C=CC(O)=C6)C=C4)C3)C(C)(C)C)C=C2)SC=N1	C52H58FN5O9S2	ERα;ERβ	P03372/Q92731	VHL	WO-2018140809-A1
TPD-TJBFJ4	SCHEMBL20442549	(2S,4R)-1-[(2S)-2-[[2-[2-[1-[2-[4-[[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]azetidin-3-yl]oxyethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOC3CN(CCOC4=CC=C(OC5=C(C6=CC=C(F)C=C6)SC6=C5C=CC(O)=C6)C=C4)C3)C(C)(C)C)C=C2)SC=N1	C51H56FN5O9S2	ERα;ERβ	P03372/Q92731	VHL	WO-2018140809-A1
TPD-G9TER5	SCHEMBL20442547	(2S,4R)-1-[(2S)-2-[[2-[2-[4-[2-[4-[[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperazin-1-yl]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCN3CCN(CCOC4=CC=C(OC5=C(C6=CC=C(F)C=C6)SC6=C5C=CC(O)=C6)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C52H59FN6O8S2	ERα;ERβ	P03372/Q92731	VHL	WO-2018140809-A1
TPD-S0J9YX	WO2018140809A1_119	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOC3=CC=C(OC4=C(C5=CC=C(CI)C=C5)SC5=C4C=CC(O)=C5)C=C3)C(C)(C)C)C=C2)SC=N1	C52H59IN4O10S2	ERα;ERβ	P03372/Q92731	VHL	WO-2018140809-A1
TPD-ZGE92C	WO2018140809A1_120	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOC3=CC=C(OC4=C(C5=CC=C(CI)C=C5)SC5=C4C=CC(O)=C5)C=C3)C(C)(C)C)C=C2)OC=N1	C52H59IN4O11S	ERα;ERβ	P03372/Q92731	VHL	WO-2018140809-A1
TPD-DBF5U9	SCHEMBL20425491	(2S,4R)-1-[(2S)-2-[[2-[4-[1-[2-[4-[[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]pyrazol-3-yl]phenyl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CC3=CC=C(C4=NN(CCOC5=CC=C(OC6=C(C7=CC=C(F)C=C7)SC7=C6C=CC(O)=C7)C=C5)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C55H53FN6O7S2	ERα;ERβ	P03372/Q92731	VHL	WO-2018140809-A1
TPD-8A8G6W	SCHEMBL20442474	(2S,4R)-1-[(2S)-2-[4-[5-[2-[4-[[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-2-yl]butanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCN3CC4CN(CCOC5=CC=C(OC6=C(C7=CC=C(F)C=C7)SC7=C6C=CC(O)=C7)C=C5)CC4C3)C(C)(C)C)C=C2)SC=N1	C54H61FN6O7S2	ERα;ERβ	P03372/Q92731	VHL	WO-2018140809-A1
TPD-2KBT4K	SCHEMBL20442478	(2S,4R)-1-[(2S)-2-[[2-[2-[(3S)-1-[2-[4-[[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]pyrrolidin-3-yl]oxyethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCO[C@H]3CCN(CCOC4=CC=C(OC5=C(C6=CC=C(F)C=C6)SC6=C5C=CC(O)=C6)C=C4)C3)C(C)(C)C)C=C2)SC=N1	C52H58FN5O9S2	ERα;ERβ	P03372/Q92731	VHL	WO-2018140809-A1
TPD-0YXV0F	SCHEMBL20442475	(2S,4R)-1-[(2S)-2-[[5-[(3S)-4-[2-[4-[[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]-3-methylpiperazin-1-yl]-5-oxopentanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCC(=O)N3CCN(CCOC4=CC=C(OC5=C(C6=CC=C(F)C=C6)SC6=C5C=CC(O)=C6)C=C4)[C@@H](C)C3)C(C)(C)C)C=C2)SC=N1	C54H61FN6O8S2	ERα;ERβ	P03372/Q92731	VHL	WO-2018140809-A1
TPD-S777RS	SCHEMBL20442477	(2S,4R)-1-[(2S)-2-[[5-[(3R)-4-[2-[4-[[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]-3-methylpiperazin-1-yl]-5-oxopentanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCC(=O)N3CCN(CCOC4=CC=C(OC5=C(C6=CC=C(F)C=C6)SC6=C5C=CC(O)=C6)C=C4)[C@H](C)C3)C(C)(C)C)C=C2)SC=N1	C54H61FN6O8S2	ERα;ERβ	P03372/Q92731	VHL	WO-2018140809-A1
TPD-ZCAWYI	SCHEMBL20442594	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[2-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOC3=CC=C(OC4=C(C5=CC=C(Br)C=C5)SC5=C4C=CC(O)=C5)C=C3)C(C)(C)C)C=C2)SC=N1	C51H57BrN4O10S2	ERα;ERβ	P03372/Q92731	VHL	WO-2018140809-A1
TPD-9KGQXP	SCHEMBL20442595	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[2-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-oxazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOC3=CC=C(OC4=C(C5=CC=C(Br)C=C5)SC5=C4C=CC(O)=C5)C=C3)C(C)(C)C)C=C2)OC=N1	C51H57BrN4O11S	ERα;ERβ	P03372/Q92731	VHL	WO-2018140809-A1
TPD-8A21CC	SCHEMBL20442593	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[2-[4-[[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl-methylamino]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCN(C)CCOC3=CC=C(OC4=C(C5=CC=C(F)C=C5)SC5=C4C=CC(O)=C5)C=C3)C(C)(C)C)C=C2)SC=N1	C52H60FN5O9S2	ERα;ERβ	P03372/Q92731	VHL	WO-2018140809-A1
TPD-B4JCPC	SCHEMBL20442596	(2S,4R)-N-[(1S)-1-(4-chlorophenyl)ethyl]-1-[(2S)-2-[[2-[2-[2-[2-[4-[[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl-methylamino]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide	C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](NC(=O)COCCOCCN(C)CCOC1=CC=C(OC2=C(C3=CC=C(F)C=C3)SC3=C2C=CC(O)=C3)C=C1)C(C)(C)C)C1=CC=C(Cl)C=C1	C48H56ClFN4O9S	ERα;ERβ	P03372/Q92731	VHL	WO-2018140809-A1
TPD-T8414J	SCHEMBL20442597	(2S,4R)-1-[(2S)-2-[3-[3-[1-[2-[4-[[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]pyrazol-3-yl]phenyl]propanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCC3=CC(C4=NN(CCOC5=CC=C(OC6=C(C7=CC=C(F)C=C7)SC7=C6C=CC(O)=C7)C=C5)C=C4)=CC=C3)C(C)(C)C)C=C2)SC=N1	C56H55FN6O7S2	ERα;ERβ	P03372/Q92731	VHL	WO-2018140809-A1
TPD-X788FF	SCHEMBL20442598	(2S,4R)-1-[(2S)-2-[4-[[1-[2-[4-[[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]pyrrolidin-3-yl]methoxy]butanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCOCC3CCN(CCOC4=CC=C(OC5=C(C6=CC=C(F)C=C6)SC6=C5C=CC(O)=C6)C=C4)C3)C(C)(C)C)C=C2)SC=N1	C53H60FN5O8S2	ERα;ERβ	P03372/Q92731	VHL	WO-2018140809-A1
TPD-CFTKQF	SCHEMBL20442761	(2S,4R)-N-[(1S)-1-(4-cyanophenyl)ethyl]-1-[(2S)-2-[[2-[2-[2-[2-[4-[[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide	C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](NC(=O)COCCOCCOCCOC1=CC=C(OC2=C(C3=CC=C(F)C=C3)SC3=C2C=CC(O)=C3)C=C1)C(C)(C)C)C1=CC=C(C#N)C=C1	C48H53FN4O10S	ERα;ERβ	P03372/Q92731	VHL	WO-2018140809-A1
TPD-Y6T5O2	SCHEMBL20442760	(2S,4R)-1-[(2S)-2-[[2-[4-[6-[4-[[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenyl]pyridin-3-yl]oxybutoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCOC3=CN=C(C4=CC=C(OC5=C(C6=CC=C(F)C=C6)SC6=C5C=CC(O)=C6)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C53H54FN5O8S2	ERα;ERβ	P03372/Q92731	VHL	WO-2018140809-A1
TPD-V4FXD5	SCHEMBL20442763	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[4-[4-[[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenyl]-2-oxopyridin-1-yl]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCN3C=CC(C4=CC=C(OC5=C(C6=CC=C(F)C=C6)SC6=C5C=CC(O)=C6)C=C4)=CC3=O)C(C)(C)C)C=C2)SC=N1	C53H54FN5O9S2	ERα;ERβ	P03372/Q92731	VHL	WO-2018140809-A1
TPD-L7CRWR	SCHEMBL20442762	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[4-[4-[[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenyl]piperidin-1-yl]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCN3CCC(C4=CC=C(OC5=C(C6=CC=C(F)C=C6)SC6=C5C=CC(O)=C6)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C53H60FN5O8S2	ERα;ERβ	P03372/Q92731	VHL	WO-2018140809-A1
TPD-OSL9PX	SCHEMBL20442759	(2S,4R)-N-[(4-cyanophenyl)methyl]-1-[(2S)-2-[[2-[2-[2-[2-[4-[[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide	CC(C)(C)[C@H](NC(=O)COCCOCCOCCOC1=CC=C(OC2=C(C3=CC=C(F)C=C3)SC3=C2C=CC(O)=C3)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C#N)C=C1	C47H51FN4O10S	ERα;ERβ	P03372/Q92731	VHL	WO-2018140809-A1
TPD-TQLABD	SCHEMBL20442758	(2S,4R)-1-[(2S)-2-[4-[1-[2-[4-[[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperidin-4-yl]oxybutanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCOC3CCN(CCOC4=CC=C(OC5=C(C6=CC=C(F)C=C6)SC6=C5C=CC(O)=C6)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C53H60FN5O8S2	ERα;ERβ	P03372/Q92731	VHL	WO-2018140809-A1
TPD-9AXXSF	SCHEMBL20442610	(2S,4R)-4-hydroxy-1-[(2S)-2-[[2-[2-[2-[2-[4-[(6-hydroxy-2-phenyl-1-benzothiophen-3-yl)oxy]phenoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-oxazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOC3=CC=C(OC4=C(C5=CC=CC=C5)SC5=C4C=CC(O)=C5)C=C3)C(C)(C)C)C=C2)OC=N1	C51H58N4O11S	ERα;ERβ	P03372/Q92731	VHL	WO-2018140809-A1
TPD-LS05XX	SCHEMBL20442611	(2S,4R)-1-[(2S)-2-[[2-[3-[2-[2-[4-[[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl-methylamino]ethyl]phenoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COC3=CC(CCN(C)CCOC4=CC=C(OC5=C(C6=CC=C(F)C=C6)SC6=C5C=CC(O)=C6)C=C4)=CC=C3)C(C)(C)C)C=C2)SC=N1	C55H58FN5O8S2	ERα;ERβ	P03372/Q92731	VHL	WO-2018140809-A1
TPD-UZPVZ7	SCHEMBL20425344	(2S,4R)-1-[(2S)-2-[[2-[2-[4-[2-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperazin-1-yl]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCN3CCN(CCOC4=CC=C(OC5=C(C6=CC=C(Br)C=C6)SC6=C5C=CC(O)=C6)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C52H59BrN6O8S2	ERα;ERβ	P03372/Q92731	VHL	WO-2018140809-A1
TPD-NYSER3	SCHEMBL20442613	(2S,4R)-1-[(2S)-2-[[2-[4-[1-[2-[4-[[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]pyrazol-3-yl]phenyl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CC3=CC=C(C4=NN(CCOC5=CC=C(OC6=C(C7=CC=C(F)C=C7)SC7=C6C=CC(O)=C7)C=C5)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C56H55FN6O7S2	ERα;ERβ	P03372/Q92731	VHL	WO-2018140809-A1
TPD-J9JQPJ	SCHEMBL20442614	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[4-[4-[[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenyl]piperidin-1-yl]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCN3CCC(C4=CC=C(OC5=C(C6=CC=C(F)C=C6)SC6=C5C=CC(O)=C6)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C54H62FN5O8S2	ERα;ERβ	P03372/Q92731	VHL	WO-2018140809-A1
TPD-IBXB1E	SCHEMBL20442612	(2S,4R)-N-[(4-cyanophenyl)methyl]-1-[(2S)-2-[[2-[2-[2-[4-[4-[[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenyl]piperidin-1-yl]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide	CC(C)(C)[C@H](NC(=O)COCCOCCN1CCC(C2=CC=C(OC3=C(C4=CC=C(F)C=C4)SC4=C3C=CC(O)=C4)C=C2)CC1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C#N)C=C1	C50H56FN5O8S	ERα;ERβ	P03372/Q92731	VHL	WO-2018140809-A1
TPD-NTMYRY	SCHEMBL20442716	(2S,4R)-N-[(4-chlorophenyl)methyl]-1-[(2S)-2-[[2-[2-[2-[4-[4-[[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenyl]piperidin-1-yl]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide	CC(C)(C)[C@H](NC(=O)COCCOCCN1CCC(C2=CC=C(OC3=C(C4=CC=C(F)C=C4)SC4=C3C=CC(O)=C4)C=C2)CC1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(Cl)C=C1	C49H56ClFN4O8S	ERα;ERβ	P03372/Q92731	VHL	WO-2018140809-A1
TPD-0SX6IF	SCHEMBL20442711	(2S,4R)-N-[(4-cyanophenyl)methyl]-1-[(2S)-2-[[2-[4-[1-[2-[4-[[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]pyrazol-3-yl]phenyl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide	CC(C)(C)[C@H](NC(=O)CC1=CC=C(C2=NN(CCOC3=CC=C(OC4=C(C5=CC=C(F)C=C5)SC5=C4C=CC(O)=C5)C=C3)C=C2)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C#N)C=C1	C52H49FN6O7S	ERα;ERβ	P03372/Q92731	VHL	WO-2018140809-A1
TPD-CU5UQD	SCHEMBL20442720	(2S,4R)-N-[(4-chlorophenyl)methyl]-1-[(2S)-2-[[2-[4-[1-[2-[4-[[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]pyrazol-3-yl]phenyl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide	CC(C)(C)[C@H](NC(=O)CC1=CC=C(C2=NN(CCOC3=CC=C(OC4=C(C5=CC=C(F)C=C5)SC5=C4C=CC(O)=C5)C=C3)C=C2)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(Cl)C=C1	C51H49ClFN5O7S	ERα;ERβ	P03372/Q92731	VHL	WO-2018140809-A1
TPD-1K5TTP	SCHEMBL20442718	(2S,4R)-N-[(1S)-1-(4-cyanophenyl)ethyl]-1-[(2S)-2-[[2-[2-[2-[4-[4-[[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenyl]piperidin-1-yl]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide	C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](NC(=O)COCCOCCN1CCC(C2=CC=C(OC3=C(C4=CC=C(F)C=C4)SC4=C3C=CC(O)=C4)C=C2)CC1)C(C)(C)C)C1=CC=C(C#N)C=C1	C51H58FN5O8S	ERα;ERβ	P03372/Q92731	VHL	WO-2018140809-A1
TPD-MU0KVK	SCHEMBL20442712	(2S,4R)-N-[(1S)-1-(4-chlorophenyl)ethyl]-1-[(2S)-2-[[2-[2-[2-[4-[4-[[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenyl]piperidin-1-yl]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide	C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](NC(=O)COCCOCCN1CCC(C2=CC=C(OC3=C(C4=CC=C(F)C=C4)SC4=C3C=CC(O)=C4)C=C2)CC1)C(C)(C)C)C1=CC=C(Cl)C=C1	C50H58ClFN4O8S	ERα;ERβ	P03372/Q92731	VHL	WO-2018140809-A1
TPD-9W89ML	SCHEMBL20442714	(2S,4R)-N-[(1S)-1-(4-cyanophenyl)ethyl]-1-[(2S)-2-[[2-[4-[1-[2-[4-[[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]pyrazol-3-yl]phenyl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide	C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](NC(=O)CC1=CC=C(C2=NN(CCOC3=CC=C(OC4=C(C5=CC=C(F)C=C5)SC5=C4C=CC(O)=C5)C=C3)C=C2)C=C1)C(C)(C)C)C1=CC=C(C#N)C=C1	C53H51FN6O7S	ERα;ERβ	P03372/Q92731	VHL	WO-2018140809-A1
TPD-BHN7L8	SCHEMBL20442694	(2S,4R)-N-[(1S)-1-(4-chlorophenyl)ethyl]-1-[(2S)-2-[[2-[4-[1-[2-[4-[[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]pyrazol-3-yl]phenyl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide	C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](NC(=O)CC1=CC=C(C2=NN(CCOC3=CC=C(OC4=C(C5=CC=C(F)C=C5)SC5=C4C=CC(O)=C5)C=C3)C=C2)C=C1)C(C)(C)C)C1=CC=C(Cl)C=C1	C52H51ClFN5O7S	ERα;ERβ	P03372/Q92731	VHL	WO-2018140809-A1
TPD-ZVGXQX	SCHEMBL20425343	(2S,4R)-1-[(2S)-2-[[2-[2-[4-[2-[4-[[2-(4-chlorophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperazin-1-yl]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCN3CCN(CCOC4=CC=C(OC5=C(C6=CC=C(Cl)C=C6)SC6=C5C=CC(O)=C6)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C52H59ClN6O8S2	ERα;ERβ	P03372/Q92731	VHL	WO-2018140809-A1
TPD-9ULC6A	WO2018140809A1_152	.	CC1=C(C2=CC=C(CNC(=O)[C@H]3C[C@H](O)CN3C(=O)[C@@H](NC(=O)COCCN3CCN(CCOC4=CC=C(OC5=C(C6=CC=C(Cl)C=C6)SC6=C5C=CC(O)=C6)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C52H59ClN6O8S2	ERα;ERβ	P03372/Q92731	VHL	WO-2018140809-A1
TPD-VQXWWO	WO2018140809A1_153	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCN3CCN(CCOC4=CC=C(OC5=C(C6=CC=C(Cl)C=C6)SC6=C5C=CC(O)=C6)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C53H61ClN6O8S2	ERα;ERβ	P03372/Q92731	VHL	WO-2018140809-A1
TPD-PCQMSM	SCHEMBL20442690	(2S,4R)-1-[(2S)-2-[[2-[2-[4-[2-[4-[[2-(4-bromophenyl)-6-methoxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperazin-1-yl]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	COC1=CC2=C(C=C1)C(OC1=CC=C(OCCN3CCN(CCOCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)NCC4=CC=C(C5=C(C)N=CS5)C=C4)C(C)(C)C)CC3)C=C1)=C(C1=CC=C(Br)C=C1)S2	C53H61BrN6O8S2	ERα;ERβ	P03372/Q92731	VHL	WO-2018140809-A1
TPD-XK3ZI6	SCHEMBL20442696	(2S,4R)-1-[(2S)-2-[[2-[2-[4-[2-[4-[[2-(4-bromophenyl)-6-methoxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperazin-1-yl]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	COC1=CC2=C(C=C1)C(OC1=CC=C(OCCN3CCN(CCOCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)N[C@@H](C)C4=CC=C(C5=C(C)N=CS5)C=C4)C(C)(C)C)CC3)C=C1)=C(C1=CC=C(Br)C=C1)S2	C54H63BrN6O8S2	ERα;ERβ	P03372/Q92731	VHL	WO-2018140809-A1
TPD-8OI1JP	SCHEMBL20442784	(2S)-1-[(2S)-2-[[2-[2-[4-[2-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperazin-1-yl]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3CCCN3C(=O)[C@@H](NC(=O)COCCN3CCN(CCOC4=CC=C(OC5=C(C6=CC=C(Br)C=C6)SC6=C5C=CC(O)=C6)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C52H59BrN6O7S2	ERα;ERβ	P03372/Q92731	VHL	WO-2018140809-A1
TPD-16UOBC	SCHEMBL20442785	(2S)-1-[(2S)-2-[[2-[2-[4-[2-[4-[[2-(4-bromophenyl)-6-methoxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperazin-1-yl]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	COC1=CC2=C(C=C1)C(OC1=CC=C(OCCN3CCN(CCOCC(=O)N[C@H](C(=O)N4CCC[C@H]4C(=O)NCC4=CC=C(C5=C(C)N=CS5)C=C4)C(C)(C)C)CC3)C=C1)=C(C1=CC=C(Br)C=C1)S2	C53H61BrN6O7S2	ERα;ERβ	P03372/Q92731	VHL	WO-2018140809-A1
TPD-TC99Z4	SCHEMBL20425503	(2S,4R)-1-[(2S)-2-[[2-[4-[2-[2-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethoxy]ethyl]piperazin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCN(CCOCCOC4=CC=C(OC5=C(C6=CC=C(Br)C=C6)SC6=C5C=CC(O)=C6)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C52H59BrN6O8S2	ERα;ERβ	P03372/Q92731	VHL	WO-2018140809-A1
TPD-5MGBLO	WO2018140809A1_159	(2S)-1-[(2S)-2-[[2-[2-[4-[2-[4-[[2-(4-bromophenyl)-6-methoxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperazin-1-yl]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-4-oxopyrrolidine-2-carboxamide	COC1=CC2=C(C=C1)C(OC1=CC=C(OCCN3CCN(CCOCC(=O)N[C@H](C(=O)N4CC(=O)C[C@H]4C(=O)NCC4=CC=C(C5=C(C)N=CS5)C=C4)C(C)(C)C)CC3)C=C1)=C(C1=CC=C(Br)C=C1)S2	C53H59BrN6O8S2	ERα;ERβ	P03372/Q92731	VHL	WO-2018140809-A1
TPD-Y0YU2F	SCHEMBL20442787	(2S,4R)-1-[(2S)-2-[[2-[4-[3-[2-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethoxy]azetidin-1-yl]piperidin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCC(N4CC(OCCOC5=CC=C(OC6=C(C7=CC=C(Br)C=C7)SC7=C6C=CC(O)=C7)C=C5)C4)CC3)C(C)(C)C)C=C2)SC=N1	C54H61BrN6O8S2	ERα;ERβ	P03372/Q92731	VHL	WO-2018140809-A1
TPD-BF4UXT	SCHEMBL20442786	(2S,4R)-1-[(2R)-2-[3-[2-[4-[2-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperazin-1-yl]ethoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-N-[(4-chlorophenyl)methyl]-4-hydroxypyrrolidine-2-carboxamide	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(Cl)C=C1)C1=CC(OCCN2CCN(CCOC3=CC=C(OC4=C(C5=CC=C(Br)C=C5)SC5=C4C=CC(O)=C5)C=C3)CC2)=NO1	C48H51BrClN5O8S	ERα;ERβ	P03372/Q92731	VHL	WO-2018140809-A1
TPD-GWQD12	SCHEMBL20442821	(2S,4R)-1-[(2S)-2-[3-[2-[4-[2-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperazin-1-yl]ethoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-N-[(4-chlorophenyl)methyl]-4-hydroxypyrrolidine-2-carboxamide	CC(C)[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(Cl)C=C1)C1=CC(OCCN2CCN(CCOC3=CC=C(OC4=C(C5=CC=C(Br)C=C5)SC5=C4C=CC(O)=C5)C=C3)CC2)=NO1	C48H51BrClN5O8S	ERα;ERβ	P03372/Q92731	VHL	WO-2018140809-A1
TPD-5Z9NNB	SCHEMBL20442822	(2S,4R)-1-[(2S)-2-[3-[2-[4-[2-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperazin-1-yl]ethoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3=CC(OCCN4CCN(CCOC5=CC=C(OC6=C(C7=CC=C(Br)C=C7)SC7=C6C=CC(O)=C7)C=C5)CC4)=NO3)C(C)C)C=C2)SC=N1	C52H55BrN6O8S2	ERα;ERβ	P03372/Q92731	VHL	WO-2018140809-A1
TPD-4G4L3R	SCHEMBL20442826	(2S,4R)-1-[(2R)-2-[3-[2-[4-[2-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperazin-1-yl]ethoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(OCCN4CCN(CCOC5=CC=C(OC6=C(C7=CC=C(Br)C=C7)SC7=C6C=CC(O)=C7)C=C5)CC4)=NO3)C(C)C)C=C2)SC=N1	C52H55BrN6O8S2	ERα;ERβ	P03372/Q92731	VHL	WO-2018140809-A1
TPD-CX6ULM	SCHEMBL20442824	(2S,4R)-1-[(2R)-2-[3-[2-[4-[2-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperazin-1-yl]ethoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-N-[(4-cyanophenyl)methyl]-4-hydroxypyrrolidine-2-carboxamide	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C#N)C=C1)C1=CC(OCCN2CCN(CCOC3=CC=C(OC4=C(C5=CC=C(Br)C=C5)SC5=C4C=CC(O)=C5)C=C3)CC2)=NO1	C49H51BrN6O8S	ERα;ERβ	P03372/Q92731	VHL	WO-2018140809-A1
TPD-ZYVSN2	SCHEMBL20442823	(2S,4R)-1-[(2S)-2-[3-[2-[4-[2-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperazin-1-yl]ethoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-N-[(4-cyanophenyl)methyl]-4-hydroxypyrrolidine-2-carboxamide	CC(C)[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C#N)C=C1)C1=CC(OCCN2CCN(CCOC3=CC=C(OC4=C(C5=CC=C(Br)C=C5)SC5=C4C=CC(O)=C5)C=C3)CC2)=NO1	C49H51BrN6O8S	ERα;ERβ	P03372/Q92731	VHL	WO-2018140809-A1
TPD-IM2UO6	SCHEMBL20442825	(2S,4R)-1-[(2S)-2-[[2-[2-[(1S,4S)-5-[2-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]-2,5-diazabicyclo[2.2.1]heptan-2-yl]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCN3C[C@@H]4C[C@H]3CN4CCOC3=CC=C(OC4=C(C5=CC=C(Br)C=C5)SC5=C4C=CC(O)=C5)C=C3)C(C)(C)C)C=C2)SC=N1	C53H59BrN6O8S2	ERα;ERβ	P03372/Q92731	VHL	WO-2018140809-A1
TPD-O72PJ2	SCHEMBL20442650	(2S,4R)-1-[(2S)-2-[[2-[2-[4-[2-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperazin-1-yl]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1R)-2-hydroxy-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CO)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCN3CCN(CCOC4=CC=C(OC5=C(C6=CC=C(Br)C=C6)SC6=C5C=CC(O)=C6)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C53H61BrN6O9S2	ERα;ERβ	P03372/Q92731	VHL	WO-2018140809-A1
TPD-MR8RG0	SCHEMBL20442651	(2S,4R)-1-[(2S)-2-[[2-[2-[(1S,4S)-5-[2-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]-2,5-diazabicyclo[2.2.1]heptan-2-yl]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1R)-2-hydroxy-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CO)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCN3C[C@@H]4C[C@H]3CN4CCOC3=CC=C(OC4=C(C5=CC=C(Br)C=C5)SC5=C4C=CC(O)=C5)C=C3)C(C)(C)C)C=C2)SC=N1	C54H61BrN6O9S2	ERα;ERβ	P03372/Q92731	VHL	WO-2018140809-A1
TPD-U7MCG5	WO2018140809A1_171	.	O=C1CCC(N2CC3=CC(NCCCOCCOCCOC4C=CC(OC5=C(C6=CC=C(Br)C=C6)SC6=C5C=CC(O)=C6)=CC4)=CC=C3C2=O)C(=O)N1	C40H40BrN3O8S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-H1BFY0	SCHEMBL21907840	3-[6-[3-[4-[2-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperazin-1-yl]propylamino]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(NCCCN4CCN(CCOC5=CC=C(OC6=C(C7=CC=C(Br)C=C7)SC7=C6C=CC(O)=C7)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C42H42BrN5O6S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-COE74A	SCHEMBL21907869	3-[6-[3-[4-[2-[4-[[2-(4-hydroxyphenyl)-6-methoxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperazin-1-yl]propylamino]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	COC1=CC2=C(C=C1)C(OC1=CC=C(OCCN3CCN(CCCNC4=CC=C5C(=O)N(C6CCC(=O)NC6=O)CC5=C4)CC3)C=C1)=C(C1=CC=C(O)C=C1)S2	C43H45N5O7S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-NTYKPW	SCHEMBL22151751	(3S)-3-[6-[2-[4-[4-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]butyl]-1,4-diazepan-1-yl]ethyl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CC[C@H](N2CC3=CC(CCN4CCCN(CCCCOC5=CC=C(OC6=C(C7=CC=C(Br)C=C7)SC7=C6C=CC(O)=C7)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C44H45BrN4O6S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-SAFMPG	SCHEMBL20442748	5-[4-[1-[2-[4-[[2-(4-Bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperidin-4-yl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(C5CCN(CCOC6=CC=C(OC7=C(C8=CC=C(Br)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C44H42BrN5O7S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-73RYBX	SCHEMBL20442706	5-[4-[[1-[2-[4-[[2-(4-Bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CC5CCN(CCOC6=CC=C(OC7=C(C8=CC=C(Br)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C45H44BrN5O7S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-YU4S7I	SCHEMBL20442561	5-[4-[[1-[2-[4-[[2-(4-Bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]azetidin-3-yl]methyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CC5CN(CCOC6=CC=C(OC7=C(C8=CC=C(Br)C=C8)SC8=C7C=CC(O)=C8)C=C6)C5)CC4)C=C3C2=O)C(=O)N1	C43H40BrN5O7S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-QVOJAY	SCHEMBL20442559	5-[4-[2-[1-[2-[4-[[2-(4-Bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]azetidin-3-yl]ethyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCC5CN(CCOC6=CC=C(OC7=C(C8=CC=C(Br)C=C8)SC8=C7C=CC(O)=C8)C=C6)C5)CC4)C=C3C2=O)C(=O)N1	C44H42BrN5O7S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-PBL2IK	SCHEMBL21906699	3-[6-[4-[[4-[4-[[6-hydroxy-2-[4-(trifluoromethyl)phenyl]-1-benzothiophen-3-yl]oxy]phenoxy]piperidin-1-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; YEVUQHKEJPIGLE-UHFFFAOYSA-N; 3-[6-[4-[[4-[4-[[6-hydroxy-2-[4-(trifluoromethyl)phenyl]-1-benzothiophen-3-yl]oxy]phenoxy]piperidin-1-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(N4CCC(CN5CCC(OC6=CC=C(OC7=C(C8=CC=C(C(F)(F)F)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C45H43F3N4O6S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-6DQEZA	SCHEMBL21906878	2-(2,6-Dioxopiperidin-3-yl)-5-[4-[[4-[4-[[6-hydroxy-2-[4-(trifluoromethyl)phenyl]-1-benzothiophen-3-yl]oxy]phenoxy]piperidin-1-yl]methyl]piperidin-1-yl]isoindole-1,3-dione; DRCUVKUSMZWTST-UHFFFAOYSA-N; 2-(2,6-Dioxopiperidin-3-yl)-5-[4-[[4-[4-[[6-hydroxy-2-[4-(trifluoromethyl)phenyl]-1-benzothiophen-3-yl]oxy]phenoxy]piperidin-1-yl]methyl]piperidin-1-yl]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC=C(N4CCC(CN5CCC(OC6=CC=C(OC7=C(C8=CC=C(C(F)(F)F)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C45H41F3N4O7S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-QWZHWZ	SCHEMBL20442560	5-[3-[[4-[2-[4-[[2-(4-Bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperazin-1-yl]methyl]azetidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC=C(N4CC(CN5CCN(CCOC6=CC=C(OC7=C(C8=CC=C(Br)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)C4)C=C3C2=O)C(=O)N1	C43H40BrN5O7S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-1WT0A0	SCHEMBL20442558	5-[1-[1-[2-[4-[[2-(4-Bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperidin-4-yl]piperidin-4-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=C(C=C(C4CCN(C5CCN(CCOC6=CC=C(OC7=C(C8=CC=C(Br)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)C=C3)C2=O)C(=O)N1	C45H43BrN4O7S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-GLHVW3	SCHEMBL20442550	5-[3-[[4-[2-[4-[[2-(4-Bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]-1,4-diazepan-1-yl]methyl]azetidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC=C(N4CC(CN5CCCN(CCOC6=CC=C(OC7=C(C8=CC=C(Br)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)C4)C=C3C2=O)C(=O)N1	C44H42BrN5O7S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-3LH6TB	SCHEMBL20442741	3-[6-[4-[1-[2-[4-[[6-hydroxy-2-[4-(trifluoromethyl)phenyl]-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperidin-4-yl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; GKTFIICDYFZDOM-UHFFFAOYSA-N; 3-[6-[4-[1-[2-[4-[[6-hydroxy-2-[4-(trifluoromethyl)phenyl]-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperidin-4-yl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(N4CCN(C5CCN(CCOC6=CC=C(OC7=C(C8=CC=C(C(F)(F)F)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C45H44F3N5O6S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-S15SUM	SCHEMBL21907867	3-[7-fluoro-6-[4-[1-[2-[4-[[6-hydroxy-2-[4-(trifluoromethyl)phenyl]-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperidin-4-yl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; QXBJEYCPIRXPJN-UHFFFAOYSA-N; 3-[7-fluoro-6-[4-[1-[2-[4-[[6-hydroxy-2-[4-(trifluoromethyl)phenyl]-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperidin-4-yl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(F)C(N4CCN(C5CCN(CCOC6=CC=C(OC7=C(C8=CC=C(C(F)(F)F)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C45H43F4N5O6S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-K7N9FF	SCHEMBL21906762	3-[6-[4-[1-[2-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperidin-4-yl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(N4CCN(C5CCN(CCOC6=CC=C(OC7=C(C8=CC=C(Br)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C44H44BrN5O6S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-89843P	SCHEMBL21907874	3-[6-[4-[1-[2-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperidin-4-yl]piperazin-1-yl]-7-fluoro-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(F)C(N4CCN(C5CCN(CCOC6=CC=C(OC7=C(C8=CC=C(Br)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C44H43BrFN5O6S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-0Y6M1X	SCHEMBL20442740	3-[6-[1-[1-[2-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperidin-4-yl]piperidin-4-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(C4CCN(C5CCN(CCOC6=CC=C(OC7=C(C8=CC=C(Br)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C45H45BrN4O6S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-NW5GPR	SCHEMBL20442744	5-[4-[4-[2-[4-[[2-(4-Bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]-1,4-diazepan-1-yl]butyl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC=C(CCCCN4CCCN(CCOC5=CC=C(OC6=C(C7=CC=C(Br)C=C7)SC7=CC(O)=CC=C76)C=C5)CC4)C=C3C2=O)C(=O)N1	C44H43BrN4O7S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-25YI0W	SCHEMBL21907138	3-[6-[4-[2-[2-[4-[[6-hydroxy-2-[4-(trifluoromethyl)phenyl]-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]-2-azaspiro[3.3]heptan-6-yl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(N4CCN(C5CC6(C5)CN(CCOC5=CC=C(OC7=C(C8=CC=C(C(F)(F)F)C=C8)SC8=C7C=CC(O)=C8)C=C5)C6)CC4)=CC=C3C2=O)C(=O)N1	C46H44F3N5O6S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-YCS3CX	SCHEMBL20442742	3-[6-[4-[4-[2-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]-1,4-diazepan-1-yl]butyl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(CCCCN4CCCN(CCOC5=CC=C(OC6=C(C7=CC=C(Br)C=C7)SC7=CC(O)=CC=C76)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C44H45BrN4O6S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-C6BJO7	SCHEMBL20442743	3-[6-[4-[[1-[2-[4-[[6-hydroxy-2-[4-(trifluoromethyl)phenyl]-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; JGCQYXFDNMAUOB-UHFFFAOYSA-N; 3-[6-[4-[[1-[2-[4-[[6-hydroxy-2-[4-(trifluoromethyl)phenyl]-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(N4CCN(CC5CCN(CCOC6=CC=C(OC7=C(C8=CC=C(C(F)(F)F)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C46H46F3N5O6S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-MRGUS4	SCHEMBL20442745	3-[7-fluoro-6-[4-[[1-[2-[4-[[6-hydroxy-2-[4-(trifluoromethyl)phenyl]-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; QTYKHOICHQVZPR-UHFFFAOYSA-N; 3-[7-fluoro-6-[4-[[1-[2-[4-[[6-hydroxy-2-[4-(trifluoromethyl)phenyl]-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(F)C(N4CCN(CC5CCN(CCOC6=CC=C(OC7=C(C8=CC=C(C(F)(F)F)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C46H45F4N5O6S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-YCYGTP	SCHEMBL20442551	2-(2,6-Dioxopiperidin-3-yl)-5-[4-[[1-[2-[4-[[6-hydroxy-2-[4-(trifluoromethyl)phenyl]-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperidin-4-yl]methyl]piperazin-1-yl]isoindole-1,3-dione; BMZMDZPZOXKXPJ-UHFFFAOYSA-N; 2-(2,6-Dioxopiperidin-3-yl)-5-[4-[[1-[2-[4-[[6-hydroxy-2-[4-(trifluoromethyl)phenyl]-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperidin-4-yl]methyl]piperazin-1-yl]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CC5CCN(CCOC6=CC=C(OC7=C(C8=CC=C(C(F)(F)F)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C46H44F3N5O7S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-QMJR2N	SCHEMBL20442554	3-[5,7-difluoro-6-[4-[1-[2-[4-[[6-hydroxy-2-[4-(trifluoromethyl)phenyl]-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperidin-4-yl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; WKFVKUVNOAFMBB-UHFFFAOYSA-N; 3-[5,7-difluoro-6-[4-[1-[2-[4-[[6-hydroxy-2-[4-(trifluoromethyl)phenyl]-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperidin-4-yl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(F)C(N4CCN(C5CCN(CCOC6=CC=C(OC7=C(C8=CC=C(C(F)(F)F)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)=C(F)C=C3C2=O)C(=O)N1	C45H42F5N5O6S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-QVXQKN	SCHEMBL20442552	3-[5-fluoro-6-[4-[[1-[2-[4-[[6-hydroxy-2-[4-(trifluoromethyl)phenyl]-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; DOHQDYLLDVSNOS-UHFFFAOYSA-N; 3-[5-fluoro-6-[4-[[1-[2-[4-[[6-hydroxy-2-[4-(trifluoromethyl)phenyl]-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(N4CCN(CC5CCN(CCOC6=CC=C(OC7=C(C8=CC=C(C(F)(F)F)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)=C(F)C=C3C2=O)C(=O)N1	C46H45F4N5O6S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-6AUBKE	SCHEMBL20442553	3-[6-[4-[1-[2-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperidin-4-yl]piperazin-1-yl]-5,7-difluoro-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(F)C(N4CCN(C5CCN(CCOC6=CC=C(OC7=C(C8=CC=C(Br)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)=C(F)C=C3C2=O)C(=O)N1	C44H42BrF2N5O6S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-96YDP9	SCHEMBL21907871	3-[5,7-difluoro-6-[4-[2-[2-[4-[[6-hydroxy-2-[4-(trifluoromethyl)phenyl]-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]-2-azaspiro[3.3]heptan-6-yl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(F)C(N4CCN(C5CC6(C5)CN(CCOC5=CC=C(OC7=C(C8=CC=C(C(F)(F)F)C=C8)SC8=C7C=CC(O)=C8)C=C5)C6)CC4)=C(F)C=C3C2=O)C(=O)N1	C46H42F5N5O6S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-LVJZX7	SCHEMBL20442555	3-[6-[4-[3-[4-[[6-hydroxy-2-[4-(trifluoromethyl)phenyl]-1-benzothiophen-3-yl]oxy]phenoxy]propyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; VNUGFHUJWXLMFR-UHFFFAOYSA-N; 3-[6-[4-[3-[4-[[6-hydroxy-2-[4-(trifluoromethyl)phenyl]-1-benzothiophen-3-yl]oxy]phenoxy]propyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCCOC5=CC=C(OC6=C(C7=CC=C(C(F)(F)F)C=C7)SC7=CC(O)=CC=C76)C=C5)CC4)=C3)C2=O)C(=O)N1	C41H37F3N4O6S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-MVJMTI	SCHEMBL20442636	3-[6-[4-[3-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]propyl]piperazin-1-yl]-7-fluoro-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCCOC5=CC=C(OC6=C(C7=CC=C(Br)C=C7)SC7=CC(O)=CC=C76)C=C5)CC4)=C3F)C2=O)C(=O)N1	C40H36BrFN4O6S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-4305VM	SCHEMBL20442535	5-[3-[[4-[4-[[2-(4-Bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenyl]piperidin-1-yl]methyl]azetidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC=C(N4CC(CN5CCC(C6=CC=C(OC7=C(C8=CC=C(Br)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)C4)C=C3C2=O)C(=O)N1	C42H37BrN4O6S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-7GXYK7	SCHEMBL20442635	5-[4-[4-[4-[[2-(4-Bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenyl]butyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCCCC5=CC=C(OC6=C(C7=CC=C(Br)C=C7)SC7=C6C=CC(O)=C7)C=C5)CC4)C=C3C2=O)C(=O)N1	C41H37BrN4O6S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-U00FNA	SCHEMBL20442570	5-[4-[3-[4-[[2-(4-Bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]azetidin-1-yl]piperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC=C(N4CCC(N5CC(OC6=CC=C(OC7=C(C8=CC=C(Br)C=C8)SC8=C7C=CC(O)=C8)C=C6)C5)CC4)C=C3C2=O)C(=O)N1	C41H35BrN4O7S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-2I1VRL	SCHEMBL20442637	5-[3-[4-[4-[[2-(4-Bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]piperidin-1-yl]azetidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC=C(N4CC(N5CCC(OC6=CC=C(OC7=C(C8=CC=C(Br)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)C4)C=C3C2=O)C(=O)N1	C41H35BrN4O7S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-1SSLFJ	SCHEMBL20442767	5-[4-[[3-[4-[[2-(4-Bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenyl]azetidin-1-yl]methyl]piperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC=C(N4CCC(CN5CC(C6=CC=C(OC7=C(C8=CC=C(Br)C=C8)SC8=C7C=CC(O)=C8)C=C6)C5)CC4)C=C3C2=O)C(=O)N1	C42H37BrN4O6S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-BPRG2K	SCHEMBL20442768	3-[6-[4-[4-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenyl]butyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(N4CCN(CCCCC5=CC=C(OC6=C(C7=CC=C(Br)C=C7)SC7=C6C=CC(O)=C7)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C41H39BrN4O5S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-KJH70S	SCHEMBL20442764	3-[6-[4-[[3-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenyl]azetidin-1-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(N4CCC(CN5CC(C6=CC=C(OC7=C(C8=CC=C(Br)C=C8)SC8=C7C=CC(O)=C8)C=C6)C5)CC4)=CC=C3C2=O)C(=O)N1	C42H39BrN4O5S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-Z5FZNU	SCHEMBL20442769	3-[6-[4-[3-[4-[[6-hydroxy-2-[4-(trifluoromethoxy)phenyl]-1-benzothiophen-3-yl]oxy]phenoxy]propyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; CQFQNCYVSZCHLT-UHFFFAOYSA-N; 3-[6-[4-[3-[4-[[6-hydroxy-2-[4-(trifluoromethoxy)phenyl]-1-benzothiophen-3-yl]oxy]phenoxy]propyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCCOC5=CC=C(OC6=C(C7=CC=C(OC(F)(F)F)C=C7)SC7=CC(O)=CC=C76)C=C5)CC4)=C3)C2=O)C(=O)N1	C41H37F3N4O7S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-8VTOV2	SCHEMBL20442765	3-[5,7-difluoro-6-[4-[3-[4-[[6-hydroxy-2-[4-(trifluoromethoxy)phenyl]-1-benzothiophen-3-yl]oxy]phenoxy]propyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; PKCWHAGQKJHPTG-UHFFFAOYSA-N; 3-[5,7-difluoro-6-[4-[3-[4-[[6-hydroxy-2-[4-(trifluoromethoxy)phenyl]-1-benzothiophen-3-yl]oxy]phenoxy]propyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=C(F)C(N4CCN(CCCOC5=CC=C(OC6=C(C7=CC=C(OC(F)(F)F)C=C7)SC7=CC(O)=CC=C76)C=C5)CC4)=C3F)C2=O)C(=O)N1	C41H35F5N4O7S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-UPN229	SCHEMBL20442766	3-[5-fluoro-6-[4-[3-[4-[[6-hydroxy-2-[4-(trifluoromethoxy)phenyl]-1-benzothiophen-3-yl]oxy]phenoxy]propyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; FXJFITSSJWIHKF-UHFFFAOYSA-N; 3-[5-fluoro-6-[4-[3-[4-[[6-hydroxy-2-[4-(trifluoromethoxy)phenyl]-1-benzothiophen-3-yl]oxy]phenoxy]propyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=C(F)C(N4CCN(CCCOC5=CC=C(OC6=C(C7=CC=C(OC(F)(F)F)C=C7)SC7=CC(O)=CC=C76)C=C5)CC4)=C3)C2=O)C(=O)N1	C41H36F4N4O7S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-HXDGGS	SCHEMBL20442752	3-[6-[4-[3-[4-[[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]propyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCCOC5=CC=C(OC6=C(C7=CC=C(F)C=C7)SC7=CC(O)=CC=C76)C=C5)CC4)=C3)C2=O)C(=O)N1	C40H37FN4O6S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-HB2BIU	SCHEMBL20442753	3-[6-[4-[3-[4-[[2-(3,4-difluorophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]propyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCCOC5=CC=C(OC6=C(C7=CC=C(F)C(F)=C7)SC7=CC(O)=CC=C76)C=C5)CC4)=C3)C2=O)C(=O)N1	C40H36F2N4O6S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-TDVRN5	SCHEMBL20442754	3-[6-[4-[3-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]propyl]piperazin-1-yl]-4-fluoro-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C2=O)C(F)=CC(N2CCN(CCCOC4=CC=C(OC5=C(C6=CC=C(Br)C=C6)SC6=CC(O)=CC=C65)C=C4)CC2)=C3)C(=O)N1	C40H36BrFN4O6S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-F7GA9T	SCHEMBL20442590	5-[4-[3-[4-[[2-(4-Bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]cyclobutyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC=C(N4CCN([C@H]5C[C@H](OC6=CC=C(OC7=C(C8=CC=C(Br)C=C8)SC8=C7C=CC(O)=C8)C=C6)C5)CC4)C=C3C2=O)C(=O)N1	C41H35BrN4O7S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-B4RPBA	SCHEMBL20442738	3-[6-[4-[3-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]cyclobutyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(N4CCN(C5CC(OC6=CC=C(OC7=C(C8=CC=C(Br)C=C8)SC8=C7C=CC(O)=C8)C=C6)C5)CC4)=CC=C3C2=O)C(=O)N1	C41H37BrN4O6S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-DFD7XZ	SCHEMBL20442755	5-[4-[2-[[4-[[2-(4-Bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenyl]methoxy]ethyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCOCC5=CC=C(OC6=C(C7=CC=C(Br)C=C7)SC7=C6C=CC(O)=C7)C=C5)CC4)C=C3C2=O)C(=O)N1	C40H35BrN4O7S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-EX6LJM	SCHEMBL20442619	3-[6-[4-[[1-[4-[[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC5CCN(C6=CC=C(OC7=C(C8=CC=C(F)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C43H42FN5O5S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-B80ODV	SCHEMBL20442623	2-(2,6-Dioxopiperidin-3-yl)-5-[4-[[1-[4-[[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=C(C=C(N4CCN(CC5CCN(C6=CC=C(OC7=C(C8=CC=C(F)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)C=C3)C2=O)C(=O)N1	C43H40FN5O6S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-USQXNW	SCHEMBL21906889	5-[4-[[1-[4-[[2-(4-Bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=C(C=C(N4CCN(CC5CCN(C6=CC=C(OC7=C(C8=CC=C(Br)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)C=C3)C2=O)C(=O)N1	C43H40BrN5O6S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-40469G	SCHEMBL20442620	3-[6-[4-[2-[1-[4-[[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenyl]piperidin-4-yl]ethyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCC5CCN(C6=CC=C(OC7=C(C8=CC=C(F)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C44H44FN5O5S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-IE3EZH	SCHEMBL20442624	3-[2-[4-[[1-[4-[[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-5-oxo-7H-pyrrolo[3,4-b]pyridin-6-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC5CCN(C6=CC=C(OC7=C(C8=CC=C(F)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)=N3)C2=O)C(=O)N1	C42H41FN6O5S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-VWH3ND	SCHEMBL20442528	3-[6-[4-[[1-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC5CCN(C6=CC=C(OC7=C(C8=CC=C(Br)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C43H42BrN5O5S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-ADVQKO	SCHEMBL20425506	3-[6-[4-[[1-[5-[[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]pyridin-2-yl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC5CCN(C6=NC=C(OC7=C(C8=CC=C(F)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C42H41FN6O5S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-B9HSW7	SCHEMBL20442803	3-[6-[4-[3-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]azetidin-1-yl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(N4CCC(N5CC(OC6=CC=C(OC7=C(C8=CC=C(Br)C=C8)SC8=C7C=CC(O)=C8)C=C6)C5)CC4)=CC=C3C2=O)C(=O)N1	C41H37BrN4O6S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-R7VI8H	SCHEMBL20442804	3-[6-[4-[[1-[4-[[6-hydroxy-2-(4-methoxyphenyl)-1-benzothiophen-3-yl]oxy]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	COC1=CC=C(C2=C(OC3=CC=C(N4CCC(CN5CCN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)CC5)CC4)C=C3)C3=C(C=C(O)C=C3)S2)C=C1	C44H45N5O6S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-S956HM	SCHEMBL20442809	3-[2-[4-[[1-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-5-oxo-7H-pyrrolo[3,4-b]pyridin-6-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC5CCN(C6=CC=C(OC7=C(C8=CC=C(Br)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)=N3)C2=O)C(=O)N1	C42H41BrN6O5S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-2SZHBJ	SCHEMBL20442805	3-[6-[4-[[1-[5-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]pyridin-2-yl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC5CCN(C6=CC=C(OC7=C(C8=CC=C(Br)C=C8)SC8=C7C=CC(O)=C8)C=N6)CC5)CC4)=C3)C2=O)C(=O)N1	C42H41BrN6O5S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-KYC0LU	SCHEMBL20442806	2-(2,6-Dioxopiperidin-3-yl)-5-[4-[[1-[4-[[6-hydroxy-2-(4-methoxyphenyl)-1-benzothiophen-3-yl]oxy]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]isoindole-1,3-dione	COC1=CC=C(C2=C(OC3=CC=C(N4CCC(CN5CCN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)C=C3)C3=C(C=C(O)C=C3)S2)C=C1	C44H43N5O7S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-1OLW70	SCHEMBL20442818	3-[6-[4-[[1-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]-2-fluorophenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC5CCN(C6=CC=C(OC7=C(C8=CC=C(Br)C=C8)SC8=C7C=CC(O)=C8)C=C6F)CC5)CC4)=C3)C2=O)C(=O)N1	C43H41BrFN5O5S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-28OJT2	SCHEMBL20442816	3-[2-[4-[[1-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]-2-fluorophenyl]piperidin-4-yl]methyl]piperazin-1-yl]-5-oxo-7H-pyrrolo[3,4-b]pyridin-6-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC5CCN(C6=CC=C(OC7=C(C8=CC=C(Br)C=C8)SC8=C7C=CC(O)=C8)C=C6F)CC5)CC4)=N3)C2=O)C(=O)N1	C42H40BrFN6O5S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-TE3EIK	SCHEMBL20442819	3-[6-[3-[4-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]piperidin-1-yl]azetidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(N4CC(N5CCC(OC6=CC=C(OC7=C(C8=CC=C(Br)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)C4)=CC=C3C2=O)C(=O)N1	C41H37BrN4O6S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-D61CIB	SCHEMBL20442820	3-[6-[3-[[4-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenyl]piperidin-1-yl]methyl]azetidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(N4CC(CN5CCC(C6=CC=C(OC7=C(C8=CC=C(Br)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)C4)=CC=C3C2=O)C(=O)N1	C42H39BrN4O5S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-PFWD9M	SCHEMBL20442646	3-[2-[4-[[1-[4-[[2-(4-bromophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]-2,6-difluorophenyl]piperidin-4-yl]methyl]piperazin-1-yl]-5-oxo-7H-pyrrolo[3,4-b]pyridin-6-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC5CCN(C6=C(F)C=C(OC7=C(C8=CC=C(Br)C=C8)SC8=C7C=CC(O)=C8)C=C6F)CC5)CC4)=N3)C2=O)C(=O)N1	C42H39BrF2N6O5S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-ICZA1U	SCHEMBL20442750	3-[6-[4-[[1-[4-[[6-hydroxy-2-(4-hydroxyphenyl)-1-benzothiophen-3-yl]oxy]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC5CCN(C6=CC=C(OC7=C(C8=CC=C(O)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C43H43N5O6S	ERα;ERβ	P03372/Q92731	CRBN	WO-2018140809-A1
TPD-LBBBE9	SCHEMBL20423219	2-[7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]-N-[3-[3-[3-(2,4-dioxopyrimidin-1-yl)quinolin-6-yl]oxypropoxy]propyl]acetamide; SCHEMBL30479947	Cc1sc2c(c1C)C(c1ccc(Cl)cc1)=NC(CC(=O)NCCCOCCCOc1ccc3ncc(-n4ccc(=O)[nH]c4=O)cc3c1)c1nnc(C)n1-2	C38H37ClN8O5S	BRD4	O60885	CRBN	WO-2018144649-A1
TPD-0244J2	SCHEMBL20423423	2-[2-[2-[4-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenyl]piperazin-1-yl]ethoxy]ethylamino]-N-[2-(2,4-dioxo-1,3-diazinan-1-yl)ethyl]benzamide; SCHEMBL20423424	CC1(C)[C@H](NC(=O)c2ccc(N3CCN(CCOCCNc4ccccc4C(=O)NCCN4CCC(=O)NC4=O)CC3)cc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C43H53ClN8O6	AR	P10275	CRBN	WO-2018144649-A1
TPD-WZ3U6A	SCHEMBL20423392	3-[4-[4-[5-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]pentyl]piperazin-1-yl]-6-oxopyridazin-1-yl]piperidine-2,6-dione	O=C1CCC(n2ncc(N3CCN(CCCCCOc4ccc([C@@H]5c6ccc(O)cc6CC[C@@H]5c5ccccc5)cc4)CC3)cc2=O)C(=O)N1	C40H45N5O5	ERα	P03372	CRBN	WO-2018144649-A1
TPD-IMINMT	SCHEMBL20423440	3-[4-[4-[5-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]pentyl]piperazin-1-yl]-6-oxopyrimidin-1-yl]piperidine-2,6-dione	O=C1CCC(n2cnc(N3CCN(CCCCCOc4ccc([C@@H]5c6ccc(O)cc6CC[C@@H]5c5ccccc5)cc4)CC3)cc2=O)C(=O)N1	C40H45N5O5	ERα	P03372	CRBN	WO-2018144649-A1
TPD-O7JMJM	SCHEMBL20423299	3-[4-[4-[[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-6-oxopyridazin-1-yl]piperidine-2,6-dione; SCHEMBL30367194	O=C1CCC(n2ncc(N3CCN(CC4CCN(c5ccc([C@@H]6c7ccc(O)cc7CC[C@@H]6c6ccccc6)cc5)CC4)CC3)cc2=O)C(=O)N1	C41H46N6O4	ERα	P03372	CRBN	WO-2018144649-A1
TPD-8OV0RJ	SCHEMBL20423454	3-[4-[6-[(3R)-1-[2-[4-[(1R,2S)-2-(4-fluorophenyl)-6-hydroxy-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]ethyl]pyrrolidin-3-yl]oxypyridin-3-yl]oxy-6-oxopyridazin-1-yl]piperidine-2,6-dione; SCHEMBL30479964	O=C1CCC(n2ncc(Oc3ccc(O[C@@H]4CCN(CCOc5ccc([C@@H]6c7ccc(O)cc7CC[C@@H]6c6ccc(F)cc6)cc5)C4)nc3)cc2=O)C(=O)N1	C42H40FN5O7	ERα	P03372	CRBN	WO-2018144649-A1
TPD-QI2PI3	SCHEMBL20423124	3-[3-[3-[1-[4-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]butyl]piperidin-4-yl]phenoxy]-5-oxo-2H-pyrrol-1-yl]piperidine-2,6-dione	O=C1CCC(N2CC(Oc3cccc(C4CCN(CCCCOc5ccc([C@@H]6c7ccc(O)cc7CC[C@@H]6c6ccccc6)cc5)CC4)c3)=CC2=O)C(=O)N1	C46H49N3O6	ERα	P03372	CRBN	WO-2018144649-A1
TPD-D767QT	WO2018144649A1_PROTAC-105	.	O=C1CCC(N2CC(Oc3cccc(C4CCN(CCCOc5ccc(C6c7ccc(O)cc7CCC6c6ccccc6)cc5)CC4)c3)=CC2=O)C(=O)N1	C45H47N3O6	ERα	P03372	CRBN	WO-2018144649-A1
TPD-AZWQRQ	SCHEMBL20423583	3-[3-[3-[1-[3-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]propyl]piperidin-4-yl]phenoxy]-5-oxo-2H-pyrrol-1-yl]piperidine-2,6-dione; SCHEMBL30367078	O=C1CCC(N2CC(Oc3cccc(C4CCN(CCCOc5ccc([C@@H]6c7ccc(O)cc7CC[C@@H]6c6ccccc6)cc5)CC4)c3)=CC2=O)C(=O)N1	C45H47N3O6	ERα	P03372	CRBN	WO-2018144649-A1
TPD-1XU9D1	SCHEMBL20437066	3-[3-[3-[1-[4-[4-[(1S,2R)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]butyl]piperidin-4-yl]phenoxy]-5-oxo-2H-pyrrol-1-yl]piperidine-2,6-dione	O=C1CCC(N2CC(Oc3cccc(C4CCN(CCCCOc5ccc([C@H]6c7ccc(O)cc7CC[C@H]6c6ccccc6)cc5)CC4)c3)=CC2=O)C(=O)N1	C46H49N3O6	ERα	P03372	CRBN	WO-2018144649-A1
TPD-XVIDDO	SCHEMBL20423473	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-5-[4-[2-[[1,3-dioxo-2-(6-oxo-2-oxa-5-azaspiro[3.5]nonan-9-yl)isoindol-4-yl]amino]ethyl]piperazin-1-yl]pyridine-2-carboxamide; SCHEMBL20423474	CC1(C)[C@H](NC(=O)c2ccc(N3CCN(CCNc4cccc5c4C(=O)N(C4CCC(=O)NC46COC6)C5=O)CC3)cn2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C42H47ClN8O6	AR	P10275	CRBN	WO-2018144649-A1
TPD-Q6Q90O	SCHEMBL20423367	3-[4-[4-[4-[3-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]propyl]piperazin-1-yl]phenyl]pyrazol-1-yl]piperidine-2,6-dione	O=C1CCC(n2cc(-c3ccc(N4CCN(CCCOc5ccc([C@@H]6c7ccc(O)cc7CC[C@@H]6c6ccccc6)cc5)CC4)cc3)cn2)C(=O)N1	C43H45N5O4	ERα	P03372	CRBN	WO-2018144649-A1
TPD-6KSTZ2	SCHEMBL20423221	3-[4-[6-[4-[3-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]propyl]piperazin-1-yl]pyridin-3-yl]pyrazol-1-yl]piperidine-2,6-dione	O=C1CCC(n2cc(-c3ccc(N4CCN(CCCOc5ccc([C@@H]6c7ccc(O)cc7CC[C@@H]6c6ccccc6)cc5)CC4)nc3)cn2)C(=O)N1	C42H44N6O4	ERα	P03372	CRBN	WO-2018144649-A1
TPD-960WOB	SCHEMBL20423793	4-[4,4-Dimethyl-3-[4-[4-[3-[2-(1-methyl-2,4-dioxopyrimidin-5-yl)-1,3-dioxoisoindol-5-yl]oxypropyl]piperazin-1-yl]phenyl]-5-oxo-2-sulfanylideneimidazolidin-1-yl]-2-(trifluoromethyl)benzonitrile; ZCZXKMFPKVITSP-UHFFFAOYSA-N; 4-[4,4-Dimethyl-3-[4-[4-[3-[2-(1-methyl-2,4-dioxopyrimidin-5-yl)-1,3-dioxoisoindol-5-yl]oxypropyl]piperazin-1-yl]phenyl]-5-oxo-2-sulfanylideneimidazolidin-1-yl]-2-(trifluoromethyl)benzonitrile	Cn1cc(N2C(=O)c3ccc(OCCCN4CCN(c5ccc(N6C(=S)N(c7ccc(C#N)c(C(F)(F)F)c7)C(=O)C6(C)C)cc5)CC4)cc3C2=O)c(=O)[nH]c1=O	C39H35F3N8O6S	AR	P10275	CRBN	WO-2018144649-A1
TPD-FNCYSG	SCHEMBL20423449	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-5-[4-[2-[[2-(5,5-dimethyl-2,4-dioxoimidazolidin-1-yl)-3-oxo-2,5,6,7,8,8a-hexahydro-1H-indolizin-6-yl]amino]ethyl]piperazin-1-yl]pyridine-2-carboxamide; SCHEMBL20423450	CC1(C)C(=O)NC(=O)N1C1CC2CCC(NCCN3CCN(c4ccc(C(=O)N[C@H]5C(C)(C)[C@H](Oc6ccc(C#N)c(Cl)c6)C5(C)C)nc4)CC3)CN2C1=O	C40H52ClN9O5	AR	P10275	CRBN	WO-2018144649-A1
TPD-8HY050	SCHEMBL20423555	4-[3-[4-[3-[3-[4-(2,4-Dioxopyrimidin-1-yl)isoquinolin-7-yl]oxypropoxy]propylamino]phenyl]-4,4-dimethyl-5-oxo-2-sulfanylideneimidazolidin-1-yl]-2-(trifluoromethyl)benzonitrile; HJSLZUFWWHEKTD-UHFFFAOYSA-N; 4-[3-[4-[3-[3-[4-(2,4-Dioxopyrimidin-1-yl)isoquinolin-7-yl]oxypropoxy]propylamino]phenyl]-4,4-dimethyl-5-oxo-2-sulfanylideneimidazolidin-1-yl]-2-(trifluoromethyl)benzonitrile	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=S)N1c1ccc(NCCCOCCCOc2ccc3c(-n4ccc(=O)[nH]c4=O)cncc3c2)cc1	C38H34F3N7O5S	AR	P10275	CRBN	WO-2018144649-A1
TPD-T96U6X	SCHEMBL20423648	4-[3-[4-[2-[2-[2-[3-(2,4-Dioxopyrimidin-1-yl)-4-methylquinolin-7-yl]oxyethoxy]ethoxy]ethylamino]phenyl]-4,4-dimethyl-5-oxo-2-sulfanylideneimidazolidin-1-yl]-2-(trifluoromethyl)benzonitrile; MKZMPZHGXUGNLD-UHFFFAOYSA-N; 4-[3-[4-[2-[2-[2-[3-(2,4-Dioxopyrimidin-1-yl)-4-methylquinolin-7-yl]oxyethoxy]ethoxy]ethylamino]phenyl]-4,4-dimethyl-5-oxo-2-sulfanylideneimidazolidin-1-yl]-2-(trifluoromethyl)benzonitrile	Cc1c(-n2ccc(=O)[nH]c2=O)cnc2cc(OCCOCCOCCNc3ccc(N4C(=S)N(c5ccc(C#N)c(C(F)(F)F)c5)C(=O)C4(C)C)cc3)ccc12	C39H36F3N7O6S	AR	P10275	CRBN	WO-2018144649-A1
TPD-U1F255	SCHEMBL20423748	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[2-[2-[3-(2,4-dioxo-1,3-diazinan-1-yl)-4-methylquinolin-7-yl]oxyethoxy]ethoxy]benzamide; SCHEMBL20423749	Cc1c(N2CCC(=O)NC2=O)cnc2cc(OCCOCCOc3ccc(C(=O)N[C@H]4C(C)(C)[C@H](Oc5ccc(C#N)c(Cl)c5)C4(C)C)cc3)ccc12	C40H42ClN5O7	AR	P10275	CRBN	WO-2018144649-A1
TPD-2GJQFO	SCHEMBL20423254	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-5-[3-[4-[1,3-dioxo-2-(6-oxo-2-oxa-5-azaspiro[3.5]nonan-9-yl)isoindol-5-yl]piperazin-1-yl]propyl]pyridine-2-carboxamide; SCHEMBL20423255	CC1(C)[C@H](NC(=O)c2ccc(CCCN3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC46COC6)C5=O)CC3)cn2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C43H48ClN7O6	AR	P10275	CRBN	WO-2018144649-A1
TPD-ZX3FJA	SCHEMBL20423429	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[2-[2-[[1-(2,6-dioxopiperidin-3-yl)-6-oxopyridazin-4-yl]amino]ethoxy]ethyl]piperazin-1-yl]benzamide; SCHEMBL20423430	CC1(C)[C@H](NC(=O)c2ccc(N3CCN(CCOCCNc4cnn(C5CCC(=O)NC5=O)c(=O)c4)CC3)cc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C39H47ClN8O6	AR	P10275	CRBN	WO-2018144649-A1
TPD-4N58TY	SCHEMBL20423814	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[[1-[5-(2,4-dioxopyrimidin-1-yl)pyridin-3-yl]piperidin-4-yl]methyl]piperazin-1-yl]benzamide; SCHEMBL20423815	CC1(C)[C@H](NC(=O)c2ccc(N3CCN(CC4CCN(c5cncc(-n6ccc(=O)[nH]c6=O)c5)CC4)CC3)cc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C41H47ClN8O4	AR	P10275	CRBN	WO-2018144649-A1
TPD-HITJ8S	SCHEMBL20443584	2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]-N-[3-[3-[3-(2,4-dioxopyrimidin-1-yl)quinolin-5-yl]oxypropoxy]propyl]acetamide	Cc1sc2c(c1C)C(c1ccc(Cl)cc1)=N[C@@H](CC(=O)NCCCOCCCOc1cccc3ncc(-n4ccc(=O)[nH]c4=O)cc13)c1nnc(C)n1-2	C38H37ClN8O5S	AR	P10275	CRBN	WO-2018144649-A1
TPD-JU5T9X	SCHEMBL20423576	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[2-[4-[2-[1-(2,6-dioxopiperidin-3-yl)-6-oxopyridazin-4-yl]oxyethyl]piperazin-1-yl]ethoxy]butoxy]benzamide; SCHEMBL20423578	CC1(C)[C@H](NC(=O)c2ccc(OCCCCOCCN3CCN(CCOc4cnn(C5CCC(=O)NC5=O)c(=O)c4)CC3)cc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C43H54ClN7O8	AR	P10275	CRBN	WO-2018144649-A1
TPD-UIB80M	SCHEMBL20423366	2-[2-[2-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]piperazin-1-yl]ethoxy]ethylamino]-N-[2-(2,4-dioxo-1,3-diazinan-1-yl)ethyl]benzamide; GSTAZSYDRCXKLK-UHFFFAOYSA-N; 2-[2-[2-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]piperazin-1-yl]ethoxy]ethylamino]-N-[2-(2,4-dioxo-1,3-diazinan-1-yl)ethyl]benzamide	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=S)N1c1ccc(N2CCN(CCOCCNc3ccccc3C(=O)NCCN3CCC(=O)NC3=O)CC2)cc1	C40H44F3N9O5S	AR	P10275	CRBN	WO-2018144649-A1
TPD-JND8L9	SCHEMBL20423436	2-[2-[2-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]anilino]ethoxy]ethylamino]-N-[2-(2,4-dioxo-1,3-diazinan-1-yl)ethyl]benzamide; FWVLXBZLWQVBHP-UHFFFAOYSA-N; 2-[2-[2-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]anilino]ethoxy]ethylamino]-N-[2-(2,4-dioxo-1,3-diazinan-1-yl)ethyl]benzamide	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=S)N1c1ccc(-c2ccc(NCCOCCNc3ccccc3C(=O)NCCN3CCC(=O)NC3=O)cc2)cc1	C42H41F3N8O5S	AR	P10275	CRBN	WO-2018144649-A1
TPD-ZTLFX6	SCHEMBL20423181	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[2-[[1,3-dioxo-2-[2-oxo-6-(trifluoromethyl)piperidin-3-yl]isoindol-4-yl]amino]ethyl]piperazin-1-yl]benzamide; SCHEMBL20423182	CC1(C)[C@H](NC(=O)c2ccc(N3CCN(CCNc4cccc5c4C(=O)N(C4CCC(C(F)(F)F)NC4=O)C5=O)CC3)cc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C42H45ClF3N7O5	AR	P10275	CRBN	WO-2018144649-A1
TPD-UJQRGA	SCHEMBL20423608	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[2-[1,3-dioxo-2-[2-oxo-6-(trifluoromethyl)piperidin-3-yl]isoindol-5-yl]oxyethyl]piperazin-1-yl]benzamide; SCHEMBL20423609	CC1(C)[C@H](NC(=O)c2ccc(N3CCN(CCOc4ccc5c(c4)C(=O)N(C4CCC(C(F)(F)F)NC4=O)C5=O)CC3)cc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C42H44ClF3N6O6	AR	P10275	CRBN	WO-2018144649-A1
TPD-5RCTKR	SCHEMBL20423370	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[2-[[1,3-dioxo-2-[2-oxo-6-(trifluoromethyl)-1H-pyridin-3-yl]isoindol-4-yl]amino]ethyl]piperazin-1-yl]benzamide; SCHEMBL20423372	CC1(C)[C@H](NC(=O)c2ccc(N3CCN(CCNc4cccc5c4C(=O)N(c4ccc(C(F)(F)F)[nH]c4=O)C5=O)CC3)cc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C42H41ClF3N7O5	AR	P10275	CRBN	WO-2018144649-A1
TPD-9QNNIP	SCHEMBL20423364	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[2-[1,3-dioxo-2-[2-oxo-6-(trifluoromethyl)-1H-pyridin-3-yl]isoindol-5-yl]oxyethyl]piperazin-1-yl]benzamide; SCHEMBL20423365	CC1(C)[C@H](NC(=O)c2ccc(N3CCN(CCOc4ccc5c(c4)C(=O)N(c4ccc(C(F)(F)F)[nH]c4=O)C5=O)CC3)cc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C42H40ClF3N6O6	AR	P10275	CRBN	WO-2018144649-A1
TPD-24K75B	SCHEMBL20423118	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[5-[6-[(2,6-dioxopiperidin-3-yl)carbamoyl]pyridin-3-yl]oxypentyl]piperazin-1-yl]pyridine-3-carboxamide; SCHEMBL20423280	CC1(C)[C@H](NC(=O)c2ccc(N3CCN(CCCCCOc4ccc(C(=O)NC5CCC(=O)NC5=O)nc4)CC3)nc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C41H49ClN8O6	AR	P10275	CRBN	WO-2018144649-A1
TPD-NQYRMU	SCHEMBL20423151	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[5-[[3-(2,6-dioxopiperidin-3-yl)-2-methyl-4-oxo-1,2-dihydroquinazolin-8-yl]oxy]pentyl]piperazin-1-yl]pyridine-3-carboxamide; SCHEMBL20423152; SCHEMBL30479988; SCHEMBL30480016	CC1Nc2c(OCCCCCN3CCN(c4ccc(C(=O)N[C@H]5C(C)(C)[C@H](Oc6ccc(C#N)c(Cl)c6)C5(C)C)cn4)CC3)cccc2C(=O)N1C1CCC(=O)NC1=O	C44H53ClN8O6	AR	P10275	CRBN	WO-2018144649-A1
TPD-FOTZH6	SCHEMBL20423386	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[6-[1-(2,6-dioxopiperidin-3-yl)-6-oxopyridazin-4-yl]oxyhexyl]piperazin-1-yl]pyridine-3-carboxamide; SCHEMBL20423388	CC1(C)[C@H](NC(=O)c2ccc(N3CCN(CCCCCCOc4cnn(C5CCC(=O)NC5=O)c(=O)c4)CC3)nc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C40H49ClN8O6	AR	P10275	CRBN	WO-2018144649-A1
TPD-VDKXVU	SCHEMBL20423580	4-[3-[4-[2-[2-[2-[2-[5-Chloro-1-(2,6-dioxopiperidin-3-yl)-6-oxopyridazin-4-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]phenyl]-4,4-dimethyl-5-oxo-2-sulfanylideneimidazolidin-1-yl]-2-(trifluoromethyl)benzonitrile; VKJNHTHGFFRTPS-UHFFFAOYSA-N; 4-[3-[4-[2-[2-[2-[2-[5-Chloro-1-(2,6-dioxopiperidin-3-yl)-6-oxopyridazin-4-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]phenyl]-4,4-dimethyl-5-oxo-2-sulfanylideneimidazolidin-1-yl]-2-(trifluoromethyl)benzonitrile	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=S)N1c1ccc(OCCOCCOCCOCCOc2cnn(C3CCC(=O)NC3=O)c(=O)c2Cl)cc1	C36H36ClF3N6O9S	AR	P10275	CRBN	WO-2018144649-A1
TPD-EKQMHM	SCHEMBL20423202	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[5-[3-(2,6-dioxopiperidin-3-yl)-2-methyl-4-oxoquinazolin-8-yl]oxypentyl]piperazin-1-yl]pyridine-3-carboxamide; SCHEMBL20423203; SCHEMBL30479992	Cc1nc2c(OCCCCCN3CCN(c4ccc(C(=O)N[C@H]5C(C)(C)[C@H](Oc6ccc(C#N)c(Cl)c6)C5(C)C)cn4)CC3)cccc2c(=O)n1C1CCC(=O)NC1=O	C44H51ClN8O6	AR	P10275	CRBN	WO-2018144649-A1
TPD-NIZKCX	SCHEMBL20423389	4-[3-[4-[2-[4-[2-[[2-(2,6-Dioxopiperidin-3-yl)-1,1,3-trioxo-1,2-benzothiazol-6-yl]amino]ethyl]piperazin-1-yl]ethoxy]phenyl]-4,4-dimethyl-5-oxo-2-sulfanylideneimidazolidin-1-yl]-2-(trifluoromethyl)benzonitrile; KOJYAUKITKKWDD-UHFFFAOYSA-N; 4-[3-[4-[2-[4-[2-[[2-(2,6-Dioxopiperidin-3-yl)-1,1,3-trioxo-1,2-benzothiazol-6-yl]amino]ethyl]piperazin-1-yl]ethoxy]phenyl]-4,4-dimethyl-5-oxo-2-sulfanylideneimidazolidin-1-yl]-2-(trifluoromethyl)benzonitrile	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=S)N1c1ccc(OCCN2CCN(CCNc3ccc4c(c3)S(=O)(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)cc1	C39H39F3N8O7S2	AR	P10275	CRBN	WO-2018144649-A1
TPD-S07S74	SCHEMBL20423275	4-[3-[4-[2-[4-[2-[[2-(2,6-Dioxopiperidin-3-yl)-1,1,3-trioxo-1,2-benzothiazol-6-yl]oxy]ethyl]piperazin-1-yl]ethoxy]phenyl]-4,4-dimethyl-5-oxo-2-sulfanylideneimidazolidin-1-yl]-2-(trifluoromethyl)benzonitrile; FYJGRNBTYNLSOW-UHFFFAOYSA-N; 4-[3-[4-[2-[4-[2-[[2-(2,6-Dioxopiperidin-3-yl)-1,1,3-trioxo-1,2-benzothiazol-6-yl]oxy]ethyl]piperazin-1-yl]ethoxy]phenyl]-4,4-dimethyl-5-oxo-2-sulfanylideneimidazolidin-1-yl]-2-(trifluoromethyl)benzonitrile	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=S)N1c1ccc(OCCN2CCN(CCOc3ccc4c(c3)S(=O)(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)cc1	C39H38F3N7O8S2	AR	P10275	CRBN	WO-2018144649-A1
TPD-XBNYQ1	SCHEMBL20423268	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[5-[[2-(2,6-dioxopiperidin-3-yl)-1,1,3-trioxo-1,2-benzothiazol-6-yl]oxy]pentyl]piperazin-1-yl]pyridine-3-carboxamide; SCHEMBL20423579	CC1(C)[C@H](NC(=O)c2ccc(N3CCN(CCCCCOc4ccc5c(c4)S(=O)(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)nc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C42H48ClN7O8S	AR	P10275	CRBN	WO-2018144649-A1
TPD-OWXV7S	SCHEMBL20423192	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[5-[[2-(2,6-dioxopiperidin-3-yl)-1,1,3-trioxo-1,2-benzothiazol-6-yl]amino]pentyl]piperazin-1-yl]pyridine-3-carboxamide; SCHEMBL20443281	CC1(C)[C@H](NC(=O)c2ccc(N3CCN(CCCCCNc4ccc5c(c4)S(=O)(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)nc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C42H49ClN8O7S	AR	P10275	CRBN	WO-2018144649-A1
TPD-5L392C	SCHEMBL20423656	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[5-[[2-(2,6-dioxopiperidin-3-yl)-1,1,3-trioxo-1,2-benzothiazol-7-yl]amino]pentyl]piperazin-1-yl]pyridine-3-carboxamide; SCHEMBL20443529	CC1(C)[C@H](NC(=O)c2ccc(N3CCN(CCCCCNc4cccc5c4S(=O)(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)nc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C42H49ClN8O7S	AR	P10275	CRBN	WO-2018144649-A1
TPD-1ZS7FS	SCHEMBL20423311	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[5-[[2-(2,6-dioxopiperidin-3-yl)-1,1,3-trioxo-1,2-benzothiazol-7-yl]oxy]pentyl]piperazin-1-yl]pyridine-3-carboxamide; SCHEMBL20443527	CC1(C)[C@H](NC(=O)c2ccc(N3CCN(CCCCCOc4cccc5c4S(=O)(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)nc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C42H48ClN7O8S	AR	P10275	CRBN	WO-2018144649-A1
TPD-TPJ1S0	SCHEMBL20423693	4-[3-[4-[2-[2-[2-[[2-(2,6-Dioxopiperidin-3-yl)-1,1,3-trioxo-1,2-benzothiazol-6-yl]oxy]ethoxy]ethoxy]ethoxy]phenyl]-4,4-dimethyl-5-oxo-2-sulfanylideneimidazolidin-1-yl]-2-(trifluoromethyl)benzonitrile; ASKZGDQWPLCGQS-UHFFFAOYSA-N; 4-[3-[4-[2-[2-[2-[[2-(2,6-Dioxopiperidin-3-yl)-1,1,3-trioxo-1,2-benzothiazol-6-yl]oxy]ethoxy]ethoxy]ethoxy]phenyl]-4,4-dimethyl-5-oxo-2-sulfanylideneimidazolidin-1-yl]-2-(trifluoromethyl)benzonitrile	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=S)N1c1ccc(OCCOCCOCCOc2ccc3c(c2)S(=O)(=O)N(C2CCC(=O)NC2=O)C3=O)cc1	C37H34F3N5O10S2	AR	P10275	CRBN	WO-2018144649-A1
TPD-9Y5SSM	SCHEMBL20423300	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[3-[3-[[2-(2,6-dioxopiperidin-3-yl)-1,1,3-trioxo-1,2-benzothiazol-6-yl]oxy]propoxy]propoxy]pyridine-3-carboxamide; SCHEMBL20443528	CC1(C)[C@H](NC(=O)c2ccc(OCCCOCCCOc3ccc4c(c3)S(=O)(=O)N(C3CCC(=O)NC3=O)C4=O)nc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C39H42ClN5O10S	AR	P10275	CRBN	WO-2018144649-A1
TPD-TGEI5P	SCHEMBL20423399	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[2-[[2-(2,4-difluorophenyl)-1-oxo-3H-isoindol-4-yl]oxy]ethyl]piperazin-1-yl]pyridine-3-carboxamide; SCHEMBL20423400; SCHEMBL30480000	CC1(C)[C@H](NC(=O)c2ccc(N3CCN(CCOc4cccc5c4CN(c4ccc(F)cc4F)C5=O)CC3)nc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C41H41ClF2N6O4	AR	P10275	CRBN	WO-2018144649-A1
TPD-21VE2O	SCHEMBL20423354	4-[3-[4-[2-[2-[4-[2-[1-(2,6-Dioxopiperidin-3-yl)-6-oxopyridazin-4-yl]oxyethyl]piperazin-1-yl]ethoxy]ethoxy]phenyl]-4,4-dimethyl-5-oxo-2-sulfanylideneimidazolidin-1-yl]-2-(trifluoromethyl)benzonitrile; CVVFXBPIYLTBIM-UHFFFAOYSA-N; 4-[3-[4-[2-[2-[4-[2-[1-(2,6-Dioxopiperidin-3-yl)-6-oxopyridazin-4-yl]oxyethyl]piperazin-1-yl]ethoxy]ethoxy]phenyl]-4,4-dimethyl-5-oxo-2-sulfanylideneimidazolidin-1-yl]-2-(trifluoromethyl)benzonitrile	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=S)N1c1ccc(OCCOCCN2CCN(CCOc3cnn(C4CCC(=O)NC4=O)c(=O)c3)CC2)cc1	C38H41F3N8O7S	AR	P10275	CRBN	WO-2018144649-A1
TPD-5R4922	SCHEMBL20423874	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[2-[2-[[2-(2,4-difluorophenyl)-1-oxo-3H-isoindol-4-yl]oxy]ethoxy]ethyl]piperazin-1-yl]pyridine-3-carboxamide; SCHEMBL20423875; SCHEMBL30479978	CC1(C)[C@H](NC(=O)c2ccc(N3CCN(CCOCCOc4cccc5c4CN(c4ccc(F)cc4F)C5=O)CC3)nc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C43H45ClF2N6O5	AR	P10275	CRBN	WO-2018144649-A1
TPD-DDL42O	SCHEMBL20423197	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[5-[2-(2,4-difluorophenyl)-1,3-dioxoisoindol-5-yl]oxypentyl]piperazin-1-yl]pyridine-3-carboxamide; SCHEMBL20423199; SCHEMBL30480003	CC1(C)[C@H](NC(=O)c2ccc(N3CCN(CCCCCOc4ccc5c(c4)C(=O)N(c4ccc(F)cc4F)C5=O)CC3)nc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C44H45ClF2N6O5	AR	P10275	CRBN	WO-2018144649-A1
TPD-CGPO5Q	SCHEMBL20423320	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[5-[2-(6-cyano-2-oxo-1H-pyridin-3-yl)-1,3-dioxoisoindol-5-yl]oxypentyl]piperazin-1-yl]pyridine-3-carboxamide; SCHEMBL20423322; SCHEMBL20423544; SCHEMBL20423546; SCHEMBL30479944	CC1(C)[C@H](NC(=O)c2ccc(N3CCN(CCCCCOc4ccc5c(c4)C(=O)N(c4ccc(C#N)[nH]c4=O)C5=O)CC3)nc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C44H45ClN8O6	AR	P10275	CRBN	WO-2018144649-A1
TPD-HY5TE1	SCHEMBL20423808	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[[4-[1,3-dioxo-2-(6-oxo-1H-pyridin-3-yl)isoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]benzamide; SCHEMBL20423811; SCHEMBL30479969	CC1(C)[C@H](NC(=O)c2ccc(N3CCC(CN4CCN(c5ccc6c(c5)C(=O)N(c5ccc(=O)[nH]c5)C6=O)CC4)CC3)cc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C45H48ClN7O5	AR	P10275	CRBN	WO-2018144649-A1
TPD-OHD9FC	SCHEMBL20423623	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[[4-[1,3-dioxo-2-(2-oxo-1H-pyridin-3-yl)isoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]benzamide; SCHEMBL20423625; SCHEMBL30479954	CC1(C)[C@H](NC(=O)c2ccc(N3CCC(CN4CCN(c5ccc6c(c5)C(=O)N(c5ccc[nH]c5=O)C6=O)CC4)CC3)cc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C45H48ClN7O5	AR	P10275	CRBN	WO-2018144649-A1
TPD-6UDSN3	SCHEMBL20423227	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[[4-[2-(2-hydroxy-6-oxo-1H-pyridin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]benzamide; SCHEMBL20423228; SCHEMBL30479955	CC1(C)[C@H](NC(=O)c2ccc(N3CCC(CN4CCN(c5ccc6c(c5)C(=O)N(c5ccc(O)[nH]c5=O)C6=O)CC4)CC3)cc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C45H48ClN7O6	AR	P10275	CRBN	WO-2018144649-A1
TPD-QENPEC	SCHEMBL20423380	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxoisoquinolin-3-yl]methoxy]ethoxy]ethyl]piperazin-1-yl]pyridine-3-carboxamide; SCHEMBL20423382	CC1(C)[C@H](NC(=O)c2ccc(N3CCN(CCOCCOCc4cc5ccccc5c(=O)n4C4CCC(=O)NC4=O)CC3)nc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C44H50ClN7O7	AR	P10275	CRBN	WO-2018144649-A1
TPD-Z32HJR	SCHEMBL20423244	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[5-[3-(2,4-dioxopyrimidin-1-yl)quinolin-6-yl]oxypentyl]piperazin-1-yl]pyridine-3-carboxamide; SCHEMBL20423245; SCHEMBL30479959	CC1(C)[C@H](NC(=O)c2ccc(N3CCN(CCCCCOc4ccc5ncc(-n6ccc(=O)[nH]c6=O)cc5c4)CC3)nc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C43H47ClN8O5	AR	P10275	CRBN	WO-2018144649-A1
TPD-FTADPY	SCHEMBL20423483	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[5-[4-[(2,6-dioxopiperidin-3-yl)-ethylcarbamoyl]phenoxy]pentyl]piperazin-1-yl]pyridine-3-carboxamide; SCHEMBL20423484	CCN(C(=O)c1ccc(OCCCCCN2CCN(c3ccc(C(=O)N[C@H]4C(C)(C)[C@H](Oc5ccc(C#N)c(Cl)c5)C4(C)C)cn3)CC2)cc1)C1CCC(=O)NC1=O	C44H54ClN7O6	AR	P10275	CRBN	WO-2018144649-A1
TPD-HB298H	SCHEMBL20423839	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[5-[4-[(2,6-dioxopiperidin-3-yl)-methylcarbamoyl]phenoxy]pentyl]piperazin-1-yl]pyridine-3-carboxamide	CN(C(=O)c1ccc(OCCCCCN2CCN(c3ccc(C(=O)N[C@H]4C(C)(C)[C@H](Oc5ccc(C#N)c(Cl)c5)C4(C)C)cn3)CC2)cc1)C1CCC(=O)NC1=O	C43H52ClN7O6	AR	P10275	CRBN	WO-2018144649-A1
TPD-3NJNGB	SCHEMBL20423586	4-[3-[4-[2-[4-[2-[5-Chloro-1-(2,6-dioxopiperidin-3-yl)-6-oxopyridazin-4-yl]oxyethyl]piperazin-1-yl]ethoxy]phenyl]-4,4-dimethyl-5-oxo-2-sulfanylideneimidazolidin-1-yl]-2-(trifluoromethyl)benzonitrile; QFDZLZVCFCCSRO-UHFFFAOYSA-N; 4-[3-[4-[2-[4-[2-[5-Chloro-1-(2,6-dioxopiperidin-3-yl)-6-oxopyridazin-4-yl]oxyethyl]piperazin-1-yl]ethoxy]phenyl]-4,4-dimethyl-5-oxo-2-sulfanylideneimidazolidin-1-yl]-2-(trifluoromethyl)benzonitrile	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=S)N1c1ccc(OCCN2CCN(CCOc3cnn(C4CCC(=O)NC4=O)c(=O)c3Cl)CC2)cc1	C36H36ClF3N8O6S	AR	P10275	CRBN	WO-2018144649-A1
TPD-BEBXAQ	SCHEMBL20423272	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[3-[6-[(2,6-dioxopiperidin-3-yl)carbamoyl]pyridin-3-yl]oxypropyl]piperazin-1-yl]pyridine-3-carboxamide; SCHEMBL20423273	CC1(C)[C@H](NC(=O)c2ccc(N3CCN(CCCOc4ccc(C(=O)NC5CCC(=O)NC5=O)nc4)CC3)nc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C39H45ClN8O6	AR	P10275	CRBN	WO-2018144649-A1
TPD-DXJXQ9	SCHEMBL20423442	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[4-[6-[(2,6-dioxopiperidin-3-yl)carbamoyl]pyridin-3-yl]oxybutyl]piperazin-1-yl]pyridine-3-carboxamide; SCHEMBL20423444	CC1(C)[C@H](NC(=O)c2ccc(N3CCN(CCCCOc4ccc(C(=O)NC5CCC(=O)NC5=O)nc4)CC3)nc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C40H47ClN8O6	AR	P10275	CRBN	WO-2018144649-A1
TPD-ZEP93S	SCHEMBL20423359	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[2-[4-[6-[(2,6-dioxopiperidin-3-yl)carbamoyl]pyridin-3-yl]piperazin-1-yl]ethyl]piperidin-1-yl]pyridine-3-carboxamide	CC1(C)[C@H](NC(=O)c2ccc(N3CCC(CCN4CCN(c5ccc(C(=O)NC6CCC(=O)NC6=O)nc5)CC4)CC3)nc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C43H52ClN9O5	AR	P10275	CRBN	WO-2018144649-A1
TPD-NDZM03	SCHEMBL20423542	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[[4-[6-[(2,6-dioxopiperidin-3-yl)carbamoyl]pyridin-3-yl]piperazin-1-yl]methyl]piperidin-1-yl]pyridine-3-carboxamide; SCHEMBL20423543	CC1(C)[C@H](NC(=O)c2ccc(N3CCC(CN4CCN(c5ccc(C(=O)NC6CCC(=O)NC6=O)nc5)CC4)CC3)nc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C42H50ClN9O5	AR	P10275	CRBN	WO-2018144649-A1
TPD-7YX3P6	SCHEMBL20423256	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[[4-[6-[(2,6-dioxopiperidin-3-yl)carbamoyl]pyridin-3-yl]piperazin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL20423257	CC1(C)[C@H](NC(=O)c2ccc(N3CCC(CN4CCN(c5ccc(C(=O)NC6CCC(=O)NC6=O)nc5)CC4)CC3)nn2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C41H49ClN10O5	AR	P10275	CRBN	WO-2018144649-A1
TPD-HJYEHI	SCHEMBL20423893	5-[4-[[1-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-N-(2,6-dioxopiperidin-3-yl)pyridine-2-carboxamide; SCHEMBL20423894	CC1(C)[C@H](NC(=O)c2ccc(N3CCC(CN4CCN(c5ccc(C(=O)NC6CCC(=O)NC6=O)nc5)CC4)CC3)cc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C43H51ClN8O5	AR	P10275	CRBN	WO-2018144649-A1
TPD-5YPMGO	SCHEMBL20423443	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-5-[4-[[4-[6-[(2,6-dioxopiperidin-3-yl)carbamoyl]pyridin-3-yl]piperazin-1-yl]methyl]piperidin-1-yl]pyrazine-2-carboxamide; SCHEMBL20423445	CC1(C)[C@H](NC(=O)c2cnc(N3CCC(CN4CCN(c5ccc(C(=O)NC6CCC(=O)NC6=O)nc5)CC4)CC3)cn2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C41H49ClN10O5	AR	P10275	CRBN	WO-2018144649-A1
TPD-A8GP63	WO2018144649A1_PROTAC-57	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCN(c6cc7c(=O)on(C8CCC(=O)NC8=O)c(=O)c7cc6F)CC5)CC4)nn3)CC2)cc1Cl	C41H43ClFN9O7	AR	P10275	CRBN	WO-2018144649-A1
TPD-YN2QQT	WO2018144649A1_PROTAC-58	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCN(c6cc7c(=O)n(C8CCC(=O)NC8=O)oc(=O)c7cc6F)CC5)CC4)nn3)CC2)cc1Cl	C41H43ClFN9O7	AR	P10275	CRBN	WO-2018144649-A1
TPD-1BLT58	SCHEMBL20423146	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[[4-[4-[(2,6-dioxopiperidin-3-yl)carbamoyl]phenyl]piperazin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL20423147; SCHEMBL30159782	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCN(c6ccc(C(=O)NC7CCC(=O)NC7=O)cc6)CC5)CC4)nn3)CC2)cc1Cl	C40H46ClN9O5	AR	P10275	CRBN	WO-2018144649-A1
TPD-ICJOC6	SCHEMBL20423475	5-[5-[4-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]ethyl]piperazin-1-yl]-1,3-dioxoisoindol-2-yl]-6-oxo-1H-pyridine-2-carbonitrile; CFMZBYCSPKSSQX-UHFFFAOYSA-N; 5-[5-[4-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]ethyl]piperazin-1-yl]-1,3-dioxoisoindol-2-yl]-6-oxo-1H-pyridine-2-carbonitrile	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=S)N1c1ccc(OCCN2CCN(c3ccc4c(c3)C(=O)N(c3ccc(C#N)[nH]c3=O)C4=O)CC2)cc1	C39H31F3N8O5S	AR	P10275	CRBN	WO-2018144649-A1
TPD-IOOOEQ	SCHEMBL20423758	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[3-[1-(2,6-dioxopiperidin-3-yl)-6-oxopyridazin-4-yl]oxypropyl]piperazin-1-yl]pyridine-3-carboxamide; SCHEMBL20423759	CC1(C)[C@H](NC(=O)c2ccc(N3CCN(CCCOc4cnn(C5CCC(=O)NC5=O)c(=O)c4)CC3)nc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C37H43ClN8O6	AR	P10275	CRBN	WO-2018144649-A1
TPD-C0U2VG	SCHEMBL20423269	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[4-[1-(2,6-dioxopiperidin-3-yl)-6-oxopyridazin-4-yl]piperazin-1-yl]butyl]pyridine-3-carboxamide; SCHEMBL20423310	CC1(C)[C@H](NC(=O)c2ccc(CCCCN3CCN(c4cnn(C5CCC(=O)NC5=O)c(=O)c4)CC3)nc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C38H45ClN8O5	AR	P10275	CRBN	WO-2018144649-A1
TPD-HTK65R	SCHEMBL20423558	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[[4-[1-(2,6-dioxopiperidin-3-yl)-6-oxopyridazin-4-yl]piperazin-1-yl]methyl]piperidin-1-yl]benzamide; SCHEMBL20423559	CC1(C)[C@H](NC(=O)c2ccc(N3CCC(CN4CCN(c5cnn(C6CCC(=O)NC6=O)c(=O)c5)CC4)CC3)cc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C41H49ClN8O5	AR	P10275	CRBN	WO-2018144649-A1
TPD-OPOYCK	WO2018144649A1_PROTAC-63	.	CC1(C)[C@H](NC(=O)c2ccc(N3CCC(CCN4CCN(c5cnn(C6CCC(=O)NC6=O)c(=O)c5)CC4)CC3)nc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C41H50ClN9O5	AR	P10275	CRBN	WO-2018144649-A1
TPD-RIO074	SCHEMBL20423681	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[[4-[2-(2,5-dioxopyrrolidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]benzamide; SCHEMBL20423685; SCHEMBL30479962	CC1(C)[C@H](NC(=O)c2ccc(N3CCC(CN4CCN(c5ccc6c(c5)C(=O)N(C5CC(=O)NC5=O)C6=O)CC4)CC3)cc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C44H48ClN7O6	AR	P10275	CRBN	WO-2018144649-A1
TPD-8D9VYU	WO2018144649A1_PROTAC-67	.	CC1(C)[C@H](NC(=O)c2ccc(N3CCN(CCCCCOc4cccc(-c5nn(C6CCC(=O)NC6=O)c(=O)[nH]5)c4)CC3)cc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C44H51ClN8O6	AR	P10275	CRBN	WO-2018144649-A1
TPD-1M439P	SCHEMBL20423447	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[[4-[3-[1-(2,6-dioxopiperidin-3-yl)-4-methyl-5-oxo-1,2,4-triazol-3-yl]phenyl]piperazin-1-yl]methyl]piperidin-1-yl]benzamide	Cn1c(-c2cccc(N3CCN(CC4CCN(c5ccc(C(=O)N[C@H]6C(C)(C)[C@H](Oc7ccc(C#N)c(Cl)c7)C6(C)C)cc5)CC4)CC3)c2)nn(C2CCC(=O)NC2=O)c1=O	C46H54ClN9O5	AR	P10275	CRBN	WO-2018144649-A1
TPD-W23EPT	SCHEMBL20423650	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[5-[4-[1-(2,6-dioxopiperidin-3-yl)-4-methyl-5-oxo-1,2,4-triazol-3-yl]phenoxy]pentyl]piperazin-1-yl]benzamide	Cn1c(-c2ccc(OCCCCCN3CCN(c4ccc(C(=O)N[C@H]5C(C)(C)[C@H](Oc6ccc(C#N)c(Cl)c6)C5(C)C)cc4)CC3)cc2)nn(C2CCC(=O)NC2=O)c1=O	C45H53ClN8O6	AR	P10275	CRBN	WO-2018144649-A1
TPD-4WX3PW	SCHEMBL20423371	4-[3-[4-[2-[4-[[1-[5-(2,4-Dioxopyrimidin-1-yl)pyridin-3-yl]piperidin-4-yl]methyl]piperazin-1-yl]ethoxy]phenyl]-4,4-dimethyl-5-oxo-2-sulfanylideneimidazolidin-1-yl]-2-(trifluoromethyl)benzonitrile; GSFAXFFNLMJSEN-UHFFFAOYSA-N; 4-[3-[4-[2-[4-[[1-[5-(2,4-Dioxopyrimidin-1-yl)pyridin-3-yl]piperidin-4-yl]methyl]piperazin-1-yl]ethoxy]phenyl]-4,4-dimethyl-5-oxo-2-sulfanylideneimidazolidin-1-yl]-2-(trifluoromethyl)benzonitrile	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=S)N1c1ccc(OCCN2CCN(CC3CCN(c4cncc(-n5ccc(=O)[nH]c5=O)c4)CC3)CC2)cc1	C40H42F3N9O4S	AR	P10275	CRBN	WO-2018144649-A1
TPD-1EPF22	SCHEMBL20423337	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxoisoquinolin-6-yl]piperazin-1-yl]methyl]piperidin-1-yl]benzamide; SCHEMBL20423401; SCHEMBL30479985	CC1(C)[C@H](NC(=O)c2ccc(N3CCC(CN4CCN(c5ccc6c(=O)n(C7CCC(=O)NC7=O)ccc6c5)CC4)CC3)cc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C46H52ClN7O5	AR	P10275	CRBN	WO-2018144649-A1
TPD-YVB1YT	SCHEMBL20423755	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-2,8-diazaspiro[4.5]decan-8-yl]methyl]piperidin-1-yl]benzamide; SCHEMBL20423756	CC1(C)[C@H](NC(=O)c2ccc(N3CCC(CN4CCC5(CC4)CC(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)cc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C41H49ClN6O6	AR	P10275	CRBN	WO-2018144649-A1
TPD-ODCERZ	SCHEMBL20423335	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-2,8-diazaspiro[4.5]decan-8-yl]propyl]benzamide; SCHEMBL20423338	CC1(C)[C@H](NC(=O)c2ccc(CCCN3CCC4(CC3)CC(=O)N(C3CCC(=O)NC3=O)C4=O)cc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C38H44ClN5O6	AR	P10275	CRBN	WO-2018144649-A1
TPD-OVMZXM	SCHEMBL20423606	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[(E)-3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-2,8-diazaspiro[4.5]decan-8-yl]prop-1-enyl]benzamide	CC1(C)[C@H](NC(=O)c2ccc(/C=C/CN3CCC4(CC3)CC(=O)N(C3CCC(=O)NC3=O)C4=O)cc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C38H42ClN5O6	AR	P10275	CRBN	WO-2018144649-A1
TPD-62ZNEL	SCHEMBL20423527	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-2,8-diazaspiro[4.5]decan-8-yl]butyl]benzamide; SCHEMBL20423528	CC1(C)[C@H](NC(=O)c2ccc(CCCCN3CCC4(CC3)CC(=O)N(C3CCC(=O)NC3=O)C4=O)cc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C39H46ClN5O6	AR	P10275	CRBN	WO-2018144649-A1
TPD-0YS981	SCHEMBL20423121	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[5-[4-(2,4-dioxopyrimidin-1-yl)isoquinolin-7-yl]oxypentyl]piperazin-1-yl]pyridine-3-carboxamide; SCHEMBL20423123; SCHEMBL30479966	CC1(C)[C@H](NC(=O)c2ccc(N3CCN(CCCCCOc4ccc5c(-n6ccc(=O)[nH]c6=O)cncc5c4)CC3)nc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C43H47ClN8O5	AR	P10275	CRBN	WO-2018144649-A1
TPD-G5CWZA	SCHEMBL20423229	4-[3-[4-[3-[3-[3-(2,4-Dioxopyrimidin-1-yl)quinolin-5-yl]oxypropoxy]propylamino]phenyl]-4,4-dimethyl-5-oxo-2-sulfanylideneimidazolidin-1-yl]-2-(trifluoromethyl)benzonitrile; DCWCYBQBRIUKSF-UHFFFAOYSA-N; 4-[3-[4-[3-[3-[3-(2,4-Dioxopyrimidin-1-yl)quinolin-5-yl]oxypropoxy]propylamino]phenyl]-4,4-dimethyl-5-oxo-2-sulfanylideneimidazolidin-1-yl]-2-(trifluoromethyl)benzonitrile	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=S)N1c1ccc(NCCCOCCCOc2cccc3ncc(-n4ccc(=O)[nH]c4=O)cc23)cc1	C38H34F3N7O5S	AR	P10275	CRBN	WO-2018144649-A1
TPD-R6L3SZ	SCHEMBL20423154	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[5-[3-(5-cyano-2,4-dioxopyrimidin-1-yl)quinolin-6-yl]oxypentyl]piperazin-1-yl]pyridine-3-carboxamide; SCHEMBL20423155; SCHEMBL30479996	CC1(C)[C@H](NC(=O)c2ccc(N3CCN(CCCCCOc4ccc5ncc(-n6cc(C#N)c(=O)[nH]c6=O)cc5c4)CC3)nc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C44H46ClN9O5	AR	P10275	CRBN	WO-2018144649-A1
TPD-GMPK2P	SCHEMBL20423829	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-4-methylidene-1-oxo-3H-isoquinolin-6-yl]piperazin-1-yl]methyl]piperidin-1-yl]benzamide; SCHEMBL20423873	C=C1CN(C2CCC(=O)NC2=O)C(=O)c2ccc(N3CCN(CC4CCN(c5ccc(C(=O)N[C@H]6C(C)(C)[C@H](Oc7ccc(C#N)c(Cl)c7)C6(C)C)cc5)CC4)CC3)cc21	C47H54ClN7O5	AR	P10275	CRBN	WO-2018144649-A1
TPD-C3OYBH	SCHEMBL20423413	3-[3-[4-[4-[[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]phenyl]-5-oxo-2H-pyrrol-1-yl]piperidine-2,6-dione; SCHEMBL30479972	O=C1CCC(N2CC(c3ccc(N4CCN(CC5CCN(c6ccc([C@@H]7c8ccc(O)cc8CC[C@@H]7c7ccccc7)cc6)CC5)CC4)cc3)=CC2=O)C(=O)N1	C47H51N5O4	ERα	P03372	CRBN	WO-2018144649-A1
TPD-YO9W6X	WO2018144649A1_PROTAC-9	.	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=S)N1c1ccc(N2CCN(CCCCNc3ccc4ncc(-n5ccc(=O)[nH]c5=O)cc4c3)CC2)cc1	C40H38F3N9O3S	AR	P10275	CRBN	WO-2018144649-A1
TPD-6H7CS7	SCHEMBL20423350	N-(2,6-dioxopiperidin-3-yl)-4-[4-[5-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]pentyl]piperazin-1-yl]-N-methylbenzamide	CN(C(=O)c1ccc(N2CCN(CCCCCOc3ccc([C@@H]4c5ccc(O)cc5CC[C@@H]4c4ccccc4)cc3)CC2)cc1)C1CCC(=O)NC1=O	C44H50N4O5	ERα	P03372	CRBN	WO-2018144649-A1
TPD-E3GU75	SCHEMBL20423560	N-(2,6-dioxopiperidin-3-yl)-5-[4-[5-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]pentyl]piperazin-1-yl]pyridine-2-carboxamide	O=C1CCC(NC(=O)c2ccc(N3CCN(CCCCCOc4ccc([C@@H]5c6ccc(O)cc6CC[C@@H]5c5ccccc5)cc4)CC3)cn2)C(=O)N1	C42H47N5O5	ERα	P03372	CRBN	WO-2018144649-A1
TPD-9DD1TR	SCHEMBL20423188	N-(2,6-dioxopiperidin-3-yl)-N-ethyl-4-[4-[5-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]pentyl]piperazin-1-yl]-2-methoxybenzamide	CCN(C(=O)c1ccc(N2CCN(CCCCCOc3ccc([C@@H]4c5ccc(O)cc5CC[C@@H]4c4ccccc4)cc3)CC2)cc1OC)C1CCC(=O)NC1=O	C46H54N4O6	ERα	P03372	CRBN	WO-2018144649-A1
TPD-5AU2MB	WO2018144649A1_PROTAC-93	.	O=C1CCC(n2ncc(Oc3ccc(OC4CCN(CCOc5ccc(C6c7ccc(O)cc7CCC6c6ccc(F)cc6)cc5)C4)nc3)cc2=O)C(=O)N1	C42H40FN5O7	ERα	P03372	CRBN	WO-2018144649-A1
TPD-XP0E6L	SCHEMBL20423456	3-[4-[6-[1-[2-[4-[(1R,2S)-2-(4-fluorophenyl)-6-hydroxy-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]ethyl]pyrrolidin-3-yl]oxypyridin-3-yl]oxy-6-oxopyridazin-1-yl]piperidine-2,6-dione	O=C1CCC(n2ncc(Oc3ccc(OC4CCN(CCOc5ccc([C@@H]6c7ccc(O)cc7CC[C@@H]6c6ccc(F)cc6)cc5)C4)nc3)cc2=O)C(=O)N1	C42H40FN5O7	ERα	P03372	CRBN	WO-2018144649-A1
TPD-TMUJXT	WO2018144649A1_PROTAC-95	.	O=C1CCC(n2ncc(Oc3ccc(N4CCN(CCOc5ccc(C6c7ccc(O)cc7CCC6c6ccc(F)cc6)cc5)CC4)nc3)cc2=O)C(=O)N1	C42H41FN6O6	ERα	P03372	CRBN	WO-2018144649-A1
TPD-3TCYZT	SCHEMBL20423276	3-[4-[6-[4-[2-[4-[(1R,2S)-2-(4-fluorophenyl)-6-hydroxy-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]ethyl]piperazin-1-yl]pyridin-3-yl]oxy-6-oxopyridazin-1-yl]piperidine-2,6-dione	O=C1CCC(n2ncc(Oc3ccc(N4CCN(CCOc5ccc([C@@H]6c7ccc(O)cc7CC[C@@H]6c6ccc(F)cc6)cc5)CC4)nc3)cc2=O)C(=O)N1	C42H41FN6O6	ERα	P03372	CRBN	WO-2018144649-A1
TPD-LOZR68	WO2018144649A1_PROTAC-97	.	O=C1CCC(n2ncc(Oc3ccc(O[C@@H]4CCN(CCOc5ccc(C6c7ccc(O)cc7CCC6c6ccc(F)cc6)cc5)C4)nc3)cc2=O)C(=O)N1	C42H40FN5O7	ERα	P03372	CRBN	WO-2018144649-A1
TPD-7G6CPH	SCHEMBL20423773	3-[4-[6-[4-[4-[(1R,2S)-2-(4-fluorophenyl)-6-hydroxy-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]butyl]pyridin-3-yl]oxy-6-oxopyridazin-1-yl]piperidine-2,6-dione	O=C1CCC(n2ncc(Oc3ccc(CCCCOc4ccc([C@@H]5c6ccc(O)cc6CC[C@@H]5c5ccc(F)cc5)cc4)nc3)cc2=O)C(=O)N1	C40H37FN4O6	ERα	P03372	CRBN	WO-2018144649-A1
TPD-LF7EDS	SCHEMBL20423805	3-[4-[6-[5-[4-[(1R,2S)-2-(4-fluorophenyl)-6-hydroxy-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]pentyl]pyridin-3-yl]oxy-6-oxopyridazin-1-yl]piperidine-2,6-dione	O=C1CCC(n2ncc(Oc3ccc(CCCCCOc4ccc([C@@H]5c6ccc(O)cc6CC[C@@H]5c5ccc(F)cc5)cc4)nc3)cc2=O)C(=O)N1	C41H39FN4O6	ERα	P03372	CRBN	WO-2018144649-A1
TPD-4K7XQJ	WO2019023553A1_1	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@H](O)CN3C(=O)[C@@H](NC(=O)COCCCOCCCCCOC3=CC=C(N4C(=S)N(C5=CC(C(F)(F)F)=C(C#N)C=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C51H60F3N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-6IMYLS	CHEMBL4646619	(2S,4R)-1-[(2S)-2-[2-(3-{[5-(4-{3-[6-cyano-5-(trifluoromethyl)pyridin-3-yl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl}phenoxy)pentyl]oxy}propoxy)acetamido]-3,3-dimethylbutanoyl]-4-hydroxy-N-{[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl}pyrrolidine-2-carboxamide; SCHEMBL17940908; SCHEMBL29817430; PD140694	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCOCCCCCOC3=CC=C(N4C(=S)N(C5=CC(C(F)(F)F)=C(C#N)N=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C50H59F3N8O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-AK3CGP	WO2019023553A1_3	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCOCCCCCOC3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3F)C(C)(C)C)C=C2)SC=N1	C51H59F4N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-ZPD7CB	WO2019023553A1_4	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCOCCCCCOC3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C52H62F3N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-6Q283P	WO2019023553A1_5	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCOCCCCCOC3=CC=C(N4C(=S)N(C5=CC=C([N+](=O)[O-])C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C50H60F3N7O10S2	AR	P10275	VHL	WO-2019023553-A1
TPD-FKPDVW	WO2019023553A1_6	.	CC1=CC(N2C(=O)C(C)(C)N(C3=CC=C(OCCCCCOCCCOCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)NCC4=CC=C(C5=C(C)N=CS5)C=C4)C(C)(C)C)C=C3)C2=S)=CC(C)=C1C#N	C52H65N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-Q7Q2GY	SCHEMBL17946912	(2S,4R)-1-[(2S)-2-[[2-[3-[5-[4-[3-(4-cyano-3-fluorophenyl)-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]pentoxy]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCOCCCCCOC3=CC=C(N4C(=S)N(C5=CC(F)=C(C#N)C=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C50H60FN7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-W4FTRO	SCHEMBL17947445	(2S,4R)-1-[(2S)-2-[[2-[3-[5-[4-[3-(3-chloro-4-cyanophenyl)-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]pentoxy]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCOCCCCCOC3=CC=C(N4C(=S)N(C5=CC(Cl)=C(C#N)C=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C50H60ClN7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-CLOB7A	SCHEMBL17947522	(2S,4R)-1-[(2S)-2-[[2-[3-[5-[4-[3-(4-cyano-3-methoxyphenyl)-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]pentoxy]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	COC1=C(C#N)C=CC(N2C(=O)C(C)(C)N(C3=CC=C(OCCCCCOCCCOCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)NCC4=CC=C(C5=C(C)N=CS5)C=C4)C(C)(C)C)C=C3)C2=S)=C1	C51H63N7O9S2	AR	P10275	VHL	WO-2019023553-A1
TPD-VAU3R3	WO2019023553A1_10	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCOCCCCCOC3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3F)C(C)(C)C)C=C2)SC=N1	C52H61F4N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-ZUDGZY	CHEMBL4638782	(2S,4R)-1-[(2S)-2-[[2-[3-[5-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]-2,6-difluorophenoxy]pentoxy]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL17946883; SCHEMBL29817595; DKNBVZGJLBYCQJ-YCDRFOERSA-N; PD140690; (2S,4R)-1-[(2S)-2-[[2-[3-[5-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]-2,6-difluorophenoxy]pentoxy]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCOCCCCCOC3=C(F)C=C(N4C(=S)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3F)C(C)(C)C)C=C2)SC=N1	C52H60F5N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-89Q7D8	SCHEMBL17947128	(2S,4R)-1-[(2S)-2-[[2-[3-[5-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]-3,3-dimethylpentoxy]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL29817160; YWEHGWGIBLBFBJ-BZPYCXPJSA-N; (2S,4R)-1-[(2S)-2-[[2-[3-[5-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]-3,3-dimethylpentoxy]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCOCCC(C)(C)CCOC3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C53H64F3N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-DEP7HO	WO2019023553A1_13	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCOCCC(O)CCOC3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C51H60F3N7O9S2	AR	P10275	VHL	WO-2019023553-A1
TPD-11NTCP	WO2019023553A1_14	.	CC(C)(C)[C@H](NC(=O)COCCCOCCCCCOC1=CC=C(N2C(=S)N(C3=CC(C(F)(F)F)=C(C#N)C=C3)C(=O)C2(C)C)C=C1)C(=O)N1C[C@@H](O)C[C@H]1C(=O)NCC1=CC=C(Cl)C=C1	C47H56ClF3N6O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-IXFF6R	WO2019023553A1_15	.	CC(C)(C)[C@H](NC(=O)COCCCOCCCCCOC1=CC=C(N2C(=S)N(C3=CC=C(C#N)C(C(F)(F)F)=C3)C(=O)C2(C)C)C=C1)C(=O)N1C[C@@H](O)C[C@H]1C(=O)NCC1=CC=C(C#N)C=C1	C48H56F3N7O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-IRD4CU	WO2019023553A1_16	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOC3=CC=C(N4C(=S)N(C5=CC(C(F)(F)F)=C(C#N)C=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C49H56F3N7O9S2	AR	P10275	VHL	WO-2019023553-A1
TPD-AVWZHM	WO2019023553A1_17	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOC3=CC=C(N4C(=O)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C49H56F3N7O10S	AR	P10275	VHL	WO-2019023553-A1
TPD-L6L7SF	SCHEMBL17947130	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]-2-fluorophenoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL29817150; QNINIFSYLDGZBT-DRTKLYQKSA-N; (2S,4R)-1-[(2S)-2-[[2-[2-[2-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]-2-fluorophenoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOC3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3F)C(C)(C)C)C=C2)SC=N1	C49H55F4N7O9S2	AR	P10275	VHL	WO-2019023553-A1
TPD-ZTALXD	SCHEMBL17941157	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[2-[4-[5,5-dimethyl-3-[4-nitro-3-(trifluoromethyl)phenyl]-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL29817079; RFFHHKHQPKZGFY-RHMQSKSJSA-N; (2S,4R)-1-[(2S)-2-[[2-[2-[2-[2-[4-[5,5-dimethyl-3-[4-nitro-3-(trifluoromethyl)phenyl]-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOC3=CC=C(N4C(=S)N(C5=CC=C([N+](=O)[O-])C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C48H56F3N7O11S2	AR	P10275	VHL	WO-2019023553-A1
TPD-TWEWXL	SCHEMBL17951940	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL29817209; XUQBWSTYEJCJCV-CVFMEUHCSA-N; (2S,4R)-1-[(2S)-2-[[2-[2-[2-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOC3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C50H58F3N7O9S2	AR	P10275	VHL	WO-2019023553-A1
TPD-ELGR2F	SCHEMBL17952286	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[2-[4-[3-[6-cyano-5-(trifluoromethyl)pyridin-3-yl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL29817520; BAVWICUZOIEOQT-RHMQSKSJSA-N; (2S,4R)-1-[(2S)-2-[[2-[2-[2-[2-[4-[3-[6-cyano-5-(trifluoromethyl)pyridin-3-yl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOC3=CC=C(N4C(=S)N(C5=CN=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C48H55F3N8O9S2	AR	P10275	VHL	WO-2019023553-A1
TPD-40QP90	SCHEMBL17947446	(2S,4R)-1-[(2S)-2-[[2-[(2R,3R)-3-[2-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]ethoxy]ethoxy]butan-2-yl]oxyacetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; QLLWMQVJMASXEI-JWIOGSMYSA-N; (2S,4R)-1-[(2S)-2-[[2-[(2R,3R)-3-[2-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]ethoxy]ethoxy]butan-2-yl]oxyacetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CO[C@H](C)[C@@H](C)OCCOCCOC3=CC=C(N4C(=S)N(C5=CC(C(F)(F)F)=C(C#N)C=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C51H60F3N7O9S2	AR	P10275	VHL	WO-2019023553-A1
TPD-9VJOW7	WO2019023553A1_23	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCO[C@H](C)[C@@H](C)OCCOC3=CC=C(N4C(=S)N(C5=CC(C(F)(F)F)=C(C#N)C=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C51H60F3N7O9S2	AR	P10275	VHL	WO-2019023553-A1
TPD-TLX38R	SCHEMBL17947653	(2S,4R)-1-[(2S)-2-[[2-[4-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]butoxy]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; ULHCJGLPFCRVDE-UMWCMSNQSA-N; (2S,4R)-1-[(2S)-2-[[2-[4-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]butoxy]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCOCCCCOC3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C51H60F3N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-PYNE6F	SCHEMBL17951943	(2S,4R)-1-[(2S)-2-[[2-[4-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]-2-fluorophenoxy]butoxy]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL29817223; WETNYWQAJOWKFW-OZSPHOIVSA-N; (2S,4R)-1-[(2S)-2-[[2-[4-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]-2-fluorophenoxy]butoxy]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCOCCCCOC3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3F)C(C)(C)C)C=C2)SC=N1	C52H61F4N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-4440EH	WO2019023553A1_26	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCOCCCCOC3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3F)C(C)(C)C)C=C2)SC=N1	C51H59F4N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-O2FX1K	WO2019023553A1_27	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@H](O)CN3C(=O)[C@@H](NC(=O)COCCCOCCCCOC3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3F)C(C)(C)C)C=C2)SC=N1	C50H57F4N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-A82IM1	WO2019023553A1_28	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@H](O)CN3C(=O)[C@@H](NC(=O)COCCCOCCCCOC3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C50H58F3N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-OHN5WU	WO2019023553A1_29	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCOCCCCOC3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3)C(C)C)C=C2)SC=N1	C49H56F3N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-Q5TQ2L	WO2019023553A1_30	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCOCCCCOC3=CC=C(N4C(=S)N(C5=CN=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C49H57F3N8O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-6YUTCX	WO2019023553A1_31	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCOCCCCOC3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(Cl)=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C49H58ClN7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-8KKTS6	SCHEMBL17951945	(2S,4R)-1-[(2S)-2-[[2-[3-[4-[4-[3-(4-cyano-3-methoxyphenyl)-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]butoxy]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL29817181	COC1=CC(N2C(=O)C(C)(C)N(C3=CC=C(OCCCCOCCCOCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)NCC4=CC=C(C5=C(C)N=CS5)C=C4)C(C)(C)C)C=C3)C2=S)=CC=C1C#N	C50H61N7O9S2	AR	P10275	VHL	WO-2019023553-A1
TPD-RFIJBM	WO2019023553A1_33	.	CC(C)(C)[C@H](NC(=O)COCCCOCCCCOC1=CC=C(N2C(=S)N(C3=CC=C(C#N)C(C(F)(F)F)=C3)C(=O)C2(C)C)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=CN=CS2)C=C1	C49H56F3N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-D4SRVG	WO2019023553A1_34	.	CC(C)(C)[C@H](NC(=O)COCCCOCCCCOC1=CC=C(N2C(=S)N(C3=CC=C(C#N)C(C(F)(F)F)=C3)C(=O)C2(C)C)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=CN=CO2)C=C1	C49H56F3N7O9S	AR	P10275	VHL	WO-2019023553-A1
TPD-GMG1GY	WO2019023553A1_35	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCOCCCCOC3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)OC=N1	C50H58F3N7O9S	AR	P10275	VHL	WO-2019023553-A1
TPD-GDAM5H	WO2019023553A1_36	.	CC(C)[C@H](NC(=O)COCCCOCCCCOC1=CC=C(N2C(=S)N(C3=CC=C(C#N)C(Cl)=C3)C(=O)C2(C)C)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=CN=CS2)C=C1	C47H54ClN7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-YR8EZE	SCHEMBL17947092	(2S,4R)-1-[(2S)-2-[[2-[3-[4-[4-[3-(5-chloro-6-cyanopyridin-3-yl)-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]butoxy]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCOCCCCOC3=CC=C(N4C(=S)N(C5=CN=C(C#N)C(Cl)=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C48H57ClN8O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-4WQ6WK	WO2019023553A1_38	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCOCCCCOC3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(Cl)=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)OC=N1	C49H58ClN7O9S	AR	P10275	VHL	WO-2019023553-A1
TPD-MGF68W	SCHEMBL17951924	(2S,4R)-1-[(2S)-2-[[2-[3-[4-[4-[3-(3-chloro-4-cyanophenyl)-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]butoxy]propoxy]acetyl]amino]-3-methylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-oxazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCOCCCCOC3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(Cl)=C5)C(=O)C4(C)C)C=C3)C(C)C)C=C2)OC=N1	C48H56ClN7O9S	AR	P10275	VHL	WO-2019023553-A1
TPD-0DEW1I	WO2019023553A1_40	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCOCCCCOC3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=N3)C(C)(C)C)C=C2)SC=N1	C49H57F3N8O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-Q3O34H	SCHEMBL17947133	(2S,4R)-1-[(2S)-2-[[2-[3-[4-[4-[3-(3-chloro-4-cyanophenyl)-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]-2-fluorophenoxy]butoxy]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL29817511	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCOCCCCOC3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(Cl)=C5)C(=O)C4(C)C)C=C3F)C(C)(C)C)C=C2)SC=N1	C49H57ClFN7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-H0CK6E	SCHEMBL17947454	(2S,4R)-1-[(2S)-2-[[2-[3-[4-[4-[3-(4-cyano-3-methoxyphenyl)-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]-2-fluorophenoxy]butoxy]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL29817026	COC1=CC(N2C(=O)C(C)(C)N(C3=CC=C(OCCCCOCCCOCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)NCC4=CC=C(C5=C(C)N=CS5)C=C4)C(C)(C)C)C(F)=C3)C2=S)=CC=C1C#N	C50H60FN7O9S2	AR	P10275	VHL	WO-2019023553-A1
TPD-T0BW8A	SCHEMBL17947134	(2S,4R)-1-[(2S)-2-[[2-[3-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-4-oxo-2-sulfanylidene-8-oxa-1,3-diazaspiro[4.5]decan-1-yl]phenoxy]butoxy]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL29817124; XFUCIVXJGAJWFO-BZPYCXPJSA-N; (2S,4R)-1-[(2S)-2-[[2-[3-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-4-oxo-2-sulfanylidene-8-oxa-1,3-diazaspiro[4.5]decan-1-yl]phenoxy]butoxy]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCOCCCCOC3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C45CCOCC5)C=C3)C(C)(C)C)C=C2)SC=N1	C52H60F3N7O9S2	AR	P10275	VHL	WO-2019023553-A1
TPD-VHRJFR	WO2019023553A1_44	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCOCCCCOC3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(Cl)=C5)C(=O)C4(C)C)C=C3F)C(C)(C)C)C=C2)OC=N1	C49H57ClFN7O9S	AR	P10275	VHL	WO-2019023553-A1
TPD-EVT8K4	SCHEMBL17947136	(2S,4R)-1-[(2S)-2-[[2-[3-[4-[4-[3-(3-chloro-4-cyanophenyl)-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]-2-fluorophenoxy]butoxy]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(1,3-oxazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL29817058	CC(C)(C)[C@H](NC(=O)COCCCOCCCCOC1=CC=C(N2C(=S)N(C3=CC=C(C#N)C(Cl)=C3)C(=O)C2(C)C)C=C1F)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=CN=CO2)C=C1	C48H55ClFN7O9S	AR	P10275	VHL	WO-2019023553-A1
TPD-WD2CZT	WO2019023553A1_46	.	CC(C)(C)[C@H](NC(=O)COCCCOCCCCOC1=CC=C(N2C(=S)N(C3=CC=C(C#N)C(Cl)=C3)C(=O)C2(C)C)C=C1F)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=CN=CS2)C=C1	C48H55ClFN7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-2WI0HQ	WO2019023553A1_47	.	CC(C)(C)[C@H](NC(=O)COCCCOCCCCOC1=CC=C(N2C(=S)N(C3=CN=C(C#N)C(C(F)(F)F)=C3)C(=O)C2(C)C)C=C1F)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=CN=CO2)C=C1	C48H54F4N8O9S	AR	P10275	VHL	WO-2019023553-A1
TPD-FRKOS1	WO2019023553A1_48	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCOCCCCOC3=CC=C(N4C(=S)N(C5=CN=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3F)C(C)(C)C)C=C2)SC=N1	C49H56F4N8O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-67CE7S	SCHEMBL17946927	(2S,4R)-1-[(2S)-2-[[2-[3-[4-[4-[3-(4-cyano-3-methoxyphenyl)-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]-2-fluorophenoxy]butoxy]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(1,3-oxazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL29817178	COC1=CC(N2C(=O)C(C)(C)N(C3=CC=C(OCCCCOCCCOCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)NCC4=CC=C(C5=CN=CO5)C=C4)C(C)(C)C)C(F)=C3)C2=S)=CC=C1C#N	C49H58FN7O10S	AR	P10275	VHL	WO-2019023553-A1
TPD-EWSR5G	SCHEMBL17947658	(2S,4R)-1-[(2S)-2-[[2-[3-[4-[4-[3-(3-chloro-4-cyanophenyl)-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]-2-fluorophenoxy]butoxy]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(2-methylpyrazol-3-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL29817028	CN1N=CC=C1C1=CC=C(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCCOCCCCOC2=CC=C(N3C(=S)N(C4=CC=C(C#N)C(Cl)=C4)C(=O)C3(C)C)C=C2F)C(C)(C)C)C=C1	C49H58ClFN8O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-ODDTC9	WO2019023553A1_51	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@H](O)CN3C(=O)[C@@H](NC(=O)COCCCOCCCCOC3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C45CCN(C)CC5)C=C3)C(C)(C)C)C=C2)SC=N1	C53H63F3N8O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-QIFM3S	SCHEMBL17951946	(2S,4R)-1-[(2S)-2-[[2-[4-[3-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]propoxy]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL29817175; DPMXDDYZNCBJKB-AKCINUCUSA-N; (2S,4R)-1-[(2S)-2-[[2-[4-[3-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]propoxy]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCOCCCOC3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C50H58F3N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-D8ZS65	SCHEMBL17952291	(2S,4R)-1-[(2S)-2-[[2-[4-[3-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]-2-fluorophenoxy]propoxy]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL29816991; VAFKQLWTGDUDRR-IPQHXDNUSA-N; (2S,4R)-1-[(2S)-2-[[2-[4-[3-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]-2-fluorophenoxy]propoxy]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCOCCCOC3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3F)C(C)(C)C)C=C2)SC=N1	C50H57F4N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-CSO8OT	SCHEMBL17940938	(2S,4R)-1-[(2S)-2-[3-[2-[5-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]pyridin-2-yl]oxyethoxy]propanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL29817480; DMBIRPJQFZDQHN-JABZAXQMSA-N; (2S,4R)-1-[(2S)-2-[3-[2-[5-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]pyridin-2-yl]oxyethoxy]propanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCOCCOC3=NC=C(C4=CC=C(N5C(=S)N(C6=CC=C(C#N)C(C(F)(F)F)=C6)C(=O)C5(C)C)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C51H53F3N8O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-JGEM76	SCHEMBL17941004	(2S,4R)-1-[(2S)-2-[3-[2-[6-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]pyridin-3-yl]oxyethoxy]propanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL29817143; FOJUOTNAVHHUNT-ZKAWRXRFSA-N; (2S,4R)-1-[(2S)-2-[3-[2-[6-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]pyridin-3-yl]oxyethoxy]propanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCOCCOC3=CN=C(C4=CC=C(N5C(=S)N(C6=CC=C(C#N)C(C(F)(F)F)=C6)C(=O)C5(C)C)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C51H53F3N8O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-ADKAA5	WO2019023553A1_88	.	CC(C)(C)C(NC(=O)CCCCN1CCN(C2=CC=C(C3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(Cl)=C5)C(=O)C4(C)C)C=C3)C=C2)CC1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=CN=CO2)C=C1	C54H60ClN9O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-JRUH92	SCHEMBL17952511	(2S,4R)-1-[(2S)-2-[[2-[4-[6-[4-[3-(3-chloro-4-cyanophenyl)-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]pyridin-3-yl]oxybutoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(1,3-oxazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL29817419	CC(C)(C)[C@H](NC(=O)COCCCCOC1=CN=C(C2=CC=C(N3C(=S)N(C4=CC=C(C#N)C(Cl)=C4)C(=O)C3(C)C)C=C2)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=CN=CO2)C=C1	C50H53ClN8O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-FYUT3Y	WO2019023553A1_90	.	CC(C)(C)[C@H](NC(=O)COCCCCOC1=NC=C(C2=CC=C(N3C(=S)N(C4=CC=C(C#N)C(Cl)=C4)C(=O)C3(C)C)C=C2)C=C1)C(=O)N1C[C@@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=CN=CO2)C=C1	C50H53ClN8O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-QGNFP9	SCHEMBL17941154	(2S,4R)-1-[(2S)-2-[4-[4-[4-[4-[3-(3-chloro-4-cyanophenyl)-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]phenyl]piperidin-1-yl]butanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(1,3-oxazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC(C)(C)[C@H](NC(=O)CCCN1CCC(C2=CC=C(C3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(Cl)=C5)C(=O)C4(C)C)C=C3)C=C2)CC1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=CN=CO2)C=C1	C54H59ClN8O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-UV766Y	WO2019023553A1_92	.	CC(C)(C)[C@H](NC(=O)COCCN1CCC(C2=CC=C(C3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(Cl)=C5)C(=O)C4(C)C)C=C3)C=C2)CC1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=CN=CO2)C=C1	C54H59ClN8O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-W5EYKK	WO2019023553A1_93	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCOC3=CC=C(C4=CC=C(N5C(=S)N(C6=CC=C(C#N)C(C(F)(F)F)=C6)C(=O)C5(C)C)C=C4)C=C3)C(C)C)C=C2)SC=N1	C52H54F3N7O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-A1Z0JU	SCHEMBL17940846	(2S,4R)-1-[(2S)-2-[[2-[4-[4-[4-[3-(3-chloro-4-cyanophenyl)-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]phenoxy]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(1,3-oxazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC(C)(C)[C@H](NC(=O)COCCCCOC1=CC=C(C2=CC=C(N3C(=S)N(C4=CC=C(C#N)C(Cl)=C4)C(=O)C3(C)C)C=C2)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=CN=CO2)C=C1	C51H54ClN7O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-PBA2FL	WO2019023553A1_95	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCOC3=CC=C(C4=CC=C(N5C(=S)N(C6=CC(C(F)(F)F)=C(C#N)C=C6)C(=O)C5(C)C)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C54H58F3N7O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-4FM4DV	SCHEMBL17941151	(2S,4R)-1-[(2S)-2-[[2-[4-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]phenoxy]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(1,3-oxazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL29817321; PCLSQNYLDUYYJP-BZPYCXPJSA-N; (2S,4R)-1-[(2S)-2-[[2-[4-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]phenoxy]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(1,3-oxazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC(C)(C)[C@H](NC(=O)COCCCCOC1=CC=C(C2=CC=C(N3C(=S)N(C4=CC(C(F)(F)F)=C(C#N)C=C4)C(=O)C3(C)C)C=C2)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=CN=CO2)C=C1	C52H54F3N7O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-6R4A19	SCHEMBL17940944	(2S,4R)-1-[(2S)-2-[[2-[4-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]phenoxy]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-oxazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL29817271; ACBQRNTUSHJDME-PPZGWQTASA-N; (2S,4R)-1-[(2S)-2-[[2-[4-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]phenoxy]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-oxazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCOC3=CC=C(C4=CC=C(N5C(=S)N(C6=CC(C(F)(F)F)=C(C#N)C=C6)C(=O)C5(C)C)C=C4)C=C3)C(C)(C)C)C=C2)OC=N1	C53H56F3N7O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-71BR7T	WO2019023553A1_98	.	CC(C)(C)[C@H](NC(=O)COCCCCOC1=CC=C(C2=CC=C(N3C(=S)N(C4=CC(C(F)(F)F)=C(C#N)C=C4)C(=O)C3(C)C)C=C2)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=CN=CS2)C=C1	C52H54F3N7O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-1SNGJF	WO2019023553A1_99	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCOC3=CC=CC(C4=CC=C(N5C(=S)N(C6=CC(C(F)(F)F)=C(C#N)C=C6)C(=O)C5(C)C)C=C4)=C3)C(C)C)C=C2)SC=N1	C52H54F3N7O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-BLUBX2	SCHEMBL17941104	(2S,4R)-1-[(2S)-2-[[2-[4-[4-[4-[3-(3-chloro-4-cyanophenyl)-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]-3-fluorophenyl]phenoxy]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-oxazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL29817048	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCOC3=CC=C(C4=CC=C(N5C(=S)N(C6=CC(Cl)=C(C#N)C=C6)C(=O)C5(C)C)C(F)=C4)C=C3)C(C)(C)C)C=C2)OC=N1	C52H55ClFN7O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-C9A28Z	SCHEMBL17941187	(2S,4R)-1-[(2S)-2-[[2-[4-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]phenoxy]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-oxazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL29823693; NXUHNQFFCSSDQH-OTNIZCNFSA-N; (2S,4R)-1-[(2S)-2-[[2-[4-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]phenoxy]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-oxazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCOC3=CC=C(C4=CC=C(N5C(=S)N(C6=CC(C(F)(F)F)=C(C#N)C=C6)C(=O)C5(C)C)C=C4)C=C3)C(C)(C)C)C=C2)OC=N1	C54H58F3N7O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-E63Z0T	WO2019023553A1_102	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCOC3=CC=C(C4=NC=C(N5C(=S)N(C6=CC(C(F)(F)F)=C(C#N)C=C6)C(=O)C5(C)C)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C52H55F3N8O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-P5L1WN	WO2019023553A1_103	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCNC3=CC=C(C4=CC=C(N5C(=S)N(C6=CC=C(C#N)C(C(F)(F)F)=C6)C(=O)C5(C)C)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C53H57F3N8O6S2	AR	P10275	VHL	WO-2019023553-A1
TPD-6QSLM0	SCHEMBL17941096	(2S,4R)-1-[(2S)-2-[[2-[4-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]phenoxy]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(3-methylimidazol-4-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL29817353; WVHXYUAMFMDTSF-PPZGWQTASA-N; (2S,4R)-1-[(2S)-2-[[2-[4-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]phenoxy]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(3-methylimidazol-4-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CN1C=NC=C1C1=CC=C(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCCCOC2=CC=C(C3=CC=C(N4C(=S)N(C5=CC(C(F)(F)F)=C(C#N)C=C5)C(=O)C4(C)C)C=C3)C=C2)C(C)(C)C)C=C1	C53H57F3N8O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-VPYNML	WO2019023553A1_105	.	CC(C)[C@H](NC(=O)COCCCCOC1=CC=C(C2=CC=C(N3C(=S)N(C4=CC(C(F)(F)F)=C(C#N)C=C4)C(=O)C3(C)C)C=C2)CC1)C(=O)N1CC(O)C[C@H]1C(=O)NCC1=CC=C(C2=C(Cl)N=CO2)C=C1	C51H53ClF3N7O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-T7YC4O	SCHEMBL17941081	(2S,4R)-1-[(2S)-2-[[2-[4-[4-[4-[3-(3-chloro-4-cyanophenyl)-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]-3-fluorophenyl]phenoxy]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(1,3-oxazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL29817152	CC(C)(C)[C@H](NC(=O)COCCCCOC1=CC=C(C2=CC=C(N3C(=S)N(C4=CC(Cl)=C(C#N)C=C4)C(=O)C3(C)C)C(F)=C2)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=CN=CO2)C=C1	C51H53ClFN7O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-4UWFTT	WO2019023553A1_107	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCOC3=CC=C(C4=CC=C(N5C(=S)N(C6=CC(Cl)=C(C#N)C=C6)C(=O)C5(C)C)C(F)=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C52H55ClFN7O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-L0C43V	WO2019023553A1_108	.	CC(C)(C)[C@H](NC(=O)COCCCCOC1=CC=C(C2=CC=C(N3C(=S)N(C4=CC(Cl)=C(C#N)C=C4)C(=O)C3(C)C)C(F)=C2)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=CN=CS2)C=C1	C51H53ClFN7O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-U0WDPH	SCHEMBL17940866	(2S,4R)-1-[(2S)-2-[[2-[4-[4-[4-[3-(3-chloro-4-cyanophenyl)-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]-2-fluorophenyl]phenoxy]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(1,3-oxazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL29817547	CC(C)(C)[C@H](NC(=O)COCCCCOC1=CC=C(C2=CC=C(N3C(=S)N(C4=CC=C(C#N)C(Cl)=C4)C(=O)C3(C)C)C=C2F)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=CN=CO2)C=C1	C51H53ClFN7O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-E6ENE6	WO2019023553A1_110	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCOC3=CC=C(C4=CC=C(N5C(=S)N(C6=CC=C(C#N)C(Cl)=C6)C(=O)C5(C)C)C=C4)C=C3)C(C)(C)C)C=C2)OC=N1	C52H56ClN7O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-CA4FY1	SCHEMBL17941021	(2S,4R)-1-[(2S)-2-[[2-[4-[4-[4-[3-(3-chloro-4-cyanophenyl)-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]phenoxy]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC(C)(C)[C@H](NC(=O)COCCCCOC1=CC=C(C2=CC=C(N3C(=S)N(C4=CC=C(C#N)C(Cl)=C4)C(=O)C3(C)C)C=C2)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=CN=CS2)C=C1	C51H54ClN7O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-EB0BZ0	SCHEMBL17940992	(2S,4R)-1-[(2S)-2-[[2-[4-[4-[4-[3-(3-chloro-4-cyanophenyl)-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]phenoxy]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCOC3=CC=C(C4=CC=C(N5C(=S)N(C6=CC=C(C#N)C(Cl)=C6)C(=O)C5(C)C)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C52H56ClN7O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-PIESV6	SCHEMBL17941132	(2S,4R)-1-[(2S)-2-[[2-[4-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]-3-fluorophenyl]phenoxy]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(1,3-oxazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL29817341; DTTRTRIKQNGZEW-FMATUXQASA-N; (2S,4R)-1-[(2S)-2-[[2-[4-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]-3-fluorophenyl]phenoxy]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(1,3-oxazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC(C)(C)[C@H](NC(=O)COCCCCOC1=CC=C(C2=CC=C(N3C(=S)N(C4=CC=C(C#N)C(C(F)(F)F)=C4)C(=O)C3(C)C)C(F)=C2)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=CN=CO2)C=C1	C52H53F4N7O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-X36479	SCHEMBL17941063	(2S,4R)-1-[(2S)-2-[[2-[3-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]phenoxy]phenoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL29817139; ACUBAXQVAHJSNU-LGDMESRFSA-N; (2S,4R)-1-[(2S)-2-[[2-[3-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]phenoxy]phenoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COC3=CC=CC(OC4=CC=C(C5=CC=C(N6C(=S)N(C7=CC=C(C#N)C(C(F)(F)F)=C7)C(=O)C6(C)C)C=C5)C=C4)=C3)C(C)(C)C)C=C2)SC=N1	C55H52F3N7O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-XEP9JN	WO2019023553A1_115	.	COC1=CC(N2C(=O)C(C)(C)N(C3=CC=C(C4=CC=C(OCCCCOCC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)NCC5=CC=C(C6=C(C)N=CO6)C=C5)C(C)(C)C)C=C4)C=C3)C2=S)=CC=C1C#N	C53H59N7O9S	AR	P10275	VHL	WO-2019023553-A1
TPD-3QBJAM	WO2019023553A1_116	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCOC3=CC=C(C4=CC=C(N5C(=S)N(C6=CC=C(C#N)C(C(F)(F)F)=C6)C(=O)C5(C)C)C(F)=C4)C=C3)C(C)(C)C)C=C2)OC=N1	C53H55F4N7O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-S8NN7F	WO2019023553A1_117	.	CC(C)(C)[C@H](NC(=O)COCCCCOC1=CC=C(C2=CC=C(N3C(=S)N(C4=CC(C(F)(F)F)=C(C#N)C=C4)C(=O)C3(C)C)C(F)=C2)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=CN=CS2)C=C1	C52H53F4N7O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-S5IPNM	WO2019023553A1_118	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCOC3=CC=C(C4=CC=C(N5C(=S)N(C6=CC=C(C#N)C(C(F)(F)F)=C6)C(=O)C5(C)C)C(F)=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C53H55F4N7O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-ME4V7F	SCHEMBL17940943	(2S,4R)-1-[(2S)-2-[[2-[4-[4-[4-[7-[4-cyano-3-(trifluoromethyl)phenyl]-8-oxo-6-sulfanylidene-5,7-diazaspiro[3.4]octan-5-yl]phenyl]phenoxy]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-oxazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL29817105; WCLMZGQHJZYBFT-IIWOMYBWSA-N; (2S,4R)-1-[(2S)-2-[[2-[4-[4-[4-[7-[4-cyano-3-(trifluoromethyl)phenyl]-8-oxo-6-sulfanylidene-5,7-diazaspiro[3.4]octan-5-yl]phenyl]phenoxy]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-oxazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCOC3=CC=C(C4=CC=C(N5C(=S)N(C6=CC=C(C#N)C(C(F)(F)F)=C6)C(=O)C56CCC6)C=C4)C=C3)C(C)(C)C)C=C2)OC=N1	C54H56F3N7O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-55H4OP	WO2019023553A1_120	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCOC3=CC=C(C4=CC=C(N5C(=S)N(C6=CC=C(C#N)C(C(F)(F)F)=C6)C(=O)C56CCC6)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C54H56F3N7O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-CT45CL	WO2019023553A1_121	.	CC(C)(C)[C@H](NC(=O)COCCCCOC1=CC(F)=C(C2=CC=C(N3C(=S)N(C4=CC=C(C#N)C(Cl)=C4)C(=O)C3(C)C)C=C2)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=CN=CO2)C=C1	C51H53ClFN7O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-NRTT0N	SCHEMBL17941162	(2S,4R)-1-[(2S)-2-[[2-[4-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]phenoxy]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(1H-pyrazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL29816994; REDLKRDFGUBXSG-SZHUYKCISA-N; (2S,4R)-1-[(2S)-2-[[2-[4-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]phenoxy]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(1H-pyrazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC(C)(C)[C@H](NC(=O)COCCCCOC1=CC=C(C2=CC=C(N3C(=S)N(C4=CC=C(C#N)C(C(F)(F)F)=C4)C(=O)C3(C)C)C=C2)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=CC=NN2)C=C1	C52H55F3N8O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-H9EA0U	SCHEMBL17940973	(2S,4R)-1-[(2S)-2-[[2-[4-[4-[4-[3-(3-chloro-4-cyano-2-fluorophenyl)-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]phenoxy]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(1,3-oxazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC(C)(C)[C@H](NC(=O)COCCCCOC1=CC=C(C2=CC=C(N3C(=S)N(C4=CC=C(C#N)C(Cl)=C4F)C(=O)C3(C)C)C=C2)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=CN=CO2)C=C1	C51H53ClFN7O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-9H5EF0	WO2019023553A1_124	.	CC(C)(C)[C@H](NC(=O)COCCCCOC1=CC=C(C2=CC=C(N3C(=S)N(C4=CC(Cl)=C(C#N)C=C4)C(=O)C34CCC4)C=C2)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=CN=CO2)C=C1	C52H54ClN7O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-FE2QCH	SCHEMBL17940945	(2S,4R)-1-[(2S)-2-[[2-[4-[4-[4-[3-(4-cyano-3-methylphenyl)-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]phenoxy]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(1,3-oxazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL29817333	CC1=C(C#N)C=CC(N2C(=O)C(C)(C)N(C3=CC=C(C4=CC=C(OCCCCOCC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)NCC5=CC=C(C6=CN=CO6)C=C5)C(C)(C)C)C=C4)C=C3)C2=S)=C1	C52H57N7O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-Z774RM	WO2019023553A1_126	.	CC(C)(C)[C@H](NC(=O)COCCCCOC1=CC=C(C2=CC=C(N3C(=S)N(C4=CC(F)=C(C#N)C=C4)C(=O)C3(C)C)C=C2)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=CN=CO2)C=C1	C51H54FN7O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-47FHHB	SCHEMBL17940864	(2S,4R)-1-[(2S)-2-[[2-[4-[3-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]phenoxy]phenoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL29817126; PUVJVTDVTLBWPB-LGDMESRFSA-N; (2S,4R)-1-[(2S)-2-[[2-[4-[3-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]phenoxy]phenoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COC3=CC=C(OC4=CC=CC(C5=CC=C(N6C(=S)N(C7=CC=C(C#N)C(C(F)(F)F)=C7)C(=O)C6(C)C)C=C5)=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C55H52F3N7O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-8XGN7Z	WO2019023553A1_128	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCOCC3=CC=C(C4=CC=C(N5C(=S)N(C6=CC(C(F)(F)F)=C(C#N)C=C6)C(=O)C5(C)C)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C53H56F3N7O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-X3E7IA	WO2019023553A1_129	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCC(O)COC3=CC=C(C4=CC=C(N5C(=S)N(C6=CC(C(F)(F)F)=C(C#N)C=C6)C(=O)C5(C)C)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C53H56F3N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-KE9LAE	WO2019023553A1_130	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COC[C@H](O)CCOC3=CC=C(C4=CC=C(N5C(=S)N(C6=CC(C(F)(F)F)=C(C#N)C=C6)C(=O)C5(C)C)CC4)C=C3)C(C)(C)C)C=C2)SC=N1	C53H58F3N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-T4APVA	WO2019023553A1_131	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCC(O)CCOC3=CC=C(C4=CC=C(N5C(=S)N(C6=CC(C(F)(F)F)=C(C#N)C=C6)C(=O)C5(C)C)C=C4)C=C3)C(C)C)C=C2)SC=N1	C52H54F3N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-YA8NHG	SCHEMBL17940875	(2S,4R)-1-[(2S)-2-[[2-[4-[4-[4-[3-(3-chloro-4-cyanophenyl)-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]phenoxy]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(1,3-oxazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](NC(=O)COCCCCOC1=CC=C(C2=CC=C(N3C(=S)N(C4=CC(Cl)=C(C#N)C=C4)C(=O)C3(C)C)C=C2)C=C1)C(C)(C)C)C1=CC=C(C2=CN=CO2)C=C1	C52H56ClN7O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-ZH4I3L	WO2019023553A1_133	.	CC(C)(C)[C@H](NC(=O)COCCCCOC1=CC=C(C2=CC=C(N3C(=S)N(C4=C(F)C=C(C#N)C(Cl)=C4)C(=O)C3(C)C)C=C2)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=CN=CO2)C=C1	C51H53ClFN7O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-7H7HCO	WO2019023553A1_134	.	CC1=C(OCCCCOCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)C=CC(C2=CC=C(N3C(=S)N(C4=CC(C(F)(F)F)=C(C#N)C=C4)C(=O)C3(C)C)C=C2)=C1	C54H58F3N7O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-9CO2CY	SCHEMBL17952349	(2S,4R)-1-[(2S)-2-[[2-[4-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]anilino]-4-oxobutoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-oxazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL29817172; HQPIAVYEBUJITD-GCXMMMFBSA-N; (2S,4R)-1-[(2S)-2-[[2-[4-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]anilino]-4-oxobutoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-oxazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCC(=O)NC3=CC=C(C4=CC=C(N5C(=S)N(C6=CC=C(C#N)C(C(F)(F)F)=C6)C(=O)C5(C)C)C=C4)C=C3)C(C)(C)C)C=C2)OC=N1	C53H55F3N8O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-JQQ791	SCHEMBL17941166	(2S,4R)-1-[(2S)-2-[[2-[4-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]-3-methylphenoxy]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL29817451; ATJHUKXEFODAGT-UJGSORPVSA-N; (2S,4R)-1-[(2S)-2-[[2-[4-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]-3-methylphenoxy]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(N3C(=S)N(C4=CC(C(F)(F)F)=C(C#N)C=C4)C(=O)C3(C)C)C=C2)C=CC(OCCCCOCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)=C1	C54H58F3N7O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-S8BWQC	SCHEMBL17940935	(2S,4R)-1-[(2S)-2-[[2-[4-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]-3-fluorophenyl]phenoxy]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; XZJXKRFVSBTTRJ-HSHIJRGOSA-N; (2S,4R)-1-[(2S)-2-[[2-[4-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]-3-fluorophenyl]phenoxy]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCOC3=CC=C(C4=CC=C(N5C(=S)N(C6=CC=C(C#N)C(C(F)(F)F)=C6)C(=O)C5(C)C)C(F)=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C54H57F4N7O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-SGS5OG	SCHEMBL17941083	(2S,4R)-1-[(2S)-2-[[2-[4-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]-3-fluorophenyl]phenoxy]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-oxazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL29817096; UTJXYWIOKSQNLN-HSHIJRGOSA-N; (2S,4R)-1-[(2S)-2-[[2-[4-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]-3-fluorophenyl]phenoxy]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-oxazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCOC3=CC=C(C4=CC=C(N5C(=S)N(C6=CC=C(C#N)C(C(F)(F)F)=C6)C(=O)C5(C)C)C(F)=C4)C=C3)C(C)(C)C)C=C2)OC=N1	C54H57F4N7O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-6YBO46	SCHEMBL17941003	(2S,4R)-1-[(2S)-2-[[2-[4-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]-2-methoxyphenoxy]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL29817552; QLUHOFDCRUDARS-MYICIHSCSA-N; (2S,4R)-1-[(2S)-2-[[2-[4-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]-2-methoxyphenoxy]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	COC1=C(OCCCCOCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)C=CC(C2=CC=C(N3C(=S)N(C4=CC(C(F)(F)F)=C(C#N)C=C4)C(=O)C3(C)C)C=C2)=C1	C54H58F3N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-CTFZDC	WO2019023553A1_140	.	COC1=C(C2=CC=C(N3C(=S)N(C4=CC(C(F)(F)F)=C(C#N)C=C4)C(=O)C3(C)C)C=C2)C=CC(OCCCCOCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(C3=C(C)N=CS3)C=C2)C(C)C)=C1	C53H56F3N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-UV8QUR	WO2019023553A1_141	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@H](O)CN3C(=O)[C@@H](NC(=O)COCCC[C@@H](C)OC3=CC=C(C4=CC=C(N5C(=S)N(C6=CC(C(F)(F)F)C(C#N)C=C6)C(=O)C5(C)C)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C54H64F3N7O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-5FL7MZ	WO2019023553A1_142	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@H](O)CN3C(=O)[C@@H](NC(=O)COCCC[C@H](C)OC3=CC=C(C4=CC=C(N5C(=S)N(C6=CC(C(F)(F)F)C(C#N)C=C6)C(=O)C5(C)C)CC4)CC3)C(C)C)C=C2)SC=N1	C53H62F3N7O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-OYJ18D	SCHEMBL17940849	(2S,4R)-1-[(2S)-2-[[2-[4-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]anilino]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-oxazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL29817293; RIGMMHCAFPOVKN-MBFMYWTBSA-N; (2S,4R)-1-[(2S)-2-[[2-[4-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]anilino]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-oxazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCNC3=CC=C(C4=CC=C(N5C(=S)N(C6=CC=C(C#N)C(C(F)(F)F)=C6)C(=O)C5(C)C)C=C4)C=C3)C(C)(C)C)C=C2)OC=N1	C54H59F3N8O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-M9MYAZ	SCHEMBL17940947	(2S,4R)-1-[(2S)-2-[[2-[5-[5-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]pyridin-2-yl]pentoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL29817162; FKCHRMHGFQACAN-LASKKICZSA-N; (2S,4R)-1-[(2S)-2-[[2-[5-[5-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]pyridin-2-yl]pentoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCCC3=CC=C(C4=CC=C(N5C(=S)N(C6=CC(C(F)(F)F)=C(C#N)C=C6)C(=O)C5(C)C)C=C4)C=N3)C(C)(C)C)C=C2)SC=N1	C53H57F3N8O6S2	AR	P10275	VHL	WO-2019023553-A1
TPD-8K9MDQ	WO2019023553A1_145	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCNC3=CC=C(C4=CC=C(N5C(=S)N(C6=CC=C(C#N)C(C(F)(F)F)=C6)C(=O)C5(C)C)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C54H59F3N8O6S2	AR	P10275	VHL	WO-2019023553-A1
TPD-V45X57	SCHEMBL17941119	(2S,4R)-1-[(2S)-2-[[2-[4-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]-3-fluorophenyl]phenoxy]butanoylamino]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL29817102; BBTBTYVIMULPJJ-BQGOKDIQSA-N; (2S,4R)-1-[(2S)-2-[[2-[4-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]-3-fluorophenyl]phenoxy]butanoylamino]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CNC(=O)CCCOC3=CC=C(C4=CC(F)=C(N5C(=S)N(C6=CC(C(F)(F)F)=C(C#N)C=C6)C(=O)C5(C)C)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C53H54F4N8O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-RSCY5A	WO2019023553A1_147	.	CC1=C(C2C=CC(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CO[C@H](C)CCCOC3=CC=C(C4=CC=C(N5C(=S)N(C6=CC(C(F)(F)F)=C(C#N)C=C6)C(=O)C5(C)C)C=C4)C=C3)C(C)(C)C)=CC2)SC=N1	C54H60F3N7O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-0TRT9Y	WO2019023553A1_148	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CO[C@@H](C)CCCOC3=CC=C(C4=CC=C(N5C(=S)N(C6=CC(C(F)(F)F)=C(C#N)C=C6)C(=O)C5(C)C)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C54H58F3N7O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-AB5GRD	WO2019023553A1_149	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCOC3=CC(F)=C(C4=CC=C(N5C(=S)N(C6=CC(C(F)(F)F)=C(C#N)C=C6)C(=O)C5(C)C)C=C4)C=C3)C(C)C)C=C2)SC=N1	C52H53F4N7O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-V7XNF3	SCHEMBL17941169	(2S,4R)-1-[(2S)-2-[[2-[2-[4-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenyl]anilino]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL17947014	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCNC3=CC=C(C4=CC=C(C(=O)NC5C(C)(C)C(OC6=CC=C(C#N)C(Cl)=C6)C5(C)C)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C54H62ClN7O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-409HNN	SCHEMBL17952534	(2S,4R)-N-[[2-[3-[2-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]ethoxy]ethoxy]propoxy]-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-4-hydroxy-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]pyrrolidine-2-carboxamide; QVCRGNUISUFFTL-UCUQKJTESA-N; (2S,4R)-N-[[2-[3-[2-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]ethoxy]ethoxy]propoxy]-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-4-hydroxy-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C(OCCCOCCOCCOC3=CC=C(N4C(=S)N(C5=CC(C(F)(F)F)=C(C#N)C=C5)C(=O)C4(C)C)C=C3)=C2)SC=N1	C55H58F3N7O9S2	AR	P10275	VHL	WO-2019023553-A1
TPD-Z7D68E	WO2019023553A1_206	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C(OCCOCCOC3=CC=C(N4C(=O)N(C5=CC(C(F)(F)F)=C(C#N)C=C5)C(=O)C4(C)C)C=C3)=C2)SC=N1	C52H52F3N7O9S	AR	P10275	VHL	WO-2019023553-A1
TPD-JNWWWD	SCHEMBL17951994	(2S,4R)-N-[[2-[4-[4-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]butoxy]butoxy]butoxy]-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-4-hydroxy-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]pyrrolidine-2-carboxamide; BSMGBNTYXXDKDD-YLJCJUPRSA-N; (2S,4R)-N-[[2-[4-[4-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]butoxy]butoxy]butoxy]-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-4-hydroxy-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C(OCCCCOCCCCOCCCCOC3=CC=C(N4C(=S)N(C5=CC(C(F)(F)F)=C(C#N)C=C5)C(=O)C4(C)C)C=C3)=C2)SC=N1	C60H68F3N7O9S2	AR	P10275	VHL	WO-2019023553-A1
TPD-MN3Y5G	SCHEMBL19600398	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[2-[2-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; KXHVWMDPUOCPRT-PPZGWQTASA-N; (2S,4R)-1-[(2S)-2-[[2-[2-[2-[2-[2-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOCCOCCOC3=CC=C(N4C(=S)N(C5=CC(C(F)(F)F)=C(C#N)C=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C53H64F3N7O11S2	AR	P10275	VHL	WO-2019023553-A1
TPD-MCTKAI	WO2019023553A1_209	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOC3=CC=C(N4C(=S)N(C5=CC(C(F)(F)F)=C(C#N)C=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C47H52F3N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-HCS21K	SCHEMBL17952370	(2S,4R)-N-[[2-[2-[2-[2-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]ethoxy]ethoxy]ethoxy]ethoxy]-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-4-hydroxy-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]pyrrolidine-2-carboxamide; GQHCFJKLAWETGU-DLDIJDMTSA-N; (2S,4R)-N-[[2-[2-[2-[2-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]ethoxy]ethoxy]ethoxy]ethoxy]-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-4-hydroxy-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C(OCCOCCOCCOCCOC3=CC=C(N4C(=S)N(C5=CC(C(F)(F)F)=C(C#N)C=C5)C(=O)C4(C)C)C=C3)=C2)SC=N1	C56H60F3N7O10S2	AR	P10275	VHL	WO-2019023553-A1
TPD-8TLEAJ	SCHEMBL17951982	(2S,4R)-N-[[2-[2-[2-[2-[2-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-4-hydroxy-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]pyrrolidine-2-carboxamide; YAOPIRGMKDEPQJ-YHVUXZCSSA-N; (2S,4R)-N-[[2-[2-[2-[2-[2-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-4-hydroxy-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C(OCCOCCOCCOCCOCCOC3=CC=C(N4C(=S)N(C5=CC(C(F)(F)F)=C(C#N)C=C5)C(=O)C4(C)C)C=C3)=C2)SC=N1	C58H64F3N7O11S2	AR	P10275	VHL	WO-2019023553-A1
TPD-NOEILQ	SCHEMBL21744365	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[2-[2-[2-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOCCOCCOCCOC3=CC=C(N4C(=S)N(C5=CC(C(F)(F)F)=C(C#N)C=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C55H68F3N7O12S2	AR	P10275	VHL	WO-2019023553-A1
TPD-8TI7CK	SCHEMBL17947570	(2S,4R)-N-[[2-[2-[2-[2-[2-[2-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-4-hydroxy-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]pyrrolidine-2-carboxamide; CKFWNQCSSJJYTM-YLJCJUPRSA-N; (2S,4R)-N-[[2-[2-[2-[2-[2-[2-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-4-hydroxy-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C(OCCOCCOCCOCCOCCOCCOC3=CC=C(N4C(=S)N(C5=CC(C(F)(F)F)=C(C#N)C=C5)C(=O)C4(C)C)C=C3)=C2)SC=N1	C60H68F3N7O12S2	AR	P10275	VHL	WO-2019023553-A1
TPD-ZYD4AT	SCHEMBL17947520	(2S,4R)-N-[[2-[2-[2-[4-[2-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]ethoxy]ethoxy]butoxy]ethoxy]ethoxy]-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-4-hydroxy-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]pyrrolidine-2-carboxamide; MVLQPRVOGWSUGX-YLJCJUPRSA-N; (2S,4R)-N-[[2-[2-[2-[4-[2-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]ethoxy]ethoxy]butoxy]ethoxy]ethoxy]-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-4-hydroxy-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C(OCCOCCOCCCCOCCOCCOC3=CC=C(N4C(=S)N(C5=CC(C(F)(F)F)=C(C#N)C=C5)C(=O)C4(C)C)C=C3)=C2)SC=N1	C60H68F3N7O11S2	AR	P10275	VHL	WO-2019023553-A1
TPD-H30979	WO2019023553A1_216	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCCCCCCCCOCCOC3=CC=C(N4C(=S)N(C5=CC(C(F)(F)F)=C(C#N)C=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C56H70F3N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-MD79PH	WO2019023553A1_218	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C(OCCOCCOCCCCCOCCOCC#CC3=CC=C(N4C(=S)N(C5=CC(C(F)(F)F)=C(C#N)C=C5)C(=O)C4(C)C)C=C3)=C2)SC=N1	C62H68F3N7O10S2	AR	P10275	VHL	WO-2019023553-A1
TPD-JRM0UV	WO2019023553A1_219	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C(OCCOCCOCCOCCOCCOCCOCCOC3=CC=C(N4C(=S)N(C5=CC(C(F)(F)F)=C(C#N)C=C5)C(=O)C4(C)C)C=C3)=C2)SC=N1	C63H74F3N7O13S2	AR	P10275	VHL	WO-2019023553-A1
TPD-WLX8SA	WO2019023553A1_220	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C(OCCOCCOCCCCCCOCCCCCOCCOCCOC3=CC=C(N4C(=S)N(C5=CC(C(F)(F)F)=C(C#N)C=C5)C(=O)C4(C)C)C=C3)=C2)SC=N1	C67H82F3N7O12S2	AR	P10275	VHL	WO-2019023553-A1
TPD-DBMTQI	WO2019023553A1_221	.	CC1=C(C2=CC=C(NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C(OCCCOCCCOCCOC3=CC=C(N4C(=S)N(C5=CC(C(F)(F)F)=C(C#N)C=C5)C(=O)C4(C)C)C=C3)=C2)SC=N1	C55H58F3N7O9S2	AR	P10275	VHL	WO-2019023553-A1
TPD-NSG9XY	WO2019023553A1_223	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCCCOCCCOCCOCCOC3=CC=C(N4C(=S)N(C5=CC(C(F)(F)F)=C(C#N)C=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C58H74F3N7O12S2	AR	P10275	VHL	WO-2019023553-A1
TPD-4B4HYF	WO2019023553A1_224	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCCCCCCCCCCCOCCOCCOC3=CC=C(N4C(=S)N(C5=CC(C(F)(F)F)=C(C#N)C=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C61H80F3N7O10S2	AR	P10275	VHL	WO-2019023553-A1
TPD-DF4UEU	SCHEMBL21743534	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[5-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]pentoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCCCCOC3=CC=C(N4C(=S)N(C5=CC(C(F)(F)F)=C(C#N)C=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C52H62F3N7O9S2	AR	P10275	VHL	WO-2019023553-A1
TPD-4TQ7EC	WO2019023553A1_226	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCOCCCCCOCCCCOC3=CC=C(N4C(=S)N(C5=CC(C(F)(F)F)=C(C#N)C=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C57H72F3N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-5QEGPO	WO2019023553A1_227	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(NC(=O)CCCCCOCCCCOCCCC#CC3=CC=C(N4C(=S)N(C5=CC(C(F)(F)F)=C(C#N)C=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C56H66F3N7O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-CBVFOY	WO2019023553A1_228	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCOCCOCCCCCCOC3=CC=C(N4C(=S)N(C5=CC(C(F)(F)F)=C(C#N)C=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C52H62F3N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-XF7LHU	SCHEMBL19598540	(2S,4S)-N-[[2-[2-[2-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]ethoxy]ethoxy]ethoxy]-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-4-hydroxy-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]pyrrolidine-2-carboxamide; OZGCBEBUDPZPIW-DTDRBBSGSA-N; (2S,4S)-N-[[2-[2-[2-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]ethoxy]ethoxy]ethoxy]-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-4-hydroxy-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C(OCCOCCOCCOC3=CC=C(N4C(=S)N(C5=CC(C(F)(F)F)=C(C#N)C=C5)C(=O)C4(C)C)C=C3)=C2)SC=N1	C54H56F3N7O9S2	AR	P10275	VHL	WO-2019023553-A1
TPD-H8S6JP	WO2019023553A1_230	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOC3=CC=C(N4C(=O)N(C5=CC(C(F)(F)F)=C(C#N)C=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C49H56F3N7O10S	AR	P10275	VHL	WO-2019023553-A1
TPD-2XUEI2	WO2019023553A1_231	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCNC(=O)CCCC3=CC=C(N4C(=O)N(C5=CC(C(F)(F)F)=C(C#N)C=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C48H53F3N8O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-T48IJJ	WO2019023553A1_232	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCC(=O)NCCCC3=CC=C(N4C(=S)N(C5=CC(C(F)(F)F)=C(C#N)C=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C50H57F3N8O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-RT0HGF	WO2019023553A1_233	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCOCCOC3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C46H50F3N7O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-C9VVV9	SCHEMBL24486187	(2S,4R)-N-[[2-[2-[2-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-2,4-dioxoimidazolidin-1-yl]phenoxy]ethoxy]ethoxy]ethoxy]-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]-4-[(2-methylpropan-2-yl)oxy]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](OC(C)(C)C)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C(OCCOCCOCCOC3=CC=C(N4C(=O)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3)=C2)SC=N1	C58H64F3N7O10S	AR	P10275	VHL	WO-2019023553-A1
TPD-KTMQB6	SCHEMBL24486092	(2S,4R)-N-[[2-[2-[2-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-2,4-dioxoimidazolidin-1-yl]phenoxy]ethoxy]ethoxy]ethoxy]-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-4-hydroxy-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C(OCCOCCOCCOC3=CC=C(N4C(=O)N(C5=CC(C(F)(F)F)=C(C#N)C=C5)C(=O)C4(C)C)C=C3)=C2)SC=N1	C54H56F3N7O10S	AR	P10275	VHL	WO-2019023553-A1
TPD-XV0FY6	SCHEMBL17951986	(2S,4R)-1-[(2S)-2-[[2-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; QOVJLLMCYXLZJQ-UZQUTMQESA-N; (2S,4R)-1-[(2S)-2-[[2-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOC3=CC=C(N4C(=S)N(C5=CC(C(F)(F)F)=C(C#N)C=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C45H48F3N7O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-EPYJAM	WO2019023553A1_237	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCOC3=CC=C(N4C(=S)N(C5=CC(C(F)(F)F)=C(C#N)C=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C45H48F3N7O6S2	AR	P10275	VHL	WO-2019023553-A1
TPD-OGRJ66	WO2019023553A1_238	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCOCCCOC3=CC=C(N4C(=S)N(C5=CC(C(F)(F)F)=C(C#N)C=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C49H56F3N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-IGT9BG	WO2019023553A1_239	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)OCCOCCCCOCCOC3=CC=C(N4C(=S)N(C5=CC(C(F)(F)F)=C(C#N)C=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C50H58F3N7O9S2	AR	P10275	VHL	WO-2019023553-A1
TPD-K78P88	SCHEMBL19598544	(2S,4R)-1-[(2S)-2-[[2-[2-[3-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]ethoxy]propoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; YZKJXDAKISSKFY-AKCINUCUSA-N; (2S,4R)-1-[(2S)-2-[[2-[2-[3-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]ethoxy]propoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCCOCCOC3=CC=C(N4C(=S)N(C5=CC(C(F)(F)F)=C(C#N)C=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C50H58F3N7O9S2	AR	P10275	VHL	WO-2019023553-A1
TPD-ZQS4R6	SCHEMBL17951987	(2S,4R)-N-[[2-[3-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]ethoxy]propoxy]-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-4-hydroxy-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]pyrrolidine-2-carboxamide; NDFXNUHKJQKRRB-RZBWGVJVSA-N; (2S,4R)-N-[[2-[3-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]ethoxy]propoxy]-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-4-hydroxy-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C(OCCCOCCOC3=CC=C(N4C(=S)N(C5=CC(C(F)(F)F)=C(C#N)C=C5)C(=O)C4(C)C)C=C3)=C2)SC=N1	C53H54F3N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-2CR044	WO2019023553A1_242	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@H](O)CN3C(=O)C(NC(=O)COCCCOCCCCCOC3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C51H60F3N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-7PXBE5	WO2019023553A1_243	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCCOC3=CC=C(N4C(=S)N(C5=CC(C(F)(F)F)=C(C#N)C=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C48H54F3N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-XCIK5J	WO2019023553A1_244	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCOCCCOC3=CC=C(N4C(=S)N(C5=CC(C(F)(F)F)=C(C#N)C=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C47H52F3N7O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-B14L3D	SCHEMBL21743537	(2S,4R)-1-[(2S)-2-[4-[2-[2-[[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]-2-fluorobenzoyl]amino]ethoxy]ethoxy]butanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCOCCOCCNC(=O)C3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3F)C(C)(C)C)C=C2)SC=N1	C50H56F4N8O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-078MM9	SCHEMBL17951997	(2S,4R)-1-[(2S)-2-[6-[5-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]pentoxy]hexanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; FQCMASSNRBXZHZ-BZPYCXPJSA-N; (2S,4R)-1-[(2S)-2-[6-[5-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]pentoxy]hexanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCOCCCCCOC3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C52H62F3N7O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-V1W32O	WO2019023553A1_247	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCCCCOC3=CC=C(N4C(=O)N(C5=CC(C(F)(F)F)=C(C#N)C=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C50H58F3N7O9S	AR	P10275	VHL	WO-2019023553-A1
TPD-HG437P	WO2019023553A1_248	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC(CCCOCCOC5=CC=C(N6C(=S)N(C7=CC(C(F)(F)F)=C(C#N)C=C7)C(=O)C6(C)C)C=C5)=C4)C3=O)C=C2)SC=N1	C53H54F3N7O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-2GEAXX	WO2019023553A1_250	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C(OCCCOCCCOC3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3)=C2)SC=N1	C54H56F3N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-TWIK4D	WO2019023553A1_251	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC(CCCCCOC5=CC=C(N6C(=S)N(C7=CC(C(F)(F)F)=C(C#N)C=C7)C(=O)C6(C)C)C=C5)=C4)C3=O)C=C2)SC=N1	C53H54F3N7O6S2	AR	P10275	VHL	WO-2019023553-A1
TPD-202JO6	SCHEMBL17952386	(2S,4R)-1-[(2S)-2-[6-[4-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]ethoxy]butyl]-3-oxo-1H-isoindol-2-yl]-3-methylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; JHIPOHGZVGJYJN-BTOBHVHUSA-N; (2S,4R)-1-[(2S)-2-[6-[4-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]ethoxy]butyl]-3-oxo-1H-isoindol-2-yl]-3-methylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC(CCCCOCCOC5=CC=C(N6C(=S)N(C7=CC(C(F)(F)F)=C(C#N)C=C7)C(=O)C6(C)C)C=C5)=C4)C3=O)C=C2)SC=N1	C54H56F3N7O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-FLE5MM	SCHEMBL21743536	(2S,4R)-N-[[2-[3-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]propoxy]-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-4-hydroxy-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C(OCCCOC3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3)=C2)SC=N1	C51H50F3N7O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-B0X7PS	SCHEMBL17952538	(2S,4R)-1-[(2S)-2-[[2-[4-[5-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]pentoxy]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; FQFCHJIDNWEFCT-BZPYCXPJSA-N; (2S,4R)-1-[(2S)-2-[[2-[4-[5-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]pentoxy]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCOCCCCCOC3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C52H62F3N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-W1X555	SCHEMBL21743884	(2S,4R)-N-[[2-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]butoxy]-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-4-hydroxy-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C(OCCCCOC3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3)=C2)SC=N1	C52H52F3N7O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-8SV5GK	WO2019023553A1_257	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3=CC=C(OCCCCOC4=CC=C(N5C(=S)N(C6=CC(C(F)(F)F)=C(C#N)C=C6)C(=O)C5(C)C)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C52H54F3N7O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-AT9YDK	WO2019023553A1_258	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3=CC=C(OCCCCCOC4=CC=C(N5C(=S)N(C6=CC(C(F)(F)F)=C(C#N)C=C6)C(=O)C5(C)C)C=C4)C=C3)C(C)C)C=C2)SC=N1	C52H54F3N7O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-HV202J	SCHEMBL17952385	(2S,4R)-1-[(2S)-2-[5-[4-[3-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]propyl]phenoxy]pentanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; KAHPLWJHAVJBIQ-ZRKJWACOSA-N; (2S,4R)-1-[(2S)-2-[5-[4-[3-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]propyl]phenoxy]pentanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCOC3=CC=C(CCCOC4=CC=C(N5C(=S)N(C6=CC(C(F)(F)F)=C(C#N)C=C6)C(=O)C5(C)C)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C55H60F3N7O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-N4MR9M	WO2019023553A1_260	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCOCCOC3=CC=C(C4=CC=C(N5C(=S)N(C6=CC(C(F)(F)F)=C(C#N)C=C6)C(=O)C5(C)C)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C53H56F3N7O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-6K60NO	SCHEMBL19600074	(2S,4R)-N-[[2-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]ethoxy]-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-4-hydroxy-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]pyrrolidine-2-carboxamide; MELFYBGHHXLVRE-LVPGGGDRSA-N; (2S,4R)-N-[[2-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]ethoxy]-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-4-hydroxy-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C(OCCOC3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3)=C2)SC=N1	C50H48F3N7O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-7OIGGO	WO2019023553A1_262	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCCOC3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C50H58F3N7O9S2	AR	P10275	VHL	WO-2019023553-A1
TPD-SLBZPJ	SCHEMBL19600364	(2S,4R)-1-[(2S)-2-[[4-[2-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]butoxy]ethoxy]benzoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; WHOKKDHMPKJKFD-LFWXKOCQSA-N; (2S,4R)-1-[(2S)-2-[[4-[2-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]butoxy]ethoxy]benzoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3=CC=C(OCCOCCCCOC4=CC=C(N5C(=S)N(C6=CC(C(F)(F)F)=C(C#N)C=C6)C(=O)C5(C)C)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C54H58F3N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-ZZQMMJ	SCHEMBL17952530	(2S,4R)-1-[(2S)-2-[[4-[2-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]ethoxy]ethoxy]benzoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; PPXRYQSJZQWLHZ-YNOIGWCPSA-N; (2S,4R)-1-[(2S)-2-[[4-[2-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]ethoxy]ethoxy]benzoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3=CC=C(OCCOCCOC4=CC=C(N5C(=S)N(C6=CC(C(F)(F)F)=C(C#N)C=C6)C(=O)C5(C)C)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C52H54F3N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-7D1BDX	SCHEMBL17952149	(2S,4R)-1-[(2S)-2-[[4-[3-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]propoxy]benzoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; HANHWACUQSQRGO-BBSCUJAXSA-N; (2S,4R)-1-[(2S)-2-[[4-[3-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]propoxy]benzoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3=CC=C(OCCCOC4=CC=C(N5C(=S)N(C6=CC(C(F)(F)F)=C(C#N)C=C6)C(=O)C5(C)C)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C51H52F3N7O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-LN7C6K	WO2019023553A1_266	.	CC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=C(OCCOCCOCCOC2=CC=C(N3C(=S)N(C4=CC=C(C#N)C(C(F)(F)F)=C4)C(=O)C3(C)C)C=C2)C=C(C2=C(C)N=CS2)C=C1)C(C)(C)C	C49H56F3N7O9S2	AR	P10275	VHL	WO-2019023553-A1
TPD-Z6XYMK	WO2019023553A1_267	.	C=CC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=C(C)N=CS2)C=C1OCCOCCOCCOC1=CC=C(N2C(=S)N(C3=CC=C(C#N)C(C(F)(F)F)=C3)C(=O)C2(C)C)C=C1)C(C)(C)C	C50H56F3N7O9S2	AR	P10275	VHL	WO-2019023553-A1
TPD-IEAP6J	WO2019023553A1_268	.	C=CC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=C(C)N=CS2)C=C1OCCOCCOCCOC1=CC=C(N2C(=O)N(C3=CC=C(C#N)C(C(F)(F)F)=C3)C(=O)C2(C)C)C=C1)C(C)(C)C	C50H56F3N7O10S	AR	P10275	VHL	WO-2019023553-A1
TPD-T9AL66	WO2019023553A1_269	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C(C)C)C(C)(C)C)C(OCCOCCOCCOC3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3)=C2)SC=N1	C51H60F3N7O9S2	AR	P10275	VHL	WO-2019023553-A1
TPD-YD11G2	SCHEMBL17952000	(2S,4R)-N-[[2-[2-[2-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]ethoxy]ethoxy]ethoxy]-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-1-[(2S)-2-(2,2-dimethylpropanoylamino)-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide; ITRCMAHRZGRLOC-AKCINUCUSA-N; (2S,4R)-N-[[2-[2-[2-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]ethoxy]ethoxy]ethoxy]-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-1-[(2S)-2-(2,2-dimethylpropanoylamino)-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C(C)(C)C)C(C)(C)C)C(OCCOCCOCCOC3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3)=C2)SC=N1	C52H62F3N7O9S2	AR	P10275	VHL	WO-2019023553-A1
TPD-NQCG77	WO2019023553A1_271	.	CC(=O)NCC(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=C(OCCOCCOCCOC2=CC=C(N3C(=S)N(C4=CC=C(C#N)C(C(F)(F)F)=C4)C(=O)C3(C)C)C=C2)C=C(C2=C(C)N=CS2)C=C1	C45H48F3N7O9S2	AR	P10275	VHL	WO-2019023553-A1
TPD-MPHU0C	WO2019023553A1_272	.	CC(=O)N[C@@H](C)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=C(C)N=CS2)C=C1OCCOCCOCCOC1=CC=C(N2C(=O)N(C3=CC=C(C#N)C(C(F)(F)F)=C3)C(=O)C2(C)C)C=C1	C46H50F3N7O10S	AR	P10275	VHL	WO-2019023553-A1
TPD-PFFG86	WO2019023553A1_273	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC(CCCCOCCCOC5=CC=C(N6C(=O)N(C7=CC(C(F)(F)F)=C(C#N)C=C7)C(=O)C6C)C=C5)=C4)C3=O)C=C2)SC=N1	C54H56F3N7O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-5YS4WN	WO2019023553A1_274	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3=CC=C(OCCOCCCOC4=CC=C(N5C(=S)N(C6=CC(C(F)(F)F)=C(C#N)C=C6)C(=O)C5(C)C)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C53H56F3N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-N8017P	SCHEMBL17952546	(2S,4R)-1-[(2S)-2-[[2-[3-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]propoxy]benzoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; ZPHAHPCZIPSOFE-QIWIAYTASA-N; (2S,4R)-1-[(2S)-2-[[2-[3-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]propoxy]benzoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3=CC=CC=C3OCCCOC3=CC=C(N4C(=S)N(C5=CC(C(F)(F)F)=C(C#N)C=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C51H52F3N7O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-PI99IW	WO2019023553A1_276	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3=CC=CC=C3OCCCCOC3=CC=C(N4C(=S)N(C5=CC(C(F)(F)F)=C(C#N)C=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)OC=N1	C52H54F3N7O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-F9H2ZQ	WO2019023553A1_277	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3=CC(CCCOC4=CC=C(N5C(=S)N(C6=CC(C(F)(F)F)=C(C#N)C=C6)C(=O)C5(C)C)C=C4)=CC=C3)C(C)(C)C)C=C2)SC=N1	C51H52F3N7O6S2	AR	P10275	VHL	WO-2019023553-A1
TPD-SM6EHV	WO2019023553A1_278	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3=CC(OCCCCOC4=CC=C(N5C(=S)N(C6=CC(C(F)(F)F)=C(C#N)C=C6)C(=O)C5(C)C)C=C4)CC=C3)C(C)(C)C)C=C2)SC=N1	C52H56F3N7O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-DVRYBI	WO2019023553A1_279	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C(OCCCCOCCCOC3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3)=C2)SC=N1	C55H58F3N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-ECWYN5	WO2019023553A1_280	.	CC[C@H](NC(C)=O)C(=O)N1C[C@@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=C(C)N=CS2)C=C1OCCOCCOCCOC1=CC=C(N2C(=S)N(C3=CC=C(C#N)C(C(F)(F)F)=C3)C(=O)C2(C)C)C=C1	C47H52F3N7O9S2	AR	P10275	VHL	WO-2019023553-A1
TPD-UVQQGN	SCHEMBL17952145	(2S,4R)-1-[(2S)-2-acetamido-3-methylbutanoyl]-N-[[2-[2-[2-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]ethoxy]ethoxy]ethoxy]-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-4-hydroxypyrrolidine-2-carboxamide; GYAVGRGZOQIWQK-UDEWTJCRSA-N; (2S,4R)-1-[(2S)-2-acetamido-3-methylbutanoyl]-N-[[2-[2-[2-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]ethoxy]ethoxy]ethoxy]-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-4-hydroxypyrrolidine-2-carboxamide	CC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=C(C)N=CS2)C=C1OCCOCCOCCOC1=CC=C(N2C(=S)N(C3=CC=C(C#N)C(C(F)(F)F)=C3)C(=O)C2(C)C)C=C1)C(C)C	C48H54F3N7O9S2	AR	P10275	VHL	WO-2019023553-A1
TPD-GTQXW4	SCHEMBL19600023	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]ethoxy]ethoxy]benzoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; LZGLOUALPVNFRK-ZKAWRXRFSA-N; (2S,4R)-1-[(2S)-2-[[2-[2-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]ethoxy]ethoxy]benzoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3=CC=CC=C3OCCOCCOC3=CC=C(N4C(=S)N(C5=CC(C(F)(F)F)=C(C#N)C=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C52H54F3N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-SP5UXL	WO2019023553A1_283	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3=CC(OCCOCCOC4=CC=C(N5C(=O)C(C)(C)N(C6=CC(C(F)(F)F)=C(C#N)C(C(F)(F)F)=C6)C5=S)N=C4)=CC=C3)C(C)(C)C)C=C2)SC=N1	C52H52F6N8O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-Q615M2	WO2019023553A1_284	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3=CC=C(OCCCOC4=CC=C(C5=CC=C(N6C(=S)N(C7=CC(C(F)(F)F)=C(C#N)C=C7)C(=O)C6(C)C)C=C5)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C57H56F3N7O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-PPUO5O	SCHEMBL17947701	(2S,4R)-1-[(2S)-2-[[4-[4-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]phenoxy]butoxy]benzoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; LQNNPDBDULBBER-NAXMREFQSA-N; (2S,4R)-1-[(2S)-2-[[4-[4-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]phenoxy]butoxy]benzoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3=CC=C(OCCCCOC4=CC=C(C5=CC=C(N6C(=S)N(C7=CC(C(F)(F)F)=C(C#N)C=C7)C(=O)C6(C)C)C=C5)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C58H58F3N7O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-Z45R6C	WO2019023553A1_286	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3=CC=C(OCCOC4=CC=C(C5=CC=C(N6C(=S)N(C7=CC=C(C#N)C(C(F)(F)F)=C7)C(=O)C6(C)C)C=C5)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C56H54F3N7O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-SMJWH2	SCHEMBL17947595	(2S,4R)-1-[(2S)-2-[[4-[1-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]butyl]piperidin-4-yl]benzoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; AXEUWYFMPRTSGA-ZAWQOTONSA-N; (2S,4R)-1-[(2S)-2-[[4-[1-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]butyl]piperidin-4-yl]benzoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3=CC=C(C4CCN(CCCCOC5=CC=C(N6C(=S)N(C7=CC(C(F)(F)F)=C(C#N)C=C7)C(=O)C6(C)C)C=C5)CC4)C=C3)C(C)(C)C)C=C2)SC=N1	C57H63F3N8O6S2	AR	P10275	VHL	WO-2019023553-A1
TPD-BB8I3B	WO2019023553A1_288	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOC3=CC(C4=CC=C(N5C(=S)N(C6=CC=C(C#N)C(C(F)(F)F)=C6)C(=O)C5(C)C)C=C4)=CC=C3)C(C)(C)C)C=C2)SC=N1	C53H56F3N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-31WJRY	SCHEMBL17947026	(2S,4R)-1-[(2S)-2-[[4-[1-[3-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]propyl]piperidin-4-yl]benzoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; MIMFKHDKHZQSIS-DMMYSGTFSA-N; (2S,4R)-1-[(2S)-2-[[4-[1-[3-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]propyl]piperidin-4-yl]benzoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3=CC=C(C4CCN(CCCOC5=CC=C(N6C(=S)N(C7=CC(C(F)(F)F)=C(C#N)C=C7)C(=O)C6(C)C)C=C5)CC4)C=C3)C(C)(C)C)C=C2)SC=N1	C56H61F3N8O6S2	AR	P10275	VHL	WO-2019023553-A1
TPD-1NDUZD	SCHEMBL17952394	(2S,4R)-1-[(2S)-2-[[2-[3-[1-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]benzoyl]piperidin-4-yl]oxypropoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; IJABCJOUJBLZSI-UMWCMSNQSA-N; (2S,4R)-1-[(2S)-2-[[2-[3-[1-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]benzoyl]piperidin-4-yl]oxypropoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCOC3CCN(C(=O)C4=CC=C(N5C(=S)N(C6=CC(C(F)(F)F)=C(C#N)C=C6)C(=O)C5(C)C)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C52H59F3N8O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-V2AUMX	WO2019023553A1_291	.	CC(C)(C)[C@H](NC(=O)C1=CC=C(OCCOC2CCN(C(=O)C3=CC=C(N4C(=S)N(C5=CC(C(F)(F)F)=C(C#N)C=C5)C(=O)C4(C)C)C=C3)CC2)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=CN=CS2)C=C1	C55H57F3N8O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-30Z5CI	WO2019023553A1_292	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCC3=CC=C(OCCCOC4=CC=C(N5C(=S)N(C6=CC=C(C#N)C(C(F)(F)F)=C6)C(=O)C5(C)C)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C53H56F3N7O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-CH02JY	SCHEMBL19600032	(2S,4R)-1-[(2S)-2-[[2-[4-[1-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]benzoyl]piperidin-4-yl]oxybutoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC(C)(C)[C@H](NC(=O)COCCCCOC1CCN(C(=O)C2=CC=C(N3C(=S)N(C4=CC(C(F)(F)F)=C(C#N)C=C4)C(=O)C3(C)C)C=C2)CC1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=CN=CS2)C=C1	C52H59F3N8O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-K0LAG9	SCHEMBL17952551	(2S,4R)-1-[(2S)-2-[[2-[5-[1-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]benzoyl]piperidin-4-yl]oxypentoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; VBQDKVXNRLPZFR-PPZGWQTASA-N; (2S,4R)-1-[(2S)-2-[[2-[5-[1-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]benzoyl]piperidin-4-yl]oxypentoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCCOC3CCN(C(=O)C4=CC=C(N5C(=S)N(C6=CC(C(F)(F)F)=C(C#N)C=C6)C(=O)C5(C)C)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C54H63F3N8O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-GW5XH6	SCHEMBL19600395	(2S,4R)-1-[(2S)-2-[[2-[5-[3-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]propoxy]pentoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; AZRRNMGNHPPVOQ-UMWCMSNQSA-N; (2S,4R)-1-[(2S)-2-[[2-[5-[3-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]propoxy]pentoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCCOCCCOC3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C51H60F3N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-000ICQ	SCHEMBL21743542	(2S,4R)-1-[(2S)-2-[[2-[2-[3-[3-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]propyl]phenoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; PILQITMFHCPQBD-UJGSORPVSA-N; (2S,4R)-1-[(2S)-2-[[2-[2-[3-[3-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]propyl]phenoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOC3=CC(CCCOC4=CC=C(N5C(=S)N(C6=CC(C(F)(F)F)=C(C#N)C=C6)C(=O)C5(C)C)C=C4)=CC=C3)C(C)(C)C)C=C2)SC=N1	C54H58F3N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-N85XX8	WO2019023553A1_297	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C(OCCO[C@@H]3CCCC[C@@H]3OCCOC3=CC=C(N4C(=S)N(C5=CC(C(F)(F)F)=C(C#N)C=C5)C(=O)C4(C)C)C=C3)=C2)SC=N1	C58H62F3N7O9S2	AR	P10275	VHL	WO-2019023553-A1
TPD-63JEEE	SCHEMBL21743896	(2S,4R)-1-[(2S)-2-[[2-[3-[3-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]ethoxy]propoxy]phenyl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; VEVQLGVPLQGELU-UJGSORPVSA-N; (2S,4R)-1-[(2S)-2-[[2-[3-[3-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]ethoxy]propoxy]phenyl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CC3=CC=CC(OCCCOCCOC4=CC=C(N5C(=S)N(C6=CC(C(F)(F)F)=C(C#N)C=C6)C(=O)C5(C)C)C=C4)=C3)C(C)(C)C)C=C2)SC=N1	C54H58F3N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-OZHP5O	WO2019023553A1_299	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4CCCOCCOC4=CC=C(N5C(=S)N(C6=CC(C(F)(F)F)=C(C#N)C=C6)C(=O)C5(C)C)C=C4)C3=O)C=C2)SC=N1	C53H54F3N7O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-4M1JKU	SCHEMBL17952024	(2S,4R)-1-[(2S)-2-[4-[2-[3-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]propoxy]ethoxy]butanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SQWCFWLAGZSECP-AKCINUCUSA-N; (2S,4R)-1-[(2S)-2-[4-[2-[3-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]propoxy]ethoxy]butanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCOCCOCCCOC3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C50H58F3N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-OE9AQI	SCHEMBL17952013	(2S,4R)-1-[(2S)-2-[4-[3-[3-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]propoxy]propoxy]butanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; XNLVGLNNMHEUKC-UMWCMSNQSA-N; (2S,4R)-1-[(2S)-2-[4-[3-[3-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]propoxy]propoxy]butanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCOCCCOCCCOC3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C51H60F3N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-YFJ0DJ	WO2019023553A1_302	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCOC3=CC=C(CCOC4=CC=C(N5C(=S)N(C6=CC=C(C#N)C(C(F)(F)F)=C6)C(=O)C5(C)C)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C53H56F3N7O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-P1PY45	SCHEMBL17952027	(2S,4R)-1-[(2S)-2-[3-[4-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]ethoxy]phenyl]propanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; UUDAUCGNPVQRAC-CENKHQFISA-N; (2S,4R)-1-[(2S)-2-[3-[4-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]ethoxy]phenyl]propanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCC3=CC=C(OCCOC4=CC=C(N5C(=S)N(C6=CC=C(C#N)C(C(F)(F)F)=C6)C(=O)C5(C)C)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C52H54F3N7O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-7YPHJ7	WO2019023553A1_304	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C(OCCO[C@@H]3CCC[C@@H]3OCCOC3=CC=C(N4C(=S)N(C5=CC(C(F)(F)F)=C(C#N)C=C5)C(=O)C4(C)C)C=C3)=C2)SC=N1	C57H60F3N7O9S2	AR	P10275	VHL	WO-2019023553-A1
TPD-VY9IRP	WO2019023553A1_305	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CC(=O)CCCOCCCCCOC3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C52H60F3N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-ZI6HL1	SCHEMBL17952020	(2S,4R)-1-[(2S)-2-[3-[4-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]ethyl]phenoxy]propanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; YHMLXUXUYZDMOE-CENKHQFISA-N; (2S,4R)-1-[(2S)-2-[3-[4-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]ethyl]phenoxy]propanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCOC3=CC=C(CCOC4=CC=C(N5C(=S)N(C6=CC=C(C#N)C(C(F)(F)F)=C6)C(=O)C5(C)C)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C52H54F3N7O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-Q4F021	WO2019023553A1_307	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCOCCCOC3=CC=C(CN4C(=S)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C50H58F3N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-2JVVRH	WO2019023553A1_308	.	CC(C)(C)[C@H](NC(=O)COCCCOCCCCOC1=CC=C(CN2C(=S)N(C3=CC=C(C#N)C(C(F)(F)F)=C3)C(=O)C2(C)C)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=CN=CS2)C=C1	C50H58F3N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-1073U5	WO2019023553A1_309	.	C=C/C(=C\C=C\N1C(=S)N(C2=CC=C(C#N)C(C(F)(F)F)=C2)C(=O)C1(C)C)C1CCN(CCOCCCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)CC1	C52H63F3N8O6S2	AR	P10275	VHL	WO-2019023553-A1
TPD-ZMY2EZ	WO2019023553A1_310	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C(C)(C)C(O)CCCOCCCCCOC3=CC=C(N4C(=O)N(C5=CC(C(F)(F)F)=C(C#N)C=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C54H66F3N7O9S	AR	P10275	VHL	WO-2019023553-A1
TPD-H8CD9L	WO2019023553A1_311	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCN3CCC(C4=CC=C(N5C(=S)N(C6=CC=C(C#N)C(C(F)(F)F)=C6)C(=O)C5(C)C)C=C4)CC3)C(C)C)C=C2)SC=N1	C51H59F3N8O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-TKBCXI	WO2019023553A1_312	.	CC(C)(C)[C@H](NC(=O)CCCCOCCOCCOC1=CC=C(N2C(=S)N(C3=CC=C(C#N)C(C(F)(F)F)=C3)C(=O)C2(C)C)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](CC1=CC=C(C2=CN=CS2)C=C1)C(=O)O	C51H58F3N7O10S2	AR	P10275	VHL	WO-2019023553-A1
TPD-54YMX6	WO2019023553A1_313	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCOCCN3CCC(COC4=CC=C(N5C(=S)N(C6=CC=C(C#N)C(C(F)(F)F)=C6)C(=O)C5(C)C)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C52H61F3N8O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-K9V8O0	WO2019023553A1_314	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC(OCCOCCOC4=CC=C(N5C(=S)N(C6=CC(C(F)(F)F)=C(C#N)C=C6)C(=O)C5(C)C)C=C4)=CC3=O)C=C2)SC=N1	C48H50F3N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-NBL0W2	WO2019023553A1_315	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCOCCCOCCOC3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C50H58F3N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-9YV0H8	WO2019023553A1_316	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CNCCCCOCCCOC3=CC=C(N4C(=S)N(C5=CC(C(F)(F)F)=C(C#N)C=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C50H59F3N8O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-4MSXTR	SCHEMBL17952026	(2S,4R)-1-[(2S)-2-[[2-[4-[3-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]propoxy]butyl-methylamino]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; FUCRFGMGNNKCEJ-UMWCMSNQSA-N; (2S,4R)-1-[(2S)-2-[[2-[4-[3-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]propoxy]butyl-methylamino]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN(C)CCCCOCCCOC3=CC=C(N4C(=S)N(C5=CC(C(F)(F)F)=C(C#N)C=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C51H61F3N8O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-Q34D7R	SCHEMBL17947541	(2S,4R)-1-[(2S)-2-[[2-[2-[1-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]ethyl]piperidin-4-yl]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; VXTKHPZNNPMCRZ-BZPYCXPJSA-N; (2S,4R)-1-[(2S)-2-[[2-[2-[1-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]ethyl]piperidin-4-yl]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCC3CCN(CCOC4=CC=C(N5C(=S)N(C6=CC=C(C#N)C(C(F)(F)F)=C6)C(=O)C5(C)C)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C52H61F3N8O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-A56H4Q	SCHEMBL19598554	(2S,4R)-1-[(2S)-2-[[2-[4-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]ethoxy]but-2-ynoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; TYLZUAXCJNBFFZ-QLMCDVMBSA-N; (2S,4R)-1-[(2S)-2-[[2-[4-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]ethoxy]but-2-ynoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCC#CCOCCOC3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C49H52F3N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-JPPR8X	SCHEMBL17947484	(2S,4R)-1-[(2S)-2-[[2-[4-[4-[3-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]butoxy]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; ZFDOSGYCPQZOEP-UMWCMSNQSA-N; (2S,4R)-1-[(2S)-2-[[2-[4-[4-[3-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]butoxy]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCOCCCCOC3=CC=CC(N4C(=S)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)=C3)C(C)(C)C)C=C2)SC=N1	C51H60F3N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-2WZWM5	SCHEMBL17947708	(2S,4R)-1-[(2S)-2-[[2-[3-[4-[3-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]butoxy]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; HPJSWVVFWBDCPU-AKCINUCUSA-N; (2S,4R)-1-[(2S)-2-[[2-[3-[4-[3-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]butoxy]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCOCCCCOC3=CC=CC(N4C(=S)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)=C3)C(C)(C)C)C=C2)SC=N1	C50H58F3N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-100I4H	WO2019023553A1_322	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCN(C)CC3CC(OC4=CC=C(N5C(=S)N(C6=CC(C(F)(F)F)=C(C#N)N=C6)C(=O)C5(C)C)C=C4)C3)C(C)(C)C)C=C2)SC=N1	C51H60F3N9O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-WCYNU2	WO2019023553A1_323	.	COC1=CC(N2C(=O)C(C)(C)N(C3=CC=C(OCCOC4=CC=C(OCC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)NCC5=CC=C(C6=C(C)N=CS6)C=C5)C(C)(C)C)C=C4)C(F)=C3)C2=S)=CC=C1C#N	C51H54FN7O9S2	AR	P10275	VHL	WO-2019023553-A1
TPD-B91PKG	SCHEMBL17947485	(2S,4R)-1-[(2S)-2-[3-[4-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]ethoxy]piperidin-1-yl]propanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; BXYPFFKOAWLUAB-ZKAWRXRFSA-N; (2S,4R)-1-[(2S)-2-[3-[4-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]ethoxy]piperidin-1-yl]propanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCN3CCC(OCCOC4=CC=C(N5C(=S)N(C6=CC=C(C#N)C(C(F)(F)F)=C6)C(=O)C5(C)C)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C51H59F3N8O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-S6G1S2	WO2019023553A1_325	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COC/C=C/COCCCCOC3=CC=C(N4C(=S)N(C5=CC(C(F)(F)F)=C(C#N)C=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C51H58F3N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-SV02MZ	SCHEMBL17952029	(2S,4R)-1-[(2S)-2-[3-[2-[2-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]ethoxy]ethoxy]ethoxy]-5-oxo-2H-pyrrol-1-yl]-3-methylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; LIPRBTHVIKREGF-JNLFEYOZSA-N; (2S,4R)-1-[(2S)-2-[3-[2-[2-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]ethoxy]ethoxy]ethoxy]-5-oxo-2H-pyrrol-1-yl]-3-methylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC(OCCOCCOCCOC4=CC=C(N5C(=S)N(C6=CC(C(F)(F)F)=C(C#N)C=C6)C(=O)C5(C)C)C=C4)=CC3=O)C=C2)SC=N1	C50H54F3N7O9S2	AR	P10275	VHL	WO-2019023553-A1
TPD-ALRO62	WO2019023553A1_327	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C(=O)CCCCOCCCCCOC3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3)C(C)C)C=C2)SC=N1	C51H58F3N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-9CJ6D4	SCHEMBL21744036	(2S,4R)-1-[(2S)-2-[[2-[[2-[[2-[[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]acetyl]amino]acetyl]amino]acetyl]amino]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CNC(=O)CNC(=O)CNC(=O)COC3=CC=C(N4C(=S)N(C5=CC(C(F)(F)F)=C(C#N)C=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C49H53F3N10O9S2	AR	P10275	VHL	WO-2019023553-A1
TPD-PHODQO	SCHEMBL17952030	(2S,4R)-1-[(2S)-2-[3-[3-[3-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]propoxy]propoxy]-5-oxo-2H-pyrrol-1-yl]-3-methylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; QMQJJGZPAGFLHD-JNLFEYOZSA-N; (2S,4R)-1-[(2S)-2-[3-[3-[3-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]propoxy]propoxy]-5-oxo-2H-pyrrol-1-yl]-3-methylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC(OCCCOCCCOC4=CC=C(N5C(=S)N(C6=CC(C(F)(F)F)=C(C#N)C=C6)C(=O)C5(C)C)C=C4)=CC3=O)C=C2)SC=N1	C50H54F3N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-Q3A7IM	SCHEMBL17947617	(2S,4R)-1-[(2S)-2-[[2-[2-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]but-2-ynoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; ZXSOFBIMNZPTPQ-QLMCDVMBSA-N; (2S,4R)-1-[(2S)-2-[[2-[2-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]but-2-ynoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCC#CCOC3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C49H52F3N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-4AYUDP	WO2019023553A1_331	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN(C)C(=O)CN(C)C(=O)CN(C)C(=O)COC3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C52H59F3N10O9S2	AR	P10275	VHL	WO-2019023553-A1
TPD-7QU5X3	WO2019023553A1_332	.	CC1=C(C2=CC=C(C[C@H](C)C(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N(C)C(=O)[C@@H]3CCCN3C(=O)[C@@H]3CCCN3C(=O)[C@@H]3CCCN3C(=O)COC3=CC=C(N4C(=S)N(C5=CC(C(F)(F)F)=C(C#N)C=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C61H70F3N9O9S2	AR	P10275	VHL	WO-2019023553-A1
TPD-NNS0KX	SCHEMBL17947292	(2S,4R)-1-[(2S)-2-[[2-[3-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]anilino]butoxy]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; HQRZBAVSCJVEQP-JIJIMACASA-N; (2S,4R)-1-[(2S)-2-[[2-[3-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]anilino]butoxy]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCOCCCCNC3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C50H59F3N8O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-J4VHCG	WO2019023553A1_335	.	CC(C)(C)[C@H](NC(=O)COCCCOCCCCOC1=CC=C(N2C(=S)N(C3=CC=C(C#N)C(C#N)=C3)C(=O)C2(C)C)C=C1F)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=CN=CO2)C=C1	C49H55FN8O9S	AR	P10275	VHL	WO-2019023553-A1
TPD-7H9K43	WO2019023553A1_336	.	C=C1N(C2=CC=C(C#N)C(Cl)=C2)C(=O)C(C)(C)N1C1=CC=C(OCCCCOCCCOCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(C3=CN=CO3)C=C2)C(C)(C)C)C=C1F	C49H57ClFN7O9	AR	P10275	VHL	WO-2019023553-A1
TPD-E3G7AR	SCHEMBL17947489	(2S,4R)-1-[(2S)-2-[[2-[3-[4-[4-[3-(3-chloro-4-cyanophenyl)-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]butoxy]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(1,3-oxazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC(C)(C)[C@H](NC(=O)COCCCOCCCCOC1=CC=C(N2C(=S)N(C3=CC=C(C#N)C(Cl)=C3)C(=O)C2(C)C)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=CN=CO2)C=C1	C48H56ClN7O9S	AR	P10275	VHL	WO-2019023553-A1
TPD-FFR1WJ	SCHEMBL17947544	(2S,4R)-1-[(2S)-2-[[2-[3-[4-[4-[3-(5-chloro-6-cyanopyridin-3-yl)-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]butoxy]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-oxazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCOCCCCOC3=CC=C(N4C(=S)N(C5=CN=C(C#N)C(Cl)=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)OC=N1	C48H57ClN8O9S	AR	P10275	VHL	WO-2019023553-A1
TPD-J4L0VR	WO2019023553A1_339	.	CC1(C)C(NC(=O)C2=CN(CCOCCCCCCOCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCC3=CC=C(C4=CN=CS4)C=C3)C(C)(C)C)N=C2)C(C)(C)C1OC1=CC(Cl)=C(C#N)C=C1	C50H65ClN8O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-IPIVF3	SCHEMBL17947546	(2S,4R)-1-[(2S)-2-[[2-[3-[4-[4-[3-(3-chloro-4-cyanophenyl)-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]butoxy]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC(C)(C)[C@H](NC(=O)COCCCOCCCCOC1=CC=C(N2C(=S)N(C3=CC=C(C#N)C(Cl)=C3)C(=O)C2(C)C)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=CN=CS2)C=C1	C48H56ClN7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-G39ALE	SCHEMBL17947709	(2S,4R)-1-[(2S)-2-[[2-[3-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]-2-fluoroanilino]butoxy]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; KCQMPPOIMFEBST-QIWIAYTASA-N; (2S,4R)-1-[(2S)-2-[[2-[3-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]-2-fluoroanilino]butoxy]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCOCCCCNC3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3F)C(C)(C)C)C=C2)SC=N1	C50H58F4N8O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-3FAAO6	WO2019023553A1_342	.	CC(C)(C)[C@H](NC(=O)COCCCOCCCCOC1=CC=C(N2C(=S)N(C3=CC=C(C#N)C(Cl)=C3)C(=O)C2(C)C)C=C1F)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=CN=CO2)C(F)=C1	C48H54ClF2N7O9S	AR	P10275	VHL	WO-2019023553-A1
TPD-CH7GCI	WO2019023553A1_343	.	CC(C)(C)[C@H](NC(=O)COCCCCN1C=C(C2=CC=C(N3C(=S)N(C4=CC=C(C#N)C(Cl)=C4)C(=O)C3(C)C)C=C2)C=N1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=CN=CO2)C=C1	C48H52ClN9O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-VBIR8N	WO2019023553A1_344	.	CC(C)(C)[C@H](NC(=O)COCCCN1C=C(C2=CC=C(N3C(=S)N(C4=CC=C(C#N)C(Cl)=C4)C(=O)C3(C)C)C=C2)C=N1)C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](CC1=CC=C(C2=CN=CO2)C=C1)C(=O)O	C49H52ClN9O9S	AR	P10275	VHL	WO-2019023553-A1
TPD-SHV6AX	SCHEMBL19598564	(2S,4R)-1-[(2S)-2-[[2-[3-[5-[4-[3-(3-chloro-4-cyanophenyl)-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]pentoxy]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(1,3-oxazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC(C)(C)[C@H](NC(=O)COCCCOCCCCCOC1=CC=C(N2C(=S)N(C3=CC=C(C#N)C(Cl)=C3)C(=O)C2(C)C)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=CN=CO2)C=C1	C49H58ClN7O9S	AR	P10275	VHL	WO-2019023553-A1
TPD-D9ANRM	WO2019023553A1_346	.	CC(C)(C)[C@H](NC(=O)COCCCCOCCCCOC1=CC=C(N2C(=O)N(C3=CC=C(C#N)C(Cl)=C3)C(=O)C2(C)C)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=CN=CO2)C=C1	C49H58ClN7O10	AR	P10275	VHL	WO-2019023553-A1
TPD-ZAPBO7	SCHEMBL17947294	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-1-[2-[5-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[4-(1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]pentoxy]ethyl]pyrazole-4-carboxamide	CC(C)(C)[C@H](NC(=O)COCCCCCOCCN1C=C(C(=O)N[C@H]2C(C)(C)[C@H](OC3=CC(Cl)=C(C#N)C=C3)C2(C)C)C=N1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=CN=CS2)C=C1	C49H63ClN8O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-KOBAJF	WO2019023553A1_348	.	CC(C)(C)[C@H](NC(=O)COCCCOCCCCOC1=CC=C(N2C(=S)N(C3=CN=C(C#N)C(Cl)=C3)C(=O)C2(C)C)C=C1F)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=CN=CO2)C=C1	C47H54ClFN8O9S	AR	P10275	VHL	WO-2019023553-A1
TPD-E95WIZ	WO2019023553A1_349	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCOCC#CC3=CC=C(N4C(=O)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C49H52F3N7O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-HU1FTO	WO2019023553A1_350	.	CC(C)(C)[C@H](NC(=O)COCCCCOCCCOC1=CC=C(N2C(=S)N(C3=CC=C(C#N)C(C(F)(F)F)=C3)C(=O)C2(C)C)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=CN=CO2)C=C1	C49H56F3N7O9S	AR	P10275	VHL	WO-2019023553-A1
TPD-NPK6QY	SCHEMBL21744489	(2S,4R)-1-[(2S)-2-[[2-[4-[4-[4-[[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]methyl]phenyl]phenyl]phenoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; OKUJODVTHTWYOM-YAXWFMJISA-N; (2S,4R)-1-[(2S)-2-[[2-[4-[4-[4-[[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]methyl]phenyl]phenyl]phenoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COC3=CC=C(C4=CC=C(C5=CC=C(COC6=CC=C(N7C(=S)N(C8=CC=C(C#N)C(C(F)(F)F)=C8)C(=O)C7(C)C)C=C6)C=C5)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C62H58F3N7O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-6FNS01	WO2019023553A1_352	.	CC(C)[C@H](NC(=O)COCCCOCCCCOC1=CC=C(N2C(=S)N(C3=CN=C(C#N)C(C(F)(F)F)=C3)C(=O)C2(C)C)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=CN=CS2)C=C1	C47H53F3N8O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-A1PZLU	WO2019023553A1_353	.	CC(C)(C)[C@H](NC(=O)COCCCOCCCCOC1=CC=C(N2C(=S)N(C3=CC=C(C#N)C(Cl)=C3F)C(=O)C2(C)C)C=C1F)C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](CC1=CC=C(C2=CN=CO2)C=C1)C(=O)O	C50H56ClF2N7O11S	AR	P10275	VHL	WO-2019023553-A1
TPD-HJTPAT	WO2019023553A1_354	.	CC(C)(C)[C@H](NC(=O)COCCCOCCCCOC1=CC=C(N2C(=S)N(C3=CC=C(C#N)C(Cl)=C3F)C(=O)C2(C)C)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=CN=CO2)C=C1	C48H55ClFN7O9S	AR	P10275	VHL	WO-2019023553-A1
TPD-2U5IQ7	SCHEMBL19598570	(2S,4R)-1-[(2S)-2-[[2-[3-[5-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]pentoxy]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(1,3-oxazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; IJWCCTGNWBBHLM-AKCINUCUSA-N; (2S,4R)-1-[(2S)-2-[[2-[3-[5-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]pentoxy]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(1,3-oxazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC(C)(C)[C@H](NC(=O)COCCCOCCCCCOC1=CC=C(N2C(=S)N(C3=CC=C(C#N)C(C(F)(F)F)=C3)C(=O)C2(C)C)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=CN=CO2)C=C1	C50H58F3N7O9S	AR	P10275	VHL	WO-2019023553-A1
TPD-VODRNV	SCHEMBL17947622	(2S,4R)-1-[(2S)-2-[[2-[4-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]butoxy]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(1,3-oxazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; DNLRJMNDLPRBER-AKCINUCUSA-N; (2S,4R)-1-[(2S)-2-[[2-[4-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]butoxy]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(1,3-oxazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC(C)(C)[C@H](NC(=O)COCCCCOCCCCOC1=CC=C(N2C(=S)N(C3=CC=C(C#N)C(C(F)(F)F)=C3)C(=O)C2(C)C)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=CN=CO2)C=C1	C50H58F3N7O9S	AR	P10275	VHL	WO-2019023553-A1
TPD-97ULSA	SCHEMBL19598571	(2S,4R)-1-[(2S)-2-[[2-[3-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]butoxy]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; KLRJAFJEPALYMA-QMOPTUDDSA-N; (2S,4R)-1-[(2S)-2-[[2-[3-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]butoxy]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCOCCCCOC3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C51H60F3N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-6OFCK5	SCHEMBL17947299	(2S,4R)-1-[(2S)-2-acetamidopentanoyl]-N-[[2-[2-[2-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]ethoxy]ethoxy]ethoxy]-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-4-hydroxypyrrolidine-2-carboxamide; QMKWYKNOTHEHOS-JDDRPVQOSA-N; (2S,4R)-1-[(2S)-2-acetamidopentanoyl]-N-[[2-[2-[2-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]ethoxy]ethoxy]ethoxy]-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-4-hydroxypyrrolidine-2-carboxamide	CCC[C@H](NC(C)=O)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=C(C)N=CS2)C=C1OCCOCCOCCOC1=CC=C(N2C(=S)N(C3=CC=C(C#N)C(C(F)(F)F)=C3)C(=O)C2(C)C)C=C1	C48H54F3N7O9S2	AR	P10275	VHL	WO-2019023553-A1
TPD-FC6IPX	SCHEMBL17947713	(2S,4R)-1-[2-[[2-[3-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]butoxy]propoxy]acetyl]amino]acetyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; CZLFXWQWKJBBBU-UXMGRTHOSA-N; (2S,4R)-1-[2-[[2-[3-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]butoxy]propoxy]acetyl]amino]acetyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)CNC(=O)COCCCOCCCCOC3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3)C=C2)SC=N1	C46H50F3N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-93BYGC	WO2019023553A1_360	.	CC[C@H](NC(=O)COCCCOCCCCOC1=CC=C(N2C(=S)N(C3=CC=C(C#N)C(C(F)(F)F)=C3)C(=O)C2(C)C)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=C(C)N=CS2)C=C1	C48H54F3N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-51OCCN	WO2019023553A1_361	.	CCC[C@H](NC(=O)COCCCOCCCCOC1=CC=C(N2C(=S)N(C3=CC=C(C#N)C(C(F)(F)F)=C3)C(=O)C2(C)C)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=C(C)N=CS2)C=C1	C49H56F3N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-JXVCCZ	WO2019023553A1_362	.	CC(C)(C)[C@H](NC(=O)COCCCOCCCCOC1=CC=C(N2C(=S)N(C3=CN=C(C#N)C(C(F)(F)F)=C3)C(=O)C2(C)C)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=CN=CO2)C=C1	C48H55F3N8O9S	AR	P10275	VHL	WO-2019023553-A1
TPD-L3G1HA	WO2019023553A1_363	.	CC(C)(C)[C@H](NC(=O)COCCCOCCCCOC1=CC=C(N2C(=S)N(C3=CC=C(C#N)C(C(F)(F)F)=C3)C(=O)C2(C)C)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=C(F)C=C(C2=CN=CO2)C=C1F	C49H54F5N7O9S	AR	P10275	VHL	WO-2019023553-A1
TPD-ANYIE6	SCHEMBL17947625	(2S,4R)-1-[(2S)-2-[[2-[3-[4-[4-[7-[4-cyano-3-(trifluoromethyl)phenyl]-8-oxo-6-sulfanylidene-5,7-diazaspiro[3.4]octan-5-yl]phenoxy]butoxy]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(1,3-oxazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; XTHXBYASOFZSDW-AKCINUCUSA-N; (2S,4R)-1-[(2S)-2-[[2-[3-[4-[4-[7-[4-cyano-3-(trifluoromethyl)phenyl]-8-oxo-6-sulfanylidene-5,7-diazaspiro[3.4]octan-5-yl]phenoxy]butoxy]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(1,3-oxazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC(C)(C)[C@H](NC(=O)COCCCOCCCCOC1=CC=C(N2C(=S)N(C3=CC=C(C#N)C(C(F)(F)F)=C3)C(=O)C23CCC3)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=CN=CO2)C=C1	C50H56F3N7O9S	AR	P10275	VHL	WO-2019023553-A1
TPD-04OHF1	SCHEMBL21743923	(2S,4R)-1-[(2S)-2-[[2-[3-[4-[4-[3-[6-cyano-5-(trifluoromethyl)pyridin-3-yl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]butoxy]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; UPBITMFDGLLQJC-IMTMYWNSSA-N; (2S,4R)-1-[(2S)-2-[[2-[3-[4-[4-[3-[6-cyano-5-(trifluoromethyl)pyridin-3-yl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]butoxy]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCOCCCCOC3=CC=C(N4C(=S)N(C5=CN=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C50H59F3N8O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-K0BHEK	SCHEMBL17947628	(2S,4R)-1-[(2S)-2-[[2-[3-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]butoxy]propoxy]acetyl]amino]propanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; IQWWINPIZQDLER-ZLAMPTBQSA-N; (2S,4R)-1-[(2S)-2-[[2-[3-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]butoxy]propoxy]acetyl]amino]propanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C)NC(=O)COCCCOCCCCOC3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3)C=C2)SC=N1	C47H52F3N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-RS0CPY	WO2019023553A1_383	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCOC3=CC=C(OC4=CC=C(N5C(=S)N(C6=CN=C(C#N)C(C(F)(F)F)=C6)C(=O)C5(C)C)C=C4)C=C3)C(C)(C)C)C=C2)OC=N1	C52H55F3N8O9S	AR	P10275	VHL	WO-2019023553-A1
TPD-YUHAYI	WO2019023553A1_384	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCOC3=CC=C(OC4=CC=C(N5C(=S)N(C6=CN=C(C#N)C(C(F)(F)F)=C6)C(=O)C5(C)C)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C52H55F3N8O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-U48Y6X	WO2019023553A1_385	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCC(=O)N3CC=C(C4=CC=C(N5C(=S)N(C6=CC=C(C#N)C(Cl)=C6)C(=O)C5(C)C)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C52H59ClN8O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-ZH2NBR	SCHEMBL17947555	(2S,4R)-1-[(2S)-2-[[2-[3-[4-[4-[3-[6-cyano-5-(trifluoromethyl)pyridin-3-yl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]phenoxy]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-oxazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; VBFALKAAHATMMI-REMRPFBRSA-N; (2S,4R)-1-[(2S)-2-[[2-[3-[4-[4-[3-[6-cyano-5-(trifluoromethyl)pyridin-3-yl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]phenoxy]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-oxazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCOC3=CC=C(OC4=CC=C(N5C(=S)N(C6=CN=C(C#N)C(C(F)(F)F)=C6)C(=O)C5(C)C)C=C4)C=C3)C(C)(C)C)C=C2)OC=N1	C51H53F3N8O9S	AR	P10275	VHL	WO-2019023553-A1
TPD-0LKZ2L	WO2019023553A1_387	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCOC3=CC=C(C(=O)NC4C(C)(C)C(OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C49H59ClN6O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-M1COCA	SCHEMBL19598585	(2S,4R)-1-[(2S)-2-[[2-[4-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenoxy]but-2-ynoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCC#CCOC3=CC=C(C(=O)N[C@H]4C(C)(C)[C@H](OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C51H59ClN6O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-GQZ125	WO2019023553A1_390	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCNC3=CC=C(C4=CC=C(N5C(=S)N(C6=CN=C(C#N)C(C(F)(F)F)=C6)C(=O)C5(C)C)C=C4)C=C3)C(C)(C)C)C=C2)OC=N1	C53H58F3N9O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-ROVPHS	WO2019023553A1_391	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCNC3=CC=C(C4=CC=C(N5C(=S)N(C6=CN=C(C#N)C(C(F)(F)F)=C6)C(=O)C5(C)C)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C52H56F3N9O6S2	AR	P10275	VHL	WO-2019023553-A1
TPD-U9KA8J	SCHEMBL19580736	(2S,4R)-1-[2-[[2-[4-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenoxy]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(NC(=O)COCCCCOC3=CC=C(C(=O)N[C@H]4C(C)(C)[C@@H](OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C50H61ClN6O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-VZ9A03	SCHEMBL21744058	(2S,4R)-1-[(2S)-2-[[2-[4-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenoxy]butanoylamino]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CNC(=O)CCCOC3=CC=C(C(=O)N[C@H]4C(C)(C)[C@@H](OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C50H60ClN7O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-2Z3NCT	WO2019023553A1_394	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCOC3=CC=C(C4=CC=C(N5C(=S)N(C6=CC=C(C#N)C(C(F)(F)F)=C6)C(=O)C5(C)C)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C53H56F3N7O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-K1DI8U	WO2019023553A1_395	.	[2H]N(CC1=CC=C(C2=C(C)N=CS2)C=C1)C(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@H](C(C)C)N1C=CC=C(OCCCCOC2=CC=C(C3=CC=C(N4C(=S)N(C5=CC(C(F)(F)F)=C(C#N)C=C5)C(=O)C4(C)C)C=C3)C=C2)C1=O	C55H54F3N7O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-4AKYUL	WO2019023553A1_396	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCC3(F)CC4(C3)CC(F)(COC3=CC=C(N5C(=S)N(C6=CC=C(C#N)C(C(F)(F)F)=C6)C(=O)C5(C)C)C=C3)C4)C(C)(C)C)C=C2)OC=N1	C53H58F5N7O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-GRPK5P	WO2019023553A1_398	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCN(C)C(=O)C3=CC=C(C(=O)N[C@H]4C(C)(C)[C@@H](OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C52H64ClN7O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-KWC0KG	WO2019023553A1_399	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCOC3=CC=C(C4=CC=C(N5C(=S)N(C6=CC=C(C#N)C(C(F)(F)F)=C6)C(=O)C5(C)C)C=C4F)C=C3)C(C)(C)C)C=C2)OC=N1	C53H55F4N7O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-BUPJH5	WO2019023553A1_400	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCOC3=CC=C(C4=CC=C(N5C(=S)N(C6=CC=C(C#N)C(C(F)(F)F)=C6)C(=O)C5(C)C)C=C4F)C=C3)C(C)(C)C)C=C2)SC=N1	C53H55F4N7O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-T1TPU8	WO2019023553A1_401	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCOC3=CC=C(C4=CC=C(N5C(=S)N(C6=CC=C(C#N)C(C(F)(F)F)=C6)C(=O)C5(C)C)C=N4)C=N3)C(C)(C)C)C=C2)SC=N1	C52H56F3N9O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-ZVQRL7	SCHEMBL17952563	(2S,4R)-1-[(2S)-2-[[2-[3-[[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]benzoyl]amino]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-oxazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; PDUYKGLSBZWKRN-BPHNBMEGSA-N; (2S,4R)-1-[(2S)-2-[[2-[3-[[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]benzoyl]amino]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-oxazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCNC(=O)C3=CC=C(C4=CC=C(N5C(=S)N(C6=CC=C(C#N)C(C(F)(F)F)=C6)C(=O)C5(C)C)C=C4)C=C3)C(C)(C)C)C=C2)OC=N1	C53H55F3N8O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-BHF20W	WO2019023553A1_403	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCOC3=CC(O)=C(C4=CC=C(N5C(=S)N(C6=CC=C(C#N)C(C(F)(F)F)=C6)C(=O)C5(C)C)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C53H56F3N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-4JZGIL	WO2019023553A1_404	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCC3CCN(C4=CC=C(C(=O)N[C@H]5C(C)(C)[C@@H](OC6=CC=C(C#N)C(Cl)=C6)C5(C)C)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C53H66ClN7O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-O3QGWL	SCHEMBL17952041	(2S,4R)-1-[(2S)-2-[[2-[(1R)-1-[4-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenoxy]phenyl]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CO[C@H](C)C3=CC=C(OC4=CC=C(C(=O)N[C@H]5C(C)(C)[C@@H](OC6=CC(Cl)=C(C#N)C=C6)C5(C)C)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C54H61ClN6O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-O1CV2R	WO2019023553A1_406	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CO[C@@H](C)C3=CC=C(OC4=CC=C(C(=O)N[C@H]5C(C)(C)[C@H](OC6=CC(Cl)=C(C#N)C=C6)C5(C)C)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C54H61ClN6O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-MFGRFP	WO2019023553A1_407	.	CC(C)(C)[C@H](NC(=O)COCCCCOC1=CC=C(C(=O)N[C@H]2C(C)(C)[C@@H](OC3=CC=C(C#N)C(Cl)=C3)C2(C)C)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=CC=CC=C2)C=C1	C52H62ClN5O8	AR	P10275	VHL	WO-2019023553-A1
TPD-0DKAI5	SCHEMBL17947714	(2S,4R)-1-[(2S)-2-[[2-[4-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]-2-hydroxyphenoxy]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; BMBNOHZHLCBCSA-MSEXGENUSA-N; (2S,4R)-1-[(2S)-2-[[2-[4-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]-2-hydroxyphenoxy]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCOC3=C(O)C=C(C4=CC=C(N5C(=S)N(C6=CC=C(C#N)C(C(F)(F)F)=C6)C(=O)C5(C)C)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C53H56F3N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-ZF4JDQ	WO2019023553A1_409	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCNC(=O)C3=CC=C(C(=O)N[C@H]4C(C)(C)[C@@H](OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C50H60ClN7O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-FWMEOM	WO2019023553A1_410	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCC3CCN(C4=CC=C(C(=O)N[C@H]5C(C)(C)[C@@H](OC6=CC=C(C#N)C(Cl)=C6)C5(C)C)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C52H64ClN7O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-4HG6V0	SCHEMBL17947634	(2S,4R)-1-[(2S)-2-[[2-[4-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]anilino]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-oxazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCNC3=CC=C(C(=O)N[C@H]4C(C)(C)[C@@H](OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C(C)(C)C)C=C2)OC=N1	C51H64ClN7O8	AR	P10275	VHL	WO-2019023553-A1
TPD-D18GJU	WO2019023553A1_412	.	CC1(C)C(NC(=O)C2=CC=C(NCCCCOCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](CC3=CC=C(C4=C(C5CC5)N=CS4)C=C3)C(=O)O)C(C)(C)C)C=C2)C(C)(C)C1OC1=CC=C(C#N)C(Cl)=C1	C54H66ClN7O9S	AR	P10275	VHL	WO-2019023553-A1
TPD-36H6KR	SCHEMBL17947566	(2S,4R)-1-[(2S)-2-[[2-[4-[3-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]prop-2-ynoxy]phenoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; FRYOXUXHFVSROQ-CENKHQFISA-N; (2S,4R)-1-[(2S)-2-[[2-[4-[3-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]prop-2-ynoxy]phenoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COC3=CC=C(OCC#CC4=CC=C(N5C(=S)N(C6=CC=C(C#N)C(C(F)(F)F)=C6)C(=O)C5(C)C)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C52H50F3N7O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-A1HHZ9	WO2019023553A1_414	.	CCOC(=O)C1=C(C2=CC=C(CN(C)C(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCOC3=CC=C(C4=CC=C(N5C(=S)N(C6=CC(C(F)(F)F)=C(C#N)C=C6)C(=O)C5(C)C)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C56H60F3N7O9S2	AR	P10275	VHL	WO-2019023553-A1
TPD-5OJXOA	WO2019023553A1_415	.	CCC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCNC3=CC=C(C(=O)NC4C(C)(C)C(OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C51H64ClN7O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-FZUMRL	SCHEMBL17947556	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]butylamino]pyridine-3-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCNC3=NC=C(C(=O)N[C@H]4C(C)(C)[C@H](OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C49H61ClN8O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-SW1CSL	WO2019023553A1_417	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COC3=CC=CC=C3CCCOC3=CC=C(C(=O)N[C@H]4C(C)(C)[C@@H](OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C55H63ClN6O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-LZQJNN	WO2019023553A1_418	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C(OCCCOCCC(O)CCOC4=CC=C(N5C(=S)N(C6=CC=C(C#N)C(C(F)(F)F)=C6)C(=O)C5(C)C)C=C4)C=N3)C=C2)SC=N1	C52H59F3N8O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-EFN1EL	WO2019023553A1_419	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C(OCCCOCCC(O)CCOC4=CC=C(N5C(=S)N(C6=CC=C(C#N)C(C(F)(F)F)=C6)C(=O)C5(C)C)C=C4)C=N3)C=C2)OC=N1	C52H59F3N8O9S	AR	P10275	VHL	WO-2019023553-A1
TPD-8DZ5E0	SCHEMBL17947718	(2S,4R)-1-[(2S)-2-[[2-[[1-[5-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]pyridin-2-yl]piperidin-4-yl]methoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; RIKQCXGESSNQDO-DQFBHCSJSA-N; (2S,4R)-1-[(2S)-2-[[2-[[1-[5-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]pyridin-2-yl]piperidin-4-yl]methoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCC3CCN(C4=NC=C(C5=CC=C(N6C(=S)N(C7=CC=C(C#N)C(C(F)(F)F)=C7)C(=O)C6(C)C)C=C5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C54H58F3N9O6S2	AR	P10275	VHL	WO-2019023553-A1
TPD-Y5I5HS	WO2019023553A1_421	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COC3=CC=C(OC4C5CC6CC4CC(OC4=CC=C(N7C(=S)N(C8=CC=C(C#N)C(C(F)(F)F)=C8)C(=O)C7(C)C)C=C4)(C6)C5)N=C3)C(C)(C)C)C=C2)SC=N1	C59H63F3N8O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-4R415U	WO2019023553A1_422	.	CC1=NC(N2CC(OC3=CC4=C(C=C3)C=C(C(=O)N[C@H](C(=O)N3C[C@](C)(O)C[C@H]3C(=O)N[C@@H](C)C3=CC=C(C5=C(C)N=CS5)C=C3)C(C)(C)C)O4)C2)=NC=C1C(=O)NC1C(C)(C)C(OC2=CC=C(C#N)C(Cl)=C2)C1(C)C	C57H64ClN9O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-U1BOPU	WO2019023553A1_423	.	CC1=NC=CN1C1=CC=C([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](C(C)C)N2C=C(OCCCOCCCCCOC3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3)C=N2)N=C1	C51H59F3N10O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-TXFJL8	SCHEMBL19598597	(2S,4R)-1-[(2S)-2-[4-[3-[5-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]pentoxy]phenoxy]pyrazol-1-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[5-(4-methyl-1,3-thiazol-5-yl)pyridin-2-yl]ethyl]pyrrolidine-2-carboxamide; KUPQIKBOUHULOJ-OIPBKTSKSA-N; (2S,4R)-1-[(2S)-2-[4-[3-[5-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]pentoxy]phenoxy]pyrazol-1-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[5-(4-methyl-1,3-thiazol-5-yl)pyridin-2-yl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C(OC4=CC=CC(OCCCCCOC5=CC=C(N6C(=S)N(C7=CC=C(C#N)C(C(F)(F)F)=C7)C(=O)C6(C)C)C=C5)=C4)C=N3)N=C2)SC=N1	C54H56F3N9O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-D6A8NM	WO2019023553A1_425	.	CC1=NC=CN1C1=CC=C([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCNC2=NC=C(C3=CC=C(C(=O)NC4C(C)(C)C(OC5=CC(Cl)=C(C#N)C=C5)C4(C)C)C=C3)C=C2)C(C)(C)C)C=C1	C54H64ClN9O7	AR	P10275	VHL	WO-2019023553-A1
TPD-YIP31Y	SCHEMBL17947345	(2S,4R)-1-[(2R)-2-[4-[3-[5-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]pentoxy]propoxy]pyrazol-1-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[5-(4-methyl-1,3-thiazol-5-yl)pyridin-2-yl]ethyl]pyrrolidine-2-carboxamide; LIIYYDNLFBGCLR-HFQBVSOISA-N; (2S,4R)-1-[(2R)-2-[4-[3-[5-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]pentoxy]propoxy]pyrazol-1-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[5-(4-methyl-1,3-thiazol-5-yl)pyridin-2-yl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C(C)C)N3C=C(OCCCOCCCCCOC4=CC=C(N5C(=S)N(C6=CC=C(C#N)C(C(F)(F)F)=C6)C(=O)C5(C)C)C=C4)C=N3)N=C2)SC=N1	C51H58F3N9O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-R0WA47	WO2019023553A1_428	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C(OCCCOCCCCCOC4=CC=C(N5C(=S)N(C6=CC=C(C#N)C(C(F)(F)F)=C6)C(=O)C5(C)C)C=C4)C=N3)N=C2)SC=N1	C51H58F3N9O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-JR4EE4	WO2019023553A1_429	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COC3=CC=C(OC4CCN(C5=NC=C(N6C(=S)N(C7=CC=C(C#N)C(C(F)(F)F)=C7)C(=O)C6(C)C)C=C5)CC4)N=C3)C(C)(C)C)C=C2)SC=N1	C53H57F3N10O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-PH38JM	SCHEMBL17947350	(2S,4R)-1-[(2S)-2-[[2-[6-[1-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]piperidin-4-yl]oxypyridin-3-yl]oxyacetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; PEGXRKBQMCYTET-KCHVANSXSA-N; (2S,4R)-1-[(2S)-2-[[2-[6-[1-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]piperidin-4-yl]oxypyridin-3-yl]oxyacetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COC3=CC=C(OC4CCN(C5=CC=C(N6C(=S)N(C7=CC=C(C#N)C(C(F)(F)F)=C7)C(=O)C6(C)C)C=C5)CC4)N=C3)C(C)(C)C)C=C2)SC=N1	C54H58F3N9O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-0B56X4	WO2019023553A1_431	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C(OCCCOCCCCCOC4=CC=C(N5C(=S)N(C6=CC=C(C#N)C(C(F)(F)F)=C6)C(=O)C5(C)C)C=C4)C=N3)N=C2)SC=N1	C50H56F3N9O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-WJ3HUT	SCHEMBL17952037	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[5-(4-methyl-1,3-thiazol-5-yl)pyridin-2-yl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethyl]carbamoyl]phenoxy]pyridine-3-carboxamide; SCHEMBL21743571	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CNC(=O)C3=CC=C(OC4=CC=C(C(=O)N[C@H]5C(C)(C)[C@@H](OC6=CC=C(C#N)C(Cl)=C6)C5(C)C)C=N4)C=C3)C(C)(C)C)N=C2)SC=N1	C52H58ClN9O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-YJUCUP	WO2019023553A1_433	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C#CC3=CC=C(OC4CCC(OC5=CC=C(C(=O)N[C@H]6C(C)(C)[C@@H](OC7=CC=C(C#N)C(Cl)=C7)C6(C)C)C=C5)CC4)N=C3)C(C)(C)C)C=C2)SC=N1	C59H66ClN7O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-O0IYZ2	WO2019023553A1_434	.	C=C/C(=C\C=C(/C)[C@H](C)NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@H](C(C)C)N1C=C(OCCCOCCCCCOC2=CC=C(N3C(=S)N(C4=CC=C(C#N)C(C(F)(F)F)=C4)C(=O)C3(C)C)C=C2)C=N1)C1=C(C)N=CS1	C53H63F3N8O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-3USL9Z	WO2019023553A1_435	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C(OCCCOCCCCCOC4=CC=C(N5C(=S)N(C6=CC=C(C#N)C(C(F)(F)F)=C6)C(=O)C5(C)C)C=C4)C=N3)C=C2)SC=N1	C52H59F3N8O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-1TY4EA	WO2019023553A1_436	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C(OCC4CCN(C5=CC=C(C(=O)N[C@H]6C(C)(C)[C@@H](OC7=CC=C(C#N)C(Cl)=C7)C6(C)C)C=C5)CC4)C=N3)C=C2)SC=N1	C53H63ClN8O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-YL2AAA	WO2019023553A1_437	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=NC=C(COC4CCN(C5=CC=C(C(=O)NC6C(C)(C)C(OC7=CC=C(C#N)C(Cl)=C7)C6(C)C)C=C5)CC4)O3)C(C)C)C=C2)SC=N1	C53H62ClN7O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-LR590C	WO2019023553A1_438	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCN3CCN(C4=CC=C(C(=O)N[C@H]5C(C)(C)[C@@H](OC6=CC=C(C#N)C(Cl)=C6)C5(C)C)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C53H67ClN8O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-DFA5SH	WO2019023553A1_439	.	CC1=C(C2=CN=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCOCCCCCOC3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)N=C2)SC=N1	C50H60F3N9O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-A0AVWR	WO2019023553A1_440	.	CC1=NOC([C@H](C(=O)N2C[C@H](O)C[C@@H]2C(=O)NCC2=CC=C(C3=C(C)N=CS3)C=C2OCCCOCCCCCOC2=CC=C(N3C(=S)N(C4=CC=C(C#N)C(C(F)(F)F)=C4)C(=O)C3(C)C)C=C2)C(C)C)=C1	C52H58F3N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-AQMVYA	WO2019023553A1_441	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOC3=CC=C(C4=CC=C(C(=O)N[C@H]5CC56CC6OC5=CC=C(C#N)C(Cl)=C5)C=C4)C=N3)C(C)(C)C)C=C2)SC=N1	C51H54ClN7O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-SO0QLG	SCHEMBL17947051	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]methyl]piperidin-1-yl]pyridine-3-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCC3CCN(C4=CC=C(C(=O)NC5C(C)(C)C(OC6=CC=C(C#N)C(Cl)=C6)C5(C)C)C=N4)CC3)C(C)(C)C)C=C2)SC=N1	C52H65ClN8O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-XGHJMX	SCHEMBL21743948	(2S,4R)-1-[(2S)-2-[[2-[3-[5-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]pentoxy]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[6-(2-oxopyrrolidin-1-yl)pyridin-3-yl]methyl]pyrrolidine-2-carboxamide	CC(C)(C)[C@H](NC(=O)COCCCOCCCCCOC1=CC=C(N2C(=S)N(C3=CC=C(C#N)C(C(F)(F)F)=C3)C(=O)C2(C)C)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(N2CCCC2=O)N=C1	C50H61F3N8O9S	AR	P10275	VHL	WO-2019023553-A1
TPD-Q8ZXF2	WO2019023553A1_444	.	CC1=NC=CN1C1=CC=C([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CNC(=O)C2=CC=C(OC3=CC=C(C(=O)N[C@H]4C(C)(C)[C@H](OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C=C2)C(C)(C)C)C=C1	C54H61ClN8O8	AR	P10275	VHL	WO-2019023553-A1
TPD-71HTN0	WO2019023553A1_445	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCNC3=NC=C(C4=CC=C(C(=O)N[C@H]5C(C)(C)[C@@H](OC6=CC(Cl)=C(C#N)C=C6)C5(C)C)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C54H63ClN8O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-XHWQPP	WO2019023553A1_446	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCNC3=NC=C(C4=CC=C(C(=O)N[C@H]5C(C)(C)[C@H](OC6=CC(Cl)=C(C#N)C=C6)C5(C)C)C=C4)C=C3)C(C)(C)C)N=C2)SC=N1	C52H60ClN9O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-1VBYIN	SCHEMBL19598602	(2S,4R)-1-[(2S)-2-[[2-[[1-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenyl]piperidin-4-yl]methoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCC3CCN(C4=CC=C(C(=O)N[C@H]5C(C)(C)[C@H](OC6=CC=C(C#N)C(Cl)=C6)C5(C)C)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C53H66ClN7O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-6IHC7Z	SCHEMBL17952131	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethyl]carbamoyl]phenoxy]pyridine-3-carboxamide; SCHEMBL19600618	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CNC(=O)C3=CC=C(OC4=CC=C(C(=O)NC5C(C)(C)C(OC6=CC=C(C#N)C(Cl)=C6)C5(C)C)C=N4)C=C3)C(C)(C)C)C=C2)SC=N1	C53H59ClN8O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-NO4QVK	SCHEMBL19600582	(2S,4R)-1-[(2S)-2-[[2-[2-[4-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenyl]phenoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(2-methylimidazol-1-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=NC=CN1C1=CC=C([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOC2=CC=C(C3=CC=C(C(=O)N[C@H]4C(C)(C)[C@@H](OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C=C2)C(C)(C)C)C=C1	C55H64ClN7O8	AR	P10275	VHL	WO-2019023553-A1
TPD-VXQMFB	SCHEMBL17947641	(2S,4R)-1-[(2S)-2-[[2-[2-[4-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenyl]phenoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOC3=CC=C(C4=CC=C(C(=O)NC5C(C)(C)C(OC6=CC=C(C#N)C(Cl)=C6)C5(C)C)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C55H63ClN6O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-6Y6UY2	WO2019023553A1_451	.	CN(C)C1=NCC(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCCOCCCCCOC2=CC=C(N3C(=S)N(C4=CC=C(C#N)C(C(F)(F)F)=C4)C(=O)C3(C)C)C=C2)C(C)(C)C)C=C1	C48H63F3N8O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-4KRMAB	WO2019023553A1_452	.	C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](NC(=O)COCCCOCCCCCOC1=CC=C(N2C(=S)N(C3=CC=C(C#N)C(C(F)(F)F)=C3)C(=O)C2(C)C)C=C1)C(C)(C)C)C1C=CC(C2=NC=CN2C)=CC1	C52H65F3N8O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-IJQ3ZY	WO2019023553A1_453	.	CC1=C(C2=CN=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCOCCCCCOC3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)[C@@H]4C)C=C3)C(C)(C)C)C=C2)SC=N1	C49H57F3N8O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-H21V2A	WO2019023553A1_454	.	CC1=C(C2=CC=C([C@@H](C)NC(=O)[C@@H]3C[C@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCCNC3=CC=C(C(=O)N[C@H]4C(C)(C)[C@@H](OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C52H66ClN7O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-J16UYO	WO2019023553A1_455	.	[C-]#[N+]C1=C(Cl)C=C(O[C@H]2C(C)(C)[C@@H](NC(=C)C3=CC=C(NCCCCCOCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)N[C@@H](C)C4=CC=C(C5=C(C)N=CS5)C=C4)C(C)(C)C)C=C3)C2(C)C)C=C1	C53H68ClN7O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-JD2MIX	SCHEMBL21744518	(2S,4R)-1-[(2S)-2-[[2-[2-[1-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenyl]piperidin-4-yl]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCC3CCN(C4=CC=C(C(=O)N[C@H]5C(C)(C)[C@@H](OC6=CC=C(C#N)C(Cl)=C6)C5(C)C)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C54H68ClN7O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-ZK3O8E	WO2019023553A1_457	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCCNC3=CC=C(C(=O)NC4C(C)(C)C(OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=N3)C(C)(C)C)C=C2)SC=N1	C51H65ClN8O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-91G6DX	SCHEMBL17940958	(2S,4R)-1-((S)-2-(2-((5-((4-((trans-3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl)carbamoyl)phenyl)amino)pentyl)oxy)acetamido)-3,3-dimethylbutanoyl)-4-hydroxy-N-((S)-1-(4-(4-methylthiazol-5-yl)phenyl)ethyl)pyrrolidine-2-carboxamide; SCHEMBL17940961; SCHEMBL19598607; SCHEMBL24486167; SCHEMBL29817301; JQTRUKZGCBXQDD-IWHLCMBKSA-N; PD140947; (2S,4R)-1-((S)-2-(2-((5-((4-((trans-3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl)carbamoyl)phenyl)amino)pentyl)oxy)acetamido)-3,3-dimethylbutanoyl)-4-hydroxy-N-((S)-1-(4-(4-methylthiazol-5-yl)phenyl)ethyl)pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCCNC3=CC=C(C(=O)N[C@H]4C(C)(C)[C@@H](OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C52H66ClN7O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-B511PY	WO2019023553A1_459	.	CC1=C(C2=CC=C([C@@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCCNC3=CC=C(C(=O)N[C@H]4C(C)(C)[C@@H](OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C52H66ClN7O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-UOE4Z3	WO2019023553A1_460	.	CC(=O)[C@@H](NC(=O)C1=CC=C(NCCCCCOCC(=O)N[C@H](C(=O)N2C[C@H](OC(=O)[C@@H](N)CCCCN)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)C=C1)C(C)(C)COC1=CC=C(C#N)C(Cl)=C1	C57H76ClN9O9S	AR	P10275	VHL	WO-2019023553-A1
TPD-3W6TMJ	WO2019023553A1_461	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](OC(=O)[C@@H]4CCCN4)CN3C(=O)[C@@H](NC(=O)COCCCCCNC3=CC=C(C(=O)NC4C(C)(C)C(OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C57H73ClN8O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-0BFM3O	SCHEMBL17952056	[(3R,5S)-1-[(2S)-2-[[2-[5-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]anilino]pentoxy]acetyl]amino]-3,3-dimethylbutanoyl]-5-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-3-yl] (2S)-2-[[(2S)-2-amino-3-methylbutanoyl]amino]-3-methylbutanoate	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](OC(=O)[C@@H](NC(=O)[C@@H](N)C(C)C)C(C)C)CN3C(=O)[C@@H](NC(=O)COCCCCCNC3=CC=C(C(=O)NC4C(C)(C)C(OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C62H84ClN9O9S	AR	P10275	VHL	WO-2019023553-A1
TPD-3SRTLE	WO2019023553A1_463	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](OC(=O)[C@@H](N)C(C)C)CN3C(=O)[C@@H](NC(=O)COCCCCCNC3=CC=C(C(=O)NC4C(C)(C)C(OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C57H75ClN8O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-6LLZ5Q	WO2019023553A1_464	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCCNC3=CC=C(C(=O)NC4C(C)(C)C(OC5=CC=C(C#N)C(C(F)(F)F)=N5)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C52H65F3N8O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-97SYC6	SCHEMBL19598616	(2S,4R)-1-[(2S)-2-[[2-[5-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenoxy]pentoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1R)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]-2-pyrrolidin-1-ylethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CN3CCCC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCCOC3=CC=C(C(=O)NC4C(C)(C)C(OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C56H72ClN7O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-E7Z03S	WO2019023553A1_466	.	CC1=C(C2=CC=C([C@@H](CN3CCCC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCCOC3=CC=C(C(=O)N[C@H]4C(C)(C)[C@@H](OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C56H72ClN7O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-0U9CNP	WO2019023553A1_467	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](OC(=O)CN)CN3C(=O)[C@@H](NC(=O)COCCCCCNC3=CC=C(C(=O)N[C@H]4C(C)(C)[C@H](OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C54H69ClN8O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-CARXOZ	SCHEMBL21743619	[(3R,5S)-1-[(2S)-2-[[2-[5-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]anilino]pentoxy]acetyl]amino]-3,3-dimethylbutanoyl]-5-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-3-yl] 2-methylpropanoate	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](OC(=O)C(C)C)CN3C(=O)[C@@H](NC(=O)COCCCCCNC3=CC=C(C(=O)N[C@H]4C(C)(C)[C@@H](OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C56H72ClN7O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-B5FCRT	SCHEMBL21744085	[(3R,5S)-1-[(2S)-2-[[2-[5-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]anilino]pentoxy]acetyl]amino]-3,3-dimethylbutanoyl]-5-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-3-yl] acetate	CC(=O)O[C@@H]1C[C@@H](C(=O)N[C@@H](C)C2=CC=C(C3=C(C)N=CS3)C=C2)N(C(=O)[C@@H](NC(=O)COCCCCCNC2=CC=C(C(=O)NC3C(C)(C)C(OC4=CC=C(C#N)C(Cl)=C4)C3(C)C)C=C2)C(C)(C)C)C1	C54H68ClN7O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-PFY21G	WO2019023553A1_470	.	CC1=C(C2=CC=C([C@H](CN(C)C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCCOC3=CC=C(C(=O)N[C@H]4C(C)(C)[C@H](OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C54H70ClN7O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-22GTR8	WO2019023553A1_471	.	CC1=C(C2=CC=C([C@@H](CN(C)C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCCOC3=CC=C(C(=O)N[C@H]4C(C)(C)[C@H](OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C54H70ClN7O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-OTOY2N	SCHEMBL17947723	(2S,4R)-1-[(2S)-2-[[2-[2-[4-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenyl]phenoxy]ethylsulfonyl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CS(=O)(=O)CCOC3=CC=C(C4=CC=C(C(=O)NC5C(C)(C)C(OC6=CC=C(C#N)C(Cl)=C6)C5(C)C)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C54H61ClN6O9S2	AR	P10275	VHL	WO-2019023553-A1
TPD-89ZKDY	SCHEMBL17952039	(2S,4R)-1-[(2S)-2-[[2-[5-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-methylcarbamoyl]anilino]pentoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCCNC3=CC=C(C(=O)N(C)C4C(C)(C)C(OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C53H68ClN7O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-O19Y2F	WO2019023553A1_474	.	CC1=C(C2=CC=C([C@@H](CN)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCCOC3=CC=C(C(=O)N[C@H]4C(C)(C)[C@@H](OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C52H66ClN7O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-1C11XD	WO2019023553A1_475	.	CC1=C(C2=CC=C([C@H](CN)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCCOC3=CC=C(C(=O)NC4C(C)(C)C(OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C52H66ClN7O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-7985Y1	WO2019023553A1_476	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCCS(=O)(=O)C3=CC=C(C(=O)N[C@H]4C(C)(C)[C@H](OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C51H63ClN6O9S2	AR	P10275	VHL	WO-2019023553-A1
TPD-Y7UAA2	WO2019023553A1_477	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCOCCCCCOC3=CC=C(N4C(=S)N(C5=CC=CC=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C49H62N6O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-N5MZX1	WO2019023553A1_478	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCOCCCCCOC3=CC=C(N4C(=S)N(C5=CC(C(F)(F)F)=CC=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C50H61F3N6O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-V2DYE1	SCHEMBL17952429	(2S,4R)-1-[(2S)-2-[[2-[3-[5-[4-[3-(4-cyanophenyl)-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]pentoxy]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCOCCCCCOC3=CC=C(N4C(=S)N(C5=CC=C(C#N)C=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C50H61N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-DA3WDT	SCHEMBL17952060	(2S,4R)-1-[(2S)-2-[[2-[5-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]anilino]pentylamino]acetyl]amino]-3,3-dimethylbutanoyl]-N-[(4-cyanophenyl)methyl]-4-hydroxypyrrolidine-2-carboxamide	CC(C)(C)[C@H](NC(=O)CNCCCCCNC1=CC=C(C(=O)N[C@H]2C(C)(C)[C@H](OC3=CC=C(C#N)C(Cl)=C3)C2(C)C)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C#N)C=C1	C48H61ClN8O6	AR	P10275	VHL	WO-2019023553-A1
TPD-OR979Q	SCHEMBL17951966	(2S,4R)-1-[(2S)-2-[[2-[2-[4-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenyl]phenoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL20574467	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOC3=CC=C(C4=CC=C(C(=O)N[C@H]5C(C)(C)[C@@H](OC6=CC=C(C#N)C(Cl)=C6)C5(C)C)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C54H61ClN6O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-VWXZ5L	SCHEMBL17952054	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-5-[5-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]pentylamino]pyridine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCCNC3=CN=C(C(=O)N[C@H]4C(C)(C)[C@@H](OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C51H65ClN8O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-DCJHBY	SCHEMBL17952426	(2S,4R)-1-[(2S)-2-[[2-[2-[[5-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenyl]pyridin-2-yl]amino]ethylamino]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CNCCNC3=NC=C(C4=CC=C(C(=O)N[C@H]5C(C)(C)[C@@H](OC6=CC=C(C#N)C(Cl)=C6)C5(C)C)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C54H64ClN9O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-M8K59N	SCHEMBL17952078	(2S,4R)-1-[(2S)-2-[[2-[2-[[5-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenyl]pyridin-2-yl]amino]ethylamino]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CNCCNC3=NC=C(C4=CC=C(C(=O)N[C@H]5C(C)(C)[C@@H](OC6=CC=C(C#N)C(Cl)=C6)C5(C)C)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C53H62ClN9O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-84VGSH	SCHEMBL17947725	(2R,4S)-1-[(2S)-2-[[2-[5-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]anilino]pentoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@H]3C[C@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCCNC3=CC=C(C(=O)N[C@H]4C(C)(C)[C@@H](OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C52H66ClN7O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-P6NJKB	WO2019023553A1_486	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCCNC3=CC=C(C(=O)NC4C(C)(C)C(OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C52H66ClN7O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-3DFUJ0	WO2019023553A1_487	.	CCC[C@H](NC(=O)COCCCCCNC1=CC=C(C(=O)N[C@H]2C(C)(C)[C@H](OC3=CC(Cl)=C(C#N)C=C3)C2(C)C)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=C(C)N=CS2)C=C1	C50H62ClN7O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-HX9IJD	WO2019023553A1_488	.	CC[C@H](NC(=O)[C@H](CC)OCCCCCNC1=CC=C(C(=O)NC2C(C)(C)C(OC3=CC=C(C#N)C(Cl)=C3)C2(C)C)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=C(C)N=CS2)C=C1	C51H64ClN7O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-CF3PUO	SCHEMBL17952052	(2S,4R)-1-[(2S)-2-[[2-[5-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]anilino]pentoxy]acetyl]amino]propanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C)NC(=O)COCCCCCNC3=CC=C(C(=O)N[C@H]4C(C)(C)[C@H](OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C=C2)SC=N1	C48H58ClN7O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-SSKPNK	SCHEMBL17952061	(2S,4R)-1-[2-[[2-[5-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]anilino]pentoxy]acetyl]amino]acetyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)CNC(=O)COCCCCCNC3=CC=C(C(=O)N[C@H]4C(C)(C)[C@@H](OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C=C2)SC=N1	C47H56ClN7O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-E2GB6D	WO2019023553A1_491	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCCNC3=CC=C(C(=O)N[C@@H]4C(=NC5=C(C#N)C(C#N)=CN=C5Cl)OCC4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C50H59ClN10O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-8KPZOO	WO2019023553A1_492	.	CC(C)(C)[C@H](NC(=O)CC1=CC=C(C#CC2=CC=C(C(=O)N[C@H]3C(C)(C)[C@@H](OC4=CC=C(C#N)C(Cl)=C4)C3(C)C)C=C2)C=N1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CCC(C#N)C=C1	C50H54ClN7O6	AR	P10275	VHL	WO-2019023553-A1
TPD-BGQ9OR	WO2019023553A1_493	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](OC(=O)[C@@H](NC(=O)[C@@H](N)C(C)C)C(C)C)CN3C(=O)[C@@H](NC(=O)COCCCCOC3=CC=C(C(=O)NC4C(C)(C)C(OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C60H79ClN8O10S	AR	P10275	VHL	WO-2019023553-A1
TPD-8MXJ5X	WO2019023553A1_494	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](OC(=O)[C@@H](N)C(C)C)CN3C(=O)[C@@H](NC(=O)COCCCCOC3=CC=C(C(=O)N[C@H]4C(C)(C)[C@H](OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C55H70ClN7O9S	AR	P10275	VHL	WO-2019023553-A1
TPD-PHJVK3	WO2019023553A1_495	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCCNC3=CC(F)=C(C(=O)N[C@H]4C(C)(C)[C@H](OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C52H65ClFN7O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-NDIQLO	SCHEMBL17952044	(2S,4R)-1-[(2S)-2-[[2-[5-[4-[[3-(3-chloro-4-cyanophenoxy)cyclobutyl]carbamoyl]anilino]pentoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCCNC3=CC=C(C(=O)N[C@H]4C[C@H](OC5=CC=C(C#N)C(Cl)=C5)C4)C=C3)C(C)(C)C)C=C2)SC=N1	C48H58ClN7O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-TT4TVP	SCHEMBL19600663	(2S,4R)-1-[(2S)-2-[[2-[5-[4-[[3-[6-cyano-5-(trifluoromethyl)pyridin-3-yl]oxy-2,2,4,4-tetramethylcyclobutyl]carbamoyl]anilino]pentoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCCNC3=CC=C(C(=O)NC4C(C)(C)C(OC5=CN=C(C#N)C(C(F)(F)F)=C5)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C52H65F3N8O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-RGN9QJ	WO2019023553A1_498	.	CC1(C)C(NC(=O)C2=CC=C(C#CC3=CC=C(NCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)NCC4=CC=C(C#N)C=C4)C(C)(C)C)N=C3)C=C2)C(C)(C)C1OC1=CC=C(C#N)C(Cl)=C1	C50H53ClN8O6	AR	P10275	VHL	WO-2019023553-A1
TPD-IJLNK9	WO2019023553A1_499	.	CC(C)(C)[C@H](NC(=O)COCCCCCNC1=CC=C(C(=O)N[C@H]2C(C)(C)C[C@H](OC3=CC=C(C#N)C(Cl)=C3)C2(C)C)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=CCNCC2)C=C1	C53H70ClN7O7	AR	P10275	VHL	WO-2019023553-A1
TPD-P5YII5	WO2019023553A1_500	.	CC(C)(C)[C@H](NC(=O)CNCCNC1=NC=C(C2=CC=C(C(=O)N[C@H]3C(C)(C)[C@H](OC4=CC=C(C#N)C(Cl)=C4)C3(C)C)C=C2)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C#N)C=C1	C50H58ClN9O6	AR	P10275	VHL	WO-2019023553-A1
TPD-LRL8C9	WO2019023553A1_501	.	CC1(C)C(NC(=O)C2=CC=C(C3=CC=C(OCCNCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)NCC4=CC=C(C#N)C=C4)C(C)(C)C)C=C3)C=C2)C(C)(C)C1OC1=CC=C(C#N)C(Cl)=C1	C51H58ClN7O7	AR	P10275	VHL	WO-2019023553-A1
TPD-R43G3B	SCHEMBL17952100	5-[4-[[[(2S,4R)-1-[(2S)-2-[[2-[5-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]anilino]pentoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carbonyl]amino]methyl]phenyl]-1,3-thiazole-4-carboxylic acid	CC(C)(C)[C@H](NC(=O)COCCCCCNC1=CC=C(C(=O)N[C@H]2C(C)(C)[C@@H](OC3=CC=C(C#N)C(Cl)=C3)C2(C)C)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=C(C(=O)O)N=CS2)C=C1	C51H62ClN7O9S	AR	P10275	VHL	WO-2019023553-A1
TPD-LYDAOT	SCHEMBL17952412	(2S,4R)-N-[[4-(4-amino-1,3-thiazol-5-yl)phenyl]methyl]-1-[(2S)-2-[[2-[5-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]anilino]pentoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide	CC(C)(C)[C@H](NC(=O)COCCCCCNC1=CC=C(C(=O)N[C@H]2C(C)(C)[C@@H](OC3=CC=C(C#N)C(Cl)=C3)C2(C)C)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=C(N)N=CS2)C=C1	C50H63ClN8O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-B5G8PK	SCHEMBL19600279	(2S,4R)-1-[(2S)-2-[[2-[5-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]anilino]pentoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(1,2,4-thiadiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1(C)C(NC(=O)C2=CC=C(NCCCCCOCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCC3=CC=C(C4=NC=NS4)C=C3)C(C)(C)C)C=C2)C(C)(C)C1OC1=CC=C(C#N)C(Cl)=C1	C49H61ClN8O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-V7F5ZR	WO2019023553A1_505	.	CC(C)(C)[C@H](NC(=O)COCCCCCNC1=CC=C(C(=O)N[C@H]2C(C)(C)[C@@H](OC3=CC=C(C#N)C(Cl)=C3)C2(C)C)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(N2C=NN=N2)C=C1	C48H61ClN10O7	AR	P10275	VHL	WO-2019023553-A1
TPD-VZ3QI2	SCHEMBL19600732	(2S,4R)-1-[(2S)-2-[[2-[5-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]anilino]pentoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(tetrazol-2-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC(C)(C)[C@H](NC(=O)COCCCCCNC1=CC=C(C(=O)N[C@H]2C(C)(C)[C@@H](OC3=CC=C(C#N)C(Cl)=C3)C2(C)C)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(N2N=CN=N2)C=C1	C48H61ClN10O7	AR	P10275	VHL	WO-2019023553-A1
TPD-P7PMYZ	WO2019023553A1_507	.	CN(C)C(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](NC(=O)COCCCCCOC1=CC=C(C(=O)N[C@H]2C(C)(C)[C@H](OC3=CC=C(C#N)C(Cl)=C3)C2(C)C)C=C1)C(C)(C)C	C42H58ClN5O8	AR	P10275	VHL	WO-2019023553-A1
TPD-88CF6W	SCHEMBL17947640	(2S,4R)-1-[(2S)-2-[[2-[5-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenoxy]pentoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[2-(methylamino)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CNCC(NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](NC(=O)COCCCCCOC1=CC=C(C(=O)N[C@H]2C(C)(C)[C@@H](OC3=CC=C(C#N)C(Cl)=C3)C2(C)C)C=C1)C(C)(C)C)C1=CC=C(C2=C(C)N=CS2)C=C1	C53H68ClN7O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-8JLOAZ	WO2019023553A1_509	.	CC(C)(C)[C@H](NC(=O)COCCCCCOC1=CC=C(C(=O)N[C@H]2C(C)(C)[C@H](OC3=CC=C(C#N)C(Cl)=C3)C2(C)C)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)O	C40H53ClN4O9	AR	P10275	VHL	WO-2019023553-A1
TPD-37JDST	SCHEMBL17952566	(2S,4R)-1-[(2S)-2-[[2-[5-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]anilino]pentoxy]acetyl]amino]-3,3-dimethylbutanoyl]-N-[(4-cyano-2-methoxyphenyl)methyl]-4-hydroxypyrrolidine-2-carboxamide	COC1=CC(C#N)=CC=C1CNC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](NC(=O)COCCCCCNC1=CC=C(C(=O)NC2C(C)(C)C(OC3=CC=C(C#N)C(Cl)=C3)C2(C)C)C=C1)C(C)(C)C	C49H62ClN7O8	AR	P10275	VHL	WO-2019023553-A1
TPD-VXA1LO	WO2019023553A1_511	.	CNC(=O)C1=CC=C(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCCCCNC2=CC=C(C(=O)N[C@@H]3[C@H](C(C)(C)C)OC4=CC=C(C#N)C=C4C3(C)C)C=C2)C(C)(C)C)C=C1	C50H67N7O8	AR	P10275	VHL	WO-2019023553-A1
TPD-J6UUEV	SCHEMBL17952567	4-[[[(2S,4R)-1-[(2S)-2-[[2-[5-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]anilino]pentoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carbonyl]amino]methyl]benzoic acid	CC(C)(C)[C@H](NC(=O)COCCCCCNC1=CC=C(C(=O)N[C@H]2C(C)(C)[C@H](OC3=CC=C(C#N)C(Cl)=C3)C2(C)C)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C(=O)O)C=C1	C48H61ClN6O9	AR	P10275	VHL	WO-2019023553-A1
TPD-9IDCJZ	WO2019023553A1_513	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCNC3=NC=C(C4=C(F)C=C(C(=O)NC5C(C)(C)C(OC6=CC=C(C#N)C(Cl)=C6)C5(C)C)C=C4F)C=C3)C(C)(C)C)C=C2)SC=N1	C53H59ClF2N8O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-9RX3WV	WO2019023553A1_514	.	CC1=C(C2=CC=C([C@@H](CN(C)C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCCOC3=CC=C(C(=O)N[C@H]4C(C)(C)[C@@H](OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C54H70ClN7O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-N0FOQJ	WO2019023553A1_515	.	CNC[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](NC(=O)COCCCCCOC1=CC=C(C(=O)NC2C(C)(C)C(OC3=CC=C(C#N)C(Cl)=C3)C2(C)C)C=C1)C(C)(C)C)C1=CC=C(C2=C(C)N=CS2)C=C1	C53H68ClN7O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-Z55W90	SCHEMBL17952068	(2S,4R)-1-[(2S)-2-[[2-[5-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]anilino]pentoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[6-(4-methyl-1,3-thiazol-5-yl)pyridin-3-yl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCCNC3=CC=C(C(=O)N[C@H]4C(C)(C)[C@@H](OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C(C)(C)C)C=N2)SC=N1	C50H63ClN8O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-FCJCLK	SCHEMBL17952066	(2S,4R)-1-[(2S)-2-[[2-[5-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]anilino]pentoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(2H-triazol-4-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](NC(=O)COCCCCCNC1=CC=C(C(=O)NC2C(C)(C)C(OC3=CC=C(C#N)C(Cl)=C3)C2(C)C)C=C1)C(C)(C)C)C1=CC=C(C2=CNN=N2)C=C1	C50H64ClN9O7	AR	P10275	VHL	WO-2019023553-A1
TPD-OEMCBG	WO2019023553A1_518	.	CC(C)(C)[C@H](NC(=O)COCCCCCNC1=CC=C(C(=O)N[C@H]2C(C)(C)[C@@H](OC3=CC=C(C#N)C(Cl)=C3)C2(C)C)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=NN=NN2)C=C1	C48H61ClN10O7	AR	P10275	VHL	WO-2019023553-A1
TPD-0CQPDM	WO2019023553A1_519	.	COC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](NC(=O)COCCCCCOC1=CC=C(C(=O)N[C@H]2C(C)(C)[C@H](OC3=CC=C(C#N)C(Cl)=C3)C2(C)C)C=C1)C(C)(C)C	C41H55ClN4O9	AR	P10275	VHL	WO-2019023553-A1
TPD-SIPM3Y	SCHEMBL17952075	(2S,4R)-1-[(2S)-2-[[2-[5-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]anilino]pentoxy]acetyl]amino]-3-methylbutanoyl]-N-[(4-cyanophenyl)methyl]-4-hydroxypyrrolidine-2-carboxamide	CC(C)[C@H](NC(=O)COCCCCCNC1=CC=C(C(=O)NC2C(C)(C)C(OC3=CC=C(C#N)C(Cl)=C3)C2(C)C)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C#N)C=C1	C47H58ClN7O7	AR	P10275	VHL	WO-2019023553-A1
TPD-KGFPG0	WO2019023553A1_521	.	CC(C)(C)[C@H](NC(=O)COCCCCCNC1=CC=C(C(=O)N[C@H]2C(C)(C)[C@H](OC3=CC=C(C#N)C(Cl)=C3)C2(C)C)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=C(C#N)N=CS2)C=C1	C51H61ClN8O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-QY1EEU	SCHEMBL17952436	(2S,4R)-1-[(2S)-2-[[2-[5-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]anilino]pentoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(4-methoxyphenyl)methyl]pyrrolidine-2-carboxamide	COC1=CC=C(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCCCCNC2=CC=C(C(=O)N[C@H]3C(C)(C)[C@H](OC4=CC=C(C#N)C(Cl)=C4)C3(C)C)C=C2)C(C)(C)C)C=C1	C48H63ClN6O8	AR	P10275	VHL	WO-2019023553-A1
TPD-T8L0R0	WO2019023553A1_523	.	CC(C)(C)[C@H](NC(=O)COCCCCCNC1=CC=C(C(=O)N[C@H]2C(C)(C)[C@H](OC3=CC=C(C#N)C(Cl)=C3)C2(C)C)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](CC1=CC=C(C#N)N=C1)C(=O)O	C49H61ClN8O9	AR	P10275	VHL	WO-2019023553-A1
TPD-PC0F2K	SCHEMBL17947644	(2S,4R)-1-[(2S)-2-[[2-[2-[4-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenyl]anilino]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-N-[(4-cyanophenyl)methyl]-4-hydroxypyrrolidine-2-carboxamide	CC(C)(C)[C@H](NC(=O)COCCNC1=CC=C(C2=CC=C(C(=O)N[C@H]3C(C)(C)[C@@H](OC4=CC=C(C#N)C(Cl)=C4)C3(C)C)C=C2)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C#N)C=C1	C51H58ClN7O7	AR	P10275	VHL	WO-2019023553-A1
TPD-KL1NI0	WO2019023553A1_525	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCN3CCC(C4=CC=C(C(=O)N[C@@H]5C6=C(Cl)C(C#N)=CC=C6OCC5(C)C)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C50H60ClN7O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-S8MSNY	WO2019023553A1_526	.	CC(C)(C)[C@H](NC(=O)COCCCCCNC1=CC=C(C(=O)N[C@H]2C(C)(C)[C@@H](OC3=CC=C(C#N)C(Cl)=C3)C2(C)C)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(N2C=CN=N2)CC1	C49H64ClN9O7	AR	P10275	VHL	WO-2019023553-A1
TPD-0N0FAB	SCHEMBL17952430	(2S,4R)-1-[(2S)-2-[[2-[5-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]anilino]pentoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(triazol-2-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1(C)C(NC(=O)C2=CC=C(NCCCCCOCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCC3=CC=C(N4N=CC=N4)C=C3)C(C)(C)C)C=C2)C(C)(C)C1OC1=CC=C(C#N)C(Cl)=C1	C49H62ClN9O7	AR	P10275	VHL	WO-2019023553-A1
TPD-Z7PWQL	WO2019023553A1_528	(2S,4R)-1-[(2S)-2-[[2-[5-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]anilino]pentoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(1H-1,2,4-triazol-5-yl)cyclohexa-1,3-dien-1-yl]methyl]pyrrolidine-2-carboxamide	CC1(C)C(NC(=O)C2=CC=C(NCCCCCOCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCC3=CC=C(C4=NN=CN4)CC3)C(C)(C)C)C=C2)C(C)(C)C1OC1=CC=C(C#N)C(Cl)=C1	C49H64ClN9O7	AR	P10275	VHL	WO-2019023553-A1
TPD-J6NQ1V	WO2019023553A1_529	.	CC(C)(C)[C@H](NC(=O)COCCCCCNC1=CC=C(C(=O)N[C@H]2C(C)(C)[C@@H](OC3=CC=C(C#N)C(Cl)=C3)C2(C)C)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(N2CCC=CC2=O)CC1	C52H68ClN7O8	AR	P10275	VHL	WO-2019023553-A1
TPD-CPPWMI	WO2019023553A1_530	.	CC(C)(C)[C@H](NC(=O)COCCCCCNC1=CC=C(C(=O)N[C@H]2C(C)(C)[C@@H](OC3=CC=C(C#N)C(Cl)=C3)C2(C)C)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(N2C=NC=N2)CC1	C49H64ClN9O7	AR	P10275	VHL	WO-2019023553-A1
TPD-GCAN3B	SCHEMBL17952047	(2S,4R)-1-[(2S)-2-[[2-[5-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]anilino]pentoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(4-pyridazin-3-ylphenyl)methyl]pyrrolidine-2-carboxamide	CC(C)(C)[C@H](NC(=O)COCCCCCNC1=CC=C(C(=O)N[C@H]2C(C)(C)[C@@H](OC3=CC=C(C#N)C(Cl)=C3)C2(C)C)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=NN=CC=C2)C=C1	C51H63ClN8O7	AR	P10275	VHL	WO-2019023553-A1
TPD-WYFN72	SCHEMBL17952098	(2S,4R)-1-[(2S)-2-[[2-[5-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]anilino]pentoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(4-pyrazin-2-ylphenyl)methyl]pyrrolidine-2-carboxamide	CC(C)(C)[C@H](NC(=O)COCCCCCNC1=CC=C(C(=O)N[C@H]2C(C)(C)[C@@H](OC3=CC=C(C#N)C(Cl)=C3)C2(C)C)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=NC=CN=C2)C=C1	C51H63ClN8O7	AR	P10275	VHL	WO-2019023553-A1
TPD-XMKUWB	WO2019023553A1_533	.	CC1(C)C(NC(=O)C2=CC=C(NCCCCCOCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCC3=CC=C(C4=NC=NC=C4)C=C3)C(C)(C)C)C=C2)C(C)(C)C1OC1=CC=C(C#N)C(Cl)=C1	C51H63ClN8O7	AR	P10275	VHL	WO-2019023553-A1
TPD-G1PW5Q	WO2019023553A1_534	.	CC(C)(C)[C@H](NC(=O)COCCCCCNC1=CC=C(C(=O)N[C@H]2C(C)(C)[C@@H](OC3=CC=C(C#N)C(Cl)=C3)C2(C)C)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=CN=CN=C2)C=C1	C51H63ClN8O7	AR	P10275	VHL	WO-2019023553-A1
TPD-Y0KHGI	WO2019023553A1_535	.	CC1(C)C(NC(=O)C2=CC=C(NCCCCCOCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCC3=CC=C(C4=NC=CC=N4)C=C3)C(C)(C)C)C=C2)C(C)(C)C1OC1=CC=C(C#N)C(Cl)=C1	C51H63ClN8O7	AR	P10275	VHL	WO-2019023553-A1
TPD-UOPKBP	SCHEMBL17952120	(2S,4R)-1-[(2S)-2-[[2-[5-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]anilino]pentoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(4-pyridin-2-ylphenyl)methyl]pyrrolidine-2-carboxamide	CC1(C)C(NC(=O)C2=CC=C(NCCCCCOCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCC3=CC=C(C4=NC=CC=C4)C=C3)C(C)(C)C)C=C2)C(C)(C)C1OC1=CC=C(C#N)C(Cl)=C1	C52H64ClN7O7	AR	P10275	VHL	WO-2019023553-A1
TPD-5WANPM	SCHEMBL24486351	(2S,4R)-1-[(2S)-2-[[2-[5-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]anilino]pentoxy]acetyl]amino]-3-methylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCCNC3=CC=C(C(=O)N[C@H]4C(C)(C)[C@@H](OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C(C)C)C=C2)SC=N1	C50H62ClN7O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-WLMV7S	SCHEMBL19600356	(2S,4R)-1-[(2S)-2-[[2-[5-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]anilino]pentoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[5-(4-methyl-1,3-thiazol-5-yl)pyridin-2-yl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCCNC3=CC=C(C(=O)N[C@H]4C(C)(C)[C@@H](OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C(C)(C)C)N=C2)SC=N1	C50H63ClN8O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-DSQ5TJ	WO2019023553A1_539	.	CC1(C)C(NC(=O)C2=CC=C(NCCCCCOCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCC3=CC=C(C#N)C=N3)C(C)(C)C)C=C2)C(C)(C)C1OC1=CC=C(C#N)C(Cl)=C1	C47H59ClN8O7	AR	P10275	VHL	WO-2019023553-A1
TPD-ANBFN2	SCHEMBL17947605	(2S,4R)-1-[(2S)-2-[[2-[2-[[5-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenyl]pyridin-2-yl]amino]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-N-[(4-cyanophenyl)methyl]-4-hydroxypyrrolidine-2-carboxamide	CC1(C)C(NC(=O)C2=CC=C(C3=CN=C(NCCOCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)NCC4=CC=C(C#N)C=C4)C(C)(C)C)C=C3)C=C2)C(C)(C)C1OC1=CC=C(C#N)C(Cl)=C1	C50H57ClN8O7	AR	P10275	VHL	WO-2019023553-A1
TPD-B0SR8J	WO2019023553A1_541	.	CC1[C@H](NC(=O)C2=CC=C(NCCCCCOCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](C)C3=CC=C(C#N)C=C3)C(C)(C)C)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C48H60ClN7O7	AR	P10275	VHL	WO-2019023553-A1
TPD-EG86R4	SCHEMBL17952573	(2S,4R)-1-[(2S)-2-[[2-[5-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]anilino]pentoxy]acetyl]amino]-3,3-dimethylbutanoyl]-N-[(4-cyanophenyl)methyl]-4-hydroxypyrrolidine-2-carboxamide	CC(C)(C)[C@H](NC(=O)COCCCCCNC1=CC=C(C(=O)N[C@H]2C(C)(C)[C@H](OC3=CC=C(C#N)C(Cl)=C3)C2(C)C)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C#N)C=C1	C48H60ClN7O7	AR	P10275	VHL	WO-2019023553-A1
TPD-B9HVXV	WO2019023553A1_543	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOC3=CC=C(C4=C(F)C=C(C(=O)N[C@H]5C(C)(C)[C@H](OC6=CC=C(C#N)C(Cl)=C6)C5(C)C)C=C4F)C=C3)C(C)(C)C)C=C2)SC=N1	C54H59ClF2N6O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-DL3MTU	WO2019023553A1_544	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCN3CCN(C4=CC=C(C(=O)N[C@H]5C(C)(C)[C@@H](OC6=CC=C(C#N)C(Cl)=C6)C5(C)C)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C52H65ClN8O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-1UYV8R	WO2019023553A1_546	.	[2H]N(CC1=CC=C(C2=C(C)N=CS2)C=C1)C(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](NC(=O)COCCCCOC1=CC=C(C2=CC=C(N3C(=S)N(C4=CC(C(F)(F)F)=C(C#N)C=C4)C(=O)C3(C)C)C=C2)C=C1)C(C)(C)C(=O)O	C53H54F3N7O9S2	AR	P10275	VHL	WO-2019023553-A1
TPD-XESGB7	WO2019023553A1_547	.	CC(C)(C)[C@H](NC(=O)COCCCCNC1=CC=C(C(=O)N[C@H]2CC3=C(C2)C2=C(Cl)C(C#N)=CC=C2OCC3)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C#N)C=C1	C46H52ClN7O7	AR	P10275	VHL	WO-2019023553-A1
TPD-7LOV3I	WO2019023553A1_548	.	C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](NC(=O)COCCCCOC1=CC=C(C(=O)N[C@H]2C[C@H](OC3=CC=C(C#N)C(Cl)=C3)C2(C)C)C=C1)C(C)(C)C)C1=CC=C(C#N)C=C1	C46H55ClN6O8	AR	P10275	VHL	WO-2019023553-A1
TPD-1J6ML7	SCHEMBL17947646	(2S,4R)-1-[(2S)-2-[[2-[2-[4-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenyl]phenoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-N-[(1S)-1-(4-cyanophenyl)ethyl]-4-hydroxypyrrolidine-2-carboxamide	C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](NC(=O)COCCOC1=CC=C(C2=CC=C(C(=O)N[C@H]3C(C)(C)[C@@H](OC4=CC(Cl)=C(C#N)C=C4)C3(C)C)C=C2)C=C1)C(C)(C)C)C1=CC=C(C#N)C=C1	C52H59ClN6O8	AR	P10275	VHL	WO-2019023553-A1
TPD-AHOJP7	SCHEMBL17947357	(2S,4R)-1-[(2S)-2-[[2-[2-[4-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenyl]phenoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-N-[(4-cyanophenyl)methyl]-4-hydroxypyrrolidine-2-carboxamide	CC1(C)C(NC(=O)C2=CC=C(C3=CC=C(OCCOCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)NCC4=CC=C(C#N)C=C4)C(C)(C)C)C=C3)C=C2)C(C)(C)C1OC1=CC=C(C#N)C(Cl)=C1	C51H57ClN6O8	AR	P10275	VHL	WO-2019023553-A1
TPD-2NHWL9	WO2019023553A1_551	.	CC(C)(C)[C@H](NC(=O)COCCCCCNC1=NC=C(C(=O)N[C@H]2C(C)(C)[C@H](OC3=CC=C(C#N)C(Cl)=C3)C2(C)C)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](CC1=CC=C(C#N)C=C1)C(=O)O	C49H61ClN8O9	AR	P10275	VHL	WO-2019023553-A1
TPD-U5H3OZ	SCHEMBL17952434	(2S,4R)-1-[(2S)-2-[[2-[5-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]anilino]pentoxy]acetyl]amino]-3,3-dimethylbutanoyl]-N-[(4-chlorophenyl)methyl]-4-hydroxypyrrolidine-2-carboxamide	CC(C)(C)[C@H](NC(=O)COCCCCCNC1=CC=C(C(=O)N[C@H]2C(C)(C)[C@H](OC3=CC=C(C#N)C(Cl)=C3)C2(C)C)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(Cl)C=C1	C47H60Cl2N6O7	AR	P10275	VHL	WO-2019023553-A1
TPD-IJ3TPJ	SCHEMBL17947530	(2S,4R)-1-[(2S)-2-[[2-[2-[[5-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenyl]pyridin-2-yl]amino]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCNC3=NC=C(C4=CC=C(C(=O)NC5C(C)(C)C(OC6=CC=C(C#N)C(Cl)=C6)C5(C)C)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C53H61ClN8O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-IKFCH0	SCHEMBL17947608	(2S,4R)-1-[(2S)-2-[[2-[4-[[5-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]pyridin-2-yl]amino]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; AWWCSWDPWRHRQB-CKAMGQHKSA-N; (2S,4R)-1-[(2S)-2-[[2-[4-[[5-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]pyridin-2-yl]amino]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCNC3=NC=C(C4=CC=C(N5C(=S)N(C6=CC=C(C#N)C(C(F)(F)F)=C6)C(=O)C5(C)C)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C52H56F3N9O6S2	AR	P10275	VHL	WO-2019023553-A1
TPD-NK0F92	WO2019023553A1_555	.	CC1(C)C(NC(=O)C2=CC=C(NCCCCCOCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCC3=CC=C(C4=C(C5CC5)N=CS4)C=C3)C(C)(C)C)C=C2)C(C)(C)C1OC1=CC=C(C#N)C(Cl)=C1	C53H66ClN7O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-YBPR3I	WO2019023553A1_556	.	CC(C)C1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCCNC3=CC=C(C(=O)N[C@H]4C(C)(C)[C@@H](OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C53H68ClN7O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-L56H4H	SCHEMBL17952572	(2S,4R)-1-[(2S)-2-[[2-[4-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenoxy]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-N-[(1S)-1-(4-ethynylphenyl)ethyl]-4-hydroxypyrrolidine-2-carboxamide	C#CC1=CC=C([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCCCOC2=CC=C(C(=O)N[C@H]3C(C)(C)[C@H](OC4=CC=C(C#N)C(Cl)=C4)C3(C)C)C=C2)C(C)(C)C)C=C1	C49H60ClN5O8	AR	P10275	VHL	WO-2019023553-A1
TPD-0A1K5W	SCHEMBL24486374	[4-[[[(2S,4R)-1-[(2S)-2-[[2-[4-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenoxy]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carbonyl]amino]methyl]phenyl]boronic acid	CC(C)(C)[C@H](NC(=O)COCCCCOC1=CC=C(C(=O)N[C@H]2C(C)(C)[C@@H](OC3=CC=C(C#N)C(Cl)=C3)C2(C)C)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(B(O)O)C=C1	C46H59BClN5O10	AR	P10275	VHL	WO-2019023553-A1
TPD-XMDFK2	SCHEMBL17947645	(2S,4R)-1-[(2S)-2-[[2-[(2S,3S)-4-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]phenoxy]-2,3-dihydroxybutoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; NSOOKXDYDSWBOB-PRJGVKDFSA-N; (2S,4R)-1-[(2S)-2-[[2-[(2S,3S)-4-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]phenoxy]-2,3-dihydroxybutoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COC[C@H](O)[C@@H](O)COC3=CC=C(C4=CC=C(N5C(=S)N(C6=CC=C(C#N)C(C(F)(F)F)=C6)C(=O)C5(C)C)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C54H58F3N7O9S2	AR	P10275	VHL	WO-2019023553-A1
TPD-OWTOAR	SCHEMBL17952103	(2S,4R)-1-[(2S)-2-[[2-[5-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]anilino]pentoxy]acetyl]amino]-3,3-dimethylbutanoyl]-N-[[4-(4-ethyl-1,3-thiazol-5-yl)phenyl]methyl]-4-hydroxypyrrolidine-2-carboxamide	CCC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCCNC3=CC=C(C(=O)N[C@H]4C(C)(C)[C@@H](OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C52H66ClN7O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-QU3NH6	SCHEMBL17952438	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[5-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]pentylamino]pyridine-3-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCCNC3=NC=C(C(=O)NC4C(C)(C)C(OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C50H63ClN8O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-8JHZGF	SCHEMBL17947730	(2S,4R)-1-[(2S)-2-[[2-[4-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]anilino]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-propan-2-yl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC(C)C1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCNC3=CC=C(C(=O)N[C@H]4C(C)(C)[C@H](OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C52H66ClN7O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-N3X2GM	WO2019023553A1_563	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCC(O)[C@H](O)COC3=CC=C(C(=O)N[C@H]4C(C)(C)[C@@H](OC5=CC(Cl)=C(C#N)C=C5)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C50H61ClN6O10S	AR	P10275	VHL	WO-2019023553-A1
TPD-2CUKWI	SCHEMBL17947616	(2S,4R)-1-[(2S)-2-[[2-[[3-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenoxy]cyclobutyl]methoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL19598626	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCC3CC(OC4=CC=C(C(=O)N[C@H]5C(C)(C)[C@@H](OC6=CC=C(C#N)C(Cl)=C6)C5(C)C)C=C4)C3)C(C)(C)C)C=C2)SC=N1	C51H61ClN6O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-I501VU	(2S,4R)-1-[(2S)-2-[[2-[[3-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]phenoxy]cyclobutyl]methoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	(2S,4R)-1-[(2S)-2-[[2-[[3-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]phenoxy]cyclobutyl]methoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL17947353; SCHEMBL19598625; FHLFHEAAJCZJLI-JTBTVGNGSA-N; FHLFHEAAJCZJLI-XYVXPXNESA-N	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCC3CC(OC4=CC=C(C5=CC=C(N6C(=S)N(C7=CC=C(C#N)C(C(F)(F)F)=C7)C(=O)C6(C)C)C=C5)C=C4)C3)C(C)(C)C)C=C2)SC=N1	C54H56F3N7O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-U5J7I8	WO2019023553A1_566	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCC(O)C(O)COC3=CC=C(C4=CC=C(N5C(=S)N(C6=CC=C(C#N)C(C(F)(F)F)=C6)C(=O)C5(C)C)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C53H56F3N7O9S2	AR	P10275	VHL	WO-2019023553-A1
TPD-6O7TTS	WO2019023553A1_567	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COC[C@H](O)[C@@H](O)COC3=CC=C(C4=CC=C(N5C(=S)N(C6=CC=C(C#N)C(C(F)(F)F)=C6)C(=O)C5(C)C)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C53H56F3N7O9S2	AR	P10275	VHL	WO-2019023553-A1
TPD-IFB22Y	SCHEMBL17952439	(2S,4R)-1-[(2S)-2-[[2-[4-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenoxy]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(4-pyrazol-1-ylphenyl)methyl]pyrrolidine-2-carboxamide	CC(C)(C)[C@H](NC(=O)COCCCCOC1=CC=C(C(=O)N[C@H]2C(C)(C)[C@@H](OC3=CC=C(C#N)C(Cl)=C3)C2(C)C)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(N2C=CC=N2)C=C1	C49H60ClN7O8	AR	P10275	VHL	WO-2019023553-A1
TPD-2L30IC	WO2019023553A1_569	.	C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](NC(=O)COCCCCOC1=CC=C(C(=O)N[C@H]2C(C)(C)[C@@H](OC3=CC=C(C#N)C(Cl)=C3)C2(C)C)C=C1)C(C)(C)C)C1=CC=C(C2=NOC=N2)C=C1	C49H60ClN7O9	AR	P10275	VHL	WO-2019023553-A1
TPD-BI8R73	WO2019023553A1_570	.	C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](NC(=O)COCCCCOC1=CC=C(C(=O)N[C@H]2C(C)(C)[C@@H](OC3=CC=C(C#N)C(Cl)=C3)C2(C)C)C=C1)C(C)(C)C)C1=CC=C(C2=NN=CS2)C=C1	C49H60ClN7O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-E8RZ8B	SCHEMBL17947535	(2S,4R)-N-[(4-cyanophenyl)methyl]-1-[(2S)-2-[[2-[4-[4-[4-[3-[6-cyano-5-(trifluoromethyl)pyridin-3-yl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]phenoxy]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide; SIOIAYDRYXLAMZ-YLAZERGNSA-N; (2S,4R)-N-[(4-cyanophenyl)methyl]-1-[(2S)-2-[[2-[4-[4-[4-[3-[6-cyano-5-(trifluoromethyl)pyridin-3-yl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]phenoxy]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide	CC(C)(C)[C@H](NC(=O)COCCCCOC1=CC=C(C2=CC=C(N3C(=S)N(C4=CN=C(C#N)C(C(F)(F)F)=C4)C(=O)C3(C)C)C=C2)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C#N)C=C1	C49H51F3N8O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-HQXDVW	WO2019023553A1_572	.	C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](NC(=O)COCCCCOC1=CC=C(C(=O)NC2C(C)(C)C(OC3=CC=C(C#N)C(Cl)=C3)C2(C)C)C=C1)C(C)(C)C)C1=CC=C(Cl)C=C1	C47H59Cl2N5O8	AR	P10275	VHL	WO-2019023553-A1
TPD-E49WVD	SCHEMBL17947729	(2S,4R)-1-[(2S)-2-[[2-[2-[4-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenyl]phenoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-N-[(4-chlorophenyl)methyl]-4-hydroxypyrrolidine-2-carboxamide	CC(C)(C)[C@H](NC(=O)COCCOC1=CC=C(C2=CC=C(C(=O)N[C@H]3C(C)(C)[C@H](OC4=CC=C(C#N)C(Cl)=C4)C3(C)C)C=C2)C=C1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(Cl)C=C1	C50H57Cl2N5O8	AR	P10275	VHL	WO-2019023553-A1
TPD-YLZ3WT	WO2019023553A1_574	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COC[C@H](O)[C@H](O)COC3=CC=C(C4=CC=C(N5C(=S)N(C6=CC=C(C#N)C(C(F)(F)F)=C6)C(=O)C5(C)C)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C54H58F3N7O9S2	AR	P10275	VHL	WO-2019023553-A1
TPD-3E5SF7	WO2019023553A1_575	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCC(O)CCOC3=CC=C(C4=CC=C(N5C(=S)N(C6=CC=C(C#N)C(C(F)(F)F)=C6)C(=O)C5(C)C)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C54H58F3N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-HEIPES	SCHEMBL17947086	(2S,4R)-1-[(2S)-2-[[2-[(2R)-4-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]phenoxy]-2-hydroxybutoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; QULZOEZONYSCJK-LYYRDYKZSA-N; (2S,4R)-1-[(2S)-2-[[2-[(2R)-4-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]phenoxy]-2-hydroxybutoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COC[C@H](O)CCOC3=CC=C(C4=CC=C(N5C(=S)N(C6=CC=C(C#N)C(C(F)(F)F)=C6)C(=O)C5(C)C)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C54H58F3N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-7T15WK	SCHEMBL17947354	(2S,4R)-1-[(2S)-2-[[2-[(2S,3S)-4-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenoxy]-2,3-dihydroxybutoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COC[C@H](O)[C@@H](O)COC3=CC=C(C(=O)N[C@H]4C(C)(C)[C@@H](OC5=CC(Cl)=C(C#N)C=C5)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C50H61ClN6O10S	AR	P10275	VHL	WO-2019023553-A1
TPD-Y5X3RC	SCHEMBL17947536	(4R)-1-[(2S)-2-[[2-[5-[4-[[(2S)-1-[3-(3-chloro-4-cyanophenyl)pyrazol-1-yl]propan-2-yl]carbamoyl]phenoxy]pentoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)C3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCCOC3=CC=C(C(=O)N[C@@H](C)CN4C=CC(C5=CC(Cl)=C(C#N)C=C5)=N4)C=C3)C(C)(C)C)C=C2)SC=N1	C50H59ClN8O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-MOI30N	WO2019023553A1_579	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CNC(=O)C3=CC=C(OC4=CC=C(C(=O)N[C@@H](C)CN5C=CC(C6=CC(Cl)=C(C#N)C=C6)=N5)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C52H54ClN9O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-P2XEMC	WO2019023553A1_580	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(OCCCCCNC4=CC=C(C(=O)N[C@@H](C)CN5C=CC(C6=CC(Cl)=C(C#N)C=C6)=N5)C=C4)=NO3)C(C)C)C=C2)SC=N1	C50H56ClN9O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-WEYAP0	WO2019023553A1_581	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCNC3=CC=C(C4=CC=C(C(=O)N[C@@H](C)CN5C=CC(C6=CC(Cl)=C(C#N)C=C6)=N5)C=C4)C=N3)C(C)(C)C)C=C2)SC=N1	C52H57ClN10O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-DJ1JIB	WO2019023553A1_582	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COC(C)CN3CCN(C4=CC=C(C(=O)N[C@@H](C)CN5C=CC(C6=CC(Cl)=C(C#N)C=C6)=N5)C=N4)CC3)C(C)(C)C)C=C2)SC=N1	C51H62ClN11O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-ASUYEO	WO2019023553A1_583	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COC3=CC=C(OC4CCC(OC5=CC=C(C(=O)N[C@@H](C)CN6C=CC(C7=CC(Cl)=C(C#N)C=C7)=N6)C=C5)CC4)C=C3)C(C)(C)C)C=C2)SC=N1	C57H63ClN8O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-SIISAT	WO2019023553A1_584	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=C(OCCCCCNC4=CC=C(C(=O)N[C@@H](C)CN5CCC(C6=CC(Cl)=C(C#N)C=C6)=N5)C=C4)C=NO3)C(C)C)C=C2)SC=N1	C50H58ClN9O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-THYTUH	WO2019023553A1_585	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3=CC4=C(C=C(OC5CN(C6=CC=C(C(=O)NCCN7C=CC(C8=CC(Cl)=C(C#N)C=C8)=N7)C=N6)C5)C=C4)O3)C(C)(C)C)C=C2)SC=N1	C53H53ClN10O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-U6UFWE	WO2019023553A1_586	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCCNC3=CC=C(C(=O)N[C@@H](C)CN4C=CC(C5=CC(Cl)=C(C#N)C=C5)=N4)C=C3)C(C)(C)C)C=C2)SC=N1	C50H60ClN9O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-PGYCPI	WO2019023553A1_587	.	[C-]#[N+]C1=C(C#N)C=CC(C2=NN(C[C@H](C)NC(=O)C3=CC=C(N4CCC(C(C)OCC(=O)N[C@H](C(=C)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=C(C)N=CS6)C=C5)C(C)(C)C)CC4)C=C3)C=C2)=C1	C54H64N10O5S	AR	P10275	VHL	WO-2019023553-A1
TPD-NC3BX1	WO2019023553A1_588	.	CNC1=C(C#N)C=CC(C2=NN(C[C@H](C)NC(=O)C3=CC=C(N4CC(OC5=NC=CC(C6=CN([C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)C)N=C6)=C5)C4)C=C3)C=C2)=C1	C54H58N12O5S	AR	P10275	VHL	WO-2019023553-A1
TPD-R400DT	WO2019023553A1_589	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C(C4=CC=NC(N5CC[C@@H](NC6=CC=C(C(=O)N[C@@H](C)CN7C=CC(C8=CC(Cl)=C(C#N)C=C8)=N7)C=N6)C5)=C4)C=N3)C=C2)SC=N1	C53H56ClN13O4S	AR	P10275	VHL	WO-2019023553-A1
TPD-ODWFP1	WO2019023553A1_590	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCC#CC#CCOC3=CC=C(C(=O)N[C@@H](C)CN4C=CC(C5=CC(Cl)=C(C#N)C=C5)=N4)C=C3)C(C)(C)C)C=C2)SC=N1	C51H53ClN8O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-IJW0SP	WO2019023553A1_591	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOC3=CC=C(C(=O)N[C@@H](C)CN4C=CC(C5=CC(Cl)=C(C#N)C=C5)=N4)C=C3)C(C)(C)C)C=C2)SC=N1	C48H55ClN8O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-6UZTQG	WO2019023553A1_594	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C(C4=CC(OC5CN(C6=NC=C(C(=O)N[C@H]7C(C)(C)[C@H](OC8=CC=C(C#N)C(Cl)=C8)C7(C)C)C=C6)C5)=NC=C4)C=N3)C=C2)SC=N1	C54H59ClN10O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-VAD4JD	WO2019023553A1_595	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C(C4=CC(OC5CN(C6=NC=C(C(=O)N[C@H]7C(C)(C)[C@@H](OC8=CC=C(C#N)C(Cl)=C8)C7(C)C)C=C6)C5)=NC=C4)C=N3)C=C2)SC=N1	C54H59ClN10O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-O8TNYW	SCHEMBL19580776	(2S,4R)-1-[(2S)-2-[4-[2-[(3R)-3-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]anilino]pyrrolidin-1-yl]pyridin-4-yl]pyrazol-1-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL19580778; SCHEMBL31591761	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C(C4=CC(N5CC[C@@H](NC6=CC=C(C(=O)N[C@H]7C(C)(C)[C@@H](OC8=CC=C(C#N)C(Cl)=C8)C7(C)C)C=C6)C5)=NC=C4)C=N3)C=C2)SC=N1	C56H63ClN10O5S	AR	P10275	VHL	WO-2019023553-A1
TPD-4F9GXD	SCHEMBL19580847	(2S,4R)-1-[(2R)-2-[4-[2-[(3R)-3-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]anilino]pyrrolidin-1-yl]pyridin-4-yl]pyrazol-1-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL19580849; SCHEMBL31591742	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C(C)C)N3C=C(C4=CC(N5CC[C@@H](NC6=CC=C(C(=O)N[C@H]7C(C)(C)[C@@H](OC8=CC=C(C#N)C(Cl)=C8)C7(C)C)C=C6)C5)=NC=C4)C=N3)C=C2)SC=N1	C56H63ClN10O5S	AR	P10275	VHL	WO-2019023553-A1
TPD-96ASB2	WO2019023553A1_598	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C(OC4CCN(C5=NC=C(C6=CC=C(N7C(=S)N(C8=CC=C(C#N)C(C(F)(F)F)=C8)C(=O)C7(C)C)C=C6)C=C5)CC4)C=N3)C=C2)SC=N1	C53H53F3N10O5S2	AR	P10275	VHL	WO-2019023553-A1
TPD-VK30I0	SCHEMBL19598637	(2S)-1-[(2S)-2-[4-[3-[5-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]pentoxy]phenoxy]pyrazol-1-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; OFWGUMLYMVJRMF-HDUSVJMWSA-N; (2S)-1-[(2S)-2-[4-[3-[5-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]pentoxy]phenoxy]pyrazol-1-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3CC(O)CN3C(=O)[C@H](C(C)C)N3C=C(OC4=CC=CC(OCCCCCOC5=CC=C(N6C(=S)N(C7=CC=C(C#N)C(C(F)(F)F)=C7)C(=O)C6(C)C)C=C5)=C4)C=N3)C=C2)SC=N1	C55H57F3N8O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-Y8JFQP	SCHEMBL19600533	(2S)-1-[(2S)-2-[4-[3-[5-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]pentoxy]phenoxy]pyrazol-1-yl]-3-methylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3CC(O)CN3C(=O)[C@H](C(C)C)N3C=C(OC4=CC=CC(OCCCCCOC5=CC=C(N6C(=S)N(C7=CC=C(C#N)C(C(F)(F)F)=C7)C(=O)C6(C)C)C=C5)=C4)C=N3)C=C2)SC=N1	C54H55F3N8O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-ABR97V	WO2019023553A1_602	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@H](O)CN3C(=O)[C@H](C(C)C)N3C=C(OC4=CC=CC(OCCCCCOC5=CC=C(N6C(=O)N(C7=CC=C(C#N)C(C(F)(F)F)=C7)C(=O)C6(C)C)C=C5)=C4)C=N3)C=C2)SC=N1	C54H55F3N8O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-FLMX03	WO2019023553A1_603	.	CC1=C(C2=CC=C([C@@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C(C4=CC(OC5CN(C6=NC=C(C(=O)NC7C(C)(C)C(OC8=CC(Cl)=C(C#N)C=C8)C7(C)C)C=N6)C5)=NC=C4)C=N3)C=C2)SC=N1	C53H58ClN11O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-7XWTCL	SCHEMBL18086789	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-2-[3-[4-[1-[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]pyrazol-4-yl]pyridin-2-yl]oxyazetidin-1-yl]pyrimidine-5-carboxamide; SCHEMBL29817129	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C(C4=CC(OC5CN(C6=NC=C(C(=O)NC7C(C)(C)C(OC8=CC(Cl)=C(C#N)C=C8)C7(C)C)C=N6)C5)=NC=C4)C=N3)C=C2)SC=N1	C53H58ClN11O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-J1Q2ON	WO2019023553A1_605	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3=CC4=C(C=C(OC[C@H]5C[C@H](COC6=CC=C(N7C(=S)N(C8=CC=C(C#N)C(C(F)(F)F)=C8)C(=O)C7(C)C)C=C6)C5)C=C4)O3)C(C)(C)C)C=C2)SC=N1	C57H58F3N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-J2H94T	WO2019023553A1_606	.	CC1=NC=CN1C1=CC=C([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCC2CCN(C3=CC=C(C(=O)NC4C(C)(C)C(OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)N=N3)CC2)C(C)(C)C)C=C1	C51H65ClN10O7	AR	P10275	VHL	WO-2019023553-A1
TPD-4RUA55	WO2019023553A1_607	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCCNC3=NN=C(C(=O)NC4C(C)(C)C(OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=N3)C(C)(C)C)C=C2)SC=N1	C49H63ClN10O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-KJOIYT	SCHEMBL19581015	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[2-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]ethyl]piperazin-1-yl]pyridine-3-carboxamide; SCHEMBL19581017; SCHEMBL29817224	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCN3CCN(C4=NC=C(C(=O)NC5C(C)(C)C(OC6=CC=C(C#N)C(Cl)=C6)C5(C)C)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C52H66ClN9O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-0HYNL0	SCHEMBL19581172	(2S,4R)-1-[(2S)-2-[4-[2-[(3S)-3-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]pyrrolidin-1-yl]pyridin-4-yl]pyrazol-1-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL31591740; BNWZMXCLRUATIL-JHARUBOLSA-N; (2S,4R)-1-[(2S)-2-[4-[2-[(3S)-3-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]pyrrolidin-1-yl]pyridin-4-yl]pyrazol-1-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C(C4=CC=NC(N5CC[C@H](OC6=CC=C(N7C(=S)N(C8=CC=C(C#N)C(C(F)(F)F)=C8)C(=O)C7(C)C)C=C6)C5)=C4)C=N3)C=C2)SC=N1	C53H53F3N10O5S2	AR	P10275	VHL	WO-2019023553-A1
TPD-8IHFDP	SCHEMBL19581308	(2S,4R)-1-[(2S)-2-[4-[3-[5-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]pentoxy]propoxy]pyrazol-1-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(2-methylimidazol-1-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL29817131; LJOIUPLCIGMUFN-GXDNTIOLSA-N; (2S,4R)-1-[(2S)-2-[4-[3-[5-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]pentoxy]propoxy]pyrazol-1-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(2-methylimidazol-1-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=NC=CN1C1=CC=C([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](C(C)C)N2C=C(OCCCOCCCCCOC3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3)C=N2)C=C1	C52H60F3N9O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-6VUEY6	WO2019023553A1_613	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCOCCC(O)CCOC3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C52H62F3N7O9S2	AR	P10275	VHL	WO-2019023553-A1
TPD-DKG85I	WO2019023553A1_614	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCOC(COCCCCCOC4=CC=C(N5C(=S)N(C6=CC=C(C#N)C(C(F)(F)F)=C6)C(=O)C5(C)C)C=C4)C3)C(C)(C)C)C=C2)SC=N1	C54H65F3N8O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-57C15T	SCHEMBL19598643	(2S,4R)-1-[(2S)-2-[[2-[4-[2-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenoxy]ethyl]piperazin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL29817513	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCN(CCOC4=CC=C(C(=O)NC5C(C)(C)C(OC6=CC=C(C#N)C(Cl)=C6)C5(C)C)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C53H67ClN8O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-C2736L	WO2019023553A1_616	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@H](O)CN3C(=O)[C@H](C(C)C)N3C=C(OCC#CC#CCOC4=CC=C(N5C(=S)N(C6=CC=C(C#N)C(C(F)(F)F)=C6)C(=O)C5(C)C)C=C4)C=N3)C=C2)SC=N1	C49H45F3N8O6S2	AR	P10275	VHL	WO-2019023553-A1
TPD-GNKGFK	WO2019023553A1_617	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=NC(C4=CC=NC(N5CCC(OC6=CC=C(N7C(=S)N(C8=CC=C(C#N)C(C(F)(F)F)=C8)C(=O)C7(C)C)C=C6)C5)=C4)=C3)C=C2)SC=N1	C53H53F3N10O5S2	AR	P10275	VHL	WO-2019023553-A1
TPD-GDAQ1I	WO2019023553A1_618	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCOCCCCCNC3=NC=C(N4C(=S)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C51H62F3N9O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-QX1866	WO2019023553A1_619	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](OC(=O)CC/C=C/CCC(=O)O)CN3C(=O)[C@@H](NC(=O)COCCCOCCCCCCCC(=O)OCCCOC3=CC=C(N4C(=S)N(C5=CC(C(F)(F)F)=C(C#N)C=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C66H82F3N7O13S2	AR	P10275	VHL	WO-2019023553-A1
TPD-1PIJFF	WO2019023553A1_620	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](OC(=O)CCCCCCC(=O)O)CN3C(=O)[C@@H](NC(=O)COCCCOCCC(CCOC3=CC=C(N4C(=S)N(C5=CC(C(F)(F)F)=C(C#N)C=C5)C(=O)C4(C)C)C=C3)OC(=O)CCCCCCC(=O)O)C(C)(C)C)C=C2)SC=N1	C68H86F3N7O15S2	AR	P10275	VHL	WO-2019023553-A1
TPD-68B2PJ	WO2019023553A1_621	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCOCCC(CCOC3=CC=C(N4C(=S)N(C5=CC(C(F)(F)F)=C(C#N)C=C5)C(=O)C4(C)C)C=C3)OC(=O)CCC3=CN(CCCCCC(=O)O[C@H](C)C4=CC=C(C5=C(C)N=CS5)C=C4)N=N3)C(C)(C)C)C=C2)SC=N1	C75H88F3N11O12S3	AR	P10275	VHL	WO-2019023553-A1
TPD-2CYM7K	SCHEMBL21743686	(2S,4R)-1-[(2S)-2-[[2-[(2S)-2-[[(2R)-2-[[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]methyl]morpholin-4-yl]methyl]morpholin-4-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL29817488	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCO[C@@H](CN4CCO[C@@H](COC5=CC=C(N6C(=S)N(C7=CC=C(C#N)C(C(F)(F)F)=C7)C(=O)C6(C)C)C=C5)C4)C3)C(C)(C)C)C=C2)SC=N1	C54H64F3N9O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-9FY27U	SCHEMBL21712848	(2S,4R)-1-[(2S)-2-[[2-[4-[2-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenoxy]ethoxy]piperidin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL29817541	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCC(OCCOC4=CC=C(C(=O)NC5C(C)(C)C(OC6=CC=C(C#N)C(Cl)=C6)C5(C)C)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C54H68ClN7O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-SMI0WX	SCHEMBL19581250	(2S,4R)-1-[(2S)-2-[5-[5-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]anilino]pentoxy]pyrazol-1-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL19581253; SCHEMBL29817505	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3N=CC=C3OCCCCCNC3=CC=C(C(=O)NC4C(C)(C)C(OC5=CC(Cl)=C(C#N)C=C5)C4(C)C)C=C3)C=C2)SC=N1	C52H63ClN8O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-E7W07E	WO2019023553A1_626	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCC3(CNC4=CC=C(C(=O)NC5C(C)(C)C(OC6=CC=C(C#N)C(Cl)=C6)C5(C)C)C=C4)COC3)C(C)(C)C)C=C2)SC=N1	C53H66ClN7O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-LNOU9Y	WO2019023553A1_627	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C(OC4=CN=C(OC5CCC(OC6=CC=C(N7C(=S)N(C8=CC=C(C#N)C(C(F)(F)F)=C8)C(=O)C7(C)C)C=C6)CC5)C=C4)C=N3)C=C2)SC=N1	C55H56F3N9O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-ZGYN7K	WO2019023553A1_628	.	[C-]#[N+]C1=CC=C(N2C(=O)C(C)(C)N(C3=CC=C(OC4CCC(OC5=NC=C(OC6=CN([C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)C)N=C6)C=C5)CC4)C=C3)C2=S)C=C1C(F)(F)F	C55H56F3N9O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-20Z8J9	WO2019023553A1_629	.	COCCOCC(=O)NC(C(=O)N1C[C@@H](OC(=O)CCC2=CN(CCCCCC(=O)OC(CCCOCCOCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](C)C3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)CCOC3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3)N=N2)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=C(C)N=CS2)C=C1)C(C)(C)C	C91H115F3N14O17S3	AR	P10275	VHL	WO-2019023553-A1
TPD-TG5IL4	SCHEMBL21712824	(2S,4R)-1-[(2S)-2-[[2-[4-[4-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenyl]phenoxy]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL29817199	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCOC3=CC=C(C4=CC=C(C(=O)NC5C(C)(C)C(OC6=CC=C(C#N)C(Cl)=C6)C5(C)C)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C57H67ClN6O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-0MS4XR	WO2019023553A1_631	.	CC1=NC=CN1C1=CC=C([C@@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](C(C)C)N2C=C(C3=CC=C(OC4CCN(C5=NC=C(N6C(=S)N(C7=CC=C(C#N)C(C(F)(F)F)=C7)C(=O)C6(C)C)C=C5)CC4)N=C3)C=N2)C=C1	C53H55F3N12O5S	AR	P10275	VHL	WO-2019023553-A1
TPD-4WZPJ2	WO2019023553A1_632	.	C#CCCC(=O)OC(CCOCCCOCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=C(C)N=CS2)C=C1)C(C)(C)C)CCOC1=CC=C(N2C(=S)N(C3=CC=C(C#N)C(C(F)(F)F)=C3)C(=O)C2(C)C)C=C1	C57H66F3N7O10S2	AR	P10275	VHL	WO-2019023553-A1
TPD-5U6R39	SCHEMBL19580956	(2S,4R)-1-[(2S)-2-[[2-[3-[5-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]pentoxy]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[3-(4-methyl-1,3-oxazol-5-yl)-1-bicyclo[1.1.1]pentanyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL31591739	CC1=C(C23CC(CNC(=O)[C@@H]4C[C@@H](O)CN4C(=O)[C@@H](NC(=O)COCCCOCCCCCOC4=CC=C(N5C(=S)N(C6=CC=C(C#N)C(C(F)(F)F)=C6)C(=O)C5(C)C)C=C4)C(C)(C)C)(C2)C3)OC=N1	C50H62F3N7O9S	AR	P10275	VHL	WO-2019023553-A1
TPD-2RUVG1	SCHEMBL19598652	(2S,4R)-1-[(2S)-2-[[2-[(2R)-1-[4-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenyl]piperazin-1-yl]propan-2-yl]oxyacetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL21712896; SCHEMBL29817386	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CO[C@H](C)CN3CCN(C4=CC=C(C(=O)NC5C(C)(C)C(OC6=CC(Cl)=C(C#N)C=C6)C5(C)C)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C54H69ClN8O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-L385XI	WO2019023553A1_635	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCOCCCCCOC3=CC=C(C(=O)NC4C(C)(C)C(OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C55H71ClN6O9S	AR	P10275	VHL	WO-2019023553-A1
TPD-3FJMRY	WO2019023553A1_636	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCN3CC4CC3CN4C3=CC=C(C(=O)NC4C(C)(C)C(OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=N3)C(C)(C)C)C=C2)SC=N1	C53H66ClN9O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-NOGXV7	SCHEMBL19598656	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[2-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]ethyl]piperazin-1-yl]pyridine-3-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCN3CCN(C4=CC=C(C(=O)NC5C(C)(C)C(OC6=CC=C(C#N)C(Cl)=C6)C5(C)C)C=N4)CC3)C(C)(C)C)C=C2)SC=N1	C51H64ClN9O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-SFP8DJ	SCHEMBL19598657	(2S,4R)-1-[(2S)-2-[[2-[(2S)-1-[4-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenyl]piperazin-1-yl]propan-2-yl]oxyacetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL31591755	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CO[C@@H](C)CN3CCN(C4=CC=C(C(=O)NC5C(C)(C)C(OC6=CC(Cl)=C(C#N)C=C6)C5(C)C)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C54H69ClN8O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-XREP05	SCHEMBL19580828	(2S,4R)-1-[(2S)-2-[[2-[4-[2-[4-[[3-[4-cyano-3-(trifluoromethyl)phenoxy]-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenoxy]ethoxy]piperidin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL29817307	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCC(OCCOC4=CC=C(C(=O)NC5C(C)(C)C(OC6=CC=C(C#N)C(C(F)(F)F)=C6)C5(C)C)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C54H66F3N7O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-87T0KV	SCHEMBL19581348	(2S,4R)-1-[2-[[2-[4-[4-[[3-[4-cyano-3-(trifluoromethyl)phenoxy]-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenoxy]butoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(NC(=O)COCCCCOC3=CC=C(C(=O)NC4C(C)(C)C(OC5=CC(C(F)(F)F)=C(C#N)C=C5)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C52H63F3N6O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-SYL4EE	WO2019023553A1_642	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)OCCC3(CCOC4=CC=C(C(=O)NC5C(C)(C)C(OC6=CC=C(C#N)C(Cl)=C6)C5(C)C)C=C4)COC3)C(C)(C)C)C=C2)SC=N1	C53H65ClN6O9S	AR	P10275	VHL	WO-2019023553-A1
TPD-PH149A	WO2019023553A1_643	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCOCCN(CCOC4=CC=C(N5C(=S)N(C6=CC=C(C#N)C(C(F)(F)F)=C6)C(=O)C5(C)C)C=C4)CCOCC3)C(C)(C)C)C=C2)SC=N1	C54H66F3N9O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-VM6XOY	WO2019023553A1_644	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CC3=CC=NC(N4CCN(C5=NC=C(C(=O)NC6C(C)(C)C(OC7=CC=C(C#N)C(Cl)=C7)C6(C)C)C=C5)CC4)=C3)C(C)(C)C)C=C2)SC=N1	C55H65ClN10O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-7QNUUW	SCHEMBL19581101	(2S,4R)-1-[(2S)-2-[[2-[4-[2-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenoxy]ethyl]piperazin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL29817356	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCN(CCOC4=CC=C(C(=O)NC5C(C)(C)C(OC6=CC=C(C#N)C(Cl)=C6)C5(C)C)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C52H65ClN8O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-PUFYTZ	SCHEMBL19580836	(2S,4R)-1-[(2S)-2-[[2-[4-[2-[4-[[3-[4-cyano-3-(trifluoromethyl)phenoxy]-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenoxy]ethyl]piperazin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL29817302; DLFRRZAVJQGGFO-CWKMZTRXSA-N; (2S,4R)-1-[(2S)-2-[[2-[4-[2-[4-[[3-[4-cyano-3-(trifluoromethyl)phenoxy]-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenoxy]ethyl]piperazin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCN(CCOC4=CC=C(C(=O)NC5C(C)(C)C(OC6=CC=C(C#N)C(C(F)(F)F)=C6)C5(C)C)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C53H65F3N8O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-IDQROL	WO2019023553A1_647	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C(OCCCOCCCN4C=NC(C5CCC(N6C(=S)N(C7=CC=C(C#N)C(C(F)(F)F)=C7)C(=O)C6(C)C)CC5)=C4)C=N3)C=C2)SC=N1	C53H63F3N10O6S2	AR	P10275	VHL	WO-2019023553-A1
TPD-O6YC4K	SCHEMBL19581085	(2S,4R)-1-[(2S)-2-[4-[3-[3-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]imidazol-1-yl]propoxy]propoxy]pyrazol-1-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL29817005; FEOQTHOQIVPDJV-GUNFGILISA-N; (2S,4R)-1-[(2S)-2-[4-[3-[3-[4-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]imidazol-1-yl]propoxy]propoxy]pyrazol-1-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C(OCCCOCCCN4C=NC(C5=CC=C(N6C(=S)N(C7=CC=C(C#N)C(C(F)(F)F)=C7)C(=O)C6(C)C)C=C5)=C4)C=N3)C=C2)SC=N1	C53H57F3N10O6S2	AR	P10275	VHL	WO-2019023553-A1
TPD-FUD6A9	SCHEMBL19598663	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[2-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]propyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]ethyl]piperazin-1-yl]pyridine-3-carboxamide; SCHEMBL31591765	CC[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](NC(=O)COCCN1CCN(C2=CC=C(C(=O)NC3C(C)(C)C(OC4=CC=C(C#N)C(Cl)=C4)C3(C)C)C=N2)CC1)C(C)(C)C)C1=CC=C(C2=C(C)N=CS2)C=C1	C53H68ClN9O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-CSB9VH	WO2019023553A1_650	.	CC1=C(C2=CC=C(C(C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=NC(CCCCOCCCCCOC4=CC=C(N5C(=S)N(C6=CC=C(C#N)C(C(F)(F)F)=C6)C(=O)C5(C)C)C=C4)=C3)C=C2)SC=N1	C53H61F3N8O6S2	AR	P10275	VHL	WO-2019023553-A1
TPD-GAFVFL	WO2019023553A1_651	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](OC(=O)[C@@H](N)CCCCN)CN3C(=O)[C@@H](NC(=O)COCCCOCCC(CCOC3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3)OC(=O)[C@@H](N)CCCCN)C(C)(C)C)C=C2)SC=N1	C64H86F3N11O11S2	AR	P10275	VHL	WO-2019023553-A1
TPD-Z6EY2C	SCHEMBL19581319	[(3R,5S)-1-[(2S)-2-[[2-[5-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]anilino]pentoxy]acetyl]amino]-3,3-dimethylbutanoyl]-5-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-3-yl] propan-2-yl carbonate; SCHEMBL29817176	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](OC(=O)OC(C)C)CN3C(=O)[C@@H](NC(=O)COCCCCCNC3=CC=C(C(=O)NC4C(C)(C)C(OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C56H72ClN7O9S	AR	P10275	VHL	WO-2019023553-A1
TPD-6REMJ9	SCHEMBL19581261	[(3R,5S)-1-[(2S)-2-[[2-[5-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]anilino]pentoxy]acetyl]amino]-3,3-dimethylbutanoyl]-5-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-3-yl]oxymethyl propan-2-yl carbonate; SCHEMBL29817179	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](OCOC(=O)OC(C)C)CN3C(=O)[C@@H](NC(=O)COCCCCCNC3=CC=C(C(=O)NC4C(C)(C)C(OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C57H74ClN7O10S	AR	P10275	VHL	WO-2019023553-A1
TPD-ZQJNLM	WO2019023553A1_654	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCN3CCN(C4=CC=C(C(=O)NC5C(C)(C)C(OC6=CC=C(C#N)C(Cl)=C6)C5(C)C)N=C4)CC3)C(C)(C)C)C=C2)SC=N1	C52H66ClN9O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-37JB4E	SCHEMBL19598662	(2S,4R)-1-[(2S)-2-[[(2S)-2-[4-[2-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenoxy]ethyl]piperazin-1-yl]-3-hydroxypropanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL29817381	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)[C@H](CO)N3CCN(CCOC4=CC=C(C(=O)N[C@H]5C(C)(C)[C@H](OC6=CC=C(C#N)C(Cl)=C6)C5(C)C)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C54H69ClN8O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-XW1QEV	WO2019023553A1_656	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCCNC3=CC=C(C(=O)NC4C(C)(C)C(OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3F)C(C)(C)C)C=C2)SC=N1	C52H65ClFN7O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-KFQ200	WO2019023553A1_657	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCCC3=CC=C(C(=O)NC4C(C)(C)C(OC5=CC(C(F)(F)F)=C(C#N)C=N5)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C52H64F3N7O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-3SEA4B	WO2019023553A1_658	.	CC1=C(C2=CC=C(C(C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3=CC(OCCN4CCN(C5=CC=C(C(=O)N[C@H]6C(C)(C)[C@H](OC7=CC=C(C#N)C(Cl)=C7)C6(C)C)C=N5)CC4)=NO3)C(C)C)C=C2)SC=N1	C52H62ClN9O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-KS75ZP	WO2019023553A1_659	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(OCCN4CCN(C5=CC=C(C(=O)N[C@H]6C(C)(C)[C@H](OC7=CC=C(C#N)C(Cl)=C7)C6(C)C)C=N5)CC4)=NO3)C(C)C)C=C2)SC=N1	C52H62ClN9O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-4FC4TS	SCHEMBL17947338	(2S,4R)-1-[(2S)-2-[[2-[2-[4-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenyl]piperazin-1-yl]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL19598600	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCN3CCN(C4=CC=C(C(=O)NC5C(C)(C)C(OC6=CC=C(C#N)C(Cl)=C6)C5(C)C)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C53H67ClN8O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-1OZCMH	WO2019023553A1_661	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCOCCCCCOC3=CC=C(N4C(=S)N(C5=CC(C(F)(F)F)=C(C#N)C=N5)C(=O)C4(C)C)C=C3)C3COC3)C=C2)SC=N1	C50H57F3N8O9S2	AR	P10275	VHL	WO-2019023553-A1
TPD-K9PAKE	SCHEMBL19581150	(2S,4R)-1-[(2S)-2-[[2-[3-[5-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]pentoxy]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-(4-imidazol-1-ylphenyl)ethyl]pyrrolidine-2-carboxamide; SCHEMBL29817186	C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](NC(=O)COCCCOCCCCCOC1=CC=C(N2C(=S)N(C3=CC=C(C#N)C(C(F)(F)F)=C3)C(=O)C2(C)C)C=C1)C(C)(C)C)C1=CC=C(N2C=CN=C2)C=C1	C51H61F3N8O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-X6GMY0	WO2019023553A1_663	.	CC1=CN(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCCCCOC3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3)C(C)(C)C)C=C2)C=N1	C51H61F3N8O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-XIO6OT	SCHEMBL19598666	(2S,4R)-1-[(2S)-2-[[(2S)-2-[2-[4-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenyl]piperazin-1-yl]ethoxy]propanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL29817468	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)[C@H](C)OCCN3CCN(C4=CC=C(C(=O)N[C@H]5C(C)(C)[C@H](OC6=CC(Cl)=C(C#N)C=C6)C5(C)C)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C54H69ClN8O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-563UWP	SCHEMBL19581405	(2S,4R)-1-[(2S)-2-[[2-[4-[3-[4-[[3-[4-cyano-3-(trifluoromethyl)phenoxy]-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenyl]propyl]piperazin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL19581408; MZUARNGNAWZKSJ-FEXCZLAUSA-N; (2S,4R)-1-[(2S)-2-[[2-[4-[3-[4-[[3-[4-cyano-3-(trifluoromethyl)phenoxy]-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenyl]propyl]piperazin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCN(CCCC4=CC=C(C(=O)N[C@H]5C(C)(C)[C@H](OC6=CC=C(C#N)C(C(F)(F)F)=C6)C5(C)C)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C55H69F3N8O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-KKRA2T	SCHEMBL19581434	(2S,4R)-1-[(2S)-2-[[2-[5-[[3-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]-1-bicyclo[1.1.1]pentanyl]amino]pentoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL19581436; SCHEMBL29817010	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCCNC34CC(C(=O)NC5C(C)(C)C(OC6=CC=C(C#N)C(Cl)=C6)C5(C)C)(C3)C4)C(C)(C)C)C=C2)SC=N1	C51H68ClN7O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-H4E0GX	WO2019023553A1_667	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCO[C@@H](CN4CCO[C@H](COC5=CC=C(N6C(=S)N(C7=CC=C(C#N)C(C(F)(F)F)=C7)C(=O)C6(C)C)C=C5)C4)C3)C(C)(C)C)C=C2)SC=N1	C54H64F3N9O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-PRV0MU	WO2019023553A1_668	.	C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](NC(=O)COCCN1CC2CC1CN2C1=NC=C(C(=O)NC2C(C)(C)C(OC3=CC(Cl)=C(C#N)C=C3)C2(C)C)C=C1)C(C)(C)C)C1=CC=C(C2=C(CO)N=CS2)C=C1	C53H66ClN9O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-N2YH6B	WO2019023553A1_669	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCN3CC4CC3CN4C3=NC=C(C(=O)NC4C(C)(C)C(OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C52H64ClN9O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-MB7E1T	SCHEMBL19581306	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-5-[5-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]pentylamino]pyridine-2-carboxamide; SCHEMBL19581309; SCHEMBL29817241	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCCNC3=CC=C(C(=O)NC4C(C)(C)C(OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)N=C3)C(C)C)C=C2)SC=N1	C50H63ClN8O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-9B7OKR	SCHEMBL19581132	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[2-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1R)-2-hydroxy-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]ethyl]piperazin-1-yl]pyridine-3-carboxamide; SCHEMBL29817463	CC1=C(C2=CC=C([C@H](CO)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCN3CCN(C4=CC=C(C(=O)NC5C(C)(C)C(OC6=CC=C(C#N)C(Cl)=C6)C5(C)C)C=N4)CC3)C(C)(C)C)C=C2)SC=N1	C52H66ClN9O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-E1N1S7	SCHEMBL19580871	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[9-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethyl]-3,9-diazaspiro[5.5]undecan-3-yl]pyridine-3-carboxamide; SCHEMBL21712832; SCHEMBL29817464	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCC4(CC3)CCN(C3=NC=C(C(=O)N[C@H]5C(C)(C)[C@@H](OC6=CC=C(C#N)C(Cl)=C6)C5(C)C)C=C3)CC4)C(C)(C)C)C=C2)SC=N1	C54H68ClN9O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-1YKNHP	SCHEMBL29817254	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[2-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-[4-(hydroxymethyl)-1,3-thiazol-5-yl]phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]ethyl]piperazin-1-yl]pyridine-3-carboxamide	C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](NC(=O)COCCN1CCN(C2=NC=C(C(=O)N[C@H]3C(C)(C)[C@H](OC4=CC=C(C#N)C(Cl)=C4)C3(C)C)C=C2)CC1)C(C)(C)C)C1=CC=C(C2=C(CO)N=CS2)C=C1	C52H66ClN9O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-SUWXOM	WO2019023553A1_674	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCN(CCC4(C5=CC=C(C(=O)NC6C(C)(C)C(OC7=CC=C(C#N)C(C(F)(F)F)=C7)C6(C)C)C=C5)COC4)CC3)C(C)(C)C)C=C2)SC=N1	C57H71F3N8O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-ZZ5Y51	WO2019023553A1_675	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCOC(CN4CCOC(COC5=CC=C(N6C(=S)N(C7=CC=C(C#N)C(C(F)(F)F)=C7)C(=O)C6(C)C)C=C5)C4)C3)C(C)(C)C)C=C2)SC=N1	C54H64F3N9O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-V0N747	WO2019023553A1_676	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(NC(=O)CN3CCO[C@@H](CN4CCOC(COC5=CC=C(N6C(=S)N(C7=CC=C(C#N)C(C(F)(F)F)=C7)C(=O)C6(C)C)C=C5)C4)C3)C(C)(C)C)C=C2)SC=N1	C54H64F3N9O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-55JSJX	WO2019023553A1_677	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)OCC3=CC=CC=C3)[C@@H](C)OCCCCCCOC3=CC=C(N4C(=S)N(C5=CC(C(F)(F)F)=C(C#N)C=C5)C(=O)C4(C)C)C=C3)C=C2)SC=N1	C54H58F3N7O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-RR36FH	SCHEMBL19598672	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-5-[3-[2-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]ethyl-methylamino]propyl]pyridine-2-carboxamide; SCHEMBL29817458	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCN(C)CCCC3=CN=C(C(=O)NC4C(C)(C)C(OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C52H67ClN8O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-HPVBHG	SCHEMBL19598673	(2S,4R)-1-[(2S)-2-[[2-[4-[2-[4-[[3-[4-cyano-3-(trifluoromethyl)phenoxy]-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenoxy]ethyl]piperazin-1-yl]-2-oxoacetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL29817047	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C(=O)N3CCN(CCOC4=CC=C(C(=O)NC5C(C)(C)C(OC6=CC=C(C#N)C(C(F)(F)F)=C6)C5(C)C)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C54H65F3N8O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-F7T33C	SCHEMBL19598674	N-[3-(4-cyano-3-methylphenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[2-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]ethyl]piperazin-1-yl]pyridine-3-carboxamide; SCHEMBL29817479	CC1=C(C#N)C=CC(OC2C(C)(C)C(NC(=O)C3=CN=C(N4CCN(CCOCC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=C(C)N=CS6)C=C5)C(C)(C)C)CC4)C=C3)C2(C)C)=C1	C53H69N9O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-OUDBRC	WO2019023553A1_681	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCN3CCN(C4=NC=C(C(=O)NC5C(C)(C)C(OC6=CC(C#N)=C(C#N)C=C6)C5(C)C)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C53H66N10O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-8VCN8K	WO2019023553A1_682	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCN3CCN(C4=NC=C(C(=O)NC5C(C)(C)C(OC6=NC(N)=C(C#N)C=N6)C5(C)C)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C50H66N12O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-WNT88M	SCHEMBL19598679	(2S,4R)-1-[(2S)-2-[[2-[4-[2-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenoxy]ethyl]piperazin-1-yl]acetyl]-methylamino]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL31591750	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N(C)C(=O)CN3CCN(CCOC4=CC=C(C(=O)N[C@H]5C(C)(C)[C@H](OC6=CC=C(C#N)C(Cl)=C6)C5(C)C)C=C4)CC3)C=C2)SC=N1	C53H67ClN8O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-84YIUD	SCHEMBL19598677	N-[3-[4-cyano-3-(trifluoromethyl)phenoxy]-2,2,4,4-tetramethylcyclobutyl]-6-[4-[2-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]ethyl]piperazin-1-yl]pyridazine-3-carboxamide; SCHEMBL29817491; GNVPIELZHKQKFU-MVNXDDALSA-N; N-[3-[4-cyano-3-(trifluoromethyl)phenoxy]-2,2,4,4-tetramethylcyclobutyl]-6-[4-[2-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]ethyl]piperazin-1-yl]pyridazine-3-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCN3CCN(C4=NN=C(C(=O)N[C@H]5C(C)(C)[C@H](OC6=CC(C(F)(F)F)=C(C#N)C=C6)C5(C)C)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C52H65F3N10O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-9XZ7DG	SCHEMBL19581361	(2S,4R)-1-[(2S)-2-[[2-[5-[3-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenyl]oxetan-3-yl]pentoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL19581363; SCHEMBL29817045	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCCC3(C4=CC=C(C(=O)NC5C(C)(C)C(OC6=CC=C(C#N)C(Cl)=C6)C5(C)C)C=C4)COC3)C(C)(C)C)C=C2)SC=N1	C55H69ClN6O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-D5DJF2	WO2019023553A1_686	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCN(CC4(CNC5=CC=C(C(=O)N[C@H]6C(C)(C)[C@H](OC7=CC=C(C#N)C(C(F)(F)F)=C7)C6(C)C)C=C5)COC4)CC3)C(C)(C)C)C=C2)SC=N1	C57H72F3N9O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-I0IH9I	WO2019023553A1_687	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCC(CCCC3=CC=C(C(=O)NC4C(C)(C)C(OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)N=C3)N3CCN(C)CC3)C(C)(C)C)C=C2)SC=N1	C58H78ClN9O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-XQ4GPP	WO2019023553A1_688	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCC(F)(F)C(F)(F)C(F)(F)COC3=CC=C(C(=O)NC4C(C)(C)C(OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C52H59ClF6N6O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-DDD1P3	WO2019023553A1_689	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCN3CCN(C4=NC=C(C(=O)NC5C(C)(C)C(OC6=CC=C(C#N)C(C(F)(F)F)=C6)C5(C)C)N=C4)CC3)C(C)(C)C)C=C2)SC=N1	C52H65F3N10O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-GJFWPX	SCHEMBL19581278	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[[3-[1-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethyl]piperidin-4-yl]oxycyclobutyl]amino]pyridine-3-carboxamide; SCHEMBL19581280; SCHEMBL29817033	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCC(O[C@H]4C[C@@H](NC5=CC=C(C(=O)N[C@H]6C(C)(C)[C@H](OC7=CC=C(C#N)C(Cl)=C7)C6(C)C)C=N5)C4)CC3)C(C)(C)C)C=C2)SC=N1	C55H70ClN9O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-SVCVP6	SCHEMBL19581264	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-5-[5-[2-[(2R)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]-3-methylimidazol-4-yl]pentylamino]pyridine-2-carboxamide; SCHEMBL19581267; SCHEMBL29817174	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=NC=C(CCCCCNC4=CC=C(C(=O)N[C@H]5C(C)(C)[C@H](OC6=CC=C(C#N)C(Cl)=C6)C5(C)C)N=C4)N3C)C(C)C)C=C2)SC=N1	C52H64ClN9O5S	AR	P10275	VHL	WO-2019023553-A1
TPD-R5MK50	WO2019023553A1_693	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCC/C(CCCC3=CC=C(C(=O)N[C@H]4C(C)(C)[C@@H](OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)N=C3)=N\O)C(C)(C)C)C=C2)SC=N1	C53H67ClN8O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-SLD7UX	SCHEMBL19581337	(2S,4R)-1-[2-[[2-[16-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenyl]-1,4,10,13-tetraoxa-7,16-diazacyclooctadec-7-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL19598682	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(NC(=O)CN3CCOCCOCCN(C4=CC=C(C(=O)NC5C(C)(C)C(OC6=CC=C(C#N)C(Cl)=C6)C5(C)C)C=C4)CCOCCOCC3)C(C)(C)C)C=C2)SC=N1	C59H79ClN8O10S	AR	P10275	VHL	WO-2019023553-A1
TPD-7RKOYK	WO2019023553A1_695	.	CCO/N=C(/CCCCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=C(C)N=CS2)C=C1)C(C)(C)C)CCCC1=CC=C(C(=O)N[C@H]2C(C)(C)[C@@H](OC3=CC=C(C#N)C(Cl)=C3)C2(C)C)N=C1	C55H71ClN8O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-P9N44N	WO2019023553A1_696	.	CC(C)[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C#N)C=C1)C1=CC(OCCN2CCN(C3=CC=C(C(=O)N[C@H]4C(C)(C)[C@@H](OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=N3)CC2)=NO1	C49H58ClN9O7	AR	P10275	VHL	WO-2019023553-A1
TPD-EC6V2Z	WO2019023553A1_697	.	CC(C)[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C#N)C=C1)C1=CC(OCCN2CCN(C3=CC=C(C(=O)NC4C(C)(C)C(OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=N3)CC2)=NO1	C49H58ClN9O7	AR	P10275	VHL	WO-2019023553-A1
TPD-NIDDXM	SCHEMBL19581223	N-[(2S)-1-[3-(3-chloro-4-cyanophenyl)pyrazol-1-yl]propan-2-yl]-5-[3-[4-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethyl]piperazin-1-yl]propoxymethyl]-1H-pyrazole-3-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCN(CCCOCC4=CC(C(=O)N[C@@H](C)CN5C=CC(C6=CC(Cl)=C(C#N)C=C6)=N5)=NN4)CC3)C(C)(C)C)C=C2)SC=N1	C50H63ClN12O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-1YMBM6	SCHEMBL19581328	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-5-[3-[2-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]ethyl-(3,3,3-trifluoropropyl)amino]propyl]pyridine-2-carboxamide; SCHEMBL19581330; SCHEMBL29817495	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCN(CCCC3=CN=C(C(=O)NC4C(C)(C)C(OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)CCC(F)(F)F)C(C)(C)C)C=C2)SC=N1	C54H68ClF3N8O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-PMGP6I	SCHEMBL19581275	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[2-[2-[[3,3-dimethyl-1-[(2S)-2-(methylcarbamoyl)pyrrolidin-1-yl]-1-oxobutan-2-yl]amino]-2-oxoethoxy]ethyl]piperazin-1-yl]pyridine-3-carboxamide	CNC(=O)[C@@H]1CCCN1C(=O)C(NC(=O)COCCN1CCN(C2=NC=C(C(=O)N[C@H]3C(C)(C)[C@@H](OC4=CC(Cl)=C(C#N)C=C4)C3(C)C)C=C2)CC1)C(C)(C)C	C41H57ClN8O6	AR	P10275	VHL	WO-2019023553-A1
TPD-N5I1IZ	WO2019023553A1_701	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=NC=C(CCCN4CCN(C5=NC=C(C(=O)NC6C(C)(C)C(OC7=CC=C(C#N)C(Cl)=C7)C6(C)C)C=C5)CC4)N3C)C(C)C)C=C2)SC=N1	C54H67ClN10O5S	AR	P10275	VHL	WO-2019023553-A1
TPD-R9S5X4	WO2019023553A1_702	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=NC=C(CCCN4CCN(C5=NC=C(C(=O)NC6C(C)(C)C(OC7=CC=C(C#N)C(Cl)=C7)C6(C)C)C=C5)CC4)N3C)C(C)O)C=C2)SC=N1	C53H65ClN10O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-YFETI4	SCHEMBL19580656	N-[3-[4-cyano-3-(trifluoromethyl)phenoxy]-2,2,4,4-tetramethylcyclobutyl]-5-[4-[2-[2-[[1-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]ethyl]-2-oxopiperazin-1-yl]pyridine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(NC(=O)COCCN3CCN(C4=CC=C(C(=O)NC5C(C)(C)C(OC6=CC=C(C#N)C(C(F)(F)F)=C6)C5(C)C)N=C4)C(=O)C3)C(C)(C)C)C=C2)SC=N1	C52H62F3N9O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-SPEP7J	WO2019023553A1_704	.	CC1=C(C2=CC=C(C(NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(NC(=O)COCCN3CCN(C4=CC=C(C(=O)NC5C(C)(C)C(OC6=CC=C(C#N)C(C(F)(F)F)=C6)C5(C)C)C=N4)CC3)C(C)(C)C)C3COC3)C=C2)SC=N1	C55H68F3N9O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-75P0IW	SCHEMBL19581302	N-[3-[4-cyano-3-(trifluoromethyl)phenoxy]-2,2,4,4-tetramethylcyclobutyl]-6-[4-[2-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(S)-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]-(oxetan-3-yl)methyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]ethyl]piperazin-1-yl]pyridine-3-carboxamide; SCHEMBL19581305	CC1=C(C2=CC=C([C@@H](NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCN3CCN(C4=CC=C(C(=O)NC5C(C)(C)C(OC6=CC=C(C#N)C(C(F)(F)F)=C6)C5(C)C)C=N4)CC3)C(C)(C)C)C3COC3)C=C2)SC=N1	C55H68F3N9O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-0JSPQV	SCHEMBL19600650	(2S,4R)-1-[(2S)-2-[[2-[4-[3-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]-2-fluoroanilino]cyclobutyl]oxypiperidin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL29817099	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCC(O[C@H]4C[C@@H](NC5=CC=C(C(=O)N[C@H]6C(C)(C)[C@H](OC7=CC=C(C#N)C(Cl)=C7)C6(C)C)C=C5F)C4)CC3)C(C)(C)C)C=C2)SC=N1	C56H70ClFN8O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-SQHKB1	SCHEMBL19581321	N-[3-[4-cyano-3-(trifluoromethyl)phenoxy]-2,2,4,4-tetramethylcyclobutyl]-6-[4-[3-[4-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethyl]piperazin-1-yl]propyl]piperazin-1-yl]pyridine-3-carboxamide; SCHEMBL19581323; ITLFIHBSUKRJKS-HDRHANLDSA-N; N-[3-[4-cyano-3-(trifluoromethyl)phenoxy]-2,2,4,4-tetramethylcyclobutyl]-6-[4-[3-[4-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethyl]piperazin-1-yl]propyl]piperazin-1-yl]pyridine-3-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCN(CCCN4CCN(C5=NC=C(C(=O)NC6C(C)(C)C(OC7=CC(C(F)(F)F)=C(C#N)C=C7)C6(C)C)C=C5)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C58H76F3N11O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-EM17WY	WO2019023553A1_708	.	CO[C@@H]1C[C@@H](C(=O)N[C@H](C)C2=CC=C(C3=C(C)N=CS3)C=C2)N(C(=O)[C@@H](NC(=O)CN2CCN(CCCC3=CC=C(C(=O)NC4C(C)(C)C(OC5=CC=C(C#N)C(C(F)(F)F)=C5)C4(C)C)C=C3)CC2)C(C)(C)C)C1	C56H71F3N8O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-EBWG5W	WO2019023553A1_709	.	CO[C@@H]1C[C@H](C(=O)N(C)CC2=CC=C(C3=C(C)N=CS3)C=C2)N(C(=O)[C@@H](N(C)C(=O)COCCCCCN(C)C2=CC=C(C(=O)N(C)[C@H]3C(C)(C)[C@H](OC4=CC=C(C#N)C(C(F)(F)F)=C4)C3(C)C)N=C2)C(C)(C)C)C1	C56H73F3N8O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-90DLJP	SCHEMBL19581097	(2S,4R)-1-[(2S)-2-[[2-[4-[3-[1-[4-[[3-[4-cyano-3-(trifluoromethyl)phenoxy]-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenyl]triazol-4-yl]propyl]piperazin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL29817237; SPDSJPPJMPDWBH-IQZKAYMSSA-N; (2S,4R)-1-[(2S)-2-[[2-[4-[3-[1-[4-[[3-[4-cyano-3-(trifluoromethyl)phenoxy]-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenyl]triazol-4-yl]propyl]piperazin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCN(CCCC4=CN(C5=CC=C(C(=O)NC6C(C)(C)C(OC7=CC=C(C#N)C(C(F)(F)F)=C7)C6(C)C)C=C5)N=N4)CC3)C(C)(C)C)C=C2)SC=N1	C56H68F3N11O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-E79KPH	SCHEMBL19580807	N-[3-[4-cyano-3-(trifluoromethyl)phenoxy]-2,2,4,4-tetramethylcyclobutyl]-6-[4-[2-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]ethyl]-2-oxopiperazin-1-yl]pyridine-3-carboxamide; SCHEMBL29817374; DUQDAWMOFLSPEF-FFAFJLKHSA-N; N-[3-[4-cyano-3-(trifluoromethyl)phenoxy]-2,2,4,4-tetramethylcyclobutyl]-6-[4-[2-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]ethyl]-2-oxopiperazin-1-yl]pyridine-3-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCN3CCN(C4=CC=C(C(=O)NC5C(C)(C)C(OC6=CC=C(C#N)C(C(F)(F)F)=C6)C5(C)C)C=N4)C(=O)C3)C(C)(C)C)C=C2)SC=N1	C52H62F3N9O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-CVM8QW	SCHEMBL19580952	(2S,4R)-1-[(2S)-2-[[2-[4-[3-[4-[[3-[4-cyano-3-(trifluoromethyl)phenoxy]-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenyl]propyl]piperazin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(R)-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]-(oxetan-3-yl)methyl]pyrrolidine-2-carboxamide; SCHEMBL21713118	CC1=C(C2=CC=C([C@H](NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCN(CCCC4=CC=C(C(=O)N[C@H]5C(C)(C)[C@@H](OC6=CC=C(C#N)C(C(F)(F)F)=C6)C5(C)C)C=C4)CC3)C(C)(C)C)C3COC3)C=C2)SC=N1	C57H71F3N8O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-V8AX76	WO2019023553A1_713	.	CC1=C(C2=CC=C([C@@H](NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCN(CCCC4=CC=C(C(=O)N[C@H]5C(C)(C)[C@@H](OC6=CC=C(C#N)C(C(F)(F)F)=C6)C5(C)C)C=C4)CC3)C(C)(C)C)C3COC3)C=C2)SC=N1	C57H71F3N8O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-DHSFYR	WO2019023553A1_714	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCN(C)C(=O)[C@@H](NC(=O)[C@H](C(C)C)N(C)CCOC3=CC=C(N4C(=S)N(C5=CC=C(C#N)C(C(F)(F)F)=C5)C(=O)C4(C)C)C=C3)C(C)C)C(C)(C)C)C=C2)SC=N1	C60H77F3N10O8S2	AR	P10275	VHL	WO-2019023553-A1
TPD-6CSZBL	SCHEMBL19581109	N-[3-(3,4-dicyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[3-[4-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethyl]piperazin-1-yl]propyl]piperazin-1-yl]pyridine-3-carboxamide; SCHEMBL19581114; SCHEMBL29817107	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCN(CCCN4CCN(C5=NC=C(C(=O)NC6C(C)(C)C(OC7=CC(C#N)=C(C#N)C=C7)C6(C)C)C=C5)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C58H76N12O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-TWZVOB	SCHEMBL19581192	N-[3-(5-cyano-6-methylpyridin-2-yl)oxy-2,2,4,4-tetramethylcyclobutyl]-6-[4-[3-[4-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethyl]piperazin-1-yl]propyl]piperazin-1-yl]pyridine-3-carboxamide; SCHEMBL19581199	CC1=C(C#N)C=CC(O[C@H]2C(C)(C)[C@@H](NC(=O)C3=CN=C(N4CCN(CCCN5CCN(CC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)(C)C)CC5)CC4)C=C3)C2(C)C)=N1	C57H78N12O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-NGXZ8P	SCHEMBL19581203	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[3-[4-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethyl]piperazin-1-yl]propyl]piperazin-1-yl]pyridine-3-carboxamide; SCHEMBL19581210; SCHEMBL29817042	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCN(CCCN4CCN(C5=NC=C(C(=O)NC6C(C)(C)C(OC7=CC(Cl)=C(C#N)C=C7)C6(C)C)C=C5)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C57H76ClN11O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-0T9EQL	WO2019023553A1_718	.	CO[C@@H]1C[C@H](C(=O)N(C)CC2=CC=C(C3=C(C)N=CS3)C=C2)N(C(=O)[C@@H](N(C)C(=O)COCCCCCN(C)C2=CC=C(C(=O)NC3C(C)(C)C(OC4=CC=C(C#N)C(C(F)(F)F)=C4)C3(C)C)N=C2)C(C)(C)C)C1	C55H71F3N8O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-JZJ7S7	SCHEMBL19581445	(2S,4R)-1-[2-[[2-[2-[1-[4-[[3-[4-cyano-3-(trifluoromethyl)phenoxy]-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenyl]triazol-4-yl]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(NC(=O)COCCC3=CN(C4=CC=C(C(=O)NC5C(C)(C)C(OC6=CC=C(C#N)C(C(F)(F)F)=C6)C5(C)C)C=C4)N=N3)C(C)(C)C)C=C2)SC=N1	C52H60F3N9O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-VAG4R6	WO2019023553A1_720	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](F)CN3C(=O)[C@@H](NC(=O)COCCN3CCN(C4=NC=C(C(=O)NC5C(C)(C)C(OC6=CC(Cl)=C(C#N)C=C6)C5(C)C)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C52H65ClFN9O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-NIOCU4	WO2019023553A1_722	.	CC(C)C[C@H](OCCN1CCN(C2=CC=C(C(=O)N[C@H]3C(C)(C)[C@H](OC4=CC=C(C#N)C(Cl)=C4)C3(C)C)C=N2)CC1)C(=O)N[C@@H](C)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(Cl)C=C1	C48H62Cl2N8O7	AR	P10275	VHL	WO-2019023553-A1
TPD-SKTYLJ	SCHEMBL19581397	(2S,4R)-1-[(2S)-2-[[2-[4-[4-[4-[[3-[4-cyano-3-(trifluoromethyl)phenoxy]-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenyl]butyl]piperazin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL19581401	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCN(CCCCC4=CC=C(C(=O)NC5C(C)(C)C(OC6=CC(C(F)(F)F)=C(C#N)C=C6)C5(C)C)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C56H71F3N8O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-IIK4BP	WO2019023553A1_724	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3CCCN3C(=O)[C@@H](NC(=O)CN3CCN(CCCC4=CC=C(C(=O)N[C@H]5C(C)(C)[C@@H](OC6=CC=C(C#N)C(C(F)(F)F)=C6)C5(C)C)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C55H69F3N8O5S	AR	P10275	VHL	WO-2019023553-A1
TPD-4OX28R	WO2019023553A1_725	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3CC(F)(F)CN3C(=O)[C@@H](NC(=O)COCCN3CCN(C4=NC=C(C(=O)NC5C(C)(C)C(OC6=CC=C(C#N)C(Cl)=C6)C5(C)C)C=C4)CC3)C(C)(C)C)C=C2)OC=N1	C52H64ClF2N9O7	AR	P10275	VHL	WO-2019023553-A1
TPD-5GJ6X0	SCHEMBL19580914	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[2-[(2S)-1-[[(2S)-1-[(2S,4R)-2-[(4-chlorophenyl)methylcarbamoyl]-4-hydroxypyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]oxyethyl]piperazin-1-yl]pyridine-3-carboxamide; SCHEMBL19580919; SCHEMBL29817098	CC(C)C[C@H](OCCN1CCN(C2=CC=C(C(=O)N[C@H]3C(C)(C)[C@@H](OC4=CC=C(C#N)C(Cl)=C4)C3(C)C)C=N2)CC1)C(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(Cl)C=C1)C(C)C	C50H66Cl2N8O7	AR	P10275	VHL	WO-2019023553-A1
TPD-EYRX53	WO2019023553A1_727	.	CC(C)C[C@H](OCCN1CCN(C2=CC=C(C(=O)N[C@H]3C(C)(C)[C@H](OC4=CC=C(C#N)C(Cl)=C4)C3(C)C)C=N2)CC1)C(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(Cl)C=C1)C(C)(C)C	C51H68Cl2N8O7	AR	P10275	VHL	WO-2019023553-A1
TPD-OKR1GF	SCHEMBL19581134	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[4-[[(2S)-1-[[(2S)-1-[(2S,4R)-2-[(4-chlorophenyl)methylcarbamoyl]-4-hydroxypyrrolidin-1-yl]-1-oxopropan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-4-oxobutyl]piperazin-1-yl]pyridine-3-carboxamide; SCHEMBL19581137; SCHEMBL29816973	CC(C)C[C@H](NC(=O)CCCN1CCN(C2=CC=C(C(=O)N[C@H]3C(C)(C)[C@@H](OC4=CC=C(C#N)C(Cl)=C4)C3(C)C)C=N2)CC1)C(=O)N[C@@H](C)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(Cl)C=C1	C50H65Cl2N9O7	AR	P10275	VHL	WO-2019023553-A1
TPD-NAUIMS	WO2019023553A1_729	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(NC(=O)OC(C)(C)C)[C@@H](C)OCCCN(C)CCC3=CC=C(C(=O)N[C@H]4C(C)(C)[C@@H](OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C=C2)SC=N1	C54H70ClN7O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-5A9MQ7	SCHEMBL19600908	(2S,4R)-1-[(2S,3R)-2-amino-3-[3-[2-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenyl]ethyl-methylamino]propoxy]butanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL29817049	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N)[C@@H](C)OCCCN(C)CCC3=CC=C(C(=O)N[C@H]4C(C)(C)[C@@H](OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C=C2)SC=N1	C49H62ClN7O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-U466YH	WO2019023553A1_731	.	CC(C)[C@H](NC(=O)[C@H](C)NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@H](C)NCC1=CC=C(Cl)C=C1)C(=O)OCCN1CCN(C2=CC=C(C(=O)NC3C(C)(C)C(OC4=CC=C(C#N)C(Cl)=C4)C3(C)C)C=N2)CC1	C50H65Cl2N9O8	AR	P10275	VHL	WO-2019023553-A1
TPD-U4IVPQ	WO2019023553A1_732	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C(OCCN3CCN(C4=CC=C(C(=O)NC5C(C)(C)C(OC6=CC=C(C#N)C(Cl)=C6)C5(C)C)C=N4)CC3)=C2)SC=N1	C56H64ClN9O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-8O2KLG	WO2019023553A1_733	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C([C@H](C)O)N3CC4=C(C=CC=C4)C3=O)C(OCCN3CCN(C4=CC=C(C(=O)NC5C(C)(C)C(OC6=CC=C(C#N)C(C(F)(F)F)=C6)C5(C)C)C=N4)CC3)=C2)SC=N1	C56H62F3N9O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-9YBGYT	SCHEMBL19600900	(2S,4R)-1-[(2S,3R)-2-acetamido-3-[3-[2-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenyl]ethyl-methylamino]propoxy]butanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL29817022	CC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=C(C)N=CS2)C=C1)[C@@H](C)OCCCN(C)CCC1=CC=C(C(=O)NC2C(C)(C)C(OC3=CC=C(C#N)C(Cl)=C3)C2(C)C)C=C1	C51H64ClN7O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-ZMVX41	WO2019023553A1_735	.	CC1=NOC(C(C(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(Cl)C=C2OCCOCCOCCOC2=CC=C(N3C(=S)N(C4=CC=C(C#N)C(C(F)(F)F)=C4)C(=O)C3(C)C)C=C2)C(C)C)=C1	C46H50ClF3N6O9S	AR	P10275	VHL	WO-2019023553-A1
TPD-QWJGTK	SCHEMBL19581096	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[2-[2-[[(2S)-1-[(2S,4R)-2-[(4-cyanophenyl)methylcarbamoyl]-4-hydroxypyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]ethyl]piperazin-1-yl]pyridine-3-carboxamide; SCHEMBL19581100; SCHEMBL29817169	CC1(C)C(NC(=O)C2=CN=C(N3CCN(CCOCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)NCC4=CC=C(C#N)C=C4)C(C)(C)C)CC3)C=C2)C(C)(C)C1OC1=CC(Cl)=C(C#N)C=C1	C48H60ClN9O7	AR	P10275	VHL	WO-2019023553-A1
TPD-TW6SRZ	WO2019023553A1_737	.	CC(C)(C)[C@H](NC(=O)COCCN1CCN(C2=NC=C(C(=O)N[C@H]3C(C)(C)[C@H](OC4=CC(Cl)=C(C#N)C=C4)C3(C)C)C=C2)CC1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(Cl)C=C1	C47H60Cl2N8O7	AR	P10275	VHL	WO-2019023553-A1
TPD-0QTXB2	SCHEMBL19581146	(2S,4R)-1-[(2S)-2-[[(2S)-2-[4-[3-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenyl]propyl]piperazin-1-yl]-4-methylpentanoyl]amino]propanoyl]-N-[(1S)-1-(4-chlorophenyl)ethyl]-4-hydroxypyrrolidine-2-carboxamide; SCHEMBL29817596	CC(C)C[C@@H](C(=O)N[C@@H](C)C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(Cl)C=C1)N1CCN(CCCC2=CC=C(C(=O)N[C@H]3C(C)(C)[C@H](OC4=CC(Cl)=C(C#N)C=C4)C3(C)C)C=C2)CC1	C51H67Cl2N7O6	AR	P10275	VHL	WO-2019023553-A1
TPD-0K8P80	WO2019023553A1_739	.	C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](NC(=O)CN1CCN(CCCC2=CC=C(C(=O)NC3C(C)(C)C(OC4=CC=C(C#N)C(Cl)=C4)C3(C)C)C=C2)CC1)C(C)(C)C)C1=CC=C(Cl)C=C1	C50H65Cl2N7O6	AR	P10275	VHL	WO-2019023553-A1
TPD-2MH2SI	WO2019023553A1_740	.	C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)C(NC(=O)COCCCCCC1=CC=C(C(=O)NC2C(C)(C)C(OC3=CC(Cl)=C(C#N)C(Cl)=C3)C2(C)C)C=C1)C(C)(C)C)C1=CC=C(Cl)C=C1	C48H60Cl3N5O7	AR	P10275	VHL	WO-2019023553-A1
TPD-GFUTG9	SCHEMBL19581393	(2S,4R)-1-[(2S)-2-[[2-[4-[[3-[[4-[[3-[4-cyano-3-(trifluoromethyl)phenoxy]-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenyl]methyl]oxetan-3-yl]methyl]piperazin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL19581396	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCN(CC4(CC5=CC=C(C(=O)N[C@H]6C(C)(C)[C@H](OC7=CC=C(C#N)C(C(F)(F)F)=C7)C6(C)C)C=C5)COC4)CC3)C(C)(C)C)C=C2)SC=N1	C57H71F3N8O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-MEG385	SCHEMBL19581008	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[2-[(2S)-1-[[(2S)-1-[(2S,4R)-2-[(4-chlorophenyl)methylcarbamoyl]-4-hydroxypyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]oxyethyl]piperazin-1-yl]pyridine-3-carboxamide; SCHEMBL21712862; SCHEMBL31591754	CC(C)[C@H](OCCN1CCN(C2=CC=C(C(=O)NC3C(C)(C)C(OC4=CC=C(C#N)C(Cl)=C4)C3(C)C)C=N2)CC1)C(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(Cl)C=C1)C(C)(C)C	C50H66Cl2N8O7	AR	P10275	VHL	WO-2019023553-A1
TPD-JMEW2R	WO2019023553A1_743	.	CC(C)[C@@H](C(=O)N1C[C@@H](O)C[C@H]1C(=O)NCC1=CC=C(Cl)C=C1OCCN1CCN(C2=CC=C(C(=O)NC3C(C)(C)C(OC4=CC=C(C#N)C(Cl)=C4)C3(C)C)C=N2)CC1)N1CC2=C(C=CC=C2)C1=O	C52H60Cl2N8O7	AR	P10275	VHL	WO-2019023553-A1
TPD-TQVA57	WO2019023553A1_744	.	CC1=C(C2=CC=C([C@H](C)NC(=O)C3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCN(CCC4(C5=CC=C(C(=O)NC6C(C)(C)C(OC7=CC=C(C#N)C(Cl)=C7)C6(C)C)C=C5)COC4)CC3)C(C)(C)C)C=C2)SC=N1	C56H71ClN8O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-FTOY0H	WO2019023553A1_745	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](NC(=O)CN3CCN(CCCC4=CC=C(C(=O)N[C@H]5C(C)(C)[C@@H](OC6=CC=C(C#N)C(C#N)=C6)C5(C)C)C=C4)CC3)C3COC3)C=C2)SC=N1	C54H65N9O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-I1N4W8	SCHEMBL19581340	(2S,4R)-1-[(2S)-2-[[2-[4-[3-[4-[[3-(3,4-dicyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenyl]propyl]piperazin-1-yl]acetyl]amino]-2-(oxetan-3-yl)acetyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL19581342; SCHEMBL29817295	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCN(CCCC4=CC=C(C(=O)NC5C(C)(C)C(OC6=CC=C(C#N)C(C#N)=C6)C5(C)C)C=C4)CC3)C3COC3)C=C2)SC=N1	C54H65N9O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-ENGGX1	SCHEMBL19598692	(2S,4R)-1-[2-[4-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenyl]butanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(NC(=O)CCCC3=CC=C(C(=O)NC4C(C)(C)C(OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C49H59ClN6O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-OIQGGH	WO2019023553A1_748	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(NC(=O)CCCCCC3=CC=C(C(=O)NC4C(C)(C)C(OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C51H63ClN6O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-Q3W2UY	SCHEMBL21712855	(2S,4R)-1-[(2S)-2-[7-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenyl]heptanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL29817029	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCC3=CC=C(C(=O)NC4C(C)(C)C(OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C52H65ClN6O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-BEWWHB	WO2019023553A1_750	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](NC(=O)CN3CCN(CCCC4=CC=C(C(=O)NC5C(C)(C)C(OC6=CC=C(C#N)C(Cl)=C6)C5(C)C)C=C4)CC3)C3COC3)C=C2)SC=N1	C53H65ClN8O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-QUTGUO	WO2019023553A1_751	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCN(CCCC4=CC=C(C(=O)NC5C(C)(C)C(OC6=CC=C(C#N)C(Cl)=C6)C5(C)C)C=C4)CC3)C3COC3)C=C2)SC=N1	C53H65ClN8O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-EWX4QK	SCHEMBL19580680	(2S,4R)-N-[[2-[4-[3-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenyl]propyl]piperazin-1-yl]-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-4-hydroxy-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]pyrrolidine-2-carboxamide; SCHEMBL29817153	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C(N3CCN(CCCC4=CC=C(C(=O)N[C@H]5C(C)(C)[C@H](OC6=CC=C(C#N)C(Cl)=C6)C5(C)C)C=C4)CC3)=C2)SC=N1	C58H67ClN8O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-JNAV5R	WO2019023553A1_753	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C(N3CCN(CCCC4=CC=C(C(=O)NC5C(C)(C)C(OC6=CC=C(C#N)C(C(F)(F)F)=C6)C5(C)C)C=C4)CC3)=C2)SC=N1	C59H67F3N8O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-FZ98TW	SCHEMBL19580634	(2S,4R)-N-[[4-chloro-2-[4-[3-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenyl]propyl]piperazin-1-yl]phenyl]methyl]-4-hydroxy-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]pyrrolidine-2-carboxamide; SCHEMBL29816993	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(Cl)C=C1N1CCN(CCCC2=CC=C(C(=O)NC3C(C)(C)C(OC4=CC=C(C#N)C(Cl)=C4)C3(C)C)C=C2)CC1)N1CC2=C(C=CC=C2)C1=O	C54H63Cl2N7O6	AR	P10275	VHL	WO-2019023553-A1
TPD-53GJDJ	SCHEMBL19581458	(2S,4R)-1-[(2S)-2-[5-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenyl]pentanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL21712834; SCHEMBL29817603	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCC3=CC=C(C(=O)N[C@H]4C(C)(C)[C@H](OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C50H61ClN6O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-TNANKJ	SCHEMBL19581345	(2S,4R)-1-[(2S)-2-[9-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenyl]nonanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL29817044	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCCC3=CC=C(C(=O)NC4C(C)(C)C(OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C54H69ClN6O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-PXQ8P6	WO2019023553A1_757	.	CC1(C)C(NC(=O)C2=CN=C(N3CCN(CCOCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)NCC4=CC=C(C5CC5)C=C4)C(C)(C)C)CC3)N=C2)C(C)(C)C1OC1=CC(Cl)=C(C#N)C=N1	C48H63ClN10O7	AR	P10275	VHL	WO-2019023553-A1
TPD-8KN6SP	SCHEMBL19581292	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[2-[2-[[(2S)-1-[(2S,4R)-2-[(4-cyclobutylphenyl)methylcarbamoyl]-4-hydroxypyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]ethyl]piperazin-1-yl]pyridine-3-carboxamide; SCHEMBL19581294; SCHEMBL29817448	CC1(C)C(NC(=O)C2=CN=C(N3CCN(CCOCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)NCC4=CC=C(C5CCC5)C=C4)C(C)(C)C)CC3)C=C2)C(C)(C)C1OC1=CC(Cl)=C(C#N)C=C1	C51H67ClN8O7	AR	P10275	VHL	WO-2019023553-A1
TPD-NZZGW5	WO2019023553A1_759	.	CC1(C)C(NC(=O)C2=CN=C(N3CCN(CCOCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)NCC4=CC=C(C5CCCC5)C=C4)C(C)(C)C)CC3)C=C2)C(C)(C)C1OC1=CC(Cl)=C(C#N)C=N1	C51H68ClN9O7	AR	P10275	VHL	WO-2019023553-A1
TPD-BNDJCU	SCHEMBL19581286	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[2-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[4-(oxan-4-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]ethyl]piperazin-1-yl]pyridine-3-carboxamide; SCHEMBL19581288; SCHEMBL29817550	CC(C)(C)[C@H](NC(=O)COCCN1CCN(C2=NC=C(C(=O)N[C@H]3C(C)(C)[C@H](OC4=CC=C(C#N)C(Cl)=C4)C3(C)C)C=C2)CC1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2CCOCC2)C=C1	C52H69ClN8O8	AR	P10275	VHL	WO-2019023553-A1
TPD-ZCKEIQ	WO2019023553A1_761	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=C(N5CCN(CCCC6=CC=C(C(=O)NC7C(C)(C)C(OC8=CC=C(C#N)C(C(F)(F)F)=C8)C7(C)C)C=C6)CC5)C=C4)C3=O)C=C2)SC=N1	C59H67F3N8O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-OHNONC	SCHEMBL19581056	(2S,4R)-1-[(2S)-2-[8-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenyl]octanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL19598694	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC3=CC=C(C(=O)NC4C(C)(C)C(OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C53H67ClN6O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-EAQMRX	SCHEMBL19581370	(2S,4R)-1-[(2S)-2-[10-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenyl]decanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL19598693	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCCCC3=CC=C(C(=O)NC4C(C)(C)C(OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C55H71ClN6O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-G7K3FY	WO2019023553A1_765	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCN3CCN(C4=NC=C(C(=O)NC5CC(OC6=CC=C(C#N)C(Cl)=C6)C5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C48H58ClN9O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-RYXC7W	SCHEMBL19581325	N-[(2S)-1-[3-[4-cyano-3-(trifluoromethyl)phenyl]pyrazol-1-yl]propan-2-yl]-5-[3-[4-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethyl]piperazin-1-yl]propoxymethyl]-1H-pyrazole-3-carboxamide; JVFMBHANTZBNAE-HDFITRACSA-N; N-[(2S)-1-[3-[4-cyano-3-(trifluoromethyl)phenyl]pyrazol-1-yl]propan-2-yl]-5-[3-[4-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethyl]piperazin-1-yl]propoxymethyl]-1H-pyrazole-3-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCN(CCCOCC4=CC(C(=O)N[C@@H](C)CN5C=CC(C6=CC(C(F)(F)F)=C(C#N)C=C6)=N5)=NN4)CC3)C(C)(C)C)C=C2)SC=N1	C51H63F3N12O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-SG3UMI	SCHEMBL19581037	N-[(2S)-1-[3-(5-cyano-6-methylpyridin-2-yl)pyrazol-1-yl]propan-2-yl]-5-[3-[4-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethyl]piperazin-1-yl]propoxymethyl]-1H-pyrazole-3-carboxamide	CC1=C(C#N)C=CC(C2=NN(C[C@H](C)NC(=O)C3=NNC(COCCCN4CCN(CC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=C(C)N=CS6)C=C5)C(C)(C)C)CC4)=C3)C=C2)=N1	C50H65N13O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-OA1EMI	SCHEMBL19581084	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[4-[[1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-4-oxobutyl]piperazin-1-yl]pyridine-3-carboxamide; SCHEMBL19598697	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(NC(=O)CCCN3CCN(C4=CC=C(C(=O)NC5C(C)(C)C(OC6=CC=C(C#N)C(Cl)=C6)C5(C)C)C=N4)CC3)C(C)(C)C)C=C2)SC=N1	C52H66ClN9O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-51CVC1	WO2019023553A1_769	.	CC(C)[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(Cl)C=C1)N1CC2=C(C=C(N3CCN(CCCC4=CC=C(C(=O)NC5C(C)(C)C(OC6=CC=C(C#N)C(C(F)(F)F)=C6)C5(C)C)C=C4)CC3)C=C2)C1=O	C55H63ClF3N7O6	AR	P10275	VHL	WO-2019023553-A1
TPD-Z4DDU7	WO2019023553A1_771	.	CC(C)[C@@H](C(=O)N1C[C@@H](O)C[C@H]1C(=O)NCC1=CC=C(C#N)C=C1)N1CC2=C(C=C(N3CCN(CCCC4=CC=C(C(=O)N[C@H]5C(C)(C)[C@H](OC6=CC=C(C#N)C(C(F)(F)F)=C6)C5(C)C)C=C4)CC3)C=C2)C1=O	C56H63F3N8O6	AR	P10275	VHL	WO-2019023553-A1
TPD-EF4DRM	WO2019023553A1_773	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=C(N5CCN(CCCC6=CC=C(C(=O)N[C@H]7C(C)(C)[C@@H](OC8=CC=C(C#N)C(Cl)=C8)C7(C)C)C=C6)CC5)C=C4)C3=O)C=C2)SC=N1	C58H67ClN8O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-7BDL5P	WO2019023553A1_774	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=C(N5CCN(CCCC6=CC=C(C(=O)N[C@H]7C(C)(C)[C@H](OC8=CC=C(C#N)C(Cl)=C8)C7(C)C)C=C6)CC5)C=C4)C3=O)C=C2)SC=N1	C58H67ClN8O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-6UIIEL	WO2019023553A1_775	.	CC1[C@H](NC(=O)C2=CN=C(N3CCN(CCOCC(=O)N[C@H](C(=O)N4C[C@@H](O)C[C@H]4C(=O)NCC4=CC(F)=CC=C4F)C(C)(C)C)CC3)C=C2)C(C)[C@@H]1OC1=CC(Cl)=C(C#N)C=C1	C45H55ClF2N8O7	AR	P10275	VHL	WO-2019023553-A1
TPD-3UGTYI	WO2019023553A1_776	.	CC(C)(C)C1=CC=C(CNC(=O)[C@@H]2C[C@H](O)CN2C(=O)[C@@H](NC(=O)COCCN2CCN(C3=NC=C(C(=O)N[C@H]4C(C)(C)[C@@H](OC5=CC(Cl)=C(C#N)C=C5)C4(C)C)C=C3)CC2)C(C)(C)C)C=C1	C51H69ClN8O7	AR	P10275	VHL	WO-2019023553-A1
TPD-CNM166	WO2019023553A1_777	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=C(N5CCN(CCCC6=CC=C(C(=O)N[C@H]7C(C)(C)[C@@H](OC8=CC=C(C#N)C(Cl)=C8)C7(C)C)C=C6)CC5)C=C4)C3=O)C=C2)SC=N1	C59H69ClN8O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-3EMNAP	WO2019023553A1_778	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=C(N5CCN(CCCC6=CC=C(C(=O)NC7C(C)(C)C(OC8=CC=C(C#N)C(Cl)=C8)C7(C)C)C=C6)CC5)C=C4)C3=O)C=C2)SC=N1	C59H69ClN8O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-1M1M28	WO2019023553A1_779	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCN3CCN(C4=NC=C(C(=O)NC5C(C)(C)C(OC6=CC=C(C#N)C(Cl)=C6)C5(C)C)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C53H68ClN9O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-B71PJW	WO2019023553A1_780	.	CC1=C(C2=CC=C([C@H](CO)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCN3CCN(C4=NC=C(C(=O)NC5C(C)(C)C(OC6=CC=C(C#N)C(Cl)=C6)C5(C)C)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C54H70ClN9O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-I99C77	SCHEMBL19580944	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[4-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1R)-2-hydroxy-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-4-oxobutyl]piperazin-1-yl]pyridine-3-carboxamide; SCHEMBL29817007	CC1=C(C2=CC=C([C@H](CO)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCN3CCN(C4=NC=C(C(=O)NC5C(C)(C)C(OC6=CC=C(C#N)C(Cl)=C6)C5(C)C)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C52H66ClN9O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-9FLRR7	SCHEMBL19580739	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[2-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]ethyl]-1,4-diazepan-1-yl]pyridine-3-carboxamide; SCHEMBL29817268	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCN3CCCN(C4=NC=C(C(=O)N[C@H]5C(C)(C)[C@@H](OC6=CC=C(C#N)C(Cl)=C6)C5(C)C)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C53H68ClN9O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-XJDOL7	WO2019023553A1_783	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCN(C[C@@H](F)CC4=CC=C(C(=O)N[C@H]5C(C)(C)[C@H](OC6=CC=C(C#N)C(Cl)=C6)C5(C)C)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C54H68ClFN8O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-FYKCN1	SCHEMBL19580801	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[5-[[1-[(2S,4R)-2-[[(1S)-1-(4-cyano-2-methoxyphenyl)ethyl]carbamoyl]-4-hydroxypyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-5-oxopentyl]piperazin-1-yl]pyridine-3-carboxamide	COC1=CC(C#N)=CC=C1[C@H](C)NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)C(NC(=O)CCCCN1CCN(C2=NC=C(C(=O)NC3C(C)(C)C(OC4=CC=C(C#N)C(Cl)=C4)C3(C)C)C=C2)CC1)C(C)(C)C	C51H66ClN9O7	AR	P10275	VHL	WO-2019023553-A1
TPD-NRE4RF	SCHEMBL19580585	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[2-[2-[[1-[(2S,4R)-2-[[(1S)-1-(4-cyano-2-methoxyphenyl)ethyl]carbamoyl]-4-hydroxypyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]ethyl]piperazin-1-yl]pyridine-3-carboxamide	COC1=CC(C#N)=CC=C1[C@H](C)NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)C(NC(=O)COCCN1CCN(C2=NC=C(C(=O)N[C@H]3C(C)(C)[C@@H](OC4=CC=C(C#N)C(Cl)=C4)C3(C)C)C=C2)CC1)C(C)(C)C	C50H64ClN9O8	AR	P10275	VHL	WO-2019023553-A1
TPD-CM828Q	WO2019023553A1_786	.	CC1=C(C2=CC=C([C@H](C)NC(=O)C3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCN3[C@H](C)CN(C4=CC=C(C(=O)N[C@H]5C(C)(C)[C@H](OC6=CC=C(C#N)C(Cl)=C6)C5(C)C)N=C4)C[C@@H]3C)C(C)(C)C)C=C2)SC=N1	C54H70ClN9O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-O9HDRX	WO2019023553A1_787	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCN3C4CCC3CN(C3=CC=C(C(=O)N[C@H]5C(C)(C)[C@H](OC6=CC=C(C#N)C(Cl)=C6)C5(C)C)C=N3)C4)C(C)(C)C)C=C2)SC=N1	C53H66ClN9O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-VOZIL6	WO2019023553A1_788	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCN3CCN(C4=CC=C(C(=O)NC5C(C)(C)C(SC6=CC=C(C#N)C(Cl)=C6)C5(C)C)N=C4)C[C@H]3CO)C(C)(C)C)C=C2)SC=N1	C53H68ClN9O7S2	AR	P10275	VHL	WO-2019023553-A1
TPD-SBNUOG	WO2019023553A1_789	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCN(CCN4CCN(C5=CC=C(C(=O)NC6C(C)(C)C(OC7=CC(Cl)=C(C#N)C=C7)C6(C)C)C=N5)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C56H74ClN11O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-ZQB8BR	SCHEMBL19581021	N-[(2S)-1-[3-(3-chloro-4-cyanophenyl)pyrazol-1-yl]propan-2-yl]-5-[[4-[2-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]ethyl]piperazin-1-yl]methyl]-1H-pyrazole-3-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCN3CCN(CC4=CC(C(=O)N[C@@H](C)CN5C=CC(C6=CC(Cl)=C(C#N)C=C6)=N5)=NN4)CC3)C(C)(C)C)C=C2)SC=N1	C49H61ClN12O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-YEEQXD	WO2019023553A1_791	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COC3CCCC[C@@H]3N3CCN(CCOC4=CC=C(C(=O)NC5C(C)(C)C(OC6=CC=C(C#N)C(Cl)=C6)C5(C)C)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C59H77ClN8O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-7TB7IH	WO2019023553A1_792	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CO[C@@H]3CCCC[C@H]3N3CCN(CCOC4=CC=C(C(=O)N[C@H]5C(C)(C)[C@@H](OC6=CC=C(C#N)C(Cl)=C6)C5(C)C)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C59H77ClN8O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-5843VV	SCHEMBL19580850	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[2-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[2-methoxy-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]ethyl]piperazin-1-yl]pyridine-3-carboxamide; SCHEMBL21712826; SCHEMBL29817278	COC1=C(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCN2CCN(C3=NC=C(C(=O)NC4C(C)(C)C(OC5=CC(Cl)=C(C#N)C=C5)C4(C)C)C=C3)CC2)C(C)(C)C)C=CC(C2=C(C)N=CS2)=C1	C52H66ClN9O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-GTOWRD	WO2019023553A1_794	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@H](O)CN3C(=O)[C@@H](NC(=O)CN3CC(N4CCN(C5=CC=C(C(=O)N[C@H]6C(C)(C)[C@@H](OC7=CC(Cl)=C(C#N)C=C7)C6(C)C)C=N5)CC4)C3)C(C)C)C=C2)SC=N1	C52H65ClN10O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-A03QQ9	WO2019023553A1_795	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCN(C4CN(C5=CC=C(C(=O)N[C@H]6C(C)(C)[C@@H](OC7=CC(Cl)=C(C#N)C=C7)C6(C)C)C=N5)C4)CC3)C(C)C)C=C2)SC=N1	C52H65ClN10O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-TYRB12	WO2019023553A1_796	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)C3CC(N4CCN(CCCC5=CC=C(C(=O)N[C@H]6C(C)(C)[C@@H](OC7=CC=C(C#N)C(Cl)=C7)C6(C)C)C=C5)CC4)=NO3)C=C2)SC=N1	C54H67ClN8O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-63NE76	WO2019023553A1_797	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)C3CC(N4CCN(CCCC5=CC=C(C(=O)NC6C(C)(C)C(OC7=CC=C(C#N)C(Cl)=C7)C6(C)C)C=C5)CC4)=NO3)C=C2)SC=N1	C54H67ClN8O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-RN2ALH	WO2019023553A1_798	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCN3CC4CC3CN4C3=CC=C(C(=O)NC4CC(OC5=CC=C(C#N)C(Cl)=C5)C4)C=N3)C(C)(C)C)C=C2)SC=N1	C50H60ClN9O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-H2KUCT	SCHEMBL19581105	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[2,2-difluoro-5-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-5-oxopentyl]piperazin-1-yl]pyridine-3-carboxamide; SCHEMBL29817358	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCC(F)(F)CN3CCN(C4=CC=C(C(=O)NC5C(C)(C)C(OC6=CC=C(C#N)C(Cl)=C6)C5(C)C)C=N4)CC3)C(C)(C)C)C=C2)SC=N1	C53H66ClF2N9O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-KTRHDN	SCHEMBL19580604	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[2,2-difluoro-5-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1R)-2-hydroxy-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-5-oxopentyl]piperazin-1-yl]pyridine-3-carboxamide; SCHEMBL29817337	CC1=C(C2=CC=C([C@H](CO)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCC(F)(F)CN3CCN(C4=CC=C(C(=O)NC5C(C)(C)C(OC6=CC=C(C#N)C(Cl)=C6)C5(C)C)C=N4)CC3)C(C)(C)C)C=C2)SC=N1	C53H66ClF2N9O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-09S867	WO2019023553A1_801	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CC4CCC3CN4CCCC3=CC=C(C(=O)NC4C(C)(C)C(OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C56H71ClN8O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-3WL19K	WO2019023553A1_802	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCN3C4CCC3CN(CCCC3=CC=C(C(=O)N[C@H]5C(C)(C)[C@@H](OC6=CC=C(C#N)C(Cl)=C6)C5(C)C)C=C3)C4)C(C)(C)C)C=C2)SC=N1	C57H73ClN8O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-ZNYZI3	SCHEMBL19580793	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[3-[4-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-4-oxobutyl]oxetan-3-yl]piperazin-1-yl]pyridine-3-carboxamide; SCHEMBL29817255	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCC3(N4CCN(C5=NC=C(C(=O)NC6C(C)(C)C(OC7=CC=C(C#N)C(Cl)=C7)C6(C)C)C=C5)CC4)COC3)C(C)(C)C)C=C2)SC=N1	C55H70ClN9O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-241NSS	WO2019023553A1_804	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCN(CCCCN4CCN(C5=CC=C(C(=O)NC6C(C)(C)C(OC7=CC(F)=C(C#N)C=C7)C6(C)C)C=N5)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C58H78FN11O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-IPEKE2	SCHEMBL19580814	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[2-[2-[4-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethyl]piperazin-1-yl]ethoxy]ethyl]piperazin-1-yl]pyridine-3-carboxamide; SCHEMBL29817147	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCN(CCOCCN4CCN(C5=CC=C(C(=O)N[C@H]6C(C)(C)[C@H](OC7=CC=C(C#N)C(Cl)=C7)C6(C)C)C=N5)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C58H78ClN11O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-36TA33	SCHEMBL19580935	(2S,4R)-1-[(2S)-2-[[2-[4-[4-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenyl]butyl]piperazin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL29817338	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCN(CCCCC4=CC=C(C(=O)NC5C(C)(C)C(OC6=CC=C(C#N)C(Cl)=C6)C5(C)C)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C55H71ClN8O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-XPJW11	WO2019023553A1_807	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CC4CC3CN4CCCC3=CC=C(C(=O)NC4C(C)(C)C(OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C55H69ClN8O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-1X8NMV	WO2019023553A1_808	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CC4CCC(C3)N4CCCC3=CC=C(C(=O)N[C@H]4C(C)(C)[C@H](OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)C(C)(C)C)C=C2)SC=N1	C56H71ClN8O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-FJC0LO	WO2019023553A1_853	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCN(CC4CCN(C5=NC=C(C(=O)NC6C(C)(C)C(OC7=CC(Cl)=C(C#N)CC7)C6(C)C)C=C5)CC4)CC3)C(C)C)C=C2)SC=N1	C55H73ClN10O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-M8M55G	WO2019023553A1_854	.	CC1=C(C2=CC=C([C@H](CO)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCN(CC4CCN(C5=NC=C(C(=O)NC6C(C)(C)C(OC7=CC(Cl)=C(C#N)C=C7)C6(C)C)C=C5)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C56H73ClN10O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-TXSHDV	WO2019023553A1_855	.	C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](NC(=O)COCCN1CCN(C2=NC=C(C(=O)NC3C(C)(C)C(OC4=CC(C(F)(F)F)=C(C#N)C=C4)C3(C)C)C=C2)CC1)C(C)(C)C)C1=CC=CC=C1	C49H63F3N8O7	AR	P10275	VHL	WO-2019023553-A1
TPD-J9N7A2	SCHEMBL19598772	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[2-[[2-[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]-3-oxo-1H-isoindol-5-yl]oxy]ethyl]piperazin-1-yl]pyridine-3-carboxamide; SCHEMBL29817146	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=CC=C(OCCN5CCN(C6=CC=C(C(=O)N[C@H]7C(C)(C)[C@H](OC8=CC=C(C#N)C(Cl)=C8)C7(C)C)C=N6)CC5)C=C4C3=O)C=C2)SC=N1	C57H66ClN9O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-K3XS9M	WO2019023553A1_857	.	CC(=O)O[C@@H]1C[C@@H](C(=O)N[C@H](C)C2=CC=C(C3=C(C)N=CS3)C=C2)N(C(=O)[C@H](C(C)C)N2CC3=C(C=C(OCCN4CCN(C5=CC=C(C(=O)NC6C(C)(C)C(OC7=CC=C(C#N)C(Cl)=C7)C6(C)C)C=N5)CC4)C=C3)C2=O)C1	C59H68ClN9O8S	AR	P10275	VHL	WO-2019023553-A1
TPD-Y48ASE	WO2019023553A1_858	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@H]3C[C@H](O)CN3C(=O)[C@@H](NC(=O)CN3C4CCC3CN(CCCOC3=CC=C(C(=O)N[C@H]5C(C)(C)[C@H](OC6=CC(Cl)=C(C#N)C=N6)C5(C)C)C=C3)C4)C(C)(C)C)C=C2)SC=N1	C55H70ClN9O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-8Z7PGB	SCHEMBL19580985	(2S,4R)-1-[(2S)-2-[[2-[4-[4-[4-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]phenyl]butyl]piperazin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1R)-2-hydroxy-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CO)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCN(CCCCC4=CC=C(C(=O)NC5C(C)(C)C(OC6=CC(Cl)=C(C#N)C=C6)C5(C)C)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C55H71ClN8O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-7OMC9Q	SCHEMBL19600889	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[3-[[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethyl]amino]cyclobutyl]piperazin-1-yl]pyridine-3-carboxamide; SCHEMBL19601059; SCHEMBL21712829	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CNC3CC(N4CCN(C5=CC=C(C(=O)N[C@H]6C(C)(C)[C@@H](OC7=CC=C(C#N)C(Cl)=C7)C6(C)C)C=N5)CC4)C3)C(C)(C)C)C=C2)SC=N1	C54H69ClN10O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-1XP5E2	SCHEMBL19601004	4-[(3R,5S)-1-[(2S)-2-[[2-[2-[4-[5-[[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]carbamoyl]pyridin-2-yl]piperazin-1-yl]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-5-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-3-yl]oxy-4-oxobutanoic acid	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](OC(=O)CCC(=O)O)CN3C(=O)[C@@H](NC(=O)COCCN3CCN(C4=NC=C(C(=O)NC5C(C)(C)C(OC6=CC=C(C#N)C(Cl)=C6)C5(C)C)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C56H70ClN9O10S	AR	P10275	VHL	WO-2019023553-A1
TPD-OYWID7	WO2019023553A1_863	.	[2H]C([2H])(NC1=CC=C(C(=O)N[C@H]2C(C)(C)[C@@H](OC3=CC(Cl)=C(C#N)C=C3)C2(C)C)C=C1)C([2H])([2H])C([2H])([2H])C([2H])([2H])C([2H])([2H])C([2H])([2H])OCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=C(C)N=CS2)C=C1)C(C)(C)C	C53H68ClN7O7S	AR	P10275	VHL	WO-2019023553-A1
TPD-93OJIO	WO2019023553A1_864	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCN(CCO/N=C(\C)C4=CC(C(=O)N[C@H](C)CN5C=CC(C6=CC(Cl)=C(C#N)C=C6)=N5)=NN4)CC3)C(C)(C)C)C=C2)SC=N1	C50H62ClN13O6S	AR	P10275	VHL	WO-2019023553-A1
TPD-B0YOVN	SCHEMBL19608689	N-[3-(3-carbamothioylphenyl)-1-[3-fluoro-2-(fluoromethyl)propyl]indol-6-yl]-3-[2-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyethoxy]ethoxy]ethoxy]propanamide	NC(=S)C1=CC(C2=CN(CC(CF)CF)C3=C2C=CC(NC(=O)CCOCCOCCOCCOC2=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C2)=C3)=CC=C1	C41H43F2N5O9S	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-N3FQ16	SCHEMBL20975149	N-[[3-(3-carbamothioylphenyl)-1-(oxan-4-yl)indol-6-yl]methyl]-3-[2-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyethoxy]ethoxy]ethoxy]propanamide	NC(=S)C1=CC(C2=CN(C3CCOCC3)C3=C2C=CC(CNC(=O)CCOCCOCCOCCOC2=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C2)=C3)=CC=C1	C43H47N5O10S	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-3RSJJ1	SCHEMBL20996089	N-[[3-(3-carbamothioylphenyl)-1-[1-(1,3-thiazol-2-yl)piperidin-4-yl]indol-6-yl]methyl]-3-[2-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyethoxy]ethoxy]ethoxy]propanamide	NC(=S)C1=CC(C2=CN(C3CCN(C4=NC=CS4)CC3)C3=C2C=CC(CNC(=O)CCOCCOCCOCCOC2=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C2)=C3)=CC=C1	C46H49N7O9S2	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-R94OKQ	SCHEMBL20996102	N-[3-(3-carbamothioylphenyl)-1-(oxan-4-yl)indol-6-yl]-3-[2-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyethoxy]ethoxy]ethoxy]propanamide	NC(=S)C1=CC(C2=CN(C3CCOCC3)C3=C2C=CC(NC(=O)CCOCCOCCOCCOC2=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C2)=C3)=CC=C1	C42H45N5O10S	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-IA5043	SCHEMBL20995334	N-[3-(3-carbamothioylphenyl)-1-[1-(1,3-thiazol-2-yl)piperidin-4-yl]indol-6-yl]-3-[2-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyethoxy]ethoxy]ethoxy]propanamide	NC(=S)C1=CC(C2=CN(C3CCN(C4=NC=CS4)CC3)C3=C2C=CC(NC(=O)CCOCCOCCOCCOC2=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C2)=C3)=CC=C1	C45H47N7O9S2	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-7LFATY	SCHEMBL20995326	N-[3-(3-carbamothioylphenyl)-1-(1-propan-2-ylsulfonylpiperidin-4-yl)indol-6-yl]-3-[2-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyethoxy]ethoxy]ethoxy]propanamide	CC(C)S(=O)(=O)N1CCC(N2C=C(C3=CC=CC(C(N)=S)=C3)C3=C2C=C(NC(=O)CCOCCOCCOCCOC2=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C2)C=C3)CC1	C45H52N6O11S2	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-KJ4BXB	SCHEMBL20995447	N-[3-(3-carbamothioylphenyl)-1-(2-methyl-1-methylsulfonylpiperidin-4-yl)indol-6-yl]-3-[2-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyethoxy]ethoxy]ethoxy]propanamide	CC1CC(N2C=C(C3=CC=CC(C(N)=S)=C3)C3=C2C=C(NC(=O)CCOCCOCCOCCOC2=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C2)C=C3)CCN1S(C)(=O)=O	C44H50N6O11S2	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-OHZ6QW	SCHEMBL20995330	N-[3-(3-carbamothioylphenyl)-1-[3-fluoro-2-(fluoromethyl)propyl]indol-6-yl]-3-[2-[2-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]but-3-ynoxy]ethoxy]ethoxy]ethoxy]propanamide	NC(=S)C1=CC(C2=CN(CC(CF)CF)C3=C2C=CC(NC(=O)CCOCCOCCOCCOCCC#CC2=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C2)=C3)=CC=C1	C45H47F2N5O9S	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-6BE93T	SCHEMBL20994707	N-[3-(3-carbamothioylphenyl)-1-[3-fluoro-2-(fluoromethyl)propyl]indol-6-yl]-3-[2-[5-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]pent-4-ynoxy]ethoxy]propanamide	NC(=S)C1=CC(C2=CN(CC(CF)CF)C3=C2C=CC(NC(=O)CCOCCOCCCC#CC2=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C2)=C3)=CC=C1	C42H41F2N5O7S	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-4NAUDT	SCHEMBL20996110	N-[[3-(3-carbamothioylphenyl)-1-(1-propan-2-ylsulfonylpiperidin-4-yl)indol-6-yl]methyl]-1-[2-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyethoxy]ethoxy]ethyl]azetidine-3-carboxamide	CC(C)S(=O)(=O)N1CCC(N2C=C(C3=CC=CC(C(N)=S)=C3)C3=C2C=C(CNC(=O)C2CN(CCOCCOCCOC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C2)C=C3)CC1	C47H55N7O10S2	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-9UPN0G	SCHEMBL20996112	N-[[3-(3-carbamothioylphenyl)-1-(1-propan-2-ylsulfonylpiperidin-4-yl)indol-6-yl]methyl]-1-[2-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyethoxy]ethoxy]ethyl]azetidine-2-carboxamide	CC(C)S(=O)(=O)N1CCC(N2C=C(C3=CC=CC(C(N)=S)=C3)C3=C2C=C(CNC(=O)C2CCN2CCOCCOCCOC2=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C2)C=C3)CC1	C47H55N7O10S2	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-RVXXKE	SCHEMBL20994705	N-[[3-(3-carbamothioylphenyl)-1-(1-propan-2-ylsulfonylpiperidin-4-yl)indol-6-yl]methyl]-1-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyethoxy]ethyl]azetidine-3-carboxamide	CC(C)S(=O)(=O)N1CCC(N2C=C(C3=CC=CC(C(N)=S)=C3)C3=C2C=C(CNC(=O)C2CN(CCOCCOC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C2)C=C3)CC1	C45H51N7O9S2	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-TWS94J	SCHEMBL20996836	N-[[3-(3-carbamothioylphenyl)-1-(1-propan-2-ylsulfonylpiperidin-4-yl)indol-6-yl]methyl]-1-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyethoxy]ethyl]azetidine-2-carboxamide	CC(C)S(=O)(=O)N1CCC(N2C=C(C3=CC=CC(C(N)=S)=C3)C3=C2C=C(CNC(=O)C2CCN2CCOCCOC2=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C2)C=C3)CC1	C45H51N7O9S2	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-F69RQ7	SCHEMBL20996899	N-[[3-(3-carbamothioylphenyl)-1-(1-propan-2-ylsulfonylpiperidin-4-yl)indol-6-yl]methyl]-1-[2-[2-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyethoxy]ethoxy]ethoxy]ethyl]azetidine-3-carboxamide	CC(C)S(=O)(=O)N1CCC(N2C=C(C3=CC=CC(C(N)=S)=C3)C3=C2C=C(CNC(=O)C2CN(CCOCCOCCOCCOC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C2)C=C3)CC1	C49H59N7O11S2	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-YK0NWF	SCHEMBL20995448	N-[[3-(3-carbamothioylphenyl)-1-(1-propan-2-ylsulfonylpiperidin-4-yl)indol-6-yl]methyl]-1-[2-[2-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyethoxy]ethoxy]ethoxy]ethyl]azetidine-2-carboxamide	CC(C)S(=O)(=O)N1CCC(N2C=C(C3=CC=CC(C(N)=S)=C3)C3=C2C=C(CNC(=O)C2CCN2CCOCCOCCOCCOC2=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C2)C=C3)CC1	C49H59N7O11S2	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-4E45AO	SCHEMBL20995331	N-[[3-(3-carbamothioylphenyl)-1-(1-propan-2-ylsulfonylpiperidin-4-yl)indol-6-yl]methyl]-1-[5-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyacetyl]amino]pentyl]azetidine-3-carboxamide	CC(C)S(=O)(=O)N1CCC(N2C=C(C3=CC=CC(C(N)=S)=C3)C3=C2C=C(CNC(=O)C2CN(CCCCCNC(=O)COC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C2)C=C3)CC1	C48H56N8O9S2	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-OW3NIU	SCHEMBL20996897	N-[[3-(3-carbamothioylphenyl)-1-(1-propan-2-ylsulfonylpiperidin-4-yl)indol-6-yl]methyl]-1-[6-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyacetyl]amino]hexyl]azetidine-3-carboxamide	CC(C)S(=O)(=O)N1CCC(N2C=C(C3=CC=CC(C(N)=S)=C3)C3=C2C=C(CNC(=O)C2CN(CCCCCCNC(=O)COC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C2)C=C3)CC1	C49H58N8O9S2	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-BLF9E2	SCHEMBL25156851	3-[6-[3-[5-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxypentylamino]-2-oxopyrrolidin-1-yl]-1-(1-propan-2-ylsulfonylpiperidin-4-yl)indol-3-yl]benzenecarbothioamide	CC(C)S(=O)(=O)N1CCC(N2C=C(C3=CC=CC(C(N)=S)=C3)C3=C2C=C(N2CCC(NCCCCCOC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C2=O)C=C3)CC1	C45H51N7O8S2	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-2N2A9H	SCHEMBL20995449	N-[1-[3-(3-carbamothioylphenyl)-1-(1-propan-2-ylsulfonylpiperidin-4-yl)indol-6-yl]-2-oxopyrrolidin-3-yl]-3-[2-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyethoxy]ethoxy]ethoxy]propanamide	CC(C)S(=O)(=O)N1CCC(N2C=C(C3=CC=CC(C(N)=S)=C3)C3=C2C=C(N2CCC(NC(=O)CCOCCOCCOCCOC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C2=O)C=C3)CC1	C49H57N7O12S2	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-7JD20W	SCHEMBL20995333	N-[3-(3-carbamothioylphenyl)-1-[3-fluoro-2-(fluoromethyl)propyl]indol-6-yl]-5-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]pent-4-ynamide	NC(=S)C1=CC=CC(C2=CN(CC(CF)CF)C3=C2C=CC(NC(=O)CCC#CC2=CC=CC4=C2C(=O)N(C2CCC(=O)NC2=O)C4=O)=C3)=C1	C37H31F2N5O5S	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-VWESY7	SCHEMBL20995332	N-[3-(3-carbamothioylphenyl)-1-[1-(trifluoromethylsulfonyl)piperidin-4-yl]indol-6-yl]-3-[2-[2-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]propanamide; PIYBCDRSHOZJEA-UHFFFAOYSA-N; N-[3-(3-carbamothioylphenyl)-1-[1-(trifluoromethylsulfonyl)piperidin-4-yl]indol-6-yl]-3-[2-[2-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]propanamide	NC(=S)C1=CC(C2=CN(C3CCN(S(=O)(=O)C(F)(F)F)CC3)C3=C2C=CC(NC(=O)CCOCCOCCOCCOCCOC2=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C2)=C3)=CC=C1	C45H49F3N6O12S2	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-KQDOC6	SCHEMBL20996119	N-[3-(3-carbamothioylphenyl)-1-(1-methylsulfonylpiperidin-4-yl)indol-6-yl]-3-[2-[2-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]propanamide	CS(=O)(=O)N1CCC(N2C=C(C3=CC(C(N)=S)=CC=C3)C3=C2C=C(NC(=O)CCOCCOCCOCCOCCOC2=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C2)C=C3)CC1	C45H52N6O12S2	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-O7C5OK	SCHEMBL20994709	N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-3-[2-[2-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]propanamide; SYRMAVHQCUTDQQ-UHFFFAOYSA-N; N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-3-[2-[2-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]propanamide	NC(=S)C1=CC=CC(C2=CN(C3CCC(F)(F)CC3)C3=C2C=CC(NC(=O)CCOCCOCCOCCOCCOC2=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C2)=C3)=C1	C45H49F2N5O10S	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-5LK1KS	SCHEMBL20971571	N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-9-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyacetyl]amino]nonanamide; SCHEMBL31194996; JHYWAXGWTLHCBF-UHFFFAOYSA-N; N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-9-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyacetyl]amino]nonanamide	NC(=S)C1=CC(C2=CN(C3CCC(F)(F)CC3)C3=C2C=CC(NC(=O)CCCCCCCCNC(=O)COC2=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C2)=C3)=CC=C1	C45H48F2N6O7S	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-F57F9D	SCHEMBL20995451	N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-3-[2-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyethoxy]ethoxy]ethoxy]propanamide; UCGZCSHCAZOGAM-UHFFFAOYSA-N; N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-3-[2-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyethoxy]ethoxy]ethoxy]propanamide	NC(=S)C1=CC(C2=CN(C3CCC(F)(F)CC3)C3=C2C=CC(NC(=O)CCOCCOCCOCCOC2=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C2)=C3)=CC=C1	C43H45F2N5O9S	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-H119DW	WO2019094772A1_26	.	CC1=C(C2=CC=C(CNC(=O)C3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCOCCOCCOCCOCCC(=O)NC3=CC4=C(C=C3)C(C3=CC=CC(C(N)=S)=C3)=CN4C3CCC(F)(F)CC3)C(C)(C)C)C=C2)SC=N1	C55H69F2N7O9S2	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-KVMIBG	SCHEMBL20996141	N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-2-[5-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyacetyl]amino]pentoxy]acetamide; QEAGMKLJXFEDHQ-UHFFFAOYSA-N; N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-2-[5-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyacetyl]amino]pentoxy]acetamide	NC(=S)C1=CC=CC(C2=CN(C3CCC(F)(F)CC3)C3=C2C=CC(NC(=O)COCCCCCNC(=O)COC2=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C2)=C3)=C1	C43H44F2N6O8S	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-6EQASM	SCHEMBL20995452	N-[3-(3-carbamothioylphenyl)-1-[1-(1,3-thiazol-2-yl)piperidin-4-yl]indol-6-yl]-3-[2-[2-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]propanamide	NC(=S)C1=CC(C2=CN(C3CCN(C4=NC=CS4)CC3)C3=C2C=CC(NC(=O)CCOCCOCCOCCOCCOC2=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C2)=C3)=CC=C1	C47H51N7O10S2	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-37ZMKK	SCHEMBL20996839	N-[3-(3-carbamothioylphenyl)-1-(oxan-4-yl)indol-6-yl]-3-[2-[2-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]propanamide	NC(=S)C1=CC(C2=CN(C3CCOCC3)C3=C2C=CC(NC(=O)CCOCCOCCOCCOCCOC2=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C2)=C3)=CC=C1	C44H49N5O11S	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-F72QI6	SCHEMBL20996900	N-[3-(3-carbamothioylphenyl)-1-(1-methylsulfonylpiperidin-4-yl)indol-6-yl]-9-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyacetyl]amino]nonanamide	CS(=O)(=O)N1CCC(N2C=C(C3=CC=CC(C(N)=S)=C3)C3=C2C=C(NC(=O)CCCCCCCCNC(=O)COC2=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C2)C=C3)CC1	C45H51N7O9S2	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-7CV5P3	SCHEMBL20994710	N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-9-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]oxy]acetyl]amino]nonanamide; GQAMXEHZYQJXDH-UHFFFAOYSA-N; N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-9-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]oxy]acetyl]amino]nonanamide	NC(=S)C1=CC(C2=CN(C3CCC(F)(F)CC3)C3=C2C=CC(NC(=O)CCCCCCCCNC(=O)COC2=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C2)=C3)=CC=C1	C45H50F2N6O6S	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-W7Y8XE	SCHEMBL20995339	3-[1-(4,4-difluorocyclohexyl)-6-[9-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]oxy]acetyl]amino]nonanoylamino]indol-3-yl]benzamide; VNAAQDKRFXUSCS-UHFFFAOYSA-N; 3-[1-(4,4-difluorocyclohexyl)-6-[9-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]oxy]acetyl]amino]nonanoylamino]indol-3-yl]benzamide	NC(=O)C1=CC(C2=CN(C3CCC(F)(F)CC3)C3=C2C=CC(NC(=O)CCCCCCCCNC(=O)COC2=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C2)=C3)=CC=C1	C45H50F2N6O7	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-OVYI1J	SCHEMBL20996902	N-[3-(3-carbamothioylphenyl)-7-chloro-1-(4,4-difluorocyclohexyl)indol-6-yl]-9-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]oxy]acetyl]amino]nonanamide; ZBMSKGQDAQLBMF-UHFFFAOYSA-N; N-[3-(3-carbamothioylphenyl)-7-chloro-1-(4,4-difluorocyclohexyl)indol-6-yl]-9-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]oxy]acetyl]amino]nonanamide	NC(=S)C1=CC(C2=CN(C3CCC(F)(F)CC3)C3=C2C=CC(NC(=O)CCCCCCCCNC(=O)COC2=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C2)=C3Cl)=CC=C1	C45H49ClF2N6O6S	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-3NIVA9	SCHEMBL20975153	N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-9-[3-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]propanoylamino]nonanamide; XGRPLHRVGOBRDK-UHFFFAOYSA-N; N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-9-[3-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]propanoylamino]nonanamide	NC(=S)C1=CC(C2=CN(C3CCC(F)(F)CC3)C3=C2C=CC(NC(=O)CCCCCCCCNC(=O)CCC2=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C2)=C3)=CC=C1	C46H52F2N6O5S	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-V471GK	SCHEMBL20996154	N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-9-[[(E)-3-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]prop-2-enoyl]amino]nonanamide; CSFPRXQJRJVFEY-NBVRZTHBSA-N; N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-9-[[(E)-3-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]prop-2-enoyl]amino]nonanamide	NC(=S)C1=CC(C2=CN(C3CCC(F)(F)CC3)C3=C2C=CC(NC(=O)CCCCCCCCNC(=O)/C=C/C2=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C2)=C3)=CC=C1	C46H50F2N6O5S	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-8E4W1P	SCHEMBL20996842	N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-9-[[2-[2-(1-methyl-2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyacetyl]amino]nonanamide; QTYKHNYHNXLSRQ-UHFFFAOYSA-N; N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-9-[[2-[2-(1-methyl-2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyacetyl]amino]nonanamide	CN1C(=O)CCC(N2C(=O)C3=CC=CC(OCC(=O)NCCCCCCCCC(=O)NC4=CC5=C(C=C4)C(C4=CC=CC(C(N)=S)=C4)=CN5C4CCC(F)(F)CC4)=C3C2=O)C1=O	C46H50F2N6O7S	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-WKTA9Z	SCHEMBL20995363	N'-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-N-[2-[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]propoxy]ethyl]hexanediamide; HBFCFVMDNDZTNI-UHFFFAOYSA-N; N'-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-N-[2-[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]propoxy]ethyl]hexanediamide	NC(=S)C1=CC(C2=CN(C3CCC(F)(F)CC3)C3=C2C=CC(NC(=O)CCCCC(=O)NCCOCCCC2=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C2)=C3)=CC=C1	C45H48F2N6O7S	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-HF3BF5	SCHEMBL20995340	N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-9-[[2-[[2-(1-methyl-2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]oxy]acetyl]amino]nonanamide; QTAAZAHFDYIXNI-UHFFFAOYSA-N; N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-9-[[2-[[2-(1-methyl-2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]oxy]acetyl]amino]nonanamide	CN1C(=O)CCC(N2CC3=C(OCC(=O)NCCCCCCCCC(=O)NC4=CC5=C(C=C4)C(C4=CC=CC(C(N)=S)=C4)=CN5C4CCC(F)(F)CC4)C=CC=C3C2=O)C1=O	C46H52F2N6O6S	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-T9OZ4T	SCHEMBL20996843	N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-7-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyacetyl]amino]heptanamide; LGULTYWKMCZCAO-UHFFFAOYSA-N; N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-7-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyacetyl]amino]heptanamide	NC(=S)C1=CC(C2=CN(C3CCC(F)(F)CC3)C3=C2C=CC(NC(=O)CCCCCCNC(=O)COC2=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C2)=C3)=CC=C1	C43H44F2N6O7S	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-8NQ393	SCHEMBL20996901	N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-3-[6-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]hexoxy]propanamide; XHKJXCFUKVKSRF-UHFFFAOYSA-N; N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-3-[6-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]hexoxy]propanamide	NC(=S)C1=CC(C2=CN(C3CCC(F)(F)CC3)C3=C2C=CC(NC(=O)CCOCCCCCCNC2=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C2)=C3)=CC=C1	C43H46F2N6O6S	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-0FPA69	SCHEMBL20975157	N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-3-[6-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyhexoxy]propanamide; VKLDTFVRSQHSAT-UHFFFAOYSA-N; N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-3-[6-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyhexoxy]propanamide	NC(=S)C1=CC(C2=CN(C3CCC(F)(F)CC3)C3=C2C=CC(NC(=O)CCOCCCCCCOC2=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C2)=C3)=CC=C1	C43H45F2N5O7S	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-MJOBDM	SCHEMBL20996904	N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-3-[6-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyhexyl-methylamino]propanamide; HMYHWRYKDNSKNN-UHFFFAOYSA-N; N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-3-[6-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyhexyl-methylamino]propanamide	CN(CCCCCCOC1=C2C(=O)N(C3CCC(=O)NC3=O)C(=O)C2=CC=C1)CCC(=O)NC1=CC2=C(C=C1)C(C1=CC=CC(C(N)=S)=C1)=CN2C1CCC(F)(F)CC1	C44H48F2N6O6S	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-UIVQOE	SCHEMBL20996845	N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-3-[6-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyhexylamino]propanamide; PVICNIGQYJIENL-UHFFFAOYSA-N; N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-3-[6-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyhexylamino]propanamide	NC(=S)C1=CC(C2=CN(C3CCC(F)(F)CC3)C3=C2C=CC(NC(=O)CCNCCCCCCOC2=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C2)=C3)=CC=C1	C43H46F2N6O6S	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-H4167J	SCHEMBL20996179	N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]but-3-ynoxy]propoxy]butanamide; XBWVREHKXDWJTL-UHFFFAOYSA-N; N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]but-3-ynoxy]propoxy]butanamide	NC(=S)C1=CC(C2=CN(C3CCC(F)(F)CC3)C3=C2C=CC(NC(=O)CCCOCCCOCCC#CC2=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C2)=C3)=CC=C1	C45H47F2N5O6S	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-3PYBPF	SCHEMBL20996847	N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]butoxy]propoxy]butanamide; OTEZFZMVWVTFBH-UHFFFAOYSA-N; N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]butoxy]propoxy]butanamide	NC(=S)C1=CC(C2=CN(C3CCC(F)(F)CC3)C3=C2C=CC(NC(=O)CCCOCCCOCCCCC2=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C2)=C3)=CC=C1	C45H51F2N5O6S	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-CN0PT6	SCHEMBL20996850	N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-3-[3-[5-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]pent-4-ynoxy]propoxy]propanamide; DZVFZWSBQSHMTP-UHFFFAOYSA-N; N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-3-[3-[5-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]pent-4-ynoxy]propoxy]propanamide	NC(=S)C1=CC(C2=CN(C3CCC(F)(F)CC3)C3=C2C=CC(NC(=O)CCOCCCOCCCC#CC2=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C2)=C3)=CC=C1	C45H47F2N5O6S	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-EZSHT3	SCHEMBL20996849	N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-3-[3-[5-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]pentoxy]propoxy]propanamide; DOVHKJZUYFEWRY-UHFFFAOYSA-N; N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-3-[3-[5-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]pentoxy]propoxy]propanamide	NC(=S)C1=CC(C2=CN(C3CCC(F)(F)CC3)C3=C2C=CC(NC(=O)CCOCCCOCCCCCC2=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C2)=C3)=CC=C1	C45H51F2N5O6S	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-SWGTI8	SCHEMBL20995344	N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-5-[5-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]pent-4-ynoxy]pentanamide; AKGPILZRVZVIMS-UHFFFAOYSA-N; N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-5-[5-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]pent-4-ynoxy]pentanamide	NC(=S)C1=CC(C2=CN(C3CCC(F)(F)CC3)C3=C2C=CC(NC(=O)CCCCOCCCC#CC2=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C2)=C3)=CC=C1	C44H45F2N5O5S	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-41SXQV	SCHEMBL20996848	N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-6-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]but-3-ynoxy]hexanamide; FGZAESCJRDDNSO-UHFFFAOYSA-N; N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-6-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]but-3-ynoxy]hexanamide	NC(=S)C1=CC(C2=CN(C3CCC(F)(F)CC3)C3=C2C=CC(NC(=O)CCCCCOCCC#CC2=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C2)=C3)=CC=C1	C44H45F2N5O5S	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-219024	SCHEMBL20996853	N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-3-[6-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]oxy]hexoxy]propanamide; AXXUYUUPYQHYSI-UHFFFAOYSA-N; N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-3-[6-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]oxy]hexoxy]propanamide	NC(=S)C1=CC(C2=CN(C3CCC(F)(F)CC3)C3=C2C=CC(NC(=O)CCOCCCCCCOC2=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C2)=C3)=CC=C1	C43H47F2N5O6S	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-3GC8N8	SCHEMBL20996855	N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-3-[6-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]hexoxy]propanamide; HSCRXYVYZMELCF-UHFFFAOYSA-N; N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-3-[6-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]hexoxy]propanamide	NC(=S)C1=CC(C2=CN(C3CCC(F)(F)CC3)C3=C2C=CC(NC(=O)CCOCCCCCCNC2=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C2)=C3)=CC=C1	C43H48F2N6O5S	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-H5CFY7	SCHEMBL20995453	N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-3-[3-[4-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]oxy]butoxy]propoxy]propanamide; WTWDPIHVDHHXQI-UHFFFAOYSA-N; N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-3-[3-[4-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]oxy]butoxy]propoxy]propanamide	NC(=S)C1=CC(C2=CN(C3CCC(F)(F)CC3)C3=C2C=CC(NC(=O)CCOCCCOCCCCOC2=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C2)=C3)=CC=C1	C44H49F2N5O7S	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-JNE2FS	SCHEMBL20996171	N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-3-[3-[4-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]butoxy]propoxy]propanamide; DDVWXHCCCXYXSY-UHFFFAOYSA-N; N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-3-[3-[4-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]butoxy]propoxy]propanamide	NC(=S)C1=CC(C2=CN(C3CCC(F)(F)CC3)C3=C2C=CC(NC(=O)CCOCCCOCCCCNC2=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C2)=C3)=CC=C1	C44H50F2N6O6S	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-KY5Z7E	SCHEMBL20995462	N-[3-(3-carbamothioylphenyl)-1-[3-fluoro-2-(fluoromethyl)propyl]indol-6-yl]-3-[2-[2-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]propanamide	NC(=S)C1=CC=CC(C2=CN(CC(CF)CF)C3=C2C=CC(NC(=O)CCOCCOCCOCCOCCOC2=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C2)=C3)=C1	C43H47F2N5O10S	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-0BP3HT	SCHEMBL20996859	N-[3-(3-carbamothioylphenyl)-1-[3-fluoro-2-(fluoromethyl)propyl]indol-6-yl]-3-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyethoxy]ethoxy]propanamide	NC(=S)C1=CC=CC(C2=CN(CC(CF)CF)C3=C2C=CC(NC(=O)CCOCCOCCOC2=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C2)=C3)=C1	C39H39F2N5O8S	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-TKH0LL	SCHEMBL20996905	N-[3-(3-carbamothioylphenyl)-1-[3-fluoro-2-(fluoromethyl)propyl]indol-6-yl]-3-[2-[2-[2-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]ethoxy]propanamide	NC(=S)C1=CC=CC(C2=CN(CC(CF)CF)C3=C2C=CC(NC(=O)CCOCCOCCOCCOCCOCCOC2=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C2)=C3)=C1	C45H51F2N5O11S	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-K7EEXM	SCHEMBL20996182	N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-7-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]oxy]acetyl]amino]heptanamide; TVSFQACBUUHHDO-UHFFFAOYSA-N; N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-7-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]oxy]acetyl]amino]heptanamide	NC(=S)C1=CC(C2=CN(C3CCC(F)(F)CC3)C3=C2C=CC(NC(=O)CCCCCCNC(=O)COC2=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C2)=C3)=CC=C1	C43H46F2N6O6S	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-GY7ZDV	SCHEMBL20994714	N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-7-[3-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]propanoylamino]heptanamide; OGVIKUPGIWAITD-UHFFFAOYSA-N; N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-7-[3-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]propanoylamino]heptanamide	NC(=S)C1=CC(C2=CN(C3CCC(F)(F)CC3)C3=C2C=CC(NC(=O)CCCCCCNC(=O)CCC2=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C2)=C3)=CC=C1	C44H48F2N6O5S	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-5FAZRX	SCHEMBL20995345	N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-2-[1-[2-[3-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]prop-2-ynoxy]ethyl]azetidin-3-yl]acetamide; RWCUJFRAQWKHJZ-UHFFFAOYSA-N; N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-2-[1-[2-[3-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]prop-2-ynoxy]ethyl]azetidin-3-yl]acetamide	NC(=S)C1=CC=CC(C2=CN(C3CCC(F)(F)CC3)C3=C2C=CC(NC(=O)CC2CN(CCOCC#CC4=C5CN(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C2)=C3)=C1	C44H44F2N6O5S	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-LU2P3W	SCHEMBL25156835	N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-2-[1-[6-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]hex-5-ynyl]azetidin-3-yl]acetamide	NC(=S)C1=CC=CC(C2=CN(C3CCC(F)(F)CC3)C3=C2C=CC(NC(=O)CC2CN(CCCCC#CC4=C5CN(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C2)=C3)=C1	C45H46F2N6O4S	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-X6GLXC	SCHEMBL20996861	N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-2-[1-[6-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]hex-5-ynoyl]azetidin-3-yl]acetamide; HXKFSHSJZXIFCY-UHFFFAOYSA-N; N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-2-[1-[6-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]hex-5-ynoyl]azetidin-3-yl]acetamide	NC(=S)C1=CC=CC(C2=CN(C3CCC(F)(F)CC3)C3=C2C=CC(NC(=O)CC2CN(C(=O)CCCC#CC4=C5CN(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C2)=C3)=C1	C45H44F2N6O5S	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-WWD2AY	SCHEMBL20994717	N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-3-[4-[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxypropyl]piperazin-1-yl]propanamide; VBZKYJRNZXNXNB-UHFFFAOYSA-N; N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-3-[4-[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxypropyl]piperazin-1-yl]propanamide	NC(=S)C1=CC(C2=CN(C3CCC(F)(F)CC3)C3=C2C=CC(NC(=O)CCN2CCN(CCCOC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC2)=C3)=CC=C1	C44H47F2N7O6S	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-LP9QHH	SCHEMBL20995346	N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-9-[[(E)-3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]prop-2-enoyl]amino]nonanamide; ZYYDNILTIAIYAM-NBVRZTHBSA-N; N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-9-[[(E)-3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]prop-2-enoyl]amino]nonanamide	NC(=S)C1=CC(C2=CN(C3CCC(F)(F)CC3)C3=C2C=CC(NC(=O)CCCCCCCCNC(=O)/C=C/C2=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C2)=C3)=CC=C1	C46H48F2N6O6S	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-WNO69G	SCHEMBL20995359	N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-9-[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]propanoylamino]nonanamide; OVPULMTXJSSFCE-UHFFFAOYSA-N; N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-9-[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]propanoylamino]nonanamide	NC(=S)C1=CC(C2=CN(C3CCC(F)(F)CC3)C3=C2C=CC(NC(=O)CCCCCCCCNC(=O)CCC2=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C2)=C3)=CC=C1	C46H50F2N6O6S	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-GPZ0F2	SCHEMBL20996906	N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]but-3-ynoxy]propoxy]butanamide; YQUIORKLPYJJJO-UHFFFAOYSA-N; N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]but-3-ynoxy]propoxy]butanamide	NC(=S)C1=CC(C2=CN(C3CCC(F)(F)CC3)C3=C2C=CC(NC(=O)CCCOCCCOCCC#CC2=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C2)=C3)=CC=C1	C45H45F2N5O7S	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-R05AQT	SCHEMBL20996211	N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]butoxy]propoxy]butanamide; LNLIDBSYFSSGEP-UHFFFAOYSA-N; N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]butoxy]propoxy]butanamide	NC(=S)C1=CC(C2=CN(C3CCC(F)(F)CC3)C3=C2C=CC(NC(=O)CCCOCCCOCCCCC2=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C2)=C3)=CC=C1	C45H49F2N5O7S	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-3Z10LF	WO2019094772A1_72	3-[1-(4,4-Difluorocyclohexyl)-6-[9-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyacetyl]amino]nonanoylamino]indol-3-yl]benzamide	NC(=O)C1=CC(C2=CN(C3CCC(F)(F)CC3)C3=C2C=CC(NC(=O)CCCCCCCCNC(=O)COC2=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C2)=C3)=CC=C1	C45H48F2N6O8	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-XZT9WF	SCHEMBL25156729	N-[8-[[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]sulfamoyl]octyl]-2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]oxy]acetamide	NC(=S)C1=CC(C2=CN(C3CCC(F)(F)CC3)C3=C2C=CC(NS(=O)(=O)CCCCCCCCNC(=O)COC2=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C2)=C3)=CC=C1	C44H50F2N6O7S2	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-XT364H	SCHEMBL20996863	N'-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-N-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]oxy]ethyl]nonanediamide; QTBZHTUEFQGUKG-UHFFFAOYSA-N; N'-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-N-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]oxy]ethyl]nonanediamide	NC(=S)C1=CC(C2=CN(C3CCC(F)(F)CC3)C3=C2C=CC(NC(=O)CCCCCCCC(=O)NCCOC2=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C2)=C3)=CC=C1	C45H50F2N6O6S	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-V0Z4C0	SCHEMBL20994720	N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-9-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]acetyl]amino]nonanamide; WARFWMYQELYLFH-UHFFFAOYSA-N; N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-9-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]acetyl]amino]nonanamide	NC(=S)C1=CC(C2=CN(C3CCC(F)(F)CC3)C3=C2C=CC(NC(=O)CCCCCCCCNC(=O)CNC2=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C2)=C3)=CC=C1	C45H51F2N7O5S	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-U40ZDY	SCHEMBL20995377	3-[1-(4,4-difluorocyclohexyl)-6-[7-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]oxy]acetyl]amino]heptanoylamino]indol-3-yl]benzamide; QCNMMYHFNVZFOD-UHFFFAOYSA-N; 3-[1-(4,4-difluorocyclohexyl)-6-[7-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]oxy]acetyl]amino]heptanoylamino]indol-3-yl]benzamide	NC(=O)C1=CC=CC(C2=CN(C3CCC(F)(F)CC3)C3=C2C=CC(NC(=O)CCCCCCNC(=O)COC2=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C2)=C3)=C1	C43H46F2N6O7	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-FGCRLX	SCHEMBL20996907	N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-6-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]oxy]acetyl]amino]hexanamide; DCHOBTORMHWOSL-UHFFFAOYSA-N; N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-6-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]oxy]acetyl]amino]hexanamide	NC(=S)C1=CC(C2=CN(C3CCC(F)(F)CC3)C3=C2C=CC(NC(=O)CCCCCNC(=O)COC2=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C2)=C3)=CC=C1	C42H44F2N6O6S	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-FXEE08	SCHEMBL20996862	N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-6-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyacetyl]amino]hexanamide; ZZCSHAIXQCLTMU-UHFFFAOYSA-N; N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-6-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyacetyl]amino]hexanamide	NC(=S)C1=CC(C2=CN(C3CCC(F)(F)CC3)C3=C2C=CC(NC(=O)CCCCCNC(=O)COC2=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C2)=C3)=CC=C1	C42H42F2N6O7S	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-KWTV1K	SCHEMBL20995381	N'-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-N-[2-[3-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]prop-2-ynoxy]ethyl]hexanediamide; STGUTPQUKNKQCY-UHFFFAOYSA-N; N'-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-N-[2-[3-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]prop-2-ynoxy]ethyl]hexanediamide	NC(=S)C1=CC(C2=CN(C3CCC(F)(F)CC3)C3=C2C=CC(NC(=O)CCCCC(=O)NCCOCC#CC2=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C2)=C3)=CC=C1	C45H46F2N6O6S	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-8RST95	SCHEMBL20995463	N-[[3-(3-carbamothioylphenyl)-1-[1-[7-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]oxy]acetyl]amino]heptylsulfonyl]piperidin-4-yl]indol-6-yl]methyl]-1-methylazetidine-3-carboxamide	CN1CC(C(=O)NCC2=CC3=C(C=C2)C(C2=CC=CC(C(N)=S)=C2)=CN3C2CCN(S(=O)(=O)CCCCCCCNC(=O)COC3=CC=CC4=C3CN(C3CCC(=O)NC3=O)C4=O)CC2)C1	C48H58N8O8S2	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-V5YKQH	SCHEMBL20996865	N-[[3-(3-carbamothioylphenyl)-1-[1-[6-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]oxy]acetyl]amino]hexylsulfamoyl]piperidin-4-yl]indol-6-yl]methyl]-1-methylazetidine-3-carboxamide	CN1CC(C(=O)NCC2=CC3=C(C=C2)C(C2=CC=CC(C(N)=S)=C2)=CN3C2CCN(S(=O)(=O)NCCCCCCNC(=O)COC3=CC=CC4=C3CN(C3CCC(=O)NC3=O)C4=O)CC2)C1	C47H57N9O8S2	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-104HKF	SCHEMBL20996866	N-[[3-(3-carbamothioylphenyl)-1-[1-[8-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]oxy]acetyl]amino]octanoyl]piperidin-4-yl]indol-6-yl]methyl]-1-methylazetidine-3-carboxamide	CN1CC(C(=O)NCC2=CC3=C(C=C2)C(C2=CC=CC(C(N)=S)=C2)=CN3C2CCN(C(=O)CCCCCCCNC(=O)COC3=CC=CC4=C3CN(C3CCC(=O)NC3=O)C4=O)CC2)C1	C49H58N8O7S	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-EJKBS5	SCHEMBL20995466	N-[[6-amino-3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-7-yl]methyl]-8-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]oxy]acetyl]amino]octanamide; XUAGCVOYWURTRM-UHFFFAOYSA-N; N-[[6-amino-3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-7-yl]methyl]-8-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]oxy]acetyl]amino]octanamide	NC(=S)C1=CC(C2=CN(C3CCC(F)(F)CC3)C3=C2C=CC(N)=C3CNC(=O)CCCCCCCNC(=O)COC2=C3CN(C4CCC(=O)NC4=O)C(=O)C3=CC=C2)=CC=C1	C45H51F2N7O6S	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-M47CO1	SCHEMBL20996242	N-[9-[6-amino-3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-7-yl]oxynonyl]-2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]oxy]acetamide; PBABHXABKFVWEG-UHFFFAOYSA-N; N-[9-[6-amino-3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-7-yl]oxynonyl]-2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]oxy]acetamide	NC(=S)C1=CC(C2=CN(C3CCC(F)(F)CC3)C3=C2C=CC(N)=C3OCCCCCCCCCNC(=O)COC2=C3CN(C4CCC(=O)NC4=O)C(=O)C3=CC=C2)=CC=C1	C45H52F2N6O6S	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-3GOK2D	SCHEMBL20996908	N-[9-[[6-amino-3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-7-yl]amino]nonyl]-2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]oxy]acetamide; CVFUYAFHDIAEJJ-UHFFFAOYSA-N; N-[9-[[6-amino-3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-7-yl]amino]nonyl]-2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]oxy]acetamide	NC(=S)C1=CC(C2=CN(C3CCC(F)(F)CC3)C3=C2C=CC(N)=C3NCCCCCCCCCNC(=O)COC2=C3CN(C4CCC(=O)NC4=O)C(=O)C3=CC=C2)=CC=C1	C45H53F2N7O5S	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-NKDAQH	SCHEMBL20994719	N-[7-[[6-amino-3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-7-yl]methylsulfamoyl]heptyl]-2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]oxy]acetamide; MOUDGGUUKWYIAB-UHFFFAOYSA-N; N-[7-[[6-amino-3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-7-yl]methylsulfamoyl]heptyl]-2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]oxy]acetamide	NC(=S)C1=CC(C2=CN(C3CCC(F)(F)CC3)C3=C2C=CC(N)=C3CNS(=O)(=O)CCCCCCCNC(=O)COC2=C3CN(C4CCC(=O)NC4=O)C(=O)C3=CC=C2)=CC=C1	C44H51F2N7O7S2	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-L4WBLD	SCHEMBL20995467	N-[8-[[6-amino-3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-7-yl]methoxy]octyl]-2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]oxy]acetamide; YKFSRBUXRFVTQE-UHFFFAOYSA-N; N-[8-[[6-amino-3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-7-yl]methoxy]octyl]-2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]oxy]acetamide	NC(=S)C1=CC(C2=CN(C3CCC(F)(F)CC3)C3=C2C=CC(N)=C3COCCCCCCCCNC(=O)COC2=C3CN(C4CCC(=O)NC4=O)C(=O)C3=CC=C2)=CC=C1	C45H52F2N6O6S	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-B3JR7K	SCHEMBL20996867	N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-9-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]acetyl]amino]nonanamide; BHRNVFIMYVDYLY-UHFFFAOYSA-N; N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-9-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]acetyl]amino]nonanamide	NC(=S)C1=CC(C2=CN(C3CCC(F)(F)CC3)C3=C2C=CC(NC(=O)CCCCCCCCNC(=O)CNC2=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C2)=C3)=CC=C1	C45H49F2N7O6S	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-RU88BO	SCHEMBL20995471	N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-9-[[2-[2-(2,7-dioxoazepan-3-yl)-1,3-dioxoisoindol-4-yl]oxyacetyl]amino]nonanamide; LJBYTPHFWUOCNM-UHFFFAOYSA-N; N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-9-[[2-[2-(2,7-dioxoazepan-3-yl)-1,3-dioxoisoindol-4-yl]oxyacetyl]amino]nonanamide	NC(=S)C1=CC(C2=CN(C3CCC(F)(F)CC3)C3=C2C=CC(NC(=O)CCCCCCCCNC(=O)COC2=C4C(=O)N(C5CCCC(=O)NC5=O)C(=O)C4=CC=C2)=C3)=CC=C1	C46H50F2N6O7S	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-K8A2DW	SCHEMBL20994718	N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-9-[[2-[2-(2,7-dioxoazepan-4-yl)-1,3-dioxoisoindol-4-yl]oxyacetyl]amino]nonanamide; KLBLTIHMVDTDBM-UHFFFAOYSA-N; N-[3-(3-carbamothioylphenyl)-1-(4,4-difluorocyclohexyl)indol-6-yl]-9-[[2-[2-(2,7-dioxoazepan-4-yl)-1,3-dioxoisoindol-4-yl]oxyacetyl]amino]nonanamide	NC(=S)C1=CC(C2=CN(C3CCC(F)(F)CC3)C3=C2C=CC(NC(=O)CCCCCCCCNC(=O)COC2=C4C(=O)N(C5CCC(=O)NC(=O)C5)C(=O)C4=CC=C2)=C3)=CC=C1	C46H50F2N6O7S	ASH1L	Q9NR48	CRBN	WO-2019094772-A1
TPD-CHECP9	WO2019148055A1_1	.	CC1(C)C(=O)N(C2=CC(C(F)(F)F)=C(C#N)C=C2)C(=S)N1C1=CC=C(OCCCOCCOCCOCCNC2=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=CC=C2)C=C1	C41H41F3N6O9S	BRD4	O60885	CRBN	WO-2019148055-A1
TPD-FRXT5L	SCHEMBL17162073	4-[3-[4-[3-[3-[2-[[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]propoxy]propoxy]phenyl]-4,4-dimethyl-5-oxo-2-sulfanylideneimidazolidin-1-yl]-2-(trifluoromethyl)benzonitrile; SCHEMBL30185468; MNISJDGXRPGROH-UHFFFAOYSA-N; 4-[3-[4-[3-[3-[2-[[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]propoxy]propoxy]phenyl]-4,4-dimethyl-5-oxo-2-sulfanylideneimidazolidin-1-yl]-2-(trifluoromethyl)benzonitrile	CC1(C)C(=O)N(C2=CC(C(F)(F)F)=C(C#N)C=C2)C(=S)N1C1=CC=C(OCCCOCCCOCCNC2=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=CC=C2)C=C1	C40H39F3N6O8S	BRD4	O60885	CRBN	WO-2019148055-A1
TPD-YW80RK	WO2019148055A1_3	.	CC1(C)C(=O)N(C2=CC(C(F)(F)F)=C(C#N)C=C2)C(=S)N1C1=CC=C(OCCOCCOCCOCCNC2=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=CC=C2)C=C1	C40H39F3N6O9S	BRD4	O60885	CRBN	WO-2019148055-A1
TPD-4QXMN8	WO2019148055A1_6	.	CC1(C)C(=O)N(C2=CC(C(F)(F)F)=C(C#N)C=C2)C(=S)N1C1=CC=C(OCCOCCOCCOCCOCCNC2=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=CC=C2)C=C1	C42H43F3N6O10S	BRD4	O60885	CRBN	WO-2019148055-A1
TPD-Q7DT7S	WO2019148055A1_7	.	C=C1C2=CC=CC(N(C)CCN(C)CCOC3=CC=C(N4C(=O)N(C5=CC(/C=C\C)=C(C#N)C=N5)C(=O)C4(C)C)C=C3)=C2C(=O)N1C1CCC(=O)NC1=O	C40H42N8O6	BRD4	O60885	CRBN	WO-2019148055-A1
TPD-EQN8G7	SCHEMBL17162108	4-[3-[4-[2-[2-[2-[[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]phenyl]-4,4-dimethyl-5-oxo-2-sulfanylideneimidazolidin-1-yl]-2-(trifluoromethyl)benzonitrile; SCHEMBL30185464; WQEIGSUDCJWNEH-UHFFFAOYSA-N; 4-[3-[4-[2-[2-[2-[[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]phenyl]-4,4-dimethyl-5-oxo-2-sulfanylideneimidazolidin-1-yl]-2-(trifluoromethyl)benzonitrile	CC1(C)C(=O)N(C2=CC(C(F)(F)F)=C(C#N)C=C2)C(=S)N1C1=CC=C(OCCOCCOCCNC2=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=CC=C2)C=C1	C38H35F3N6O8S	BRD4	O60885	CRBN	WO-2019148055-A1
TPD-M7VOO6	SCHEMBL17162045	4-[3-[4-[3-[2-[2-[[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]propoxy]phenyl]-4,4-dimethyl-5-oxo-2-sulfanylideneimidazolidin-1-yl]-2-(trifluoromethyl)benzonitrile; SCHEMBL31348243; WINHYUVKLDGXAY-UHFFFAOYSA-N; 4-[3-[4-[3-[2-[2-[[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]propoxy]phenyl]-4,4-dimethyl-5-oxo-2-sulfanylideneimidazolidin-1-yl]-2-(trifluoromethyl)benzonitrile	CC1(C)C(=O)N(C2=CC(C(F)(F)F)=C(C#N)C=C2)C(=S)N1C1=CC=C(OCCCOCCOCCNC2=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=CC=C2)C=C1	C39H37F3N6O8S	BRD4	O60885	CRBN	WO-2019148055-A1
TPD-X3IH1M	SCHEMBL17162106	4-[3-[4-[4-[2-[2-[2-[[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]butoxy]phenyl]-4,4-dimethyl-5-oxo-2-sulfanylideneimidazolidin-1-yl]-2-(trifluoromethyl)benzonitrile; SCHEMBL29474864; XEYJIDBWIHFLLZ-UHFFFAOYSA-N; 4-[3-[4-[4-[2-[2-[2-[[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]butoxy]phenyl]-4,4-dimethyl-5-oxo-2-sulfanylideneimidazolidin-1-yl]-2-(trifluoromethyl)benzonitrile	CC1(C)C(=O)N(C2=CC(C(F)(F)F)=C(C#N)C=C2)C(=S)N1C1=CC=C(OCCCCOCCOCCOCCNC2=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=CC=C2)C=C1	C42H43F3N6O9S	BRD4	O60885	CRBN	WO-2019148055-A1
TPD-E1308E	WO2019148055A1_11	.	CC1(C)C(NC(=O)C2=CC=C(OCCCCCOCCCNC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)C=C2)C(C)(C)C1OC1=CC(Cl)=C(C#N)C=N1	C42H47ClN6O8	BRD4	O60885	CRBN	WO-2019148055-A1
TPD-S36OZ5	WO2019148055A1_12	.	CC1(C)C(=O)N(C2=CC(C(F)(F)F)=C(C#N)C=C2)C(=S)N1C1=CC=C(OCCCOCCOCCOCCNC2=C3C(=O)N(C4(C)CCC(=O)NC4=O)C(=O)C3=CC=C2)C=C1	C42H43F3N6O9S	BRD4	O60885	CRBN	WO-2019148055-A1
TPD-UZWYM9	CHEMBL4448938	4-[3-[4-[4-[5-[[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]pentoxy]phenyl]phenyl]-4,4-dimethyl-5-oxo-2-sulfanylideneimidazolidin-1-yl]-2-(trifluoromethyl)benzonitrile; SCHEMBL17162105; SCHEMBL29474863; LTNVQSMHVCBXCG-UHFFFAOYSA-N; PD140930; 4-[3-[4-[4-[5-[[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]pentoxy]phenyl]phenyl]-4,4-dimethyl-5-oxo-2-sulfanylideneimidazolidin-1-yl]-2-(trifluoromethyl)benzonitrile	CC1(C)C(=O)N(C2=CC=C(C#N)C(C(F)(F)F)=C2)C(=S)N1C1=CC=C(C2=CC=C(OCCCCCNC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)C=C2)C=C1	C43H37F3N6O6S	BRD4	O60885	CRBN	WO-2019148055-A1
TPD-XQYH1W	WO2019148055A1_14	.	CC1=NN=C(N(CC(=O)NC2=CC=C(OCCOCCOCCOCCS(=O)(=O)C3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)C=C2)C(=O)CC2=CC=C(Cl)C=C2)N1C1=CC(C)=C(C)S1	C46H48ClN7O12S2	BRD4	O60885	CRBN	WO-2019148055-A1
TPD-G03D0S	SCHEMBL17169755	2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]-N-[4-[2-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]phenyl]acetamide; PD140928	CC1=NN=C2[C@H](CC(=O)NC3=CC=C(OCCOCCOCCOCCOCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C3)N=C(C3=CC=C(Cl)C=C3)C3=C(SC(C)=C3C)N12	C48H51ClN8O10S	BRD4	O60885	CRBN	WO-2019148055-A1
TPD-5YNA2K	SCHEMBL17169756	2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]-N-[4-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]phenyl]acetamide; PD140926	CC1=NN=C2[C@H](CC(=O)NC3=CC=C(OCCOCCOCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C3)N=C(C3=CC=C(Cl)C=C3)C3=C(SC(C)=C3C)N12	C44H43ClN8O8S	BRD4	O60885	CRBN	WO-2019148055-A1
TPD-0X11PG	SCHEMBL17162043	N-(3-(5-bromo-2-(4-(2-(2-(2-(2-(2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindolin-4-ylamino)ethoxy)ethoxy)ethoxy)ethoxy)phenylamino)pyrimidin-4-ylamino)propyl)-N-methylcyclobutanecarboxamide; SCHEMBL29474844; QRKKOIZEVBIEPL-UHFFFAOYSA-N; N-(3-(5-bromo-2-(4-(2-(2-(2-(2-(2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindolin-4-ylamino)ethoxy)ethoxy)ethoxy)ethoxy)phenylamino)pyrimidin-4-ylamino)propyl)-N-methylcyclobutanecarboxamide	CN(CCCNC1=NC(NC2=CC=C(OCCOCCOCCOCCNC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)C=C2)=NC=C1Br)C(=O)C1CCC1	C40H49BrN8O9	BRD4	O60885	CRBN	WO-2019148055-A1
TPD-Q6CUSH	WO2019148055A1_18	.	N#CC1=C(NCCCNC(=O)C2CCC2)N=C(NC2=CC=C(OCCOCCOCCOCCOCCOCCNC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)C=C2)N=C1	C44H55N9O11	BRD4	O60885	CRBN	WO-2019148055-A1
TPD-ZOR6UT	WO2019148055A1_19	.	N#CC1=CC=C(NC2=CC=C(OCCOCCOCCOCCOCCNC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)C=C2)N=C1NCCCNC(=O)C1CCC1	C43H52N8O10	BRD4	O60885	CRBN	WO-2019148055-A1
TPD-G6M1YQ	SCHEMBL17162082	4-[4-[(Z)-[3-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethyl]-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl]-2-methoxyphenoxy]-3-(trifluoromethyl)benzonitrile; SCHEMBL29474866; QIBFIGPKOZNXAE-QRQIAZFYSA-N; 4-[4-[(Z)-[3-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethyl]-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl]-2-methoxyphenoxy]-3-(trifluoromethyl)benzonitrile	COC1=CC(/C=C2\SC(=O)N(CCOCCNC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)C2=O)=CC=C1OC1=C(C(F)(F)F)C=C(C#N)C=C1	C36H28F3N5O9S	BRD4	O60885	CRBN	WO-2019148055-A1
TPD-1M2C1L	WO2019148055A1_22	.	COC1=CC(/C=C2\SC(=O)N(CCOCCOCCNC3=CC=CC4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)C2=O)=CC=C1OC1=C(C(F)(F)F)C=C(C#N)C=C1	C38H32F3N5O10S	BRD4	O60885	CRBN	WO-2019148055-A1
TPD-RK2WQQ	WO2019148055A1_23	.	CC1=NN=C2[C@H](CC(=O)N[C@@H](C)C3=CC=C(C#CCCCCNC4=CC=CC5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)C=C3)N=C(C3=CC=C(Cl)C=C3)C3=C(SC(C)=C3C)N12	C46H43ClN8O5S	BRD4	O60885	CRBN	WO-2019148055-A1
TPD-PGDYVT	SCHEMBL17174615	2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]-N-[3-[3-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]propoxy]propyl]acetamide; SCHEMBL29457005	CC1=NN=C2[C@H](CC(=O)NCCCOCCCNC3=CC=CC4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)N=C(C3=CC=C(Cl)C=C3)C3=C(SC(C)=C3C)N12	C38H39ClN8O6S	BRD4	O60885	CRBN	WO-2019148055-A1
TPD-ZG8WMN	SCHEMBL17174036	2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]-N-[3-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]propyl]acetamide; SCHEMBL29456991	CC1=NN=C2[C@H](CC(=O)NCCCNC3=CC=CC4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)N=C(C3=CC=C(Cl)C=C3)C3=C(SC(C)=C3C)N12	C35H33ClN8O5S	BRD4	O60885	CRBN	WO-2019148055-A1
TPD-X68XVU	WO2019148055A1_26	.	CC1=NN=C2[C@H](CC(=O)NC(=O)C3=CC=C(OCCOCCNC4=CC=CC5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)C=C3)N=C(C3=CC=C(Cl)C=C3)C3=C(SC(C)=C3C)N12	C43H39ClN8O8S	BRD4	O60885	CRBN	WO-2019148055-A1
TPD-V56Z7W	SCHEMBL17173843	2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]-N-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethyl]acetamide; SCHEMBL29456986; PD140919	CC1=NN=C2[C@H](CC(=O)NCCOCCNC3=CC=CC4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)N=C(C3=CC=C(Cl)C=C3)C3=C(SC(C)=C3C)N12	C36H35ClN8O6S	BRD4	O60885	CRBN	WO-2019148055-A1
TPD-4I2BFQ	WO2019148055A1_28	.	CC1=NN=C2[C@H](CC(=O)NC(=O)C3=CC=C(OCCCCN(C)C4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C3)N=C(C3=CC=C(C#N)C=C3)C3=C(SC(C)=C3C)N12	C45H41N9O7S	BRD4	O60885	CRBN	WO-2019148055-A1
TPD-VEO89V	WO2019148055A1_29	.	CC1=NN=C2[C@H](CC(=O)NC(C)C3=CC=C(C#CCCOCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C3)N=C(C3=CC=C(Cl)C=C3)C3=C(SC(C)=C3C)N12	C46H43ClN8O6S	BRD4	O60885	CRBN	WO-2019148055-A1
TPD-RGL40H	WO2019148055A1_30	.	CC1=NN=C2[C@H](CC(=O)N[C@H](C)C3=CC=C(OCCCS(=O)(=O)C4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C3)N=C(C3=CC=C(Cl)C=C3)C3=C(SC(C)=C3C)N12	C43H40ClN7O8S2	BRD4	O60885	CRBN	WO-2019148055-A1
TPD-3BIJH7	WO2019148055A1_31	.	CC1=NN=C2[C@H](CC(=O)NC3=CC=C(C4=CC=C(OCCCNC5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)C=C4)N=C3)N=C(C3=CC=C(Cl)C=C3)C3=C(SC(C)=C3C)N12	C46H40ClN9O6S	BRD4	O60885	CRBN	WO-2019148055-A1
TPD-6OY8AN	WO2019148055A1_32	.	CC1=NN=C(SCC(=O)NC2=CC(F)=C(OCCCOCCNC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)C=C2)N1C1=C(C(=O)C2=CC=C(C#N)C=C2)C(C)=C(C)S1	C43H39FN8O8S2	BRD4	O60885	CRBN	WO-2019148055-A1
TPD-D4X5SF	SCHEMBL17169767	2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]-N-[4-[4-[3-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]propoxy]butoxy]-2-fluorophenyl]acetamide; SCHEMBL29457002	CC1=NN=C2[C@H](CC(=O)NC3=CC=C(OCCCCOCCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C3F)N=C(C3=CC=C(Cl)C=C3)C3=C(SC(C)=C3C)N12	C45H44ClFN8O7S	BRD4	O60885	CRBN	WO-2019148055-A1
TPD-9TTUXC	SCHEMBL17169763	2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]-N-[4-[4-[3-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]propoxy]butoxy]-3-fluorophenyl]acetamide	CC1=NN=C2[C@H](CC(=O)NC3=CC=C(OCCCCOCCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C(F)=C3)N=C(C3=CC=C(Cl)C=C3)C3=C(SC(C)=C3C)N12	C45H44ClFN8O7S	BRD4	O60885	CRBN	WO-2019148055-A1
TPD-9AGP2S	SCHEMBL17162078	2-[(9R)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]-N-[4-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethoxy]phenyl]acetamide; SCHEMBL29457003	CC1=NN=C2[C@@H](CC(=O)NC3=CC=C(OCCOCCOCCOCCNC4=C5CN(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C3)N=C(C3=CC=C(Cl)C=C3)C3=C(SC(C)=C3C)N12	C46H49ClN8O8S	BRD4	O60885	CRBN	WO-2019148055-A1
TPD-C797H6	WO2019148055A1_36	.	CC1=C(C)C2=C(S1)N1C=NN=C1[C@H](CC(=O)N[C@@H](C)C1=CC=C(C3=NC=C(OCCOCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=N3)C=C1)N=C2C1=CC=C(Cl)C=C1	C47H43ClN10O7S	BRD4	O60885	CRBN	WO-2019148055-A1
TPD-GBDRD0	WO2019148055A1_37	.	CC(=O)NC(=O)C(C)N1C(=O)C2=CC=CC(NCCOCCOCCNC(=O)C[C@@H]3N=C(C4=CC=C(Cl)C=C4)C4=C(SC(C)=C4C)N4C(C)=NN=C34)=C2C1=O	C38H41ClN8O7S	BRD4	O60885	CRBN	WO-2019148055-A1
TPD-99WQ2W	SCHEMBL17552898	2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]-N-[(1R)-1-[4-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]ethoxy]ethoxy]phenyl]ethyl]acetamide; SCHEMBL29474868	CC1=NN=C2[C@H](CC(=O)N[C@H](C)C3=CC=C(OCCOCCNC4=C5CN(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C3)N=C(C3=CC=C(Cl)C=C3)C3=C(SC(C)=C3C)N12	C44H45ClN8O6S	BRD4	O60885	CRBN	WO-2019148055-A1
TPD-PA2JAL	SCHEMBL17553349	2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]-N-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]ethoxy]ethyl]acetamide	CC1=NN=C2[C@H](CC(=O)NCCOCCNC3=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)N=C(C3=CC=C(Cl)C=C3)C3=C(SC(C)=C3C)N12	C36H37ClN8O5S	BRD4	O60885	CRBN	WO-2019148055-A1
TPD-H58IYS	SCHEMBL17536579	2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]-N-[(1S)-1-[4-[5-[3-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]propoxy]pyrimidin-2-yl]phenyl]ethyl]acetamide	CC1=NN=C2[C@H](CC(=O)N[C@@H](C)C3=CC=C(C4=NC=C(OCCCNC5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)C=N4)C=C3)N=C(C3=CC=C(Cl)C=C3)C3=C(SC(C)=C3C)N12	C47H43ClN10O6S	BRD4	O60885	CRBN	WO-2019148055-A1
TPD-KEW56D	SCHEMBL17552900	2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]-N-[(1S)-1-[4-[3-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]propoxy]phenyl]ethyl]acetamide; SCHEMBL29474836	CC1=NN=C2[C@H](CC(=O)N[C@@H](C)C3=CC=C(OCCCOCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C3)N=C(C3=CC=C(Cl)C=C3)C3=C(SC(C)=C3C)N12	C45H45ClN8O7S	BRD4	O60885	CRBN	WO-2019148055-A1
TPD-7XL0XA	WO2019148055A1_42	.	CC1=NN=C2[C@H](CC(=O)N[C@@H](C)C3=CC=C(OCCOCCNC4=C5CN(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C3)N=C(C3=CC=C(Cl)C=C3)C3=C(SC(C)=C3C)N12	C44H45ClN8O6S	BRD4	O60885	CRBN	WO-2019148055-A1
TPD-HV0CJM	SCHEMBL17553383	2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]-N-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]butyl]acetamide; SCHEMBL29474823	CC1=NN=C2[C@H](CC(=O)NCCCCNC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)N=C(C3=CC=C(Cl)C=C3)C3=C(SC(C)=C3C)N12	C36H35ClN8O5S	BRD4	O60885	CRBN	WO-2019148055-A1
TPD-D1934C	SCHEMBL17553409	2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]-N-[5-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]pentyl]acetamide; SCHEMBL29474853	CC1=NN=C2[C@H](CC(=O)NCCCCCNC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)N=C(C3=CC=C(Cl)C=C3)C3=C(SC(C)=C3C)N12	C37H37ClN8O5S	BRD4	O60885	CRBN	WO-2019148055-A1
TPD-22KB62	SCHEMBL17553401	2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]-N-[3-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]propyl]acetamide; SCHEMBL29474830	CC1=NN=C2[C@H](CC(=O)NCCCNC3=CC=CC4=C3CN(C3CCC(=O)NC3=O)C4=O)N=C(C3=CC=C(Cl)C=C3)C3=C(SC(C)=C3C)N12	C35H35ClN8O4S	BRD4	O60885	CRBN	WO-2019148055-A1
TPD-IMZ3X6	SCHEMBL17553382	2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]-N-[4-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]butyl]acetamide; SCHEMBL29474862	CC1=NN=C2[C@H](CC(=O)NCCCCNC3=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)N=C(C3=CC=C(Cl)C=C3)C3=C(SC(C)=C3C)N12	C36H37ClN8O4S	BRD4	O60885	CRBN	WO-2019148055-A1
TPD-MVIZFI	SCHEMBL26846785	2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]-N-[(1S)-1-[4-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]-3-fluorophenyl]ethyl]acetamide; SCHEMBL29474858	CC1=NN=C2[C@H](CC(=O)N[C@@H](C)C3=CC(F)=C(OCCOCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C3)N=C(C3=CC=C(Cl)C=C3)C3=C(SC(C)=C3C)N12	C44H42ClFN8O7S	BRD4	O60885	CRBN	WO-2019148055-A1
TPD-R4ZJFK	SCHEMBL17553347	2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]-N-[4-[2-[2-[2-[2-[[2-(3-methyl-2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethoxy]phenyl]acetamide; SCHEMBL29474859	CC1=NN=C2[C@H](CC(=O)NC3=CC=C(OCCOCCOCCOCCNC4=C5C(=O)N(C6(C)CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C3)N=C(C3=CC=C(Cl)C=C3)C3=C(SC(C)=C3C)N12	C47H49ClN8O9S	BRD4	O60885	CRBN	WO-2019148055-A1
TPD-W9F5W4	SCHEMBL17553350	2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]-N-[4-[2-[2-[2-[2-[[2-(1-methyl-2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethoxy]phenyl]acetamide; SCHEMBL29474867	CC1=NN=C2[C@H](CC(=O)NC3=CC=C(OCCOCCOCCOCCNC4=C5C(=O)N(C6CCC(=O)N(C)C6=O)C(=O)C5=CC=C4)C=C3)N=C(C3=CC=C(Cl)C=C3)C3=C(SC(C)=C3C)N12	C47H49ClN8O9S	BRD4	O60885	CRBN	WO-2019148055-A1
TPD-1FIRBF	SCHEMBL17552903	2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]-N-[(1R)-1-[3-[3-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]propoxy]phenyl]ethyl]acetamide; SCHEMBL29474845	CC1=NN=C2[C@H](CC(=O)N[C@H](C)C3=CC=CC(OCCCNC4=CC=CC5=C4CN(C4CCC(=O)NC4=O)C5=O)=C3)N=C(C3=CC=C(Cl)C=C3)C3=C(SC(C)=C3C)N12	C43H43ClN8O5S	BRD4	O60885	CRBN	WO-2019148055-A1
TPD-NT8MWE	WO2019148055A1_52	.	CC1=C(C)C2=C(S1)N1N=NN=C1[C@H](CC(=O)N[C@H]1CCN(C(=O)C3=CC=C(NCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C3)C1)N=C2C1=CC=C(Cl)C=C1	C43H40ClN11O6S	BRD4	O60885	CRBN	WO-2019148055-A1
TPD-P8PYDQ	SCHEMBL17553351	2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]-N-[2-[2-[[3-(2,6-dioxopiperidin-3-yl)-2-methyl-4-oxoquinazolin-5-yl]amino]ethoxy]ethyl]acetamide	CC1=NN=C2[C@H](CC(=O)NCCOCCNC3=C4C(=O)N(C5CCC(=O)NC5=O)C(C)=NC4=CC=C3)N=C(C3=CC=C(Cl)C=C3)C3=C(SC(C)=C3C)N12	C37H38ClN9O5S	BRD4	O60885	CRBN	WO-2019148055-A1
TPD-QRDDCM	WO2019148055A1_54	.	CC1=NN=C2[C@H](CC(=O)NCCCOCCCNC3=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)N=C(C3=CC=C(Cl)C=C3)C3=C(SC(C)=C3C)N12	C38H41ClN8O5S	BRD4	O60885	CRBN	WO-2019148055-A1
TPD-CWOPWX	SCHEMBL17552905	2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]-N-[(3S)-1-[4-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]benzoyl]pyrrolidin-3-yl]acetamide; SCHEMBL29474834	CC1=NN=C2[C@H](CC(=O)N[C@H]3CCN(C(=O)C4=CC=C(OCCNC5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)C=C4)C3)N=C(C3=CC=C(Cl)C=C3)C3=C(SC(C)=C3C)N12	C45H42ClN9O7S	BRD4	O60885	CRBN	WO-2019148055-A1
TPD-SH7Q3G	SCHEMBL17553392	2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]-N-[4-[2-[2-[2-[[3-(2,6-dioxopiperidin-3-yl)-2-methyl-4-oxoquinazolin-5-yl]amino]ethoxy]ethoxy]ethoxy]phenyl]acetamide	CC1=NN=C2[C@H](CC(=O)NC3=CC=C(OCCOCCOCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(C)=NC5=CC=C4)C=C3)N=C(C3=CC=C(Cl)C=C3)C3=C(SC(C)=C3C)N12	C45H46ClN9O7S	BRD4	O60885	CRBN	WO-2019148055-A1
TPD-9XJF14	SCHEMBL21331489	2-[2-[4-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]ethoxy]-N-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]acetamide; PD140765	NC1=C2C(C3=CC=C(OC4=CC=CC=C4)C=C3)=NN(C3CCN(CCOCC(=O)NC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)C2=NC=N1	C39H37N9O7	BTK	Q06187	CRBN	WO-2019177902-A1
TPD-L4B7H0	SCHEMBL21331490	2-[2-[2-[4-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]ethoxy]ethoxy]-N-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]acetamide; PD140767	NC1=NC=NC2=C1C(C1=CC=C(OC3=CC=CC=C3)C=C1)=NN2C1CCN(CCOCCOCC(=O)NC2=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=CC=C2)CC1	C41H41N9O8	BTK	Q06187	CRBN	WO-2019177902-A1
TPD-9EM6AI	SCHEMBL21331493	3-[3-[3-[4-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propoxy]propoxy]-N-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]propanamide; MT-781	NC1=C2C(C3=CC=C(OC4=CC=CC=C4)C=C3)=NN(C3CCN(CCCOCCCOCCC(=O)NC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)C2=NC=N1	C44H47N9O8	BTK	Q06187	CRBN	WO-2019177902-A1
TPD-J5K807	WO2019177902A1_104	.	NC1=NC=NC2=C1C(C1=CC=C(OC3=CC=CC=C3)C=C1)=NN2C1CCN(CCCCCCOCCOCC(=O)NC2=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=CC=C2)CC1	C45H49N9O8	BTK	Q06187	CRBN	WO-2019177902-A1
TPD-CGO2NU	SCHEMBL21331475	2-[4-[4-[4-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]butoxy]butoxy]-N-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]acetamide; MT-809	NC1=NC=NC2=C1C(C1=CC=C(OC3=CC=CC=C3)C=C1)=NN2C1CCN(CCCCOCCCCOCC(=O)NC2=CC=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=C2)CC1	C45H49N9O8	BTK	Q06187	CRBN	WO-2019177902-A1
TPD-MQR5Y6	SCHEMBL21331478	2-[4-[4-[4-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]butoxy]butoxy]-N-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]acetamide; MT-541	NC1=NC=NC2=C1C(C1=CC=C(OC3=CC=CC=C3)C=C1)=NN2C1CCN(CCCCOCCCCOCC(=O)NC2=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=CC=C2)CC1	C45H49N9O8	BTK	Q06187	CRBN	WO-2019177902-A1
TPD-VMCKYP	SCHEMBL21331535	2-[6-[6-[4-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]hexoxy]hexoxy]-N-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]acetamide	NC1=NC=NC2=C1C(C1=CC=C(OC3=CC=CC=C3)C=C1)=NN2C1CCN(CCCCCCOCCCCCCOCC(=O)NC2=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=CC=C2)CC1	C49H57N9O8	BTK	Q06187	CRBN	WO-2019177902-A1
TPD-O9AAF5	WO2019177902A1_110	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C(OCCOCC(=O)N3CCC(N4N=C(C5=CC=C(OC6=CC=CC=C6)C=C5)C5=C4N=CN=C5N)CC3)=C2)SC=N1	C55H58N10O8S	BTK	Q06187	VHL	WO-2019177902-A1
TPD-HEJK75	SCHEMBL21341774	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[2-[2-[4-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]ethoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOCCN3CCC(N4N=C(C5=CC=C(OC6=CC=CC=C6)C=C5)C5=C4N=CN=C5N)CC3)C(C)(C)C)C=C2)SC=N1	C54H68N10O9S	BTK	Q06187	VHL	WO-2019177902-A1
TPD-SUOPI3	WO2019177902A1_112	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCCCCCN3CCC(N4N=C(C5=CC=C(OC6=CC=CC=C6)C=C5)C5=C4N=CN=C5N)CC3)C(C)(C)C)C=C2)SC=N1	C56H72N10O8S	BTK	Q06187	VHL	WO-2019177902-A1
TPD-MG2WPK	SCHEMBL21331503	(2S,4R)-1-[(2S)-2-[[2-[5-[6-[4-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]hexoxy]pentoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCCOCCCCCCN3CCC(N4N=C(C5=CC=C(OC6=CC=CC=C6)C=C5)C5=C4N=CN=C5N)CC3)C(C)(C)C)C=C2)SC=N1	C57H74N10O7S	BTK	Q06187	VHL	WO-2019177902-A1
TPD-19Q570	SCHEMBL21341886	(2S,4R)-1-[(2S)-2-[6-[2-[6-[4-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]hexoxy]ethoxy]hexanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCOCCOCCCCCCN3CCC(N4N=C(C5=CC=C(OC6=CC=CC=C6)C=C5)C5=C(N)N=CN=C54)CC3)C(C)(C)C)C=C2)SC=N1	C58H76N10O7S	BTK	Q06187	VHL	WO-2019177902-A1
TPD-3KK4S0	SCHEMBL21341775	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[2-[4-[4-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]butoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOCCCCN3CCC(N4N=C(C5=CC=C(OC6=CC=CC=C6)C=C5)C5=C4N=CN=C5N)CC3)C(C)(C)C)C=C2)SC=N1	C56H72N10O9S	BTK	Q06187	VHL	WO-2019177902-A1
TPD-MNEW8J	SCHEMBL21341896	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[2-[2-[4-[4-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]cyclohexyl]piperazin-1-yl]ethoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOCCN3CCN(C4CCC(N5N=C(C6=CC=C(OC7=CC=CC=C7)C=C6)C6=C5N=CN=C6N)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C59H77N11O9S	BTK	Q06187	VHL	WO-2019177902-A1
TPD-8F9UX4	SCHEMBL21341607	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[2-[6-[4-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]hexoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOCCCCCCN3CCC(N4N=C(C5=CC=C(OC6=CC=CC=C6)C=C5)C5=C4N=CN=C5N)CC3)C(C)(C)C)C=C2)SC=N1	C58H76N10O9S	BTK	Q06187	VHL	WO-2019177902-A1
TPD-4THP5A	SCHEMBL21342083	(2S,4R)-1-[(2S)-2-[6-[2-[2-[6-[4-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]hexoxy]ethoxy]ethoxy]hexanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCOCCOCCOCCCCCCN3CCC(N4N=C(C5=CC=C(OC6=CC=CC=C6)C=C5)C5=C(N)N=CN=C54)CC3)C(C)(C)C)C=C2)SC=N1	C60H80N10O8S	BTK	Q06187	VHL	WO-2019177902-A1
TPD-D2VM6N	SCHEMBL21331530	(2S,4R)-1-[(2S)-2-[6-[5-[6-[4-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]hexoxy]pentoxy]hexanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCOCCCCCOCCCCCCN3CCC(N4N=C(C5=CC=C(OC6=CC=CC=C6)C=C5)C5=C(N)N=CN=C54)CC3)C(C)(C)C)C=C2)SC=N1	C61H82N10O7S	BTK	Q06187	VHL	WO-2019177902-A1
TPD-SDH52Q	WO2019177902A1_120	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOCCOCCCCCCN3CCC(N4N=C(C5=CC=C(OC6=CC=CC=C6)C=C5)C5=C(N)N=CN=C54)CC3)C(C)C)C=C2)SC=N1	C59H78N10O10S	BTK	Q06187	VHL	WO-2019177902-A1
TPD-KSSSYT	WO2019177902A1_121	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCOCCOCCOCCOCCCCCCN3CCC(N4N=C(C5=CC=C(OC6=CC=CC=C6)C=C5)C5=C(N)N=CN=C54)CC3)C(C)(C)C)C=C2)SC=N1	C63H86N10O9S	BTK	Q06187	VHL	WO-2019177902-A1
TPD-WCU1J0	SCHEMBL21341601	(2S,4R)-1-[(2S)-2-[6-[2-[2-[2-[2-[6-[4-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]hexoxy]ethoxy]ethoxy]ethoxy]ethoxy]hexanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCOCCOCCOCCOCCOCCCCCCN3CCC(N4N=C(C5=CC=C(OC6=CC=CC=C6)C=C5)C5=C(N)N=CN=C54)CC3)C(C)(C)C)C=C2)SC=N1	C64H88N10O10S	BTK	Q06187	VHL	WO-2019177902-A1
TPD-61GMK6	SCHEMBL21341892	3-[3-[3-[4-[4-amino-3-[4-phenoxy-3-(prop-2-enoylamino)phenyl]pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propoxy]propoxy]-N-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]propanamide	C=CC(=O)NC1=C(OC2=CC=CC=C2)C=CC(C2=NN(C3CCN(CCCOCCCOCCC(=O)NC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)C3=NC=NC(N)=C23)=C1	C47H50N10O9	BTK	Q06187	CRBN	WO-2019177902-A1
TPD-SSA3YH	SCHEMBL21341893	N-[5-[4-amino-1-[1-[4-[4-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]-2-oxoethoxy]butoxy]butyl]piperidin-4-yl]pyrazolo[3,4-d]pyrimidin-3-yl]-2-phenoxyphenyl]prop-2-enamide	C=CC(=O)NC1=C(OC2=CC=CC=C2)C=CC(C2=NN(C3CCN(CCCCOCCCCOCC(=O)NC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)C3=C2C(N)=NC=N3)=C1	C48H52N10O9	BTK	Q06187	CRBN	WO-2019177902-A1
TPD-A2YF3E	SCHEMBL21341602	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[6-[4-[4-amino-3-[4-phenoxy-3-(prop-2-enoylamino)phenyl]pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]hexoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	C=CC(=O)NC1=C(OC2=CC=CC=C2)C=CC(C2=NN(C3CCN(CCCCCCOCCOCCOCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)NCC4=CC=C(C5=C(C)N=CS5)C=C4)C(C)(C)C)CC3)C3=NC=NC(N)=C23)=C1	C59H75N11O9S	BTK	Q06187	VHL	WO-2019177902-A1
TPD-T6J4IH	WO2020035049A1_C001	.	CC(C)C1=C2N=C(NCCCCCCN)C=C(NCC3=CC=C(CCCCCCNC(=O)COC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C3)N2N=C1	C43H55N9O6	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-JFV51J	WO2020035049A1_C002	.	CC(C)C1=C2N=C(NCCCCCCN)C=C(NCC3=CC(CCCCCCNC(=O)COC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)=CC=C3)N2N=C1	C43H55N9O6	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-7E70CI	CHEMBL4867830	2-(2,6-Dioxopiperidin-3-yl)-4-[7-[4-[[[2-(1-methylpiperidin-4-yl)oxy-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]phenyl]heptoxy]isoindole-1,3-dione; SCHEMBL21741600; PD172406	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(CCCCCCCOC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C3)N2N=C1	C41H50N8O6	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-BAKKET	WO2020035049A1_C004	.	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(CCCOCCOCCOC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C3)N2N=C1	C41H50N8O8	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-GBTRDQ	WO2020035049A1_C005	.	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(CCCCCCOC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C3N(C)C)N2N=C1	C42H53N9O6	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-0U73VO	SCHEMBL21741578	4-[6-[3-(Dimethylamino)-2-[[[2-(1-methylpiperidin-4-yl)oxy-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]phenyl]hexoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=C(N(C)C)C=CC=C3CCCCCCOC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)N2N=C1	C42H53N9O6	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-OOA4M5	CHEMBL4865385	4-[7-[3-(Dimethylamino)-4-[[[2-(1-methylpiperidin-4-yl)oxy-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]phenyl]heptoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione; SCHEMBL21741581; PD172400	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(CCCCCCCOC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C3N(C)C)N2N=C1	C43H55N9O6	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-J5UI4O	CHEMBL4850062	4-[7-[2-(Dimethylamino)-3-[[[2-(1-methylpiperidin-4-yl)oxy-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]phenyl]heptoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione; SCHEMBL21741580; PD172399	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=C(N(C)C)C(CCCCCCCOC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)=CC=C3)N2N=C1	C43H55N9O6	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-FNCT8Q	SCHEMBL21741591	4-[6-[3-(Dimethylamino)-4-[[[2-(1-methylpiperidin-4-yl)oxy-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]phenyl]hexylamino]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(CCCCCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C3N(C)C)N2N=C1	C42H54N10O5	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-A6D5GL	CHEMBL4855880	N-[6-[3-(dimethylamino)-4-[[[2-(1-methylpiperidin-4-yl)oxy-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]phenyl]hexyl]-2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyacetamide; PD172394	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(CCCCCCNC(=O)COC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C3N(C)C)N2N=C1	C44H56N10O7	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-799D5C	CHEMBL4849856	N-[6-[4-(dimethylamino)-3-[[[2-(1-methylpiperidin-4-yl)oxy-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]phenyl]hexyl]-2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyacetamide; SCHEMBL21741602; PD172395	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC(CCCCCCNC(=O)COC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)=CC=C3N(C)C)N2N=C1	C44H56N10O7	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-GTUZDD	WO2020035049A1_C012	.	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(NC(=O)CCCCCCNC(=O)COC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C3)N2N=C1	C43H52N10O8	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-L3ZN3U	CHEMBL4853149	7-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyacetyl]amino]-N-[3-[[[2-(1-methylpiperidin-4-yl)oxy-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]phenyl]heptanamide; SCHEMBL21741579; PD172401	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC(NC(=O)CCCCCCNC(=O)COC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)=CC=C3)N2N=C1	C43H52N10O8	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-7VK6BZ	CHEMBL4873076	N-[4-(dimethylamino)-3-[[[2-(1-methylpiperidin-4-yl)oxy-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]phenyl]-7-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyacetyl]amino]heptanamide; PD172397	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC(NC(=O)CCCCCCNC(=O)COC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)=CC=C3N(C)C)N2N=C1	C45H57N11O8	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-WPMAZV	CHEMBL4871849	N-[3-(dimethylamino)-4-[[[2-(1-methylpiperidin-4-yl)oxy-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]phenyl]-7-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyacetyl]amino]heptanamide; PD172396	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(NC(=O)CCCCCCNC(=O)COC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C3N(C)C)N2N=C1	C45H57N11O8	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-CYHA8G	WO2020035049A1_C016	.	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(NC(=O)CCCCCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C3N(C)C)N2N=C1	C43H55N11O6	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-HS3SIA	CHEMBL4877871	7-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]-N-[4-[[[2-(1-methylpiperidin-4-yl)oxy-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]phenyl]heptanamide; SCHEMBL21741583; PD172403	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(NC(=O)CCCCCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C3)N2N=C1	C41H50N10O6	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-F57ALN	SCHEMBL21741604	5-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxy-N-[4-[[[2-(1-methylpiperidin-4-yl)oxy-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]phenyl]pentanamide	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(NC(=O)CCCCOC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C3)N2N=C1	C39H45N9O7	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-TH8NEE	SCHEMBL21741881	5-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]oxy]-N-[4-[[[2-(1-methylpiperidin-4-yl)oxy-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]phenyl]pentanamide	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(NC(=O)CCCCOC4=C5CN(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C3)N2N=C1	C39H47N9O6	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-79UAAX	CHEMBL4849935	6-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxy-N-[4-[[[2-(1-methylpiperidin-4-yl)oxy-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]phenyl]hexanamide; PD172405	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(NC(=O)CCCCCOC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C3)N2N=C1	C40H47N9O7	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-2AH9VB	PD172416	6-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]oxy]-N-[4-[[[2-(1-methylpiperidin-4-yl)oxy-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]phenyl]hexanamide	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(NC(=O)CCCCCOC4=C5CN(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C3)N2N=C1	C40H49N9O6	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-Y8VQU2	CHEMBL4872741	7-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxy-N-[4-[[[2-(1-methylpiperidin-4-yl)oxy-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]phenyl]heptanamide; PD172404	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(NC(=O)CCCCCCOC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C3)N2N=C1	C41H49N9O7	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-LSB7XL	CHEMBL4860712	7-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]oxy]-N-[4-[[[2-(1-methylpiperidin-4-yl)oxy-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]phenyl]heptanamide; PD172415	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(NC(=O)CCCCCCOC4=C5CN(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C3)N2N=C1	C41H51N9O6	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-K0XWRB	CHEMBL4852223	8-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxy-N-[4-[[[2-(1-methylpiperidin-4-yl)oxy-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]phenyl]octanamide; PD172407	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(NC(=O)CCCCCCCOC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C3)N2N=C1	C42H51N9O7	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-96VAIY	CHEMBL4853696	8-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]oxy]-N-[4-[[[2-(1-methylpiperidin-4-yl)oxy-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]phenyl]octanamide; PD172414	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(NC(=O)CCCCCCCOC4=C5CN(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C3)N2N=C1	C42H53N9O6	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-ITQHLQ	CHEMBL4859664	9-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxy-N-[4-[[[2-(1-methylpiperidin-4-yl)oxy-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]phenyl]nonanamide; PD172408	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(NC(=O)CCCCCCCCOC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C3)N2N=C1	C43H53N9O7	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-4QTW7L	WO2020035049A1_C027	.	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(NC(=O)CCCCCCCCOC4=C5CN(C6CCC(=O)NC6=O)C(=O)C5C=CC=C4)C=C3)N2N=C1	C44H57N9O6	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-H8WDY8	WO2020035049A1_C028	.	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(NC(=O)CCCCCCCCCOC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C3)N2N=C1	C44H55N9O7	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-ZFAHSR	CHEMBL4871519	10-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]oxy]-N-[4-[[[2-(1-methylpiperidin-4-yl)oxy-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]phenyl]decanamide; PD172412	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(NC(=O)CCCCCCCCCOC4=C5CN(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C3)N2N=C1	C44H57N9O6	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-LKK76Z	SCHEMBL21741882	2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyethoxy]-N-[4-[[[2-(1-methylpiperidin-4-yl)oxy-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]phenyl]acetamide	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(NC(=O)COCCOC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C3)N2N=C1	C38H43N9O8	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-K8AJN8	CHEMBL4873421	2-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyethoxy]ethoxy]-N-[4-[[[2-(1-methylpiperidin-4-yl)oxy-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]phenyl]acetamide; PD172409	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(NC(=O)COCCOCCOC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C3)N2N=C1	C40H47N9O9	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-AXHVUS	CHEMBL4858363	2-[2-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyethoxy]ethoxy]ethoxy]-N-[4-[[[2-(1-methylpiperidin-4-yl)oxy-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]phenyl]acetamide; PD172411	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(NC(=O)COCCOCCOCCOC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C3)N2N=C1	C42H51N9O10	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-LDCG0C	WO2020035049A1_C033	8-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxy-N-[3-[[[2-(1-methylpiperidin-4-yl)oxy-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]phenyl]octanamide	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC(NC(=O)CCCCCCCOC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)=CC=C3)N2N=C1	C42H51N9O7	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-XTJGJS	WO2020035049A1_C034	.	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(NC(=O)CCCCCCCOC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C3N3C=CN=C3)N2N=C1	C45H53N11O7	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-0DXMG8	WO2020035049A1_C035	.	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=C(N(C)C)C(NC(=O)CCCCCCCOC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)=CC=C3)N2N=C1	C44H56N10O7	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-ND5CIP	SCHEMBL21741840	N-[3-(dimethylamino)-4-[[[2-(1-methylpiperidin-4-yl)oxy-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]phenyl]-8-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyoctanamide	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(NC(=O)CCCCCCCOC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C3N(C)C)N2N=C1	C44H56N10O7	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-MZA6UU	SCHEMBL21741584	8-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxy-N-[4-[[[2-[[(2R)-1-hydroxybutan-2-yl]amino]-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]phenyl]octanamide	CC[C@H](CO)NC1=NC2=C(C(C)C)C=NN2C(NCC2=CC=C(NC(=O)CCCCCCCOC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)C=C2)=N1	C40H49N9O7	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-C8CYHB	SCHEMBL21741585	8-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxy-N-[4-[[[2-[[(2S)-1-hydroxybutan-2-yl]amino]-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]phenyl]octanamide	CC[C@@H](CO)NC1=NC2=C(C(C)C)C=NN2C(NCC2=CC=C(NC(=O)CCCCCCCOC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)C=C2)=N1	C40H49N9O7	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-QXXPG2	WO2020035049A1_C039	.	CC(C)C1=C2N=C(O[C@@H]3CCCNC3)N=C(NCC3=CC=C(NC(=O)CCCCCCCOC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C3)N2N=C1	C41H49N9O7	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-ZESS7F	WO2020035049A1_C040	8-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxy-N-[4-[[[2-[(3S)-piperidin-3-yl]oxy-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]phenyl]octanamide	CC(C)C1=C2N=C(O[C@H]3CCCNC3)N=C(NCC3=CC=C(NC(=O)CCCCCCCOC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C3)N2N=C1	C41H49N9O7	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-IB054M	CHEMBL4851888	7-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]-N-[4-[[[2-(1-methylpiperidin-4-yl)oxy-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]phenyl]heptanamide; PD172417	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(NC(=O)CCCCCCC4=CC=CC5=C4CN(C4CCC(=O)NC4=O)C5=O)C=C3)N2N=C1	C41H51N9O5	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-J9RNCJ	WO2020035049A1_C042	5-[3-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]propoxy]-N-[4-[[[2-(1-methylpiperidin-4-yl)oxy-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]phenyl]pentanamide	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(NC(=O)CCCCOCCCC4=CC=CC5=C4CN(C4CCC(=O)NC4=O)C5=O)C=C3)N2N=C1	C42H53N9O6	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-LFWQNP	WO2020035049A1_C043	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCC(=O)CC3=CC=CC(CNC4=NC(OC5CCN(C)CC5)=NC5=C(C(C)C)C=NN45)=C3N(C)C)C(C)(C)C)C=C2)SC=N1	C54H75N11O6S	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-I1B7VE	WO2020035049A1_C044	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCC3=CC=CC(CNC4=NC(OC5CCN(C)CC5)=NC5=C(C(C)C)C=NN45)=C3N(C)C)C(C)(C)C)C=C2)SC=N1	C52H73N11O5S	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-KQTDDM	WO2020035049A1_C045	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCC(=O)NC3=CC=C(CNC4=NC(OC5CCN(C)CC5)=NC5=C(C(C)C)C=NN45)C=C3)C(C)(C)C)C=C2)SC=N1	C51H69N11O6S	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-Y9DOLR	WO2020035049A1_C046	.	CC1=C2C(C#N)=CNC2=C(NS(=O)(=O)C2=CC=C(CNC(=O)CCCCCCCCC(=O)NC3=CC=C(CNC4=NC(OC5CCN(C)CC5)=NC5=C(C(C)C)C=NN45)C=C3)C=C2)C=C1	C48H59N11O5S	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-JDBIPZ	WO2020035049A1_C047	.	CC1=C2C(C#N)=CNC2=C(NS(=O)(=O)C2=CC=C(CNC(=O)COCCOCC(=O)NC3=CC=C(CNC4=NC(OC5CCN(C)CC5)=NC5=C(C(C)C)C=NN45)C=C3)C=C2)C=C1	C44H51N11O7S	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-9TNHCO	WO2020035049A1_C048	.	CC1=C2C(C#N)=CNC2=C(NS(=O)(=O)C2=CC=C(CNC(=O)CCCCC(=O)NC3=CC=C(CNC4=NC(OC5CCN(C)CC5)=NC5=C(C(C)C)C=NN45)C=C3)C=C2)C=C1	C44H51N11O5S	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-6XJTFJ	SCHEMBL21741857	N-[[4-[(3-cyano-4-methyl-1H-indol-7-yl)sulfamoyl]phenyl]methyl]-N'-[4-[[[2-(1-methylpiperidin-4-yl)oxy-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]phenyl]octanediamide	CC1=CC=C(NS(=O)(=O)C2=CC=C(CNC(=O)CCCCCCC(=O)NC3=CC=C(CNC4=NC(OC5CCN(C)CC5)=NC5=C(C(C)C)C=NN45)C=C3)C=C2)C2=C1C(C#N)=CN2	C46H55N11O5S	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-IH5RIU	SCHEMBL21741636	8-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]oxy]-N-[4-[[[5-(1-methylpiperidin-4-yl)oxy-3-propan-2-ylpyrazolo[1,5-a]pyrimidin-7-yl]amino]methyl]phenyl]octanamide	CC(C)C1=C2N=C(OC3CCN(C)CC3)C=C(NCC3=CC=C(NC(=O)CCCCCCCOC4=C5CN(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C3)N2N=C1	C43H54N8O6	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-F98UMV	SCHEMBL21741639	8-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]oxy]-N-[4-[[[5-[[(2R)-1-hydroxybutan-2-yl]amino]-3-propan-2-ylpyrazolo[1,5-a]pyrimidin-7-yl]amino]methyl]phenyl]octanamide	CC[C@H](CO)NC1=NC2=C(C(C)C)C=NN2C(NCC2=CC=C(NC(=O)CCCCCCCOC3=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)C=C2)=C1	C41H52N8O6	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-4Q397G	WO2020035049A1_C052	.	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(NC(=O)CCCCOCCOC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C3)N2N=C1	C41H49N9O8	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-WJPMXR	WO2020035049A1_C053	5-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]oxy]ethoxy]-N-[4-[[[2-(1-methylpiperidin-4-yl)oxy-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]phenyl]pentanamide	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(NC(=O)CCCCOCCOC4=C5CN(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C3)N2N=C1	C41H51N9O7	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-JX3WNK	WO2020035049A1_C080	2-[2-[3-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]propoxy]ethoxy]-N-[4-[[[2-(1-methylpiperidin-4-yl)oxy-8-propylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]phenyl]acetamide	CCCC1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(NC(=O)COCCOCCCC4=C5CN(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C3)N2N=C1	C41H51N9O7	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-B8A6N9	WO2020035049A1_C082	.	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(N[C@@H](C)C3=CC=C(NC(=O)COCCOCCCC4=CC=CC5=C4CN(C4CCC(=O)NC4=O)C5=O)C=C3)N2N=C1	C42H53N9O7	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-UT13IB	WO2020035049A1_C083	2-[2-[3-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]propoxy]ethoxy]-N-[6-[[[2-(1-methylpiperidin-4-yl)oxy-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]pyridin-3-yl]acetamide	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=NC=C(NC(=O)COCCOCCCC4=C5CN(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C3)N2N=C1	C40H50N10O7	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-1RJ1H0	WO2020035049A1_C084	2-[2-[3-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]propoxy]ethoxy]-N-[5-[[[2-(1-methylpiperidin-4-yl)oxy-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]pyrimidin-2-yl]acetamide	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CN=C(NC(=O)COCCOCCCC4=C5CN(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)N=C3)N2N=C1	C39H49N11O7	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-D4L0IT	WO2020035049A1_C085	2-[2-[3-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]propoxy]ethoxy]-N-[5-[[[2-(1-methylpiperidin-4-yl)oxy-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]pyridin-2-yl]acetamide	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CN=C(NC(=O)COCCOCCCC4=C5CN(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C3)N2N=C1	C40H50N10O7	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-S24JEZ	WO2020035049A1_C086	2-[2-[3-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]propoxy]ethoxy]-N-[8-[[[2-(1-methylpiperidin-4-yl)oxy-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]quinolin-5-yl]acetamide	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(NC(=O)COCCOCCCC4=C5CN(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C4=C3N=CC=C4)N2N=C1	C44H52N10O7	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-8Q4BKG	WO2020035049A1_C087	2-[2-[3-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]propoxy]ethoxy]-N-[8-[[[2-(1-methylpiperidin-4-yl)oxy-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]isoquinolin-5-yl]acetamide	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(NC(=O)COCCOCCCC4=C5CN(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C4=C3C=NC=C4)N2N=C1	C44H52N10O7	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-7Z1UOA	WO2020035049A1_C088	.	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(NC(=O)COCCOCCCC4=C5CN(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C4=C3OCO4)N2N=C1	C42H51N9O9	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-2316NK	WO2020035049A1_C089	2-[2-[3-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]propoxy]ethoxy]-N-[4-[[[2-(1-methylpiperidin-4-yl)oxy-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]cyclohexyl]acetamide	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3CCC(NC(=O)COCCOCCCC4=CC=CC5=C4CN(C4CCC(=O)NC4=O)C5=O)CC3)N2N=C1	C41H57N9O7	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-SZ4L8W	WO2020035049A1_C090	.	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(C(=O)NCCCCCCCOC4=C5CN(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C3)N2N=C1	C42H53N9O6	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-AIEB8S	WO2020035049A1_C091	.	CC(C)C1=CN(/C(=N\C(=[N-])OC2CCN(C)CC2)NCC2=CC=C(C(=O)NCCOCCOCCCC3=CC=CC4=C3CN(C3CCC(=O)NC3=O)C4=O)C=C2)N=C1	C42H54N9O7-	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-SLSK8X	WO2020035049A1_C093	N-[5-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]pentyl]-4-[[[2-(1-methylpiperidin-4-yl)oxy-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]benzamide	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(C(=O)NCCCCCC4=CC=CC5=C4CN(C4CCC(=O)NC4=O)C5=O)C=C3)N2N=C1	C40H49N9O5	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-NNNWTC	WO2020035049A1_C095	6-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]-N-[6-[4-[[[2-(1-methylpiperidin-4-yl)oxy-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]phenyl]pyridin-3-yl]hexanamide	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(C4=NC=C(NC(=O)CCCCCC5=CC=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)C=C4)C=C3)N2N=C1	C45H52N10O5	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-VX9GKS	WO2020035049A1_C096	.	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(NC(=O)NCCCCCC4=CC=CC5=C4CN(C4CCC(=O)NC4=O)C5=O)C=C3)N2N=C1	C40H50N10O5	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-HQOIB3	WO2020035049A1_C097	.	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(NC(=O)COCCOC/C=C/C4=C5CN(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C3)N2N=C1	C41H49N9O7	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-EIHKOL	WO2020035049A1_C098	.	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(NC(=O)COCCOCCOCC#CC4=C5CN(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C3)N2N=C1	C43H51N9O8	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-WSBNW1	WO2020035049A1_C099	.	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(NC(=O)COCCOCCOCC#CC4=CC=C(F)C5=C4CN(C4CCC(=O)NC4=O)C5=O)C=C3)N2N=C1	C43H50FN9O8	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-IHSTRA	WO2020035049A1_C100	2-[2-[2-[3-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]propoxy]ethoxy]ethoxy]-N-[4-[[[2-(1-methylpiperidin-4-yl)oxy-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]phenyl]acetamide	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(NC(=O)COCCOCCOCCCC4=CC=C5C(=O)N(C6CCC(=O)NC6=O)CC5=C4)C=C3)N2N=C1	C43H55N9O8	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-PGLCMD	WO2020035049A1_C101	2-[2-[2-[3-[2-(2,6-dioxopiperidin-3-yl)-3-oxo-1H-isoindol-5-yl]propoxy]ethoxy]ethoxy]-N-[4-[[[2-(1-methylpiperidin-4-yl)oxy-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]phenyl]acetamide	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(NC(=O)COCCOCCOCCCC4=CC=C5CN(C6CCC(=O)NC6=O)C(=O)C5=C4)C=C3)N2N=C1	C43H55N9O8	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-T4ZW92	WO2020035049A1_C102	5-[3-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-pyrrolo[3,4-c]pyridin-4-yl]propoxy]-N-[4-[[[2-(1-methylpiperidin-4-yl)oxy-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]phenyl]pentanamide	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(NC(=O)CCCCOCCCC4=C5CN(C6CCC(=O)NC6=O)C(=O)C5=CC=N4)C=C3)N2N=C1	C41H52N10O6	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-P93ZXU	WO2020035049A1_C103	5-[3-[2-(2,6-dioxopiperidin-3-yl)-3-oxo-1H-pyrrolo[3,4-c]pyridin-7-yl]propoxy]-N-[4-[[[2-(1-methylpiperidin-4-yl)oxy-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]phenyl]pentanamide	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(NC(=O)CCCCOCCCC4=C5CN(C6CCC(=O)NC6=O)C(=O)C5=CN=C4)C=C3)N2N=C1	C41H52N10O6	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-WL8GJB	WO2020035049A1_C104	5-[3-[6-(2,6-dioxopiperidin-3-yl)-7-oxo-5H-pyrrolo[3,4-b]pyridin-4-yl]propoxy]-N-[4-[[[2-(1-methylpiperidin-4-yl)oxy-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]phenyl]pentanamide	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(NC(=O)CCCCOCCCC4=C5CN(C6CCC(=O)NC6=O)C(=O)C5=NC=C4)C=C3)N2N=C1	C41H52N10O6	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-X5RG0W	WO2020035049A1_C105	5-[3-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1-oxo-3H-isoindol-4-yl]propoxy]-N-[4-[[[2-(1-methylpiperidin-4-yl)oxy-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]phenyl]pentanamide	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(NC(=O)CCCCOCCCC4=C5CN(C6CCC(=O)NC6=O)C(=O)C5=CC(F)=C4)C=C3)N2N=C1	C42H52FN9O6	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-CNWZ6G	WO2020035049A1_C106	.	CC1=CC=C(NS(=O)(=O)C2=CC=C(S(=O)(=O)NCCCCCCCC(=O)NC3=CC=C(CNC4=NC(OC5CCN(C)CC5)=NC5=C(C(C)C)C=NN45)C=C3)C=C2)C2=C1C(C#N)=CN2	C45H55N11O6S2	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-MTRBCE	SCHEMBL21741640	10-[[3-[(3-cyano-4-methyl-1H-indol-7-yl)sulfamoyl]phenyl]sulfonylamino]-N-[4-[[[2-(1-methylpiperidin-4-yl)oxy-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]phenyl]decanamide	CC1=CC=C(NS(=O)(=O)C2=CC=CC(S(=O)(=O)NCCCCCCCCCC(=O)NC3=CC=C(CNC4=NC(OC5CCN(C)CC5)=NC5=C(C(C)C)C=NN45)C=C3)=C2)C2=C1C(C#N)=CN2	C47H59N11O6S2	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-56QUSH	SCHEMBL21741637	2-[2-[2-[[4-[(3-chloro-1H-indol-7-yl)sulfamoyl]phenyl]methylamino]ethoxy]ethoxy]-N-[4-[[[2-(1-methylpiperidin-4-yl)oxy-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]phenyl]acetamide	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(NC(=O)COCCOCCNCC4=CC=C(S(=O)(=O)NC5=CC=CC6=C5NC=C6Cl)C=C4)C=C3)N2N=C1	C42H51ClN10O6S	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-9Q8H5O	WO2020035049A1_C109	.	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(NC(=O)CCCCCCC(=O)NCC4=CC=C(S(=O)(=O)NC5=NC6=C(N=C5)C(Cl)=CC=C6)C=C4)C=C3)N2N=C1	C44H52ClN11O5S	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-0ZML57	WO2020035049A1_C110	.	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(NC(=O)CCCCCCCNS(=O)(=O)C4=CC=C(S(=O)(=O)NC5=NC6=C(C=CC=C6)N=C5)C=C4)C=C3)N2N=C1	C43H53N11O6S2	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-YOHUEE	WO2020035049A1_C111	.	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(NC(=O)CCCCCCCNCC4=CC=C(S(=O)(=O)NC(=O)C5=C(Cl)C=C(Cl)C=C5)S4)C=C3)N2N=C1	C41H51Cl2N9O5S2	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-8EX9B7	WO2020035049A1_C112	.	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(NC(=O)CCCCCCCNS(=O)(=O)C4=CC=C(S(=O)(=O)NC(=O)C5=CC=C(Cl)C=C5Cl)S4)C=C3)N2N=C1	C40H49Cl2N9O7S3	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-SDAGOG	WO2020035049A1_C116	3-[7-[5-[4-[4-[[[2-(1-methylpiperidin-4-yl)oxy-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]phenyl]piperazin-1-yl]pentyl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(N4CCN(CCCCCC5=CC=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)N2N=C1	C43H56N10O4	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-YKYMI8	CHEMBL4865751	4-[5-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]pentyl]-N-[4-[[[2-(1-methylpiperidin-4-yl)oxy-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]phenyl]piperazine-1-carboxamide; PD172422	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(NC(=O)N4CCN(CCCCCC5=CC=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)N2N=C1	C44H57N11O5	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-PTY3VB	WO2020035049A1_C118	.	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(NC(=O)N4CCN(CCCCC5=CC=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)N2N=C1	C43H55N11O5	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-NOMA16	WO2020035049A1_C120	N-[3,5-difluoro-4-[[[2-(1-methylpiperidin-4-yl)oxy-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]phenyl]-3-[3-[3-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]propyl]azetidin-1-yl]propanamide	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=C(F)C=C(NC(=O)CCN4CC(CCCC5=CC=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)C4)C=C3F)N2N=C1	C43H52F2N10O5	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-49076K	WO2020035049A1_C121	N-[3-cyano-4-[[[2-(1-methylpiperidin-4-yl)oxy-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]phenyl]-5-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]ethyl]pyrazol-1-yl]pentanamide	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(NC(=O)CCCCN4C=C(CCC5=CC=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)C=N4)C=C3C#N)N2N=C1	C45H52N12O5	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-LXR494	SCHEMBL21741589	N-[3-chloro-4-[[[2-(1-methylpiperidin-4-yl)oxy-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]phenyl]-2-[4-[5-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]pentyl]piperazin-1-yl]acetamide	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=C(Cl)C=C(NC(=O)CN4CCN(CCCCCC5=CC=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)N2N=C1	C45H58ClN11O5	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-T2OH9V	SCHEMBL21741587	N-[4-[[[5-(cyclopentylamino)-3-propan-2-ylpyrazolo[1,5-a]pyrimidin-7-yl]amino]methyl]phenyl]-4-[5-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]pentyl]piperazine-1-carboxamide	CC(C)C1=C2N=C(NC3CCCC3)C=C(NCC3=CC=C(NC(=O)N4CCN(CCCCCC5=CC=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)N2N=C1	C44H56N10O4	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-GVWZGH	SCHEMBL21741572	4-[5-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]pentyl]-N-[4-[[[5-(4-hydroxypiperidin-1-yl)-3-propan-2-ylpyrazolo[1,5-a]pyrimidin-7-yl]amino]methyl]phenyl]piperazine-1-carboxamide	CC(C)C1=C2N=C(N3CCC(O)CC3)C=C(NCC3=CC=C(NC(=O)N4CCN(CCCCCC5=CC=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)N2N=C1	C44H56N10O5	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-0ISBGS	SCHEMBL21741624	N-[4-[[[5-[[(2R,3R)-1,3-dihydroxybutan-2-yl]amino]-3-propan-2-ylpyrazolo[1,5-a]pyrimidin-7-yl]amino]methyl]phenyl]-4-[5-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]pentyl]piperazine-1-carboxamide	CC(C)C1=C2N=C(N[C@H](CO)[C@@H](C)O)C=C(NCC3=CC=C(NC(=O)N4CCN(CCCCCC5=C6CN(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)CC4)C=C3)N2N=C1	C43H56N10O6	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-ZA8I1B	SCHEMBL21741620	N-[4-[[[5-[[(2S,3S)-1,3-dihydroxybutan-2-yl]amino]-3-propan-2-ylpyrazolo[1,5-a]pyrimidin-7-yl]amino]methyl]phenyl]-4-[5-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]pentyl]piperazine-1-carboxamide	CC(C)C1=C2N=C(N[C@@H](CO)[C@H](C)O)C=C(NCC3=CC=C(NC(=O)N4CCN(CCCCCC5=C6CN(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)CC4)C=C3)N2N=C1	C43H56N10O6	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-NV6O2U	SCHEMBL21741622	4-[5-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]pentyl]-N-[4-[[(3-propan-2-yl-5-pyrrolidin-1-ylpyrazolo[1,5-a]pyrimidin-7-yl)amino]methyl]phenyl]piperazine-1-carboxamide	CC(C)C1=C2N=C(N3CCCC3)C=C(NCC3=CC=C(NC(=O)N4CCN(CCCCCC5=CC=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)N2N=C1	C43H54N10O4	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-ONHENJ	SCHEMBL21741615	4-[5-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]pentyl]-N-[4-[[[5-[(3S)-3-hydroxypiperidin-1-yl]-3-propan-2-ylpyrazolo[1,5-a]pyrimidin-7-yl]amino]methyl]phenyl]piperazine-1-carboxamide	CC(C)C1=C2N=C(N3CCC[C@H](O)C3)C=C(NCC3=CC=C(NC(=O)N4CCN(CCCCCC5=CC=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)N2N=C1	C44H56N10O5	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-YW2HBZ	SCHEMBL21741616	4-[5-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]pentyl]-N-[4-[[[5-[(1-methylsulfonylpiperidin-4-yl)amino]-3-propan-2-ylpyrazolo[1,5-a]pyrimidin-7-yl]amino]methyl]phenyl]piperazine-1-carboxamide	CC(C)C1=C2N=C(NC3CCN(S(C)(=O)=O)CC3)C=C(NCC3=CC=C(NC(=O)N4CCN(CCCCCC5=CC=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)N2N=C1	C45H59N11O6S	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-SQNNXC	WO2020035049A1_C130	.	CC(C)C1=C2N=C(N3CCS(=O)(=O)CC3)C=C(NCC3=CC=C(NC(=O)N4CCN(CCCCCC5=C6CN(C7CCC(=O)NC7=O)C(=O)C6CC=C5)CC4)C=C3)N2N=C1	C43H56N10O6S	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-7DEO5R	SCHEMBL21741626	4-[5-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]pentyl]-N-[4-[[[5-[(3R)-3-hydroxypiperidin-1-yl]-3-propan-2-ylpyrazolo[1,5-a]pyrimidin-7-yl]amino]methyl]phenyl]piperazine-1-carboxamide	CC(C)C1=C2N=C(N3CCC[C@@H](O)C3)C=C(NCC3=CC=C(NC(=O)N4CCN(CCCCCC5=CC=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)N2N=C1	C44H56N10O5	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-QSVT0F	SCHEMBL21741617	6-[4-[5-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]pentyl]piperazin-1-yl]-N-[4-[[[5-[[(2R)-1-hydroxybutan-2-yl]amino]-3-propan-2-ylpyrazolo[1,5-a]pyrimidin-7-yl]amino]methyl]phenyl]hexanamide	CC[C@H](CO)NC1=NC2=C(C(C)C)C=NN2C(NCC2=CC=C(NC(=O)CCCCCN3CCN(CCCCCC4=CC=CC5=C4CN(C4CCC(=O)NC4=O)C5=O)CC3)C=C2)=C1	C48H66N10O5	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-WQFVWB	SCHEMBL21741618	4-[4-[5-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]pentyl]piperazin-1-yl]-N-[4-[[[5-[[(2R)-1-hydroxybutan-2-yl]amino]-3-propan-2-ylpyrazolo[1,5-a]pyrimidin-7-yl]amino]methyl]phenyl]butanamide	CC[C@H](CO)NC1=NC2=C(C(C)C)C=NN2C(NCC2=CC=C(NC(=O)CCCN3CCN(CCCCCC4=CC=CC5=C4CN(C4CCC(=O)NC4=O)C5=O)CC3)C=C2)=C1	C46H62N10O5	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-F5AL8D	WO2020035049A1_C134	.	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(NC(=O)CCCN4CCN(CCCC5=CC=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)N2N=C1	C45H59N11O5	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-OALBP7	SCHEMBL21741623	4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]butyl]piperazin-1-yl]-N-[4-[[[2-(1-methylpiperidin-4-yl)oxy-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]phenyl]butanamide	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(NC(=O)CCCN4CCN(CCCCC5=CC=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)N2N=C1	C46H61N11O5	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-6SZW8G	CHEMBL4848803	4-[4-[5-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]pentyl]piperazin-1-yl]-N-[4-[[[2-(1-methylpiperidin-4-yl)oxy-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]phenyl]butanamide; SCHEMBL21741782; PD172419	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(NC(=O)CCCN4CCN(CCCCCC5=CC=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)N2N=C1	C47H63N11O5	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-J3CLWS	SCHEMBL21741789	5-[4-[3-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]propyl]piperazin-1-yl]-N-[4-[[[2-(1-methylpiperidin-4-yl)oxy-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]phenyl]pentanamide	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(NC(=O)CCCCN4CCN(CCCC5=CC=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)N2N=C1	C46H61N11O5	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-W8YVDO	SCHEMBL21741790	5-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]butyl]piperazin-1-yl]-N-[4-[[[2-(1-methylpiperidin-4-yl)oxy-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]phenyl]pentanamide	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(NC(=O)CCCCN4CCN(CCCCC5=CC=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)N2N=C1	C47H63N11O5	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-KLULFT	WO2020035049A1_C139	.	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(NC(=O)CCCCN4CCN(CCCCCC5=CC=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)N2N=C1	C48H65N11O5	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-L1WU83	CHEMBL4875639	6-[4-[3-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]propyl]piperazin-1-yl]-N-[4-[[[2-(1-methylpiperidin-4-yl)oxy-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]phenyl]hexanamide; SCHEMBL21741794; PD172420	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(NC(=O)CCCCCN4CCN(CCCC5=CC=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)N2N=C1	C47H63N11O5	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-WP8I8W	WO2020035049A1_C141	.	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(NC(=O)CCCCCN4CCN(CCCCC5=CC=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)N2N=C1	C48H65N11O5	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-CV7S5J	CHEMBL4870840	6-[4-[5-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]pentyl]piperazin-1-yl]-N-[4-[[[2-(1-methylpiperidin-4-yl)oxy-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]phenyl]hexanamide; SCHEMBL21741792; PD172418	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(NC(=O)CCCCCN4CCN(CCCCCC5=CC=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)N2N=C1	C49H67N11O5	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-2QK5BL	WO2020035049A1_C143	.	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(NC(=O)CCCCC#CC4=CC=CC5=C4CN(C4CCC(=O)NC4=O)C5=O)C=C3)N2N=C1	C41H47N9O5	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-OWEWC7	SCHEMBL21741797	8-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxy-N-[6-[[[2-(1-methylpiperidin-4-yl)oxy-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]pyridin-3-yl]octanamide	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(NC(=O)CCCCCCCOC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=N3)N2N=C1	C41H50N10O7	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-IWUSKN	SCHEMBL21741793	6-[4-[3-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]prop-2-ynyl]piperazin-1-yl]-N-[4-[[[2-(1-methylpiperidin-4-yl)oxy-8-propan-2-ylpyrazolo[1,5-a][1,3,5]triazin-4-yl]amino]methyl]phenyl]hexanamide	CC(C)C1=C2N=C(OC3CCN(C)CC3)N=C(NCC3=CC=C(NC(=O)CCCCCN4CCN(CC#CC5=CC=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)N2N=C1	C47H59N11O5	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-QXB531	SCHEMBL21741791	8-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxy-N-[4-[[[5-[(1-methylpiperidin-4-yl)amino]-3-propan-2-ylpyrazolo[1,5-a]pyrimidin-7-yl]amino]methyl]phenyl]octanamide	CC(C)C1=C2N=C(NC3CCN(C)CC3)C=C(NCC3=CC=C(NC(=O)CCCCCCCOC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C3)N2N=C1	C43H53N9O6	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-JMEZYZ	SCHEMBL21741786	7-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]-N-[4-[[[5-[(1-methylpiperidin-4-yl)amino]-3-propan-2-ylpyrazolo[1,5-a]pyrimidin-7-yl]amino]methyl]phenyl]heptanamide	CC(C)C1=C2N=C(NC3CCN(C)CC3)C=C(NCC3=CC=C(NC(=O)CCCCCCC4=CC=CC5=C4CN(C4CCC(=O)NC4=O)C5=O)C=C3)N2N=C1	C42H53N9O4	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-GZQBM4	WO2020035049A1_C148	.	CC[C@@H](CO)NC1=NC2=C(C(C)C)C=NN2C(NCC2=CC=C(NC(=O)CCCCCCC3C=CC=C4C(=O)N(C5CCC(=O)NC5=O)CC43)C=C2)=C1	C40H52N8O5	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-I70NOG	SCHEMBL21722286	7-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]-N-[4-[[[5-[[(2R)-1-hydroxybutan-2-yl]amino]-3-propan-2-ylpyrazolo[1,5-a]pyrimidin-7-yl]amino]methyl]phenyl]heptanamide	CC[C@H](CO)NC1=NC2=C(C(C)C)C=NN2C(NCC2=CC=C(NC(=O)CCCCCCC3=CC=CC4=C3CN(C3CCC(=O)NC3=O)C4=O)C=C2)=C1	C40H50N8O5	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-K2U5XB	PROTAC CDK9 degrader-4	PROTAC CDK9 degrader-4; 2411021-01-5; orb1984561; CHEMBL4849244; SCHEMBL21741644; EX-A8550; AKOS040757675; DA-66949; PD172423; HY-115728; CS-0254141; 4-[5-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]pentyl]-N-[4-[[[5-[[(2S)-1-hydroxybutan-2-yl]amino]-3-propan-2-ylpyrazolo[1,5-a]pyrimidin-7-yl]amino]methyl]phenyl]piperazine-1-carboxamide	CC[C@@H](CO)NC1=NC2=C(C(C)C)C=NN2C(NCC2=CC=C(NC(=O)N3CCN(CCCCCC4=C5CN(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)C=C2)=C1	C43H56N10O5	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-FU560C	SCHEMBL21741641	4-[5-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]pentyl]-N-[4-[[[5-[[(2R)-1-hydroxybutan-2-yl]amino]-3-propan-2-ylpyrazolo[1,5-a]pyrimidin-7-yl]amino]methyl]phenyl]piperazine-1-carboxamide	CC[C@H](CO)NC1=NC2=C(C(C)C)C=NN2C(NCC2=CC=C(NC(=O)N3CCN(CCCCCC4=C5CN(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)C=C2)=C1	C43H56N10O5	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-Y9FYDI	SCHEMBL21741647	4-[5-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]pentyl]-N-[4-[[[5-[(1-methylpiperidin-4-yl)amino]-3-propan-2-ylpyrazolo[1,5-a]pyrimidin-7-yl]amino]methyl]phenyl]piperazine-1-carboxamide	CC(C)C1=C2N=C(NC3CCN(C)CC3)C=C(NCC3=CC=C(NC(=O)N4CCN(CCCCCC5=C6CN(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)CC4)C=C3)N2N=C1	C45H59N11O4	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-5ZRJ81	SCHEMBL21741649	4-[5-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]pentyl]-N-[4-[[[5-(oxan-4-ylamino)-3-propan-2-ylpyrazolo[1,5-a]pyrimidin-7-yl]amino]methyl]phenyl]piperazine-1-carboxamide	CC(C)C1=C2N=C(NC3CCOCC3)C=C(NCC3=CC=C(NC(=O)N4CCN(CCCCCC5=CC=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)N2N=C1	C44H56N10O5	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-4KHOA7	WO2020035049A1_C154	.	CC[C@@H](CO)NC1=NC2=C(C(C)C)C=NN2C(NCC2=CC=C(NC(=O)N3CCN(CCCCCC4=CC=CC5=C4CN(C4CCC(=O)NC4=O)C5=O)CC3)C=C2)=N1	C42H55N11O5	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-RLQ08W	SCHEMBL21741643	4-[5-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]pentyl]-N-[4-[[[5-[(3R)-3-hydroxypyrrolidin-1-yl]-3-propan-2-ylpyrazolo[1,5-a]pyrimidin-7-yl]amino]methyl]phenyl]piperazine-1-carboxamide	CC(C)C1=C2N=C(N3CC[C@@H](O)C3)C=C(NCC3=CC=C(NC(=O)N4CCN(CCCCCC5=CC=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)N2N=C1	C43H54N10O5	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-TVQ7WV	SCHEMBL21741648	4-[5-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]pentyl]-N-[4-[[[5-[(3S)-3-hydroxypyrrolidin-1-yl]-3-propan-2-ylpyrazolo[1,5-a]pyrimidin-7-yl]amino]methyl]phenyl]piperazine-1-carboxamide	CC(C)C1=C2N=C(N3CC[C@H](O)C3)C=C(NCC3=CC=C(NC(=O)N4CCN(CCCCCC5=CC=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)N2N=C1	C43H54N10O5	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-LS6R1C	WO2020035049A1_C157	.	CC(C)C1=C2N=C(N3CCC[C@H]3CO)C=C(NCC3=CC=C(NC(=O)N4CCN(CCCCCC5=C6CN(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)CC4)C=C3)N2N=C1	C44H56N10O5	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-35YGU6	SCHEMBL21741787	4-[5-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]pentyl]-N-[4-[[[5-[(2R)-2-(hydroxymethyl)pyrrolidin-1-yl]-3-propan-2-ylpyrazolo[1,5-a]pyrimidin-7-yl]amino]methyl]phenyl]piperazine-1-carboxamide	CC(C)C1=C2N=C(N3CCC[C@@H]3CO)C=C(NCC3=CC=C(NC(=O)N4CCN(CCCCCC5=CC=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)N2N=C1	C44H56N10O5	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-LOV9BG	SCHEMBL21741795	4-[5-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]pentyl]-N-[4-[[[5-[(2R)-2-(2-hydroxyethyl)piperidin-1-yl]-3-propan-2-ylpyrazolo[1,5-a]pyrimidin-7-yl]amino]methyl]phenyl]piperazine-1-carboxamide	CC(C)C1=C2N=C(N3CCCC[C@@H]3CCO)C=C(NCC3=CC=C(NC(=O)N4CCN(CCCCCC5=CC=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)N2N=C1	C46H60N10O5	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-VFV7T8	SCHEMBL21722278	4-[5-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]pentyl]-N-[4-[[[5-[(2S)-2-(2-hydroxyethyl)piperidin-1-yl]-3-propan-2-ylpyrazolo[1,5-a]pyrimidin-7-yl]amino]methyl]phenyl]piperazine-1-carboxamide	CC(C)C1=C2N=C(N3CCCC[C@H]3CCO)C=C(NCC3=CC=C(NC(=O)N4CCN(CCCCCC5=C6CN(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)CC4)C=C3)N2N=C1	C46H60N10O5	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-3486ST	SCHEMBL21741799	N-[4-[[[5-[[(2S,3R)-1,3-dihydroxybutan-2-yl]amino]-3-propan-2-ylpyrazolo[1,5-a]pyrimidin-7-yl]amino]methyl]phenyl]-4-[5-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]pentyl]piperazine-1-carboxamide	CC(C)C1=C2N=C(N[C@@H](CO)[C@@H](C)O)C=C(NCC3=CC=C(NC(=O)N4CCN(CCCCCC5=C6CN(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)CC4)C=C3)N2N=C1	C43H56N10O6	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-XRN80Z	SCHEMBL21741788	4-[5-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]pentyl]-N-[4-[[[3-propan-2-yl-5-[[(2S,3S)-1,3,4-trihydroxybutan-2-yl]amino]pyrazolo[1,5-a]pyrimidin-7-yl]amino]methyl]phenyl]piperazine-1-carboxamide	CC(C)C1=C2N=C(N[C@@H](CO)[C@H](O)CO)C=C(NCC3=CC=C(NC(=O)N4CCN(CCCCCC5=CC=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)N2N=C1	C43H56N10O7	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-K8RTCO	SCHEMBL21741784	2-[4-[5-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]pentyl]piperazin-1-yl]-N-[4-[[[5-[[(2R)-1-hydroxybutan-2-yl]amino]-3-propan-2-ylpyrazolo[1,5-a]pyrimidin-7-yl]amino]methyl]phenyl]acetamide	CC[C@H](CO)NC1=NC2=C(C(C)C)C=NN2C(NCC2=CC=C(NC(=O)CN3CCN(CCCCCC4=C5CN(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)C=C2)=C1	C44H58N10O5	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-MZS3AJ	WO2020035049A1_C164	.	CC[C@@H](CO)NC1=NC2=C(C(C)C)C=NN2C(NCC2=CC=C(NC(=O)CCN3CCN(CCCCCC4=CC=CC5=C4CN(C4CCC(=O)NC4=O)C5=O)CC3)C=C2)=C1	C45H60N10O5	CDK7;CDK9	P50613/P50750	CRBN	WO-2020035049-A1
TPD-DRA1NJ	CHEMBL4633400	(2S,4R)-1-[(2S)-3,3-dimethyl-2-[[2-[2-[2-[[2-[4-(methylamino)phenyl]-1,3-benzothiazol-6-yl]oxy]ethoxy]ethoxy]acetyl]amino]butanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL21771117; PD140720	CNC1=CC=C(C2=NC3=C(C=C(OCCOCCOCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)N[C@@H](C)C4=CC=C(C5=C(C)N=CS5)C=C4)C(C)(C)C)C=C3)S2)C=C1	C43H52N6O7S2	α-syn	P37840	VHL	WO-2020041331-A1
TPD-VLH2QZ	WO2020041331A1_2	.	CNC1=CC=C(C2=NC3=C(C=C(OCCOCCOCCOCC(=O)N[C@H](C(=O)N4C[C@H](O)CC4C(=O)N[C@@H](C)C4=CC=C(C5=C(C)N=CS5)C=C4)C(C)(C)C)C=C3)S2)C=C1	C45H56N6O8S2	α-syn	P37840	VHL	WO-2020041331-A1
TPD-9Q2MZJ	SCHEMBL21820254	(2S,4R)-1-[(2S)-3,3-dimethyl-2-[[2-[2-[2-[2-[2-[[2-[4-(methylamino)phenyl]-1,3-benzothiazol-6-yl]oxy]ethoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]butanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL30497584	CNC1=CC=C(C2=NC3=C(C=C(OCCOCCOCCOCCOCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)N[C@@H](C)C4=CC=C(C5=C(C)N=CS5)C=C4)C(C)(C)C)C=C3)S2)C=C1	C47H60N6O9S2	α-syn	P37840	VHL	WO-2020041331-A1
TPD-4PAMCT	CHEMBL4634581	(2S,4R)-1-[(2S)-3,3-dimethyl-2-[[2-[2-[2-[2-[2-[2-[[2-[4-(methylamino)phenyl]-1,3-benzothiazol-6-yl]oxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]butanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL21820347; SCHEMBL30497521; PD140718	CNC1=CC=C(C2=NC3=C(C=C(OCCOCCOCCOCCOCCOCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)N[C@@H](C)C4=CC=C(C5=C(C)N=CS5)C=C4)C(C)(C)C)C=C3)S2)C=C1	C49H64N6O10S2	α-syn	P37840	VHL	WO-2020041331-A1
TPD-CQRS35	PROTAC |A-synuclein degrader 3	PROTAC ; A-synuclein degrader 3; PROTAC alpha-synuclein degrader 3; 2412273-77-7; orb2278512; CHEMBL4634339; SCHEMBL21820337; SCHEMBL30497585; EX-A11337; HY-136001; CS-0119142	CNC1=CC=C(C2=NC3=C(C=C(OCCOCCOCCOCCOCCOCCOCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)N[C@@H](C)C4=CC=C(C5=C(C)N=CS5)C=C4)C(C)(C)C)C=C3)S2)C=C1	C51H68N6O11S2	α-syn	P37840	VHL	WO-2020041331-A1
TPD-W46FZG	WO2020041331A1_6	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOC3=CC=C(CN4C(=O)C(=CC=CC5=CC=C(NOO)C=C5)C5=CC=CC=C54)C=C3)C(C)(C)C)C=C2)SC=N1	C53H60N6O10S	α-syn	P37840	VHL	WO-2020041331-A1
TPD-SGCCMQ	WO2020041331A1_8	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOC3=CC4=C(C=C3)NC3=CC=C(NOO)C=C3S4)C(C)(C)C)C=C2)SC=N1	C41H50N6O9S2	α-syn	P37840	VHL	WO-2020041331-A1
TPD-OLV7BJ	WO2020041331A1_9	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOC3=CC4=C(C=C3)NC3=CC=C(NOO)C=C3S4)C(C)(C)C)C=C2)SC=N1	C43H54N6O10S2	α-syn	P37840	VHL	WO-2020041331-A1
TPD-R938NR	WO2020041331A1_10	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOCCOC3=CC4=C(C=C3)NC3=CC=C(NOO)C=C3S4)C(C)(C)C)C=C2)SC=N1	C45H58N6O11S2	α-syn	P37840	VHL	WO-2020041331-A1
TPD-V4ZPQI	WO2020041331A1_11	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOCCOCCOC3=CC4=C(C=C3)NC3=CC=C(NOO)C=C3S4)C(C)(C)C)C=C2)SC=N1	C47H62N6O12S2	α-syn	P37840	VHL	WO-2020041331-A1
TPD-NBYFGU	WO2020041331A1_12	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOCCOCCOCCOC3=CC4=C(C=C3)NC3=CC=C(NOO)C=C3S4)C(C)(C)C)C=C2)SC=N1	C49H66N6O13S2	α-syn	P37840	VHL	WO-2020041331-A1
TPD-223GYE	WO2020041331A1_13	.	O=C1CCC(N2C(=O)C3=C(C=C(OCCOCCOCCOCCOC4=CC5=C(C=C4)NC4=CC=C(NOO)C=C4S5)C=C3)C2=O)C(=O)N1	C33H34N4O11S	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-KX48D3	WO2020041331A1_14	.	O=C1CCC(N2C(=O)C3=C(C=C(OCCOCCOCCOCCOCCOC4=CC5=C(C=C4)NC4=CC=C(NOO)C=C4S5)C=C3)C2=O)C(=O)N1	C35H38N4O12S	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-PZCQZH	SCHEMBL21771138	2-(2,6-Dioxopiperidin-3-yl)-5-[2-[2-[2-[methyl(3-phenothiazin-10-ylpropyl)amino]ethoxy]ethoxy]ethoxy]isoindole-1,3-dione; SCHEMBL30497538	CN(CCCN1C2=C(C=CC=C2)SC2=C1C=CC=C2)CCOCCOCCOC1=CC2=C(C=C1)C(=O)N(C1CCC(=O)NC1=O)C2=O	C35H38N4O7S	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-NDYVU6	SCHEMBL21752033	2-(2,6-Dioxopiperidin-3-yl)-5-[2-[2-[2-[2-[methyl(3-phenothiazin-10-ylpropyl)amino]ethoxy]ethoxy]ethoxy]ethoxy]isoindole-1,3-dione; SCHEMBL30497567	CN(CCCN1C2=C(C=CC=C2)SC2=C1C=CC=C2)CCOCCOCCOCCOC1=CC2=C(C=C1)C(=O)N(C1CCC(=O)NC1=O)C2=O	C37H42N4O8S	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-TL9JB8	SCHEMBL21752054	2-(2,6-Dioxopiperidin-3-yl)-5-[4-[3-[1-[4-(6-methoxy-1,3-benzothiazol-2-yl)phenyl]azetidin-3-yl]oxypropyl]piperazin-1-yl]isoindole-1,3-dione; SCHEMBL30497545	COC1=CC=C2N=C(C3=CC=C(N4CC(OCCCN5CCN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)C=C3)SC2=C1	C37H38N6O6S	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-TCZR45	WO2020041331A1_18	.	O=C1CCC(N2C(=O)C3=C(C=C(N4CCN(CCN5CCC(O[C@H]6C[C@H](OC7=CC8=C(C=C7)NC7=CC=C(NOO)C=C7S8)C6)CC5)CC4)C=C3)C2=O)C(=O)N1	C40H45N7O8S	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-WAOVRF	WO2020041331A1_19	.	O=C1CCC(N2C(=O)C3=C(C=C(OCCCCCN4CCC(O[C@H]5C[C@H](OC6=CC7=C(C=C6)NC6=CC=C(NOO)C=C6S7)C5)CC4)C=C3)C2=O)C(=O)N1	C39H43N5O9S	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-ZFV7TU	SCHEMBL21751984	5-[2-[2-[2-[2-[[7-(dimethylamino)-10H-phenothiazin-3-yl]oxy]ethoxy]ethoxy]ethoxy]ethoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN(C)C1=CC=C2NC3=C(C=C(OCCOCCOCCOCCOC4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C=C3)SC2=C1	C35H38N4O9S	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-1NJGWT	SCHEMBL21771140	5-[2-[2-[2-[2-[2-[[7-(dimethylamino)-10H-phenothiazin-3-yl]oxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione; SCHEMBL30497574	CN(C)C1=CC=C2NC3=C(C=C(OCCOCCOCCOCCOCCOC4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C=C3)SC2=C1	C37H42N4O10S	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-OMYUDC	SCHEMBL21751971	2-(2,6-Dioxopiperidin-3-yl)-5-[5-[4-[1-(3-phenothiazin-10-ylpropyl)azetidin-3-yl]oxypiperidin-1-yl]pentoxy]isoindole-1,3-dione; SCHEMBL30497589	O=C1CCC(N2C(=O)C3=C(C=C(OCCCCCN4CCC(OC5CN(CCCN6C7=C(C=CC=C7)SC7=C6C=CC=C7)C5)CC4)C=C3)C2=O)C(=O)N1	C41H47N5O6S	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-1V23VW	SCHEMBL21771327	2-(2,6-Dioxopiperidin-3-yl)-5-[4-[2-[4-[1-(3-phenothiazin-10-ylpropyl)azetidin-3-yl]oxypiperidin-1-yl]ethyl]piperazin-1-yl]isoindole-1,3-dione; SCHEMBL30497536	O=C1CCC(N2C(=O)C3=C(C=C(N4CCN(CCN5CCC(OC6CN(CCCN7C8=C(C=CC=C8)SC8=C7C=CC=C8)C6)CC5)CC4)C=C3)C2=O)C(=O)N1	C42H49N7O5S	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-ZJL8AS	SCHEMBL21771343	5-[4-[3-[3-[[2-[4-(Dimethylamino)phenyl]-1,3-benzothiazol-6-yl]oxy]cyclobutyl]oxypropyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione; SCHEMBL21820324	CN(C)C1=CC=C(C2=NC3=C(C=C(O[C@H]4C[C@H](OCCCN5CCN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)C=C3)S2)C=C1	C39H42N6O6S	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-25HADY	SCHEMBL21752007	2-(2,6-Dioxopiperidin-3-yl)-5-[5-[4-[1-[4-(6-methoxy-1,3-benzothiazol-2-yl)phenyl]azetidin-3-yl]oxypiperidin-1-yl]pentoxy]isoindole-1,3-dione; SCHEMBL30497596	COC1=CC=C2N=C(C3=CC=C(N4CC(OC5CCN(CCCCCOC6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)C=C3)SC2=C1	C40H43N5O7S	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-RIQGXB	SCHEMBL21771321	2-(2,6-Dioxopiperidin-3-yl)-5-[4-[2-[4-[1-[4-(6-methoxy-1,3-benzothiazol-2-yl)phenyl]azetidin-3-yl]oxypiperidin-1-yl]ethyl]piperazin-1-yl]isoindole-1,3-dione; SCHEMBL30497544	COC1=CC=C2N=C(C3=CC=C(N4CC(OC5CCN(CCN6CCN(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)C4)C=C3)SC2=C1	C41H45N7O6S	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-Y4P0IL	SCHEMBL21771143	5-[5-[4-[3-[[2-[4-(Dimethylamino)phenyl]-1,3-benzothiazol-6-yl]oxy]cyclobutyl]oxypiperidin-1-yl]pentoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione; SCHEMBL21820363	CN(C)C1=CC=C(C2=NC3=C(C=C(O[C@H]4C[C@H](OC5CCN(CCCCCOC6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)C=C3)S2)C=C1	C42H47N5O7S	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-ES5SNL	SCHEMBL21771145	2-(2,6-Dioxopiperidin-3-yl)-5-[4-[3-[1-(3-phenothiazin-10-ylpropyl)azetidin-3-yl]oxypropyl]piperazin-1-yl]isoindole-1,3-dione; SCHEMBL30497588	O=C1CCC(N2C(=O)C3=C(C=C(N4CCN(CCCOC5CN(CCCN6C7=C(C=CC=C7)SC7=C6C=CC=C7)C5)CC4)C=C3)C2=O)C(=O)N1	C38H42N6O5S	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-L08KFW	SCHEMBL21771144	5-[4-[2-[4-[3-[[2-[4-(Dimethylamino)phenyl]-1,3-benzothiazol-6-yl]oxy]cyclobutyl]oxypiperidin-1-yl]ethyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione; SCHEMBL21820305	CN(C)C1=CC=C(C2=NC3=C(C=C(O[C@H]4C[C@H](OC5CCN(CCN6CCN(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)C4)C=C3)S2)C=C1	C43H49N7O6S	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-IRERB0	WO2020041331A1_30	.	O=C1CCC(N2C(=O)C3=C(C=C(N4CCN(CCCO[C@H]5C[C@H](OC6=CC7=C(C=C6)NC6=CC=C(NOO)C=C6S7)C5)CC4)C=C3)C2=O)C(=O)N1	C36H38N6O8S	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-BK50TB	SCHEMBL26017982	2-(2,6-Dioxopiperidin-3-yl)-5-[5-[4-[3-[4-[[3-[3-(4-nitrophenyl)prop-2-enylidene]-2-oxoindol-1-yl]methyl]phenoxy]cyclobutyl]oxypiperidin-1-yl]pentoxy]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC=C(OCCCCCN4CCC(O[C@H]5C[C@H](OC6=CC=C(CN7C(=O)C(=CC=CC8=CC=C([N+](=O)[O-])C=C8)C8=CC=CC=C87)C=C6)C5)CC4)C=C3C2=O)C(=O)N1	C51H51N5O10	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-PLB8ND	WO2020041331A1_33	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCCN3CCC(O[C@H]4C[C@H](OC5=CC6=C(C=C5)NC5=CC=C(NOO)C=C5S6)C4)CC3)C(C)(C)C)C=C2)SC=N1	C51H67N7O9S2	α-syn	P37840	VHL	WO-2020041331-A1
TPD-12C0L8	WO2020041331A1_34	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCN(CCN4CCC(O[C@H]5C[C@H](OC6=CC7=C(C=C6)NC6=CC=C(NOO)C=C6S7)C5)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C52H69N9O8S2	α-syn	P37840	VHL	WO-2020041331-A1
TPD-IMSSYV	WO2020041331A1_35	.	COC1=CC(/C=C/C2=NC3=C(C=C2)C=C(OCCOCCOCCOCC(=O)N[C@H](C(=O)C2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C4=C(C)N=CS4)C=C2)C(C)(C)C)C=C3)=CC=N1	C49H59N5O9S	α-syn	P37840	VHL	WO-2020041331-A1
TPD-NNKWP1	SCHEMBL21771346	2-(2,6-dioxopiperidin-3-yl)-5-[2-[2-[2-[2-[2-[(E)-2-(2-methoxypyridin-4-yl)ethenyl]quinolin-6-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]isoindole-1,3-dione; SCHEMBL30497555	COC1=CC(/C=C/C2=NC3=C(C=C2)C=C(OCCOCCOCCOCCOC2=CC4=C(C=C2)C(=O)N(C2CCC(=O)NC2=O)C4=O)C=C3)=CC=N1	C38H38N4O10	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-OT54SQ	SCHEMBL21771348	2-(2,6-dioxopiperidin-3-yl)-5-[5-[4-[3-[2-[(E)-2-(2-methoxypyridin-4-yl)ethenyl]quinolin-6-yl]oxycyclobutyl]oxypiperidin-1-yl]pentoxy]isoindole-1,3-dione	COC1=CC(/C=C/C2=NC3=C(C=C2)C=C(O[C@H]2C[C@H](OC4CCN(CCCCCOC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C2)C=C3)=CC=N1	C44H47N5O8	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-VX0QZ8	SCHEMBL21771350	2-(2,6-Dioxopiperidin-3-yl)-5-[5-[4-[3-[2-[5-(2-methoxypyridin-4-yl)-1,2,4-oxadiazol-3-yl]quinolin-6-yl]oxycyclobutyl]oxypiperidin-1-yl]pentoxy]isoindole-1,3-dione	COC1=CC(C2=NC(C3=NC4=C(C=C3)C=C(O[C@H]3C[C@H](OC5CCN(CCCCCOC6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C3)C=C4)=NO2)=CC=N1	C44H45N7O9	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-0IIGD9	SCHEMBL21771344	2-(2,6-dioxopiperidin-3-yl)-5-[4-[2-[4-[3-[2-[(E)-2-(2-methoxypyridin-4-yl)ethenyl]quinolin-6-yl]oxycyclobutyl]oxypiperidin-1-yl]ethyl]piperazin-1-yl]isoindole-1,3-dione	COC1=CC(/C=C/C2=NC3=C(C=C2)C=C(O[C@H]2C[C@H](OC4CCN(CCN5CCN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)C2)C=C3)=CC=N1	C45H49N7O7	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-B92V55	SCHEMBL21771510	2-(2,6-Dioxopiperidin-3-yl)-5-[4-[2-[4-[3-[2-[5-(2-methoxypyridin-4-yl)-1,2,4-oxadiazol-3-yl]quinolin-6-yl]oxycyclobutyl]oxypiperidin-1-yl]ethyl]piperazin-1-yl]isoindole-1,3-dione	COC1=CC(C2=NC(C3=NC4=C(C=C3)C=C(O[C@H]3C[C@H](OC5CCN(CCN6CCN(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)C3)C=C4)=NO2)=CC=N1	C45H47N9O8	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-O4VUH0	WO2020041331A1_41	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(OCCOCCOCCOC4=CC5=C(C=C4)NC4=CC=C(NOO)C=C4S5)=NO3)C(C)C)C=C2)SC=N1	C43H50N6O10S2	α-syn	P37840	VHL	WO-2020041331-A1
TPD-V8WLHW	WO2020041331A1_42	.	COC1=CC(/C=C/C2=NC3=C(C=C2)C=C(OCCOCCOCCOC2=NOC([C@H](C(=O)N4C[C@H](O)CC4C(=O)N[C@@H](C)C4=CC=C(C5=C(C)N=CS5)C=C4)C(C)C)=C2)C=C3)=CC=N1	C48H54N6O9S	α-syn	P37840	VHL	WO-2020041331-A1
TPD-L1NJ93	SCHEMBL21771511	(2S,4R)-4-hydroxy-1-[(2R)-2-[3-[4-[2-[4-[1-[4-(6-methoxy-1,3-benzothiazol-2-yl)phenyl]azetidin-3-yl]oxypiperidin-1-yl]ethyl]piperazin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	COC1=CC=C2N=C(C3=CC=C(N4CC(OC5CCN(CCN6CCN(C7=NOC([C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)C8=CC=C(C9=C(C)N=CS9)C=C8)C(C)C)=C7)CC6)CC5)C4)C=C3)SC2=C1	C53H65N9O6S2	α-syn	P37840	VHL	WO-2020041331-A1
TPD-IBVEEB	SCHEMBL21771513	(2S,4R)-4-hydroxy-1-[(2R)-3-methyl-2-[3-[2-[2-[2-[2-[[2-[4-(methylamino)phenyl]-1,3-benzothiazol-6-yl]oxy]ethoxy]ethoxy]ethoxy]ethoxy]-1,2-oxazol-5-yl]butanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CNC1=CC=C(C2=NC3=C(C=C(OCCOCCOCCOCCOC4=NOC([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=C(C)N=CS6)C=C5)C(C)C)=C4)C=C3)S2)C=C1	C47H56N6O9S2	α-syn	P37840	VHL	WO-2020041331-A1
TPD-M1W0PX	WO2020041331A1_45	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCN(CCN5CCC(O[C@H]6C[C@H](OC7=CC8=C(C=C7)NC7=CC=C(NOO)C=C7S8)C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C52H65N9O8S2	α-syn	P37840	VHL	WO-2020041331-A1
TPD-G8HFCL	WO2020041331A1_46	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(OCCCCCN4CCC(O[C@H]5C[C@H](OC6=CC7=C(C=C6)NC6=CC=C(NOO)C=C6S7)C5)CC4)=NO3)C(C)C)C=C2)SC=N1	C51H63N7O9S2	α-syn	P37840	VHL	WO-2020041331-A1
TPD-8BA0WZ	SCHEMBL21771141	2-(2,6-dioxopiperidin-3-yl)-5-[2-[2-[2-[2-[(E)-2-(2-methoxypyridin-4-yl)ethenyl]quinolin-6-yl]oxyethoxy]ethoxy]ethoxy]isoindole-1,3-dione; SCHEMBL30497519	COC1=NC=CC(/C=C/C2=CC=C3C=C(OCCOCCOCCOC4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C=CC3=N2)=C1	C36H34N4O9	α-syn	P37840	VHL	WO-2020041331-A1
TPD-JQM0UG	SCHEMBL21771142	(2S,4R)-4-hydroxy-1-[(2S)-2-[[2-[2-[2-[2-[2-[2-[(E)-2-(2-methoxypyridin-4-yl)ethenyl]quinolin-6-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL30497586	COC1=NC=CC(/C=C/C2=NC3=C(C=C2)C=C(OCCOCCOCCOCCOCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C4=C(C)N=CS4)C=C2)C(C)(C)C)C=C3)=C1	C50H62N6O10S	α-syn	P37840	VHL	WO-2020041331-A1
TPD-U740UD	SCHEMBL21771330	2-[4-[2-[2-[2-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]ethoxy]ethoxy]ethyl]piperazin-1-yl]-N-[1-(1H-indol-3-yl)hexan-2-yl]-1,3-thiazole-5-carboxamide; SCHEMBL30497539	CCCCC(CC1=CNC2=C1C=CC=C2)NC(=O)C1=CN=C(N2CCN(CCOCCOCCOCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](C)C3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)CC2)S1	C53H73N9O8S2	α-syn	P37840	VHL	WO-2020041331-A1
TPD-I03Y0Q	SCHEMBL21771331	2-[4-[2-[2-[2-[2-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]ethoxy]ethoxy]ethoxy]ethyl]piperazin-1-yl]-N-[1-(1H-indol-3-yl)hexan-2-yl]-1,3-thiazole-5-carboxamide; SCHEMBL30497565	CCCCC(CC1=CNC2=C1C=CC=C2)NC(=O)C1=CN=C(N2CCN(CCOCCOCCOCCOCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](C)C3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)CC2)S1	C55H77N9O9S2	α-syn	P37840	VHL	WO-2020041331-A1
TPD-29IX2H	SCHEMBL21820357	2-[4-[2-[2-[2-[2-[2-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethyl]piperazin-1-yl]-N-[1-(1H-indol-3-yl)hexan-2-yl]-1,3-thiazole-5-carboxamide	CCCCC(CC1=CNC2=C1C=CC=C2)NC(=O)C1=CN=C(N2CCN(CCOCCOCCOCCOCCOCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](C)C3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)CC2)S1	C57H81N9O10S2	α-syn	P37840	VHL	WO-2020041331-A1
TPD-KTZEHL	SCHEMBL21751989	2-[4-[2-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxyethoxy]ethoxy]ethyl]piperazin-1-yl]-N-[1-(1H-indol-3-yl)hexan-2-yl]-1,3-thiazole-5-carboxamide; SCHEMBL30497581	CCCCC(CC1=CNC2=C1C=CC=C2)NC(=O)C1=CN=C(N2CCN(CCOCCOCCOC3=CC=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)CC2)S1	C41H49N7O8S	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-P0JE9H	WO2020041331A1_53	.	CCCC(CC1=CNC2=C1C=CC=C2)NC(=O)C1=CN=C(N2CCN(CCOCCOCCOCCOC3=CC=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)CC2)S1	C42H51N7O9S	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-P8HP7N	SCHEMBL21771337	2-[4-[2-[2-[2-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]ethyl]piperazin-1-yl]-N-[1-(1H-indol-3-yl)hexan-2-yl]-1,3-thiazole-5-carboxamide; SCHEMBL30497580	CCCCC(CC1=CNC2=C1C=CC=C2)NC(=O)C1=CN=C(N2CCN(CCOCCOCCOCCOCCOC3=CC=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)CC2)S1	C45H57N7O10S	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-P4RR5B	SCHEMBL21771332	2-[4-[4-[2-[2-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]ethoxy]ethoxy]phenyl]piperazin-1-yl]-N-[1-(1H-indol-3-yl)hexan-2-yl]-1,3-thiazole-5-carboxamide; SCHEMBL30497571	CCCCC(CC1=CNC2=C1C=CC=C2)NC(=O)C1=CN=C(N2CCN(C3=CC=C(OCCOCCOCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)N[C@@H](C)C4=CC=C(C5=C(C)N=CS5)C=C4)C(C)(C)C)C=C3)CC2)S1	C57H73N9O8S2	α-syn	P37840	VHL	WO-2020041331-A1
TPD-S5D3DQ	SCHEMBL21771338	2-[4-[4-[2-[2-[2-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]ethoxy]ethoxy]ethoxy]phenyl]piperazin-1-yl]-N-[1-(1H-indol-3-yl)hexan-2-yl]-1,3-thiazole-5-carboxamide; SCHEMBL30497576	CCCCC(CC1=CNC2=C1C=CC=C2)NC(=O)C1=CN=C(N2CCN(C3=CC=C(OCCOCCOCCOCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)N[C@@H](C)C4=CC=C(C5=C(C)N=CS5)C=C4)C(C)(C)C)C=C3)CC2)S1	C59H77N9O9S2	α-syn	P37840	VHL	WO-2020041331-A1
TPD-P7QQDB	SCHEMBL21752053	2-[4-[4-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxyethoxy]ethoxy]phenyl]piperazin-1-yl]-N-[1-(1H-indol-3-yl)hexan-2-yl]-1,3-thiazole-5-carboxamide; SCHEMBL30497522	CCCCC(CC1=CNC2=C1C=CC=C2)NC(=O)C1=CN=C(N2CCN(C3=CC=C(OCCOCCOC4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)C=C3)CC2)S1	C45H49N7O8S	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-QXL8DR	SCHEMBL21771335	2-[4-[4-[2-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxyethoxy]ethoxy]ethoxy]phenyl]piperazin-1-yl]-N-[1-(1H-indol-3-yl)hexan-2-yl]-1,3-thiazole-5-carboxamide; SCHEMBL30497529	CCCCC(CC1=CNC2=C1C=CC=C2)NC(=O)C1=CN=C(N2CCN(C3=CC=C(OCCOCCOCCOC4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)C=C3)CC2)S1	C47H53N7O9S	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-AHUPLA	WO2020041331A1_59	.	O=C1CCC(N2C(=O)C3=CC=C(OCCOCCOC4=CC=C(CN5C(=O)/C(=C/C=C/C6=CC=C(NOO)C=C6)C6=C5C=CC=C6)C=C4)C=C3C2=O)C(=O)N1	C41H36N4O10	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-WK1R7N	SCHEMBL21820308	2-(2,6-dioxopiperidin-3-yl)-5-[2-[2-[4-[[(3Z)-3-[(E)-3-(4-nitrophenyl)prop-2-enylidene]-2-oxoindol-1-yl]methyl]phenoxy]ethoxy]ethoxy]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC=C(OCCOCCOC4=CC=C(CN5C(=O)/C(=C\C=C\C6=CC=C([N+](=O)[O-])C=C6)C6=C5C=CC=C6)C=C4)C=C3C2=O)C(=O)N1	C41H34N4O10	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-UTZXWB	WO2020041331A1_61	.	O=NC1=CC=C(/C=C/C=C2/C(=O)N(CC3=CC=C(OCCOCCOCCOC4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)C=C3)C3=C2C=CC=C3)C=C1	C43H38N4O10	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-DML84Q	SCHEMBL21820288	2-(2,6-dioxopiperidin-3-yl)-5-[2-[2-[2-[4-[[(3Z)-3-[(E)-3-(4-nitrophenyl)prop-2-enylidene]-2-oxoindol-1-yl]methyl]phenoxy]ethoxy]ethoxy]ethoxy]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC=C(OCCOCCOCCOC4=CC=C(CN5C(=O)/C(=C\C=C\C6=CC=C([N+](=O)[O-])C=C6)C6=C5C=CC=C6)C=C4)C=C3C2=O)C(=O)N1	C43H38N4O11	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-WTX0AH	WO2020041331A1_63	.	O=C1CCC(N2C(=O)C3=CC=C(OCCOCCOCCOCCOC4=CC=C(CN5C(=O)/C(=C/C=C/C6=CC=C(NOO)C=C6)C6=C5C=CC=C6)C=C4)C=C3C2=O)C(=O)N1	C45H44N4O12	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-FVZRYA	WO2020041331A1_64	.	O=NC1=CC=C(/C=C/C=C2\C(=O)N(CC3=CC=C(OCCOCCOCCOCCOC4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)C=C3)C3=C2C=CC=C3)C=C1	C45H42N4O11	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-YPQ1UV	WO2020041331A1_65	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3=CC(OCCOCCOC4=CC=C(CN5C(=O)/C(=C/C=C/C6=CC=C(NOO)C=C6)C6=C5C=CC=C6)C=C4)=NO3)C(C)C)C=C2)SC=N1	C53H56N6O10S	α-syn	P37840	VHL	WO-2020041331-A1
TPD-ZLT1LD	WO2020041331A1_66	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(OCCOCCOC4=CC=C(CN5C(=O)/C(=C/C=C/C6=CC=C(NOO)C=C6)C6=C5C=CC=C6)C=C4)=NO3)C(C)C)C=C2)SC=N1	C53H56N6O10S	α-syn	P37840	VHL	WO-2020041331-A1
TPD-IQZ5PP	WO2020041331A1_67	.	CC1=C(C2=CC=C([C@H](C)NC(=O)C3C[C@@H](O)CN3C(=O)[C@H](C3=CC(OCCOCCOC4=CC=C(CN5C(=O)/C(=C\C=C\C6=CC=C([N+](=O)[O-])C=C6)C6=C5C=CC=C6)C=C4)=NO3)C(C)C)C=C2)SC=N1	C53H54N6O10S	α-syn	P37840	VHL	WO-2020041331-A1
TPD-RNJJOU	WO2020041331A1_68	.	CC1=C(C2=CC=C([C@H](C)NC(=O)C3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(OCCOCCOC4=CC=C(CN5C(=O)/C(=C\C=C\C6=CC=C([N+](=O)[O-])C=C6)C6=C5C=CC=C6)C=C4)=NO3)C(C)C)C=C2)SC=N1	C53H54N6O10S	α-syn	P37840	VHL	WO-2020041331-A1
TPD-K1HBAK	WO2020041331A1_69	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3=CC(OCCOCCOCCOCCOC4=CC=C(CN5C(=O)/C(=C/C=C/C6=CC=C(NOO)C=C6)C6=C5C=CC=C6)C=C4)=NO3)C(C)C)C=C2)SC=N1	C57H64N6O12S	α-syn	P37840	VHL	WO-2020041331-A1
TPD-AVYFRZ	SCHEMBL26018026	(2S,4R)-4-hydroxy-1-[(2R)-3-methyl-2-[3-[2-[2-[2-[2-[4-[[(3E)-3-[(E)-3-(4-nitrophenyl)prop-2-enylidene]-2-oxoindol-1-yl]methyl]phenoxy]ethoxy]ethoxy]ethoxy]ethoxy]-1,2-oxazol-5-yl]butanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL30497572	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(OCCOCCOCCOCCOC4=CC=C(CN5C(=O)/C(=C/C=C/C6=CC=C([N+](=O)[O-])C=C6)C6=C5C=CC=C6)C=C4)=NO3)C(C)C)C=C2)SC=N1	C57H62N6O12S	α-syn	P37840	VHL	WO-2020041331-A1
TPD-YZ5VWU	SCHEMBL26018027	(2S,4R)-4-hydroxy-1-[(2S)-3-methyl-2-[3-[2-[2-[2-[2-[4-[[(3Z)-3-[(E)-3-(4-nitrophenyl)prop-2-enylidene]-2-oxoindol-1-yl]methyl]phenoxy]ethoxy]ethoxy]ethoxy]ethoxy]-1,2-oxazol-5-yl]butanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL30497587	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3=CC(OCCOCCOCCOCCOC4=CC=C(CN5C(=O)/C(=C\C=C\C6=CC=C([N+](=O)[O-])C=C6)C6=C5C=CC=C6)C=C4)=NO3)C(C)C)C=C2)SC=N1	C57H62N6O12S	α-syn	P37840	VHL	WO-2020041331-A1
TPD-HJT0V1	SCHEMBL26018029	(2S,4R)-4-hydroxy-1-[(2R)-3-methyl-2-[3-[2-[2-[2-[2-[4-[[(3Z)-3-[(E)-3-(4-nitrophenyl)prop-2-enylidene]-2-oxoindol-1-yl]methyl]phenoxy]ethoxy]ethoxy]ethoxy]ethoxy]-1,2-oxazol-5-yl]butanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL30497546	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(OCCOCCOCCOCCOC4=CC=C(CN5C(=O)/C(=C\C=C\C6=CC=C([N+](=O)[O-])C=C6)C6=C5C=CC=C6)C=C4)=NO3)C(C)C)C=C2)SC=N1	C57H62N6O12S	α-syn	P37840	VHL	WO-2020041331-A1
TPD-ZEW8DR	WO2020041331A1_73	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3=CC(OCCOCCOCCOC4=CC=C(CN5C(=O)/C(=C/C=C/C6=CC=C(NOO)C=C6)C6=C5C=CC=C6)C=C4)=NO3)C(C)C)C=C2)SC=N1	C55H60N6O11S	α-syn	P37840	VHL	WO-2020041331-A1
TPD-PIVLVP	WO2020041331A1_74	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(OCCOCCOCCOC4=CC=C(CN5C(=O)/C(=C/C=C/C6=CC=C(NOO)C=C6)C6=C5C=CC=C6)C=C4)=NO3)C(C)C)C=C2)SC=N1	C55H60N6O11S	α-syn	P37840	VHL	WO-2020041331-A1
TPD-F501UL	SCHEMBL26018030	(2S,4R)-4-hydroxy-1-[(2S)-3-methyl-2-[3-[2-[2-[2-[4-[[(3Z)-3-[(E)-3-(4-nitrophenyl)prop-2-enylidene]-2-oxoindol-1-yl]methyl]phenoxy]ethoxy]ethoxy]ethoxy]-1,2-oxazol-5-yl]butanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL30497575	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3=CC(OCCOCCOCCOC4=CC=C(CN5C(=O)/C(=C\C=C\C6=CC=C([N+](=O)[O-])C=C6)C6=C5C=CC=C6)C=C4)=NO3)C(C)C)C=C2)SC=N1	C55H58N6O11S	α-syn	P37840	VHL	WO-2020041331-A1
TPD-CNJY0B	SCHEMBL26018031	(2S,4R)-4-hydroxy-1-[(2R)-3-methyl-2-[3-[2-[2-[2-[4-[[(3Z)-3-[(E)-3-(4-nitrophenyl)prop-2-enylidene]-2-oxoindol-1-yl]methyl]phenoxy]ethoxy]ethoxy]ethoxy]-1,2-oxazol-5-yl]butanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL30497534	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(OCCOCCOCCOC4=CC=C(CN5C(=O)/C(=C\C=C\C6=CC=C([N+](=O)[O-])C=C6)C6=C5C=CC=C6)C=C4)=NO3)C(C)C)C=C2)SC=N1	C55H58N6O11S	α-syn	P37840	VHL	WO-2020041331-A1
TPD-CSSYTT	WO2020041331A1_77	.	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCCO[C@H]5C[C@H](OC6=CC=C(CN7C(=O)/C(=C/C=C/C8=CC=C(NOO)C=C8)C8=C7C=CC=C8)C=C6)C5)CC4)C=C3C2=O)C(=O)N1	C48H48N6O9	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-IKF68U	SCHEMBL26018033	2-(2,6-dioxopiperidin-3-yl)-5-[4-[3-[3-[4-[[(3Z)-3-[(E)-3-(4-nitrophenyl)prop-2-enylidene]-2-oxoindol-1-yl]methyl]phenoxy]cyclobutyl]oxypropyl]piperazin-1-yl]isoindole-1,3-dione; SCHEMBL30497542	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCCO[C@H]5C[C@H](OC6=CC=C(CN7C(=O)/C(=C\C=C\C8=CC=C([N+](=O)[O-])C=C8)C8=C7C=CC=C8)C=C6)C5)CC4)C=C3C2=O)C(=O)N1	C48H46N6O9	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-X95IIG	WO2020041331A1_79	.	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCN5CCC(O[C@H]6C[C@H](OC7=CC=C(CN8C(=O)/C(=C/C=C/C9=CC=C(NOO)C=C9)C9=C8C=CC=C9)C=C7)C6)CC5)CC4)C=C3C2=O)C(=O)N1	C52H55N7O9	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-1ARME7	SCHEMBL26018038	2-(2,6-dioxopiperidin-3-yl)-5-[4-[2-[4-[3-[4-[[(3Z)-3-[(E)-3-(4-nitrophenyl)prop-2-enylidene]-2-oxoindol-1-yl]methyl]phenoxy]cyclobutyl]oxypiperidin-1-yl]ethyl]piperazin-1-yl]isoindole-1,3-dione; SCHEMBL30497566	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCN5CCC(O[C@H]6C[C@H](OC7=CC=C(CN8C(=O)/C(=C\C=C\C9=CC=C([N+](=O)[O-])C=C9)C9=C8C=CC=C9)C=C7)C6)CC5)CC4)C=C3C2=O)C(=O)N1	C52H53N7O9	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-B3R1J9	WO2020041331A1_81	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3=CC(N4CCN(CCC5CCN(C6=CC7=C(C=C6)NC6=C(C=C(NOO)C=C6)S7)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C48H59N9O6S2	α-syn	P37840	VHL	WO-2020041331-A1
TPD-9AFH8D	WO2020041331A1_82	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCN(CCC5CCN(C6=CC7=C(C=C6)NC6=C(C=C(NOO)C=C6)S7)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C48H59N9O6S2	α-syn	P37840	VHL	WO-2020041331-A1
TPD-7161H5	WO2020041331A1_83	.	O=C1CCC(N2C(=O)C3=C(C=C(N4CCN(CCC5CCN(C6=CC7=C(C=C6)NC6=C(C=C(NOO)C=C6)S7)CC5)CC4)C=C3)C2=O)C(=O)N1	C36H39N7O6S	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-SE4J9X	WO2020041331A1_84	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3=CC(N4CCN(CCCO[C@H]5C[C@H](OC6=CC7=C(C=C6)NC6=C(C=C(NOO)C=C6)S7)C5)CC4)=NO3)C(C)C)C=C2)SC=N1	C48H58N8O8S2	α-syn	P37840	VHL	WO-2020041331-A1
TPD-JHAX7D	WO2020041331A1_85	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCN(CCCO[C@H]5C[C@H](OC6=CC7=C(C=C6)NC6=C(C=C(NOO)C=C6)S7)C5)CC4)=NO3)C(C)C)C=C2)SC=N1	C48H58N8O8S2	α-syn	P37840	VHL	WO-2020041331-A1
TPD-JBZ5LN	SCHEMBL21771298	4-[2-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxyethoxy]ethoxy]ethoxy]-2-fluoro-N-[4-(4-pyridin-2-ylpiperazin-1-yl)phenyl]benzamide	O=C1CCC(N2C(=O)C3=CC=C(OCCOCCOCCOC4=CC=C(C(=O)NC5=CC=C(N6CCN(C7=NC=CC=C7)CC6)C=C5)C(F)=C4)C=C3C2=O)C(=O)N1	C41H41FN6O9	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-WO1FJC	SCHEMBL21771294	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[2-[3-fluoro-4-[[4-(4-pyridin-2-ylpiperazin-1-yl)phenyl]carbamoyl]phenoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOC3=CC=C(C(=O)NC4=CC=C(N5CCN(C6=NC=CC=C6)CC5)C=C4)C(F)=C3)C(C)(C)C)C=C2)SC=N1	C53H65FN8O9S	α-syn	P37840	VHL	WO-2020041331-A1
TPD-IEQUJI	SCHEMBL21771290	4-[4-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]ethyl]piperidin-1-yl]-2-fluoro-N-[4-(4-pyridin-2-ylpiperazin-1-yl)phenyl]benzamide	O=C1CCC(N2C(=O)C3=C(C=C(N4CCN(CCC5CCN(C6=CC=C(C(=O)NC7=CC=C(N8CCN(C9=NC=CC=C9)CC8)C=C7)C(F)=C6)CC5)CC4)C=C3)C2=O)C(=O)N1	C46H50FN9O5	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-HL5CQ6	SCHEMBL21771537	(2S,4R)-1-[(2R)-2-[3-[4-[2-[1-[3-fluoro-4-[[4-(4-pyridin-2-ylpiperazin-1-yl)phenyl]carbamoyl]phenyl]piperidin-4-yl]ethyl]piperazin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCN(CCC5CCN(C6=CC=C(C(=O)NC7=CC=C(N8CCN(C9=NC=CC=C9)CC8)C=C7)C(F)=C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C58H70FN11O5S	α-syn	P37840	VHL	WO-2020041331-A1
TPD-1M46GA	SCHEMBL21771532	4-[3-[1-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]ethyl]piperidin-4-yl]oxycyclobutyl]oxy-2-fluoro-N-[4-(4-pyridin-2-ylpiperazin-1-yl)phenyl]benzamide	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCN5CCC(O[C@H]6C[C@H](OC7=CC=C(C(=O)NC8=CC=C(N9CCN(C%10=NC=CC=C%10)CC9)C=C8)C(F)=C7)C6)CC5)CC4)C=C3C2=O)C(=O)N1	C50H56FN9O7	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-G0GQKT	SCHEMBL21771538	4-[3-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]propoxy]cyclobutyl]oxy-2-fluoro-N-[4-(4-pyridin-2-ylpiperazin-1-yl)phenyl]benzamide	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCCO[C@H]5C[C@H](OC6=CC=C(C(=O)NC7=CC=C(N8CCN(C9=NC=CC=C9)CC8)C=C7)C(F)=C6)C5)CC4)C=C3C2=O)C(=O)N1	C46H49FN8O7	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-ZQUKBC	SCHEMBL21771536	4-[3-[1-[5-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxypentyl]piperidin-4-yl]oxycyclobutyl]oxy-2-fluoro-N-[4-(4-pyridin-2-ylpiperazin-1-yl)phenyl]benzamide	O=C1CCC(N2C(=O)C3=C(C=C(OCCCCCN4CCC(O[C@H]5C[C@H](OC6=CC=C(C(=O)NC7=CC=C(N8CCN(C9=NC=CC=C9)CC8)C=C7)C(F)=C6)C5)CC4)C=C3)C2=O)C(=O)N1	C49H54FN7O8	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-6J24P3	SCHEMBL21771533	2-(2,6-dioxopiperidin-3-yl)-5-[2-[2-[2-[4-[(E)-2-[5-(1,3-thiazol-2-yl)-1,2-oxazol-3-yl]ethenyl]phenoxy]ethoxy]ethoxy]ethoxy]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC=C(OCCOCCOCCOC4=CC=C(/C=C/C5=NOC(C6=NC=CS6)=C5)C=C4)C=C3C2=O)C(=O)N1	C33H30N4O9S	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-FPYWAY	SCHEMBL21771146	(2S,4R)-1-[(2S)-3,3-dimethyl-2-[[2-[2-[2-[2-[4-[(E)-2-[5-(1,3-thiazol-2-yl)-1,2-oxazol-3-yl]ethenyl]phenoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]butanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOC3=CC=C(/C=C/C4=NOC(C5=NC=CS5)=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C45H54N6O9S2	α-syn	P37840	VHL	WO-2020041331-A1
TPD-VOCF17	SCHEMBL21771148	2-(2,6-dioxopiperidin-3-yl)-5-[4-[2-[1-[4-[(E)-2-[5-(1,3-thiazol-2-yl)-1,2-oxazol-3-yl]ethenyl]phenyl]piperidin-4-yl]ethyl]piperazin-1-yl]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=C(C=C(N4CCN(CCC5CCN(C6=CC=C(/C=C/C7=NOC(C8=NC=CS8)=C7)C=C6)CC5)CC4)C=C3)C2=O)C(=O)N1	C38H39N7O5S	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-TY75R7	SCHEMBL21771147	(2S,4R)-4-hydroxy-1-[(2R)-3-methyl-2-[3-[4-[2-[1-[4-[(E)-2-[5-(1,3-thiazol-2-yl)-1,2-oxazol-3-yl]ethenyl]phenyl]piperidin-4-yl]ethyl]piperazin-1-yl]-1,2-oxazol-5-yl]butanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCN(CCC5CCN(C6=CC=C(/C=C/C7=NOC(C8=NC=CS8)=C7)C=C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C50H59N9O5S2	α-syn	P37840	VHL	WO-2020041331-A1
TPD-D6ZR2O	SCHEMBL21771150	2-(2,6-dioxopiperidin-3-yl)-5-[4-[2-[4-[3-[4-[(E)-2-[5-(1,3-thiazol-2-yl)-1,2-oxazol-3-yl]ethenyl]phenoxy]cyclobutyl]oxypiperidin-1-yl]ethyl]piperazin-1-yl]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCN5CCC(O[C@H]6C[C@H](OC7=CC=C(/C=C/C8=NOC(C9=NC=CS9)=C8)C=C7)C6)CC5)CC4)C=C3C2=O)C(=O)N1	C42H45N7O7S	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-ZDUIAR	SCHEMBL21771151	2-(2,6-dioxopiperidin-3-yl)-5-[4-[3-[3-[4-[(E)-2-[5-(1,3-thiazol-2-yl)-1,2-oxazol-3-yl]ethenyl]phenoxy]cyclobutyl]oxypropyl]piperazin-1-yl]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCCO[C@H]5C[C@H](OC6=CC=C(/C=C/C7=NOC(C8=NC=CS8)=C7)C=C6)C5)CC4)C=C3C2=O)C(=O)N1	C38H38N6O7S	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-L5YC5S	SCHEMBL21771149	2-(2,6-dioxopiperidin-3-yl)-5-[5-[4-[3-[4-[(E)-2-[5-(1,3-thiazol-2-yl)-1,2-oxazol-3-yl]ethenyl]phenoxy]cyclobutyl]oxypiperidin-1-yl]pentoxy]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=C(C=C(OCCCCCN4CCC(O[C@H]5C[C@H](OC6=CC=C(/C=C/C7=NOC(C8=NC=CS8)=C7)C=C6)C5)CC4)C=C3)C2=O)C(=O)N1	C41H43N5O8S	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-YTVQ64	SCHEMBL26040838	2-(2,6-dioxopiperidin-3-yl)-5-[2-[2-[2-[(3-nitro-10H-pyrido[3,2-b][1,4]benzothiazin-7-yl)oxy]ethoxy]ethoxy]ethoxy]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC=C(OCCOCCOCCOC4=CC5=C(C=C4)NC4=NC=C([N+](=O)[O-])C=C4S5)C=C3C2=O)C(=O)N1	C30H27N5O10S	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-PQMJWE	WO2020041331A1_101	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOC3=CC4=C(C=C3)NC3=NC=C(NOO)C=C3S4)C(C)(C)C)C=C2)SC=N1	C42H53N7O10S2	α-syn	P37840	VHL	WO-2020041331-A1
TPD-EJCU2W	WO2020041331A1_102	.	O=C1CCC(N2C(=O)C3=C(C=C(N4CCN(CCC5CCN(C6=CC7=C(C=C6)NC6=NC=C(NOO)C=C6S7)CC5)CC4)C=C3)C2=O)C(=O)N1	C35H38N8O6S	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-6AZ901	WO2020041331A1_103	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCN(CCC5CCN(C6=CC7=C(C=C6)NC6=NC=C(NOO)C=C6S7)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C47H58N10O6S2	α-syn	P37840	VHL	WO-2020041331-A1
TPD-FWESHH	WO2020041331A1_104	.	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCN5CCC(O[C@H]6C[C@H](OC7=CC8=C(C=C7)NC7=NC=C(NOO)C=C7S8)C6)CC5)CC4)C=C3C2=O)C(=O)N1	C39H44N8O8S	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-3FC87C	WO2020041331A1_105	.	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCCO[C@H]5C[C@H](OC6=CC7=C(C=C6)NC6=NC=C(NOO)C=C6S7)C5)CC4)C=C3C2=O)C(=O)N1	C35H37N7O8S	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-2QZKAF	WO2020041331A1_106	.	O=C1CCC(N2C(=O)C3=C(C=C(OCCCCCN4CCC(O[C@H]5C[C@H](OC6=CC7=C(C=C6)NC6=NC=C(NOO)C=C6S7)C5)CC4)C=C3)C2=O)C(=O)N1	C38H42N6O9S	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-0DC5TB	SCHEMBL21771353	N-[4-[2-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxyethoxy]ethoxy]ethoxy]naphthalen-1-yl]thiophene-2-sulfonamide	O=C1CCC(N2C(=O)C3=C(C=C(OCCOCCOCCOC4=C5C=CC=CC5=C(NS(=O)(=O)C5=CC=CS5)C=C4)C=C3)C2=O)C(=O)N1	C33H31N3O10S2	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-VKH74U	SCHEMBL21771355	(2S,4R)-1-[(2S)-3,3-dimethyl-2-[[2-[2-[2-[4-(thiophen-2-ylsulfonylamino)naphthalen-1-yl]oxyethoxy]ethoxy]acetyl]amino]butanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOC3=C4C=CC=CC4=C(NS(=O)(=O)C4=CC=CS4)C=C3)C(C)(C)C)C=C2)SC=N1	C43H51N5O9S3	α-syn	P37840	VHL	WO-2020041331-A1
TPD-LF94O3	SCHEMBL21771356	N-[3-[[1-[2-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxyethoxy]ethoxy]ethyl]-1,2,4-triazol-3-yl]sulfanyl]-4-hydroxynaphthalen-1-yl]thiophene-2-sulfonamide	O=C1CCC(N2C(=O)C3=C(C=C(OCCOCCOCCN4C=NC(SC5=CC(NS(=O)(=O)C6=CC=CS6)=C6C=CC=CC6=C5O)=N4)C=C3)C2=O)C(=O)N1	C35H32N6O10S3	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-6DUMDZ	SCHEMBL21771357	(2S,4R)-4-hydroxy-1-[(2S)-2-[[2-[2-[2-[2-[3-[1-hydroxy-4-(thiophen-2-ylsulfonylamino)naphthalen-2-yl]sulfanyl-1,2,4-triazol-1-yl]ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCN3C=NC(SC4=CC(NS(=O)(=O)C5=CC=CS5)=C5C=CC=CC5=C4O)=N3)C(C)(C)C)C=C2)SC=N1	C47H56N8O10S4	α-syn	P37840	VHL	WO-2020041331-A1
TPD-R7OF23	SCHEMBL21771564	4-[2-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxyethoxy]ethoxy]ethoxy]-N-[4-(4-pyridin-3-ylpiperazin-1-yl)phenyl]benzamide	O=C1CCC(N2C(=O)C3=CC=C(OCCOCCOCCOC4=CC=C(C(=O)NC5=CC=C(N6CCN(C7=CC=CN=C7)CC6)C=C5)C=C4)C=C3C2=O)C(=O)N1	C41H42N6O9	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-BYGKHX	SCHEMBL21771566	N-[4-[4-(5-cyanopyridin-2-yl)piperazin-1-yl]phenyl]-4-[2-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxyethoxy]ethoxy]ethoxy]benzamide	N#CC1=CC=C(N2CCN(C3=CC=C(NC(=O)C4=CC=C(OCCOCCOCCOC5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C=C4)C=C3)CC2)N=C1	C42H41N7O9	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-FJD7FK	SCHEMBL21771568	(2S,4R)-1-[(2S)-3,3-dimethyl-2-[[2-[2-[2-[2-[4-[[4-(4-pyridin-2-ylpiperazin-1-yl)phenyl]carbamoyl]phenoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]butanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOC3=CC=C(C(=O)NC4=CC=C(N5CCN(C6=CC=CC=N6)CC5)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C53H66N8O9S	α-syn	P37840	VHL	WO-2020041331-A1
TPD-1OLASI	SCHEMBL21771559	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[2-[4-[[4-[4-(5-cyanopyridin-2-yl)piperazin-1-yl]phenyl]carbamoyl]phenoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOC3=CC=C(C(=O)NC4=CC=C(N5CCN(C6=CC=C(C#N)C=N6)CC5)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C54H65N9O9S	α-syn	P37840	VHL	WO-2020041331-A1
TPD-3RQV6F	SCHEMBL21771562	(2S,4R)-1-[(2S)-3,3-dimethyl-2-[[2-[2-[2-[2-[4-[[4-(4-pyridin-3-ylpiperazin-1-yl)phenyl]carbamoyl]phenoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]butanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOC3=CC=C(C(=O)NC4=CC=C(N5CCN(C6=CC=CN=C6)CC5)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C53H66N8O9S	α-syn	P37840	VHL	WO-2020041331-A1
TPD-DA5Z0R	WO2020041331A1_116	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOC3=CC=C(C4=CC5=C(C=C4)N=C(C4=CN=C(N6CCCC6)C=C4)S5)C=N3)C(C)(C)C)C=C2)SC=C1	C53H63N7O8S2	α-syn	P37840	VHL	WO-2020041331-A1
TPD-LG1ZPK	SCHEMBL21771289	(2S,4R)-1-[(2S)-3,3-dimethyl-2-[[2-[2-[2-[2-[1-[5-(6-pyridin-3-yl-1,3-benzothiazol-2-yl)pyridin-2-yl]pyrrolidin-3-yl]oxyethoxy]ethoxy]ethoxy]acetyl]amino]butanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOC3CCN(C4=NC=C(C5=NC6=C(C=C(C7=CC=CN=C7)C=C6)S5)C=C4)C3)C(C)(C)C)C=C2)SC=N1	C52H62N8O8S2	α-syn	P37840	VHL	WO-2020041331-A1
TPD-VDJMS3	SCHEMBL21771293	(2S,4R)-1-[(2S)-3,3-dimethyl-2-[[2-[2-[2-[2-[3-oxo-4-[2-(6-pyrrolidin-1-ylpyridin-3-yl)-1,3-benzothiazol-6-yl]piperazin-1-yl]ethoxy]ethoxy]ethoxy]acetyl]amino]butanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCN3CCN(C4=CC5=C(C=C4)N=C(C4=CN=C(N6CCCC6)C=C4)S5)C(=O)C3)C(C)(C)C)C=C2)SC=N1	C51H65N9O8S2	α-syn	P37840	VHL	WO-2020041331-A1
TPD-DD3UX6	SCHEMBL21771296	(2S,4R)-1-[(2S)-3,3-dimethyl-2-[[2-[2-[2-[2-[1-[5-[6-(4-methyl-2-oxopiperazin-1-yl)-1,3-benzothiazol-2-yl]pyridin-2-yl]pyrrolidin-3-yl]oxyethoxy]ethoxy]ethoxy]acetyl]amino]butanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOC3CCN(C4=NC=C(C5=NC6=C(C=C(N7CCN(C)CC7=O)C=C6)S5)C=C4)C3)C(C)(C)C)C=C2)SC=N1	C52H67N9O9S2	α-syn	P37840	VHL	WO-2020041331-A1
TPD-S3ND5T	SCHEMBL21771297	(2S,4R)-1-[(2S)-3,3-dimethyl-2-[[2-[2-[2-[2-[1-[5-(5-pyridin-3-yl-1,3-benzothiazol-2-yl)pyridin-2-yl]pyrrolidin-3-yl]oxyethoxy]ethoxy]ethoxy]acetyl]amino]butanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOC3CCN(C4=NC=C(C5=NC6=C(C=CC(C7=CC=CN=C7)=C6)S5)C=C4)C3)C(C)(C)C)C=C2)SC=N1	C52H62N8O8S2	α-syn	P37840	VHL	WO-2020041331-A1
TPD-DMRTC8	SCHEMBL21771291	(2S,4R)-1-[(2S)-3,3-dimethyl-2-[[2-[2-[2-[2-[5-[2-(6-pyrrolidin-1-ylpyridin-3-yl)-1,3-benzothiazol-5-yl]pyridin-2-yl]oxyethoxy]ethoxy]ethoxy]acetyl]amino]butanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOC3=CC=C(C4=CC5=C(C=C4)SC(C4=CN=C(N6CCCC6)C=C4)=N5)C=N3)C(C)(C)C)C=C2)SC=N1	C52H62N8O8S2	α-syn	P37840	VHL	WO-2020041331-A1
TPD-HM539P	SCHEMBL21771352	(2S,4R)-1-[(2S)-3,3-dimethyl-2-[[2-[2-[2-[2-[1-[5-(2-pyridin-3-ylthieno[2,3-b]pyridin-6-yl)pyridin-2-yl]pyrrolidin-3-yl]oxyethoxy]ethoxy]ethoxy]acetyl]amino]butanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOC3CCN(C4=CC=C(C5=CC=C6C=C(C7=CC=CN=C7)SC6=N5)C=N4)C3)C(C)(C)C)C=C2)SC=N1	C52H62N8O8S2	α-syn	P37840	VHL	WO-2020041331-A1
TPD-0FB9QH	SCHEMBL21771349	(2S,4R)-1-[(2S)-3,3-dimethyl-2-[[2-[2-[2-[2-[5-[6-(6-pyrrolidin-1-ylpyridin-3-yl)thieno[2,3-b]pyridin-2-yl]pyridin-2-yl]oxyethoxy]ethoxy]ethoxy]acetyl]amino]butanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOC3=CC=C(C4=CC5=CC=C(C6=CC=C(N7CCCC7)N=C6)N=C5S4)C=N3)C(C)(C)C)C=C2)SC=N1	C52H62N8O8S2	α-syn	P37840	VHL	WO-2020041331-A1
TPD-VNP33F	SCHEMBL21771347	2-(2,6-Dioxopiperidin-3-yl)-5-[2-[2-[2-[1-[5-(4-oxo-5-pyridin-3-yl-6,7-dihydro-[1,3]thiazolo[5,4-c]pyridin-2-yl)pyridin-2-yl]pyrrolidin-3-yl]oxyethoxy]ethoxy]ethoxy]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=C(C=C(OCCOCCOCCOC4CCN(C5=NC=C(C6=NC7=C(S6)C(=O)N(C6=CC=CN=C6)CC7)C=C5)C4)C=C3)C2=O)C(=O)N1	C39H39N7O9S	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-JMPB4V	SCHEMBL21771351	2-(2,6-Dioxopiperidin-3-yl)-5-[2-[2-[2-[5-[4-oxo-2-(6-pyrrolidin-1-ylpyridin-3-yl)-6,7-dihydro-[1,3]thiazolo[5,4-c]pyridin-5-yl]pyridin-2-yl]oxyethoxy]ethoxy]ethoxy]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=C(C=C(OCCOCCOCCOC4=CC=C(N5CCC6=C(SC(C7=CN=C(N8CCCC8)C=C7)=N6)C5=O)C=N4)C=C3)C2=O)C(=O)N1	C39H39N7O9S	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-T8D3K7	SCHEMBL21771354	(2S,4R)-1-[(2S)-3,3-dimethyl-2-[[2-[2-[2-[2-[1-[5-(4-oxo-5-pyridin-3-yl-6,7-dihydro-[1,3]thiazolo[5,4-c]pyridin-2-yl)pyridin-2-yl]pyrrolidin-3-yl]oxyethoxy]ethoxy]ethoxy]acetyl]amino]butanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOC3CCN(C4=NC=C(C5=NC6=C(S5)C(=O)N(C5=CC=CN=C5)CC6)C=C4)C3)C(C)(C)C)C=C2)SC=N1	C51H63N9O9S2	α-syn	P37840	VHL	WO-2020041331-A1
TPD-YNA8T6	SCHEMBL21771345	(2S,4R)-1-[(2S)-3,3-dimethyl-2-[[2-[2-[2-[2-[5-[4-oxo-2-(6-pyrrolidin-1-ylpyridin-3-yl)-6,7-dihydro-[1,3]thiazolo[5,4-c]pyridin-5-yl]pyridin-2-yl]oxyethoxy]ethoxy]ethoxy]acetyl]amino]butanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOC3=CC=C(N4CCC5=C(SC(C6=CN=C(N7CCCC7)C=C6)=N5)C4=O)C=N3)C(C)(C)C)C=C2)SC=N1	C51H63N9O9S2	α-syn	P37840	VHL	WO-2020041331-A1
TPD-W8VBDA	SCHEMBL21771555	2-(2,6-Dioxopiperidin-3-yl)-5-[2-[2-[2-[5-[6-(6-pyrrolidin-1-ylpyridin-3-yl)thieno[2,3-b]pyridin-2-yl]pyridin-2-yl]oxyethoxy]ethoxy]ethoxy]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC=C(OCCOCCOCCOC4=CC=C(C5=CC6=CC=C(C7=CC=C(N8CCCC8)N=C7)N=C6S5)C=N4)C=C3C2=O)C(=O)N1	C40H38N6O8S	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-ST38GL	SCHEMBL21771548	2-(2,6-Dioxopiperidin-3-yl)-5-[2-[2-[2-[1-[5-(2-pyridin-3-ylthieno[2,3-b]pyridin-6-yl)pyridin-2-yl]pyrrolidin-3-yl]oxyethoxy]ethoxy]ethoxy]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC=C(OCCOCCOCCOC4CCN(C5=CC=C(C6=CC=C7C=C(C8=CC=CN=C8)SC7=N6)C=N5)C4)C=C3C2=O)C(=O)N1	C40H38N6O8S	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-8VR0A7	SCHEMBL21771550	2-(2,6-Dioxopiperidin-3-yl)-5-[2-[2-[2-[5-[2-(6-pyrrolidin-1-ylpyridin-3-yl)-1,3-benzothiazol-5-yl]pyridin-2-yl]oxyethoxy]ethoxy]ethoxy]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=C(C=C(OCCOCCOCCOC4=CC=C(C5=CC6=C(C=C5)SC(C5=CN=C(N7CCCC7)C=C5)=N6)C=N4)C=C3)C2=O)C(=O)N1	C40H38N6O8S	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-2I93PB	SCHEMBL21771554	2-(2,6-Dioxopiperidin-3-yl)-5-[2-[2-[2-[1-[5-(5-pyridin-3-yl-1,3-benzothiazol-2-yl)pyridin-2-yl]pyrrolidin-3-yl]oxyethoxy]ethoxy]ethoxy]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=C(C=C(OCCOCCOCCOC4CCN(C5=NC=C(C6=NC7=C(C=CC(C8=CC=CN=C8)=C7)S6)C=C5)C4)C=C3)C2=O)C(=O)N1	C40H38N6O8S	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-DIX5EX	SCHEMBL21771551	2-(2,6-Dioxopiperidin-3-yl)-5-[2-[2-[2-[5-[2-(6-pyrrolidin-1-ylpyridin-3-yl)-1,3-benzothiazol-6-yl]pyridin-2-yl]oxyethoxy]ethoxy]ethoxy]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=C(C=C(OCCOCCOCCOC4=CC=C(C5=CC6=C(C=C5)N=C(C5=CN=C(N7CCCC7)C=C5)S6)C=N4)C=C3)C2=O)C(=O)N1	C40H38N6O8S	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-N15UMT	SCHEMBL21771556	2-(2,6-Dioxopiperidin-3-yl)-5-[2-[2-[2-[1-[5-(6-pyridin-3-yl-1,3-benzothiazol-2-yl)pyridin-2-yl]pyrrolidin-3-yl]oxyethoxy]ethoxy]ethoxy]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=C(C=C(OCCOCCOCCOC4CCN(C5=NC=C(C6=NC7=C(C=C(C8=CC=CN=C8)C=C7)S6)C=C5)C4)C=C3)C2=O)C(=O)N1	C40H38N6O8S	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-P5MIJE	SCHEMBL21771552	2-(2,6-Dioxopiperidin-3-yl)-5-[2-[2-[2-[3-oxo-4-[2-(6-pyrrolidin-1-ylpyridin-3-yl)-1,3-benzothiazol-6-yl]piperazin-1-yl]ethoxy]ethoxy]ethoxy]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=C(C=C(OCCOCCOCCN4CCN(C5=CC6=C(C=C5)N=C(C5=CN=C(N7CCCC7)C=C5)S6)C(=O)C4)C=C3)C2=O)C(=O)N1	C39H41N7O8S	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-YU3JAU	SCHEMBL21771557	2-(2,6-Dioxopiperidin-3-yl)-5-[2-[2-[2-[1-[5-[6-(4-methyl-2-oxopiperazin-1-yl)-1,3-benzothiazol-2-yl]pyridin-2-yl]pyrrolidin-3-yl]oxyethoxy]ethoxy]ethoxy]isoindole-1,3-dione	CN1CCN(C2=CC3=C(C=C2)N=C(C2=CN=C(N4CCC(OCCOCCOCCOC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)C=C2)S3)C(=O)C1	C40H43N7O9S	α-syn	P37840	CRBN	WO-2020041331-A1
TPD-RJ1AVX	SCHEMBL19475717	2-[8-(1,3-benzothiazol-2-ylcarbamoyl)-3,4-dihydro-1H-isoquinolin-2-yl]-5-[3-[4-[3-[4-[4-[4-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxymethyl]triazol-1-yl]butanoyl]piperazin-1-yl]prop-1-ynyl]-2-fluorophenoxy]propyl]-1,3-thiazole-4-carboxylic acid; PD142081	O=C1CCC(N2C(=O)C3=CC=CC(NCCOCCOCCOCC4=CN(CCCC(=O)N5CCN(CC#CC6=CC(F)=C(OCCCC7=C(C(=O)O)N=C(N8CCC9=CC=CC(C(=O)NC%10=NC%11=C(C=CC=C%11)S%10)=C9C8)S7)C=C6)CC5)N=N4)=C3C2=O)C(=O)N1	C63H65FN12O12S2	BCL2L1	Q07817	CRBN	WO-2020081880-A1
TPD-UN4HMW	SCHEMBL19503633	2-[8-(1,3-benzothiazol-2-ylcarbamoyl)-3,4-dihydro-1H-isoquinolin-2-yl]-5-[3-[4-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxymethyl]triazol-1-yl]propyl]-1,3-thiazole-4-carboxylic acid	O=C1CCC(N2C(=O)C3=CC=CC(NCCOCCOCCOCC4=CN(CCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)N=N4)=C3C2=O)C(=O)N1	C46H46N10O10S2	BCL2L1	Q07817	CRBN	WO-2020081880-A1
TPD-Q6HBMU	SCHEMBL19475829	2-[8-(1,3-benzothiazol-2-ylcarbamoyl)-3,4-dihydro-1H-isoquinolin-2-yl]-5-[3-[4-[3-[4-[4-[4-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]-2-oxoethoxy]ethoxy]ethoxymethyl]triazol-1-yl]butanoyl]piperazin-1-yl]prop-1-ynyl]-2-fluorophenoxy]propyl]-1,3-thiazole-4-carboxylic acid; PD142079	O=C1CCC(N2CC3=C(NC(=O)COCCOCCOCC4=CN(CCCC(=O)N5CCN(CC#CC6=CC(F)=C(OCCCC7=C(C(=O)O)N=C(N8CCC9=CC=CC(C(=O)NC%10=NC%11=C(C=CC=C%11)S%10)=C9C8)S7)C=C6)CC5)N=N4)C=CC=C3C2=O)C(=O)N1	C63H65FN12O12S2	BCL2L1	Q07817	CRBN	WO-2020081880-A1
TPD-6YBEG7	orb2813994	2-[8-(1,3-benzothiazol-2-ylcarbamoyl)-3,4-dihydro-1H-isoquinolin-2-yl]-5-[3-[4-[3-[4-[4-[4-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxymethyl]triazol-1-yl]butanoyl]piperazin-1-yl]prop-1-ynyl]-2-fluorophenoxy]propyl]-1,3-thiazole-4-carboxylic acid; CHEMBL4777606; SCHEMBL19475882; XZ424	O=C1CCC(N2C(=O)C3=CC=CC(NCCOCCOCC4=CN(CCCC(=O)N5CCN(CC#CC6=CC(F)=C(OCCCC7=C(C(=O)O)N=C(N8CCC9=CC=CC(C(=O)NC%10=NC%11=C(C=CC=C%11)S%10)=C9C8)S7)C=C6)CC5)N=N4)=C3C2=O)C(=O)N1	C61H61FN12O11S2	BCL2L1	Q07817	CRBN	WO-2020081880-A1
TPD-XLTX75	SCHEMBL19475870	4-[4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[(2R)-4-[4-[4-[4-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxymethyl]triazol-1-yl]butanoyl]piperazin-1-yl]-1-phenylsulfanylbutan-2-yl]amino]-3-(trifluoromethylsulfonyl)phenyl]sulfonylbenzamide; SCHEMBL19475878; XJPCOLHEXNGRQM-WNIUGPFTSA-N; 4-[4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[(2R)-4-[4-[4-[4-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxymethyl]triazol-1-yl]butanoyl]piperazin-1-yl]-1-phenylsulfanylbutan-2-yl]amino]-3-(trifluoromethylsulfonyl)phenyl]sulfonylbenzamide	CC1(C)CCC(C2=CC=C(Cl)C=C2)=C(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC(S(=O)(=O)C(F)(F)F)=C(N[C@H](CCN5CCN(C(=O)CCCN6C=C(COCCOCCOCCNC7=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=CC=C7)N=N6)CC5)CSC5=CC=CC=C5)C=C4)C=C3)CC2)C1	C73H86ClF3N12O13S3	BCL2L1	Q07817	CRBN	WO-2020081880-A1
TPD-KR3DTL	SCHEMBL19475757	2-[8-(1,3-benzothiazol-2-ylcarbamoyl)-3,4-dihydro-1H-isoquinolin-2-yl]-5-[3-[2-fluoro-4-[3-[4-[4-[4-[2-[2-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]ethoxy]ethoxymethyl]triazol-1-yl]butanoyl]piperazin-1-yl]prop-1-ynyl]phenoxy]propyl]-1,3-thiazole-4-carboxylic acid; SCHEMBL19475760	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCC3=CN(CCCC(=O)N4CCN(CC#CC5=CC(F)=C(OCCCC6=C(C(=O)O)N=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=C(C=CC=C%10)S9)=C8C7)S6)C=C5)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C72H82FN13O12S3	BCL2L1	Q07817	VHL	WO-2020081880-A1
TPD-JHXWGA	SCHEMBL19475796	4-[(3R)-3-[4-[[4-[4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]benzoyl]sulfamoyl]-2-(trifluoromethylsulfonyl)anilino]-4-phenylsulfanylbutyl]-N-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethyl]piperazine-1-carboxamide; HUJOFFBNGNRZLG-LKVFYHIZSA-N; PD142181; 4-[(3R)-3-[4-[[4-[4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]benzoyl]sulfamoyl]-2-(trifluoromethylsulfonyl)anilino]-4-phenylsulfanylbutyl]-N-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethyl]piperazine-1-carboxamide	CC1(C)CCC(C2=CC=C(Cl)C=C2)=C(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC(S(=O)(=O)C(F)(F)F)=C(N[C@H](CCN5CCN(C(=O)NCCOCCOCCNC6=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)CC5)CSC5=CC=CC=C5)C=C4)C=C3)CC2)C1	C67H78ClF3N10O12S3	BCL2L1	Q07817	CRBN	WO-2020081880-A1
TPD-85CZU2	SCHEMBL19475737	4-[4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[(2R)-4-[4-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]acetyl]piperazin-1-yl]-1-phenylsulfanylbutan-2-yl]amino]-3-(trifluoromethylsulfonyl)phenyl]sulfonylbenzamide; SCHEMBL19475744; PD142185	CC1(C)CCC(C2=CC=C(Cl)C=C2)=C(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC(S(=O)(=O)C(F)(F)F)=C(N[C@H](CCN5CCN(C(=O)COCCOCCOCCNC6=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)CC5)CSC5=CC=CC=C5)C=C4)C=C3)CC2)C1	C68H79ClF3N9O13S3	BCL2L1	Q07817	CRBN	WO-2020081880-A1
TPD-OMMPEC	SCHEMBL19475841	4-[4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[(2R)-4-[4-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]acetyl]piperazin-1-yl]-1-phenylsulfanylbutan-2-yl]amino]-3-(trifluoromethylsulfonyl)phenyl]sulfonylbenzamide; SCHEMBL19475852; VJVKHPKQMHHKQT-YJUSKGKKSA-N; PD142187; 4-[4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[(2R)-4-[4-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]acetyl]piperazin-1-yl]-1-phenylsulfanylbutan-2-yl]amino]-3-(trifluoromethylsulfonyl)phenyl]sulfonylbenzamide	CC1(C)CCC(C2=CC=C(Cl)C=C2)=C(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC(S(=O)(=O)C(F)(F)F)=C(N[C@H](CCN5CCN(C(=O)COCCOCCNC6=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)CC5)CSC5=CC=CC=C5)C=C4)C=C3)CC2)C1	C66H75ClF3N9O12S3	BCL2L1	Q07817	CRBN	WO-2020081880-A1
TPD-YLNTSN	SCHEMBL19475672	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]acetyl]piperidin-4-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC=C(NCC5CCN(C(=O)COCCOCCOCCNC6=CC=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C([N+](=O)[O-])=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C66H74ClN11O14S	BCL2L1	Q07817	CRBN	WO-2020081880-A1
TPD-P13BG8	SCHEMBL19475774	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[4-[4-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxymethyl]triazol-1-yl]butanoyl]piperidin-4-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC=C(NCC5CCN(C(=O)CCCN6C=C(COCCOCCOCCNC7=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=CC=C7)N=N6)CC5)C([N+](=O)[O-])=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C71H81ClN14O14S	BCL2L1	Q07817	CRBN	WO-2020081880-A1
TPD-W2NAZ5	SCHEMBL19475694	N-[2-[2-[2-[[4-[[4-[[4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzoyl]sulfamoyl]-2-nitroanilino]methyl]piperidine-1-carbonyl]amino]ethoxy]ethoxy]ethyl]-N'-[(2S)-1-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]butanediamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCC(=O)NCCOCCOCCNC(=O)N3CCC(CNC4=CC=C(S(=O)(=O)NC(=O)C5=CC=C(N6CCN(CC7=C(C8=CC=C(Cl)C=C8)CC(C)(C)CC7)CC6)C=C5OC5=CN=C6NC=CC6=C5)C=C4[N+](=O)[O-])CC3)C(C)(C)C)C=C2)SC=N1	C78H97ClN14O14S2	BCL2L1	Q07817	VHL	WO-2020081880-A1
TPD-WWE1JT	SCHEMBL19475705	N-[2-[2-[2-[[4-[(3R)-3-[4-[[4-[4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]benzoyl]sulfamoyl]-2-(trifluoromethylsulfonyl)anilino]-4-phenylsulfanylbutyl]piperazine-1-carbonyl]amino]ethoxy]ethoxy]ethyl]-N'-[(2S)-1-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]butanediamide; ZCDDZBYIYTWMLY-QAXPGBGFSA-N	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCC(=O)NCCOCCOCCNC(=O)N3CCN(CC[C@H](CSC4=CC=CC=C4)NC4=C(S(=O)(=O)C(F)(F)F)C=C(S(=O)(=O)NC(=O)C5=CC=C(N6CCN(CC7=C(C8=CC=C(Cl)C=C8)CCC(C)(C)C7)CC6)C=C5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C80H102ClF3N12O13S4	BCL2L1	Q07817	VHL	WO-2020081880-A1
TPD-PJV0CX	SCHEMBL19475656	4-[4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[(2R)-4-[4-[2-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethoxy]acetyl]piperazin-1-yl]-1-phenylsulfanylbutan-2-yl]amino]-3-(trifluoromethylsulfonyl)phenyl]sulfonylbenzamide; SCHEMBL19475661; PD142183	CC1(C)CCC(C2=CC=C(Cl)C=C2)=C(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC(S(=O)(=O)C(F)(F)F)=C(N[C@H](CCN5CCN(C(=O)COCCOCCOCCOCCNC6=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)CC5)CSC5=CC=CC=C5)C=C4)C=C3)CC2)C1	C70H83ClF3N9O14S3	BCL2L1	Q07817	CRBN	WO-2020081880-A1
TPD-FQLFXG	SCHEMBL19475863	4-[4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[(2R)-4-[4-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethyl]piperazin-1-yl]-1-phenylsulfanylbutan-2-yl]amino]-3-(trifluoromethylsulfonyl)phenyl]sulfonylbenzamide; SCHEMBL19475869; DYOGHZZIPKJNPD-LKVFYHIZSA-N; PD142175; 4-[4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[(2R)-4-[4-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethyl]piperazin-1-yl]-1-phenylsulfanylbutan-2-yl]amino]-3-(trifluoromethylsulfonyl)phenyl]sulfonylbenzamide	CC1(C)CCC(C2=CC=C(Cl)C=C2)=C(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC(S(=O)(=O)C(F)(F)F)=C(N[C@H](CCN5CCN(CCOCCOCCNC6=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)CC5)CSC5=CC=CC=C5)C=C4)C=C3)CC2)C1	C66H77ClF3N9O11S3	BCL2L1	Q07817	CRBN	WO-2020081880-A1
TPD-5ISMDQ	SCHEMBL19475682	4-[4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[(2R)-4-[4-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethyl]piperazin-1-yl]-1-phenylsulfanylbutan-2-yl]amino]-3-(trifluoromethylsulfonyl)phenyl]sulfonylbenzamide; SCHEMBL19475691; IYIOGVQABFXBJW-IQRNJRIOSA-N; PD142177; 4-[4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[(2R)-4-[4-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethyl]piperazin-1-yl]-1-phenylsulfanylbutan-2-yl]amino]-3-(trifluoromethylsulfonyl)phenyl]sulfonylbenzamide	CC1(C)CCC(C2=CC=C(Cl)C=C2)=C(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC(S(=O)(=O)C(F)(F)F)=C(N[C@H](CCN5CCN(CCOCCNC6=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)CC5)CSC5=CC=CC=C5)C=C4)C=C3)CC2)C1	C64H73ClF3N9O10S3	BCL2L1	Q07817	CRBN	WO-2020081880-A1
TPD-ET1VHY	WO2020081880A1_XZ15418	.	CC1(C)CCC(C2=CC=C(Cl)C=C2)=C(CC2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC(S(=O)(=O)C(F)(F)F)=C(N[C@H](CCN5CCN(CCOCCOCCOCCNC6=C7C(=O)C(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)CC5)CSC5=CC=CC=C5)C=C4)C=C3)CC2)C1	C70H83ClF3N7O12S3	BCL2L1	Q07817	CRBN	WO-2020081880-A1
TPD-J4XX7P	SCHEMBL19475665	4-[4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[(2R)-4-[4-[2-[4-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxymethyl]triazol-1-yl]acetyl]piperazin-1-yl]-1-phenylsulfanylbutan-2-yl]amino]-3-(trifluoromethylsulfonyl)phenyl]sulfonylbenzamide; SCHEMBL19475671; DYYRHXFGKFWYQO-QJKVXZADSA-N; 4-[4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[(2R)-4-[4-[2-[4-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxymethyl]triazol-1-yl]acetyl]piperazin-1-yl]-1-phenylsulfanylbutan-2-yl]amino]-3-(trifluoromethylsulfonyl)phenyl]sulfonylbenzamide	CC1(C)CCC(C2=CC=C(Cl)C=C2)=C(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC(S(=O)(=O)C(F)(F)F)=C(N[C@H](CCN5CCN(C(=O)CN6C=C(COCCOCCNC7=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=CC=C7)N=N6)CC5)CSC5=CC=CC=C5)C=C4)C=C3)CC2)C1	C69H78ClF3N12O12S3	BCL2L1	Q07817	CRBN	WO-2020081880-A1
TPD-3PTG8K	SCHEMBL24172484	N-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]-2-oxoethyl]-methylamino]ethyl]-2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyacetamide; AC-1-027	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(=O)CN(C)CCNC(=O)COc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)cn3)nc2n(C2CCCC2)c1=O	C44H49N11O9	CDK4;CDK6	P11802/Q00534	CRBN	WO-2020092662-A1
TPD-3LSYPY	AC-1-112	N-[2-[2-[2-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]-2-oxoethyl]amino]ethoxy]ethoxy]ethoxy]ethyl]-2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyacetamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(=O)CNCCOCCOCCOCCNC(=O)COc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)cn3)nc2n(C2CCCC2)c1=O	C49H59N11O12	CDK4;CDK6	P11802/Q00534	CRBN	WO-2020092662-A1
TPD-OFODJ4	SCHEMBL21635230	N-[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]ethyl]-2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyacetamide; SCHEMBL30339173; AC-1-212	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CCNC(=O)COc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)cn3)nc2n(C2CCCC2)c1=O	C41H44N10O8	CDK4;CDK6	P11802/Q00534	CRBN	WO-2020092662-A1
TPD-DPMWAY	SCHEMBL23779421	N-[6-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]hexyl]-2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyacetamide; PD142096	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CCCCCCNC(=O)COc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H52N10O8	CDK4;CDK6	P11802/Q00534	CRBN	WO-2020092662-A1
TPD-2R1XZM	SCHEMBL24172345	2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxy-N-[2-[4-[[6-[[5-fluoro-4-(7-fluoro-2-methyl-3-propan-2-ylbenzimidazol-5-yl)pyrimidin-2-yl]amino]pyridin-3-yl]methyl]piperazin-1-yl]ethyl]acetamide; PD140955	Cc1nc2c(F)cc(-c3nc(Nc4ccc(CN5CCN(CCNC(=O)COc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)cn4)ncc3F)cc2n1C(C)C	C42H43F2N11O6	CDK4;CDK6	P11802/Q00534	CRBN	WO-2020092662-A1
TPD-AG4HR9	YX-2-107	CID 166642460; 2417408-46-7; orb1982695; CHEMBL5281294; SCHEMBL24172331; AC-37780; BP-42228; DA-68793; HY-148530; CS-0634381; H38906; N-(4-((2-(4-(6-((6-Acetyl-8-cyclopentyl-5-methyl-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-2-yl)amino)pyridin-3-yl)piperazin-1-yl)-2-oxoethyl)amino)butyl)-2-((2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindolin-4-yl)oxy)acetamide; N-[4-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]-2-oxoethyl]amino]butyl]-2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyacetamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(=O)CNCCCCNC(=O)COc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)cn3)nc2n(C2CCCC2)c1=O	C45H51N11O9	CDK4;CDK6	P11802/Q00534	CRBN	WO-2020092662-A1
TPD-G2ZSAU	SCHEMBL24172347	(2S,4R)-1-[(2S)-2-[6-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]-2-oxoethyl]amino]hexanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(=O)CNCCCCCC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)NCc5ccc(-c6scnc6C)cc5)C(C)(C)C)CC4)cn3)nc2n(C2CCCC2)c1=O	C54H70N12O7S	CDK4;CDK6	P11802/Q00534	VHL	WO-2020092662-A1
TPD-ZY9MXT	SCHEMBL24172482	N-[2-[[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]-2-oxoethyl]-methylamino]ethyl]-2-[4-[(4S,5R)-2-(4-tert-butyl-2-ethoxyphenyl)-4,5-bis(4-chlorophenyl)-4,5-dimethylimidazole-1-carbonyl]piperazin-1-yl]acetamide; PD140956	CCOc1cc(C(C)(C)C)ccc1C1=N[C@@](C)(c2ccc(Cl)cc2)[C@@](C)(c2ccc(Cl)cc2)N1C(=O)N1CCN(CC(=O)NCCN(C)CC(=O)N2CCN(c3ccc(Nc4ncc5c(C)c(C(C)=O)c(=O)n(C6CCCC6)c5n4)nc3)CC2)CC1	C65H79Cl2N13O6	CDK4;CDK6	P11802/Q00534	VHL	WO-2020092662-A1
TPD-BUMWJ2	WO2020092662A1_YX-2-238	.	CN[C@@H](C)C(=O)N[C@H](C(=O)N1Cc2cc(OCC(=O)NCCNCC(=O)N3CCN(c4ccc(Nc5ncc6c(C)c(C(C)=O)c(=O)n(C7CCCC7)c6n5)nc4)CC3)ccc2C[C@H]1C(=O)N[C@@H]1CCCc2ccccc21)C(C)(C)C	C60H77N13O8	CDK4;CDK6	P11802/Q00534	VHL	WO-2020092662-A1
TPD-GV2V4Q	WO2020092662A1_YX-2-79	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(=O)CCc5cn(CCOCCOCCOCC(=O)N[C@@H](C)C(=O)N6C[C@H](O)C[C@H]6C(=O)NCc6ccc(-c7scnc7C)cc6)nn5)CC4)cn3)nc2n(C2CCCC2)c1=O	C56H70N14O10S	CDK4;CDK6	P11802/Q00534	VHL	WO-2020092662-A1
TPD-R1WKGM	SCHEMBL24172471	2-[4-[3-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]-3-oxopropyl]triazol-1-yl]-N-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyacetyl]amino]butyl]acetamide	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(C(=O)CCc5cn(CC(=O)NCCCCNC(=O)COc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)nn5)CC4)cn3)nc2n(C2CCCC2)c1=O	C50H56N14O10	CDK4;CDK6	P11802/Q00534	CRBN	WO-2020092662-A1
TPD-E12ZI9	WO2020142228A1_HXC78	.	Cc1cc([C@H](C(=O)N2C[C@H](O)C[C@@H]2C(=O)N[C@@H](CC(=O)NCCOCCOCCOCCNC(=O)c2cc3c4c(c2)-c2cc(O)cc5c2C4(OC3=O)c2ccc(O)cc2O5)c2ccc(-c3scnc3C)cc2)C(C)C)on1	C56H58N6O14S	AR	P10275	VHL	WO-2020142228-A1
TPD-7RRPNM	SCHEMBL22198038	(2S,4R)-N-[(1S)-3-[2-[2-[2-[2-[5-[(3aS,4S,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]pentanoylamino]ethoxy]ethoxy]ethoxy]ethylamino]-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]-3-oxopropyl]-4-hydroxy-1-[(2R)-3-methyl-2-(3-methyl-1,2-oxazol-5-yl)butanoyl]pyrrolidine-2-carboxamide	Cc1cc([C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](CC(=O)NCCOCCOCCOCCNC(=O)CCCC[C@@H]2SC[C@@H]3NC(=O)N[C@@H]32)c2ccc(-c3scnc3C)cc2)C(C)C)on1	C45H64N8O10S2	AR	P10275	VHL	WO-2020142228-A1
TPD-HJ5A82	GMB-101	(2S,4R)-1-[(2S)-3,3-dimethyl-2-[[2-[2-[[3-[6-[4-(trifluoromethoxy)anilino]pyrimidin-4-yl]benzoyl]amino]ethoxy]acetyl]amino]butanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL22440773; DTXGFSWBHDABPE-MNYREFGISA-N; (2S,4R)-1-[(2S)-3,3-dimethyl-2-[[2-[2-[[3-[6-[4-(trifluoromethoxy)anilino]pyrimidin-4-yl]benzoyl]amino]ethoxy]acetyl]amino]butanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCNC(=O)c2cccc(-c3cc(Nc4ccc(OC(F)(F)F)cc4)ncn3)c2)C(C)(C)C)cc1	C44H47F3N8O7S	BCR-ABL	Q16189	VHL	WO-2020198055-A1
TPD-X0IPLB	SCHEMBL22440746	(2S,4R)-1-[(2S)-3,3-dimethyl-2-[[2-[2-[2-[[3-[6-[4-(trifluoromethoxy)anilino]pyrimidin-4-yl]benzoyl]amino]ethoxy]ethoxy]acetyl]amino]butanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; ILQZPNKSGAYTFS-RDGUTDORSA-N; (2S,4R)-1-[(2S)-3,3-dimethyl-2-[[2-[2-[2-[[3-[6-[4-(trifluoromethoxy)anilino]pyrimidin-4-yl]benzoyl]amino]ethoxy]ethoxy]acetyl]amino]butanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCNC(=O)c2cccc(-c3cc(Nc4ccc(OC(F)(F)F)cc4)ncn3)c2)C(C)(C)C)cc1	C46H51F3N8O8S	BCR-ABL	Q16189	VHL	WO-2020198055-A1
TPD-OK37TM	SCHEMBL22440780	(2S,4R)-1-[(2S)-3,3-dimethyl-2-[3-[2-[2-[2-[2-[[3-[6-[4-(trifluoromethoxy)anilino]pyrimidin-4-yl]benzoyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]propanoylamino]butanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; LFHKRKSFSYGSEO-BTBOVKSYSA-N; (2S,4R)-1-[(2S)-3,3-dimethyl-2-[3-[2-[2-[2-[2-[[3-[6-[4-(trifluoromethoxy)anilino]pyrimidin-4-yl]benzoyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]propanoylamino]butanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCOCCOCCOCCOCCNC(=O)c2cccc(-c3cc(Nc4ccc(OC(F)(F)F)cc4)ncn3)c2)C(C)(C)C)cc1	C51H61F3N8O10S	BCR-ABL	Q16189	VHL	WO-2020198055-A1
TPD-U64F3W	SCHEMBL22440822	(2S,4R)-1-[(2S)-2-[[2-[2-[[3-(6-anilinopyrimidin-4-yl)benzoyl]amino]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCNC(=O)c2cccc(-c3cc(Nc4ccccc4)ncn3)c2)C(C)(C)C)cc1	C43H48N8O6S	BCR-ABL	Q16189	VHL	WO-2020198055-A1
TPD-EVIHUY	SCHEMBL22440766	(2S,4R)-1-[(2S)-3,3-dimethyl-2-[[2-[2-[3-[6-[4-(trifluoromethoxy)anilino]pyrimidin-4-yl]phenoxy]ethoxy]acetyl]amino]butanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; JYTRHTWBEBADME-SBJIGXGQSA-N; PD141988; (2S,4R)-1-[(2S)-3,3-dimethyl-2-[[2-[2-[3-[6-[4-(trifluoromethoxy)anilino]pyrimidin-4-yl]phenoxy]ethoxy]acetyl]amino]butanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOc2cccc(-c3cc(Nc4ccc(OC(F)(F)F)cc4)ncn3)c2)C(C)(C)C)cc1	C43H46F3N7O7S	BCR-ABL	Q16189	VHL	WO-2020198055-A1
TPD-L543XS	WO2020198055A1_6	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCCCCCCCCCCOc2cccc(-c3cc(Nc4ccc(OC(F)(F)F)cc4)ncn3)c2)C(C)(C)C)cc1	C52H64F3N7O7S	BCR-ABL	Q16189	VHL	WO-2020198055-A1
TPD-UJ7KUM	SCHEMBL22440786	(2S,4R)-1-[(2S)-3,3-dimethyl-2-[3-[2-[2-[3-[6-[4-(trifluoromethoxy)anilino]pyrimidin-4-yl]phenoxy]ethoxy]ethoxy]propanoylamino]butanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; HYFVPOSPBYLWAI-LNZHUCSUSA-N; (2S,4R)-1-[(2S)-3,3-dimethyl-2-[3-[2-[2-[3-[6-[4-(trifluoromethoxy)anilino]pyrimidin-4-yl]phenoxy]ethoxy]ethoxy]propanoylamino]butanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCOCCOCCOc2cccc(-c3cc(Nc4ccc(OC(F)(F)F)cc4)ncn3)c2)C(C)(C)C)cc1	C46H52F3N7O8S	BCR-ABL	Q16189	VHL	WO-2020198055-A1
TPD-CFEEIO	SCHEMBL22440794	(2S,4R)-4-hydroxy-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]-N-[[5-(4-methyl-1,3-thiazol-5-yl)-2-[4-[3-[6-[4-(trifluoromethoxy)anilino]pyrimidin-4-yl]phenoxy]butoxy]phenyl]methyl]pyrrolidine-2-carboxamide; SFSLUNJLLNWOKI-RJYSFZSUSA-N; (2S,4R)-4-hydroxy-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]-N-[[5-(4-methyl-1,3-thiazol-5-yl)-2-[4-[3-[6-[4-(trifluoromethoxy)anilino]pyrimidin-4-yl]phenoxy]butoxy]phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(OCCCCOc2cccc(-c3cc(Nc4ccc(OC(F)(F)F)cc4)ncn3)c2)c(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](C(C)C)N2Cc3ccccc3C2=O)c1	C50H50F3N7O7S	BCR-ABL	Q16189	VHL	WO-2020198055-A1
TPD-3ZWHJO	SCHEMBL22440754	(2S,4R)-4-hydroxy-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]-N-[[5-(4-methyl-1,3-thiazol-5-yl)-2-[4-[4-[3-[6-[4-(trifluoromethoxy)anilino]pyrimidin-4-yl]phenoxy]butoxy]butoxy]phenyl]methyl]pyrrolidine-2-carboxamide; KGDBNBZSFZCQGG-AOIYGEQBSA-N; (2S,4R)-4-hydroxy-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]-N-[[5-(4-methyl-1,3-thiazol-5-yl)-2-[4-[4-[3-[6-[4-(trifluoromethoxy)anilino]pyrimidin-4-yl]phenoxy]butoxy]butoxy]phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(OCCCCOCCCCOc2cccc(-c3cc(Nc4ccc(OC(F)(F)F)cc4)ncn3)c2)c(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](C(C)C)N2Cc3ccccc3C2=O)c1	C54H58F3N7O8S	BCR-ABL	Q16189	VHL	WO-2020198055-A1
TPD-ZYTMZW	GMB-475	(2S,4R)-1-((S)-3,3-dimethyl-2-(2-(2-(4-(6-((4-(trifluoromethoxy)phenyl)amino)pyrimidin-4-yl)phenoxy)ethoxy)acetamido)butanoyl)-4-hydroxy-N-(4-(4-methylthiazol-5-yl)benzyl)pyrrolidine-2-carboxamide; 2490599-18-1; (2S,4R)-1-((S)-3,3-dimethyl-2-(2-(2-(4-(6-((4-(trifluoromethoxy)phenyl)amino)pyrimidin-4-yl)phenoxy)ethoxy)acetamido)butanoyl)-4-hydroxy-N-(4-(4-methylthiazol-5-yl)benzyl)pyrrolidine-2-carboxamide; (2S,4R)-1-[(2S)-3,3-dimethyl-2-[[2-[2-[4-[6-[4-(trifluoromethoxy)anilino]pyrimidin-4-yl]phenoxy]ethoxy]acetyl]amino]butanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; 2489876-37-9; C43H46F3N7O7S; GMB-475?; orb1298891; CHEMBL5190713; SCHEMBL22440821; ONDVWISBMHHLGZ-SBJIGXGQSA-N; GLXC-22826; EX-A3614; s8888; AKOS037649355; AC-37884; BP-28372; BS-18108; HY-125834; CS-0100935; D81569; (2S,4R)-1-[(2S)-3,3-dimethyl-2-[[2-[2-[4-[6-[4-(trifluoromethoxy)anilino]pyrimidin-4-yl]phenoxy]ethoxy]acetyl]amino]butanoyl]-4-hydroxy-N-[[4-(4-methylthiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOc2ccc(-c3cc(Nc4ccc(OC(F)(F)F)cc4)ncn3)cc2)C(C)(C)C)cc1	C43H46F3N7O7S	BCR-ABL	Q16189	VHL	WO-2020198055-A1
TPD-ADMMK8	SCHEMBL22440816	(2S,4R)-1-[(2S)-3,3-dimethyl-2-[[2-[2-[4-[6-[4-(trifluoromethoxy)anilino]pyrimidin-4-yl]pyrazol-1-yl]ethoxy]acetyl]amino]butanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; IHEJQWQYBWMXBL-YRGOHLIBSA-N; (2S,4R)-1-[(2S)-3,3-dimethyl-2-[[2-[2-[4-[6-[4-(trifluoromethoxy)anilino]pyrimidin-4-yl]pyrazol-1-yl]ethoxy]acetyl]amino]butanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCn2cc(-c3cc(Nc4ccc(OC(F)(F)F)cc4)ncn3)cn2)C(C)(C)C)cc1	C40H44F3N9O6S	BCR-ABL	Q16189	VHL	WO-2020198055-A1
TPD-6C0Y2D	WO2020198055A1_12	.	COc1cc(C(=O)NCCCCOCCCCOc2cccc(-c3cc(Nc4ccc(OC(F)(F)F)cc4)ncn3)c2)ccc1NC[C@@H]1C[C@@H](CC(C)(C)C)[C@](C#N)(c2ccc(Cl)cc2F)[C@H]1c1cccc(Cl)c1F	C57H59Cl2F5N6O5	BCR-ABL	Q16189	VHL	WO-2020198055-A1
TPD-QA643O	SCHEMBL22440753	2-(2,6-Dioxopiperidin-3-yl)-4-[4-[4-[3-[6-[4-(trifluoromethoxy)anilino]pyrimidin-4-yl]phenoxy]butoxy]butylamino]isoindole-1,3-dione; YCYZMESGGZYUDG-UHFFFAOYSA-N; 2-(2,6-Dioxopiperidin-3-yl)-4-[4-[4-[3-[6-[4-(trifluoromethoxy)anilino]pyrimidin-4-yl]phenoxy]butoxy]butylamino]isoindole-1,3-dione	O=C1CCC(N2C(=O)c3cccc(NCCCCOCCCCOc4cccc(-c5cc(Nc6ccc(OC(F)(F)F)cc6)ncn5)c4)c3C2=O)C(=O)N1	C38H37F3N6O7	BCR-ABL	Q16189	CRBN	WO-2020198055-A1
TPD-8AVLJS	WO2020198055A1_14	.	Cc1ncsc1-c1ccc(CCC(=O)[C@H]2C[C@H](O)CN2C(=O)[C@@H](NC(=O)COCCOc2ccc(-c3cc(Nc4ccc(OC(F)(F)F)cc4)ncn3)cc2)C(C)(C)C)cc1	C44H47F3N6O7S	BCR-ABL	Q16189	VHL	WO-2020198055-A1
TPD-VH6SNS	GMB-805	CID 155138636; 2489876-41-5; SCHEMBL22458192; ZZAMCOWPQNSLBF-CPIPLPSASA-N; GLXC-23318; EX-A5218; N-(4-(Chlorodifluoromethoxy)phenyl)-6-((2-(2-(((S)-1-((2S,4R)-4-hydroxy-2-((4-(4-methylthiazol-5-yl)benzyl)carbamoyl)pyrrolidin-1-yl)-3,3-dimethyl-1-oxobutan-2-yl)amino)-2-oxoethoxy)ethyl)amino)-5-(1H-pyrazol-3-yl)nicotinamide; N-(4-(chlorodifluoromethoxy)phenyl)-6-((2-(2-(((S)-1-((2S,4R)-4-hydroxy-2-((4-(4-methylthiazol-5-yl)benzyl)carbamoyl)pyrrolidin-1-yl)-3,3-dimethyl-1-oxobutan-2-yl)amino)-2-oxoethoxy)ethyl)amino)-5-(1H-pyrazol-5-yl)nicotinamide; N-[4-[chloro(difluoro)methoxy]phenyl]-6-[2-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]ethylamino]-5-(1H-pyrazol-5-yl)pyridine-3-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCNc2ncc(C(=O)Nc3ccc(OC(F)(F)Cl)cc3)cc2-c2ccn[nH]2)C(C)(C)C)cc1	C42H46ClF2N9O7S	BCR-ABL	Q16189	VHL	WO-2020198055-A1
TPD-BBQF9E	WO2020198055A1_16	N-[4-[chloro(difluoro)methoxy]phenyl]-6-[(3S)-3-[3-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-3-oxopropoxy]pyrrolidin-1-yl]-5-(1H-pyrazol-5-yl)pyridine-3-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCO[C@H]2CCN(c3ncc(C(=O)Nc4ccc(OC(F)(F)Cl)cc4)cc3-c3ccn[nH]3)C2)C(C)(C)C)cc1	C45H50ClF2N9O7S	BCR-ABL	Q16189	VHL	WO-2020198055-A1
TPD-G8Z6XQ	SCHEMBL22440749	N-[4-[chloro(difluoro)methoxy]phenyl]-6-[4-[[3-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-3-oxopropoxy]methyl]piperidin-1-yl]-5-(1H-pyrazol-5-yl)pyridine-3-carboxamide; QFILAJIWUBTSKP-RHMQSKSJSA-N; N-[4-[chloro(difluoro)methoxy]phenyl]-6-[4-[[3-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-3-oxopropoxy]methyl]piperidin-1-yl]-5-(1H-pyrazol-5-yl)pyridine-3-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCOCC2CCN(c3ncc(C(=O)Nc4ccc(OC(F)(F)Cl)cc4)cc3-c3ccn[nH]3)CC2)C(C)(C)C)cc1	C47H54ClF2N9O7S	BCR-ABL	Q16189	VHL	WO-2020198055-A1
TPD-37TFDQ	SCHEMBL22440785	N-[4-[chloro(difluoro)methoxy]phenyl]-6-[(3S)-3-[[3-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-3-oxopropoxy]methyl]pyrrolidin-1-yl]-5-(1H-pyrazol-5-yl)pyridine-3-carboxamide; WQHQQDRDSJKPRQ-UVIROJIRSA-N; N-[4-[chloro(difluoro)methoxy]phenyl]-6-[(3S)-3-[[3-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-3-oxopropoxy]methyl]pyrrolidin-1-yl]-5-(1H-pyrazol-5-yl)pyridine-3-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCOC[C@H]2CCN(c3ncc(C(=O)Nc4ccc(OC(F)(F)Cl)cc4)cc3-c3ccn[nH]3)C2)C(C)(C)C)cc1	C46H52ClF2N9O7S	BCR-ABL	Q16189	VHL	WO-2020198055-A1
TPD-K83ZNL	WO2020198055A1_19	.	Cc1ncsc1-c1ccc(CCC(=O)C2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCNc2ncc(C(=O)Nc3ccc(OC(F)(F)Cl)cc3)cc2-c2ccn[nH]2)C(C)(C)C)cc1	C43H47ClF2N8O7S	BCR-ABL	Q16189	VHL	WO-2020198055-A1
TPD-SMKUQ6	WO2020201080A1_1	.	C[C@@H]1Cc2c([nH]c3ccccc23)C(C2=CNC(N3CCC(CN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)CC3)N=C2)N1CC(C)(C)F	C43H54FN9O3	ERα	P03372	CRBN	WO-2020201080-A1
TPD-QXV3K8	CHEMBL4781967	3-[6-[4-[2-[1-[5-[(1R,3R)-2-(2-fluoro-2-methylpropyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyrimidin-2-yl]piperidin-4-yl]ethyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL22498050; BDBM50547907; PD155484	C[C@@H]1Cc2c([nH]c3ccccc23)[C@@H](c2cnc(N3CCC(CCN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)CC3)nc2)N1CC(C)(C)F	C44H54FN9O3	ERα	P03372	CRBN	WO-2020201080-A1
TPD-YZNNRC	SCHEMBL22498034	2-(2,6-dioxopiperidin-3-yl)-5-[4-[[1-[5-[(1R,3R)-2-(2-fluoro-2-methylpropyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyrimidin-2-yl]piperidin-4-yl]methyl]piperazin-1-yl]isoindole-1,3-dione	C[C@@H]1Cc2c([nH]c3ccccc23)[C@@H](c2cnc(N3CCC(CN4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)nc2)N1CC(C)(C)F	C43H50FN9O4	ERα	P03372	CRBN	WO-2020201080-A1
TPD-NI8OF0	CHEMBL4785047	3-[6-[4-[2-[1-[5-[(1R,3R)-2-(2-fluoro-2-methylpropyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyrimidin-2-yl]piperidin-4-yl]oxyethyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL22498432; BDBM50547908; PD155482	C[C@@H]1Cc2c([nH]c3ccccc23)[C@@H](c2cnc(N3CCC(OCCN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)CC3)nc2)N1CC(C)(C)F	C44H54FN9O4	ERα	P03372	CRBN	WO-2020201080-A1
TPD-MIXG1P	CHEMBL4791102	3-[6-[4-[5-[3,5-difluoro-4-[(1R,3R)-2-(2-fluoro-2-methylpropyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]phenoxy]pentyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL22498446; BDBM50547909; PD155480	C[C@@H]1Cc2c([nH]c3ccccc23)[C@@H](c2c(F)cc(OCCCCCN3CCN(c4ccc5c(c4)CN(C4CCC(=O)NC4=O)C5=O)CC3)cc2F)N1CC(C)(C)F	C44H51F3N6O4	ERα	P03372	CRBN	WO-2020201080-A1
TPD-Z58A3M	CHEMBL4747484	3-[6-[4-[[4-[[1-[5-[(1R,3R)-2-(2-fluoro-2-methylpropyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyrimidin-2-yl]piperidin-4-yl]methyl]piperazin-1-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL22497999; BDBM50547910; PD155478	C[C@@H]1Cc2c([nH]c3ccccc23)[C@@H](c2cnc(N3CCC(CN4CCN(CC5CCN(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC5)CC4)CC3)nc2)N1CC(C)(C)F	C49H63FN10O3	ERα	P03372	CRBN	WO-2020201080-A1
TPD-NSGO8O	SCHEMBL22520710	(3S)-3-[6-[9-[[1-[5-[(1R,3R)-2-(2-fluoro-2-methylpropyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyrimidin-2-yl]piperidin-4-yl]methyl]-3,9-diazaspiro[5.5]undecan-3-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C[C@@H]1Cc2c([nH]c3ccccc23)[C@@H](c2cnc(N3CCC(CN4CCC5(CC4)CCN(c4ccc6c(c4)CN([C@H]4CCC(=O)NC4=O)C6=O)CC5)CC3)nc2)N1CC(C)(C)F	C48H60FN9O3	ERα	P03372	CRBN	WO-2020201080-A1
TPD-38BA3J	SCHEMBL22497954	3-[6-[4-[3-[1-[5-[(1R,3R)-2-(2-fluoro-2-methylpropyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyrimidin-2-yl]piperidin-4-yl]propyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C[C@@H]1Cc2c([nH]c3ccccc23)[C@@H](c2cnc(N3CCC(CCCN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)CC3)nc2)N1CC(C)(C)F	C45H56FN9O3	ERα	P03372	CRBN	WO-2020201080-A1
TPD-EDEYWF	SCHEMBL22497967	3-[6-[4-[[3-[5-[(1R,3R)-2-(2-fluoro-2-methylpropyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyrimidin-2-yl]-3,9-diazaspiro[5.5]undecan-9-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C[C@@H]1Cc2c([nH]c3ccccc23)[C@@H](c2cnc(N3CCC4(CCN(CC5CCN(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC5)CC4)CC3)nc2)N1CC(C)(C)F	C48H60FN9O3	ERα	P03372	CRBN	WO-2020201080-A1
TPD-OZ9VL1	CHEMBL4752165	3-[6-[4-[2-[3-[5-[(1R,3R)-2-(2-fluoro-2-methylpropyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyrimidin-2-yl]-3,9-diazaspiro[5.5]undecan-9-yl]ethyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL22498035; BDBM50547911; PD155476	C[C@@H]1Cc2c([nH]c3ccccc23)[C@@H](c2cnc(N3CCC4(CCN(CCC5CCN(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC5)CC4)CC3)nc2)N1CC(C)(C)F	C49H62FN9O3	ERα	P03372	CRBN	WO-2020201080-A1
TPD-WR9VK4	CHEMBL4760508	3-[6-[9-[2-[1-[5-[(1R,3R)-2-(2-fluoro-2-methylpropyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyrimidin-2-yl]piperidin-4-yl]ethyl]-3,9-diazaspiro[5.5]undecan-3-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL22497950; BDBM50547912; PD155474	C[C@@H]1Cc2c([nH]c3ccccc23)[C@@H](c2cnc(N3CCC(CCN4CCC5(CC4)CCN(c4ccc6c(c4)CN(C4CCC(=O)NC4=O)C6=O)CC5)CC3)nc2)N1CC(C)(C)F	C49H62FN9O3	ERα	P03372	CRBN	WO-2020201080-A1
TPD-BLI1WJ	CHEMBL4745409	3-[6-[4-[2-[1-[5-[(1R,3R)-2-(2-fluoro-2-methylpropyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyrimidin-2-yl]piperidin-4-yl]ethyl]piperazin-1-yl]-4-methoxy-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL22498066; BDBM50547913; PD155472	COc1cc(N2CCN(CCC3CCN(c4ncc([C@@H]5c6[nH]c7ccccc7c6C[C@@H](C)N5CC(C)(C)F)cn4)CC3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C45H56FN9O4	ERα	P03372	CRBN	WO-2020201080-A1
TPD-SH5V0E	SCHEMBL22498060	3-[6-[4-[3-[1-[5-[(1R,3R)-2-(2-fluoro-2-methylpropyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyrimidin-2-yl]piperidin-4-yl]propyl]piperazin-1-yl]-4-methoxy-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	COc1cc(N2CCN(CCCC3CCN(c4ncc([C@@H]5c6[nH]c7ccccc7c6C[C@@H](C)N5CC(C)(C)F)cn4)CC3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C46H58FN9O4	ERα	P03372	CRBN	WO-2020201080-A1
TPD-OHZXTA	SCHEMBL22498004	3-[6-[4-[[1-[[1-[5-[(1R,3R)-2-(2-fluoro-2-methylpropyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyrimidin-2-yl]piperidin-4-yl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C[C@@H]1Cc2c([nH]c3ccccc23)[C@@H](c2cnc(N3CCC(CN4CCC(CN5CCN(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC5)CC4)CC3)nc2)N1CC(C)(C)F	C49H63FN10O3	ERα	P03372	CRBN	WO-2020201080-A1
TPD-YEZ2VB	SCHEMBL22498014	3-[6-[4-[2-[1-[5-[(1R,3R)-3-methyl-2-(2,2,2-trifluoroethyl)-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyrimidin-2-yl]piperidin-4-yl]ethyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C[C@@H]1Cc2c([nH]c3ccccc23)[C@@H](c2cnc(N3CCC(CCN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)CC3)nc2)N1CC(F)(F)F	C42H48F3N9O3	ERα	P03372	CRBN	WO-2020201080-A1
TPD-IYMNJ4	SCHEMBL22498011	3-[6-[4-[[3-[[1-[5-[(1R,3R)-2-(2-fluoro-2-methylpropyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyrimidin-2-yl]piperidin-4-yl]methyl-methylamino]azetidin-1-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C[C@@H]1Cc2c([nH]c3ccccc23)[C@@H](c2cnc(N3CCC(CN(C)C4CN(CC5CCN(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC5)C4)CC3)nc2)N1CC(C)(C)F	C49H63FN10O3	ERα	P03372	CRBN	WO-2020201080-A1
TPD-WSI4AA	SCHEMBL22498059	3-[6-[4-[2-[3-[5-[(1R,3R)-2-(2-fluoro-2-methylpropyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyrimidin-2-yl]-7-oxa-3,10-diazaspiro[5.6]dodecan-10-yl]ethyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C[C@@H]1Cc2c([nH]c3ccccc23)[C@@H](c2cnc(N3CCC4(CCN(CCC5CCN(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC5)CCO4)CC3)nc2)N1CC(C)(C)F	C49H62FN9O4	ERα	P03372	CRBN	WO-2020201080-A1
TPD-H5BOBW	SCHEMBL22498007	3-[6-[4-[[3-[5-[(1R,3R)-2-(2-fluoro-2-methylpropyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyrimidin-2-yl]-7-oxa-3,10-diazaspiro[5.6]dodecan-10-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C[C@@H]1Cc2c([nH]c3ccccc23)[C@@H](c2cnc(N3CCC4(CCN(CC5CCN(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC5)CCO4)CC3)nc2)N1CC(C)(C)F	C48H60FN9O4	ERα	P03372	CRBN	WO-2020201080-A1
TPD-SGNSHE	CHEMBL4800591	3-[6-[10-[[1-[5-[(1R,3R)-2-(2-fluoro-2-methylpropyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyrimidin-2-yl]piperidin-4-yl]methyl]-7-oxa-3,10-diazaspiro[5.6]dodecan-3-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL22497995; BDBM50547914; PD155470	C[C@@H]1Cc2c([nH]c3ccccc23)[C@@H](c2cnc(N3CCC(CN4CCOC5(CC4)CCN(c4ccc6c(c4)CN(C4CCC(=O)NC4=O)C6=O)CC5)CC3)nc2)N1CC(C)(C)F	C48H60FN9O4	ERα	P03372	CRBN	WO-2020201080-A1
TPD-OFD9CV	CHEMBL4792381	3-[6-[10-[2-[1-[5-[(1R,3R)-2-(2-fluoro-2-methylpropyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyrimidin-2-yl]piperidin-4-yl]ethyl]-7-oxa-3,10-diazaspiro[5.6]dodecan-3-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL22497990; BDBM50547915; PD155468	C[C@@H]1Cc2c([nH]c3ccccc23)[C@@H](c2cnc(N3CCC(CCN4CCOC5(CC4)CCN(c4ccc6c(c4)CN(C4CCC(=O)NC4=O)C6=O)CC5)CC3)nc2)N1CC(C)(C)F	C49H62FN9O4	ERα	P03372	CRBN	WO-2020201080-A1
TPD-0NNPVN	SCHEMBL22498001	3-[6-[9-[[1-[6-[(1S,3R)-2-(2-fluoro-2-methylpropyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyridin-3-yl]piperidin-4-yl]methyl]-3,9-diazaspiro[5.5]undecan-3-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL29629082	C[C@@H]1Cc2c([nH]c3ccccc23)[C@@H](c2ccc(N3CCC(CN4CCC5(CC4)CCN(c4ccc6c(c4)CN(C4CCC(=O)NC4=O)C6=O)CC5)CC3)cn2)N1CC(C)(C)F	C49H61FN8O3	ERα	P03372	CRBN	WO-2020201080-A1
TPD-LP37OC	SCHEMBL22497988	3-[6-[9-[[7-[5-[(1R,3R)-2-(2-fluoro-2-methylpropyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyrimidin-2-yl]-7-azaspiro[3.5]nonan-2-yl]methyl]-3,9-diazaspiro[5.5]undecan-3-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C[C@@H]1Cc2c([nH]c3ccccc23)[C@@H](c2cnc(N3CCC4(CC3)CC(CN3CCC5(CC3)CCN(c3ccc6c(c3)CN(C3CCC(=O)NC3=O)C6=O)CC5)C4)nc2)N1CC(C)(C)F	C51H64FN9O3	ERα	P03372	CRBN	WO-2020201080-A1
TPD-JIPFF1	SCHEMBL22498427	3-[6-[9-[2-[3-[5-[(1R,3R)-2-(2-fluoro-2-methylpropyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyrimidin-2-yl]oxycyclobutyl]ethyl]-3,9-diazaspiro[5.5]undecan-3-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C[C@@H]1Cc2c([nH]c3ccccc23)[C@@H](c2cnc(OC3CC(CCN4CCC5(CC4)CCN(c4ccc6c(c4)CN(C4CCC(=O)NC4=O)C6=O)CC5)C3)nc2)N1CC(C)(C)F	C48H59FN8O4	ERα	P03372	CRBN	WO-2020201080-A1
TPD-UMC1E3	SCHEMBL22498042	3-[6-[9-[5-[5-[(1R,3R)-2-(2-fluoro-2-methylpropyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyrimidin-2-yl]oxypentyl]-3,9-diazaspiro[5.5]undecan-3-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C[C@@H]1Cc2c([nH]c3ccccc23)[C@@H](c2cnc(OCCCCCN3CCC4(CC3)CCN(c3ccc5c(c3)CN(C3CCC(=O)NC3=O)C5=O)CC4)nc2)N1CC(C)(C)F	C47H59FN8O4	ERα	P03372	CRBN	WO-2020201080-A1
TPD-PBCLBB	SCHEMBL22497975	3-[6-[4-[2-[9-[5-[(1R,3R)-2-(2-fluoro-2-methylpropyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyrimidin-2-yl]-4-oxo-3,9-diazaspiro[5.5]undecan-3-yl]ethyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C[C@@H]1Cc2c([nH]c3ccccc23)[C@@H](c2cnc(N3CCC4(CCN(CCN5CCN(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC5)C(=O)C4)CC3)nc2)N1CC(C)(C)F	C48H59FN10O4	ERα	P03372	CRBN	WO-2020201080-A1
TPD-253C6I	SCHEMBL22497956	3-[6-[4-[2-[3-[5-[(1R,3R)-2-(2-fluoro-2-methylpropyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyrimidin-2-yl]-3,9-diazaspiro[5.5]undecan-9-yl]ethyl]-3-oxopiperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C[C@@H]1Cc2c([nH]c3ccccc23)[C@@H](c2cnc(N3CCC4(CCN(CCN5CCN(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC5=O)CC4)CC3)nc2)N1CC(C)(C)F	C48H59FN10O4	ERα	P03372	CRBN	WO-2020201080-A1
TPD-WX8KAQ	SCHEMBL22498010	3-[6-[4-[[7-[5-[(1R,3R)-2-(2-fluoro-2-methylpropyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyrimidin-2-yl]-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C[C@@H]1Cc2c([nH]c3ccccc23)[C@@H](c2cnc(N3CCC4(CC3)CC(CN3CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC3)C4)nc2)N1CC(C)(C)F	C46H56FN9O3	ERα	P03372	CRBN	WO-2020201080-A1
TPD-LF19WH	CHEMBL4745755	3-[6-[2-[[7-[5-[(1R,3R)-2-(2-fluoro-2-methylpropyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyrimidin-2-yl]-7-azaspiro[3.5]nonan-2-yl]methyl]-2,7-diazaspiro[3.5]nonan-7-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL22497994; BDBM50547916; PD155466	C[C@@H]1Cc2c([nH]c3ccccc23)[C@@H](c2cnc(N3CCC4(CC3)CC(CN3CC5(CCN(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC5)C3)C4)nc2)N1CC(C)(C)F	C49H60FN9O3	ERα	P03372	CRBN	WO-2020201080-A1
TPD-NMGG4F	SCHEMBL22497958	3-[6-[4-[[7-[5-[(1R,3R)-2-(2-fluoro-2-methylpropyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyrimidin-2-yl]-2,7-diazaspiro[3.5]nonan-2-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C[C@@H]1Cc2c([nH]c3ccccc23)[C@@H](c2cnc(N3CCC4(CC3)CN(CC3CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC3)C4)nc2)N1CC(C)(C)F	C46H56FN9O3	ERα	P03372	CRBN	WO-2020201080-A1
TPD-QTAKE7	SCHEMBL22497965	3-[6-[6-[[1-[5-[(1R,3R)-2-(2-fluoro-2-methylpropyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyrimidin-2-yl]piperidin-4-yl]methyl]-2,6-diazaspiro[3.3]heptan-2-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C[C@@H]1Cc2c([nH]c3ccccc23)[C@@H](c2cnc(N3CCC(CN4CC5(C4)CN(c4ccc6c(c4)CN(C4CCC(=O)NC4=O)C6=O)C5)CC3)nc2)N1CC(C)(C)F	C44H52FN9O3	ERα	P03372	CRBN	WO-2020201080-A1
TPD-PJW23Q	SCHEMBL22497955	3-[6-[4-[[6-[5-[(1R,3R)-2-(2-fluoro-2-methylpropyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyrimidin-2-yl]-6-azaspiro[2.5]octan-2-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C[C@@H]1Cc2c([nH]c3ccccc23)[C@@H](c2cnc(N3CCC4(CC3)CC4CN3CCN(c4ccc5c(c4)CN(C4CCC(=O)NC4=O)C5=O)CC3)nc2)N1CC(C)(C)F	C45H54FN9O3	ERα	P03372	CRBN	WO-2020201080-A1
TPD-ALQDVH	SCHEMBL22498045	3-[6-[3-[2-[1-[5-[(1R,3R)-2-(2-fluoro-2-methylpropyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyrimidin-2-yl]piperidin-4-yl]ethyl-methylamino]azetidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C[C@@H]1Cc2c([nH]c3ccccc23)[C@@H](c2cnc(N3CCC(CCN(C)C4CN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)C4)CC3)nc2)N1CC(C)(C)F	C44H54FN9O3	ERα	P03372	CRBN	WO-2020201080-A1
TPD-MW7Q2I	SCHEMBL22497993	3-[6-[(1R,4R)-5-[3-[1-[5-[(1R,3R)-2-(2-fluoro-2-methylpropyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyrimidin-2-yl]piperidin-4-yl]propyl]-2,5-diazabicyclo[2.2.1]heptan-2-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL29629038	C[C@@H]1Cc2c([nH]c3ccccc23)[C@@H](c2cnc(N3CCC(CCCN4C[C@H]5C[C@@H]4CN5c4ccc5c(c4)CN(C4CCC(=O)NC4=O)C5=O)CC3)nc2)N1CC(C)(C)F	C46H56FN9O3	ERα	P03372	CRBN	WO-2020201080-A1
TPD-LRX5HA	SCHEMBL22498024	3-[6-[4-[3-[1-[5-[(1R,3R)-3-methyl-2-(2,2,2-trifluoroethyl)-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyrimidin-2-yl]piperidin-4-yl]propyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C[C@@H]1Cc2c([nH]c3ccccc23)[C@@H](c2cnc(N3CCC(CCCN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)CC3)nc2)N1CC(F)(F)F	C43H50F3N9O3	ERα	P03372	CRBN	WO-2020201080-A1
TPD-MF60RE	SCHEMBL22498127	3-[6-[4-[[1-[5-[(1R,3R)-3-methyl-2-(2,2,2-trifluoroethyl)-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyrimidin-2-yl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C[C@@H]1Cc2c([nH]c3ccccc23)[C@@H](c2cnc(N3CCC(CN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)CC3)nc2)N1CC(F)(F)F	C41H46F3N9O3	ERα	P03372	CRBN	WO-2020201080-A1
TPD-2S7DKD	SCHEMBL22498008	3-[6-[4-[1-[1-[5-[(1R,3R)-2-(2-fluoro-2-methylpropyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyrimidin-2-yl]piperidin-4-yl]ethyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CC(C1CCN(c2ncc([C@@H]3c4[nH]c5ccccc5c4C[C@@H](C)N3CC(C)(C)F)cn2)CC1)N1CCN(c2ccc3c(c2)CN(C2CCC(=O)NC2=O)C3=O)CC1	C44H54FN9O3	ERα	P03372	CRBN	WO-2020201080-A1
TPD-ZTFSHF	SCHEMBL22498017	3-[6-[4-[2-[1-[5-[(1R,3R)-2-(2-fluoro-2-methylpropyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyrimidin-2-yl]azetidin-3-yl]ethyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C[C@@H]1Cc2c([nH]c3ccccc23)[C@@H](c2cnc(N3CC(CCN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)C3)nc2)N1CC(C)(C)F	C42H50FN9O3	ERα	P03372	CRBN	WO-2020201080-A1
TPD-HE83F1	SCHEMBL22497978	3-[6-[4-[3-[1-[5-[(1R,3R)-2-(2-fluoro-2-methylpropyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyrimidin-2-yl]piperidin-4-yl]oxypropyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C[C@@H]1Cc2c([nH]c3ccccc23)[C@@H](c2cnc(N3CCC(OCCCN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)CC3)nc2)N1CC(C)(C)F	C45H56FN9O4	ERα	P03372	CRBN	WO-2020201080-A1
TPD-0SOT1G	CHEMBL4789907	3-[6-[4-[[1-[5-[(1R,3R)-2-(2-fluoro-2-methylpropyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyrimidin-2-yl]piperidin-4-yl]methyl]piperazin-1-yl]-4-methoxy-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL22497963; BDBM50547917; PD155464	COc1cc(N2CCN(CC3CCN(c4ncc([C@@H]5c6[nH]c7ccccc7c6C[C@@H](C)N5CC(C)(C)F)cn4)CC3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C44H54FN9O4	ERα	P03372	CRBN	WO-2020201080-A1
TPD-L6Y6FK	SCHEMBL22497959	3-[6-[4-[5-[5-[(1R,3R)-2-(2-fluoro-2-methylpropyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyrimidin-2-yl]oxypentyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C[C@@H]1Cc2c([nH]c3ccccc23)[C@@H](c2cnc(OCCCCCN3CCN(c4ccc5c(c4)CN(C4CCC(=O)NC4=O)C5=O)CC3)nc2)N1CC(C)(C)F	C42H51FN8O4	ERα	P03372	CRBN	WO-2020201080-A1
TPD-MSN50I	CHEMBL4754618	3-[6-[4-[[9-[5-[(1R,3R)-2-(2-fluoro-2-methylpropyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyrimidin-2-yl]oxy-3-azaspiro[5.5]undecan-3-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL22498113; BDBM50547918; PD155462	C[C@@H]1Cc2c([nH]c3ccccc23)[C@@H](c2cnc(OC3CCC4(CC3)CCN(CC3CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC3)CC4)nc2)N1CC(C)(C)F	C49H61FN8O4	ERα	P03372	CRBN	WO-2020201080-A1
TPD-53JEBZ	WO2020232115A1_7	.	CCOc1cc(C)ccc1C1=N[C@@H](c2ccc(Cl)cc2)[C@@H](c2ccc(Cl)cc2)N1C(=O)N1CCN(C(=O)CCC#Cc2cccc3c2CN(C2CCC(=O)NC2=O)C3=O)CC1	C47H44Cl2N6O6	MDM2	Q00987	CRBN	WO-2020232115-A1
TPD-7B4FRX	WO2020232115A1_8	.	CCOc1cc(C)ccc1C1=N[C@@H](c2ccc(Cl)cc2)[C@@H](c2ccc(Cl)cc2)N1C(=O)N1CCN(C(=O)CCCC#Cc2cccc3c2CN(C2CCC(=O)NC2=O)C3=O)CC1	C48H46Cl2N6O6	MDM2	Q00987	CRBN	WO-2020232115-A1
TPD-H1EGQ6	WO2020232115A1_9	.	CCOc1cc(C)ccc1C1=N[C@@H](c2ccc(Cl)cc2)[C@@H](c2ccc(Cl)cc2)N1C(=O)N1CCN(C(=O)CCCCC#Cc2cccc3c2CN(C2CCC(=O)NC2=O)C3=O)CC1	C49H48Cl2N6O6	MDM2	Q00987	CRBN	WO-2020232115-A1
TPD-HDKPE2	WO2020232115A1_14	.	CCOc1cc(C)ccc1C1=N[C@H](c2ccc(Cl)cc2)[C@H](c2ccc(Cl)cc2)N1C(=O)N1CCN(C(=O)CNC(=O)CCC#Cc2cccc3c2CN(C2CCC(=O)NC2=O)C3=O)CC1	C49H47Cl2N7O7	MDM2	Q00987	CRBN	WO-2020232115-A1
TPD-XO14VT	WO2020232115A1_15	.	CCOc1cc(C)ccc1C1=N[C@H](c2ccc(Cl)cc2)[C@H](c2ccc(Cl)cc2)N1C(=O)N1CCN(C(=O)CNC(=O)CCCC#Cc2cccc3c2CN(C2CCC(=O)NC2=O)C3=O)CC1	C50H49Cl2N7O7	MDM2	Q00987	CRBN	WO-2020232115-A1
TPD-PEMZ0K	WO2020232115A1_16	.	CCOc1cc(C)ccc1C1=N[C@H](c2ccc(Cl)cc2)[C@H](c2ccc(Cl)cc2)N1C(=O)N1CCN(C(=O)CNC(=O)CCCCC#Cc2cccc3c2CN(C2CCC(=O)NC2=O)C3=O)CC1	C51H51Cl2N7O7	MDM2	Q00987	CRBN	WO-2020232115-A1
TPD-B49FLJ	WO2020232115A1_20	.	CCOc1cc(C)ccc1C1=N[C@@H](c2ccc(Cl)cc2)[C@@H](c2ccc(Cl)cc2)N1C(=O)N1CCN(CC#Cc2cccc3c2CN(C2CCC(=O)NC2=O)C3=O)CC1	C45H42Cl2N6O5	MDM2	Q00987	CRBN	WO-2020232115-A1
TPD-6GZZF0	WO2020232115A1_21	.	CCOc1cc(C)ccc1C1=N[C@@H](c2ccc(Cl)cc2)[C@@H](c2ccc(Cl)cc2)N1C(=O)N1CCN(CCC#Cc2cccc3c2CN(C2CCC(=O)NC2=O)C3=O)CC1	C46H44Cl2N6O5	MDM2	Q00987	CRBN	WO-2020232115-A1
TPD-9W0GAL	WO2020232115A1_22	.	CCOc1cc(C)ccc1C1=N[C@@H](c2ccc(Cl)cc2)[C@@H](c2ccc(Cl)cc2)N1C(=O)N1CCN(CCCC#Cc2cccc3c2CN(C2CCC(=O)NC2=O)C3=O)CC1	C47H46Cl2N6O5	MDM2	Q00987	CRBN	WO-2020232115-A1
TPD-H7EBG2	WO2020232115A1_25	4-[4-[(4S,5R)-4,5-bis(4-chlorophenyl)-2-(2-ethoxy-4-methylphenyl)-4,5-dihydroimidazole-1-carbonyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CCOc1cc(C)ccc1C1=N[C@@H](c2ccc(Cl)cc2)[C@@H](c2ccc(Cl)cc2)N1C(=O)N1CCN(c2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)CC1	C42H38Cl2N6O6	MDM2	Q00987	CRBN	WO-2020232115-A1
TPD-EDNE5W	WO2020232115A1_26	.	CCOc1cc(C)ccc1C1=N[C@@H](c2ccc(Cl)cc2)[C@@H](c2ccc(Cl)cc2)N1C(=O)N1CCN(C(=O)CNc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)CC1	C44H41Cl2N7O7	MDM2	Q00987	CRBN	WO-2020232115-A1
TPD-IKPXTE	WO2020232115A1_32	.	CCOc1cc(C)ccc1C1=N[C@H](c2ccc(Cl)cc2)[C@H](c2ccc(Cl)cc2)N1C(=O)N1CCN(CC#Cc2cccc3c2CN(C2CCC(=O)NC2=O)C3=O)CC1	C45H42Cl2N6O5	MDM2	Q00987	CRBN	WO-2020232115-A1
TPD-WPC6JZ	WO2020232115A1_33	.	CCOc1cc(C)ccc1C1=N[C@H](c2ccc(Cl)cc2)[C@H](c2ccc(Cl)cc2)N1C(=O)N1CCN(CCC#Cc2cccc3c2CN(C2CCC(=O)NC2=O)C3=O)CC1	C46H44Cl2N6O5	MDM2	Q00987	CRBN	WO-2020232115-A1
TPD-REP5NZ	WO2020232115A1_34	.	CCOc1cc(C)ccc1C1=N[C@H](c2ccc(Cl)cc2)[C@H](c2ccc(Cl)cc2)N1C(=O)N1CCN(CCCC#Cc2cccc3c2CN(C2CCC(=O)NC2=O)C3=O)CC1	C47H46Cl2N6O5	MDM2	Q00987	CRBN	WO-2020232115-A1
TPD-GD848V	CHEMBL5278232	4-[2-[2-[2-[2-[(E)-7-[(3R)-3-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]-7-oxohept-5-enoxy]ethoxy]ethoxy]ethoxy]ethoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	Nc1ncnc2c1c(-c1ccc(Oc3ccccc3)cc1)nn2[C@@H]1CCCN(C(=O)/C=C/CCCCOCCOCCOCCOCCOc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)C1	C50H56N8O11	BTK	Q06187	CRBN	WO-2020252397-A1
TPD-KMADSL	PD142816	5-Amino-3-[4-(2,4-difluorophenoxy)phenyl]-1-[1-[2-[2-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]acetyl]piperidin-3-yl]pyrazole-4-carboxamide	NC(=O)c1c(-c2ccc(Oc3ccc(F)cc3F)cc2)nn(C2CCCN(C(=O)COCCOCCOCCOCCOCCNc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)c1N	C46H52F2N8O12	BTK	Q06187	CRBN	WO-2020252397-A1
TPD-SLNGI0	2366132-45-6	4-(1,1-Dimethylethyl)-N-[3-[6-[[4-[[4-[6-[[2-[[2-(2,6-dioxo-3-piperidinyl)-2,3-dihydro-1,3-dioxo-1H-isoindol-4-yl]amino]acetyl]amino]hexyl]-1-piperazinyl]carbonyl]phenyl]amino]-4,5-dihydro-4-methyl-5-oxo-2-pyrazinyl]-2-methylphenyl]benzamide; 4-(1,1-Dimethylethyl)-N-(3-(6-((4-((4-(6-((2-((2-(2,6-dioxo-3-piperidinyl)-2,3-dihydro-1,3-dioxo-1H-isoindol-4-yl)amino)acetyl)amino)hexyl)-1-piperazinyl)carbonyl)phenyl)amino)-4,5-dihydro-4-methyl-5-oxo-2-pyrazinyl)-2-methylphenyl)benzamide; 4-(1,1-Dimethylethyl)-N-[3-[6-[[4-[[4-[6-[[2-[[2-(2,6-dioxo-3-piperidinyl)-2,3-dihydro-1,3-dioxo-1H-isoindol-4-yl]amino]acetyl]amino]hexyl]-1-piperazinyl]carbonyl]phenyl]amino]-4,5-dihydro-4-methyl-5-oxo-2-pyrazinyl]-2-methylphenyl]benzamide; 861-635-4; DD-03-171; DD 03-171; CHEMBL4754443; 4-(tert-Butyl)-N-(3-(6-((4-(4-(6-(2-((2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindolin-4-yl)amino)acetamido)hexyl)piperazine-1-carbonyl)phenyl)amino)-4-methyl-5-oxo-4,5-dihydropyrazin-2-yl)-2-methylphenyl)benzamide; orb1694562; SCHEMBL22946097; SCHEMBL29625487; GTPL10535; GLXC-20433; RUD13245; BDBM50546201; AKOS040754650; 4-tert-butyl-N-[3-[6-[4-[4-[6-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]acetyl]amino]hexyl]piperazine-1-carbonyl]anilino]-4-methyl-5-oxopyrazin-2-yl]-2-methylphenyl]benzamide; HY-122830; CS-0089906; 4-(tert-Butyl)-N-(3-(6-((4-(4-(6-(2-((2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindolin-4-yl)amino)acetamido)hexyl)piperazine-1-carbon yl)phenyl)amino)-4-methyl-5-oxo-4,5-dihydropyrazin-2-yl)-2-methylphenyl)benzamide	Cc1c(NC(=O)c2ccc(C(C)(C)C)cc2)cccc1-c1cn(C)c(=O)c(Nc2ccc(C(=O)N3CCN(CCCCCCNC(=O)CNc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)cc2)n1	C55H62N10O8	BTK	Q06187	CRBN	WO-2020252397-A1
TPD-X0UH6U	IRC-1-DiMe	N-[3-[[(E)-5-[(3R)-3-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]-2-methyl-5-oxopent-3-en-2-yl]-methylamino]propyl]-2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]acetamide	CN(CCCNC(=O)CNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O)C(C)(C)/C=C/C(=O)N1CCC[C@@H](n2nc(-c3ccc(Oc4ccccc4)cc3)c3c(N)ncnc32)C1	C47H51N11O7	BTK	Q06187	CRBN	WO-2020252397-A1
TPD-IGDBCE	IRC-1	N-[3-[[(E)-4-[(3R)-3-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]-4-oxobut-2-enyl]-methylamino]propyl]-2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]acetamide	CN(C/C=C/C(=O)N1CCC[C@@H](n2nc(-c3ccc(Oc4ccccc4)cc3)c3c(N)ncnc32)C1)CCCNC(=O)CNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O	C45H47N11O7	BTK	Q06187	CRBN	WO-2020252397-A1
TPD-C4YQIL	PD155230	N-[2-[2-[[(E)-4-[(3R)-3-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]-4-oxobut-2-enyl]-methylamino]ethoxy]ethyl]-2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]amino]acetamide	CN(C/C=C/C(=O)N1CCC[C@@H](n2nc(-c3ccc(Oc4ccccc4)cc3)c3c(N)ncnc32)C1)CCOCCNC(=O)CNc1ccc2c(c1)C(=O)N(C1CCC(=O)NC1=O)C2=O	C46H49N11O8	BTK	Q06187	CRBN	WO-2020252397-A1
TPD-0BSXUZ	PD155238	N-[2-[2-[[(E)-4-[(3R)-3-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]-4-oxobut-2-enyl]-methylamino]ethoxy]ethyl]-2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]acetamide	CN(C/C=C/C(=O)N1CCC[C@@H](n2nc(-c3ccc(Oc4ccccc4)cc3)c3c(N)ncnc32)C1)CCOCCNC(=O)CNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O	C46H49N11O8	BTK	Q06187	CRBN	WO-2020252397-A1
TPD-JJUW4F	WO2020252397A1_IRC-CN	.	CN(CCCNC(=O)CNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O)C(C)(C)/C=C(\C#N)C(=O)NC/C=C/C(=O)N1CCC[C@@H](n2nc(-c3ccc(Oc4ccccc4)cc3)c3c(N)ncnc32)C1	C52H55N13O8	BTK	Q06187	CRBN	WO-2020252397-A1
TPD-B9CGEO	SCHEMBL22778081	N-[3-[[5-[(3R)-3-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]-4-cyano-2-methyl-5-oxopent-3-en-2-yl]-methylamino]propyl]-2-[[2-(1-methyl-2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]acetamide	CN1C(=O)CCC(N2C(=O)c3cccc(NCC(=O)NCCCN(C)C(C)(C)C=C(C#N)C(=O)N4CCC[C@@H](n5nc(-c6ccc(Oc7ccccc7)cc6)c6c(N)ncnc65)C4)c3C2=O)C1=O	C49H52N12O7	BTK	Q06187	CRBN	WO-2020252397-A1
TPD-CXNOC0	CHEMBL5195741	N-[3-[[5-[(3R)-3-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]-4-cyano-2-methyl-5-oxopent-3-en-2-yl]-methylamino]propyl]-2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]acetamide	CN(CCCNC(=O)CNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O)C(C)(C)C=C(C#N)C(=O)N1CCC[C@@H](n2nc(-c3ccc(Oc4ccccc4)cc3)c3c(N)ncnc32)C1	C48H50N12O7	BTK	Q06187	CRBN	WO-2020252397-A1
TPD-RCEHRO	WO2020252397A1_RC-10	.	CN(CCOCCNC(=O)CNc1ccc2c(c1)C(=O)N(C1CCC(=O)NC1=O)C2=O)C(C)(C)C=C(C#N)C(=O)N1CCC[C@@H](n2nc(-c3ccc(Oc4ccccc4)cc3)c3c(N)ncnc32)C1	C49H52N12O8	BTK	Q06187	CRBN	WO-2020252397-A1
TPD-L751J9	WO2020252397A1_RC-11	.	CN(CCCCCCCc1cccc2c1CN(C1CCC(=O)NC1=O)C2=O)C(C)(C)C=C(C#N)C(=O)N1CCC[C@@H](n2nc(-c3ccc(Oc4ccccc4)cc3)c3c(N)ncnc32)C1	C50H56N10O5	BTK	Q06187	CRBN	WO-2020252397-A1
TPD-6O7R93	WO2020252397A1_RC-12	.	CN(CCCCCC#Cc1cccc2c1CN(C1CCC(=O)NC1=O)C2=O)C(C)(C)C=C(C#N)C(=O)N1CCC[C@@H](n2nc(-c3ccc(Oc4ccccc4)cc3)c3c(N)ncnc32)C1	C50H52N10O5	BTK	Q06187	CRBN	WO-2020252397-A1
TPD-Y0NRG3	WO2020252397A1_RC-13	.	CN(CCCCCCNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O)C(C)(C)/C=C(\C#N)C(=O)N1CCC[C@@H](n2nc(-c3ccc(Oc4ccccc4)cc3)c3c(N)ncnc32)C1	C49H53N11O6	BTK	Q06187	CRBN	WO-2020252397-A1
TPD-8RFFNH	SCHEMBL22778001	N-[1-[(E)-5-[(3R)-3-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]-4-cyano-2-methyl-5-oxopent-3-en-2-yl]piperidin-4-yl]-2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]acetamide	CC(C)(/C=C(\C#N)C(=O)N1CCC[C@@H](n2nc(-c3ccc(Oc4ccccc4)cc3)c3c(N)ncnc32)C1)N1CCC(NC(=O)CNc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)CC1	C49H50N12O7	BTK	Q06187	CRBN	WO-2020252397-A1
TPD-XD9V3O	WO2020252397A1_RC-2	.	CN(CCCCNC(=O)CNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O)C(C)(C)C=C(C#N)C(=O)N1CCC[C@@H](n2nc(-c3ccc(Oc4ccccc4)cc3)c3c(N)ncnc32)C1	C49H52N12O7	BTK	Q06187	CRBN	WO-2020252397-A1
TPD-KFH156	SCHEMBL22777949	N-[2-[2-[[(E)-5-[(3R)-3-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]-4-cyano-2-methyl-5-oxopent-3-en-2-yl]-methylamino]ethoxy]ethyl]-2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]acetamide; PD155256	CN(CCOCCNC(=O)CNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O)C(C)(C)/C=C(\C#N)C(=O)N1CCC[C@@H](n2nc(-c3ccc(Oc4ccccc4)cc3)c3c(N)ncnc32)C1	C49H52N12O8	BTK	Q06187	CRBN	WO-2020252397-A1
TPD-Q3WJSG	WO2020252397A1_RC-4	.	CN(CCOCCOCCNC(=O)CNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O)C(C)(C)C=C(C#N)C(=O)N1CCC[C@@H](n2nc(-c3ccc(Oc4ccccc4)cc3)c3c(N)ncnc32)C1	C51H56N12O9	BTK	Q06187	CRBN	WO-2020252397-A1
TPD-U5654A	SCHEMBL22777947	N-[2-[2-[2-[2-[[5-[(3R)-3-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]-4-cyano-2-methyl-5-oxopent-3-en-2-yl]-methylamino]ethoxy]ethoxy]ethoxy]ethyl]-2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]acetamide	CN(CCOCCOCCOCCNC(=O)CNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O)C(C)(C)C=C(C#N)C(=O)N1CCC[C@@H](n2nc(-c3ccc(Oc4ccccc4)cc3)c3c(N)ncnc32)C1	C53H60N12O10	BTK	Q06187	CRBN	WO-2020252397-A1
TPD-9LGUO9	WO2020252397A1_RC-7	.	CN(CCCCNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O)C(C)(C)C=C(C#N)C(=O)N1CCC[C@@H](n2nc(-c3ccc(Oc4ccccc4)cc3)c3c(N)ncnc32)C1	C47H49N11O6	BTK	Q06187	CRBN	WO-2020252397-A1
TPD-FJXM8G	WO2020252397A1_RC-8	.	CN(CCCNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O)C(C)(C)C=C(C#N)C(=O)N1CCC[C@@H](n2nc(-c3ccc(Oc4ccccc4)cc3)c3c(N)ncnc32)C1	C46H47N11O6	BTK	Q06187	CRBN	WO-2020252397-A1
TPD-IH8OH2	WO2020252397A1_RC-9	.	CN(CCCNC(=O)COc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O)C(C)(C)C=C(C#N)C(=O)N1CCC[C@@H](n2nc(-c3ccc(Oc4ccccc4)cc3)c3c(N)ncnc32)C1	C48H49N11O8	BTK	Q06187	CRBN	WO-2020252397-A1
TPD-VY2YRU	RNC-1	N-[3-[[4-[(3R)-3-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]-4-oxobutyl]-methylamino]propyl]-2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]acetamide	CN(CCCNC(=O)CNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O)CCCC(=O)N1CCC[C@@H](n2nc(-c3ccc(Oc4ccccc4)cc3)c3c(N)ncnc32)C1	C45H49N11O7	BTK	Q06187	CRBN	WO-2020252397-A1
TPD-K8CYP6	PD155228	N-[2-[2-[[4-[(3R)-3-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]-4-oxobutyl]-methylamino]ethoxy]ethyl]-2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]amino]acetamide	CN(CCCC(=O)N1CCC[C@@H](n2nc(-c3ccc(Oc4ccccc4)cc3)c3c(N)ncnc32)C1)CCOCCNC(=O)CNc1ccc2c(c1)C(=O)N(C1CCC(=O)NC1=O)C2=O	C46H51N11O8	BTK	Q06187	CRBN	WO-2020252397-A1
TPD-MZ3PX6	PD155236	N-[2-[2-[[4-[(3R)-3-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]-4-oxobutyl]-methylamino]ethoxy]ethyl]-2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]acetamide	CN(CCCC(=O)N1CCC[C@@H](n2nc(-c3ccc(Oc4ccccc4)cc3)c3c(N)ncnc32)C1)CCOCCNC(=O)CNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O	C46H51N11O8	BTK	Q06187	CRBN	WO-2020252397-A1
TPD-XC0O79	WO2020252397A1_RNC-CN-Ctrl	.	CN(CCCNC(=O)CNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O)C(C)(C)CC(C#N)C(=O)NCCCC(=O)N1CCC[C@@H](n2nc(-c3ccc(Oc4ccccc4)cc3)c3c(N)ncnc32)C1	C52H59N13O8	BTK	Q06187	CRBN	WO-2020252397-A1
TPD-NRWH8E	RNC-1-CN-DiMe	RNC-1-CN-DiMe	CN(CCCNC(=O)CNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O)C(C)(C)CC(C#N)C(=O)N1CCC[C@@H](n2nc(-c3ccc(Oc4ccccc4)cc3)c3c(N)ncnc32)C1	C48H52N12O7	BTK	Q06187	CRBN	WO-2020252397-A1
TPD-PULWOP	WO2020252397A1_RNC-CN	.	CN(CCCNC(=O)CNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O)C(C)(C)/C=C(\C#N)C(=O)NCCCC(=O)N1CCC[C@@H](n2nc(-c3ccc(Oc4ccccc4)cc3)c3c(N)ncnc32)C1	C52H57N13O8	BTK	Q06187	CRBN	WO-2020252397-A1
TPD-BI5D0Z	SCHEMBL22778112	N-[4-[(3R)-3-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]-4-oxobutyl]-N-[3-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]acetyl]amino]propyl]-5-(dithiolan-3-yl)pentanamide	Nc1ncnc2c1c(-c1ccc(Oc3ccccc3)cc1)nn2[C@@H]1CCCN(C(=O)CCCN(CCCNC(=O)CNc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)C(=O)CCCCC2CCSS2)C1	C52H59N11O8S2	BTK	Q06187	CRBN	WO-2020252397-A1
TPD-R2244O	SCHEMBL22940936	(7S)-7-[1-[1-[2-[3-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]propoxy]ethyl]triazole-4-carbonyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	NC(=O)C1=C2NCC[C@@H](C3CCN(C(=O)C4=CN(CCOCCCC5=C6CN(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)N=N4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C45H48N10O7	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-8JJTW8	SCHEMBL22940354	(7S)-7-[1-[1-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethyl]triazole-4-carbonyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	NC(=O)C1=C2NCC[C@@H](C3CCN(C(=O)C4=CN(CCOCCNC5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)N=N4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C44H45N11O8	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-K1FT9B	SCHEMBL22940352	(7S)-7-[1-[1-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethyl]triazole-4-carbonyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	NC(=O)C1=C2NCC[C@@H](C3CCN(C(=O)C4=CN(CCOCCOCCNC5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)N=N4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C46H49N11O9	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-54QCFY	SCHEMBL22940170	(7S)-7-[1-[1-[2-[2-[3-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]prop-2-ynoxy]ethoxy]ethyl]triazole-4-carbonyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	NC(=O)C1=C2NCC[C@@H](C3CCN(C(=O)C4=CN(CCOCCOCC#CC5=C6CN(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)N=N4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C47H48N10O8	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-6CN922	WO2021018018A1_5	.	NC(=O)C1=C2NCCC(C3CCN(C(=O)C4=CN(CCOCCOCCCC5=C6CN(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)N=N4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C47H52N10O8	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-EGJXMO	WO2021018018A1_6	.	NC(=O)C1=C2NCCC(C3CCN(C(=O)C4=CN(CCOCCOCCOCCCC5=C6CN(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)N=N4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C49H56N10O9	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-MZCVMA	SCHEMBL22940194	(7S)-7-[1-[1-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]amino]ethoxy]ethoxy]ethyl]triazole-4-carbonyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide; SCHEMBL29795765	NC(=O)C1=C2NCC[C@@H](C3CCN(C(=O)C4=CN(CCOCCOCCNC5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)N=N4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C46H49N11O9	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-SVKCV9	SCHEMBL22940928	(7S)-7-[1-[1-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethyl]triazole-4-carbonyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	NC(=O)C1=C2NCC[C@@H](C3CCN(C(=O)C4=CN(CCOCCOCCOCCNC5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)N=N4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C48H53N11O10	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-E0HCGR	SCHEMBL22941270	(7S)-7-[1-[1-[2-[2-[2-[3-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]prop-2-ynoxy]ethoxy]ethoxy]ethyl]triazole-4-carbonyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	NC(=O)C1=C2NCC[C@@H](C3CCN(C(=O)C4=CN(CCOCCOCCOCC#CC5=C6CN(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)N=N4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C49H52N10O9	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-MWVMCL	SCHEMBL22940126	(7S)-7-[1-[1-[2-[2-[2-[2-[3-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]propoxy]ethoxy]ethoxy]ethoxy]ethyl]triazole-4-carbonyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	NC(=O)C1=C2NCC[C@@H](C3CCN(C(=O)C4=CN(CCOCCOCCOCCOCCCC5=C6CN(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)N=N4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C51H60N10O10	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-TWEQXE	WO2021018018A1_11	.	NC(=O)C1=C2NC=CC=C2N(C2CCN(C(=O)C3=CN(CCOCCOCCOCCOCC#CC4=C5CN(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)N=N3)CC2)N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C52H54N10O10	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-XVX95X	SCHEMBL22940929	(7S)-7-[1-[1-[2-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethyl]triazole-4-carbonyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide; SCHEMBL29414353	NC(=O)C1=C2NCC[C@@H](C3CCN(C(=O)C4=CN(CCOCCOCCOCCOCCNC5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)N=N4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C50H57N11O11	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-QM2QCU	CHEMBL4749185	(7S)-7-[1-[1-[2-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethyl]triazole-4-carbonyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide; SCHEMBL22940927; PD173240	NC(=O)C1=C2NCC[C@@H](C3CCN(C(=O)C4=CN(CCOCCOCCOCCOCCNC5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)N=N4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C50H57N11O11	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-TRH818	WO2021018018A1_14	.	CN(CCOCCOCCOCCOCCOCCNC1=CC2=C(C=C1)C(=O)N(C1CCC(=O)NC1=O)C2=O)/N=N\CC(=O)N1CCC([C@@H]2CCNC3=C(C(N)=O)C(C4=CC=C(OC5=CC=CC=C5)C=C4)=NN32)CC1	C52H65N11O12	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-K03Z89	WO2021018018A1_15	.	NC(=O)C1C(C2=CC=C(OC3=CCCCC3)C=C2)=NN(C(=O)C2CCN(C(=O)CN3C=C(COCCOCCOCCOCCOCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)N=N3)CC2)[C@H]2CCN[C@H]12	C53H67N11O13	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-RZ1X2D	WO2021018018A1_16	.	O=C1CCC(N2C(=O)C3=CC=CC(NCCOCCOCCOCCOCCOCCOCCN4C=C(C(=O)N5CCC(N6N=C(C7=CC=C(OC8=CC=CC=C8)C=C7)C7=C6N=CNC7=O)CC5)N=N4)=C3C2=O)C(=O)N1	C52H59N11O13	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-XCKVOL	WO2021018018A1_17	.	CN(CCOCCOCCOCCOCCOCCOCCOCCNC1=C2C(=O)N(C3CCC(=O)NC3=O)C(=O)C2=CC=C1)/N=N\CC(=O)N1CCC([C@@H]2CCNC3=C(C(N)=O)C(C4=CC=C(OC5=CC=CC=C5)C=C4)=NN32)CC1	C56H73N11O14	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-Q9GK9E	SCHEMBL22940938	(7S)-7-[1-[4-[1-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethyl]triazol-4-yl]butanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	NC(=O)C1=C2NCC[C@@H](C3CCN(C(=O)CCCC4=CN(CCOCCNC5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)N=N4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C47H51N11O8	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-QGDG39	SCHEMBL22940939	(7S)-7-[1-[4-[1-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyacetyl]amino]butyl]triazol-4-yl]butanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide; SCHEMBL29795742	NC(=O)C1=C2NCC[C@@H](C3CCN(C(=O)CCCC4=CN(CCCCNC(=O)COC5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)N=N4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C49H53N11O9	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-8HEDZN	SCHEMBL22940380	(7S)-7-[1-[4-[1-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethyl]triazol-4-yl]butanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	NC(=O)C1=C2NCC[C@@H](C3CCN(C(=O)CCCC4=CN(CCOCCOCCNC5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)N=N4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C49H55N11O9	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-UIHBWG	SCHEMBL22940241	(7S)-7-[1-[4-[1-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethyl]triazol-4-yl]butanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	NC(=O)C1=C2NCC[C@@H](C3CCN(C(=O)CCCC4=CN(CCOCCOCCOCCNC5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)N=N4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C51H59N11O10	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-J38OB5	SCHEMBL22940240	(7S)-7-[1-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]amino]-2-oxoethoxy]ethyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	NC(=O)C1=C2NCC[C@@H](C3CCN(CCOCC(=O)NC4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C41H42N8O8	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-94LDDS	SCHEMBL22940206	(7S)-7-[1-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]amino]-2-oxoethoxy]ethoxy]ethoxy]ethyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	NC(=O)C1=C2NCC[C@@H](C3CCN(CCOCCOCCOCC(=O)NC4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C45H50N8O10	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-O2WDA3	SCHEMBL22940243	(7S)-7-[1-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]amino]-2-oxoethoxy]ethoxy]ethyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	NC(=O)C1=C2NCC[C@@H](C3CCN(CCOCCOCC(=O)NC4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C43H46N8O9	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-Q6TO58	SCHEMBL22940242	(7S)-7-[1-[2-[8-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]oxy]acetyl]amino]octoxy]acetyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	NC(=O)C1=C2NCC[C@@H](C3CCN(C(=O)COCCCCCCCCNC(=O)COC4=C5CN(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C49H58N8O9	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-1W74JC	WO2021018018A1_26	.	NC(=O)C1=C2NCC[C@@H](C3CCN(C(=O)COCCCCCCCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C47H54N8O8	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-T2JO07	SCHEMBL22940506	(7S)-7-[1-[2-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethoxy]acetyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	NC(=O)C1=C2NCC[C@@H](C3CCN(C(=O)COCCOCCOCCOCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C47H54N8O11	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-9L8I8I	SCHEMBL22940499	(7S)-7-[1-[2-[2-[2-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]propanoylamino]ethoxy]ethoxy]acetyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	NC(=O)C1=C2NCC[C@@H](C3CCN(C(=O)COCCOCCNC(=O)CCN4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C50H58N10O10	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-IY1Z55	WO2021018018A1_29	.	NC(=O)C1=C2NCCC(C3CCN(C(=O)COCCOCCOCCOCCNC(=O)COC4=C5CN(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C49H58N8O12	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-I4AX28	SCHEMBL22940219	(7S)-7-[1-[5-[2-[[2-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]acetyl]amino]ethoxy]pentanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	NC(=O)C1=C2NCC[C@@H](C3CCN(C(=O)CCCCOCCNC(=O)CN4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C50H58N10O9	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-UZF162	SCHEMBL22940502	(7S)-7-[1-[5-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]pentanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	NC(=O)C1=C2NCC[C@@H](C3CCN(C(=O)CCCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C42H44N8O7	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-LQ7II4	SCHEMBL22940226	(7S)-7-[1-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]butanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	NC(=O)C1=C2NCC[C@@H](C3CCN(C(=O)CCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C41H42N8O7	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-ROT19H	SCHEMBL22940500	(7S)-7-[1-[3-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]acetyl]-methylamino]propanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	CN(CCC(=O)N1CCC([C@@H]2CCNC3=C(C(N)=O)C(C4=CC=C(OC5=CC=CC=C5)C=C4)=NN32)CC1)C(=O)CNC1=C2C(=O)N(C3CCC(=O)NC3=O)C(=O)C2=CC=C1	C43H45N9O8	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-NELJ94	SCHEMBL22940251	(7S)-7-[1-[4-[[2-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]butanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	NC(=O)C1=C2NCC[C@@H](C3CCN(C(=O)CCCNC(=O)COCCOCCOCCOCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C51H61N9O12	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-OUPQ9B	WO2021018018A1_35	.	NC(=O)C1=C2NCC[C@@H](C3CCN(C(=O)COCCOCCNC(=O)CCCCN4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)N2N=C1C1=CC=C(OC2=CC=CCC2)C=C1	C52H64N10O10	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-LH4ZV6	SCHEMBL22940398	(7S)-7-[1-[3-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethyl-methylamino]propanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	CN(CCOCCNC1=C2C(=O)N(C3CCC(=O)NC3=O)C(=O)C2=CC=C1)CCC(=O)N1CCC([C@@H]2CCNC3=C(C(N)=O)C(C4=CC=C(OC5=CC=CC=C5)C=C4)=NN32)CC1	C45H51N9O8	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-VRUYTR	SCHEMBL22940323	(7S)-7-[1-[3-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethyl-methylamino]propanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide; SCHEMBL29795796	CN(CCNC1=CC=CC2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O)CCC(=O)N1CCC([C@@H]2CCNC3=C(C(N)=O)C(C4=CC=C(OC5=CC=CC=C5)C=C4)=NN32)CC1	C43H47N9O7	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-45J5QW	SCHEMBL22941134	(7S)-7-[1-[4-[6-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]hexyl-methylamino]butanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	CN(CCCCCCNC1=C2C(=O)N(C3CCC(=O)NC3=O)C(=O)C2=CC=C1)CCCC(=O)N1CCC([C@@H]2CCNC3=C(C(N)=O)C(C4=CC=C(OC5=CC=CC=C5)C=C4)=NN32)CC1	C48H57N9O7	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-FE9B6W	CHEMBL4764736	(7S)-7-[1-[3-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]phenyl]propanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide; SCHEMBL22940292; SCHEMBL29795753; PD173250	NC(=O)C1=C2NCC[C@@H](C3CCN(C(=O)CCC4=CC=C(N5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)C=C4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C50H51N9O7	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-530S6R	WO2021018018A1_41	.	NC(=O)C1=C2NCCC(C3CCN(C(=O)COCCOCCNC(=O)CN4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C49H56N10O10	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-7Y7750	WO2021018018A1_42	.	NC(=O)C1=C2NCC[C@@H](C3CCN(C(=O)COCCOCCNC(=O)CCCN4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C51H60N10O10	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-VETUGT	SCHEMBL22940320	(7S)-7-[1-[1-[[4-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethylcarbamoyl]phenyl]methyl]piperidin-4-yl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide; SCHEMBL29795924; SCHEMBL29795926	NC(=O)C1=C2NCC[C@@H](C3CCN(C4CCN(CC5=CC=C(C(=O)NCCNC6=CC=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7=O)C=C5)CC4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C52H56N10O7	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-K0Z0KJ	SCHEMBL22940442	(7S)-7-[1-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]phenyl]butanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide; SCHEMBL29795828	NC(=O)C1=C2NCC[C@@H](C3CCN(C(=O)CCCC4=CC=C(N5CCN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C=C4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C51H53N9O7	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-LM125T	SCHEMBL22940259	(7S)-7-[1-[3-[4-[4-[[[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]acetyl]amino]methyl]phenyl]piperazin-1-yl]propanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	NC(=O)C1=C2NCC[C@@H](C3CCN(C(=O)CCN4CCN(C5=CC=C(CNC(=O)CNC6=C7CN(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)C=C5)CC4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C53H59N11O7	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-8D1296	SCHEMBL22940236	(7S)-7-[1-[(E)-4-[5-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]pentyl-methylamino]but-2-enoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide; SCHEMBL29795752	CN(C/C=C/C(=O)N1CCC([C@@H]2CCNC3=C(C(N)=O)C(C4=CC=C(OC5=CC=CC=C5)C=C4)=NN32)CC1)CCCCCNC1=CC=CC2=C1CN(C1CCC(=O)NC1=O)C2=O	C47H55N9O6	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-YRENF3	SCHEMBL22941214	(7S)-7-[1-[(E)-4-[6-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]hexyl-methylamino]but-2-enoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	CN(C/C=C/C(=O)N1CCC([C@@H]2CCNC3=C(C(N)=O)C(C4=CC=C(OC5=CC=CC=C5)C=C4)=NN32)CC1)CCCCCCNC1=C2CN(C3CCC(=O)NC3=O)C(=O)C2=CC=C1	C48H57N9O6	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-3O565I	SCHEMBL22940428	(7S)-7-[1-[(E)-3-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethyl-methylamino]prop-2-enoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide; SCHEMBL29795731	CN(/C=C/C(=O)N1CCC([C@@H]2CCNC3=C(C(N)=O)C(C4=CC=C(OC5=CC=CC=C5)C=C4)=NN32)CC1)CCOCCNC1=C2C(=O)N(C3CCC(=O)NC3=O)C(=O)C2=CC=C1	C45H49N9O8	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-DLT37G	SCHEMBL22941139	(7S)-7-[1-[(E)-3-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethyl-methylamino]prop-2-enoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide; SCHEMBL29795777	CN(/C=C/C(=O)N1CCC([C@@H]2CCNC3=C(C(N)=O)C(C4=CC=C(OC5=CC=CC=C5)C=C4)=NN32)CC1)CCNC1=CC=CC2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O	C43H45N9O7	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-MNXZNB	SCHEMBL22940349	(7S)-7-[1-[(E)-4-[6-[3-(4-amino-1,3-dioxoisoindol-2-yl)-2,6-dioxopiperidin-1-yl]hexyl-methylamino]but-2-enoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	CN(C/C=C/C(=O)N1CCC([C@@H]2CCNC3=C(C(N)=O)C(C4=CC=C(OC5=CC=CC=C5)C=C4)=NN32)CC1)CCCCCCN1C(=O)CCC(N2C(=O)C3=CC=CC(N)=C3C2=O)C1=O	C48H55N9O7	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-0MQOQP	SCHEMBL22940202	(7S)-7-[1-[(E)-4-[6-[3-(7-amino-3-oxo-1H-isoindol-2-yl)-2,6-dioxopiperidin-1-yl]hexyl-methylamino]but-2-enoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	CN(C/C=C/C(=O)N1CCC([C@@H]2CCNC3=C(C(N)=O)C(C4=CC=C(OC5=CC=CC=C5)C=C4)=NN32)CC1)CCCCCCN1C(=O)CCC(N2CC3=C(N)C=CC=C3C2=O)C1=O	C48H57N9O6	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-LT31SD	SCHEMBL22940346	(7S)-7-[1-[(E)-4-[2-[2-[2-[2-[3-(7-amino-3-oxo-1H-isoindol-2-yl)-2,6-dioxopiperidin-1-yl]ethoxy]ethoxy]ethoxy]ethyl-methylamino]but-2-enoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	CN(C/C=C/C(=O)N1CCC([C@@H]2CCNC3=C(C(N)=O)C(C4=CC=C(OC5=CC=CC=C5)C=C4)=NN32)CC1)CCOCCOCCOCCN1C(=O)CCC(N2CC3=C(N)C=CC=C3C2=O)C1=O	C50H61N9O9	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-YZT2TD	SCHEMBL22940351	(7S)-7-[1-[(E)-4-[5-[3-(7-amino-3-oxo-1H-isoindol-2-yl)-2,6-dioxopiperidin-1-yl]pentyl-methylamino]but-2-enoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	CN(C/C=C/C(=O)N1CCC([C@@H]2CCNC3=C(C(N)=O)C(C4=CC=C(OC5=CC=CC=C5)C=C4)=NN32)CC1)CCCCCN1C(=O)CCC(N2CC3=C(N)C=CC=C3C2=O)C1=O	C47H55N9O6	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-31LHRD	WO2021018018A1_54	.	C=C/C=C(\C=C)OC1=CC=C(C2=NN3C(=C2C(N)=O)NCC[C@H]3C2CCN(C(=O)/C=C/CN(C)CCCN3C(=O)CCC(N4CC5=C(N)C=CC=C5C4=O)C3=O)CC2)C=C1	C45H53N9O6	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-OMP8M6	SCHEMBL22940348	(7S)-7-[1-[(E)-4-[2-[2-[2-[3-(7-amino-3-oxo-1H-isoindol-2-yl)-2,6-dioxopiperidin-1-yl]ethoxy]ethoxy]ethyl-methylamino]but-2-enoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	CN(C/C=C/C(=O)N1CCC([C@@H]2CCNC3=C(C(N)=O)C(C4=CC=C(OC5=CC=CC=C5)C=C4)=NN32)CC1)CCOCCOCCN1C(=O)CCC(N2CC3=C(N)C=CC=C3C2=O)C1=O	C48H57N9O8	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-QTRU02	WO2021018018A1_56	.	NC(=O)C1=C2NCC[C@@H](C3CCN(C(=O)CCN4CCN(C5=CC=C(CNC(=O)CCN6C(=O)CC[C@H](N7CC8=C(N)C=CC=C8C7=O)C6=O)C=C5)CC4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C54H61N11O7	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-LQK17X	SCHEMBL22940507	(7S)-7-[1-[3-[4-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]amino]acetyl]amino]phenyl]propanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide; SCHEMBL29795751	NC(=O)C1=C2NCC[C@@H](C3CCN(C(=O)CCC4=CC=C(NC(=O)CNC5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C=C4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C48H47N9O8	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-L2AF40	CHEMBL4782596	(7S)-7-[1-[4-[4-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]amino]acetyl]amino]phenyl]butanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide; SCHEMBL29795862; PD173252	NC(=O)C1=C2NCC[C@@H](C3CCN(C(=O)CCCC4=CC=C(NC(=O)CNC5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C=C4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C49H49N9O8	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-GCE2FZ	SCHEMBL22940425	(7S)-7-[1-[5-[4-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]amino]acetyl]amino]phenyl]pentanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide; SCHEMBL29795920	NC(=O)C1=C2NCC[C@@H](C3CCN(C(=O)CCCCC4=CC=C(NC(=O)CNC5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C=C4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C50H51N9O8	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-6I30ZR	SCHEMBL22940509	(7S)-7-[1-[3-[4-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]amino]acetyl]amino]cyclohexyl]propanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide; SCHEMBL29795770	NC(=O)C1=C2NCC[C@@H](C3CCN(C(=O)CC[C@H]4CC[C@H](NC(=O)CNC5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C48H53N9O8	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-89J5LV	WO2021018018A1_61	.	NC(=O)C1=C2NCC[C@H](C3CCN(C(=O)CCC[C@H]4CC[C@@H](NC(=O)CNC5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C49H55N9O8	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-12FJYJ	SCHEMBL22940444	(7S)-7-[1-[5-[4-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]amino]acetyl]amino]cyclohexyl]pentanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide; SCHEMBL29795855	NC(=O)C1=C2NCC[C@@H](C3CCN(C(=O)CCCC[C@H]4CC[C@H](NC(=O)CNC5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C50H57N9O8	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-CVDB6N	CHEMBL4749156	(7S)-7-[1-[3-[4-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]amino]acetyl]piperazin-1-yl]propanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide; SCHEMBL29795725; PD173254	NC(=O)C1=C2NCC[C@@H](C3CCN(C(=O)CCN4CCN(C(=O)CNC5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C46H50N10O8	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-6A3TKZ	WO2021018018A1_64	.	CN(CCC(=O)N1CCC([C@@H]2CCNC3=C(C(N)=O)C(C4=CC=C(OC5=CC=CC=C5)C=C4)=NN32)CC1)CC1CCN(C2=CC=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=C2)CC1	C47H53N9O7	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-66J4TT	SCHEMBL22940901	(7S)-7-[1-[5-[4-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]amino]acetyl]piperazin-1-yl]pentanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide; SCHEMBL29795762	NC(=O)C1=C2NCC[C@@H](C3CCN(C(=O)CCCCN4CCN(C(=O)CNC5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C48H54N10O8	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-80F07Q	SCHEMBL22940257	(7S)-7-[1-[3-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]amino]ethoxy]ethyl-methylamino]propanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide; SCHEMBL29795864	CN(CCOCCNC1=CC=C2C(=O)N(C3CCC(=O)NC3=O)C(=O)C2=C1)CCC(=O)N1CCC([C@@H]2CCNC3=C(C(N)=O)C(C4=CC=C(OC5=CC=CC=C5)C=C4)=NN32)CC1	C45H51N9O8	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-IM78Z1	SCHEMBL22940460	(7S)-7-[1-[3-[[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]amino]cyclohexyl]methyl-methylamino]propanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide; SCHEMBL29795782	CN(CCC(=O)N1CCC([C@@H]2CCNC3=C(C(N)=O)C(C4=CC=C(OC5=CC=CC=C5)C=C4)=NN32)CC1)CC1CCC(NC2=CC3=C(C=C2)C(=O)N(C2CCC(=O)NC2=O)C3=O)CC1	C48H55N9O7	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-HINQJ0	SCHEMBL22940277	(7S)-7-[1-[3-[[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]phenyl]methyl-methylamino]propanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide; SCHEMBL29795806	CN(CCC(=O)N1CCC([C@@H]2CCNC3=C(C(N)=O)C(C4=CC=C(OC5=CC=CC=C5)C=C4)=NN32)CC1)CC1=CC=C(CN2CCN(C3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)C=C1	C53H58N10O7	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-IRO1KH	WO2021018018A1_70	.	CN(CCC(=O)N1CCC([C@@H]2CCNC3=C(C(N)=O)C(C4=CCC(OC5=CC=CC=C5)C=C4)=NN32)CC1)CC1=CC=C(N2CCN(C3=CC=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)CC2)C=C1	C52H58N10O7	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-RZH13A	WO2021018018A1_71	.	CC(=O)NC(=O)N(C)C1=CC=C(N(C)CCN(C)C2=CC=C(CN(C)CCC(=O)N3CCC([C@@H]4CCNC5=C(C(N)=O)C(C6=CC=C(OC7=CC=CC=C7)C=C6)=NN54)CC3)C=C2)C=C1	C49H60N10O5	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-UH5PFP	SCHEMBL22940270	(7S)-7-[1-[3-[2-[4-[4-[(2,6-dioxopiperidin-3-yl)amino]phenyl]piperazin-1-yl]ethyl-methylamino]propanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	CN(CCC(=O)N1CCC([C@@H]2CCNC3=C(C(N)=O)C(C4=CC=C(OC5=CC=CC=C5)C=C4)=NN32)CC1)CCN1CCN(C2=CC=C(NC3CCC(=O)NC3=O)C=C2)CC1	C45H56N10O5	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-Q103P7	WO2021018018A1_73	.	CC(=O)NC(=O)N(C)C1=CC=C(N(C)CCC(CN(C)CCC(=O)N2CCC([C@@H]3CCNC4=C(C(N)=O)C(C5=CC=C(OC6=CC=CC=C6)C=C5)=NN43)CC2)C2CCN(C3=CC=C(N(C)C(=O)NC(C)=O)C=C3)CC2)C=C1	C58H74N12O7	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-0225UE	SCHEMBL22940327	(7S)-7-[1-[3-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)-2-fluorophenyl]piperidin-4-yl]methyl-methylamino]propanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	CN(CCC(=O)N1CCC([C@@H]2CCNC3=C(C(N)=O)C(C4=CC=C(OC5=CC=CC=C5)C=C4)=NN32)CC1)CC1CCN(C2=C(F)C=C(N3CCC(=O)NC3=O)C=C2)CC1	C44H52FN9O5	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-OCMU3C	SCHEMBL22940328	(7S)-7-[1-[3-[[1-[6-(2,4-dioxo-1,3-diazinan-1-yl)-4-fluoropyridin-3-yl]piperidin-4-yl]methyl-methylamino]propanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	CN(CCC(=O)N1CCC([C@@H]2CCNC3=C(C(N)=O)C(C4=CC=C(OC5=CC=CC=C5)C=C4)=NN32)CC1)CC1CCN(C2=C(F)C=C(N3CCC(=O)NC3=O)N=C2)CC1	C43H51FN10O5	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-FA8YFC	SCHEMBL22940289	(7S)-7-[1-[3-[[1-[5-(2,4-dioxo-1,3-diazinan-1-yl)pyrazin-2-yl]piperidin-4-yl]methyl-methylamino]propanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide; SCHEMBL29795825	CN(CCC(=O)N1CCC([C@@H]2CCNC3=C(C(N)=O)C(C4=CC=C(OC5=CC=CC=C5)C=C4)=NN32)CC1)CC1CCN(C2=NC=C(N3CCC(=O)NC3=O)N=C2)CC1	C42H51N11O5	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-QUUDFV	SCHEMBL22940329	(7S)-7-[1-[3-[[1-[5-(2,4-dioxo-1,3-diazinan-1-yl)pyrimidin-2-yl]piperidin-4-yl]methyl-methylamino]propanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	CN(CCC(=O)N1CCC([C@@H]2CCNC3=C(C(N)=O)C(C4=CC=C(OC5=CC=CC=C5)C=C4)=NN32)CC1)CC1CCN(C2=NC=C(N3CCC(=O)NC3=O)C=N2)CC1	C42H51N11O5	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-JRAM5I	SCHEMBL22940325	(7S)-7-[1-[3-[7-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]-2,7-diazaspiro[3.5]nonan-2-yl]propanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	NC(=O)C1=C2NCC[C@@H](C3CCN(C(=O)CCN4CC5(CCN(C6=CC=C(N7CCC(=O)NC7=O)C=C6)CC5)C4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C44H51N9O5	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-I3WVEH	SCHEMBL22940326	(7S)-7-[1-[(E)-3-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl-methylamino]prop-2-enoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	CN(/C=C/C(=O)N1CCC([C@@H]2CCNC3=C(C(N)=O)C(C4=CC=C(OC5=CC=CC=C5)C=C4)=NN32)CC1)CC1CCN(C2=CC=C(N3CCC(=O)NC3=O)C=C2)CC1	C44H51N9O5	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-92MW4Z	SCHEMBL22940360	(7S)-7-[1-[(E)-3-[2-[2-[4-(2,4-dioxo-1,3-diazinan-1-yl)anilino]ethoxy]ethyl-methylamino]prop-2-enoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	CN(/C=C/C(=O)N1CCC([C@@H]2CCNC3=C(C(N)=O)C(C4=CC=C(OC5=CC=CC=C5)C=C4)=NN32)CC1)CCOCCNC1=CC=C(N2CCC(=O)NC2=O)C=C1	C42H49N9O6	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-8NJDNJ	SCHEMBL22940358	(7S)-7-[1-[3-[2-[4-[3-(2,4-dioxo-1,3-diazinan-1-yl)benzoyl]piperidin-1-yl]ethyl-methylamino]propanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide; SCHEMBL29795776	CN(CCC(=O)N1CCC([C@@H]2CCNC3=C(C(N)=O)C(C4=CC=C(OC5=CC=CC=C5)C=C4)=NN32)CC1)CCN1CCC(C(=O)C2=CC(N3CCC(=O)NC3=O)=CC=C2)CC1	C46H55N9O6	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-57O1I9	SCHEMBL22940283	(7S)-7-[1-[(E)-3-[2-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyacetyl]amino]ethyl-methylamino]prop-2-enoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide; SCHEMBL29795727	CN(/C=C/C(=O)N1CCC([C@@H]2CCNC3=C(C(N)=O)C(C4=CC=C(OC5=CC=CC=C5)C=C4)=NN32)CC1)CCNC(=O)COC1=C2C(=O)N(C3CCC(=O)NC3=O)C(=O)C2=CC=C1	C45H47N9O9	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-X5EJX1	SCHEMBL22940357	(7S)-7-[1-[3-[[4-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperazin-1-yl]cyclohexyl]methyl-methylamino]propanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	CN(CCC(=O)N1CCC([C@@H]2CCNC3=C(C(N)=O)C(C4=CC=C(OC5=CC=CC=C5)C=C4)=NN32)CC1)CC1CCC(N2CCN(C3=CC=C(N4CCC(=O)NC4=O)C=C3)CC2)CC1	C49H62N10O5	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-YA1ANZ	SCHEMBL22940361	(7S)-7-[1-[3-[2-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperazin-1-yl]ethyl-methylamino]propanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	CN(CCC(=O)N1CCC([C@@H]2CCNC3=C(C(N)=O)C(C4=CC=C(OC5=CC=CC=C5)C=C4)=NN32)CC1)CCN1CCN(C2=CC=C(N3CCC(=O)NC3=O)C=C2)CC1	C44H54N10O5	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-LUDYA9	SCHEMBL22940359	(7S)-7-[1-[3-[[2-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperazin-1-yl]-2-oxoethyl]-methylamino]propanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	CN(CCC(=O)N1CCC([C@@H]2CCNC3=C(C(N)=O)C(C4=CC=C(OC5=CC=CC=C5)C=C4)=NN32)CC1)CC(=O)N1CCN(C2=CC=C(N3CCC(=O)NC3=O)C=C2)CC1	C44H52N10O6	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-OQ9NCU	SCHEMBL22940456	(7S)-7-[1-[3-[[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethylamino]-2-oxoethyl]-methylamino]propanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide; SCHEMBL29795774	CN(CCC(=O)N1CCC([C@@H]2CCNC3=C(C(N)=O)C(C4=CC=C(OC5=CC=CC=C5)C=C4)=NN32)CC1)CC(=O)NCCNC1=C2C(=O)N(C3CCC(=O)NC3=O)C(=O)C2=CC=C1	C45H50N10O8	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-BGHOCM	SCHEMBL22940494	(7S)-7-[1-[3-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyethoxy]ethyl-methylamino]propanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide; SCHEMBL29795759	CN(CCOCCOC1=C2C(=O)N(C3CCC(=O)NC3=O)C(=O)C2=CC=C1)CCC(=O)N1CCC([C@@H]2CCNC3=C(C(N)=O)C(C4=CC=C(OC5=CC=CC=C5)C=C4)=NN32)CC1	C45H50N8O9	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-GQRRTO	SCHEMBL22940495	(7S)-7-[1-[3-[[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyethylamino]-2-oxoethyl]-methylamino]propanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide; SCHEMBL29795830	CN(CCC(=O)N1CCC([C@@H]2CCNC3=C(C(N)=O)C(C4=CC=C(OC5=CC=CC=C5)C=C4)=NN32)CC1)CC(=O)NCCOC1=C2C(=O)N(C3CCC(=O)NC3=O)C(=O)C2=CC=C1	C45H49N9O9	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-2O2VSU	SCHEMBL22940298	(7S)-7-[1-[1-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethyl]piperidine-3-carbonyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide; SCHEMBL29795859	NC(=O)C1=C2NCC[C@@H](C3CCN(C(=O)C4CCCN(CCOCCNC5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)C4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C47H53N9O8	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-VL3GAY	SCHEMBL22940496	(7S)-7-[1-[3-[3-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]piperidin-1-yl]propanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide; SCHEMBL29795841	NC(=O)C1=C2NCC[C@@H](C3CCN(C(=O)CCN4CCCC(OCCNC5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)C4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C47H53N9O8	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-KCOG3N	SCHEMBL22940294	(7S)-7-[1-[1-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethyl]piperidine-4-carbonyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide; SCHEMBL29795718	NC(=O)C1=C2NCC[C@@H](C3CCN(C(=O)C4CCN(CCOCCNC5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)CC4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C47H53N9O8	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-EY3ZGZ	SCHEMBL22940453	(7S)-7-[1-[3-[4-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]piperidin-1-yl]propanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide; SCHEMBL29795845	NC(=O)C1=C2NCC[C@@H](C3CCN(C(=O)CCN4CCC(OCCNC5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)CC4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C47H53N9O8	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-MY20BN	SCHEMBL22940897	(7S)-7-[1-[[1-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethyl]piperidin-4-yl]carbamoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide; SCHEMBL29795784	NC(=O)C1=C2NCC[C@@H](C3CCN(C(=O)NC4CCN(CCOCCNC5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)CC4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C47H54N10O8	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-SI0OWX	SCHEMBL22940905	(7S)-7-[1-[[1-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethyl]azetidin-3-yl]carbamoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide; SCHEMBL29795969	NC(=O)C1=C2NCC[C@@H](C3CCN(C(=O)NC4CN(CCOCCNC5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)C4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C45H50N10O8	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-1QQQMV	SCHEMBL22940906	(7S)-7-[1-[3-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]propanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide; SCHEMBL29795792	NC(=O)C1=C2NCC[C@@H](C3CCN(C(=O)CCN4CCC(CN5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C50H58N10O7	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-CE96PX	SCHEMBL22940479	(7S)-7-[1-[3-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperazin-1-yl]methyl]piperidin-1-yl]propanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	NC(=O)C1=C2NCC[C@@H](C3CCN(C(=O)CCN4CCC(CN5CCN(C6=CC=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C47H58N10O5	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-B6HE9B	SCHEMBL22940904	(7S)-7-[1-[3-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]methylcarbamoylamino]ethyl-methylamino]propanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide; SCHEMBL29795743	CN(CCNC(=O)NCC1=CC=C2C(=O)N(C3CCC(=O)NC3=O)C(=O)C2=C1)CCC(=O)N1CCC([C@@H]2CCNC3=C(C(N)=O)C(C4=CC=C(OC5=CC=CC=C5)C=C4)=NN32)CC1	C45H50N10O8	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-4FB8HH	SCHEMBL22940907	(7S)-7-[1-[3-[[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]methylcarbamoylamino]cyclohexyl]-methylamino]propanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide; SCHEMBL29795835	CN(CCC(=O)N1CCC([C@@H]2CCNC3=C(C(N)=O)C(C4=CC=C(OC5=CC=CC=C5)C=C4)=NN32)CC1)C1CCC(NC(=O)NCC2=CC=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=C2)CC1	C49H56N10O8	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-JOS4VO	SCHEMBL29414327	(7S)-7-[1-[3-[7-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-2,7-diazaspiro[3.5]nonan-2-yl]propanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	NC(=O)C1=C2NCC[C@@H](C3CCN(C(=O)CCN4CC5(CCN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C47H51N9O7	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-YC2H12	WO2021018018A1_100	.	CC(CCC1(C)CN(CCC(=O)N2CCC([C@@H]3CCNC4=C(C(N)=O)C(C5=CC=C(OC6=CC=CC=C6)C=C5)=NN43)CC2)C1)NC1=CC=C2C(=O)N(C3CCC(=O)NC3=O)C(=O)C2=C1	C48H55N9O7	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-1RZTTD	WO2021018018A1_101	.	NC(=O)C1=C2NCC[C@@H](C3CCN(C(=O)CCN4CC5(CCC(NC6=CC=C(N7CCC(=O)NC7=O)C=C6)CC5)C4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C45H53N9O5	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-UPY7C5	WO2021018018A1_103	.	CC(CCC(C)NC1=CC=C2C(=O)N(C3CCC(=O)NC3=O)C(=O)C2=C1)CN(C)C1CC(C(=O)N2CCC([C@@H]3CCNC4=C(C(N)=O)C(C5=CC=C(OC6=CC=CC=C6)C=C5)=NN43)CC2)C1	C50H59N9O7	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-VUX0ZG	SCHEMBL29795802	(7S)-7-[1-[3-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl-methylamino]cyclobutanecarbonyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	CN(CC1CCN(C2=CC=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=C2)CC1)C1CC(C(=O)N2CCC([C@@H]3CCNC4=C(C(N)=O)C(C5=CC=C(OC6=CC=CC=C6)C=C5)=NN43)CC2)C1	C49H55N9O7	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-DKG0QH	SCHEMBL29795839	(7S)-7-[1-[3-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl-methylamino]cyclobutanecarbonyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	CN(CC1CCN(C2=CC=C(N3CCC(=O)NC3=O)C=C2)CC1)C1CC(C(=O)N2CCC([C@@H]3CCNC4=C(C(N)=O)C(C5=CC=C(OC6=CC=CC=C6)C=C5)=NN43)CC2)C1	C46H55N9O5	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-7F7JJ4	SCHEMBL29795763	(7S)-7-[1-[3-[[1-[3-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl-methylamino]cyclobutanecarbonyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	CN(CC1CCN(C2=CC(N3CCC(=O)NC3=O)=CC=C2)CC1)C1CC(C(=O)N2CCC([C@@H]3CCNC4=C(C(N)=O)C(C5=CC=C(OC6=CC=CC=C6)C=C5)=NN43)CC2)C1	C46H55N9O5	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-OO3NEE	SCHEMBL29795850	(7S)-7-[1-[3-[[1-[3-(2,4-dioxo-1,3-diazinan-1-yl)benzoyl]piperidin-4-yl]methyl-methylamino]cyclobutanecarbonyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	CN(CC1CCN(C(=O)C2=CC(N3CCC(=O)NC3=O)=CC=C2)CC1)C1CC(C(=O)N2CCC([C@@H]3CCNC4=C(C(N)=O)C(C5=CC=C(OC6=CC=CC=C6)C=C5)=NN43)CC2)C1	C47H55N9O6	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-56GBVQ	SCHEMBL28706491	(7S)-7-[1-[3-[methyl-[[1-(7-oxo-6,8-dihydro-5H-1,8-naphthyridine-4-carbonyl)piperidin-4-yl]methyl]amino]cyclobutanecarbonyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide; SCHEMBL29795808	CN(CC1CCN(C(=O)C2=CC=NC3=C2CCC(=O)N3)CC1)C1CC(C(=O)N2CCC([C@@H]3CCNC4=C(C(N)=O)C(C5=CC=C(OC6=CC=CC=C6)C=C5)=NN43)CC2)C1	C45H53N9O5	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-MNHWG8	SCHEMBL28712681	(7S)-7-[1-[3-[methyl-[[1-(7-oxo-6,8-dihydro-5H-1,8-naphthyridine-3-carbonyl)piperidin-4-yl]methyl]amino]cyclobutanecarbonyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	CN(CC1CCN(C(=O)C2=CC3=C(N=C2)NC(=O)CC3)CC1)C1CC(C(=O)N2CCC([C@@H]3CCNC4=C(C(N)=O)C(C5=CC=C(OC6=CC=CC=C6)C=C5)=NN43)CC2)C1	C45H53N9O5	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-PF2OVT	WO2021018018A1_110	.	NC(=O)C1=C2NCC[C@@H](C3CCC(N4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C48H55N9O6	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-EHPYLB	SCHEMBL29795821	(7S)-7-[4-[[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperidin-4-yl]amino]cyclohexyl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	NC(=O)C1=C2NCC[C@@H](C3CCC(NC4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C49H57N9O6	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-KQB891	SCHEMBL22940295	(7S)-7-[4-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]cyclohexyl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	NC(=O)C1=C2NCC[C@@H](C3CCC(N4CCN(CC5CCN(C6=CC=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C45H55N9O4	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-C69CRN	SCHEMBL22940481	(7S)-7-[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindole-5-carbonyl]piperidin-4-yl]methyl]piperazin-1-yl]cyclohexyl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide; SCHEMBL29795858	NC(=O)C1=C2NCC[C@@H](C3CCC(N4CCN(CC5CCN(C(=O)C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C49H55N9O7	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-LPVZOR	SCHEMBL22940273	(7S)-7-[4-[4-[[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindole-5-carbonyl]piperidin-4-yl]phenyl]methyl]piperazin-1-yl]cyclohexyl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide; SCHEMBL29795955	NC(=O)C1=C2NCC[C@@H](C3CCC(N4CCN(CC5=CC=C(C6CCN(C(=O)C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)C=C5)CC4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C55H59N9O7	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-KI4MAS	SCHEMBL22940311	(7S)-7-[4-[4-[[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindole-5-carbonyl]piperazin-1-yl]phenyl]methyl]piperazin-1-yl]cyclohexyl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide; SCHEMBL29795936	NC(=O)C1=C2NCC[C@@H](C3CCC(N4CCN(CC5=CC=C(N6CCN(C(=O)C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)C=C5)CC4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C54H58N10O7	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-WU3IOF	SCHEMBL22941193	(7S)-7-[4-[4-[[1-[3-(2,4-dioxo-1,3-diazinan-1-yl)benzoyl]piperidin-4-yl]methyl]piperazin-1-yl]cyclohexyl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	NC(=O)C1=C2NCC[C@@H](C3CCC(N4CCN(CC5CCN(C(=O)C6=CC=CC(N7CCC(=O)NC7=O)=C6)CC5)CC4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C46H55N9O5	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-CKZX2N	SCHEMBL28691079	(7S)-7-[4-[4-[[4-[1-[3-(2,4-dioxo-1,3-diazinan-1-yl)benzoyl]piperidin-4-yl]phenyl]methyl]piperazin-1-yl]cyclohexyl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide; SCHEMBL29795812	NC(=O)C1=C2NCC[C@@H](C3CCC(N4CCN(CC5=CC=C(C6CCN(C(=O)C7=CC=CC(N8CCC(=O)NC8=O)=C7)CC6)C=C5)CC4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C52H59N9O5	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-JTY3KL	SCHEMBL22941217	(7S)-7-[1-[3-[2-[4-[3-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperazin-1-yl]ethyl-methylamino]propanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide; SCHEMBL29795811	CN(CCC(=O)N1CCC([C@@H]2CCNC3=C(C(N)=O)C(C4=CC=C(OC5=CC=CC=C5)C=C4)=NN32)CC1)CCN1CCN(C2=CC(N3CCC(=O)NC3=O)=CC=C2)CC1	C44H54N10O5	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-V3JKAH	WO2021018018A1_119	.	NC(=O)C1=C2NCC[C@@H](C3CCC(N4CCN(CC5=CC=C(N6CCN(C(=O)C7=CC=CC(N8CCC(=O)NC8=O)=C7)CC6)C=C5)CC4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C51H58N10O5	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-Y1NY90	SCHEMBL22940322	(7S)-7-[4-[[1-[[1-[3-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperidin-4-yl]amino]cyclohexyl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide; SCHEMBL28712701	NC(=O)C1=C2NCC[C@@H](C3CCC(NC4CCN(CC5CCN(C6=CC=CC(N7CCC(=O)NC7=O)=C6)CC5)CC4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C46H57N9O4	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-006615	SCHEMBL22940266	(7S)-7-[4-[[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindole-5-carbonyl]piperidin-4-yl]methyl]piperidin-4-yl]amino]cyclohexyl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide; SCHEMBL29795754	NC(=O)C1=C2NCC[C@@H](C3CCC(NC4CCN(CC5CCN(C(=O)C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C50H57N9O7	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-LDVU4J	WO2021018018A1_122	.	CN(CCC(=O)N1CCC([C@H]2CCNC3=C(C(N)=O)C(C4=CC=C(OC5=CC=CC=C5)C=C4)=NN32)CC1)CCN1CCN(C(=O)C2=CC(N3CCC(=O)NC3=O)=CC=C2)CC1	C45H54N10O6	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-RR6S2D	SCHEMBL22940949	(7S)-7-[4-[[1-[[4-[1-[3-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]phenyl]methyl]piperidin-4-yl]amino]cyclohexyl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	NC(=O)C1=C2NCC[C@@H](C3CCC(NC4CCN(CC5=CC=C(C6CCN(C7=CC=CC(N8CCC(=O)NC8=O)=C7)CC6)C=C5)CC4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C52H61N9O4	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-8PHYJT	SCHEMBL22940313	(7S)-7-[4-[[1-[[4-[4-[3-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperazin-1-yl]phenyl]methyl]piperidin-4-yl]amino]cyclohexyl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide; SCHEMBL28935128	NC(=O)C1=C2NCC[C@@H](C3CCC(NC4CCN(CC5=CC=C(N6CCN(C7=CC=CC(N8CCC(=O)NC8=O)=C7)CC6)C=C5)CC4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C51H60N10O4	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-VM3Z68	SCHEMBL29795873	(7S)-7-[4-[[1-[[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindole-5-carbonyl]piperidin-4-yl]phenyl]methyl]piperidin-4-yl]amino]cyclohexyl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	NC(=O)C1=C2NCC[C@@H](C3CCC(NC4CCN(CC5=CC=C(C6CCN(C(=O)C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)C=C5)CC4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C56H61N9O7	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-55L76L	SCHEMBL22940291	(7S)-7-[1-[3-[7-[[3-(2,4-dioxo-1,3-diazinan-1-yl)benzoyl]amino]-2-azaspiro[3.5]nonan-2-yl]propanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	NC(=O)C1=C2NCC[C@@H](C3CCN(C(=O)CCN4CC5(CCC(NC(=O)C6=CC=CC(N7CCC(=O)NC7=O)=C6)CC5)C4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C46H53N9O6	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-K8XRT7	SCHEMBL22940909	(7S)-7-[4-[[1-[[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindole-5-carbonyl]piperazin-1-yl]phenyl]methyl]piperidin-4-yl]amino]cyclohexyl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide; SCHEMBL29795769	NC(=O)C1=C2NCC[C@@H](C3CCC(NC4CCN(CC5=CC=C(N6CCN(C(=O)C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)C=C5)CC4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C55H60N10O7	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-LR45D5	SCHEMBL22941416	(7S)-7-[1-[3-[7-[3-(2,4-dioxo-1,3-diazinan-1-yl)benzoyl]-2,7-diazaspiro[3.5]nonan-2-yl]propanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	NC(=O)C1=C2NCC[C@@H](C3CCN(C(=O)CCN4CC5(CCN(C(=O)C6=CC=CC(N7CCC(=O)NC7=O)=C6)CC5)C4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C45H51N9O6	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-NI089Y	SCHEMBL22940316	(7S)-7-[1-[3-[[4-[4-[3-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperazin-1-yl]phenyl]methyl-methylamino]propanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	CN(CCC(=O)N1CCC([C@@H]2CCNC3=C(C(N)=O)C(C4=CC=C(OC5=CC=CC=C5)C=C4)=NN32)CC1)CC1=CC=C(N2CCN(C3=CC=CC(N4CCC(=O)NC4=O)=C3)CC2)C=C1	C49H56N10O5	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-SRUELR	SCHEMBL22940312	(7S)-7-[1-[3-[[6-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)benzoyl]piperazin-1-yl]pyridin-3-yl]methyl-methylamino]propanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	CN(CCC(=O)N1CCC([C@@H]2CCNC3=C(C(N)=O)C(C4=CC=C(OC5=CC=CC=C5)C=C4)=NN32)CC1)CC1=CC=C(N2CCN(C(=O)C3=CC=C(N4CCC(=O)NC4=O)C=C3)CC2)N=C1	C49H55N11O6	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-LUKTQV	SCHEMBL22940478	(7S)-7-[1-[3-[2-[4-[3-[(2,6-dioxopiperidin-3-yl)amino]phenyl]piperazin-1-yl]ethyl-methylamino]propanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide; SCHEMBL29795869	CN(CCC(=O)N1CCC([C@@H]2CCNC3=C(C(N)=O)C(C4=CC=C(OC5=CC=CC=C5)C=C4)=NN32)CC1)CCN1CCN(C2=CC(NC3CCC(=O)NC3=O)=CC=C2)CC1	C45H56N10O5	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-73TDX4	SCHEMBL22940468	(7S)-7-[1-[3-[2-[4-[3-[(2,6-dioxopiperidin-3-yl)amino]benzoyl]piperazin-1-yl]ethyl-methylamino]propanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide; SCHEMBL29795772	CN(CCC(=O)N1CCC([C@@H]2CCNC3=C(C(N)=O)C(C4=CC=C(OC5=CC=CC=C5)C=C4)=NN32)CC1)CCN1CCN(C(=O)C2=CC(NC3CCC(=O)NC3=O)=CC=C2)CC1	C46H56N10O6	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-2LHN2P	SCHEMBL29795729	(7S)-7-[1-[3-[[4-[4-[3-(2,4-dioxo-1,3-diazinan-1-yl)benzoyl]piperazin-1-yl]phenyl]methyl-methylamino]propanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	CN(CCC(=O)N1CCC([C@@H]2CCNC3=C(C(N)=O)C(C4=CC=C(OC5=CC=CC=C5)C=C4)=NN32)CC1)CC1=CC=C(N2CCN(C(=O)C3=CC=CC(N4CCC(=O)NC4=O)=C3)CC2)C=C1	C50H56N10O6	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-3X2G0Y	SCHEMBL29795756	(7S)-7-[1-[3-[[4-[4-[5-(2,4-dioxo-1,3-diazinan-1-yl)pyridine-2-carbonyl]piperazin-1-yl]phenyl]methyl-methylamino]propanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	CN(CCC(=O)N1CCC([C@@H]2CCNC3=C(C(N)=O)C(C4=CC=C(OC5=CC=CC=C5)C=C4)=NN32)CC1)CC1=CC=C(N2CCN(C(=O)C3=CC=C(N4CCC(=O)NC4=O)C=N3)CC2)C=C1	C49H55N11O6	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-B0ATRA	SCHEMBL22940911	(7S)-7-[1-[3-[2-[4-[4-[(2,6-dioxopiperidin-3-yl)amino]pyridine-2-carbonyl]piperazin-1-yl]ethyl-methylamino]propanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide; SCHEMBL29795893	CN(CCC(=O)N1CCC([C@@H]2CCNC3=C(C(N)=O)C(C4=CC=C(OC5=CC=CC=C5)C=C4)=NN32)CC1)CCN1CCN(C(=O)C2=CC(NC3CCC(=O)NC3=O)=CC=N2)CC1	C45H55N11O6	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-PINB6T	SCHEMBL22941248	(7S)-7-[1-[3-[[5-[4-[3-(2,4-dioxo-1,3-diazinan-1-yl)benzoyl]piperazin-1-yl]pyridin-2-yl]methyl-methylamino]propanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	CN(CCC(=O)N1CCC([C@@H]2CCNC3=C(C(N)=O)C(C4=CC=C(OC5=CC=CC=C5)C=C4)=NN32)CC1)CC1=CC=C(N2CCN(C(=O)C3=CC=CC(N4CCC(=O)NC4=O)=C3)CC2)C=N1	C49H55N11O6	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-5E166N	WO2021018018A1_137	.	CN(CCC(=O)N1CCC([C@@H]2CCNC3=C(C(N)=O)C(C4=CC=C(OC5=CC=CC=C5)C=C4)=NN32)CC1)CC1=NC=C(N2CCN(C(=O)C3=CC=C(N4CCC(=O)NC4=O)C=C3)CC2)C=C1	C49H55N11O6	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-37J1DT	SCHEMBL22940147	(7S)-7-[1-[3-[2-[4-[5-[(2,6-dioxopiperidin-3-yl)amino]-2-fluorobenzoyl]piperazin-1-yl]ethyl-methylamino]propanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	CN(CCC(=O)N1CCC([C@@H]2CCNC3=C(C(N)=O)C(C4=CC=C(OC5=CC=CC=C5)C=C4)=NN32)CC1)CCN1CCN(C(=O)C2=CC(NC3CCC(=O)NC3=O)=CC=C2F)CC1	C46H55FN10O6	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-ALU8KD	WO2021018018A1_139	.	CN(CCC(=O)N1CCC([C@@H]2CCNC3=C(C(N)=O)C(C4=CC=C(OC5=CC=CC=C5)C=C4)=NN32)CC1)CC1=CC=C(N2CCN(C(=O)C3=C(F)C=CC(N4CCC(=O)NC4=O)=C3)CC2)C=C1	C50H55FN10O6	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-5F84XH	SCHEMBL29795780	(7S)-7-[1-[3-[[5-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)benzoyl]piperazin-1-yl]pyrimidin-2-yl]methyl-methylamino]propanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	CN(CCC(=O)N1CCC([C@@H]2CCNC3=C(C(N)=O)C(C4=CC=C(OC5=CC=CC=C5)C=C4)=NN32)CC1)CC1=NC=C(N2CCN(C(=O)C3=CC=C(N4CCC(=O)NC4=O)C=C3)CC2)C=N1	C48H54N12O6	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-S5NMJQ	SCHEMBL22941407	(7S)-7-[1-[3-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)benzoyl]piperidin-4-yl]methyl-methylamino]propanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	CN(CCC(=O)N1CCC([C@@H]2CCNC3=C(C(N)=O)C(C4=CC=C(OC5=CC=CC=C5)C=C4)=NN32)CC1)CC1CCN(C(=O)C2=CC=C(N3CCC(=O)NC3=O)C=C2)CC1	C45H53N9O6	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-AP30DW	SCHEMBL22940342	(7S)-7-[1-[3-[[1-[3-(2,4-dioxo-1,3-diazinan-1-yl)benzoyl]piperidin-4-yl]methyl-methylamino]propanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	CN(CCC(=O)N1CCC([C@@H]2CCNC3=C(C(N)=O)C(C4=CC=C(OC5=CC=CC=C5)C=C4)=NN32)CC1)CC1CCN(C(=O)C2=CC=CC(N3CCC(=O)NC3=O)=C2)CC1	C45H53N9O6	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-LTP0CU	SCHEMBL22941403	(7S)-7-[1-[3-[7-[3-(2,4-dioxo-1,3-diazinan-1-yl)anilino]-2-azaspiro[3.5]nonan-2-yl]propanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide; SCHEMBL29795886	NC(=O)C1=C2NCC[C@@H](C3CCN(C(=O)CCN4CC5(CCC(NC6=CC(N7CCC(=O)NC7=O)=CC=C6)CC5)C4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C45H53N9O5	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-2X3Y1R	SCHEMBL22940517	(7S)-7-[1-[3-[7-[3-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]-2,7-diazaspiro[3.5]nonan-2-yl]propanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	NC(=O)C1=C2NCC[C@@H](C3CCN(C(=O)CCN4CC5(CCN(C6=CC=CC(N7CCC(=O)NC7=O)=C6)CC5)C4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C44H51N9O5	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-LRQ650	SCHEMBL22940512	(7S)-7-[1-[3-[[4-[4-[3-(2,4-dioxo-1,3-diazinan-1-yl)benzoyl]piperazin-1-yl]cyclohexyl]methyl-methylamino]propanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide; SCHEMBL29795867	CN(CCC(=O)N1CCC([C@@H]2CCNC3=C(C(N)=O)C(C4=CC=C(OC5=CC=CC=C5)C=C4)=NN32)CC1)CC1CCC(N2CCN(C(=O)C3=CC(N4CCC(=O)NC4=O)=CC=C3)CC2)CC1	C50H62N10O6	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-WGLKUR	SCHEMBL22940465	(7S)-7-[1-[3-[[4-[4-[3-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperazin-1-yl]cyclohexyl]methyl-methylamino]propanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide; SCHEMBL29795882	CN(CCC(=O)N1CCC([C@@H]2CCNC3=C(C(N)=O)C(C4=CC=C(OC5=CC=CC=C5)C=C4)=NN32)CC1)CC1CCC(N2CCN(C3=CC(N4CCC(=O)NC4=O)=CC=C3)CC2)CC1	C49H62N10O5	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-KBUZPI	WO2021018018A1_147	(7S)-7-[1-[2-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]cyclohexyl]acetyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	NC(=O)C1=C2NCC[C@@H](C3CCN(C(=O)CC4CCC(N5CCN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C49H55N9O7	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-7DN8RZ	SCHEMBL29795800	(7S)-7-[1-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]cyclohexyl]butanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	NC(=O)C1=C2NCC[C@@H](C3CCN(C(=O)CCCC4CCC(N5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C51H59N9O7	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-6SJTTI	SCHEMBL22940510	(7S)-7-[1-[5-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyacetyl]amino]butylamino]-5-oxopentanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	NC(=O)C1=C2NCC[C@@H](C3CCN(C(=O)CCCC(=O)NCCCCNC(=O)COC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C48H53N9O10	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-WB76EN	SCHEMBL22940511	(7S)-7-[1-[1-[[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazine-1-carbonyl]phenyl]methyl]piperidin-4-yl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide; SCHEMBL29414347	NC(=O)C1=C2NCC[C@@H](C3CCN(C4CCN(CC5=CC=C(C(=O)N6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)C=C5)CC4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C54H58N10O7	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-DVIL0V	CHEMBL4752555	(7S)-7-[1-[3-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]cyclohexyl]propanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide; SCHEMBL22940302; SCHEMBL29795789; PD173258	NC(=O)C1=C2NCC[C@@H](C3CCN(C(=O)CCC4CCC(N5CCN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C50H57N9O7	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-GXGC5U	CHEMBL4789332	(7S)-7-[1-[4-[4-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]amino]acetyl]piperazin-1-yl]butanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide; SCHEMBL22940457; SCHEMBL29795876; PD173260	NC(=O)C1=C2NCC[C@@H](C3CCN(C(=O)CCCN4CCN(C(=O)CNC5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C47H52N10O8	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-HUZUII	WO2021018018A1_153	.	CN(CCC(=O)N1CCC([C@@H]2CCNC3=C(C(N)=O)C(C4=CC=C(OC5=CC=CC=C5)C=C4)=NN32)CC1)CC1=CC=C(N2CCN(C3=CC=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)CC2)C=C1	C52H56N10O7	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-7G637K	SCHEMBL22940498	(7S)-7-[1-[3-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]propanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	NC(=O)C1=C2NCC[C@@H](C3CCN(C(=O)CCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C40H40N8O7	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-LDFZNY	CHEMBL4764218	(7S)-7-[1-[3-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)benzoyl]piperidin-4-yl]methyl-methylamino]cyclobutanecarbonyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide; SCHEMBL22940488; PD173262	CN(CC1CCN(C(=O)C2=CC=C(N3CCC(=O)NC3=O)C=C2)CC1)C1CC(C(=O)N2CCC([C@@H]3CCNC4=C(C(N)=O)C(C5=CC=C(OC6=CC=CC=C6)C=C5)=NN43)CC2)C1	C47H55N9O6	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-2OXQM9	SCHEMBL22940473	(7S)-7-[1-[3-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]piperidin-1-yl]propanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	NC(=O)C1=C2NCC[C@@H](C3CCN(C(=O)CCN4CCC(N5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C49H56N10O7	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-W21PET	SCHEMBL22940941	(7S)-7-[1-[(E)-4-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethyl-methylamino]but-2-enoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	CN(C/C=C/C(=O)N1CCC([C@@H]2CCNC3=C(C(N)=O)C(C4=CC=C(OC5=CC=CC=C5)C=C4)=NN32)CC1)CCOCCOCCOCCNC1=C2CN(C3CCC(=O)NC3=O)C(=O)C2=CC=C1	C50H61N9O9	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-8KEVPQ	SCHEMBL29795849	(7S)-7-[1-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]propanoyl]piperidin-4-yl]-2-(4-phenoxyphenyl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide	NC(=O)C1=C2NCC[C@@H](C3CCN(C(=O)CCN4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)N2N=C1C1=CC=C(OC2=CC=CC=C2)C=C1	C44H47N9O7	BTK	Q06187	CRBN	WO-2021018018-A1
TPD-645JYO	CHEMBL4784942	4-[[4-[1-[(1R)-2-cyano-1-cyclopentylethyl]pyrazol-4-yl]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]-N-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]butyl]benzamide; SCHEMBL22939040; PD173238	N#CC[C@H](C1CCCC1)n1cc(-c2nc(Nc3ccc(C(=O)NCCCCNc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)cc3)nc3[nH]ccc23)cn1	C41H41N11O5	JAK2	O60674	CRBN	WO-2021022076-A1
TPD-QST1OF	SCHEMBL22939001	4-[[4-[1-[3-(cyanomethyl)-1-ethylsulfonylazetidin-3-yl]pyrazol-4-yl]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]-N-[3-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]amino]propyl]benzamide	CCS(=O)(=O)N1CC(CC#N)(n2cc(-c3nc(Nc4ccc(C(=O)NCCCNc5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)cc4)nc4[nH]ccc34)cn2)C1	C39H38N12O7S	JAK2	O60674	CRBN	WO-2021022076-A1
TPD-39MCNC	SCHEMBL22938977	4-[[4-[1-[3-(cyanomethyl)-1-ethylsulfonylazetidin-3-yl]pyrazol-4-yl]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]-N-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]propyl]benzamide	CCS(=O)(=O)N1CC(CC#N)(n2cc(-c3nc(Nc4ccc(C(=O)NCCCN5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)cc4)nc4[nH]ccc34)cn2)C1	C43H45N13O7S	JAK2	O60674	CRBN	WO-2021022076-A1
TPD-YCDZWJ	WO2021022076A1_59	.	C=C1c2c(OCC(=O)NCCCNC(=O)c3ccc(Nc4nc(-c5cnn(C6(CC#N)CN(S(=O)(=O)CC)C6)c5)c5cc[nH]c5n4)cc3)cccc2C(=O)N1C1CCC(=O)NC1=O	C42H42N12O8S	JAK2	O60674	CRBN	WO-2021022076-A1
TPD-85FGL7	SCHEMBL22939054	4-[[4-[1-[3-(cyanomethyl)-1-ethylsulfonylazetidin-3-yl]pyrazol-4-yl]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]-N-[4-[[2-(1-methyl-2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]butyl]benzamide	CCS(=O)(=O)N1CC(CC#N)(n2cc(-c3nc(Nc4ccc(C(=O)NCCCCNc5cccc6c5C(=O)N(C5CCC(=O)N(C)C5=O)C6=O)cc4)nc4[nH]ccc34)cn2)C1	C41H42N12O7S	JAK2	O60674	CRBN	WO-2021022076-A1
TPD-4JPZ9U	SCHEMBL22939179	4-[[4-[1-[3-(cyanomethyl)-1-ethylsulfonylazetidin-3-yl]pyrazol-4-yl]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]-N-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]amino]butyl]benzamide	CCS(=O)(=O)N1CC(CC#N)(n2cc(-c3nc(Nc4ccc(C(=O)NCCCCNc5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)cc4)nc4[nH]ccc34)cn2)C1	C40H40N12O7S	JAK2	O60674	CRBN	WO-2021022076-A1
TPD-MGWB7M	SCHEMBL23168921	4-[8-[4-[5-[6-Amino-5-[[3-(3-hydroxy-3-methylbut-1-ynyl)phenyl]methoxy]pyridin-3-yl]-1,3-thiazol-2-yl]piperidin-1-yl]-8-oxooctoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CC(C)(O)C#Cc1cccc(COc2cc(-c3cnc(C4CCN(C(=O)CCCCCCCOc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)s3)cnc2N)c1	C46H50N6O8S	HPK1	Q92918	CRBN	WO-2021057872-A1
TPD-12UKRE	WO2021057872A1_C10	.	CC(C)(O)C#Cc1cccc(COc2cc(-c3cnc(C4CCN(C(=O)CCOCCCCCCCOc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)s3)cnc2N)c1	C48H54N6O9S	HPK1	Q92918	CRBN	WO-2021057872-A1
TPD-6WWM3D	WO2021057872A1_C11	4-[8-[3-[4-[5-[6-Amino-5-[[3-(3-hydroxy-3-methylbut-1-ynyl)phenyl]methoxy]pyridin-3-yl]-1,3-thiazol-2-yl]piperidin-1-yl]-3-oxopropoxy]octoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CC(C)(O)C#Cc1cccc(COc2cc(-c3cnc(C4CCN(C(=O)CCOCCCCCCCCOc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)s3)cnc2N)c1	C49H56N6O9S	HPK1	Q92918	CRBN	WO-2021057872-A1
TPD-HV9E9K	WO2021057872A1_C12	.	CC(C)(O)C#Cc1cccc(COc2cc(-c3cnc(C4CCN(C(=O)CCOCCCCCCCCCOc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)s3)cnc2N)c1	C50H58N6O9S	HPK1	Q92918	CRBN	WO-2021057872-A1
TPD-9O3CHK	WO2021057872A1_C13	N-[3-[4-[5-[6-amino-5-[[3-(3-hydroxy-3-methylbut-1-ynyl)phenyl]methoxy]pyridin-3-yl]-1,3-thiazol-2-yl]piperidin-1-yl]-3-oxopropyl]-4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxybutanamide	CC(C)(O)C#Cc1cccc(COc2cc(-c3cnc(C4CCN(C(=O)CCNC(=O)CCCOc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)s3)cnc2N)c1	C45H47N7O9S	HPK1	Q92918	CRBN	WO-2021057872-A1
TPD-O8Y2AB	WO2021057872A1_C14	N-[3-[4-[5-[6-amino-5-[[3-(3-hydroxy-3-methylbut-1-ynyl)phenyl]methoxy]pyridin-3-yl]-1,3-thiazol-2-yl]piperidin-1-yl]-3-oxopropyl]-5-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxypentanamide	CC(C)(O)C#Cc1cccc(COc2cc(-c3cnc(C4CCN(C(=O)CCNC(=O)CCCCOc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)s3)cnc2N)c1	C46H49N7O9S	HPK1	Q92918	CRBN	WO-2021057872-A1
TPD-X4SUMP	WO2021057872A1_C15	N-[3-[4-[5-[6-amino-5-[[3-(3-hydroxy-3-methylbut-1-ynyl)phenyl]methoxy]pyridin-3-yl]-1,3-thiazol-2-yl]piperidin-1-yl]-3-oxopropyl]-6-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyhexanamide	CC(C)(O)C#Cc1cccc(COc2cc(-c3cnc(C4CCN(C(=O)CCNC(=O)CCCCCOc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)s3)cnc2N)c1	C47H51N7O9S	HPK1	Q92918	CRBN	WO-2021057872-A1
TPD-SCQAZO	WO2021057872A1_C16	N-[3-[4-[5-[6-amino-5-[[3-(3-hydroxy-3-methylbut-1-ynyl)phenyl]methoxy]pyridin-3-yl]-1,3-thiazol-2-yl]piperidin-1-yl]-3-oxopropyl]-7-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyheptanamide	CC(C)(O)C#Cc1cccc(COc2cc(-c3cnc(C4CCN(C(=O)CCNC(=O)CCCCCCOc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)s3)cnc2N)c1	C48H53N7O9S	HPK1	Q92918	CRBN	WO-2021057872-A1
TPD-49K5IQ	WO2021057872A1_C17	4-[5-[4-[4-[5-[6-Amino-5-[[3-(3-hydroxy-3-methylbut-1-ynyl)phenyl]methoxy]pyridin-3-yl]-1,3-thiazol-2-yl]piperidine-1-carbonyl]piperidin-1-yl]-5-oxopentoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CC(C)(O)C#Cc1cccc(COc2cc(-c3cnc(C4CCN(C(=O)C5CCN(C(=O)CCCCOc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)s3)cnc2N)c1	C49H53N7O9S	HPK1	Q92918	CRBN	WO-2021057872-A1
TPD-ISC5UP	WO2021057872A1_C18	4-[6-[4-[4-[5-[6-Amino-5-[[3-(3-hydroxy-3-methylbut-1-ynyl)phenyl]methoxy]pyridin-3-yl]-1,3-thiazol-2-yl]piperidine-1-carbonyl]piperidin-1-yl]-6-oxohexoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CC(C)(O)C#Cc1cccc(COc2cc(-c3cnc(C4CCN(C(=O)C5CCN(C(=O)CCCCCOc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)s3)cnc2N)c1	C50H55N7O9S	HPK1	Q92918	CRBN	WO-2021057872-A1
TPD-VGJJE3	WO2021057872A1_C19	4-[7-[4-[4-[5-[6-Amino-5-[[3-(3-hydroxy-3-methylbut-1-ynyl)phenyl]methoxy]pyridin-3-yl]-1,3-thiazol-2-yl]piperidine-1-carbonyl]piperidin-1-yl]-7-oxoheptoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CC(C)(O)C#Cc1cccc(COc2cc(-c3cnc(C4CCN(C(=O)C5CCN(C(=O)CCCCCCOc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)s3)cnc2N)c1	C51H57N7O9S	HPK1	Q92918	CRBN	WO-2021057872-A1
TPD-E9F4VJ	SCHEMBL23168731	4-[8-[4-[5-[6-Amino-5-[[3-(3-hydroxy-3-methylbut-1-ynyl)phenyl]methoxy]pyridin-3-yl]-1,3-thiazol-2-yl]piperidin-1-yl]-8-oxooctoxy]-2-(1-methyl-2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN1C(=O)CCC(N2C(=O)c3cccc(OCCCCCCCC(=O)N4CCC(c5ncc(-c6cnc(N)c(OCc7cccc(C#CC(C)(C)O)c7)c6)s5)CC4)c3C2=O)C1=O	C47H52N6O8S	HPK1	Q92918	CRBN	WO-2021057872-A1
TPD-IHP06P	WO2021057872A1_C20	.	CC(O)C#Cc1cccc(COc2cc(-c3cnc(C4CCN(C(=O)Cn5cc(COCCOc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)nn5)CC4)s3)cnc2N)c1	C44H43N9O9S	HPK1	Q92918	CRBN	WO-2021057872-A1
TPD-L8PDC0	orb2813958	4-[10-[4-[5-[6-Amino-5-[[3-(3-hydroxy-3-methylbut-1-ynyl)phenyl]methoxy]pyridin-3-yl]-1,3-thiazol-2-yl]piperidin-1-yl]-10-oxodecoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione; CHEMBL5172420; SCHEMBL23168730	CC(C)(O)C#Cc1cccc(COc2cc(-c3cnc(C4CCN(C(=O)CCCCCCCCCOc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)s3)cnc2N)c1	C48H54N6O8S	HPK1	Q92918	CRBN	WO-2021057872-A1
TPD-PMCVEE	SCHEMBL23168910	4-[10-[4-[5-[6-Amino-5-[[3-(3-hydroxy-3-methylbut-1-ynyl)phenyl]methoxy]pyridin-3-yl]-1,3-thiazol-2-yl]piperidin-1-yl]-10-oxodecoxy]-2-(1-methyl-2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN1C(=O)CCC(N2C(=O)c3cccc(OCCCCCCCCCC(=O)N4CCC(c5ncc(-c6cnc(N)c(OCc7cccc(C#CC(C)(C)O)c7)c6)s5)CC4)c3C2=O)C1=O	C49H56N6O8S	HPK1	Q92918	CRBN	WO-2021057872-A1
TPD-KWYTS1	SCHEMBL23168908	4-[2-[2-[2-[3-[4-[5-[6-Amino-5-[[3-(3-hydroxy-3-methylbut-1-ynyl)phenyl]methoxy]pyridin-3-yl]-1,3-thiazol-2-yl]piperidin-1-yl]-3-oxopropoxy]ethoxy]ethoxy]ethoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CC(C)(O)C#Cc1cccc(COc2cc(-c3cnc(C4CCN(C(=O)CCOCCOCCOCCOc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)s3)cnc2N)c1	C47H52N6O11S	HPK1	Q92918	CRBN	WO-2021057872-A1
TPD-K73BI4	HPK1 Degrader SS47	SS47; 2636072-62-1; SS47 (TFA); HPK1 Degrader SS47; PROTAC SS47; orb1982877; CHEMBL5204123; GLXC-25881; EX-A7964; DA-78019; HY-146231; CS-0527875; 4-((15-(4-(5-(6-Amino-5-((3-(3-hydroxy-3-methylbut-1-yn-1-yl)benzyl)oxy)pyridin-3-yl)thiazol-2-yl)piperidin-1-yl)-15-oxo-3,6,9,12-tetraoxapentadecyl)oxy)-2-(2,6-dioxopiperidin-3-yl)isoindoline-1,3-dione; 4-[2-[2-[2-[2-[3-[4-[5-[6-amino-5-[[3-(3-hydroxy-3-methyl-but-1-ynyl)phenyl]methoxy]-3-pyridyl]thiazol-2-yl]-1-piperidyl]-3-oxo-propoxy]ethoxy]ethoxy]ethoxy]ethoxy]-2-(2,6-dioxo-3-piperidyl)isoindoline-1,3-dione	CC(C)(O)C#Cc1cccc(COc2cc(-c3cnc(C4CCN(C(=O)CCOCCOCCOCCOCCOc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)s3)cnc2N)c1	C49H56N6O12S	HPK1	Q92918	CRBN	WO-2021057872-A1
TPD-1B6ZQX	SCHEMBL23168948	4-[5-[3-[4-[5-[6-Amino-5-[[3-(3-hydroxy-3-methylbut-1-ynyl)phenyl]methoxy]pyridin-3-yl]-1,3-thiazol-2-yl]piperidin-1-yl]-3-oxopropoxy]pentoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CC(C)(O)C#Cc1cccc(COc2cc(-c3cnc(C4CCN(C(=O)CCOCCCCCOc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)s3)cnc2N)c1	C46H50N6O9S	HPK1	Q92918	CRBN	WO-2021057872-A1
TPD-VBUNC5	SCHEMBL23168949	4-[6-[3-[4-[5-[6-Amino-5-[[3-(3-hydroxy-3-methylbut-1-ynyl)phenyl]methoxy]pyridin-3-yl]-1,3-thiazol-2-yl]piperidin-1-yl]-3-oxopropoxy]hexoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CC(C)(O)C#Cc1cccc(COc2cc(-c3cnc(C4CCN(C(=O)CCOCCCCCCOc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)s3)cnc2N)c1	C47H52N6O9S	HPK1	Q92918	CRBN	WO-2021057872-A1
TPD-DZ1NBE	CHEMBL4875679	6-[[7-(3-chloro-4-cyanophenyl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]amino]-N-[6-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]hexyl]-2-fluoropyridine-3-carboxamide; SCHEMBL23173145	N#CC1=CC=C(N2CCC3=C(C2)N=CN=C3NC2=CC=C(C(=O)NCCCCCCN3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)C(F)=N2)C=C1Cl	C43H43ClFN11O5	AR	P10275	CRBN	WO-2021058017-A1
TPD-1N93PU	CHEMBL4875118	2-chloro-4-[4-[[5-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidine-1-carbonyl]-6-fluoropyridin-2-yl]amino]-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]benzonitrile; SCHEMBL23173088	N#CC1=CC=C(N2CCC3=C(C2)N=CN=C3NC2=NC(F)=C(C(=O)N3CCC(CN4CCN(C5=CC6=C(C=C5F)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)C=C2)C=C1Cl	C43H40ClF2N11O5	AR	P10275	CRBN	WO-2021058017-A1
TPD-NNATRU	SCHEMBL23173496	2-chloro-4-[4-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidine-1-carbonyl]anilino]-8H-pyrido[3,4-d]pyrimidin-7-yl]benzonitrile	N#CC1=CC=C(N2C=CC3=C(C2)N=CN=C3NC2=CC=C(C(=O)N3CCC(CN4CCN(C5=CC6=C(C=C5F)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)C=C2)C=C1Cl	C44H40ClFN10O5	AR	P10275	CRBN	WO-2021058017-A1
TPD-UPZ4FZ	SCHEMBL23173461	2-chloro-4-[4-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidine-1-carbonyl]anilino]-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]benzonitrile	N#CC1=CC=C(N2CCC3=C(C2)N=CN=C3NC2=CC=C(C(=O)N3CCC(CN4CCN(C5=CC6=C(C=C5F)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)C=C2)C=C1Cl	C44H42ClFN10O5	AR	P10275	CRBN	WO-2021058017-A1
TPD-004EZ5	SCHEMBL23173096	2-chloro-4-[4-[[6-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidine-1-carbonyl]pyridin-3-yl]amino]-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]benzonitrile	N#CC1=CC=C(N2CCC3=C(C2)N=CN=C3NC2=CC=C(C(=O)N3CCC(CN4CCN(C5=CC6=C(C=C5F)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)N=C2)C=C1Cl	C43H41ClFN11O5	AR	P10275	CRBN	WO-2021058017-A1
TPD-2GRWSG	SCHEMBL23173188	2-chloro-4-[4-[[5-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidine-1-carbonyl]pyridin-2-yl]amino]-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]benzonitrile	N#CC1=CC=C(N2CCC3=C(C2)N=CN=C3NC2=NC=C(C(=O)N3CCC(CN4CCN(C5=CC6=C(C=C5F)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)C=C2)C=C1Cl	C43H41ClFN11O5	AR	P10275	CRBN	WO-2021058017-A1
TPD-ZOAAXB	SCHEMBL23173772	2-chloro-4-[4-[[5-[3-[[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]azetidine-1-carbonyl]-6-fluoropyridin-2-yl]amino]-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]benzonitrile	N#CC1=CC=C(N2CCC3=C(C2)N=CN=C3NC2=NC(F)=C(C(=O)N3CC(CN4CCN(C5=CC6=C(C=C5F)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C3)C=C2)C=C1Cl	C41H36ClF2N11O5	AR	P10275	CRBN	WO-2021058017-A1
TPD-HZ8BH7	CHEMBL4871512	2-chloro-4-[4-[[5-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]-methylamino]piperidine-1-carbonyl]-6-fluoropyridin-2-yl]amino]-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]benzonitrile; SCHEMBL23173063	CN(C1CCN(C(=O)C2=C(F)N=C(NC3=NC=NC4=C3CCN(C3=CC=C(C#N)C(Cl)=C3)C4)C=C2)CC1)C1CCN(C2=CC3=C(C=C2)C(=O)N(C2CCC(=O)NC2=O)C3=O)CC1	C44H43ClFN11O5	AR	P10275	CRBN	WO-2021058017-A1
TPD-MJAUU1	CHEMBL4860986	2-chloro-4-[4-[[5-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperidin-4-yl]-methylamino]piperidine-1-carbonyl]-6-fluoropyridin-2-yl]amino]-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]benzonitrile; SCHEMBL23173671	CN(C1CCN(C(=O)C2=C(F)N=C(NC3=NC=NC4=C3CCN(C3=CC=C(C#N)C(Cl)=C3)C4)C=C2)CC1)C1CCN(C2=CC3=C(C=C2F)C(=O)N(C2CCC(=O)NC2=O)C3=O)CC1	C44H42ClF2N11O5	AR	P10275	CRBN	WO-2021058017-A1
TPD-7DW01Y	CHEMBL4858794	2-chloro-4-[4-[[5-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidine-1-carbonyl]-6-fluoropyridin-2-yl]amino]-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]benzonitrile; SCHEMBL23173050	N#CC1=CC=C(N2CCC3=C(C2)N=CN=C3NC2=NC(F)=C(C(=O)N3CCC(CN4CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)C=C2)C=C1Cl	C43H41ClFN11O5	AR	P10275	CRBN	WO-2021058017-A1
TPD-S46ZHD	SCHEMBL23173650	2-chloro-4-[4-[[6-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidine-1-carbonyl]pyridazin-3-yl]amino]-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]benzonitrile	N#CC1=CC=C(N2CCC3=C(C2)N=CN=C3NC2=CC=C(C(=O)N3CCC(CN4CCN(C5=CC6=C(C=C5F)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)N=N2)C=C1Cl	C42H40ClFN12O5	AR	P10275	CRBN	WO-2021058017-A1
TPD-R8ABHW	WO2021058017A1_2	.	N#CC1=CC=C(N2CCC3=C(C2)N=CN=C3NC2=CC=C(C(=O)NCCOCCOCCCC3=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)C(F)N2)C=C1Cl	C40H41ClFN9O6	AR	P10275	CRBN	WO-2021058017-A1
TPD-NIS401	SCHEMBL23173089	6-[[7-(3-chloro-4-cyanophenyl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]amino]-N-[3-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]propyl]-2-fluoropyridine-3-carboxamide	N#CC1=CC=C(N2CCC3=C(C2)N=CN=C3NC2=CC=C(C(=O)NCCCN3CCC(CN4CCN(C5=C(F)C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)C(F)=N2)C=C1Cl	C46H47ClF2N12O5	AR	P10275	CRBN	WO-2021058017-A1
TPD-7M05HA	CHEMBL4864381	6-[[7-(3-chloro-4-cyanophenyl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]amino]-N-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperidin-4-yl]-2-fluoropyridine-3-carboxamide; SCHEMBL23173083	N#CC1=CC=C(N2CCC3=C(C2)N=CN=C3NC2=NC(F)=C(C(=O)NC3CCN(CC4CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)C=C2)C=C1Cl	C44H43ClFN11O5	AR	P10275	CRBN	WO-2021058017-A1
TPD-DOEGT7	CHEMBL4856387	6-[[7-(3-chloro-4-cyanophenyl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]amino]-N-[2-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]-2-oxoethyl]-2-fluoropyridine-3-carboxamide; SCHEMBL23173475	N#CC1=CC=C(N2CCC3=C(C2)N=CN=C3NC2=NC(F)=C(C(=O)NCC(=O)N3CCC(CN4CCN(C5=CC6=C(C=C5F)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)C=C2)C=C1Cl	C45H43ClF2N12O6	AR	P10275	CRBN	WO-2021058017-A1
TPD-EOA0Z1	CHEMBL4874415	6-[[7-(3-chloro-4-cyanophenyl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]amino]-N-[3-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]-3-oxopropyl]-2-fluoropyridine-3-carboxamide; SCHEMBL23173233	N#CC1=CC=C(N2CCC3=C(C2)N=CN=C3NC2=CC=C(C(=O)NCCC(=O)N3CCC(CN4CCN(C5=C(F)C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)C(F)=N2)C=C1Cl	C46H45ClF2N12O6	AR	P10275	CRBN	WO-2021058017-A1
TPD-A55JM8	WO2021058017A1_24	.	[H][C@]1(CN2CCN(C3=C(F)C=C4C(=O)N(C5CCC(=O)N=NC5=O)C(=O)C4=C3)CC2)CC[C@]([H])(NC(=O)C2=CC=C(NC3=NC=NC4=C3CCN(C3=CC=C(C#N)C(Cl)=C3)C4)N=C2F)CC1	C44H41ClF2N12O5	AR	P10275	CRBN	WO-2021058017-A1
TPD-9VMKT0	CHEMBL4874007	6-[[7-(3-chloro-4-cyanophenyl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]amino]-N-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperidin-4-yl]-2-fluoropyridine-3-carboxamide; SCHEMBL23173149	N#CC1=CC=C(N2CCC3=C(C2)N=CN=C3NC2=NC(F)=C(C(=O)NC3CCN(C4CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)C=C2)C=C1Cl	C43H41ClFN11O5	AR	P10275	CRBN	WO-2021058017-A1
TPD-B3IQ04	WO2021058017A1_26	.	N#CC1=CC=C(N2CCC3=C(C2)N=CN=C3NC2=CC=C(C(=O)NC3CCN(CC4CCN(C5=C(F)C=C6C(=O)N(C7CCC(=O)N=NC7=O)C(=O)C6=C5)CC4)CC3)C=N2)C=C1Cl	C44H42ClFN12O5	AR	P10275	CRBN	WO-2021058017-A1
TPD-7315QN	WO2021058017A1_27	.	N#CC1=CC=C(N2CCC3=C(C2)N=CN=C3NC2=CC=C(C(=O)NC3CCN(CC4CCN(C5=C(F)C=C6C(=O)N(C7CCC(=O)N=NC7=O)C(=O)C6=C5)CC4)CC3)N=N2)C=C1Cl	C43H41ClFN13O5	AR	P10275	CRBN	WO-2021058017-A1
TPD-MAVBMH	WO2021058017A1_28	.	N#CC1=CC=C(N2CCC3=C(C2)N=CN=C3NC2=CN=C(C(=O)NC3CCN(CC4CCN(C5=C(F)C=C6C(=O)N(C7CCC(=O)N=NC7=O)C(=O)C6=C5)CC4)CC3)C=N2)C=C1Cl	C43H41ClFN13O5	AR	P10275	CRBN	WO-2021058017-A1
TPD-W9ORP2	WO2021058017A1_29	.	[H][C@]1(CN2CCN(C3=CC=C4C(=O)N(C5CCC(=O)N=NC5=O)C(=O)C4=C3)C[C@@H]2C)CC[C@]([H])(NC(=O)C2=CC=C(NC3=NC=NC4=C3CCN(C3=CC=C(C#N)C(Cl)=C3)C4)N=C2F)CC1	C45H44ClFN12O5	AR	P10275	CRBN	WO-2021058017-A1
TPD-9OEZJ0	SCHEMBL23173075	6-[[7-(3-chloro-4-cyanophenyl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]amino]-N-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethyl]-2-fluoropyridine-3-carboxamide	N#CC1=CC=C(N2CCC3=C(C2)N=CN=C3NC2=CC=C(C(=O)NCCOCCNC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)C(F)=N2)C=C1Cl	C37H32ClFN10O6	AR	P10275	CRBN	WO-2021058017-A1
TPD-UQ1N53	WO2021058017A1_30	.	[H][C@]1(CN2CCN(C3=CC=C4C(=O)N(C5CCC(=O)N=NC5=O)C(=O)C4=C3)C[C@H]2C)CC[C@]([H])(NC(=O)C2=CC=C(NC3=NC=NC4=C3CCN(C3=CC=C(C#N)C(Cl)=C3)C4)N=C2F)CC1	C45H44ClFN12O5	AR	P10275	CRBN	WO-2021058017-A1
TPD-EMW1Q1	SCHEMBL23173561	6-[[7-(3-chloro-4-cyanophenyl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]amino]-N-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperidin-4-yl]-2-fluoropyridine-3-carboxamide	N#CC1=CC=C(N2CCC3=C(C2)N=CN=C3NC2=NC(F)=C(C(=O)NC3CCN(C4CCN(C5=CC6=C(C=C5F)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)C=C2)C=C1Cl	C43H40ClF2N11O5	AR	P10275	CRBN	WO-2021058017-A1
TPD-QJTDSP	SCHEMBL23173132	6-[[7-(3-chloro-4-cyanophenyl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]amino]-N-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]-2-fluoro-N-methylpyridine-3-carboxamide	CN(C(=O)C1=C(F)N=C(NC2=NC=NC3=C2CCN(C2=CC=C(C#N)C(Cl)=C2)C3)C=C1)C1CCN(C2=CC3=C(C=C2)C(=O)N(C2CCC(=O)NC2=O)C3=O)CC1	C39H34ClFN10O5	AR	P10275	CRBN	WO-2021058017-A1
TPD-T4H4SQ	SCHEMBL23173232	6-[[7-(3-chloro-4-cyanophenyl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]amino]-N-[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperidin-4-yl]-2-fluoro-N-methylpyridine-3-carboxamide	CN(C(=O)C1=C(F)N=C(NC2=NC=NC3=C2CCN(C2=CC=C(C#N)C(Cl)=C2)C3)C=C1)C1CCN(C2=CC3=C(C=C2F)C(=O)N(C2CCC(=O)NC2=O)C3=O)CC1	C39H33ClF2N10O5	AR	P10275	CRBN	WO-2021058017-A1
TPD-M2BU7J	SCHEMBL23173219	6-[[7-(3-chloro-4-cyanophenyl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]amino]-N-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]-2-fluoropyridine-3-carboxamide	N#CC1=CC=C(N2CCC3=C(C2)N=CN=C3NC2=CC=C(C(=O)NCC3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)C(F)=N2)C=C1Cl	C39H34ClFN10O5	AR	P10275	CRBN	WO-2021058017-A1
TPD-G2775F	SCHEMBL23173246	6-[[7-(3-chloro-4-cyanophenyl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]amino]-N-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]-2-fluoropyridine-3-carboxamide	N#CC1=CC=C(N2CCC3=C(C2)N=CN=C3NC2=NC(F)=C(C(=O)NC3CCN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)C=C2)C=C1Cl	C38H32ClFN10O5	AR	P10275	CRBN	WO-2021058017-A1
TPD-GBVVV2	SCHEMBL23173507	5-[[7-(3-chloro-4-cyanophenyl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]amino]-N-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperidin-4-yl]pyridine-2-carboxamide	N#CC1=CC=C(N2CCC3=C(C2)N=CN=C3NC2=CC=C(C(=O)NC3CCN(CC4CCN(C5=C(F)C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)N=C2)C=C1Cl	C44H43ClFN11O5	AR	P10275	CRBN	WO-2021058017-A1
TPD-XKVWFV	SCHEMBL23173125	6-[[7-(3-chloro-4-cyanophenyl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]amino]-N-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperidin-4-yl]-2-fluoropyridine-3-carboxamide	N#CC1=CC=C(N2CCC3=C(C2)N=CN=C3NC2=CC=C(C(=O)NC3CCN(CC4CCN(C5=C(F)C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)C(F)=N2)C=C1Cl	C44H42ClF2N11O5	AR	P10275	CRBN	WO-2021058017-A1
TPD-2JJBJC	SCHEMBL23173164	4-[[7-(3-chloro-4-cyanophenyl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]amino]-N-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperidin-4-yl]benzamide	N#CC1=CC=C(N2CCC3=C(C2)N=CN=C3NC2=CC=C(C(=O)NC3CCN(CC4CCN(C5=C(F)C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)C=C2)C=C1Cl	C45H44ClFN10O5	AR	P10275	CRBN	WO-2021058017-A1
TPD-ZRZAPF	SCHEMBL23173985	6-[[7-(3-chloro-4-cyanophenyl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]amino]-N-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperidin-4-yl]-2-fluoro-N-methylpyridine-3-carboxamide	CN(C(=O)C1=CC=C(NC2=NC=NC3=C2CCN(C2=CC=C(C#N)C(Cl)=C2)C3)N=C1F)C1CCN(CC2CCN(C3=CC=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)CC2)CC1	C45H45ClFN11O5	AR	P10275	CRBN	WO-2021058017-A1
TPD-0PI4OQ	SCHEMBL23173189	6-[[7-(3-chloro-4-cyanophenyl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]amino]-N-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethyl]-2-fluoropyridine-3-carboxamide	N#CC1=CC=C(N2CCC3=C(C2)N=CN=C3NC2=CC=C(C(=O)NCCOCCOCCNC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)C(F)=N2)C=C1Cl	C39H36ClFN10O7	AR	P10275	CRBN	WO-2021058017-A1
TPD-EOPSNP	SCHEMBL23173157	6-[[7-(3-chloro-4-cyanophenyl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]amino]-N-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperidin-4-yl]-2-fluoro-N-methylpyridine-3-carboxamide	CN(C(=O)C1=CC=C(NC2=NC=NC3=C2CCN(C2=CC=C(C#N)C(Cl)=C2)C3)N=C1F)C1CCN(CC2CCN(C3=C(F)C=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)CC2)CC1	C45H44ClF2N11O5	AR	P10275	CRBN	WO-2021058017-A1
TPD-PN2H5H	SCHEMBL23173159	6-[[7-(3-chloro-4-cyanophenyl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]amino]-N-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]cyclohexyl]-2-fluoropyridine-3-carboxamide; SCHEMBL23173249	N#CC1=CC=C(N2CCC3=C(C2)N=CN=C3NC2=CC=C(C(=O)NC3CCC(N4CCN(C5=C(F)C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)C(F)=N2)C=C1Cl	C43H40ClF2N11O5	AR	P10275	CRBN	WO-2021058017-A1
TPD-UD3YLC	SCHEMBL23173163	6-[[7-(3-chloro-4-cyanophenyl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]amino]-N-[3-[[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]cyclobutyl]-2-fluoropyridine-3-carboxamide	N#CC1=CC=C(N2CCC3=C(C2)N=CN=C3NC2=CC=C(C(=O)N[C@H]3C[C@H](CN4CCN(C5=C(F)C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)C3)C(F)=N2)C=C1Cl	C42H38ClF2N11O5	AR	P10275	CRBN	WO-2021058017-A1
TPD-9TKRUC	SCHEMBL23173122	6-[[7-(3-chloro-4-cyanophenyl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]amino]-N-[2-[4-[[4-[3-(2,4-dioxo-1,3-diazinan-1-yl)benzoyl]piperazin-1-yl]methyl]piperidin-1-yl]-2-oxoethyl]-2-fluoropyridine-3-carboxamide	N#CC1=CC=C(N2CCC3=C(C2)N=CN=C3NC2=CC=C(C(=O)NCC(=O)N3CCC(CN4CCN(C(=O)C5=CC=CC(N6CCC(=O)NC6=O)=C5)CC4)CC3)C(F)=N2)C=C1Cl	C43H44ClFN12O5	AR	P10275	CRBN	WO-2021058017-A1
TPD-SG524T	SCHEMBL23173116	6-[[7-(3-chloro-4-cyanophenyl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]amino]-N-[4-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperazin-1-yl]cyclohexyl]-2-fluoropyridine-3-carboxamide; SCHEMBL23173807; SCHEMBL23173808	N#CC1=CC=C(N2CCC3=C(C2)N=CN=C3NC2=CC=C(C(=O)NC3CCC(N4CCN(C5=CC=C(N6CCC(=O)NC6=O)C=C5)CC4)CC3)C(F)=N2)C=C1Cl	C40H41ClFN11O3	AR	P10275	CRBN	WO-2021058017-A1
TPD-B6PLNS	SCHEMBL23173226	6-[[7-(3-chloro-4-cyanophenyl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]amino]-N-[2-[4-[[4-[3-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperazin-1-yl]methyl]piperidin-1-yl]-2-oxoethyl]-2-fluoropyridine-3-carboxamide	N#CC1=CC=C(N2CCC3=C(C2)N=CN=C3NC2=CC=C(C(=O)NCC(=O)N3CCC(CN4CCN(C5=CC=CC(N6CCC(=O)NC6=O)=C5)CC4)CC3)C(F)=N2)C=C1Cl	C42H44ClFN12O4	AR	P10275	CRBN	WO-2021058017-A1
TPD-7WDZ01	SCHEMBL23173243	6-[[7-(3-chloro-4-cyanophenyl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]amino]-N-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperazin-1-yl]methyl]cyclohexyl]-2-fluoropyridine-3-carboxamide; SCHEMBL23173497	[H][C@]1(CN2CCN(C3=CC=C(N4CCC(=O)NC4=O)C=C3)CC2)CC[C@]([H])(NC(=O)C2=CC=C(NC3=NC=NC4=C3CCN(C3=CC=C(C#N)C(Cl)=C3)C4)N=C2F)CC1	C41H43ClFN11O3	AR	P10275	CRBN	WO-2021058017-A1
TPD-DLV4ML	SCHEMBL23173260	6-[[7-(3-chloro-4-cyanophenyl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]amino]-N-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]amino]spiro[3.5]nonan-7-yl]-2-fluoropyridine-3-carboxamide	N#CC1=CC=C(N2CCC3=C(C2)N=CN=C3NC2=CC=C(C(=O)NC3CCC4(CC3)CC(NC3=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C3)C4)C(F)=N2)C=C1Cl	C42H38ClFN10O5	AR	P10275	CRBN	WO-2021058017-A1
TPD-4B94MI	WO2021058017A1_49	.	N#CC1=CC=C(N2CCC3=C(C2)N=CN=C3NC2=CC=C(C(=O)NC3CC4(C3)CN(CC3CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC3)C4)C(F)=N2)C=C1Cl	C45H43ClFN11O5	AR	P10275	CRBN	WO-2021058017-A1
TPD-RYS0YC	WO2021058017A1_5	.	N#CC1=CC=C(N2CCC3=C(C2)N=CN=C3NC2=NC(F)=C(C(=O)NCCOCCOCCOCCCC3=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)C=C2)C=C1Cl	C42H43ClFN9O7	AR	P10275	CRBN	WO-2021058017-A1
TPD-W16T22	SCHEMBL23173148	6-[[7-(3-chloro-4-cyanophenyl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]amino]-N-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]-2-azaspiro[3.3]heptan-6-yl]-2-fluoropyridine-3-carboxamide	N#CC1=CC=C(N2CCC3=C(C2)N=CN=C3NC2=CC=C(C(=O)NC3CC4(C3)CN(C3CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC3)C4)C(F)=N2)C=C1Cl	C44H41ClFN11O5	AR	P10275	CRBN	WO-2021058017-A1
TPD-M5ZB2F	SCHEMBL23173686	6-[[7-(3-chloro-4-cyanophenyl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]amino]-N-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]spiro[3.3]heptan-6-yl]-2-fluoropyridine-3-carboxamide	N#CC1=CC=C(N2CCC3=C(C2)N=CN=C3NC2=CC=C(C(=O)NC3CC4(C3)CC(N3CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC3)C4)C(F)=N2)C=C1Cl	C44H41ClFN11O5	AR	P10275	CRBN	WO-2021058017-A1
TPD-227OER	SCHEMBL23173699	6-[[7-(3-chloro-4-cyanophenyl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]amino]-N-[7-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]spiro[3.5]nonan-2-yl]-2-fluoropyridine-3-carboxamide	N#CC1=CC=C(N2CCC3=C(C2)N=CN=C3NC2=CC=C(C(=O)NC3CC4(CCC(N5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C3)C(F)=N2)C=C1Cl	C46H45ClFN11O5	AR	P10275	CRBN	WO-2021058017-A1
TPD-31BABS	SCHEMBL23173127	6-[[7-(3-chloro-4-cyanophenyl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]amino]-N-[6-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]spiro[3.3]heptan-2-yl]-2-fluoropyridine-3-carboxamide	N#CC1=CC=C(N2CCC3=C(C2)N=CN=C3NC2=CC=C(C(=O)NC3CC4(CC(CN5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)C4)C3)C(F)=N2)C=C1Cl	C45H43ClFN11O5	AR	P10275	CRBN	WO-2021058017-A1
TPD-9LJE6Y	SCHEMBL23173707	6-[[7-(3-chloro-4-cyanophenyl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]amino]-N-[7-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazine-1-carbonyl]spiro[3.5]nonan-2-yl]-2-fluoropyridine-3-carboxamide	N#CC1=CC=C(N2CCC3=C(C2)N=CN=C3NC2=CC=C(C(=O)NC3CC4(CCC(C(=O)N5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C3)C(F)=N2)C=C1Cl	C47H45ClFN11O6	AR	P10275	CRBN	WO-2021058017-A1
TPD-AMCPJS	WO2021058017A1_55	.	N#CC1=CC=C(N2CCC3=C(C2)N=CN=C3NC2=CC=C(C(=O)NC3CC4(C3)CC(C(=O)N3CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC3)C4)C(F)=N2)C=C1Cl	C45H41ClFN11O6	AR	P10275	CRBN	WO-2021058017-A1
TPD-DC130J	WO2021058017A1_56	.	N#CC1=CC=C(N2CCC3=C(C2)N=CN=C3NC2=CC=C(C(=O)NC3CCC4(CC3)CN(C3CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC3)C4)C(F)=N2)C=C1Cl	C46H45ClFN11O5	AR	P10275	CRBN	WO-2021058017-A1
TPD-ACZA34	SCHEMBL23173824	6-[[7-(3-chloro-4-cyanophenyl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]amino]-N-[7-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]-7-azaspiro[3.5]nonan-2-yl]-2-fluoropyridine-3-carboxamide	N#CC1=CC=C(N2CCC3=C(C2)N=CN=C3NC2=CC=C(C(=O)NC3CC4(CCN(C5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C3)C(F)=N2)C=C1Cl	C46H45ClFN11O5	AR	P10275	CRBN	WO-2021058017-A1
TPD-BFAIBE	SCHEMBL23173234	6-[[7-(3-chloro-4-cyanophenyl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]amino]-N-[7-[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]-7-azaspiro[3.5]nonan-2-yl]-2-fluoropyridine-3-carboxamide	N#CC1=CC=C(N2CCC3=C(C2)N=CN=C3NC2=CC=C(C(=O)NC3CC4(CCN(C5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)CC5)CC4)C3)C(F)=N2)C=C1Cl	C46H47ClFN11O4	AR	P10275	CRBN	WO-2021058017-A1
TPD-BC7Q10	SCHEMBL23173229	6-[[7-(3-chloro-4-cyanophenyl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]amino]-N-[8-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyoctyl]-2-fluoropyridine-3-carboxamide	N#CC1=CC=C(N2CCC3=C(C2)N=CN=C3NC2=NC(F)=C(C(=O)NCCCCCCCCOC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)C=C2)C=C1Cl	C41H39ClFN9O6	AR	P10275	CRBN	WO-2021058017-A1
TPD-Y56PZS	SCHEMBL23173711	6-[[7-(3-chloro-4-cyanophenyl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]amino]-N-[3-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]-3-azaspiro[5.5]undecan-9-yl]-2-fluoropyridine-3-carboxamide	N#CC1=CC=C(N2CCC3=C(C2)N=CN=C3NC2=CC=C(C(=O)NC3CCC4(CC3)CCN(C3CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC3)CC4)C(F)=N2)C=C1Cl	C48H49ClFN11O5	AR	P10275	CRBN	WO-2021058017-A1
TPD-G74JVR	SCHEMBL23173684	6-[[7-(3-chloro-4-cyanophenyl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]amino]-N-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]cyclohexyl]-2-fluoropyridine-3-carboxamide; SCHEMBL23173688	[H][C@]1(CN2CCN(C3=C(F)C=C4C(=O)N(C5CCC(=O)NC5=O)CC4=C3)CC2)CC[C@]([H])(NC(=O)C2=CC=C(NC3=NC=NC4=C3CCN(C3=CC=C(C#N)C(Cl)=C3)C4)N=C2F)CC1	C44H44ClF2N11O4	AR	P10275	CRBN	WO-2021058017-A1
TPD-7PGBI4	SCHEMBL23173524	6-[[7-(3-chloro-4-cyanophenyl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]amino]-N-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]cyclohexyl]-2-fluoropyridine-3-carboxamide; SCHEMBL23173532	[H][C@]1(CN2CCN(C3=CC=C4C(=O)N(C5CCC(=O)NC5=O)CC4=C3)CC2)CC[C@]([H])(NC(=O)C2=CC=C(NC3=NC=NC4=C3CCN(C3=CC=C(C#N)C(Cl)=C3)C4)N=C2F)CC1	C44H45ClFN11O4	AR	P10275	CRBN	WO-2021058017-A1
TPD-ZKGZ94	WO2021058017A1_63	.	[H][C@]1(CN2CCN(C3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)CC2)CC[C@]([H])(NC(=O)C2=CC=C(NC3=NC=NC4=C3CCN(C3=CC=C(C#N)C(Cl)=C3)C4)N=C2F)CC1	C44H43ClFN11O5	AR	P10275	CRBN	WO-2021058017-A1
TPD-CTPA01	SCHEMBL23173527	6-[[7-(3-chloro-4-cyanophenyl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]amino]-N-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1-oxo-3H-isoindol-4-yl]piperazin-1-yl]methyl]cyclohexyl]-2-fluoropyridine-3-carboxamide; SCHEMBL23173534	[H][C@]1(CN2CCN(C3=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC(F)=C3)CC2)CC[C@]([H])(NC(=O)C2=CC=C(NC3=NC=NC4=C3CCN(C3=CC=C(C#N)C(Cl)=C3)C4)N=C2F)CC1	C44H44ClF2N11O4	AR	P10275	CRBN	WO-2021058017-A1
TPD-YNYXQV	SCHEMBL23173766	6-[[7-[4-cyano-3-(trifluoromethyl)phenyl]-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]amino]-N-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]cyclohexyl]-2-fluoropyridine-3-carboxamide; SCHEMBL23173767	[H][C@]1(CN2CCN(C3=C(F)C=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)CC2)CC[C@]([H])(NC(=O)C2=CC=C(NC3=NC=NC4=C3CCN(C3=CC=C(C#N)C(C(F)(F)F)=C3)C4)N=C2F)CC1	C45H42F5N11O5	AR	P10275	CRBN	WO-2021058017-A1
TPD-1D0QPD	WO2021058017A1_66	.	[H][C@]1(CN2CCN(C3=C(F)C=C4C(=O)N(C5CCC(=O)NC5=O)CC4=C3)CC2)CC[C@]([H])(NC(=O)C2=CC=C(NC3=NC=NC4=C3CCN(C3=CC=C(C#N)C(C(F)(F)F)=C3)C4)N=C2F)CC1	C45H44F5N11O4	AR	P10275	CRBN	WO-2021058017-A1
TPD-TGRHWK	SCHEMBL23173719	6-[[7-[4-cyano-3-(trifluoromethyl)phenyl]-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]amino]-N-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]cyclohexyl]-2-fluoropyridine-3-carboxamide	[H][C@]1(CN2CCN(C3=CC=C4C(=O)N(C5CCC(=O)NC5=O)CC4=C3)CC2)CC[C@]([H])(NC(=O)C2=CC=C(NC3=NC=NC4=C3CCN(C3=CC=C(C#N)C(C(F)(F)F)=C3)C4)N=C2F)CC1	C45H45F4N11O4	AR	P10275	CRBN	WO-2021058017-A1
TPD-XNFZ1C	WO2021058017A1_68	.	[H][C@]1(CN2CCN(C3=CC=C(N4CCC(=O)NC4=O)C=C3F)CC2)CC[C@]([H])(NC(=O)C2=CC=C(NC3=NC=NC4=C3CCN(C3=CC=C(C#N)C(C(F)(F)F)=C3)C4)N=C2F)CC1	C42H42F5N11O3	AR	P10275	CRBN	WO-2021058017-A1
TPD-LZTK5B	SCHEMBL23173716	6-[[7-[4-cyano-3-(trifluoromethyl)phenyl]-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]amino]-N-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)-2-methylphenyl]piperazin-1-yl]methyl]cyclohexyl]-2-fluoropyridine-3-carboxamide	[H][C@]1(CN2CCN(C3=CC=C(N4CCC(=O)NC4=O)C=C3C)CC2)CC[C@]([H])(NC(=O)C2=CC=C(NC3=NC=NC4=C3CCN(C3=CC=C(C#N)C(C(F)(F)F)=C3)C4)N=C2F)CC1	C43H45F4N11O3	AR	P10275	CRBN	WO-2021058017-A1
TPD-5HQJG9	SCHEMBL23173779	6-[[7-[4-cyano-3-(trifluoromethyl)phenyl]-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]amino]-N-[4-[[4-[5-(2,4-dioxo-1,3-diazinan-1-yl)pyridin-2-yl]piperazin-1-yl]methyl]cyclohexyl]-2-fluoropyridine-3-carboxamide; SCHEMBL23173782	[H][C@]1(CN2CCN(C3=CC=C(N4CCC(=O)NC4=O)C=N3)CC2)CC[C@]([H])(NC(=O)C2=CC=C(NC3=NC=NC4=C3CCN(C3=CC=C(C#N)C(C(F)(F)F)=C3)C4)N=C2F)CC1	C41H42F4N12O3	AR	P10275	CRBN	WO-2021058017-A1
TPD-GHMGUY	WO2021058017A1_71	.	[H][C@]1(CN2CCN(C3=CC=C(N4CCC(=O)NC4=O)C=C3)CC2)CC[C@]([H])(NC(=O)C2=CC=C(NC3=NC=NC4=C3CCN(C3=CC=C(C#N)C(C(F)(F)F)=C3)C4)N=C2F)CC1	C42H43F4N11O3	AR	P10275	CRBN	WO-2021058017-A1
TPD-6OJ9NN	WO2021058017A1_72	.	[H][C@]1(CN2CCN(C3=CC=C(N4CCC(=O)NC4=O)C=C3)CC2)CC[C@@]([H])(NC(=O)C2=CC=C(NC3=NC=NC4=C3CCN(C3=CC=C(C#N)C(C(F)(F)F)=C3)C4)N=C2F)CC1	C42H43F4N11O3	AR	P10275	CRBN	WO-2021058017-A1
TPD-H45JFP	SCHEMBL23173732	6-[[7-[4-cyano-3-(trifluoromethyl)phenyl]-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]amino]-N-[1-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)-2-fluorophenyl]piperidin-4-yl]methyl]piperidin-4-yl]-2-fluoropyridine-3-carboxamide	N#CC1=CC=C(N2CCC3=C(C2)N=CN=C3NC2=CC=C(C(=O)NC3CCN(CC4CCN(C5=CC=C(N6CCC(=O)NC6=O)C=C5F)CC4)CC3)C(F)=N2)C=C1C(F)(F)F	C42H42F5N11O3	AR	P10275	CRBN	WO-2021058017-A1
TPD-XLUUIJ	SCHEMBL23173228	6-[[7-[4-cyano-3-(trifluoromethyl)phenyl]-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]amino]-N-[1-[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)-2-fluorophenyl]piperidin-4-yl]piperidin-4-yl]-2-fluoropyridine-3-carboxamide	N#CC1=CC=C(N2CCC3=C(C2)N=CN=C3NC2=CC=C(C(=O)NC3CCN(C4CCN(C5=CC=C(N6CCC(=O)NC6=O)C=C5F)CC4)CC3)C(F)=N2)C=C1C(F)(F)F	C41H40F5N11O3	AR	P10275	CRBN	WO-2021058017-A1
TPD-0KLNPT	SCHEMBL23173989	6-[[7-[4-cyano-3-(trifluoromethyl)phenyl]-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]amino]-N-[4-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)-2-fluorophenyl]piperazin-1-yl]cyclohexyl]-2-fluoropyridine-3-carboxamide	N#CC1=CC=C(N2CCC3=C(C2)N=CN=C3NC2=CC=C(C(=O)NC3CCC(N4CCN(C5=CC=C(N6CCC(=O)NC6=O)C=C5F)CC4)CC3)C(F)=N2)C=C1C(F)(F)F	C41H40F5N11O3	AR	P10275	CRBN	WO-2021058017-A1
TPD-741V6H	WO2021058017A1_76	.	N#CC1=CC=C(N2CCC3=C(C2)N=CN=C3NC2=CC=C(C(=O)NC3CCC(CN4CCN(C5=CC=C(N6CCC(=O)NC6=O)C=C5F)CC4)CC3)C(F)=N2)C=C1C(F)(F)F	C42H42F5N11O3	AR	P10275	CRBN	WO-2021058017-A1
TPD-DYPC94	SCHEMBL23173820	6-[[7-[4-cyano-3-(trifluoromethyl)phenyl]-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]amino]-N-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)-2-fluorophenyl]piperazin-1-yl]methyl]phenyl]-2-fluoropyridine-3-carboxamide	N#CC1=CC=C(N2CCC3=C(C2)N=CN=C3NC2=CC=C(C(=O)NC3=CC=C(CN4CCN(C5=CC=C(N6CCC(=O)NC6=O)C=C5F)CC4)C=C3)C(F)=N2)C=C1C(F)(F)F	C42H36F5N11O3	AR	P10275	CRBN	WO-2021058017-A1
TPD-MZVQOH	SCHEMBL23173567	6-[[7-[4-cyano-3-(trifluoromethyl)phenyl]-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]amino]-N-[4-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperazin-1-yl]phenyl]-2-fluoropyridine-3-carboxamide	N#CC1=CC=C(N2CCC3=C(C2)N=CN=C3NC2=CC=C(C(=O)NC3=CC=C(N4CCN(C5=CC=C(N6CCC(=O)NC6=O)C=C5)CC4)C=C3)C(F)=N2)C=C1C(F)(F)F	C41H35F4N11O3	AR	P10275	CRBN	WO-2021058017-A1
TPD-U3W2GU	SCHEMBL23173822	6-[[7-[4-cyano-3-(trifluoromethyl)phenyl]-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]amino]-N-[[4-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperazin-1-yl]phenyl]methyl]-2-fluoropyridine-3-carboxamide	N#CC1=CC=C(N2CCC3=C(C2)N=CN=C3NC2=CC=C(C(=O)NCC3=CC=C(N4CCN(C5=CC=C(N6CCC(=O)NC6=O)C=C5)CC4)C=C3)C(F)=N2)C=C1C(F)(F)F	C42H37F4N11O3	AR	P10275	CRBN	WO-2021058017-A1
TPD-BKFLHQ	SCHEMBL23173101	2-chloro-4-[4-[[5-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazine-1-carbonyl]-6-fluoropyridin-2-yl]amino]-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]benzonitrile	N#CC1=CC=C(N2CCC3=C(C2)N=CN=C3NC2=NC(F)=C(C(=O)N3CCN(CC4CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)C=C2)C=C1Cl	C43H41ClFN11O5	AR	P10275	CRBN	WO-2021058017-A1
TPD-3X3QR1	SCHEMBL23173550	6-[[7-(6-chloro-5-cyanopyridin-2-yl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]amino]-N-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]cyclohexyl]-2-fluoropyridine-3-carboxamide	[H][C@]1(CN2CCN(C3=C(F)C=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)CC2)CC[C@]([H])(NC(=O)C2=CC=C(NC3=NC=NC4=C3CCN(C3=CC=C(C#N)C(Cl)=N3)C4)N=C2F)CC1	C43H41ClF2N12O5	AR	P10275	CRBN	WO-2021058017-A1
TPD-00ZR26	SCHEMBL23173265	6-[[7-(6-chloro-5-cyanopyridin-2-yl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]amino]-N-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]cyclohexyl]-2-fluoropyridine-3-carboxamide	[H][C@]1(CN2CCN(C3=C(F)C=C4C(=O)N(C5CCC(=O)NC5=O)CC4=C3)CC2)CC[C@]([H])(NC(=O)C2=CC=C(NC3=NC=NC4=C3CCN(C3=CC=C(C#N)C(Cl)=N3)C4)N=C2F)CC1	C43H43ClF2N12O4	AR	P10275	CRBN	WO-2021058017-A1
TPD-S8WXHE	SCHEMBL23173735	6-[[7-(6-chloro-5-cyanopyridin-2-yl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]amino]-N-[4-[[4-[4-[(2,6-dioxopiperidin-3-yl)amino]phenyl]piperazin-1-yl]methyl]cyclohexyl]-2-fluoropyridine-3-carboxamide; SCHEMBL23173737	[H][C@]1(CN2CCN(C3=CC=C(NC4CCC(=O)NC4=O)C=C3)CC2)CC[C@]([H])(NC(=O)C2=CC=C(NC3=NC=NC4=C3CCN(C3=CC=C(C#N)C(Cl)=N3)C4)N=C2F)CC1	C41H44ClFN12O3	AR	P10275	CRBN	WO-2021058017-A1
TPD-YDCPOT	SCHEMBL23173558	6-[[7-(6-chloro-5-cyanopyridin-2-yl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]amino]-N-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperazin-1-yl]methyl]cyclohexyl]-2-fluoropyridine-3-carboxamide; SCHEMBL23173559	[H][C@]1(CN2CCN(C3=CC=C(N4CCC(=O)NC4=O)C=C3)CC2)CC[C@]([H])(NC(=O)C2=CC=C(NC3=NC=NC4=C3CCN(C3=CC=C(C#N)C(Cl)=N3)C4)N=C2F)CC1	C40H42ClFN12O3	AR	P10275	CRBN	WO-2021058017-A1
TPD-BNW55L	SCHEMBL23173255	6-[[7-(6-chloro-5-cyanopyridin-2-yl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]amino]-N-[4-[[4-[4-(2,6-dioxopiperidin-3-yl)phenyl]piperazin-1-yl]methyl]cyclohexyl]-2-fluoropyridine-3-carboxamide	[H][C@]1(CN2CCN(C3=CC=C(C4CCC(=O)NC4=O)C=C3)CC2)CC[C@]([H])(NC(=O)C2=CC=C(NC3=NC=NC4=C3CCN(C3=CC=C(C#N)C(Cl)=N3)C4)N=C2F)CC1	C41H43ClFN11O3	AR	P10275	CRBN	WO-2021058017-A1
TPD-E6193G	SCHEMBL23173114	6-[[7-(6-chloro-5-cyanopyridin-2-yl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]amino]-N-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]cyclohexyl]-2-fluoropyridine-3-carboxamide	[H][C@]1(NC(=O)C2=CC=C(NC3=NC=NC4=C3CCN(C3=CC=C(C#N)C(Cl)=N3)C4)N=C2F)CC[C@]([H])(N2CCN(C3=C(F)C=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)CC2)CC1	C42H39ClF2N12O5	AR	P10275	CRBN	WO-2021058017-A1
TPD-X6UG09	SCHEMBL23173277	6-[[7-(6-chloro-5-cyanopyridin-2-yl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]amino]-N-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]cyclohexyl]-2-fluoropyridine-3-carboxamide	[H][C@]1(NC(=O)C2=CC=C(NC3=NC=NC4=C3CCN(C3=CC=C(C#N)C(Cl)=N3)C4)N=C2F)CC[C@]([H])(C2CCN(C3=C(F)C=C4C(=O)N(C5CCC(=O)NC5=O)CC4=C3)CC2)CC1	C43H42ClF2N11O4	AR	P10275	CRBN	WO-2021058017-A1
TPD-EYMMOO	SCHEMBL23173280	6-[[7-(6-chloro-5-cyanopyridin-2-yl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]amino]-N-[4-[4-[4-[(2,6-dioxopiperidin-3-yl)amino]phenyl]piperazin-1-yl]cyclohexyl]-2-fluoropyridine-3-carboxamide	[H][C@]1(NC(=O)C2=CC=C(NC3=NC=NC4=C3CCN(C3=CC=C(C#N)C(Cl)=N3)C4)N=C2F)CC[C@]([H])(N2CCN(C3=CC=C(NC4CCC(=O)NC4=O)C=C3)CC2)CC1	C40H42ClFN12O3	AR	P10275	CRBN	WO-2021058017-A1
TPD-02XK3D	SCHEMBL23173830	6-[[7-(6-chloro-5-cyanopyridin-2-yl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]amino]-N-[4-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperazin-1-yl]cyclohexyl]-2-fluoropyridine-3-carboxamide	[H][C@]1(NC(=O)C2=CC=C(NC3=NC=NC4=C3CCN(C3=CC=C(C#N)C(Cl)=N3)C4)N=C2F)CC[C@]([H])(N2CCN(C3=CC=C(N4CCC(=O)NC4=O)C=C3)CC2)CC1	C39H40ClFN12O3	AR	P10275	CRBN	WO-2021058017-A1
TPD-MFTS0V	SCHEMBL23173531	6-[[7-[5-cyano-6-(trifluoromethyl)pyridin-2-yl]-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]amino]-N-[4-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperazin-1-yl]cyclohexyl]-2-fluoropyridine-3-carboxamide	[H][C@]1(NC(=O)C2=CC=C(NC3=NC=NC4=C3CCN(C3=CC=C(C#N)C(C(F)(F)F)=N3)C4)N=C2F)CC[C@]([H])(N2CCN(C3=CC=C(N4CCC(=O)NC4=O)C=C3)CC2)CC1	C40H40F4N12O3	AR	P10275	CRBN	WO-2021058017-A1
TPD-E8EIC1	SCHEMBL23173979	2-chloro-4-[4-[[5-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperazine-1-carbonyl]-6-fluoropyridin-2-yl]amino]-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]benzonitrile	N#CC1=CC=C(N2CCC3=C(C2)N=CN=C3NC2=NC(F)=C(C(=O)N3CCN(C4CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)C=C2)C=C1Cl	C42H39ClFN11O5	AR	P10275	CRBN	WO-2021058017-A1
TPD-VGHO6Z	SCHEMBL23173269	6-[[7-(6-chloro-5-cyanopyridin-2-yl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]amino]-N-[4-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperazin-1-yl]butyl]-2-fluoropyridine-3-carboxamide	N#CC1=CC=C(N2CCC3=C(C2)N=CN=C3NC2=CC=C(C(=O)NCCCCN3CCN(C4=CC=C(N5CCC(=O)NC5=O)C=C4)CC3)C(F)=N2)N=C1Cl	C37H38ClFN12O3	AR	P10275	CRBN	WO-2021058017-A1
TPD-RAPK9N	SCHEMBL23173253	6-[[7-(6-chloro-5-cyanopyridin-2-yl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]amino]-N-[3-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperazin-1-yl]propyl]-2-fluoropyridine-3-carboxamide	N#CC1=CC=C(N2CCC3=C(C2)N=CN=C3NC2=CC=C(C(=O)NCCCN3CCN(C4=CC=C(N5CCC(=O)NC5=O)C=C4)CC3)C(F)=N2)N=C1Cl	C36H36ClFN12O3	AR	P10275	CRBN	WO-2021058017-A1
TPD-NWYWC3	SCHEMBL23173275	6-[[7-(6-chloro-5-cyanopyridin-2-yl)-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-4-yl]amino]-N-[2-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperazin-1-yl]ethyl]-2-fluoropyridine-3-carboxamide	N#CC1=CC=C(N2CCC3=C(C2)N=CN=C3NC2=CC=C(C(=O)NCCN3CCN(C4=CC=C(N5CCC(=O)NC5=O)C=C4)CC3)C(F)=N2)N=C1Cl	C35H34ClFN12O3	AR	P10275	CRBN	WO-2021058017-A1
TPD-XS0SAF	SCHEMBL23225985	4-[2-[2-[2-[2-[4-[(3R)-3-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidine-1-carbonyl]triazol-1-yl]ethoxy]ethoxy]ethoxy]ethoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	Nc1ncnc2c1c(-c1ccc(Oc3ccccc3)cc1)nn2[C@@H]1CCCN(C(=O)c2cn(CCOCCOCCOCCOc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)nn2)C1	C46H47N11O10	BTK	Q06187	CRBN	WO-2021068380-A1
TPD-XYO3Z9	SCHEMBL23225986	5-[2-[2-[2-[2-[4-[(3R)-3-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidine-1-carbonyl]triazol-1-yl]ethoxy]ethoxy]ethoxy]ethylamino]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	Nc1ncnc2c1c(-c1ccc(Oc3ccccc3)cc1)nn2[C@@H]1CCCN(C(=O)c2cn(CCOCCOCCOCCNc3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)nn2)C1	C46H48N12O9	BTK	Q06187	CRBN	WO-2021068380-A1
TPD-DMCZO0	SCHEMBL23226042	2-[(3R)-3-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]-N-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethyl]acetamide	Nc1ncnc2c1c(-c1ccc(Oc3ccccc3)cc1)nn2[C@@H]1CCCN(CC(=O)NCCOCCOCCOCCNc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)C1	C45H50N10O9	BTK	Q06187	CRBN	WO-2021068380-A1
TPD-GCIPAN	WO2021068380A1_4	.	Nc1ncnc2c1c(-c1ccc(Oc3ccccc3)cc1)nn2[C@@H]1CCCN(CC(=O)NCCOCCOCCNc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)C1	C43H46N10O8	BTK	Q06187	CRBN	WO-2021068380-A1
TPD-T6A60H	SCHEMBL23226045	2-[(3R)-3-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]-N-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]amino]ethoxy]ethoxy]ethoxy]ethyl]acetamide	Nc1ncnc2c1c(-c1ccc(Oc3ccccc3)cc1)nn2[C@@H]1CCCN(CC(=O)NCCOCCOCCOCCNc2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)C1	C45H50N10O9	BTK	Q06187	CRBN	WO-2021068380-A1
TPD-09VA30	SCHEMBL23226043	3-[7-[2-[2-[2-[2-[4-[(3R)-3-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidine-1-carbonyl]triazol-1-yl]ethoxy]ethoxy]ethoxy]ethylamino]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	Nc1ncnc2c1c(-c1ccc(Oc3ccccc3)cc1)nn2[C@@H]1CCCN(C(=O)c2cn(CCOCCOCCOCCNc3cccc4c3CN(C3CCC(=O)NC3=O)C4=O)nn2)C1	C46H50N12O8	BTK	Q06187	CRBN	WO-2021068380-A1
TPD-IPPULD	SCHEMBL23226006	3-[5-[2-[2-[2-[2-[4-[(3R)-3-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidine-1-carbonyl]triazol-1-yl]ethoxy]ethoxy]ethoxy]ethylamino]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	Nc1ncnc2c1c(-c1ccc(Oc3ccccc3)cc1)nn2[C@@H]1CCCN(C(=O)c2cn(CCOCCOCCOCCNc3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4)nn2)C1	C46H50N12O8	BTK	Q06187	CRBN	WO-2021068380-A1
TPD-YKRJNH	SCHEMBL23226008	2-[(3R)-3-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]-N-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethyl]acetamide	Nc1ncnc2c1c(-c1ccc(Oc3ccccc3)cc1)nn2[C@@H]1CCCN(CC(=O)NCCOCCOCCOCCNc2cccc3c2CN(C2CCC(=O)NC2=O)C3=O)C1	C45H52N10O8	BTK	Q06187	CRBN	WO-2021068380-A1
TPD-IDL3QN	SCHEMBL23226005	4-[2-[2-[2-[2-[4-[4-[4-Amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidine-1-carbonyl]triazol-1-yl]ethoxy]ethoxy]ethoxy]ethylamino]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	Nc1ncnc2c1c(-c1ccc(Oc3ccccc3)cc1)nn2C1CCN(C(=O)c2cn(CCOCCOCCOCCNc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)nn2)CC1	C46H48N12O9	BTK	Q06187	CRBN	WO-2021068380-A1
TPD-P63BD8	SCHEMBL23226007	4-[[9-[3-[4-Amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]-9-oxononyl]amino]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione; PD173369	Nc1ncnc2c1c(-c1ccc(Oc3ccccc3)cc1)nn2C1CCCN(C(=O)CCCCCCCCNc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)C1	C44H47N9O6	BTK	Q06187	CRBN	WO-2021068380-A1
TPD-PAGQSH	SCHEMBL23226009	4-[[7-[3-[4-Amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]-7-oxoheptyl]amino]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione; PD173363	Nc1ncnc2c1c(-c1ccc(Oc3ccccc3)cc1)nn2C1CCCN(C(=O)CCCCCCNc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)C1	C42H43N9O6	BTK	Q06187	CRBN	WO-2021068380-A1
TPD-8F5TLV	SCHEMBL23226047	4-[8-[3-[4-Amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]octylamino]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	Nc1ncnc2c1c(-c1ccc(Oc3ccccc3)cc1)nn2C1CCCN(CCCCCCCCNc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)C1	C43H47N9O5	BTK	Q06187	CRBN	WO-2021068380-A1
TPD-IX9V1Y	SCHEMBL23225989	5-[[8-[3-[4-Amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]-8-oxooctyl]amino]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione; PD173367	Nc1ncnc2c1c(-c1ccc(Oc3ccccc3)cc1)nn2C1CCCN(C(=O)CCCCCCCNc2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)C1	C43H45N9O6	BTK	Q06187	CRBN	WO-2021068380-A1
TPD-8RBI83	SCHEMBL23225994	8-[3-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]-N-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]octanamide	Nc1ncnc2c1c(-c1ccc(Oc3ccccc3)cc1)nn2C1CCCN(CCCCCCCC(=O)Nc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)C1	C43H45N9O6	BTK	Q06187	CRBN	WO-2021068380-A1
TPD-443349	SCHEMBL23225988	3-[6-[8-[3-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]-8-oxooctyl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	Nc1ncnc2c1c(-c1ccc(Oc3ccccc3)cc1)nn2C1CCCN(C(=O)CCCCCCCc2ccc3c(c2)CN(C2CCC(=O)NC2=O)C3=O)C1	C43H46N8O5	BTK	Q06187	CRBN	WO-2021068380-A1
TPD-0NDH7H	SCHEMBL23225990	3-[7-[8-[3-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]octyl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	Nc1ncnc2c1c(-c1ccc(Oc3ccccc3)cc1)nn2C1CCCN(CCCCCCCCc2cccc3c2CN(C2CCC(=O)NC2=O)C3=O)C1	C43H48N8O4	BTK	Q06187	CRBN	WO-2021068380-A1
TPD-KKSNGB	SCHEMBL23225996	3-[7-[8-[3-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]-8-oxooctyl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	Nc1ncnc2c1c(-c1ccc(Oc3ccccc3)cc1)nn2C1CCCN(C(=O)CCCCCCCc2cccc3c2CN(C2CCC(=O)NC2=O)C3=O)C1	C43H46N8O5	BTK	Q06187	CRBN	WO-2021068380-A1
TPD-HL2APC	SCHEMBL23603037	2-Chloro-4-[5-[4-[3-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]azetidin-1-yl]phenyl]-3,3-dimethyl-2-oxoindol-1-yl]benzonitrile	CC1(C)C(=O)N(c2ccc(C#N)c(Cl)c2)c2ccc(-c3ccc(N4CC(CN5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)cc3)cc21	C44H40ClN7O5	AR	P10275	CRBN	WO-2021129653-A1
TPD-MZ142C	SCHEMBL23602981	4-[5-[4-[3-[[4-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]azetidin-1-yl]phenyl]-3,3-dimethyl-2-oxoindol-1-yl]-2-methoxybenzonitrile	COc1cc(N2C(=O)C(C)(C)c3cc(-c4ccc(N5CC(CN6CCN(c7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)C5)cc4)ccc32)ccc1C#N	C45H43N7O6	AR	P10275	CRBN	WO-2021129653-A1
TPD-J9NKAE	SCHEMBL23602987	4-[5-[4-[3-[[4-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]azetidin-1-yl]phenyl]-3,3-dimethyl-2-oxoindol-1-yl]-2-(trifluoromethyl)benzonitrile	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)c2ccc(-c3ccc(N4CC(CN5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)cc3)cc21	C45H40F3N7O5	AR	P10275	CRBN	WO-2021129653-A1
TPD-7FBYRQ	SCHEMBL23602976	2-chloro-4-[5-[4-[3-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]azetidin-1-yl]phenyl]-3,3-dimethyl-2-oxoindol-1-yl]benzonitrile	CC1(C)C(=O)N(c2ccc(C#N)c(Cl)c2)c2ccc(-c3ccc(N4CC(CN5CCN(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC5)C4)cc3)cc21	C44H42ClN7O4	AR	P10275	CRBN	WO-2021129653-A1
TPD-EHNUL7	SCHEMBL23603009	2-Chloro-4-[5-[4-[3-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]-3-fluoroazetidin-1-yl]phenyl]-3,3-dimethyl-2-oxoindol-1-yl]benzonitrile	CC1(C)C(=O)N(c2ccc(C#N)c(Cl)c2)c2ccc(-c3ccc(N4CC(F)(CN5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)cc3)cc21	C44H39ClFN7O5	AR	P10275	CRBN	WO-2021129653-A1
TPD-I7G8UJ	SCHEMBL23603004	2-Chloro-4-[5-[5-[3-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]azetidin-1-yl]pyrimidin-2-yl]-3,3-dimethyl-2-oxoindol-1-yl]benzonitrile	CC1(C)C(=O)N(c2ccc(C#N)c(Cl)c2)c2ccc(-c3ncc(N4CC(CN5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)cn3)cc21	C42H38ClN9O5	AR	P10275	CRBN	WO-2021129653-A1
TPD-UXRU3T	SCHEMBL23602980	2-Chloro-4-[5-[4-[3-[[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]azetidin-1-yl]phenyl]-3,3-dimethyl-2-oxoindol-1-yl]benzonitrile	CC1(C)C(=O)N(c2ccc(C#N)c(Cl)c2)c2ccc(-c3ccc(N4CC(CN5CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)cc3)cc21	C44H39ClFN7O5	AR	P10275	CRBN	WO-2021129653-A1
TPD-KX8T9I	SCHEMBL23603005	2-Chloro-4-[5-[6-[3-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]azetidin-1-yl]pyridazin-3-yl]-3,3-dimethyl-2-oxoindol-1-yl]benzonitrile	CC1(C)C(=O)N(c2ccc(C#N)c(Cl)c2)c2ccc(-c3ccc(N4CC(CN5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)nn3)cc21	C42H38ClN9O5	AR	P10275	CRBN	WO-2021129653-A1
TPD-Z4E72Q	WO2021129653A1_9	.	CC1(C)C(=O)N(c2ccc(C#N)c(Cl)c2)c2ccc(C3=CC=C(N4CC(CN5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)NC3)cc21	C43H41ClN8O5	AR	P10275	CRBN	WO-2021129653-A1
TPD-K0O9JP	SCHEMBL23603463	2-Chloro-4-[5-[5-[3-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]azetidin-1-yl]pyrazin-2-yl]-3,3-dimethyl-2-oxoindol-1-yl]benzonitrile	CC1(C)C(=O)N(c2ccc(C#N)c(Cl)c2)c2ccc(-c3cnc(N4CC(CN5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)cn3)cc21	C42H38ClN9O5	AR	P10275	CRBN	WO-2021129653-A1
TPD-1GP5MF	SCHEMBL23602988	3-Chloro-5-[5-[4-[3-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]azetidin-1-yl]phenyl]-3,3-dimethyl-2-oxoindol-1-yl]pyridine-2-carbonitrile	CC1(C)C(=O)N(c2cnc(C#N)c(Cl)c2)c2ccc(-c3ccc(N4CC(CN5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)cc3)cc21	C43H39ClN8O5	AR	P10275	CRBN	WO-2021129653-A1
TPD-MEYUDF	SCHEMBL23603272	2-Chloro-4-[5-[4-[1-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]ethyl]pyrazol-4-yl]phenyl]-3,3-dimethyl-2-oxoindol-1-yl]benzonitrile	CC1(C)C(=O)N(c2ccc(C#N)c(Cl)c2)c2ccc(-c3ccc(-c4cnn(CCN5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)c4)cc3)cc21	C45H39ClN8O5	AR	P10275	CRBN	WO-2021129653-A1
TPD-ONK8WG	SCHEMBL23603277	2-Chloro-4-[5-[4-[1-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]propyl]pyrazol-4-yl]phenyl]-3,3-dimethyl-2-oxoindol-1-yl]benzonitrile	CC1(C)C(=O)N(c2ccc(C#N)c(Cl)c2)c2ccc(-c3ccc(-c4cnn(CCCN5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)c4)cc3)cc21	C46H41ClN8O5	AR	P10275	CRBN	WO-2021129653-A1
TPD-ROG0GJ	SCHEMBL23603069	2-Chloro-4-[5-[6-[3-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]azetidin-1-yl]-2-fluoropyridin-3-yl]-3,3-dimethyl-2-oxoindol-1-yl]benzonitrile	CC1(C)C(=O)N(c2ccc(C#N)c(Cl)c2)c2ccc(-c3ccc(N4CC(CN5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)nc3F)cc21	C43H38ClFN8O5	AR	P10275	CRBN	WO-2021129653-A1
TPD-6HZFZN	SCHEMBL23603274	4-[5-[6-[3-[[4-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]azetidin-1-yl]-2-fluoropyridin-3-yl]-3,3-dimethyl-2-oxoindol-1-yl]-2-(trifluoromethyl)benzonitrile	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)c2ccc(-c3ccc(N4CC(CN5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)nc3F)cc21	C44H38F4N8O5	AR	P10275	CRBN	WO-2021129653-A1
TPD-CV2JGR	SCHEMBL23630348	2-[4-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]piperazin-1-yl]-N-[(2S)-1-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]pyridine-4-carboxamide; SCHEMBL29943860	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)c2ccnc(N3CCN(c4cc(-c5ccccc5O)nnc4N)CC3)c2)C(C)(C)C)cc1	C42H48N10O5S	SMARCA2	P51531	VHL	WO-2021142247-A1
TPD-CQBVQE	SCHEMBL23630591	6-[4-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]piperazin-1-yl]-N-[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]pyridine-2-carboxamide; SCHEMBL29943874; SCHEMBL29943876; PD215567	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)c2cccc(N3CCN(c4cc(-c5ccccc5O)nnc4N)CC3)n2)C(C)(C)C)cc1	C43H50N10O5S	SMARCA2	P51531	VHL	WO-2021142247-A1
TPD-1AETO6	N-(2-{4-[(6M)-3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]piperazin-1-yl}pyridine-4-carbonyl)-3-methyl-L-valyl-(4R)-4-hydroxy-N-{(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl}-L-prolinamide	N-(2-{4-[(6M)-3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]piperazin-1-yl}pyridine-4-carbonyl)-3-methyl-L-valyl-(4R)-4-hydroxy-N-{(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl}-L-prolinamide; PROTAC SMARCA2 degrader-8; orb2664212; SCHEMBL23630481; SCHEMBL29943904; PD215565; HY-161882; 2669027-50-1; YHB	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)c2ccnc(N3CCN(c4cc(-c5ccccc5O)nnc4N)CC3)c2)C(C)(C)C)cc1	C43H50N10O5S	SMARCA2	P51531	VHL	WO-2021142247-A1
TPD-YGQWZ2	SCHEMBL23630506	(2S,4R)-1-[(2S)-2-[[3-[4-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]piperazin-1-yl]benzoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL29943872; PD215571	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)c2cccc(N3CCN(c4cc(-c5ccccc5O)nnc4N)CC3)c2)C(C)(C)C)cc1	C44H51N9O5S	SMARCA2	P51531	VHL	WO-2021142247-A1
TPD-MN4KUP	SCHEMBL23630469	2-[4-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]piperazin-1-yl]-N-[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]-1,3-thiazole-4-carboxamide; SCHEMBL29943882; PD215573	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)c2csc(N3CCN(c4cc(-c5ccccc5O)nnc4N)CC3)n2)C(C)(C)C)cc1	C41H48N10O5S2	SMARCA2	P51531	VHL	WO-2021142247-A1
TPD-H87ALF	SCHEMBL23630327	(2S,4R)-1-[(2S)-2-[[5-[4-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]piperazin-1-yl]thiophene-2-carbonyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL29943890	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)c2ccc(N3CCN(c4cc(-c5ccccc5O)nnc4N)CC3)s2)C(C)(C)C)cc1	C42H49N9O5S2	SMARCA2	P51531	VHL	WO-2021142247-A1
TPD-W1O8C0	SCHEMBL23630391	6-[4-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]piperazin-1-yl]-N-[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]pyridine-3-carboxamide; SCHEMBL29943929; PD215569	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)c2ccc(N3CCN(c4cc(-c5ccccc5O)nnc4N)CC3)nc2)C(C)(C)C)cc1	C43H50N10O5S	SMARCA2	P51531	VHL	WO-2021142247-A1
TPD-BE83OU	SCHEMBL23630476	(2S,4R)-1-[(2S)-2-[[2-[2-[4-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]piperazin-1-yl]pyridin-4-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL29943982; PD215575	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)Cc2ccnc(N3CCN(c4cc(-c5ccccc5O)nnc4N)CC3)c2)C(C)(C)C)cc1	C44H52N10O5S	SMARCA2	P51531	VHL	WO-2021142247-A1
TPD-NWQE4I	SCHEMBL23630380	(2S,4R)-1-[(2S)-2-[3-[2-[4-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]piperazin-1-yl]pyridin-4-yl]propanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL29943878; PD215577	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCc2ccnc(N3CCN(c4cc(-c5ccccc5O)nnc4N)CC3)c2)C(C)(C)C)cc1	C45H54N10O5S	SMARCA2	P51531	VHL	WO-2021142247-A1
TPD-BMS87I	SCHEMBL23630494	6-[4-[6-amino-3-(2-hydroxyphenyl)-1,2,4-triazin-5-yl]piperazin-1-yl]-N-[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]pyridine-2-carboxamide; SCHEMBL29943863; PD215579	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)c2cccc(N3CCN(c4nc(-c5ccccc5O)nnc4N)CC3)n2)C(C)(C)C)cc1	C42H49N11O5S	SMARCA2	P51531	VHL	WO-2021142247-A1
TPD-AD8L4K	SCHEMBL23630448	N-[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]-2-[4-[6-(2-hydroxyphenyl)pyridazin-4-yl]piperazin-1-yl]pyridine-4-carboxamide; SCHEMBL29943873; PD215581	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)c2ccnc(N3CCN(c4cnnc(-c5ccccc5O)c4)CC3)c2)C(C)(C)C)cc1	C43H49N9O5S	SMARCA2	P51531	VHL	WO-2021142247-A1
TPD-0VS0IO	CHEMBL5073757	N-[4-[(2-aminophenyl)carbamoyl]phenyl]-N'-[(2S)-1-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]dodecanediamide; PD142065	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCCCCCC(=O)Nc2ccc(C(=O)Nc3ccccc3N)cc2)C(C)(C)C)cc1	C47H61N7O6S	HDAC1;HDAC2	Q13547/Q92769	VHL	WO-2021148811-A1
TPD-D40TFY	SCHEMBL23682388	N'-[4-[(2-aminophenyl)carbamoyl]phenyl]-N-[(3S,5S)-1-[(2S)-2-cyclohexyl-2-[[(2S)-2-(methylamino)propanoyl]amino]acetyl]-5-[[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]carbamoyl]pyrrolidin-3-yl]dodecanediamide; SCHEMBL30406288	CN[C@@H](C)C(=O)N[C@H](C(=O)N1C[C@@H](NC(=O)CCCCCCCCCCC(=O)Nc2ccc(C(=O)Nc3ccccc3N)cc2)C[C@H]1C(=O)N[C@@H]1CCCc2ccccc21)C1CCCCC1	C52H72N8O6	HDAC1;HDAC2	Q13547/Q92769	VHL	WO-2021148811-A1
TPD-WUFQQP	SCHEMBL23682378	(2S,4S)-4-[[2-[2-[2-[2-[4-[(2-aminophenyl)carbamoyl]anilino]-2-oxoethoxy]ethoxy]ethoxy]acetyl]amino]-1-[(2S)-2-cyclohexyl-2-[[(2S)-2-(methylamino)propanoyl]amino]acetyl]-N-[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]pyrrolidine-2-carboxamide	CN[C@@H](C)C(=O)N[C@H](C(=O)N1C[C@@H](NC(=O)COCCOCCOCC(=O)Nc2ccc(C(=O)Nc3ccccc3N)cc2)C[C@H]1C(=O)N[C@@H]1CCCc2ccccc21)C1CCCCC1	C48H64N8O9	HDAC1;HDAC2	Q13547/Q92769	VHL	WO-2021148811-A1
TPD-S4EV3M	CHEMBL5188888	[1-[8-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-8-oxooctyl]triazol-4-yl]methyl N-[[4-[(2-aminophenyl)carbamoyl]phenyl]methyl]carbamate	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCCn2cc(COC(=O)NCc3ccc(C(=O)Nc4ccccc4N)cc3)nn2)C(C)(C)C)cc1	C48H60N10O7S	HDAC1;HDAC2	Q13547/Q92769	VHL	WO-2021148811-A1
TPD-57MD61	SCHEMBL23682491	N-(2-aminophenyl)-4-[12-[3-[2-[(2S)-1-[(2S)-2-cyclohexyl-2-[[(2S)-2-(methylamino)propanoyl]amino]acetyl]pyrrolidin-2-yl]-1,3-thiazole-4-carbonyl]phenoxy]dodecanoylamino]benzamide	CN[C@@H](C)C(=O)N[C@H](C(=O)N1CCC[C@H]1c1nc(C(=O)c2cccc(OCCCCCCCCCCCC(=O)Nc3ccc(C(=O)Nc4ccccc4N)cc3)c2)cs1)C1CCCCC1	C51H67N7O6S	HDAC1;HDAC2	Q13547/Q92769	VHL	WO-2021148811-A1
TPD-54ATKS	WO2021148811A1_NC-PROTAC4	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCCCCCC(=O)Nc2ccc(C(=O)Nc3ccccc3N)cc2)C(C)(C)C)cc1	C47H61N7O6S	HDAC1;HDAC2	Q13547/Q92769	VHL	WO-2021148811-A1
TPD-VM7942	PD142070	N-(2-aminophenyl)-4-[6-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyacetyl]amino]hexanoylamino]benzamide	Nc1ccccc1NC(=O)c1ccc(NC(=O)CCCCCNC(=O)COc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)cc1	C34H34N6O8	HDAC1;HDAC2	Q13547/Q92769	VHL	WO-2021148811-A1
TPD-NPHFMA	PD142069	N-(2-aminophenyl)-4-[12-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyacetyl]amino]dodecanoylamino]benzamide	Nc1ccccc1NC(=O)c1ccc(NC(=O)CCCCCCCCCCCNC(=O)COc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)cc1	C40H46N6O8	HDAC1;HDAC2	Q13547/Q92769	VHL	WO-2021148811-A1
TPD-28SCFL	WO2021148811A1_PROTAC3	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCC(=O)Nc2ccc(C(=O)Nc3ccccc3N)cc2)C(C)(C)C)cc1	C43H53N7O6S	HDAC1;HDAC2	Q13547/Q92769	VHL	WO-2021148811-A1
TPD-EE7WR0	SCHEMBL27212265	N-(2-aminophenyl)-4-[9-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyacetyl]amino]nonanoylamino]benzamide	Nc1ccccc1NC(=O)c1ccc(NC(=O)CCCCCCCCNC(=O)COc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)cc1	C37H40N6O8	HDAC1;HDAC2	Q13547/Q92769	VHL	WO-2021148811-A1
TPD-F2QLVD	WO2021148811A1_PROTAC7	.	Nc1ccccc1NC(=O)c1ccc(NC(=O)COCCOCCOCCNC(=O)COc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)cc1	C36H38N6O11	HDAC1;HDAC2	Q13547/Q92769	VHL	WO-2021148811-A1
TPD-QLX77C	WO2021148811A1_PROTAC9	.	Nc1ccccc1NC(=O)c1ccc(NC(=O)COCCOCCNC(=O)COc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)cc1	C34H34N6O10	HDAC1;HDAC2	Q13547/Q92769	VHL	WO-2021148811-A1
TPD-6OEQQU	SCHEMBL23702571	(4S)-1-[4-[4-[3-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethoxy]propanoyl]piperazin-1-yl]phenyl]-7,8-dimethoxy-N,4-dimethyl-4,5-dihydro-2,3-benzodiazepine-3-carboxamide	CNC(=O)N1N=C(C2=CC=C(N3CCN(C(=O)CCOCCOCCOCCOCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)C=C2)C2=C(C=C(OC)C(OC)=C2)C[C@@H]1C	C48H60N8O12	BRD4	O60885	CRBN	WO-2021152113-A1
TPD-79ZJ5R	SCHEMBL23702528	(4S)-1-[4-[4-[3-[2-[2-[2-[2-[[2-[(3S)-2,6-dioxopiperidin-3-yl]-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethoxy]propanoyl]piperazin-1-yl]phenyl]-7,8-dimethoxy-N,4-dimethyl-4,5-dihydro-2,3-benzodiazepine-3-carboxamide	CNC(=O)N1N=C(C2=CC=C(N3CCN(C(=O)CCOCCOCCOCCOCCNC4=CC=CC5=C4C(=O)N([C@H]4CCC(=O)NC4=O)C5=O)CC3)C=C2)C2=C(C=C(OC)C(OC)=C2)C[C@@H]1C	C48H60N8O12	BRD4	O60885	CRBN	WO-2021152113-A1
TPD-MERCNF	CHEMBL5178566	(4S)-1-[4-[4-[3-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]propanoyl]piperazin-1-yl]phenyl]-7,8-dimethoxy-N,4-dimethyl-4,5-dihydro-2,3-benzodiazepine-3-carboxamide; SCHEMBL23702523; BDBM50590048	CNC(=O)N1N=C(C2=CC=C(N3CCN(C(=O)CCOCCOCCOCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)C=C2)C2=C(C=C(OC)C(OC)=C2)C[C@@H]1C	C46H56N8O11	BRD4	O60885	CRBN	WO-2021152113-A1
TPD-2Q9NZ5	SCHEMBL23702553	(4S)-1-[4-[4-[3-[2-[2-[2-[[2-[(3S)-2,6-dioxopiperidin-3-yl]-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]propanoyl]piperazin-1-yl]phenyl]-7,8-dimethoxy-N,4-dimethyl-4,5-dihydro-2,3-benzodiazepine-3-carboxamide	CNC(=O)N1N=C(C2=CC=C(N3CCN(C(=O)CCOCCOCCOCCNC4=CC=CC5=C4C(=O)N([C@H]4CCC(=O)NC4=O)C5=O)CC3)C=C2)C2=C(C=C(OC)C(OC)=C2)C[C@@H]1C	C46H56N8O11	BRD4	O60885	CRBN	WO-2021152113-A1
TPD-CEUNNZ	CHEMBL4858472	(4S)-1-[4-[4-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]-2-oxoethoxy]ethoxy]ethoxy]acetyl]piperazin-1-yl]phenyl]-7,8-dimethoxy-N,4-dimethyl-4,5-dihydro-2,3-benzodiazepine-3-carboxamide; SCHEMBL23702548; BDBM50573453	CNC(=O)N1N=C(C2=CC=C(N3CCN(C(=O)COCCOCCOCC(=O)NC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)C=C2)C2=C(C=C(OC)C(OC)=C2)C[C@@H]1C	C45H52N8O12	BRD4	O60885	CRBN	WO-2021152113-A1
TPD-TAGYBJ	Brd4-IN-2	BRD4-IN-2; CHEMBL4854720; 2679925-55-2; orb1690683; SCHEMBL23702543; BDBM50573454; AKOS040757961; DA-51381; HY-141843; CS-0254874; (4S)-1-[4-[4-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]-2-oxoethoxy]ethoxy]acetyl]piperazin-1-yl]phenyl]-7,8-dimethoxy-N,4-dimethyl-4,5-dihydro-2,3-benzodiazepine-3-carboxamide	CNC(=O)N1N=C(C2=CC=C(N3CCN(C(=O)COCCOCC(=O)NC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)C=C2)C2=C(C=C(OC)C(OC)=C2)C[C@@H]1C	C43H48N8O11	BRD4	O60885	CRBN	WO-2021152113-A1
TPD-K47317	CHEMBL4848064	(4S)-1-[4-[4-[5-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyacetyl]amino]pentanoyl]piperazin-1-yl]phenyl]-7,8-dimethoxy-N,4-dimethyl-4,5-dihydro-2,3-benzodiazepine-3-carboxamide; SCHEMBL23702555; BDBM50573455	CNC(=O)N1N=C(C2=CC=C(N3CCN(C(=O)CCCCNC(=O)COC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)C=C2)C2=C(C=C(OC)C(OC)=C2)C[C@@H]1C	C44H50N8O10	BRD4	O60885	CRBN	WO-2021152113-A1
TPD-VJEWOR	CHEMBL4851953	(4S)-1-[4-[4-[2-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]-2-oxoethoxy]ethoxy]ethoxy]ethoxy]acetyl]piperazin-1-yl]phenyl]-7,8-dimethoxy-N,4-dimethyl-4,5-dihydro-2,3-benzodiazepine-3-carboxamide; SCHEMBL23702540; BDBM50573456	CNC(=O)N1N=C(C2=CC=C(N3CCN(C(=O)COCCOCCOCCOCC(=O)NC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)C=C2)C2=C(C=C(OC)C(OC)=C2)C[C@@H]1C	C47H56N8O13	BRD4	O60885	CRBN	WO-2021152113-A1
TPD-JXMN28	SCHEMBL23702550	(4R)-1-[4-[4-[3-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethoxy]propanoyl]piperazin-1-yl]phenyl]-7,8-dimethoxy-N,4-dimethyl-4,5-dihydro-2,3-benzodiazepine-3-carboxamide	CNC(=O)N1N=C(C2=CC=C(N3CCN(C(=O)CCOCCOCCOCCOCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)C=C2)C2=C(C=C(OC)C(OC)=C2)C[C@H]1C	C48H60N8O12	BRD4	O60885	CRBN	WO-2021152113-A1
TPD-AMFFD0	SCHEMBL23702522	(4R)-1-[4-[4-[3-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]propanoyl]piperazin-1-yl]phenyl]-7,8-dimethoxy-N,4-dimethyl-4,5-dihydro-2,3-benzodiazepine-3-carboxamide	CNC(=O)N1N=C(C2=CC=C(N3CCN(C(=O)CCOCCOCCOCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)C=C2)C2=C(C=C(OC)C(OC)=C2)C[C@H]1C	C46H56N8O11	BRD4	O60885	CRBN	WO-2021152113-A1
TPD-MWVEWJ	SCHEMBL23702564	(4S)-1-[4-[2-[2-[2-[2-[[2-[(3S)-2,6-dioxopiperidin-3-yl]-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethylcarbamoyl]phenyl]-7,8-dimethoxy-N,4-dimethyl-4,5-dihydro-2,3-benzodiazepine-3-carboxamide	CNC(=O)N1N=C(C2=CC=C(C(=O)NCCOCCOCCOCCNC3=CC=CC4=C3C(=O)N([C@H]3CCC(=O)NC3=O)C4=O)C=C2)C2=C(C=C(OC)C(OC)=C2)C[C@@H]1C	C42H49N7O11	BRD4	O60885	CRBN	WO-2021152113-A1
TPD-MRP2GU	CHEMBL4864279	(4S)-1-[4-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyacetyl]amino]butylcarbamoyl]phenyl]-7,8-dimethoxy-N,4-dimethyl-4,5-dihydro-2,3-benzodiazepine-3-carboxamide; SCHEMBL23702537; BDBM50573457	CNC(=O)N1N=C(C2=CC=C(C(=O)NCCCCNC(=O)COC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)C=C2)C2=C(C=C(OC)C(OC)=C2)C[C@@H]1C	C40H43N7O10	BRD4	O60885	CRBN	WO-2021152113-A1
TPD-ZJ8VG3	SCHEMBL23702565	(4S)-1-[4-[2-[2-[2-[2-[2-[[2-[(3S)-2,6-dioxopiperidin-3-yl]-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethylcarbamoyl]phenyl]-7,8-dimethoxy-N,4-dimethyl-4,5-dihydro-2,3-benzodiazepine-3-carboxamide	CNC(=O)N1N=C(C2=CC=C(C(=O)NCCOCCOCCOCCOCCNC3=CC=CC4=C3C(=O)N([C@H]3CCC(=O)NC3=O)C4=O)C=C2)C2=C(C=C(OC)C(OC)=C2)C[C@@H]1C	C44H53N7O12	BRD4	O60885	CRBN	WO-2021152113-A1
TPD-SWF6CZ	CHEMBL4855093	(4S)-1-[4-[4-[3-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]amino]ethoxy]ethoxy]ethoxy]propanoyl]piperazin-1-yl]phenyl]-7,8-dimethoxy-N,4-dimethyl-4,5-dihydro-2,3-benzodiazepine-3-carboxamide; SCHEMBL23702566; BDBM50573458	CNC(=O)N1N=C(C2=CC=C(N3CCN(C(=O)CCOCCOCCOCCNC4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)C=C2)C2=C(C=C(OC)C(OC)=C2)C[C@@H]1C	C46H56N8O11	BRD4	O60885	CRBN	WO-2021152113-A1
TPD-17BBJ5	SCHEMBL23702542	(4S)-1-[4-[4-[3-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]amino]ethoxy]ethoxy]ethoxy]ethoxy]propanoyl]piperazin-1-yl]phenyl]-7,8-dimethoxy-N,4-dimethyl-4,5-dihydro-2,3-benzodiazepine-3-carboxamide	CNC(=O)N1N=C(C2=CC=C(N3CCN(C(=O)CCOCCOCCOCCOCCNC4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)C=C2)C2=C(C=C(OC)C(OC)=C2)C[C@@H]1C	C48H60N8O12	BRD4	O60885	CRBN	WO-2021152113-A1
TPD-FR2EPP	WO2021152113A1_16	.	CNC(=O)N1N=C(C2=CC=C(C(=O)NCCOCCOCCOCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCC3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)C=C2)C2=CC(OC)=C(OC)C=C2C[C@@H]1C	C51H66N8O11S	BRD4	O60885	CRBN	WO-2021152113-A1
TPD-KH6JND	WO2021152113A1_17	(4S)-1-[4-[2-[2-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]ethoxy]ethylcarbamoyl]phenyl]-7,8-dimethoxy-N,4-dimethyl-4,5-dihydro-2,3-benzodiazepine-3-carboxamide	CNC(=O)N1N=C(C2=CC=C(C(=O)NCCOCCOCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCC3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)C=C2)C2=CC(OC)=C(OC)C=C2C[C@@H]1C	C49H62N8O10S	BRD4	O60885	CRBN	WO-2021152113-A1
TPD-WWK6TZ	WO2021152113A1_18	.	CNC(=O)N1N=C(C2=CC=C(C(=O)NCCOCCOCCOCCOCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCC3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)C=C2)C2=CC(OC)=C(OC)C=C2C[C@@H]1C	C53H70N8O12S	BRD4	O60885	CRBN	WO-2021152113-A1
TPD-B3CAG0	SCHEMBL24950310	2-[4-[4-[[5-chloro-4-(2-propan-2-ylsulfonylanilino)pyrimidin-2-yl]amino]-2-methyl-5-propan-2-yloxyphenyl]piperidin-1-yl]-N-[[1-(2,6-dioxopiperidin-3-yl)benzo[e][1]benzofuran-7-yl]methyl]acetamide	CC1=C(C2CCN(CC(=O)NCC3=CC4=C(C=C3)C3=C(C=C4)OC=C3C3CCC(=O)NC3=O)CC2)C=C(OC(C)C)C(NC2=NC=C(Cl)C(NC3=CC=CC=C3S(=O)(=O)C(C)C)=N2)=C1	C48H52ClN7O7S	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-39NPVX	WO2021185291A1_WX003	.	CCS(=O)(=O)C1=CC=CC=C1NC1=NC(NC2=CC(C)=C(C3CCN(C(=O)COC4=CC=C5OC=C(C6CCC(=O)NC6=O)C5=C4)CC3)C=C2OC(C)C)=NC=C1Cl	C42H45ClN6O8S	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-FSINIM	SCHEMBL24950412	2-[4-(4-amino-2-methyl-5-propan-2-yloxyphenyl)piperidin-1-yl]-N-[2-[[3-(2,6-dioxopiperidin-3-yl)-1-benzofuran-5-yl]oxy]ethyl]acetamide	CC1=C(C2CCN(CC(=O)NCCOC3=CC=C4OC=C(C5CCC(=O)NC5=O)C4=C3)CC2)C=C(OC(C)C)C(N)=C1	C32H40N4O6	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-XR3W27	SCHEMBL26161768	2-[4-[4-[(4-amino-5-chloropyrimidin-2-yl)amino]-2-methyl-5-propan-2-yloxyphenyl]piperidin-1-yl]-N-[2-[[3-(2,6-dioxopiperidin-3-yl)-1-benzofuran-5-yl]oxy]ethyl]acetamide	CC1=C(C2CCN(CC(=O)NCCOC3=CC=C4OC=C(C5CCC(=O)NC5=O)C4=C3)CC2)C=C(OC(C)C)C(NC2=NC=C(Cl)C(N)=N2)=C1	C36H42ClN7O6	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-9EAFH4	SCHEMBL24949407	3-[5-[2-[4-[4-[[5-Chloro-4-(2-propan-2-ylsulfonylanilino)pyrimidin-2-yl]amino]-2-methyl-5-propan-2-yloxyphenyl]piperidin-1-yl]ethoxy]-1-benzofuran-3-yl]piperidine-2,6-dione	CC1=C(C2CCN(CCOC3=CC=C4OC=C(C5CCC(=O)NC5=O)C4=C3)CC2)C=C(OC(C)C)C(NC2=NC=C(Cl)C(NC3=CC=CC=C3S(=O)(=O)C(C)C)=N2)=C1	C43H49ClN6O7S	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-XWAJII	SCHEMBL24950272	2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]-N-[2-[1-(2,6-dioxopiperidin-3-yl)benzo[e][1]benzofuran-7-yl]oxyethyl]acetamide	CC1=NN=C2[C@H](CC(=O)NCCOC3=CC=C4C(=C3)C=CC3=C4C(C4CCC(=O)NC4=O)=CO3)N=C(C3=CC=C(Cl)C=C3)C3=C(SC(C)=C3C)N12	C38H33ClN6O5S	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-TSY1BY	SCHEMBL24949408	2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]-N-[2-[2-[2-[1-(2,6-dioxopiperidin-3-yl)benzo[e][1]benzofuran-7-yl]oxyethoxy]ethoxy]ethyl]acetamide	CC1=NN=C2[C@H](CC(=O)NCCOCCOCCOC3=CC=C4C(=C3)C=CC3=C4C(C4CCC(=O)NC4=O)=CO3)N=C(C3=CC=C(Cl)C=C3)C3=C(SC(C)=C3C)N12	C42H41ClN6O7S	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-S2RV6J	SCHEMBL24950383	2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]-N-[6-[[1-(2,6-dioxopiperidin-3-yl)benzo[e][1]benzofuran-7-yl]amino]hexyl]acetamide	CC1=NN=C2[C@H](CC(=O)NCCCCCCNC3=CC=C4C(=C3)C=CC3=C4C(C4CCC(=O)NC4=O)=CO3)N=C(C3=CC=C(Cl)C=C3)C3=C(SC(C)=C3C)N12	C42H42ClN7O4S	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-ETU6TA	SCHEMBL24949431	2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]-N-[2-[[1-(2,6-dioxopiperidin-3-yl)benzo[e][1]benzofuran-7-yl]amino]ethyl]acetamide	CC1=NN=C2[C@H](CC(=O)NCCNC3=CC=C4C(=C3)C=CC3=C4C(C4CCC(=O)NC4=O)=CO3)N=C(C3=CC=C(Cl)C=C3)C3=C(SC(C)=C3C)N12	C38H34ClN7O4S	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-WN5OX3	SCHEMBL24950241	2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]-N-[2-[2-[1-(2,6-dioxopiperidin-3-yl)benzo[e][1]benzofuran-7-yl]oxyethoxy]ethyl]acetamide	CC1=NN=C2[C@H](CC(=O)NCCOCCOC3=CC4=C(C=C3)C3=C(C=C4)OC=C3C3CCC(=O)NC3=O)N=C(C3=CC=C(Cl)C=C3)C3=C(SC(C)=C3C)N12	C40H37ClN6O6S	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-NZDE8H	SCHEMBL24950344	2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]-N-[6-[1-(2,6-dioxopiperidin-3-yl)benzo[e][1]benzofuran-7-yl]oxyhexyl]acetamide	CC1=NN=C2[C@H](CC(=O)NCCCCCCOC3=CC=C4C(=C3)C=CC3=C4C(C4CCC(=O)NC4=O)=CO3)N=C(C3=CC=C(Cl)C=C3)C3=C(SC(C)=C3C)N12	C42H41ClN6O5S	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-9G50WG	SCHEMBL24950195	N-[4-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]butyl]-2-[1-(2,6-dioxopiperidin-3-yl)benzo[e][1]benzofuran-7-yl]oxyacetamide	CC(=O)C1=C(C)C2=C(N=C(NC3=CC=C(N4CCN(CCCCNC(=O)COC5=CC6=C(C=C5)C5=C(C=C6)OC=C5C5CCC(=O)NC5=O)CC4)C=N3)N=C2)N(C2CCCC2)C1=O	C47H51N9O7	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-J1PS6I	SCHEMBL24949426	5-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]-N-[2-[[1-(2,6-dioxopiperidin-3-yl)benzo[e][1]benzofuran-7-yl]amino]ethyl]pentanamide	CC(=O)C1=C(C)C2=C(N=C(NC3=CC=C(N4CCN(CCCCC(=O)NCCNC5=CC=C6C(=C5)C=CC5=C6C(C6CCC(=O)NC6=O)=CO5)CC4)C=N3)N=C2)N(C2CCCC2)C1=O	C48H54N10O6	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-QWH716	SCHEMBL26161784	2-[4-[(3S)-1-[6-[[2-[1-(2,6-dioxopiperidin-3-yl)benzo[e][1]benzofuran-7-yl]oxyacetyl]amino]hexyl]piperidin-3-yl]phenyl]indazole-7-carboxamide	NC(=O)C1=CC=CC2=CN(C3=CC=C([C@@H]4CCCN(CCCCCCNC(=O)COC5=CC6=CC=C7OC=C(C8CCC(=O)NC8=O)C7=C6C=C5)C4)C=C3)N=C21	C44H46N6O6	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-B5DMP0	SCHEMBL26158952	2-[4-[(3S)-1-[3-[[2-[1-(2,6-dioxopiperidin-3-yl)benzo[e][1]benzofuran-7-yl]oxyacetyl]amino]propyl]piperidin-3-yl]phenyl]indazole-7-carboxamide	NC(=O)C1=CC=CC2=CN(C3=CC=C([C@@H]4CCCN(CCCNC(=O)COC5=CC6=CC=C7OC=C(C8CCC(=O)NC8=O)C7=C6C=C5)C4)C=C3)N=C21	C41H40N6O6	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-Q7V4ZJ	SCHEMBL24950233	5-[4-(3-chloro-4-fluoroanilino)-7-methoxyquinazolin-6-yl]oxy-N-[2-[1-(2,6-dioxopiperidin-3-yl)benzo[e][1]benzofuran-7-yl]oxyethyl]pentanamide	COC1=CC2=C(C=C1OCCCCC(=O)NCCOC1=CC3=C(C=C1)C1=C(C=C3)OC=C1C1CCC(=O)NC1=O)C(NC1=CC(Cl)=C(F)C=C1)=NC=N2	C39H35ClFN5O7	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-JT9TT0	SCHEMBL26161793	N-[2-[1-(2,6-dioxopiperidin-3-yl)benzo[e][1]benzofuran-7-yl]oxyethyl]-N-methyl-2-[6-[6-(trifluoromethoxy)-1H-benzimidazol-2-yl]pyridin-3-yl]oxyacetamide	CN(CCOC1=CC=C2C(=C1)C=CC1=C2C(C2CCC(=O)NC2=O)=CO1)C(=O)COC1=CN=C(C2=NC3=CC(OC(F)(F)F)=CC=C3N2)C=C1	C35H28F3N5O7	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-0DU19B	SCHEMBL26161794	N-[2-[2-[1-(2,6-dioxopiperidin-3-yl)benzo[e][1]benzofuran-7-yl]oxyethoxy]ethyl]-2-[6-[6-(trifluoromethoxy)-1H-benzimidazol-2-yl]pyridin-3-yl]oxyacetamide	O=C(COC1=CN=C(C2=NC3=CC(OC(F)(F)F)=CC=C3N2)C=C1)NCCOCCOC1=CC=C2C(=C1)C=CC1=C2C(C2CCC(=O)NC2=O)=CO1	C36H30F3N5O8	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-1MBQPD	SCHEMBL26161795	3-[(1S,3R)-3-(4-chlorophenyl)sulfonyl-3-(2,5-difluorophenyl)cyclohexyl]-N-[2-[2-[2-[1-(2,6-dioxopiperidin-3-yl)benzo[e][1]benzofuran-7-yl]oxyethoxy]ethoxy]ethyl]propanamide	O=C(CC[C@@H]1CCC[C@@](C2=C(F)C=CC(F)=C2)(S(=O)(=O)C2=CC=C(Cl)C=C2)C1)NCCOCCOCCOC1=CC=C2C(=C1)C=CC1=C2C(C2CCC(=O)NC2=O)=CO1	C44H45ClF2N2O9S	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-BY4DPG	SCHEMBL26161796	3-[(1S,3R)-3-(4-chlorophenyl)sulfonyl-3-(2,5-difluorophenyl)cyclohexyl]-N-[2-[2-[1-(2,6-dioxopiperidin-3-yl)benzo[e][1]benzofuran-7-yl]oxyethoxy]ethyl]propanamide	O=C(CC[C@@H]1CCC[C@@](C2=C(F)C=CC(F)=C2)(S(=O)(=O)C2=CC=C(Cl)C=C2)C1)NCCOCCOC1=CC=C2C(=C1)C=CC1=C2C(C2CCC(=O)NC2=O)=CO1	C42H41ClF2N2O8S	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-MMH0UB	SCHEMBL24949125	3-[7-[3-[4-[4-[[1-[6-(2-Hydroxypropan-2-yl)pyridin-2-yl]-3-oxo-2-prop-2-enylpyrazolo[3,4-d]pyrimidin-6-yl]amino]phenyl]piperazin-1-yl]propylamino]benzo[e][1]benzofuran-1-yl]piperidine-2,6-dione	C=CCN1C(=O)C2=CN=C(NC3=CC=C(N4CCN(CCCNC5=CC6=CC=C7OC=C(C8CCC(=O)NC8=O)C7=C6C=C5)CC4)C=C3)N=C2N1C1=NC(C(C)(C)O)=CC=C1	C46H48N10O5	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-W7DGBU	SCHEMBL24949144	3-[7-[2-[4-[4-[[1-[6-(2-Hydroxypropan-2-yl)pyridin-2-yl]-3-oxo-2-prop-2-enylpyrazolo[3,4-d]pyrimidin-6-yl]amino]phenyl]piperazin-1-yl]-2-oxoethoxy]benzo[e][1]benzofuran-1-yl]piperidine-2,6-dione	C=CCN1C(=O)C2=CN=C(NC3=CC=C(N4CCN(C(=O)COC5=CC6=C(C=C5)C5=C(C=C6)OC=C5C5CCC(=O)NC5=O)CC4)C=C3)N=C2N1C1=NC(C(C)(C)O)=CC=C1	C45H43N9O7	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-RYOPOU	SCHEMBL24950348	2-[1-(2,6-dioxopiperidin-3-yl)benzo[e][1]benzofuran-7-yl]oxy-N-[3-[4-[4-[[1-[6-(2-hydroxypropan-2-yl)pyridin-2-yl]-3-oxo-2-prop-2-enylpyrazolo[3,4-d]pyrimidin-6-yl]amino]phenyl]piperazin-1-yl]propyl]acetamide	C=CCN1C(=O)C2=CN=C(NC3=CC=C(N4CCN(CCCNC(=O)COC5=CC6=C(C=C5)C5=C(C=C6)OC=C5C5CCC(=O)NC5=O)CC4)C=C3)N=C2N1C1=NC(C(C)(C)O)=CC=C1	C48H50N10O7	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-YTO6Y4	SCHEMBL24949480	3-[7-[[3-[4-[4-[[1-[6-(2-Hydroxypropan-2-yl)pyridin-2-yl]-3-oxo-2-prop-2-enylpyrazolo[3,4-d]pyrimidin-6-yl]amino]phenyl]piperazin-1-yl]-3-oxopropyl]amino]benzo[e][1]benzofuran-1-yl]piperidine-2,6-dione	C=CCN1C(=O)C2=CN=C(NC3=CC=C(N4CCN(C(=O)CCNC5=CC6=C(C=C5)C5=C(C=C6)OC=C5C5CCC(=O)NC5=O)CC4)C=C3)N=C2N1C1=NC(C(C)(C)O)=CC=C1	C46H46N10O6	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-9L81AC	SCHEMBL24950277	3-[[1-(2,6-dioxopiperidin-3-yl)benzo[e][1]benzofuran-7-yl]amino]-N-[3-[4-[4-[[1-[6-(2-hydroxypropan-2-yl)pyridin-2-yl]-3-oxo-2-prop-2-enylpyrazolo[3,4-d]pyrimidin-6-yl]amino]phenyl]piperazin-1-yl]propyl]propanamide	C=CCN1C(=O)C2=CN=C(NC3=CC=C(N4CCN(CCCNC(=O)CCNC5=CC6=C(C=C5)C5=C(C=C6)OC=C5C5CCC(=O)NC5=O)CC4)C=C3)N=C2N1C1=NC(C(C)(C)O)=CC=C1	C49H53N11O6	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-J3EK1D	SCHEMBL24949489	6-(4-bromo-2-fluoroanilino)-N-[2-[2-[2-[1-(2,6-dioxopiperidin-3-yl)benzo[e][1]benzofuran-7-yl]oxyethoxy]ethoxy]ethyl]-7-fluoro-3-methylbenzimidazole-5-carboxamide	CN1C=NC2=C1C=C(C(=O)NCCOCCOCCOC1=CC3=C(C=C1)C1=C(C=C3)OC=C1C1CCC(=O)NC1=O)C(NC1=CC=C(Br)C=C1F)=C2F	C38H34BrF2N5O7	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-Z1RUU6	SCHEMBL24949487	6-(4-bromo-2-fluoroanilino)-N-[6-[[1-(2,6-dioxopiperidin-3-yl)benzo[e][1]benzofuran-7-yl]amino]hexyl]-7-fluoro-3-methylbenzimidazole-5-carboxamide	CN1C=NC2=C1C=C(C(=O)NCCCCCCNC1=CC=C3C(=C1)C=CC1=C3C(C3CCC(=O)NC3=O)=CO1)C(NC1=CC=C(Br)C=C1F)=C2F	C38H35BrF2N6O4	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-THU6F5	SCHEMBL24950244	6-(4-bromo-2-fluoroanilino)-N-[2-[[1-(2,6-dioxopiperidin-3-yl)benzo[e][1]benzofuran-7-yl]amino]ethyl]-7-fluoro-3-methylbenzimidazole-5-carboxamide	CN1C=NC2=C1C=C(C(=O)NCCNC1=CC=C3C(=C1)C=CC1=C3C(C3CCC(=O)NC3=O)=CO1)C(NC1=CC=C(Br)C=C1F)=C2F	C34H27BrF2N6O4	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-1VCTTY	SCHEMBL24949448	6-(4-bromo-2-fluoroanilino)-N-[2-[2-[1-(2,6-dioxopiperidin-3-yl)benzo[e][1]benzofuran-7-yl]oxyethoxy]ethyl]-7-fluoro-3-methylbenzimidazole-5-carboxamide	CN1C=NC2=C1C=C(C(=O)NCCOCCOC1=CC=C3C(=C1)C=CC1=C3C(C3CCC(=O)NC3=O)=CO1)C(NC1=CC=C(Br)C=C1F)=C2F	C36H30BrF2N5O6	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-6L7VFO	SCHEMBL24950247	6-(4-bromo-2-fluoroanilino)-N-[6-[1-(2,6-dioxopiperidin-3-yl)benzo[e][1]benzofuran-7-yl]oxyhexyl]-7-fluoro-3-methylbenzimidazole-5-carboxamide	CN1C=NC2=C1C=C(C(=O)NCCCCCCOC1=CC=C3C(=C1)C=CC1=C3C(C3CCC(=O)NC3=O)=CO1)C(NC1=CC=C(Br)C=C1F)=C2F	C38H34BrF2N5O5	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-24F5D4	WO2021185291A1_WX032	.	CC1=NC(NC2=NC=C(C(=O)NC3=C(C)C=CC=C3CI)S2)=CC(N2CCN(CCCCCC(=O)NCC3=CC4=C(C=C3)C3=C(C=C4)OC=C3C3CCC(=O)NC3=O)CC2)=N1	C45H48IN9O5S	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-XL1BGC	SCHEMBL24949600	N-(2-chloro-6-methylphenyl)-2-[[6-[4-[6-[6-[[1-(2,6-dioxopiperidin-3-yl)benzo[e][1]benzofuran-7-yl]amino]hexylamino]-6-oxohexyl]piperazin-1-yl]-2-methylpyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide	CC1=NC(NC2=NC=C(C(=O)NC3=C(C)C=CC=C3Cl)S2)=CC(N2CCN(CCCCCC(=O)NCCCCCCNC3=CC4=C(C=C3)C3=C(C=C4)OC=C3C3CCC(=O)NC3=O)CC2)=N1	C49H57ClN10O5S	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-DQ6V3D	SCHEMBL24950374	N-(2-chloro-6-methylphenyl)-2-[[6-[4-[6-[2-[2-[2-[1-(2,6-dioxopiperidin-3-yl)benzo[e][1]benzofuran-7-yl]oxyethoxy]ethoxy]ethylamino]-6-oxohexyl]piperazin-1-yl]-2-methylpyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide	CC1=NC(NC2=NC=C(C(=O)NC3=C(C)C=CC=C3Cl)S2)=CC(N2CCN(CCCCCC(=O)NCCOCCOCCOC3=CC4=C(C=C3)C3=C(C=C4)OC=C3C3CCC(=O)NC3=O)CC2)=N1	C49H56ClN9O8S	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-RL1I39	SCHEMBL24950238	N-(2-chloro-6-methylphenyl)-2-[[6-[4-[6-[2-[[1-(2,6-dioxopiperidin-3-yl)benzo[e][1]benzofuran-7-yl]amino]ethylamino]-6-oxohexyl]piperazin-1-yl]-2-methylpyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide	CC1=NC(NC2=NC=C(C(=O)NC3=C(C)C=CC=C3Cl)S2)=CC(N2CCN(CCCCCC(=O)NCCNC3=CC4=C(C=C3)C3=C(C=C4)OC=C3C3CCC(=O)NC3=O)CC2)=N1	C45H49ClN10O5S	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-Z5XA46	SCHEMBL24950232	4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]-N-[2-[[3-(2,6-dioxopiperidin-3-yl)-1-benzofuran-5-yl]oxy]ethyl]-2-fluorobenzamide	CC1(C)C(=O)N(C2=CC(C(F)(F)F)=C(C#N)C=C2)C(=S)N1C1=CC(F)=C(C(=O)NCCOC2=CC=C3OC=C(C4CCC(=O)NC4=O)C3=C2)C=C1	C35H27F4N5O6S	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-58YWEQ	SCHEMBL24950230	4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]-N-[4-[[3-(2,6-dioxopiperidin-3-yl)-1-benzofuran-5-yl]oxy]butyl]-2-fluorobenzamide	CC1(C)C(=O)N(C2=CC(C(F)(F)F)=C(C#N)C=C2)C(=S)N1C1=CC(F)=C(C(=O)NCCCCOC2=CC=C3OC=C(C4CCC(=O)NC4=O)C3=C2)C=C1	C37H31F4N5O6S	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-T8ES8Y	SCHEMBL24950338	4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]-N-[2-[2-[2-[[3-(2,6-dioxopiperidin-3-yl)-1-benzofuran-5-yl]oxy]ethoxy]ethoxy]ethyl]-2-fluorobenzamide	CC1(C)C(=O)N(C2=CC(C(F)(F)F)=C(C#N)C=C2)C(=S)N1C1=CC(F)=C(C(=O)NCCOCCOCCOC2=CC=C3OC=C(C4CCC(=O)NC4=O)C3=C2)C=C1	C39H35F4N5O8S	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-7G3NEI	SCHEMBL24949491	4-[3-[4-[2-[[3-(2,6-Dioxopiperidin-3-yl)-1-benzofuran-5-yl]oxy]ethoxy]-3-fluorophenyl]-4,4-dimethyl-5-oxo-2-sulfanylideneimidazolidin-1-yl]-2-(trifluoromethyl)benzonitrile	CC1(C)C(=O)N(C2=CC(C(F)(F)F)=C(C#N)C=C2)C(=S)N1C1=CC(F)=C(OCCOC2=CC=C3OC=C(C4CCC(=O)NC4=O)C3=C2)C=C1	C34H26F4N4O6S	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-OQZA8D	SCHEMBL24949443	2-[4-[2-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]-2-fluorophenoxy]ethyl]phenyl]-N-[3-(2,6-dioxopiperidin-3-yl)-1,2-benzoxazol-5-yl]acetamide	CC1(C)C(=O)N(C2=CC(C(F)(F)F)=C(C#N)C=C2)C(=S)N1C1=CC=C(OCCC2=CC=C(CC(=O)NC3=CC=C4ON=C(C5CCC(=O)NC5=O)C4=C3)C=C2)C(F)=C1	C41H32F4N6O6S	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-N4D773	SCHEMBL24949193	3-[5-[[1-[6-(2-Hydroxypropan-2-yl)pyridin-2-yl]-3-oxo-2-prop-2-enylpyrazolo[3,4-d]pyrimidin-6-yl]amino]-1-benzofuran-3-yl]piperidine-2,6-dione	C=CCN1C(=O)C2=CN=C(NC3=CC=C4OC=C(C5CCC(=O)NC5=O)C4=C3)N=C2N1C1=NC(C(C)(C)O)=CC=C1	C29H27N7O5	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-JEAEYC	WO2021185291A1_WX042	.	CC1=NNC2[C@H](CC(=O)NCCCNC(=O)COC3=CC=C4OC=C(C5CCC(=O)NC5=O)C4=C3)N=C(C3=CC=C(Cl)C=C3)C3=C(SC(C)=C3C)N12	C37H38ClN7O6S	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-7IE1K5	SCHEMBL24948998	3-[5-[2-[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]ethylamino]ethoxy]-1-benzofuran-3-yl]piperidine-2,6-dione	CC1=NN=C2[C@H](CCNCCOC3=CC4=C(C=C3)OC=C4C3CCC(=O)NC3=O)N=C(C3=CC=C(Cl)C=C3)C3=C(SC(C)=C3C)N12	C34H33ClN6O4S	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-M0OTX5	SCHEMBL24948996	3-[5-[2-[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]ethyl-methylamino]ethoxy]-1-benzofuran-3-yl]piperidine-2,6-dione	CC1=NN=C2[C@H](CCN(C)CCOC3=CC4=C(C=C3)OC=C4C3CCC(=O)NC3=O)N=C(C3=CC=C(Cl)C=C3)C3=C(SC(C)=C3C)N12	C35H35ClN6O4S	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-JBUOBZ	SCHEMBL24948900	3-[5-[3-[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]ethyl-methylamino]propyl]-1-benzofuran-3-yl]piperidine-2,6-dione	CC1=NN=C2[C@H](CCN(C)CCCC3=CC4=C(C=C3)OC=C4C3CCC(=O)NC3=O)N=C(C3=CC=C(Cl)C=C3)C3=C(SC(C)=C3C)N12	C36H37ClN6O3S	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-99IZGE	SCHEMBL24948899	CID 168752646	O=C1CCC(C2=COC3=C2C2=CC=C(OCCCCCCNC(=O)C4=CC=C(NC(=O)[C@@H]5NC6(CCCCC6)[C@@]6(C(=O)NC7=C6C=CC(Cl)=C7)[C@H]5C5=CC=CC(Cl)=C5F)C=C4)C=C2C=C3)C(=O)N1	C53H50Cl2FN5O7	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-LSZEPE	WO2021185291A1_WX047	.	O=C1CCC(C2=COC3=C2C2=CC=C(OCCOCCNC(=O)C4=CC=C(NC(=O)C5NC6(CCCCC6)[C@@]6(C(=O)NC7=C6C=CC(Cl)=C7)[C@H]5C5=CC=CC(Cl)=C5F)C=C4)C=C2C=C3)C(=O)N1	C51H46Cl2FN5O8	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-6BUPOA	SCHEMBL24950363	4-[4-[[4-chloro-3-(trifluoromethyl)phenyl]carbamoylamino]phenoxy]-N-[3-[[3-(2,6-dioxopiperidin-3-yl)-1-benzofuran-5-yl]oxy]propyl]pyridine-2-carboxamide	O=C1CCC(C2=COC3=C2C=C(OCCCNC(=O)C2=CC(OC4=CC=C(NC(=O)NC5=CC(C(F)(F)F)=C(Cl)C=C5)C=C4)=CC=N2)C=C3)C(=O)N1	C36H29ClF3N5O7	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-WYMNZH	SCHEMBL24950325	4-[4-[[4-chloro-3-(trifluoromethyl)phenyl]carbamoylamino]phenoxy]-N-[6-[[3-(2,6-dioxopiperidin-3-yl)-1-benzofuran-5-yl]oxy]hexyl]pyridine-2-carboxamide	O=C1CCC(C2=COC3=C2C=C(OCCCCCCNC(=O)C2=CC(OC4=CC=C(NC(=O)NC5=CC(C(F)(F)F)=C(Cl)C=C5)C=C4)=CC=N2)C=C3)C(=O)N1	C39H35ClF3N5O7	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-4QMIBS	SCHEMBL24950229	4-[4-[[4-chloro-3-(trifluoromethyl)phenyl]carbamoylamino]phenoxy]-N-[2-[2-[[3-(2,6-dioxopiperidin-3-yl)-1-benzofuran-5-yl]oxy]ethoxy]ethyl]pyridine-2-carboxamide	O=C1CCC(C2=COC3=C2C=C(OCCOCCNC(=O)C2=CC(OC4=CC=C(NC(=O)NC5=CC(C(F)(F)F)=C(Cl)C=C5)C=C4)=CC=N2)C=C3)C(=O)N1	C37H31ClF3N5O8	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-9ST7C1	SCHEMBL24950264	4-[4-[[4-chloro-3-(trifluoromethyl)phenyl]carbamoylamino]phenoxy]-N-[2-[[3-(2,6-dioxopiperidin-3-yl)-1-benzofuran-5-yl]oxy]ethyl]pyridine-2-carboxamide	O=C1CCC(C2=COC3=C2C=C(OCCNC(=O)C2=CC(OC4=CC=C(NC(=O)NC5=CC(C(F)(F)F)=C(Cl)C=C5)C=C4)=CC=N2)C=C3)C(=O)N1	C35H27ClF3N5O7	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-BZWXBO	SCHEMBL26161880	4-[3-[4-[[1-[4-[2-[[3-(2,6-Dioxopiperidin-3-yl)-1-benzofuran-5-yl]oxy]ethyl]piperazin-1-yl]cyclopropyl]methoxy]-3-fluorophenyl]-4,4-dimethyl-5-oxo-2-sulfanylideneimidazolidin-1-yl]-2-(trifluoromethyl)benzonitrile	CC1(C)C(=O)N(C2=CC(C(F)(F)F)=C(C#N)C=C2)C(=S)N1C1=CC=C(OCC2(N3CCN(CCOC4=CC5=C(C=C4)OC=C5C4CCC(=O)NC4=O)CC3)CC2)C(F)=C1	C42H40F4N6O6S	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-FUNEF6	SCHEMBL24950240	4-[3-[4-[[1-[4-[2-[[3-(2,6-Dioxopiperidin-3-yl)-1-benzofuran-6-yl]oxy]ethyl]piperazin-1-yl]cyclopropyl]methoxy]-3-fluorophenyl]-4,4-dimethyl-5-oxo-2-sulfanylideneimidazolidin-1-yl]-2-(trifluoromethyl)benzonitrile	CC1(C)C(=O)N(C2=CC(C(F)(F)F)=C(C#N)C=C2)C(=S)N1C1=CC(F)=C(OCC2(N3CCN(CCOC4=CC5=C(C=C4)C(C4CCC(=O)NC4=O)=CO5)CC3)CC2)C=C1	C42H40F4N6O6S	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-CDRBY1	SCHEMBL24950417	2-[4-[1-[[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]-2-fluorophenoxy]methyl]cyclopropyl]piperazin-1-yl]-N-[3-(2,6-dioxopiperidin-3-yl)-1-benzofuran-6-yl]acetamide	CC1(C)C(=O)N(C2=CC(C(F)(F)F)=C(C#N)C=C2)C(=S)N1C1=CC(F)=C(OCC2(N3CCN(CC(=O)NC4=CC5=C(C=C4)C(C4CCC(=O)NC4=O)=CO5)CC3)CC2)C=C1	C42H39F4N7O6S	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-071AEH	SCHEMBL24950380	N-[3-(2,6-dioxopiperidin-3-yl)-1-benzofuran-5-yl]-2-[2-[2-[2-[4-[[5-hydroxy-2-(4-hydroxyphenyl)-3-methylindol-1-yl]methyl]phenoxy]ethoxy]ethoxy]ethoxy]acetamide	CC1=C(C2=CC=C(O)C=C2)N(CC2=CC=C(OCCOCCOCCOCC(=O)NC3=CC=C4OC=C(C5CCC(=O)NC5=O)C4=C3)C=C2)C2=C1C=C(O)C=C2	C43H43N3O10	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-AF4ZVZ	SCHEMBL24950215	3-[5-[3-[4-[2-[4-[[5-Hydroxy-2-(4-hydroxyphenyl)-3-methylindol-1-yl]methyl]phenoxy]ethyl]piperazin-1-yl]propyl]-1-benzofuran-3-yl]piperidine-2,6-dione	CC1=C(C2=CC=C(O)C=C2)N(CC2=CC=C(OCCN3CCN(CCCC4=CC=C5OC=C(C6CCC(=O)NC6=O)C5=C4)CC3)C=C2)C2=C1C=C(O)C=C2	C44H46N4O6	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-FH0WWR	SCHEMBL24950542	3-[5-[4-[5-[4-[[5-Hydroxy-2-(4-hydroxyphenyl)-3-methylindol-1-yl]methyl]phenoxy]pentyl]piperazin-1-yl]-1-benzofuran-3-yl]piperidine-2,6-dione	CC1=C(C2=CC=C(O)C=C2)N(CC2=CC=C(OCCCCCN3CCN(C4=CC=C5OC=C(C6CCC(=O)NC6=O)C5=C4)CC3)C=C2)C2=C1C=C(O)C=C2	C44H46N4O6	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-CBGL5S	SCHEMBL26161896	2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]-N-[3-[[3-(2,6-dioxopiperidin-3-yl)-1-benzofuran-5-yl]oxy]propyl]acetamide	CC1=NN=C2[C@H](CC(=O)NCCCOC3=CC=C4OC=C(C5CCC(=O)NC5=O)C4=C3)N=C(C3=CC=C(Cl)C=C3)C3=C(SC(C)=C3C)N12	C35H33ClN6O5S	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-SWGXE9	SCHEMBL24950304	2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]-N-[2-[[3-(2,6-dioxopiperidin-3-yl)-1-benzofuran-5-yl]oxy]ethyl]acetamide	CC1=NN=C2[C@H](CC(=O)NCCOC3=CC=C4OC=C(C5CCC(=O)NC5=O)C4=C3)N=C(C3=CC=C(Cl)C=C3)C3=C(SC(C)=C3C)N12	C34H31ClN6O5S	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-5JP3A6	SCHEMBL24950399	2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]-N-[4-[[3-(2,6-dioxopiperidin-3-yl)-1-benzofuran-5-yl]oxy]butyl]acetamide	CC1=NN=C2[C@H](CC(=O)NCCCCOC3=CC=C4OC=C(C5CCC(=O)NC5=O)C4=C3)N=C(C3=CC=C(Cl)C=C3)C3=C(SC(C)=C3C)N12	C36H35ClN6O5S	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-5NVRKN	SCHEMBL24950398	2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]-N-[4-[[2-[[3-(2,6-dioxopiperidin-3-yl)-1-benzofuran-5-yl]oxy]acetyl]amino]butyl]acetamide	CC1=NN=C2[C@H](CC(=O)NCCCCNC(=O)COC3=CC=C4OC=C(C5CCC(=O)NC5=O)C4=C3)N=C(C3=CC=C(Cl)C=C3)C3=C(SC(C)=C3C)N12	C38H38ClN7O6S	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-BIDAYT	SCHEMBL26158964	2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]-N-[2-[2-[2-[[3-(2,6-dioxopiperidin-3-yl)-1-benzofuran-5-yl]oxy]ethoxy]ethoxy]ethyl]acetamide	CC1=NN=C2[C@H](CC(=O)NCCOCCOCCOC3=CC=C4OC=C(C5CCC(=O)NC5=O)C4=C3)N=C(C3=CC=C(Cl)C=C3)C3=C(SC(C)=C3C)N12	C38H39ClN6O7S	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-6DVWPU	SCHEMBL26159098	4-[[[4-[(4-chlorophenyl)methyl-cyclopentylsulfamoyl]phenyl]sulfonyl-(piperidin-4-ylmethyl)amino]methyl]-N-[2-[2-[2-[[3-(2,6-dioxopiperidin-3-yl)-1-benzofuran-5-yl]oxy]ethoxy]ethoxy]ethyl]benzamide	O=C1CCC(C2=COC3=CC=C(OCCOCCOCCNC(=O)C4=CC=C(CN(CC5CCNCC5)S(=O)(=O)C5=CC=C(S(=O)(=O)N(CC6=CC=C(Cl)C=C6)C6CCCC6)C=C5)C=C4)C=C32)C(=O)N1	C51H60ClN5O11S2	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-O912J1	SCHEMBL24950409	4-[[[4-[(4-chlorophenyl)methyl-cyclopentylsulfamoyl]phenyl]sulfonyl-(piperidin-4-ylmethyl)amino]methyl]-N-[2-[2-[[3-(2,6-dioxopiperidin-3-yl)-1-benzofuran-5-yl]oxy]ethoxy]ethyl]benzamide	O=C1CCC(C2=COC3=CC=C(OCCOCCNC(=O)C4=CC=C(CN(CC5CCNCC5)S(=O)(=O)C5=CC=C(S(=O)(=O)N(CC6=CC=C(Cl)C=C6)C6CCCC6)C=C5)C=C4)C=C32)C(=O)N1	C49H56ClN5O10S2	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-UEDRDW	SCHEMBL24950371	4-[[[4-[(4-chlorophenyl)methyl-cyclopentylsulfamoyl]phenyl]sulfonyl-(piperidin-4-ylmethyl)amino]methyl]-N-[3-[[3-(2,6-dioxopiperidin-3-yl)-1-benzofuran-5-yl]oxy]propyl]benzamide	O=C1CCC(C2=COC3=CC=C(OCCCNC(=O)C4=CC=C(CN(CC5CCNCC5)S(=O)(=O)C5=CC=C(S(=O)(=O)N(CC6=CC=C(Cl)C=C6)C6CCCC6)C=C5)C=C4)C=C32)C(=O)N1	C48H54ClN5O9S2	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-86IG2B	SCHEMBL26158966	4-[[[4-[(4-chlorophenyl)methyl-cyclopentylsulfamoyl]phenyl]sulfonyl-(piperidin-4-ylmethyl)amino]methyl]-N-[4-[[3-(2,6-dioxopiperidin-3-yl)-1-benzofuran-5-yl]oxy]butyl]benzamide	O=C1CCC(C2=COC3=CC=C(OCCCCNC(=O)C4=CC=C(CN(CC5CCNCC5)S(=O)(=O)C5=CC=C(S(=O)(=O)N(CC6=CC=C(Cl)C=C6)C6CCCC6)C=C5)C=C4)C=C32)C(=O)N1	C49H56ClN5O9S2	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-5LM2DR	SCHEMBL24950252	3-[5-[4-[[1-[4-[[5-Hydroxy-2-(4-hydroxyphenyl)-3-methylindol-1-yl]methyl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-1-benzofuran-3-yl]piperidine-2,6-dione	CC1=C(C2=CC=C(O)C=C2)N(CC2=CC=C(N3CCC(CN4CCN(C5=CC=C6OC=C(C7CCC(=O)NC7=O)C6=C5)CC4)CC3)C=C2)C2=C1C=C(O)C=C2	C45H47N5O5	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-RM9KC8	SCHEMBL24950190	3-[5-[4-[2-[1-[4-[[5-Hydroxy-2-(4-hydroxyphenyl)-3-methylindol-1-yl]methyl]phenyl]piperidin-4-yl]ethyl]piperazin-1-yl]-1-benzofuran-3-yl]piperidine-2,6-dione	CC1=C(C2=CC=C(O)C=C2)N(CC2=CC=C(N3CCC(CCN4CCN(C5=CC=C6OC=C(C7CCC(=O)NC7=O)C6=C5)CC4)CC3)C=C2)C2=C1C=C(O)C=C2	C46H49N5O5	BRD4;c-Myc	O60885/P01106	CRBN	WO-2021185291-A1
TPD-0LQH87	CHEMBL5201103	2-[[5-chloro-2-[4-[4-[8-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]acetyl]amino]octyl]piperazin-1-yl]-2-methoxyanilino]pyrimidin-4-yl]amino]-N-methylbenzamide; BDBM50593928; PD216457	CNC(=O)c1ccccc1Nc1nc(Nc2ccc(N3CCN(CCCCCCCCNC(=O)CNc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)cc2OC)ncc1Cl	C46H54ClN11O7	FAK	Q05397	CRBN	WO-2021190413-A1
TPD-IL42BK	CHEMBL5170596	2-[[5-chloro-2-[4-[4-[3-[3-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethylamino]-3-oxopropoxy]propyl]piperazin-1-yl]-2-methoxyanilino]pyrimidin-4-yl]amino]-N-methylbenzamide; BDBM50593929; PD216458	CNC(=O)c1ccccc1Nc1nc(Nc2ccc(N3CCN(CCCOCCC(=O)NCCNc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)cc2OC)ncc1Cl	C44H50ClN11O8	FAK	Q05397	CRBN	WO-2021190413-A1
TPD-1NSHI8	CHEMBL5191088	2-[[5-chloro-2-[4-[4-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethyl]piperazin-1-yl]-2-methoxyanilino]pyrimidin-4-yl]amino]-N-methylbenzamide; BDBM50593930; PD216459	CNC(=O)c1ccccc1Nc1nc(Nc2ccc(N3CCN(CCOCCOCCOCCNc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)cc2OC)ncc1Cl	C44H51ClN10O9	FAK	Q05397	CRBN	WO-2021190413-A1
TPD-0QZGCF	Fak protac B5	FAK PROTAC B5; 2471525-44-5; CHEMBL5172031; orb1983069; BDBM50593931; AT44275; DA-63362; PD216460; HY-143458; CS-0438140	CNC(=O)c1ccccc1Nc1nc(Nc2ccc(N3CCN(CCCCC(=O)Nc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)cc2OC)ncc1Cl	C41H43ClN10O7	FAK	Q05397	CRBN	WO-2021190413-A1
TPD-SQ6FJE	CHEMBL5203043	2-[[5-chloro-2-[4-[4-[6-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]-6-oxohexyl]piperazin-1-yl]-2-methoxyanilino]pyrimidin-4-yl]amino]-N-methylbenzamide; BDBM50593932; PD216461	CNC(=O)c1ccccc1Nc1nc(Nc2ccc(N3CCN(CCCCCC(=O)Nc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)cc2OC)ncc1Cl	C42H45ClN10O7	FAK	Q05397	CRBN	WO-2021190413-A1
TPD-RCCXJR	CHEMBL5183755	2-[[5-chloro-2-[4-[4-[7-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]-7-oxoheptyl]piperazin-1-yl]-2-methoxyanilino]pyrimidin-4-yl]amino]-N-methylbenzamide; BDBM50593933; PD216462	CNC(=O)c1ccccc1Nc1nc(Nc2ccc(N3CCN(CCCCCCC(=O)Nc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)cc2OC)ncc1Cl	C43H47ClN10O7	FAK	Q05397	CRBN	WO-2021190413-A1
TPD-KITH5W	CHEMBL5177296	2-[[5-chloro-2-[4-[4-[8-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]-8-oxooctyl]piperazin-1-yl]-2-methoxyanilino]pyrimidin-4-yl]amino]-N-methylbenzamide; BDBM50593934; PD216463	CNC(=O)c1ccccc1Nc1nc(Nc2ccc(N3CCN(CCCCCCCC(=O)Nc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)cc2OC)ncc1Cl	C44H49ClN10O7	FAK	Q05397	CRBN	WO-2021190413-A1
TPD-FU8MX5	CHEMBL5186599	2-[[5-chloro-2-[4-[4-[9-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]-9-oxononyl]piperazin-1-yl]-2-methoxyanilino]pyrimidin-4-yl]amino]-N-methylbenzamide; BDBM50593935; PD216464	CNC(=O)c1ccccc1Nc1nc(Nc2ccc(N3CCN(CCCCCCCCC(=O)Nc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)cc2OC)ncc1Cl	C45H51ClN10O7	FAK	Q05397	CRBN	WO-2021190413-A1
TPD-44HYKN	CHEMBL5207575	2-[[5-chloro-2-[4-[4-[10-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]-10-oxodecyl]piperazin-1-yl]-2-methoxyanilino]pyrimidin-4-yl]amino]-N-methylbenzamide; BDBM50593936; PD216465	CNC(=O)c1ccccc1Nc1nc(Nc2ccc(N3CCN(CCCCCCCCCC(=O)Nc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)cc2OC)ncc1Cl	C46H53ClN10O7	FAK	Q05397	CRBN	WO-2021190413-A1
TPD-18450H	CHEMBL5201498	2-[[5-chloro-2-[4-[4-[5-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethylamino]-5-oxopentyl]piperazin-1-yl]-2-methoxyanilino]pyrimidin-4-yl]amino]-N-methylbenzamide; BDBM50593937; PD216466	CNC(=O)c1ccccc1Nc1nc(Nc2ccc(N3CCN(CCCCC(=O)NCCNc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)cc2OC)ncc1Cl	C43H48ClN11O7	FAK	Q05397	CRBN	WO-2021190413-A1
TPD-76EM81	CHEMBL5173827	2-[[5-chloro-2-[4-[4-[6-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethylamino]-6-oxohexyl]piperazin-1-yl]-2-methoxyanilino]pyrimidin-4-yl]amino]-N-methylbenzamide; BDBM50593938; PD216467	CNC(=O)c1ccccc1Nc1nc(Nc2ccc(N3CCN(CCCCCC(=O)NCCNc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)cc2OC)ncc1Cl	C44H50ClN11O7	FAK	Q05397	CRBN	WO-2021190413-A1
TPD-5C6G5Q	CHEMBL5181306	2-[[5-chloro-2-[4-[4-[7-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethylamino]-7-oxoheptyl]piperazin-1-yl]-2-methoxyanilino]pyrimidin-4-yl]amino]-N-methylbenzamide; BDBM50593939; PD216468	CNC(=O)c1ccccc1Nc1nc(Nc2ccc(N3CCN(CCCCCCC(=O)NCCNc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)cc2OC)ncc1Cl	C45H52ClN11O7	FAK	Q05397	CRBN	WO-2021190413-A1
TPD-9RSLK7	CHEMBL5178915	2-[[5-chloro-2-[4-[4-[8-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethylamino]-8-oxooctyl]piperazin-1-yl]-2-methoxyanilino]pyrimidin-4-yl]amino]-N-methylbenzamide; BDBM50593940; PD216469	CNC(=O)c1ccccc1Nc1nc(Nc2ccc(N3CCN(CCCCCCCC(=O)NCCNc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)cc2OC)ncc1Cl	C46H54ClN11O7	FAK	Q05397	CRBN	WO-2021190413-A1
TPD-DADA0D	CHEMBL5183462	2-[[5-chloro-2-[4-[4-[10-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethylamino]-10-oxodecyl]piperazin-1-yl]-2-methoxyanilino]pyrimidin-4-yl]amino]-N-methylbenzamide; BDBM50593941; PD216470	CNC(=O)c1ccccc1Nc1nc(Nc2ccc(N3CCN(CCCCCCCCCC(=O)NCCNc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)cc2OC)ncc1Cl	C48H58ClN11O7	FAK	Q05397	CRBN	WO-2021190413-A1
TPD-2VK9LL	WO2021190413A1_15	.	COc1cc(N2CCN(CCCCC(=O)Nc3cccc4c3CN(C3CCC(=O)NC3=O)C4=O)CC2)ccc1Nc1ncc(Cl)c(Nc2ccccc2C(N)=O)n1	C40H43ClN10O6	FAK	Q05397	CRBN	WO-2021190413-A1
TPD-SAJPDK	WO2021190413A1_16	.	CNC(=O)c1ccccc1Nc1nc(Nc2ccc(N3CCN(CCCCCC(=O)Nc4cccc5c4CN(C4CCC(=O)NC4=O)C5=O)CC3)cc2OC)ncc1Cl	C42H47ClN10O6	FAK	Q05397	CRBN	WO-2021190413-A1
TPD-EEKHJ1	WO2021190413A1_17	.	CNC(=O)c1ccccc1Nc1nc(Nc2ccc(N3CCN(CCCCCCCC(=O)Nc4cccc5c4CN(C4CCC(=O)NC4=O)C5=O)CC3)cc2OC)ncc1Cl	C44H51ClN10O6	FAK	Q05397	CRBN	WO-2021190413-A1
TPD-FRU9S5	WO2021190413A1_18	.	CNC(=O)c1ccccc1Nc1nc(Nc2ccc(N3CCN(CCCCCCCCCC(=O)Nc4cccc5c4CN(C4CCC(=O)NC4=O)C5=O)CC3)cc2OC)ncc1Cl	C46H55ClN10O6	FAK	Q05397	CRBN	WO-2021190413-A1
TPD-ZUXGC2	CHEMBL5184768	[8-[[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]-8-oxooctyl] 4-[4-[[5-chloro-4-[2-(methylcarbamoyl)anilino]pyrimidin-2-yl]amino]-3-methoxyphenyl]piperazine-1-carbodithioate; BDBM50593942; PD216471	CNC(=O)c1ccccc1Nc1nc(Nc2ccc(N3CCN(C(=S)SCCCCCCCC(=O)Nc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)cc2OC)ncc1Cl	C45H49ClN10O7S2	FAK	Q05397	CRBN	WO-2021190413-A1
TPD-LEIA51	CHEMBL5203801	[10-[[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]-10-oxodecyl] 4-[4-[[5-chloro-4-[2-(methylcarbamoyl)anilino]pyrimidin-2-yl]amino]-3-methoxyphenyl]piperazine-1-carbodithioate; BDBM50593943; PD216472	CNC(=O)c1ccccc1Nc1nc(Nc2ccc(N3CCN(C(=S)SCCCCCCCCCC(=O)Nc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)cc2OC)ncc1Cl	C47H53ClN10O7S2	FAK	Q05397	CRBN	WO-2021190413-A1
TPD-IYSKS2	SCHEMBL23983475	3-tert-butyl-N-[[4-[6-[4-[1-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperidin-4-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]methyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(C5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)cc4)cc23)ccc1CNC(=O)c1nc(C(C)(C)C)no1	C48H54N10O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-ZZTOQ0	SCHEMBL23983317	3-tert-butyl-N-[[4-[6-[4-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperidin-4-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]methyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(C5CCN(CC6CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)cc4)cc23)ccc1CNC(=O)c1nc(C(C)(C)C)no1	C51H53FN10O6	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-BDR46W	SCHEMBL23983261	3-tert-butyl-N-[[4-[6-[4-[1-[2-[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]ethyl]piperidin-4-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]methyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(C5CCN(CCC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)cc4)cc23)ccc1CNC(=O)c1nc(C(C)(C)C)no1	C49H56N10O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-KLBKR1	WO2021219070A1_4	.	Cc1cc(-c2ncnc3[nH]c(-c4ccc(C5CCN(CCC6CCN(c7ccc(C8CCC(=O)NC8=O)cc7)CC6)CC5)cc4)cc23)ccc1CNC(=O)c1nc(C(C)C)no1	C49H55N9O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-DOIM7X	SCHEMBL23983267	3-tert-butyl-N-[[4-[6-[4-[1-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]azetidin-3-yl]methyl]piperidin-4-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]methyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(C5CCN(CC6CN(c7ccc(N8CCC(=O)NC8=O)cc7)C6)CC5)cc4)cc23)ccc1CNC(=O)c1nc(C(C)(C)C)no1	C46H50N10O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-YY4OEI	SCHEMBL23983428	3-tert-butyl-N-[[4-[6-[4-[1-[3-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]propyl]piperidin-4-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]methyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(C5CCN(CCCC6CN(c7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)C6)CC5)cc4)cc23)ccc1CNC(=O)c1nc(C(C)(C)C)no1	C51H54N10O6	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-IDOZUH	SCHEMBL23983260	3-tert-butyl-N-[(1R)-1-[4-[6-[4-[1-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperidin-4-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(C5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)cc4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C49H56N10O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-EPLYUH	SCHEMBL23983331	3-tert-butyl-N-[(1S)-1-[4-[6-[4-[1-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperidin-4-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(C5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)cc4)cc23)ccc1[C@H](C)NC(=O)c1nc(C(C)(C)C)no1	C49H56N10O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-6RF99A	SCHEMBL23983257	1-[4-[4-[[4-[4-[4-[3-(4,4-dimethyl-9-oxo-1,10-diazatricyclo[6.4.0.02,6]dodeca-2(6),7-dien-10-yl)-2-methylphenyl]-7H-pyrrolo[2,3-d]pyrimidin-6-yl]phenyl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-1,3-diazinane-2,4-dione	Cc1c(-c2ncnc3[nH]c(-c4ccc(C5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)cc4)cc23)cccc1N1CCn2c(cc3c2CC(C)(C)C3)C1=O	C52H57N9O3	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-0BNKRQ	SCHEMBL23983469	1-[4-[4-[[4-[5-[4-[3-(4,4-dimethyl-9-oxo-1,10-diazatricyclo[6.4.0.02,6]dodeca-2(6),7-dien-10-yl)-2-methylphenyl]-7H-pyrrolo[2,3-d]pyrimidin-6-yl]pyridin-2-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]-1,3-diazinane-2,4-dione	Cc1c(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)nc4)cc23)cccc1N1CCn2c(cc3c2CC(C)(C)C3)C1=O	C50H55N11O3	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-V59RPN	SCHEMBL23983492	1-[4-[4-[[4-[4-[4-[3-(4,4-dimethyl-9-oxo-1,10-diazatricyclo[6.4.0.02,6]dodeca-2(6),7-dien-10-yl)-2-methylphenyl]-7H-pyrrolo[2,3-d]pyrimidin-6-yl]phenyl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]-1,3-diazinane-2,4-dione	Cc1c(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)cc4)cc23)cccc1N1CCn2c(cc3c2CC(C)(C)C3)C1=O	C51H56N10O3	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-PZD0O3	SCHEMBL23984159	3-tert-butyl-N-[[4-[6-[4-[1-[3-(2,4-dioxo-1,3-diazinan-1-yl)-4-methoxybenzoyl]piperidin-4-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]methyl]-1,2,4-oxadiazole-5-carboxamide; SCHEMBL30281682	COc1ccc(C(=O)N2CCC(c3ccc(-c4cc5c(-c6ccc(CNC(=O)c7nc(C(C)(C)C)no7)c(C)c6)ncnc5[nH]4)cc3)CC2)cc1N1CCC(=O)NC1=O	C44H45N9O6	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-6FS1O2	SCHEMBL23983313	3-tert-butyl-N-[[4-[6-[4-[1-[2-[1-[5-(2,4-dioxo-1,3-diazinan-1-yl)-6-methylpyridin-2-yl]piperidin-4-yl]ethyl]piperidin-4-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]methyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(C5CCN(CCC6CCN(c7ccc(N8CCC(=O)NC8=O)c(C)n7)CC6)CC5)cc4)cc23)ccc1CNC(=O)c1nc(C(C)(C)C)no1	C49H57N11O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-OUBSSX	Btk-IN-29	BTK-IN-29; Catadegbrutinib; 2736508-60-2; BGB116673; (R)-3-(TERT-BUTYL)-N-[1-[4-[6-[6-[4-[[1-[4-[2,4-DIOXOTETRAHYDROPYRIMIDIN-1(2H)-YL]PHENYL]-4-PIPERIDYL]METHYL]-1-PIPERAZINYL]-3-PYRIDYL]-7H-PYRROLO[2,3-D]PYRIMIDIN-4-YL]-2-METHYLPHENYL]ETHYL]-1,2,4-OXADIAZOLE-5-CARBOXAMIDE; catadegbrutinib [INN]; PF6GPZ4DYT; orb2566761; SCHEMBL23984154; GTPL13736; EX-A8331; BGB-116673; compound 14 [WO2021219070A1]; SY396764; HY-160141; CS-0911695; G86483; 1,2,4-Oxadiazole-5-carboxamide, 3-(1,1-dimethylethyl)-N-[(1R)-1-[2-methyl-4-[6-[6-[4-[[1-[4-(tetrahydro-2,4-dioxo-1(2H)-pyrimidinyl)phenyl]-4-piperidinyl]methyl]-1-piperazinyl]-3-pyridinyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]phenyl]ethyl]-; 3-tert-butyl-N-[(1R)-1-[4-[6-[6-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-3-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide; 3-tert-butyl-N-{(1R)-1-[13-methyl-82,84-dioxo-27H-2(4,6)-pyrrolo[2,3-d]pyrimidina-8(1)-[1,3]diazinana-4(1,4)-piperazina-3(5,2)-pyridina-6(4,1)-piperidina-1(1),7(1,4)-dibenzenaoctaphan-14-yl]ethyl}-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)nc4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C47H54N12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-JGIBZM	SCHEMBL23983343	3-tert-butyl-N-[[4-[6-[4-[1-[2-[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)-3-fluorophenyl]piperidin-4-yl]ethyl]piperidin-4-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]methyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(C5CCN(CCC6CCN(c7ccc(N8CCC(=O)NC8=O)c(F)c7)CC6)CC5)cc4)cc23)ccc1CNC(=O)c1nc(C(C)(C)C)no1	C49H55FN10O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-AZZ3TT	SCHEMBL23983337	3-tert-butyl-N-[[4-[6-[1-[1-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperidin-4-yl]pyrazol-4-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-fluorophenyl]methyl]-1,2,4-oxadiazole-5-carboxamide	CC(C)(C)c1noc(C(=O)NCc2ccc(-c3ncnc4[nH]c(-c5cnn(C6CCN(CC7CCN(c8ccc(N9CCC(=O)NC9=O)cc8)CC7)CC6)c5)cc34)cc2F)n1	C44H49FN12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-63VU8C	SCHEMBL23983340	3-tert-butyl-N-[[4-[6-[4-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperidin-4-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]methyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(C5CCN(CC6CCN(c7ccc8c(c7)CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)cc4)cc23)ccc1CNC(=O)c1nc(C(C)(C)C)no1	C51H56N10O5	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-IW0HZH	SCHEMBL23983863	3-tert-butyl-N-[[4-[6-[4-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]methyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)cc4)cc23)ccc1CNC(=O)c1nc(C(C)(C)C)no1	C47H53N11O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-E89FQX	2736508-65-7	3-(1,1-Dimethylethyl)-N-[(1R)-1-[2-methyl-4-[6-[5-[4-[[1-[4-(tetrahydro-2,4-dioxo-1(2H)-pyrimidinyl)phenyl]-4-piperidinyl]methyl]-1-piperazinyl]-2-pyridinyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]phenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide; BGB16673; PROTAC BTK Degrader-12; orb2945760; SCHEMBL23983861; EX-A8316; AT46732; 3-(1,1-Dimethylethyl)-N-[(1R)-1-[2-methyl-4-[6-[5-[4-[[1-[4-(tetrahydro-2,4-dioxo-1(2H)-pyrimidinyl)phenyl]-4-piperidinyl]methyl]-1-piperazinyl]-2-pyridinyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]phenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide; HY-170413	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)cn4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C47H54N12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-Y8LJTC	SCHEMBL23983458	3-tert-butyl-N-[(1R)-1-[4-[6-[4-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)cc4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C48H55N11O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-2PVV3S	SCHEMBL23983551	3-tert-butyl-N-[(1R)-1-[4-[6-[4-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-fluorophenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	C[C@@H](NC(=O)c1nc(C(C)(C)C)no1)c1ccc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)cc4)cc23)cc1F	C47H52FN11O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-6KZC1I	SCHEMBL25203593	3-tert-butyl-N-[[4-[6-[4-[1-[2-[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)-3-methylphenyl]piperidin-4-yl]ethyl]piperidin-4-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]methyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(C5CCN(CCC6CCN(c7ccc(N8CCC(=O)NC8=O)c(C)c7)CC6)CC5)cc4)cc23)ccc1CNC(=O)c1nc(C(C)(C)C)no1	C50H58N10O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-BZBEVX	SCHEMBL23983494	3-tert-butyl-N-[[4-[6-[4-[1-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperidin-4-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-fluorophenyl]methyl]-1,2,4-oxadiazole-5-carboxamide	CC(C)(C)c1noc(C(=O)NCc2ccc(-c3ncnc4[nH]c(-c5ccc(C6CCN(CC7CCN(c8ccc(N9CCC(=O)NC9=O)cc8)CC7)CC6)cc5)cc34)cc2F)n1	C47H51FN10O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-ON6TGG	SCHEMBL23983318	3-tert-butyl-N-[[4-[6-[4-[1-[2-[1-[3-chloro-4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]ethyl]piperidin-4-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]methyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(C5CCN(CCC6CCN(c7ccc(N8CCC(=O)NC8=O)c(Cl)c7)CC6)CC5)cc4)cc23)ccc1CNC(=O)c1nc(C(C)(C)C)no1	C49H55ClN10O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-70IEDS	SCHEMBL23983269	3-tert-butyl-N-[(1R)-1-[4-[8-[4-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]phenyl]-7H-purin-6-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)cc4)nc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C47H54N12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-CDC0QB	SCHEMBL25245174	3-tert-butyl-N-[(1R)-1-[4-[6-[6-[4-[2-[1-[3-chloro-4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]ethyl]piperazin-1-yl]pyridin-3-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CCC6CCN(c7ccc(N8CCC(=O)NC8=O)c(Cl)c7)CC6)CC5)nc4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C48H55ClN12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-VA1JHC	SCHEMBL23984156	3-tert-butyl-N-[[4-[6-[4-[1-[[1-[3-(2,4-dioxo-1,3-diazinan-1-yl)-4-methoxybenzoyl]piperidin-4-yl]methyl]piperidin-4-yl]oxyphenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]methyl]-1,2,4-oxadiazole-5-carboxamide	COc1ccc(C(=O)N2CCC(CN3CCC(Oc4ccc(-c5cc6c(-c7ccc(CNC(=O)c8nc(C(C)(C)C)no8)c(C)c7)ncnc6[nH]5)cc4)CC3)CC2)cc1N1CCC(=O)NC1=O	C50H56N10O7	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-2YKC9C	SCHEMBL23983325	N-[3-[6-[4-[1-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperidin-4-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-5-fluoro-2-methylphenyl]-2-fluoro-4-(2-hydroxypropan-2-yl)benzamide	Cc1c(NC(=O)c2ccc(C(C)(C)O)cc2F)cc(F)cc1-c1ncnc2[nH]c(-c3ccc(C4CCN(CC5CCN(c6ccc(N7CCC(=O)NC7=O)cc6)CC5)CC4)cc3)cc12	C50H52F2N8O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-X25T17	SCHEMBL23983322	N-[3-[6-[4-[1-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperidin-4-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-5-fluoro-2-methylphenyl]-2-fluoro-4-prop-1-en-2-ylbenzamide	C=C(C)c1ccc(C(=O)Nc2cc(F)cc(-c3ncnc4[nH]c(-c5ccc(C6CCN(CC7CCN(c8ccc(N9CCC(=O)NC9=O)cc8)CC7)CC6)cc5)cc34)c2C)c(F)c1	C50H50F2N8O3	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-RXE289	SCHEMBL23983263	5-tert-butyl-N-[[4-[6-[4-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]methyl]-1,2,4-oxadiazole-3-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)cc4)cc23)ccc1CNC(=O)c1noc(C(C)(C)C)n1	C47H53N11O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-KV0QRK	SCHEMBL23983319	5-tert-butyl-N-[(1R)-1-[4-[6-[4-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-fluorophenyl]ethyl]-1,2,4-oxadiazole-3-carboxamide	C[C@@H](NC(=O)c1noc(C(C)(C)C)n1)c1ccc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)cc4)cc23)cc1F	C47H52FN11O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-MLM0D6	SCHEMBL23983282	3-tert-butyl-N-[[4-[6-[4-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-fluorophenyl]methyl]-1,2,4-oxadiazole-5-carboxamide	CC(C)(C)c1noc(C(=O)NCc2ccc(-c3ncnc4[nH]c(-c5ccc(N6CCN(CC7CCN(c8ccc(N9CCC(=O)NC9=O)cc8)CC7)CC6)cc5)cc34)cc2F)n1	C46H50FN11O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-IXUEHF	SCHEMBL23983281	3-tert-butyl-N-[(1R)-1-[4-[6-[6-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-3-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-fluorophenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	C[C@@H](NC(=O)c1nc(C(C)(C)C)no1)c1ccc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)nc4)cc23)cc1F	C46H51FN12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-PZCY9R	SCHEMBL25204442	5-tert-butyl-N-[(1R)-1-[4-[6-[6-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-3-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-fluorophenyl]ethyl]-1,2,4-oxadiazole-3-carboxamide	C[C@@H](NC(=O)c1noc(C(C)(C)C)n1)c1ccc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)nc4)cc23)cc1F	C46H51FN12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-WM51HH	SCHEMBL25242086	1-tert-butyl-N-[[4-[6-[4-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]methyl]pyrazole-4-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)cc4)cc23)ccc1CNC(=O)c1cnn(C(C)(C)C)c1	C48H55N11O3	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-IPNDUY	SCHEMBL23983684	N-[[4-[6-[4-[1-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperidin-4-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-fluoro-5-methylphenyl]methyl]-2-fluoro-4-(2-hydroxypropan-2-yl)benzamide	Cc1cc(CNC(=O)c2ccc(C(C)(C)O)cc2F)c(F)cc1-c1ncnc2[nH]c(-c3ccc(C4CCN(CC5CCN(c6ccc(N7CCC(=O)NC7=O)cc6)CC5)CC4)cc3)cc12	C51H54F2N8O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-7V3G85	SCHEMBL23983366	1-tert-butyl-N-[[4-[6-[4-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]methyl]triazole-4-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)cc4)cc23)ccc1CNC(=O)c1cn(C(C)(C)C)nn1	C47H54N12O3	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-FPVGG4	SCHEMBL23983584	3-tert-butyl-N-[(1R)-1-[4-[6-[4-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-fluorophenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)c(F)c4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C48H54FN11O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-IVFFC5	SCHEMBL23983500	3-tert-butyl-N-[[4-[6-[4-[1-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)-2-fluorophenyl]piperidin-4-yl]methyl]piperidin-4-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]methyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(C5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7F)CC6)CC5)cc4)cc23)ccc1CNC(=O)c1nc(C(C)(C)C)no1	C48H53FN10O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-FEFED8	SCHEMBL23983687	1-tert-butyl-N-[[4-[6-[4-[1-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperidin-4-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]methyl]triazole-4-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(C5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)cc4)cc23)ccc1CNC(=O)c1cn(C(C)(C)C)nn1	C48H55N11O3	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-Z1CW2D	SCHEMBL25203139	5-tert-butyl-N-[(1R)-1-[4-[6-[4-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-3-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)cc4)cc23)ccc1[C@@H](C)NC(=O)c1noc(C(C)(C)C)n1	C48H55N11O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-616P7O	SCHEMBL25245520	3-tert-butyl-N-[[4-[6-[6-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-3-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-fluorophenyl]methyl]-1,2,4-oxadiazole-5-carboxamide	CC(C)(C)c1noc(C(=O)NCc2ccc(-c3ncnc4[nH]c(-c5ccc(N6CCN(CC7CCN(c8ccc(N9CCC(=O)NC9=O)cc8)CC7)CC6)nc5)cc34)cc2F)n1	C45H49FN12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-0CESXZ	SCHEMBL23984253	3-tert-butyl-N-[(1R)-1-[4-[6-[4-[4-[[1-[2-(2,4-dioxo-1,3-diazinan-1-yl)-5-fluorophenyl]piperidin-4-yl]methyl]piperazin-1-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7cc(F)ccc7N7CCC(=O)NC7=O)CC6)CC5)cc4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C48H54FN11O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-79HBJY	SCHEMBL25666868	3-tert-butyl-N-[(1R)-1-[4-[6-[4-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)-3-methylphenyl]piperidin-4-yl]methyl]piperazin-1-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)c(C)c7)CC6)CC5)cc4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C49H57N11O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-OJI1R7	SCHEMBL23983459	3-tert-butyl-N-[(1R)-1-[4-[6-[4-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)-3-methoxyphenyl]piperidin-4-yl]methyl]piperazin-1-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	COc1cc(N2CCC(CN3CCN(c4ccc(-c5cc6c(-c7ccc([C@@H](C)NC(=O)c8nc(C(C)(C)C)no8)c(C)c7)ncnc6[nH]5)cc4)CC3)CC2)ccc1N1CCC(=O)NC1=O	C49H57N11O5	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-YB4EG0	SCHEMBL23983393	2-tert-butyl-N-[[4-[6-[4-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]methyl]-1,3-thiazole-4-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)cc4)cc23)ccc1CNC(=O)c1csc(C(C)(C)C)n1	C48H54N10O3S	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-502FA3	SCHEMBL23984209	2-tert-butyl-N-[[4-[6-[4-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]methyl]-1,3-thiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)cc4)cc23)ccc1CNC(=O)c1cnc(C(C)(C)C)s1	C48H54N10O3S	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-6ZI8IL	2736508-94-2	3-tert-butyl-N-[(1R)-1-[4-[6-[6-[4-[[1-[4-(2,6-dioxopiperidin-3-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-3-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide; orb2802225; SCHEMBL23984259; EX-A8331A; 1,2,4-Oxadiazole-5-carboxamide, 3-(1,1-dimethylethyl)-N-[(1R)-1-[4-[6-[6-[4-[[1-[4-(2,6-dioxo-3-piperidinyl)phenyl]-4-piperidinyl]methyl]-1-piperazinyl]-3-pyridinyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(C8CCC(=O)NC8=O)cc7)CC6)CC5)nc4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C48H55N11O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-NTKSDO	SCHEMBL23984181	3-tert-butyl-N-[[4-[6-[4-[1-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperidin-4-yl]oxyphenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]methyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(OC5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)cc4)cc23)ccc1CNC(=O)c1nc(C(C)(C)C)no1	C48H54N10O5	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-XZECFP	SCHEMBL23984254	N-[[4-[6-[4-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]methyl]-5-(1,1,1-trifluoro-2-methylpropan-2-yl)-1,2,4-oxadiazole-3-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)cc4)cc23)ccc1CNC(=O)c1noc(C(C)(C)C(F)(F)F)n1	C47H50F3N11O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-515U9N	WO2021219070A1_51	.	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)cc4)cc23)ccc1CNC(=O)C1=NOC2N1C(F)(F)C21CC1	C47H49F2N11O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-56STKI	SCHEMBL23984213	3-tert-butyl-N-[(1R)-1-[4-[6-[6-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)-3-methylphenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-3-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-fluorophenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(N2CCC(CN3CCN(c4ccc(-c5cc6c(-c7ccc([C@@H](C)NC(=O)c8nc(C(C)(C)C)no8)c(F)c7)ncnc6[nH]5)cn4)CC3)CC2)ccc1N1CCC(=O)NC1=O	C47H53FN12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-YRR9L7	SCHEMBL25227518	3-tert-butyl-N-[(1R)-1-[4-[6-[6-[4-[2-[1-[4-(2,6-dioxopiperidin-3-yl)phenyl]piperidin-4-yl]ethyl]piperazin-1-yl]pyridin-3-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CCC6CCN(c7ccc(C8CCC(=O)NC8=O)cc7)CC6)CC5)nc4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C49H57N11O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-YICUHL	SCHEMBL25227515	3-tert-butyl-N-[(1R)-1-[4-[6-[6-[4-[2-[1-[4-[(3S)-2,6-dioxopiperidin-3-yl]phenyl]piperidin-4-yl]ethyl]piperazin-1-yl]pyridin-3-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CCC6CCN(c7ccc([C@@H]8CCC(=O)NC8=O)cc7)CC6)CC5)nc4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C49H57N11O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-CDIP7A	SCHEMBL23983386	3-tert-butyl-N-[(1R)-1-[4-[6-[4-[4-[[1-[4-(2,6-dioxopiperidin-3-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(C8CCC(=O)NC8=O)cc7)CC6)CC5)cc4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C49H56N10O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-S98R8H	SCHEMBL23983696	5-tert-butyl-N-[(1R)-1-[4-[6-[6-[4-[[1-[4-(2,6-dioxopiperidin-3-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-3-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-3-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(C8CCC(=O)NC8=O)cc7)CC6)CC5)nc4)cc23)ccc1[C@@H](C)NC(=O)c1noc(C(C)(C)C)n1	C48H55N11O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-A47XUX	SCHEMBL25206610	5-tert-butyl-N-[(1R)-1-[4-[6-[5-[4-[[1-[4-(2,6-dioxopiperidin-3-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-2-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-3-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(C8CCC(=O)NC8=O)cc7)CC6)CC5)cn4)cc23)ccc1[C@@H](C)NC(=O)c1noc(C(C)(C)C)n1	C48H55N11O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-1NDQ9D	SCHEMBL25205770	3-tert-butyl-N-[(1R)-1-[4-[6-[6-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)-3-methylphenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-3-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)c(C)c7)CC6)CC5)nc4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C48H56N12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-KG0W8O	SCHEMBL23983416	3-tert-butyl-N-[(1R)-1-[4-[6-[5-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)-3-methylphenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-2-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)c(C)c7)CC6)CC5)cn4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C48H56N12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-98QP6N	SCHEMBL23983578	3-tert-butyl-N-[(1R)-1-[4-[6-[1-[1-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperidin-4-yl]-3,5-dimethylpyrazol-4-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4c(C)nn(C5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)c4C)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C48H58N12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-970E8D	SCHEMBL23983570	3-tert-butyl-N-[(1R)-1-[4-[6-[1-[1-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)-3-methylphenyl]piperidin-4-yl]methyl]piperidin-4-yl]-3,5-dimethylpyrazol-4-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4c(C)nn(C5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)c(C)c7)CC6)CC5)c4C)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C49H60N12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-OBS6BD	SCHEMBL23983573	5-tert-butyl-N-[(1R)-1-[4-[6-[1-[1-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperidin-4-yl]-3,5-dimethylpyrazol-4-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-3-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4c(C)nn(C5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)c4C)cc23)ccc1[C@@H](C)NC(=O)c1noc(C(C)(C)C)n1	C48H58N12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-V9U751	SCHEMBL25203981	3-tert-butyl-N-[(1R)-1-[4-[8-[6-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-3-yl]-7H-purin-6-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)nc4)nc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C46H53N13O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-SW5Q27	SCHEMBL25233676	3-tert-butyl-N-[(1R)-1-[4-[8-[5-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-2-yl]-7H-purin-6-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)cn4)nc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C46H53N13O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-K9IM5Y	SCHEMBL25209853	3-tert-butyl-N-[(1R)-1-[4-[8-[6-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)-3-methylphenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-3-yl]-7H-purin-6-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)c(C)c7)CC6)CC5)nc4)nc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C47H55N13O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-6IZXUW	SCHEMBL23983593	3-tert-butyl-N-[(1R)-1-[4-[8-[5-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)-3-methylphenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-2-yl]-7H-purin-6-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)c(C)c7)CC6)CC5)cn4)nc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C47H55N13O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-PAM0EC	SCHEMBL23983608	3-tert-butyl-N-[(1R)-1-[4-[8-[4-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)-3-methylphenyl]piperidin-4-yl]methyl]piperazin-1-yl]phenyl]-7H-purin-6-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)c(C)c7)CC6)CC5)cc4)nc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C48H56N12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-J23WGN	SCHEMBL23983427	5-tert-butyl-N-[(1R)-1-[4-[8-[4-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]phenyl]-7H-purin-6-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-3-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)cc4)nc23)ccc1[C@@H](C)NC(=O)c1noc(C(C)(C)C)n1	C47H54N12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-8A180N	SCHEMBL23983510	5-tert-butyl-N-[(1R)-1-[4-[8-[6-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-3-yl]-7H-purin-6-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-3-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)nc4)nc23)ccc1[C@@H](C)NC(=O)c1noc(C(C)(C)C)n1	C46H53N13O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-AAJET5	SCHEMBL23983512	5-tert-butyl-N-[(1R)-1-[4-[8-[5-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-2-yl]-7H-purin-6-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-3-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)cn4)nc23)ccc1[C@@H](C)NC(=O)c1noc(C(C)(C)C)n1	C46H53N13O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-1AC2YG	SCHEMBL23984219	5-tert-butyl-N-[(1R)-1-[4-[8-[6-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)-3-methylphenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-3-yl]-7H-purin-6-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-3-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)c(C)c7)CC6)CC5)nc4)nc23)ccc1[C@@H](C)NC(=O)c1noc(C(C)(C)C)n1	C47H55N13O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-J1HXMK	SCHEMBL25206570	5-tert-butyl-N-[(1R)-1-[4-[8-[5-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)-3-methylphenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-2-yl]-7H-purin-6-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-3-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)c(C)c7)CC6)CC5)cn4)nc23)ccc1[C@@H](C)NC(=O)c1noc(C(C)(C)C)n1	C47H55N13O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-NCJI3U	SCHEMBL23983314	5-tert-butyl-N-[(1R)-1-[4-[8-[4-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)-3-methylphenyl]piperidin-4-yl]methyl]piperazin-1-yl]phenyl]-7H-purin-6-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-3-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)c(C)c7)CC6)CC5)cc4)nc23)ccc1[C@@H](C)NC(=O)c1noc(C(C)(C)C)n1	C48H56N12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-RPL51S	SCHEMBL23983524	3-tert-butyl-N-[(1R)-1-[4-[6-[4-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-(hydroxymethyl)phenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	C[C@@H](NC(=O)c1nc(C(C)(C)C)no1)c1ccc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)cc4)cc23)cc1CO	C48H55N11O5	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-7WZJWN	SCHEMBL25666890	3-tert-butyl-N-[(1R)-1-[4-[6-[4-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-(methoxymethyl)phenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	COCc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)cc4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C49H57N11O5	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-OD3EBC	SCHEMBL25203974	3-tert-butyl-N-[(1R)-1-[4-[6-[6-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-3-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-(methoxymethyl)phenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	COCc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)nc4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C48H56N12O5	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-DZ20WE	SCHEMBL25237335	3-tert-butyl-N-[(1R)-1-[4-[6-[5-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-2-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-(methoxymethyl)phenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	COCc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)cn4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C48H56N12O5	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-Z0BWHU	SCHEMBL23984227	3-tert-butyl-N-[(1R)-1-[4-[6-[4-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-3-fluoro-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1c([C@@H](C)NC(=O)c2nc(C(C)(C)C)no2)ccc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)cc4)cc23)c1F	C48H54FN11O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-INVQRE	SCHEMBL23983298	3-tert-butyl-N-[(1R)-1-[4-[6-[6-[(2S)-4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]-2-methylpiperazin-1-yl]pyridin-3-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-fluorophenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	C[C@@H](NC(=O)c1nc(C(C)(C)C)no1)c1ccc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)C[C@@H]5C)nc4)cc23)cc1F	C47H53FN12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-KQA804	SCHEMBL23983730	3-tert-butyl-N-[(1R)-1-[4-[6-[6-[(2R)-4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]-2-methylpiperazin-1-yl]pyridin-3-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-fluorophenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	C[C@@H]1CN(CC2CCN(c3ccc(N4CCC(=O)NC4=O)cc3)CC2)CCN1c1ccc(-c2cc3c(-c4ccc([C@@H](C)NC(=O)c5nc(C(C)(C)C)no5)c(F)c4)ncnc3[nH]2)cn1	C47H53FN12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-04KTBP	WO2021219070A1_82	.	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)c(F)c7)CC6)CC5)cn4)cc23)ccc1[C@@H](C)NC(=O)C1=NC(C(C)(C)C)NO1	C47H55FN12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-T7C38D	SCHEMBL25235584	3-tert-butyl-N-[(1R)-1-[4-[6-[6-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)-3-fluorophenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-3-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)c(F)c7)CC6)CC5)nc4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C47H53FN12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-5Z5K9E	SCHEMBL25210566	N-[(1R)-1-[4-[6-[4-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-5-[1-(trifluoromethyl)cyclopropyl]-1,2,4-oxadiazole-3-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)cc4)cc23)ccc1[C@@H](C)NC(=O)c1noc(C2(C(F)(F)F)CC2)n1	C48H50F3N11O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-QBBS0K	SCHEMBL23984294	N-[(1R)-1-[4-[6-[4-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-5-(1,1,1-trifluoro-2-methylpropan-2-yl)-1,2,4-oxadiazole-3-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)cc4)cc23)ccc1[C@@H](C)NC(=O)c1noc(C(C)(C)C(F)(F)F)n1	C48H52F3N11O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-SJ8UGV	SCHEMBL25209879	N-[(1R)-1-[4-[6-[6-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-3-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-5-[1-(trifluoromethyl)cyclopropyl]-1,2,4-oxadiazole-3-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)nc4)cc23)ccc1[C@@H](C)NC(=O)c1noc(C2(C(F)(F)F)CC2)n1	C47H49F3N12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-FVYTFY	SCHEMBL25251534	N-[(1R)-1-[4-[6-[5-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-2-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-5-[1-(trifluoromethyl)cyclopropyl]-1,2,4-oxadiazole-3-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)cn4)cc23)ccc1[C@@H](C)NC(=O)c1noc(C2(C(F)(F)F)CC2)n1	C47H49F3N12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-N6MNWR	WO2021219070A1_88	.	Cc1cc(-c2ncnc3[nH]c(C4=CNC(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)C=C4)cc23)ccc1[C@@H](C)NC(=O)c1noc(C(C)(C)C(F)(F)F)n1	C47H53F3N12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-U85RFO	SCHEMBL23984297	N-[(1R)-1-[4-[6-[5-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-2-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-5-(1,1,1-trifluoro-2-methylpropan-2-yl)-1,2,4-oxadiazole-3-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)cn4)cc23)ccc1[C@@H](C)NC(=O)c1noc(C(C)(C)C(F)(F)F)n1	C47H51F3N12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-JI6ARL	SCHEMBL23983677	N-[(1R)-1-[4-[6-[4-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-5-(1-methylcyclopropyl)-1,2,4-oxadiazole-3-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)cc4)cc23)ccc1[C@@H](C)NC(=O)c1noc(C2(C)CC2)n1	C48H53N11O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-47BD24	SCHEMBL23983336	3-tert-butyl-N-[(1R)-1-[4-[6-[4-[4-[[1-[5-(2,4-dioxo-1,3-diazinan-1-yl)pyridin-2-yl]piperidin-4-yl]methyl]piperazin-1-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cn7)CC6)CC5)cc4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C47H54N12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-317WXW	SCHEMBL23984215	3-tert-butyl-N-[(1R)-1-[4-[6-[4-[4-[[1-[6-(2,4-dioxo-1,3-diazinan-1-yl)pyridin-3-yl]piperidin-4-yl]methyl]piperazin-1-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)nc7)CC6)CC5)cc4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C47H54N12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-CN3BEM	SCHEMBL23984289	3-tert-butyl-N-[(1R)-1-[4-[6-[5-[4-[[1-[5-(2,4-dioxo-1,3-diazinan-1-yl)pyridin-2-yl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-2-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cn7)CC6)CC5)cn4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C46H53N13O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-GBWOML	SCHEMBL23984286	3-tert-butyl-N-[(1R)-1-[4-[6-[5-[4-[[1-[6-(2,4-dioxo-1,3-diazinan-1-yl)pyridin-3-yl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-2-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)nc7)CC6)CC5)cn4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C46H53N13O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-NMFEOG	SCHEMBL25255186	3-tert-butyl-N-[(1R)-1-[4-[6-[6-[4-[[1-[5-(2,4-dioxo-1,3-diazinan-1-yl)pyridin-2-yl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-3-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cn7)CC6)CC5)nc4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C46H53N13O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-BB0NGY	SCHEMBL23984203	3-tert-butyl-N-[(1R)-1-[4-[6-[6-[4-[[1-[6-(2,4-dioxo-1,3-diazinan-1-yl)pyridin-3-yl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-3-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)nc7)CC6)CC5)nc4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C46H53N13O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-T9E484	SCHEMBL23984243	3-tert-butyl-N-[(1R)-1-[4-[6-[4-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCC(CN6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)cc4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C48H55N11O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-3N8MQW	SCHEMBL23984226	3-tert-butyl-N-[(1R)-1-[4-[6-[4-[4-[[4-[5-(2,4-dioxo-1,3-diazinan-1-yl)pyridin-2-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCC(CN6CCN(c7ccc(N8CCC(=O)NC8=O)cn7)CC6)CC5)cc4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C47H54N12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-STVPYL	SCHEMBL23983311	3-tert-butyl-N-[(1R)-1-[4-[6-[4-[4-[[4-[6-(2,4-dioxo-1,3-diazinan-1-yl)pyridin-3-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCC(CN6CCN(c7ccc(N8CCC(=O)NC8=O)nc7)CC6)CC5)cc4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C47H54N12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-SJ9LBC	SCHEMBL23984214	3-tert-butyl-N-[(1R)-1-[4-[6-[6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperazin-1-yl]methyl]piperidin-1-yl]pyridin-3-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCC(CN6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)nc4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C47H54N12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-HGZVJZ	SCHEMBL23984241	3-tert-butyl-N-[(1R)-1-[4-[6-[5-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperazin-1-yl]methyl]piperidin-1-yl]pyridin-2-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCC(CN6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)cn4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C47H54N12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-RPC0EA	SCHEMBL23984220	3-tert-butyl-N-[(1R)-1-[4-[6-[6-[4-[[4-[5-(2,4-dioxo-1,3-diazinan-1-yl)pyridin-2-yl]piperazin-1-yl]methyl]piperidin-1-yl]pyridin-3-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCC(CN6CCN(c7ccc(N8CCC(=O)NC8=O)cn7)CC6)CC5)nc4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C46H53N13O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-M9055D	SCHEMBL23983598	3-tert-butyl-N-[(1R)-1-[4-[6-[5-[4-[[4-[5-(2,4-dioxo-1,3-diazinan-1-yl)pyridin-2-yl]piperazin-1-yl]methyl]piperidin-1-yl]pyridin-2-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCC(CN6CCN(c7ccc(N8CCC(=O)NC8=O)cn7)CC6)CC5)cn4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C46H53N13O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-JVVDCQ	SCHEMBL25215520	5-tert-butyl-N-[(1R)-1-[4-[6-[6-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-3-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-3-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)nc4)cc23)ccc1[C@@H](C)NC(=O)c1noc(C(C)(C)C)n1	C47H54N12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-JL2DMR	WO2021219070A1_105	.	Cc1cc(-c2ncnc3c2CC(c2ccc(N4CCN(CC5CCN(c6ccc(N7CCC(=O)NC7=O)cc6)CC5)C[C@H]4C)nc2)N3)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C48H58N12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-1XLBCB	SCHEMBL25233908	3-tert-butyl-N-[(1R)-1-[4-[6-[6-[(2S)-4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]-2-methylpiperazin-1-yl]pyridin-3-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)C[C@@H]5C)nc4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C48H56N12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-L4HY4Z	SCHEMBL23983651	5-tert-butyl-N-[(1R)-1-[4-[6-[4-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-5-fluoro-2-methylphenyl]ethyl]-1,2,4-oxadiazole-3-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)cc4)cc23)c(F)cc1[C@@H](C)NC(=O)c1noc(C(C)(C)C)n1	C48H54FN11O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-HFPL8O	SCHEMBL23984245	5-tert-butyl-N-[(1R)-1-[4-[6-[5-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-2-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-fluorophenyl]ethyl]-1,2,4-oxadiazole-3-carboxamide	C[C@@H](NC(=O)c1noc(C(C)(C)C)n1)c1ccc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)cn4)cc23)cc1F	C46H51FN12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-ZWX4ZG	SCHEMBL25209055	3-tert-butyl-N-[[4-[6-[4-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-(hydroxymethyl)phenyl]methyl]-1,2,4-oxadiazole-5-carboxamide	CC(C)(C)c1noc(C(=O)NCc2ccc(-c3ncnc4[nH]c(-c5ccc(N6CCN(CC7CCN(c8ccc(N9CCC(=O)NC9=O)cc8)CC7)CC6)cc5)cc34)cc2CO)n1	C47H53N11O5	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-LMPNXH	SCHEMBL25212156	3-tert-butyl-N-[(1R)-1-[2-methyl-4-[6-[5-[4-[[1-[4-(3-methyl-2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-2-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]phenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)N(C)C8=O)cc7)CC6)CC5)cn4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C48H56N12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-DF48JP	SCHEMBL23984237	3-tert-butyl-N-[(1R)-1-[4-[6-[4-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)-3-fluorophenyl]piperidin-4-yl]methyl]piperazin-1-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)c(F)c7)CC6)CC5)cc4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C48H54FN11O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-QCCG8D	SCHEMBL23983605	3-tert-butyl-N-[(1R)-1-[4-[8-[4-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)-3-methylphenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-methylphenyl]-7H-purin-6-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)c(C)c7)CC6)CC5)c(C)c4)nc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C49H58N12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-AKN2PV	WO2021219070A1_113	.	COc1cc(C2Nc3ncnc(-c4ccc([C@@H](C)NC(=O)c5nc(C(C)(C)C)no5)c(C)c4)c3N2)ccc1N1CCN(CC2CCN(c3ccc(N4CCC(=O)NC4=O)c(C)c3)CC2)CC1	C49H60N12O5	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-CLF0F1	SCHEMBL23984217	3-tert-butyl-N-[(1R)-1-[4-[8-[4-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)-3-methylphenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-methylphenyl]-7H-purin-6-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(N2CCN(CC3CCN(c4ccc(N5CCC(=O)NC5=O)c(C)c4)CC3)CC2)ccc1-c1nc2c(-c3ccc([C@@H](C)NC(=O)c4nc(C(C)(C)C)no4)c(C)c3)ncnc2[nH]1	C49H58N12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-684QDR	SCHEMBL23983502	5-tert-butyl-N-[(1R)-1-[4-[6-[4-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-3-fluoro-2-methylphenyl]ethyl]-1,2,4-oxadiazole-3-carboxamide	Cc1c([C@@H](C)NC(=O)c2noc(C(C)(C)C)n2)ccc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)cc4)cc23)c1F	C48H54FN11O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-XSG7DL	SCHEMBL23983617	3-tert-butyl-N-[(1R)-1-[4-[6-[3-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4cccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)c4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C48H55N11O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-DOWCH6	SCHEMBL25217011	5-tert-butyl-N-[(1R)-1-[4-[6-[6-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-3-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2-oxazole-3-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)nc4)cc23)ccc1[C@@H](C)NC(=O)c1cc(C(C)(C)C)on1	C48H55N11O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-KIXAXB	SCHEMBL25204608	5-tert-butyl-N-[(1R)-1-[4-[6-[4-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-(hydroxymethyl)phenyl]ethyl]-1,2,4-oxadiazole-3-carboxamide	C[C@@H](NC(=O)c1noc(C(C)(C)C)n1)c1ccc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)cc4)cc23)cc1CO	C48H55N11O5	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-VA2KEC	SCHEMBL25251516	3-tert-butyl-N-[(1R)-1-[4-[6-[5-[4-[[1-[3-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-2-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7cccc(N8CCC(=O)NC8=O)c7)CC6)CC5)cn4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C47H54N12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-0R6AB4	SCHEMBL23983324	5-tert-butyl-N-[(1R)-1-[4-[6-[1-[1-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperidin-4-yl]-3,5-dimethylpyrazol-4-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-(hydroxymethyl)phenyl]ethyl]-1,2,4-oxadiazole-3-carboxamide	Cc1nn(C2CCN(CC3CCN(c4ccc(N5CCC(=O)NC5=O)cc4)CC3)CC2)c(C)c1-c1cc2c(-c3ccc([C@@H](C)NC(=O)c4noc(C(C)(C)C)n4)c(CO)c3)ncnc2[nH]1	C48H58N12O5	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-P0ZVX3	SCHEMBL23984222	1-tert-butyl-N-[(1R)-1-[4-[6-[1-[1-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperidin-4-yl]-3,5-dimethylpyrazol-4-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]triazole-4-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4c(C)nn(C5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)c4C)cc23)ccc1[C@@H](C)NC(=O)c1cn(C(C)(C)C)nn1	C48H59N13O3	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-UIO5JB	SCHEMBL23983702	1-tert-butyl-N-[(1R)-1-[4-[6-[1-[1-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperidin-4-yl]-3,5-dimethylpyrazol-4-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-(hydroxymethyl)phenyl]ethyl]triazole-4-carboxamide	Cc1nn(C2CCN(CC3CCN(c4ccc(N5CCC(=O)NC5=O)cc4)CC3)CC2)c(C)c1-c1cc2c(-c3ccc([C@@H](C)NC(=O)c4cn(C(C)(C)C)nn4)c(CO)c3)ncnc2[nH]1	C48H59N13O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-7ZR8PO	SCHEMBL23983682	N-[(1R)-1-[4-[6-[5-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)-3-methylphenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-2-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-5-[1-(hydroxymethyl)cyclopropyl]-1,2,4-oxadiazole-3-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)c(C)c7)CC6)CC5)cn4)cc23)ccc1[C@@H](C)NC(=O)c1noc(C2(CO)CC2)n1	C48H54N12O5	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-EPDNH8	SCHEMBL23983719	N-[(1R)-1-[4-[6-[5-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-2-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-5-(1-methylcyclopropyl)-1,2,4-oxadiazole-3-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)cn4)cc23)ccc1[C@@H](C)NC(=O)c1noc(C2(C)CC2)n1	C47H52N12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-CCJJ3M	SCHEMBL25245193	N-[(1R)-1-[4-[6-[5-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)-3-methylphenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-2-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-5-(1-methylcyclopropyl)-1,2,4-oxadiazole-3-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)c(C)c7)CC6)CC5)cn4)cc23)ccc1[C@@H](C)NC(=O)c1noc(C2(C)CC2)n1	C48H54N12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-G61EVE	SCHEMBL23983722	N-[(1R)-1-[4-[6-[6-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)-3-methylphenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-3-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-5-(1-methylcyclopropyl)-1,2,4-oxadiazole-3-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)c(C)c7)CC6)CC5)nc4)cc23)ccc1[C@@H](C)NC(=O)c1noc(C2(C)CC2)n1	C48H54N12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-9ZQBVP	SCHEMBL23983717	5-tert-butyl-N-[(1R)-1-[4-[6-[5-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-2-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-3-fluoro-2-methylphenyl]ethyl]-1,2,4-oxadiazole-3-carboxamide	Cc1c([C@@H](C)NC(=O)c2noc(C(C)(C)C)n2)ccc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)cn4)cc23)c1F	C47H53FN12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-O4XVMJ	SCHEMBL25216217	5-tert-butyl-N-[(1R)-1-[4-[6-[5-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)-3-methylphenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-2-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-3-fluoro-2-methylphenyl]ethyl]-1,2,4-oxadiazole-3-carboxamide	Cc1cc(N2CCC(CN3CCN(c4ccc(-c5cc6c(-c7ccc([C@@H](C)NC(=O)c8noc(C(C)(C)C)n8)c(C)c7F)ncnc6[nH]5)nc4)CC3)CC2)ccc1N1CCC(=O)NC1=O	C48H55FN12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-OSEUQR	SCHEMBL25202760	5-tert-butyl-N-[(1R)-1-[4-[6-[5-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)-3-methylphenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-2-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-3-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)c(C)c7)CC6)CC5)cn4)cc23)ccc1[C@@H](C)NC(=O)c1noc(C(C)(C)C)n1	C48H56N12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-SK1481	SCHEMBL25229129	5-tert-butyl-N-[(1R)-1-[4-[6-[5-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)-3-methylphenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-2-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-5-fluoro-2-methylphenyl]ethyl]-1,2,4-oxadiazole-3-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)c(C)c7)CC6)CC5)cn4)cc23)c(F)cc1[C@@H](C)NC(=O)c1noc(C(C)(C)C)n1	C48H55FN12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-0IRUMJ	SCHEMBL25211325	5-tert-butyl-N-[(1R)-1-[4-[6-[6-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-3-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-5-fluoro-2-methylphenyl]ethyl]-1,2,4-oxadiazole-3-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)nc4)cc23)c(F)cc1[C@@H](C)NC(=O)c1noc(C(C)(C)C)n1	C47H53FN12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-XFMSVJ	SCHEMBL23983643	5-tert-butyl-N-[(1R)-1-[4-[6-[6-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)-3-methylphenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-3-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-5-fluoro-2-methylphenyl]ethyl]-1,2,4-oxadiazole-3-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)c(C)c7)CC6)CC5)nc4)cc23)c(F)cc1[C@@H](C)NC(=O)c1noc(C(C)(C)C)n1	C48H55FN12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-SS1G13	SCHEMBL23983610	5-tert-butyl-N-[(1R)-1-[4-[6-[5-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-2-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-3-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)cn4)cc23)ccc1[C@@H](C)NC(=O)c1noc(C(C)(C)C)n1	C47H54N12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-8MU3HP	SCHEMBL25210550	5-tert-butyl-N-[(1R)-1-[4-[6-[5-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-2-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-5-fluoro-2-methylphenyl]ethyl]-1,2,4-oxadiazole-3-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)cn4)cc23)c(F)cc1[C@@H](C)NC(=O)c1noc(C(C)(C)C)n1	C47H53FN12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-SG66XK	SCHEMBL23984256	3-tert-butyl-N-[(1R)-1-[1-[6-[6-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-3-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]piperidin-4-yl]ethyl]-1,2,4-oxadiazole-5-carboxamide	C[C@@H](NC(=O)c1nc(C(C)(C)C)no1)C1CCN(c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)nc4)cc23)CC1	C45H57N13O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-GMF6KB	SCHEMBL23983625	5-tert-butyl-N-[(1R)-1-[4-[6-[5-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-2-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-(hydroxymethyl)phenyl]ethyl]-1,2,4-oxadiazole-3-carboxamide	C[C@@H](NC(=O)c1noc(C(C)(C)C)n1)c1ccc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)cn4)cc23)cc1CO	C47H54N12O5	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-QGTHJR	SCHEMBL25243511	5-tert-butyl-N-[(1R)-1-[4-[6-[5-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)-3-methylphenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-2-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-(hydroxymethyl)phenyl]ethyl]-1,2,4-oxadiazole-3-carboxamide	Cc1cc(N2CCC(CN3CCN(c4ccc(-c5cc6c(-c7ccc([C@@H](C)NC(=O)c8noc(C(C)(C)C)n8)c(CO)c7)ncnc6[nH]5)nc4)CC3)CC2)ccc1N1CCC(=O)NC1=O	C48H56N12O5	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-V0ZCAQ	SCHEMBL23984246	3-tert-butyl-N-[(1R)-1-[4-[6-[1-[1-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperidin-4-yl]-3,5-dimethylpyrazol-4-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-(hydroxymethyl)phenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1nn(C2CCN(CC3CCN(c4ccc(N5CCC(=O)NC5=O)cc4)CC3)CC2)c(C)c1-c1cc2c(-c3ccc([C@@H](C)NC(=O)c4nc(C(C)(C)C)no4)c(CO)c3)ncnc2[nH]1	C48H58N12O5	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-21C50J	SCHEMBL23983347	3-tert-butyl-N-[(1R)-1-[4-[6-[1-[1-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperidin-4-yl]-3,5-dimethylpyrazol-4-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-5-fluoro-2-(hydroxymethyl)phenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1nn(C2CCN(CC3CCN(c4ccc(N5CCC(=O)NC5=O)cc4)CC3)CC2)c(C)c1-c1cc2c(-c3cc(CO)c([C@@H](C)NC(=O)c4nc(C(C)(C)C)no4)cc3F)ncnc2[nH]1	C48H57FN12O5	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-A9DY53	SCHEMBL23984225	5-tert-butyl-N-[(1R)-1-[4-[6-[6-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-3-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-3-fluoro-2-methylphenyl]ethyl]-1,2,4-oxadiazole-3-carboxamide	Cc1c([C@@H](C)NC(=O)c2noc(C(C)(C)C)n2)ccc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)nc4)cc23)c1F	C47H53FN12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-QQUVDM	SCHEMBL23984293	5-tert-butyl-N-[(1R)-1-[4-[6-[6-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)-3-methylphenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-3-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-3-fluoro-2-methylphenyl]ethyl]-1,2,4-oxadiazole-3-carboxamide	Cc1cc(N2CCC(CN3CCN(c4ccc(-c5cc6c(-c7ccc([C@@H](C)NC(=O)c8noc(C(C)(C)C)n8)c(C)c7F)ncnc6[nH]5)cn4)CC3)CC2)ccc1N1CCC(=O)NC1=O	C48H55FN12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-IK8S87	SCHEMBL23983612	3-tert-butyl-N-[(1R)-1-[4-[6-[6-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-3-yl]-5-fluoro-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)nc4)c(F)c23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C47H53FN12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-O6FZCI	SCHEMBL23983338	3-tert-butyl-N-[(1R)-1-[4-[6-[4-[4-[[1-[4-(2,6-dioxopiperidin-3-yl)phenyl]pyrrolidin-3-yl]methyl]piperazin-1-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(C8CCC(=O)NC8=O)cc7)C6)CC5)cc4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C48H54N10O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-VCHLQ9	SCHEMBL23983564	5-tert-butyl-N-[(1R)-1-[4-[6-[6-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-3-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-(hydroxymethyl)phenyl]ethyl]-1,2,4-oxadiazole-3-carboxamide	C[C@@H](NC(=O)c1noc(C(C)(C)C)n1)c1ccc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)nc4)cc23)cc1CO	C47H54N12O5	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-2NKI63	SCHEMBL25206103	5-tert-butyl-N-[(1R)-1-[4-[6-[6-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)-3-methylphenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-3-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-(hydroxymethyl)phenyl]ethyl]-1,2,4-oxadiazole-3-carboxamide	Cc1cc(N2CCC(CN3CCN(c4ccc(-c5cc6c(-c7ccc([C@@H](C)NC(=O)c8noc(C(C)(C)C)n8)c(CO)c7)ncnc6[nH]5)cn4)CC3)CC2)ccc1N1CCC(=O)NC1=O	C48H56N12O5	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-LVOUPR	SCHEMBL23983515	3-tert-butyl-N-[(1R)-1-[2-methyl-4-[6-[6-[4-[[1-[4-(3-methyl-2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-3-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]phenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)N(C)C8=O)cc7)CC6)CC5)nc4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C48H56N12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-JQEWB8	SCHEMBL23983391	3-tert-butyl-N-[(1S)-1-[4-[6-[5-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-2-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)cn4)cc23)ccc1[C@H](C)NC(=O)c1nc(C(C)(C)C)no1	C47H54N12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-9K9BIS	SCHEMBL25205750	3-tert-butyl-N-[(1S)-1-[4-[6-[6-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-3-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)nc4)cc23)ccc1[C@H](C)NC(=O)c1nc(C(C)(C)C)no1	C47H54N12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-TASQ9N	SCHEMBL23983565	5-tert-butyl-N-[(1R)-1-[4-[6-[1-[1-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperidin-4-yl]-3,5-dimethylpyrazol-4-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-5-fluoro-2-(hydroxymethyl)phenyl]ethyl]-1,2,4-oxadiazole-3-carboxamide	Cc1nn(C2CCN(CC3CCN(c4ccc(N5CCC(=O)NC5=O)cc4)CC3)CC2)c(C)c1-c1cc2c(-c3cc(CO)c([C@@H](C)NC(=O)c4noc(C(C)(C)C)n4)cc3F)ncnc2[nH]1	C48H57FN12O5	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-R4U1A7	SCHEMBL25206636	3-tert-butyl-N-[(1R)-5-[6-[5-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-2-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2,3-dihydro-1H-inden-1-yl]-1,2,4-oxadiazole-5-carboxamide	CC(C)(C)c1noc(C(=O)N[C@@H]2CCc3cc(-c4ncnc5[nH]c(-c6ccc(N7CCN(CC8CCN(c9ccc(N%10CCC(=O)NC%10=O)cc9)CC8)CC7)cn6)cc45)ccc32)n1	C47H52N12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-6SFML4	SCHEMBL23984218	3-tert-butyl-N-[(1R)-5-[6-[6-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-3-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2,3-dihydro-1H-inden-1-yl]-1,2,4-oxadiazole-5-carboxamide	CC(C)(C)c1noc(C(=O)N[C@@H]2CCc3cc(-c4ncnc5[nH]c(-c6ccc(N7CCN(CC8CCN(c9ccc(N%10CCC(=O)NC%10=O)cc9)CC8)CC7)nc6)cc45)ccc32)n1	C47H52N12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-VSJ2W9	SCHEMBL23983568	3-tert-butyl-N-[(1R)-1-[4-[6-[4-[1-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperidin-4-yl]-3,5-dimethylpyrazol-1-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-n4nc(C)c(C5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)c4C)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C48H58N12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-YAL28A	SCHEMBL25217013	3-tert-butyl-N-[(1R)-1-[4-[6-[4-[4-[3-[4-(2,6-dioxopiperidin-3-yl)phenyl]cyclobutyl]piperazin-1-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(C6CC(c7ccc(C8CCC(=O)NC8=O)cc7)C6)CC5)cc4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C47H51N9O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-UWX8P5	SCHEMBL23983420	3-tert-butyl-N-[(1R)-1-[4-[6-[5-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-2-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-fluorophenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	C[C@@H](NC(=O)c1nc(C(C)(C)C)no1)c1ccc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)cn4)cc23)cc1F	C46H51FN12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-TMO37K	SCHEMBL23983424	3-tert-butyl-N-[(1R)-1-[4-[6-[1-[1-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperidin-4-yl]-3,5-dimethylpyrazol-4-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-N-methyl-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4c(C)nn(C5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)c4C)cc23)ccc1[C@@H](C)N(C)C(=O)c1nc(C(C)(C)C)no1	C49H60N12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-6T0QDY	SCHEMBL23983364	5-tert-butyl-N-[(1R)-5-[6-[4-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2,3-dihydro-1H-inden-1-yl]-1,2,4-oxadiazole-3-carboxamide	CC(C)(C)c1nc(C(=O)N[C@@H]2CCc3cc(-c4ncnc5[nH]c(-c6ccc(N7CCN(CC8CCN(c9ccc(N%10CCC(=O)NC%10=O)cc9)CC8)CC7)cc6)cc45)ccc32)no1	C48H53N11O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-V9VZR4	SCHEMBL23984262	3-tert-butyl-N-[(1R)-1-[4-[6-[4-[1-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]azetidin-3-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(C5CN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)C5)cc4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C47H52N10O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-TBR2AM	SCHEMBL23983430	3-tert-butyl-N-[(1R)-1-[4-[6-[4-[1-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]pyrrolidin-3-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(C5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)C5)cc4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C48H54N10O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-UT32TT	SCHEMBL23983425	3-tert-butyl-N-[(1R)-1-[4-[6-[6-[1-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]-2,5-dihydropyrrol-3-yl]pyridin-3-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(C5=CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)C5)nc4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C47H51N11O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-JWIZSF	SCHEMBL23983426	3-tert-butyl-N-[(1R)-1-[4-[6-[2-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyrimidin-5-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4cnc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)nc4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C46H53N13O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-NQNHF0	WO2021219070A1_161	.	Cc1cc(-c2nccc3[nH]c(-c4c(C)nn(C5CCN(C(=O)CNCC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)c4C)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C51H62N12O5	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-P4172X	SCHEMBL23983421	3-tert-butyl-N-[(1R)-1-[4-[6-[6-[1-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]pyrrolidin-3-yl]pyridin-3-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(C5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)C5)nc4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C47H53N11O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-2NQ14Y	SCHEMBL23983680	3-tert-butyl-N-[(1R)-1-[4-[6-[1-[1-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]pyrrolidin-3-yl]-3,5-dimethylpyrazol-4-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4c(C)nn(C5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)C5)c4C)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C47H56N12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-4A9ZIX	SCHEMBL25214806	3-tert-butyl-N-[(1R)-1-[4-[6-[4-[6-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]-2,6-diazaspiro[3.3]heptan-2-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CC6(CN(CC7CCN(c8ccc(N9CCC(=O)NC9=O)cc8)CC7)C6)C5)cc4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C49H55N11O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-YJCJ2W	SCHEMBL23983451	N-[(1R)-1-[4-[6-[5-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-2-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-3-(1-methylcyclopropyl)-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)cn4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C2(C)CC2)no1	C47H52N12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-AA4LRP	SCHEMBL25666897	N-[(1R)-1-[4-[6-[6-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-3-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-5-(1-methylcyclopropyl)-1,2,4-oxadiazole-3-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)nc4)cc23)ccc1[C@@H](C)NC(=O)c1noc(C2(C)CC2)n1	C47H52N12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-R6LQ04	WO2021219070A1_167	.	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)cc4)cc23)ccc1[C@@H](C)NC(=O)C1NC(C(C)(C)C)=NO1	C49H59N11O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-IKT03I	SCHEMBL23983452	3-tert-butyl-N-[(1R)-1-[4-[6-[2-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-1,3-thiazol-5-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4cnc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)s4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C45H52N12O4S	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-43DCVD	SCHEMBL23983455	3-tert-butyl-N-[(1R)-1-[4-[6-[1-[1-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]azetidin-3-yl]-3,5-dimethylpyrazol-4-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4c(C)nn(C5CN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)C5)c4C)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C46H54N12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-Z4M97M	SCHEMBL23983358	3-tert-butyl-N-[(1R)-1-[4-[6-[5-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-2-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-(hydroxymethyl)phenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	C[C@@H](NC(=O)c1nc(C(C)(C)C)no1)c1ccc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)cn4)cc23)cc1CO	C47H54N12O5	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-ENZJ8J	SCHEMBL25231211	5-tert-butyl-N-[(1R)-1-[4-[6-[5-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-2-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-5-fluoro-2-(hydroxymethyl)phenyl]ethyl]-1,2,4-oxadiazole-3-carboxamide	C[C@@H](NC(=O)c1noc(C(C)(C)C)n1)c1cc(F)c(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)cn4)cc23)cc1CO	C47H53FN12O5	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-LCRJN4	SCHEMBL23983407	3-tert-butyl-N-[(1R)-1-[4-[6-[5-[1-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]-3-hydroxyazetidin-3-yl]pyridin-2-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(C5(O)CN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)C5)cn4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C46H51N11O5	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-WVFTJ7	SCHEMBL23983476	3-tert-butyl-N-[(1R)-1-[4-[6-[5-[1-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]-3-fluoroazetidin-3-yl]pyridin-2-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(C5(F)CN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)C5)cn4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C46H50FN11O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-PCO0ML	SCHEMBL23983453	3-tert-butyl-N-[(1R)-1-[4-[6-[5-[1-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]-3,6-dihydro-2H-pyridin-4-yl]-1,4-dimethylpyrazol-3-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4nn(C)c(C5=CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)c4C)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C48H56N12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-G7EFQK	SCHEMBL23983478	3-tert-butyl-N-[(1R)-1-[4-[6-[1-[1-[2-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methylamino]ethyl]piperidin-4-yl]-3,5-dimethylpyrazol-4-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4c(C)nn(C5CCN(CCNCC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)c4C)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C50H63N13O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-OWOLRJ	SCHEMBL23984242	3-tert-butyl-N-[(1R)-1-[4-[6-[5-[1-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]pyrrolidin-3-yl]pyridin-2-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(C5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)C5)cn4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C47H53N11O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-YO76BA	SCHEMBL23983454	3-tert-butyl-N-[(1R)-1-[4-[6-[5-[1-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]-3-fluoropyrrolidin-3-yl]pyridin-2-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(C5(F)CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)C5)cn4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C47H52FN11O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-3PXEX0	SCHEMBL23984274	3-tert-butyl-N-[(1R)-1-[4-[6-[5-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-2-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-5-fluoro-2-(hydroxymethyl)phenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	C[C@@H](NC(=O)c1nc(C(C)(C)C)no1)c1cc(F)c(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)cn4)cc23)cc1CO	C47H53FN12O5	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-NARR5A	SCHEMBL23983369	3-tert-butyl-N-[(1R)-1-[4-[6-[6-[1-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]azetidin-3-yl]pyridin-3-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(C5CN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)C5)nc4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C46H51N11O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-9UFTSL	SCHEMBL23983447	3-tert-butyl-N-[(1R)-1-[4-[6-[5-[1-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]-3-hydroxypyrrolidin-3-yl]pyridin-2-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(C5(O)CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)C5)cn4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C47H53N11O5	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-18HX9Y	SCHEMBL23983449	3-tert-butyl-N-[(1R)-1-[4-[6-[5-[4-[[4-(2,6-dioxopiperidin-3-yl)-3-fluorophenyl]methyl]piperazin-1-yl]pyridin-2-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(Cc6ccc(C7CCC(=O)NC7=O)c(F)c6)CC5)cn4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C43H45FN10O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-W80D97	SCHEMBL23983367	3-tert-butyl-N-[(1R)-1-[4-[6-[4-[8-[[1-[5-(2,4-dioxo-1,3-diazinan-1-yl)pyridin-2-yl]piperidin-4-yl]methyl]-8-azabicyclo[3.2.1]octan-3-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(C5CC6CCC(C5)N6CC5CCN(c6ccc(N7CCC(=O)NC7=O)cn6)CC5)cc4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C50H57N11O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-KA8VUU	SCHEMBL23983752	3-tert-butyl-N-[(1R)-1-[4-[6-[4-[8-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]-8-azabicyclo[3.2.1]octan-3-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(C5CC6CCC(C5)N6CC5CCN(c6ccc(N7CCC(=O)NC7=O)cc6)CC5)cc4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C51H58N10O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-02UDT8	SCHEMBL23983400	3-tert-butyl-N-[(1R)-1-[4-[6-[5-[4-[[1-[4-(2,4-dioxoimidazolidin-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-2-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CC(=O)NC8=O)cc7)CC6)CC5)cn4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C46H52N12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-4HOBS2	SCHEMBL23984277	5-tert-butyl-N-[(1R)-1-[4-[6-[5-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-2-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,3,4-oxadiazole-2-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)cn4)cc23)ccc1[C@@H](C)NC(=O)c1nnc(C(C)(C)C)o1	C47H54N12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-9B9YA4	SCHEMBL23983669	3-tert-butyl-N-[(1R)-1-[4-[6-[5-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-1,3-thiazol-2-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ncc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)s4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C45H52N12O4S	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-BTKJ2F	SCHEMBL25201467	3-tert-butyl-N-[(1R)-1-[4-[6-[6-[4-[[1-[4-(2,4-dioxopyrimidin-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-3-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(-n8ccc(=O)[nH]c8=O)cc7)CC6)CC5)nc4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C47H52N12O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-ZY4C0S	SCHEMBL25243813	3-tert-butyl-N-[(1R)-1-[4-[6-[6-[4-[3-[4-[[(3S)-2,6-dioxopiperidin-3-yl]amino]phenyl]cyclobutyl]piperazin-1-yl]pyridin-3-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide; SCHEMBL25666947	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN([C@H]6C[C@@H](c7ccc(N[C@H]8CCC(=O)NC8=O)cc7)C6)CC5)nc4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C46H51N11O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-Z4VM2C	SCHEMBL25202308	3-tert-butyl-N-[(1R)-1-[4-[6-[6-[4-[3-[4-[[(3R)-2,6-dioxopiperidin-3-yl]amino]phenyl]cyclobutyl]piperazin-1-yl]pyridin-3-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide; SCHEMBL25666946	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(C6CC(c7ccc(N[C@@H]8CCC(=O)NC8=O)cc7)C6)CC5)nc4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C46H51N11O4	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-Q5I9XL	SCHEMBL23983410	3-tert-butyl-N-[(1R)-1-[4-[6-[4-[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]-3-oxopiperazin-1-yl]phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(CC6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)C(=O)C5)cc4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C48H53N11O5	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-C4ZQT3	SCHEMBL23983389	3-tert-butyl-N-[(1R)-1-[4-[6-[6-[4-[3-[4-[(3S)-2,6-dioxopiperidin-3-yl]oxyphenyl]cyclobutyl]piperazin-1-yl]pyridin-3-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide; SCHEMBL25205849	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN([C@H]6C[C@@H](c7ccc(O[C@H]8CCC(=O)NC8=O)cc7)C6)CC5)nc4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C46H50N10O5	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-T312UQ	SCHEMBL25202773	3-tert-butyl-N-[(1R)-1-[4-[6-[6-[4-[3-[4-[(3R)-2,6-dioxopiperidin-3-yl]oxyphenyl]cyclobutyl]piperazin-1-yl]pyridin-3-yl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2-methylphenyl]ethyl]-1,2,4-oxadiazole-5-carboxamide; SCHEMBL25666953	Cc1cc(-c2ncnc3[nH]c(-c4ccc(N5CCN(C6CC(c7ccc(O[C@@H]8CCC(=O)NC8=O)cc7)C6)CC5)nc4)cc23)ccc1[C@@H](C)NC(=O)c1nc(C(C)(C)C)no1	C46H50N10O5	BTK	Q06187	CRBN	WO-2021219070-A1
TPD-5EMBM9	WO2021219071A1_Compound2	.	CC1(C)Cc2cc3n(c2C1)CCN(c1cccc(-c2ncnc4[nH]c(-c5ccc(N6CCN(CC7CCN(c8ccc(N9CCC(=O)NC9=O)cc8)CC7)CC6)nc5)cc24)c1)C3=O	C49H53N11O3	BTK	Q06187	CRBN	WO-2021219071-A1
TPD-6XUDTL	WO2021222138A1_1	.	O=C1CCC(N2C(=O)c3cccc(NC(=O)CCCCCCCCCCC(=O)N4CCC(C(=O)NCCCn5cc(-c6ccc(OC(F)(F)F)cc6)c6cc(CN7CCN(Cc8c(Cl)cccc8Cl)CC7)ccc65)CC4)c3C2=O)C(=O)N1	C61H69Cl2F3N8O8	KRAS	P01116	CRBN	WO-2021222138-A1
TPD-C8KJ74	WO2021222138A1_2	.	O=C1CCC(N2C(=O)c3cccc(NCCOCCOCCOCCN4CCC(C(=O)NCCCn5cc(-c6ccc(OC(F)(F)F)cc6)c6cc(CN7CCN(Cc8c(Cl)cccc8Cl)CC7)ccc65)CC4)c3C2=O)C(=O)N1	C57H65Cl2F3N8O9	KRAS	P01116	CRBN	WO-2021222138-A1
TPD-S1755A	WO2021222138A1_3	.	O=C(COc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O)NCCCC(=O)N1CCC(C(=O)NCCCN2C=C(c3ccc(OC(F)(F)F)cc3)C3=CC(CN4CCN(Cc5c(Cl)cccc5Cl)CC4)=CCC32)CC1	C55H59Cl2F3N8O9	KRAS	P01116	CRBN	WO-2021222138-A1
TPD-N51DEA	WO2021222138A1_4	.	O=C1CCC(N2C(=O)c3cccc(NCCOCCOCCC(=O)N4CCC(C(=O)NCCCn5cc(-c6ccc(OC(F)(F)F)cc6)c6cc(CN7CCN(Cc8c(Cl)cccc8Cl)CC7)ccc65)CC4)c3C2=O)C(=O)N1	C56H61Cl2F3N8O9	KRAS	P01116	CRBN	WO-2021222138-A1
TPD-GPD14G	WO2021222138A1_5	.	O=C1CCC(N2C(=O)c3cccc(NCCOCCOCCOCCOCC(=O)N4CCC(C(=O)NCCCN5CC(c6ccc(OC(F)(F)F)cc6)c6cc(CN7CCN(Cc8c(Cl)cccc8Cl)CC7)ccc65)CC4)c3C2=O)C(=O)N1	C59H69Cl2F3N8O11	KRAS	P01116	CRBN	WO-2021222138-A1
TPD-ZOPZGL	WO2021222138A1_6	.	NC1(C(=O)NCCCN2CC(c3ccc(OC(F)(F)F)cc3)c3cc(CN4CCN(Cc5c(Cl)cccc5Cl)CC4)ccc32)CCN(C(=O)COCCOCCOCCOCCNc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)CC1	C59H70Cl2F3N9O11	KRAS	P01116	CRBN	WO-2021222138-A1
TPD-1S9TYI	WO2021222138A1_7	.	NC1(C(=O)NCCCn2cc(-c3ccc(OC(F)(F)F)cc3)c3cc(CN4CCN(Cc5c(Cl)cccc5Cl)CC4)ccc32)CCN(C(=O)CCOCCOCCOCCOCCNc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)CC1	C60H70Cl2F3N9O11	KRAS	P01116	CRBN	WO-2021222138-A1
TPD-GF5OKR	WO2021222138A1_8	.	NC1(C(=O)NCCCn2cc(-c3ccc(OC(F)(F)F)cc3)c3cc(CN4CCN(Cc5c(Cl)cccc5Cl)CC4)ccc32)CCN(C(=O)CCOCCOCCOCCNc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)CC1	C58H66Cl2F3N9O10	KRAS	P01116	CRBN	WO-2021222138-A1
TPD-OODL1J	WO2021222138A1_9	.	NC1(C(=O)NCCCn2cc(-c3ccc(OC(F)(F)F)cc3)c3cc(CN4CCN(Cc5c(Cl)cccc5Cl)CC4)ccc32)CCN(C(=O)CCOCCOCCOCCOCCOCCNc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)CC1	C62H74Cl2F3N9O12	KRAS	P01116	CRBN	WO-2021222138-A1
TPD-SUB8A7	WO2021222138A1_10	.	O=C1CCC(N2C(=O)c3cccc(NCCOCCOCCOCCOCC(=O)N4CCC(C(=O)NCCCn5cc(-c6ccccc6)c6cc(CN7CCN(Cc8c(Cl)cccc8Cl)CC7)ccc65)CC4)c3C2=O)C(=O)N1	C58H68Cl2N8O10	KRAS	P01116	CRBN	WO-2021222138-A1
TPD-7FUHFI	WO2021222138A1_11	.	O=C1CCC(N2C(=O)c3cccc(NCCOCCOCCOCCOCCOCCC(=O)N4CCC(C(=O)NCCCn5cc(-c6ccc(OC(F)(F)F)cc6)c6cc(CN7CCN(Cc8c(Cl)cccc8Cl)CC7)ccc65)CC4)c3C2=O)C(=O)N1	C62H73Cl2F3N8O12	KRAS	P01116	CRBN	WO-2021222138-A1
TPD-WRVXQ9	WO2021222138A1_12	.	O=C1CCC(N2C(=O)c3cccc(NCCOCCOCCOCCOCC(=O)NC4(C(=O)NCCCn5cc(-c6ccc(OC(F)(F)F)cc6)c6cc(CN7CCN(Cc8c(Cl)cccc8Cl)CC7)ccc65)CCNCC4)c3C2=O)C(=O)N1	C59H68Cl2F3N9O11	KRAS	P01116	CRBN	WO-2021222138-A1
TPD-Y3OM7A	WO2021222138A1_13	.	O=C(CCCNC(=O)COCCOCCOCCOCCNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O)NCCCn1cc(-c2ccc(OC(F)(F)F)cc2)c2cc(CN3CCN(Cc4c(Cl)cccc4Cl)CC3)ccc21	C57H65Cl2F3N8O11	KRAS	P01116	CRBN	WO-2021222138-A1
TPD-8BW6MX	WO2021222138A1_14	.	O=C1CCC(N2C(=O)c3cccc(NCCOCCOCCOCCOCC(=O)N4CCCC(C(=O)NCCCn5cc(-c6ccc(OC(F)(F)F)cc6)c6cc(CN7CCN(Cc8c(Cl)cccc8Cl)CC7)ccc65)C4)c3C2=O)C(=O)N1	C59H67Cl2F3N8O11	KRAS	P01116	CRBN	WO-2021222138-A1
TPD-Y2ZG9S	WO2021222138A1_15	.	O=C1CCC(N2C(=O)c3cccc(NCCOCCOCCOCCC(=O)N4CCC(C(=O)NCCCn5cc(-c6ccc(OC(F)(F)F)cc6)c6cc(CN7CCN(Cc8c(Cl)cccc8Cl)CC7)ccc65)CC4)c3C2=O)C(=O)N1	C58H65Cl2F3N8O10	KRAS	P01116	CRBN	WO-2021222138-A1
TPD-NEECDV	WO2021222138A1_16	.	O=C1CCC(N2C(=O)c3cccc(NCCOCCOCCOCCOCCC(=O)N4CCC(C(=O)NCCCn5cc(-c6ccc(OC(F)(F)F)cc6)c6cc(CN7CCN(Cc8c(Cl)cccc8Cl)CC7)ccc65)CC4)c3C2=O)C(=O)N1	C60H69Cl2F3N8O11	KRAS	P01116	CRBN	WO-2021222138-A1
TPD-2NQJ2K	WO2021222138A1_17	.	Cc1ncsc1-c1ccc(CNC(=O)[C@H]2C[C@H](O)CN2C(=O)C(NC(=O)CCOCCOCCOCCOCCC(=O)N2CCC(N)(C(=O)NCCCn3cc(-c4ccc(OC(F)(F)F)cc4)c4cc(CN5CCN(Cc6c(Cl)cccc6Cl)CC5)ccc43)CC2)C(C)(C)C)cc1	C70H89Cl2F3N10O11S	KRAS	P01116	CRBN	WO-2021222138-A1
TPD-CTUL0E	WO2021222138A1_18	.	Cc1cccc(Cl)c1CN1CCN(Cc2ccc3c(c2)c(-c2ccc(OC(F)(F)F)cc2)cn3CCCNC(=O)C2CCN(C(=O)CCOCCOCCOCCOCCC(=O)N[C@@H](C(=O)N3C[C@@H](O)C[C@@H]3C(=O)NCc3ccc(-c4scnc4C)cc3)C(C)(C)C)CC2)CC1	C71H91ClF3N9O11S	KRAS	P01116	VHL	WO-2021222138-A1
TPD-JJCGDY	WO2021222138A1_19	.	O=C1CCC(N2C(=O)c3cccc(NCCOCCOCCOCCOCC(=O)N4CCC(C(=O)NCCCn5cc(-c6ccc(OC(F)(F)F)cc6)c6cc(CN7CCC(NCc8c(Cl)cccc8Cl)CC7)ccc65)CC4)c3C2=O)C(=O)N1	C60H69Cl2F3N8O11	KRAS	P01116	CRBN	WO-2021222138-A1
TPD-2R0QSK	WO2021222138A1_20	.	CC1CN(Cc2c(Cl)cccc2Cl)CCN1Cc1ccc2c(c1)c(-c1ccc(OC(F)(F)F)cc1)cn2CCCNC(=O)C1CCN(C(=O)COCCOCCOCCOCCNc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)CC1	C60H69Cl2F3N8O11	KRAS	P01116	CRBN	WO-2021222138-A1
TPD-DCMN12	WO2021222138A1_21	.	O=C1CCC(N2C(=O)c3cccc(NCCOCCOCCOCCOCC(=O)N4CCCCC4C(=O)NCCCn4cc(-c5ccc(OC(F)(F)F)cc5)c5cc(CN6CCN(Cc7c(Cl)cccc7Cl)CC6)ccc54)c3C2=O)C(=O)N1	C59H67Cl2F3N8O11	KRAS	P01116	CRBN	WO-2021222138-A1
TPD-U06VKF	WO2021222138A1_22	.	O=C1CCC(N2C(=O)c3cccc(NCCOCCOCCOCCOCC(=O)N4CCCC4C(=O)NCCCn4cc(-c5ccc(OC(F)(F)F)cc5)c5cc(CN6CCN(Cc7c(Cl)cccc7Cl)CC6)ccc54)c3C2=O)C(=O)N1	C58H65Cl2F3N8O11	KRAS	P01116	CRBN	WO-2021222138-A1
TPD-V67H5Q	WO2021222138A1_23	.	CC1(C(=O)NCCCn2cc(-c3ccc(OC(F)(F)F)cc3)c3cc(CN4CCN(Cc5c(Cl)cccc5Cl)CC4)ccc32)CCN(C(=O)COCCOCCOCCOCCNc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)CC1	C60H69Cl2F3N8O11	KRAS	P01116	CRBN	WO-2021222138-A1
TPD-R4RZ61	WO2021222138A1_24	.	O=C1CCC(N2C(=O)c3cccc(NCCOCCOCCOCCOCC(=O)N4CCNC(C(=O)NCCCN5CC(c6ccc(OC(F)(F)F)cc6)c6cc(CN7CCN(Cc8c(Cl)cccc8Cl)CC7)ccc65)C4)c3C2=O)C(=O)N1	C58H68Cl2F3N9O11	KRAS	P01116	CRBN	WO-2021222138-A1
TPD-XK7VJM	WO2021222138A1_25	.	Cc1ncsc1-c1ccc(CNC(=O)C2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCOCCOCCOCCOCCC(O)N2CCCC(C(=O)NCCCn3cc(-c4ccc(OC(F)(F)F)cc4)c4cc(CN5CCN(C/C=C(Cl)/C=C\C=C\Cl)CC5)ccc43)C2)C(C)(C)C)cc1	C70H92Cl2F3N9O11S	KRAS	P01116	VHL	WO-2021222138-A1
TPD-Q5I6GZ	WO2021222138A1_26	.	Cc1ncsc1-c1ccc(CNC(=O)C2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCOCCOCCOCCOCCC(=O)N2CCCCC2C(=O)NCCCn2cc(-c3ccc(OC(F)(F)F)cc3)c3cc(CN4CCN(Cc5c(Cl)cccc5Cl)CC4)ccc32)C(C)(C)C)cc1	C70H88Cl2F3N9O11S	KRAS	P01116	VHL	WO-2021222138-A1
TPD-83MOGA	WO2021222138A1_27	.	O=C1CCC(N2C(=O)c3cccc(NCCOCCOCCOCCOCCC(=O)N4CCC(C(=O)NCCCN5CC(c6ccc(OC(F)(F)F)cc6)c6ccc(CN7CCN(Cc8c(Cl)cccc8Cl)CC7)cc65)CC4)c3C2=O)C(=O)N1	C60H71Cl2F3N8O11	KRAS	P01116	CRBN	WO-2021222138-A1
TPD-CJGDLS	WO2021222138A1_28	.	O=C1CCC(N2C(=O)c3cccc(NCCOCCOCCOCCOCCC(=O)N4CCC(C(=O)NCCCN5CC(c6ccc(OC(F)(F)F)cc6)c6cccc(CN7CCN(Cc8c(Cl)cccc8Cl)CC7)c65)CC4)c3C2=O)C(=O)N1	C60H71Cl2F3N8O11	KRAS	P01116	CRBN	WO-2021222138-A1
TPD-1KWEDG	WO2021222138A1_29	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCOCCOCCOCCOCCC(=O)N2CCC(C(=O)NCCCn3cc(-c4ccc(OC(F)(F)F)cc4)c4ccc(CN5CCN(Cc6c(Cl)cccc6Cl)CC5)cc43)CC2)C(C)(C)C)cc1	C70H88Cl2F3N9O11S	KRAS	P01116	VHL	WO-2021222138-A1
TPD-JT72JO	WO2021222138A1_30	.	Cc1ncsc1-c1ccc(CNC(=O)[C@H]2C[C@H](O)CN2C(=O)[C@H](NC(=O)CCOCCOCCOCCOCCC(=O)NCCCC(=O)NCCCn2cc(-c3ccc(OC(F)(F)F)cc3)c3cc(CN4CCN(Cc5c(Cl)cccc5Cl)CC4)ccc32)C(C)(C)C)cc1	C68H86Cl2F3N9O11S	KRAS	P01116	VHL	WO-2021222138-A1
TPD-CCW2J9	WO2021222138A1_31	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCOCCOCCOCCOCCC(=O)N2CCC(C(=O)NCCCn3cc(-c4ccc(OC(F)(F)F)cc4)c4cccc(CN5CCN(Cc6c(Cl)cccc6Cl)CC5)c43)CC2)C(C)(C)C)cc1	C70H88Cl2F3N9O11S	KRAS	P01116	VHL	WO-2021222138-A1
TPD-PMEM1C	WO2021222138A1_32	.	O=C1CCC(N2C(=O)c3cccc(NCCCCCCCCC(=O)N4CCC(C(=O)NCCCn5cc(-c6ccc(OC(F)(F)F)cc6)c6cc(CN7CCN(Cc8c(Cl)cccc8Cl)CC7)ccc65)CC4)c3C2=O)C(=O)N1	C58H65Cl2F3N8O7	KRAS	P01116	CRBN	WO-2021222138-A1
TPD-6QVQL3	WO2021222138A1_33	.	Cc1ncsc1-c1ccc(CNC(=O)[C@H]2C[C@H](O)CN2C(=O)C(NC(=O)CCCCCCCCCCC(=O)N2CCC(C(=O)NCCCn3cc(-c4ccc(OC(F)(F)F)cc4)c4cc(CN5CCN(Cc6c(Cl)cccc6Cl)CC5)ccc43)CC2)C(C)(C)C)cc1	C70H88Cl2F3N9O7S	KRAS	P01116	VHL	WO-2021222138-A1
TPD-NJVSP6	WO2021222138A1_34	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCOCCOCCOCCN2CCC(C(=O)NCCCn3cc(-c4ccc(OC(F)(F)F)cc4)c4cc(CN5CCN(Cc6c(Cl)cccc6Cl)CC5)ccc43)CC2)C(C)(C)C)cc1	C67H84Cl2F3N9O9S	KRAS	P01116	VHL	WO-2021222138-A1
TPD-22BSUD	WO2021222138A1_35	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCOCCN2CCC(C(=O)NCCCn3cc(-c4ccc(OC(F)(F)F)cc4)c4cc(CN5CCN(Cc6c(Cl)cccc6Cl)CC5)ccc43)CC2)C(C)(C)C)cc1	C63H76Cl2F3N9O7S	KRAS	P01116	VHL	WO-2021222138-A1
TPD-NC7GLU	WO2021222138A1_36	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@H](O)CN2C(=O)[C@@H](NC(=O)CN2CCN(CCCN3CCC(C(=O)NCCCn4cc(-c5ccc(OC(F)(F)F)cc5)c5cc(CN6CCN(Cc7c(Cl)cccc7Cl)CC6)ccc54)CC3)CC2)C(C)(C)C)cc1	C67H84Cl2F3N11O6S	KRAS	P01116	VHL	WO-2021222138-A1
TPD-U5RVH9	WO2021222138A1_37	.	O=C1CCC(N2C(=O)c3ccc(NCCOCCOCCOCCC(=O)N4CCC(C(=O)NCCCn5cc(-c6ccc(OC(F)(F)F)cc6)c6cc(CN7CCN(Cc8c(Cl)cccc8Cl)CC7)ccc65)CC4)cc3C2=O)C(=O)N1	C58H65Cl2F3N8O10	KRAS	P01116	CRBN	WO-2021222138-A1
TPD-26RW3U	WO2021222138A1_38	.	O=C1CCC(N2C(=O)c3ccc(NCCOCCOCCOCCOCCC(=O)N4CCC(C(=O)NCCCN5CC(c6ccc(OC(F)(F)F)cc6)c6cc(CN7CCN(Cc8c(Cl)cccc8Cl)CC7)ccc65)CC4)cc3C2=O)C(=O)N1	C60H71Cl2F3N8O11	KRAS	P01116	CRBN	WO-2021222138-A1
TPD-EEWWQ4	WO2021222138A1_39	.	O=C1CCC(N2Cc3c(NCCOCCOCCOCCOCCC(=O)N4CCC(C(=O)NCCCN5CC(C6C=CC(OC(F)(F)F)=CC6)c6cc(CN7CCN(Cc8c(Cl)cccc8Cl)CC7)ccc65)CC4)cccc3C2=O)C(=O)N1	C60H75Cl2F3N8O10	KRAS	P01116	CRBN	WO-2021222138-A1
TPD-ANZVDF	WO2021222138A1_40	.	NC1(C(=O)NCCCn2cc(-c3ccc(OC(F)(F)F)cc3)c3cc(CN4CCN(Cc5c(Cl)cccc5Cl)CC4)ccc32)CCN(C(=O)CCOCCOCCOCCOCCNc2cccc3c2CN(C2CCC(=O)NC2=O)C3=O)CC1	C60H72Cl2F3N9O10	KRAS	P01116	CRBN	WO-2021222138-A1
TPD-45SS23	WO2021222138A1_41	.	O=C(COc1ccc2c(c1)CCCN2C(=O)CCl)NCCOCCOCCOCCOCCC(=O)N1CCC(C(=O)NCCCNc2ccc(CN3CCN(Cc4c(Cl)cccc4Cl)CC3)cc2Cc2ccc(OC(F)(F)F)cc2)CC1	C59H75Cl3F3N7O10	KRAS	P01116	CRBN	WO-2021222138-A1
TPD-XG31K2	WO2021222138A1_42	.	O=C(COc1ccc2c(c1)CCCN2C(=O)CCl)NCCOCCOCCOCCOCCOCCC(=O)N1CCC(C(=O)NCCCn2cc(-c3ccc(OC(F)(F)F)cc3)c3cc(CN4CCN(Cc5c(Cl)cccc5Cl)CC4)ccc32)CC1	C62H77Cl3F3N7O11	KRAS	P01116	CRBN	WO-2021222138-A1
TPD-YEKK2E	WO2021222138A1_43	.	NC1(C(=O)NCCCn2cc(-c3ccc(OC(F)(F)F)cc3)c3cc(CN4CCN(Cc5c(Cl)cccc5Cl)CC4)ccc32)CCN(C(=O)CCOCCOCCOCCOCCNC(=O)COc2ccc3c(c2)CCCN3C(=O)CCl)CC1	C60H74Cl3F3N8O10	KRAS	P01116	CRBN	WO-2021222138-A1
TPD-HS38LP	WO2021222138A1_44	.	O=C(COc1ccc2c(c1)CCCN2C(=O)CCl)NCCOCCOCCOCCC(=O)N1CCC(C(=O)NCCCn2cc(-c3ccc(OC(F)(F)F)cc3)c3cc(CN4CCN(Cc5c(Cl)cccc5Cl)CC4)ccc32)CC1	C58H69Cl3F3N7O9	KRAS	P01116	CRBN	WO-2021222138-A1
TPD-ECFKEG	WO2021222138A1_45	.	NC1(C(=O)NCCCn2cc(-c3ccc(OC(F)(F)F)cc3)c3cc(CN4CCN(Cc5c(Cl)cccc5Cl)CC4)ccc32)CCN(C(=O)CCOCCOCCOCCNC(=O)COc2ccc3c(c2)CCCN3C(=O)CCl)CC1	C58H70Cl3F3N8O9	KRAS	P01116	CRBN	WO-2021222138-A1
TPD-2S4QI4	WO2021222138A1_46	.	NC1(C(=C=O)NCCCn2cc(-c3ccc(OC(F)(F)F)cc3)c3cc(CN4CCN(Cc5c(Cl)cccc5Cl)CC4)ccc32)CCN(C(=O)COc2ccc3c(c2)CCCN3C(=O)CCl)CC1	C50H53Cl3F3N7O5	KRAS	P01116	CRBN	WO-2021222138-A1
TPD-DFPT5G	SCHEMBL24031529	2-chloro-4-[3-[6-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-7,8-dihydro-5H-pyrrolo[3,4-g]isoquinolin-6-yl]-2-oxoethyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC(Cl)=C(C#N)C=C2)C(C)(C)[C@H]1N1CC2=C(C=CC(N3CCN(CC(=O)N4CCC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)=C2)C1=O	C45H46ClN7O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-26VRBT	SCHEMBL24031538	2-chloro-4-[3-[6-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]-2-oxoethyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC(Cl)=C(C#N)C=C2)C(C)(C)[C@H]1N1CC2=C(C=CC(N3CCN(CC(=O)N4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)=C2)C1=O	C44H44ClN7O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-ZH0XLP	SCHEMBL24031533	2-chloro-4-[4-[6-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-7,8-dihydro-5H-pyrrolo[3,4-g]isoquinolin-6-yl]-2-oxoethyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]cyclohexyl]oxybenzonitrile	N#CC1=C(Cl)C=C(O[C@H]2CC[C@H](N3CC4=C(C=CC(N5CCN(CC(=O)N6CCC7=C(C=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)C6)CC5)=C4)C3=O)CC2)C=C1	C43H42ClN7O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-K1WMAH	SCHEMBL24031530	2-chloro-4-[4-[6-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]-2-oxoethyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]cyclohexyl]oxybenzonitrile	N#CC1=C(Cl)C=C(O[C@H]2CC[C@H](N3CC4=C(C=CC(N5CCN(CC(=O)N6CC7=C(C=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)C6)CC5)=C4)C3=O)CC2)C=C1	C42H40ClN7O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-UYPSXG	SCHEMBL24031924	2-chloro-4-[3-[6-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]piperidine-1-carbonyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC(Cl)=C(C#N)C=C2)C(C)(C)[C@H]1N1CC2=CC(C(=O)N3CCC(N4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)=CC=C2C1=O	C44H43ClN6O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-KS4M34	SCHEMBL26801952	2-chloro-4-[3-[6-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidine-1-carbonyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC(Cl)=C(C#N)C=C2)C(C)(C)[C@H]1N1CC2=CC(C(=O)N3CCC(CN4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)=CC=C2C1=O	C45H45ClN6O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-AKB3B0	SCHEMBL26801954	2-chloro-4-[3-[6-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]ethyl]piperidine-1-carbonyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC(Cl)=C(C#N)C=C2)C(C)(C)[C@H]1N1CC2=CC(C(=O)N3CCC(CCN4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)=CC=C2C1=O	C46H47ClN6O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-8237LF	SCHEMBL26801957	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]benzamide	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=CC=C(N4CCC(CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C3)CC2)C=C1Cl	C41H41ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-OLAGO1	SCHEMBL26801961	2-Chloro-4-[4-[4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidine-1-carbonyl]anilino]cyclohexyl]oxybenzonitrile	N#CC1=CC=C(O[C@H]2CC[C@H](NC3=CC=C(C(=O)N4CCC(CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C3)CC2)C=C1Cl	C41H41ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-96MJNA	WO2021231927A1_10	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC3=CC=C(C(=O)N4CCC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C3)CC2)C=C1Cl	C40H39ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-TQV9S1	SCHEMBL24031729	2-Chloro-4-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]piperidine-1-carbonyl]phenoxy]cyclohexyl]oxybenzonitrile	N#CC1=CC=C(O[C@H]2CC[C@H](OC3=CC=C(C(=O)N4CCC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C3)CC2)C=C1Cl	C40H38ClN5O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-3528SC	WO2021231927A1_12	.	N#CC1=CC=C(O[C@H]2CC[C@H](OC3=CC=C(C(=O)N4CCC(CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C3)CC2)C=C1Cl	C41H40ClN5O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-O68RDE	WO2021231927A1_13	.	C[C@H]1C[C@H](NC(=O)C2=CC=C(N3CCC(N4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=C2)CC[C@H]1CC1=CC=C(C#N)C(Cl)=C1	C42H43ClN6O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-T0D6JP	SCHEMBL24031728	N-[(1R,3S,4R)-4-(3-chloro-4-cyanophenoxy)-3-methylcyclohexyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]benzamide	C[C@H]1C[C@H](NC(=O)C2=CC=C(N3CCC(CN4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=C2)CC[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C42H43ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-DMT53O	WO2021231927A1_15	.	C[C@H]1C[C@@H](NC(=O)C2=CC=C(N3CCC(CN4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=C2)CC[C@@H]1OC1=CC=C(C#N)C(Cl)=C1	C42H43ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-U8E4CR	WO2021231927A1_16	.	C[C@H]1C[C@@H](NC(=O)C2=CC=C(N3CCC(N4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=C2)CC[C@@H]1OC1=CC=C(C#N)C(Cl)=C1	C41H41ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-Q71E9X	WO2021231927A1_17	.	N#CC1=CC=C(N[C@H]2CC[C@H](NC(=O)C3=CC=C(N4CCC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C3)CC2)C=C1Cl	C40H40ClN7O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-JDIA8J	WO2021231927A1_18	.	N#CC1=CC=C(N[C@H]2CC[C@H](NC(=O)C3=CC=C(N4CCC(CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C3)CC2)C=C1Cl	C41H42ClN7O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-3GOXEE	SCHEMBL30690849	N-[4-(3-chloro-4-cyano-N-methylanilino)cyclohexyl]-4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]piperidin-1-yl]benzamide	CN(C1=CC=C(C#N)C(Cl)=C1)C1CCC(NC(=O)C2=CC=C(N3CCC(N4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=C2)CC1	C41H42ClN7O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-4GLPP6	SCHEMBL23051559	N-[4-(3-chloro-4-cyano-N-methylanilino)cyclohexyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]benzamide; SCHEMBL26667228; SCHEMBL29760409	CN(C1=CC=C(C#N)C(Cl)=C1)[C@H]1CC[C@H](NC(=O)C2=CC=C(N3CCC(CN4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=C2)CC1	C42H44ClN7O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-BGL4DB	WO2021231927A1_21	.	N#CC1=C(Cl)C=C(O[C@H]2CC[C@H](NC(=O)C3=CC=C(N4CC(CN5CC6=CC7=C(C=C6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C4)C=C3)CC2)C=C1	C39H37ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-MRSA7J	SCHEMBL24031624	N-[4-(3-chloro-4-cyanoanilino)cyclohexyl]-4-[3-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]azetidin-1-yl]benzamide	N#CC1=C(Cl)C=C(N[C@H]2CC[C@H](NC(=O)C3=CC=C(N4CC(CN5CC6=CC7=C(C=C6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C4)C=C3)CC2)C=C1	C39H38ClN7O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-12IWBC	WO2021231927A1_23	.	CC1=C(Cl)C=C(N(C)[C@H]2CC[C@H](NC(=O)C3=CC=C(N4CC(CN5CC6=CC7=C(C=C6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C4)C=C3)CC2)C=C1	C40H43ClN6O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-RML06U	SCHEMBL24031875	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]acetyl]-3,4-dihydro-1H-isoquinoline-6-carboxamide	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=CC=C4CN(C(=O)CN5CC6=CC7=C(C=C6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CCC4=C3)CC2)C=C1Cl	C40H37ClN6O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-59YST6	WO2021231927A1_25	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=CC=C4CCN(C(=O)CN5CC6=CC7=C(C=C6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CCC4=C3)CC2)C=C1Cl	C41H39ClN6O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-0B67MC	WO2021231927A1_26	.	N#CC1=CC=C(N2CC[C@H]3C[C@H](NC(=O)C4=CC=C(N5CCC(CN6CC7=C(C=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)C6)CC5)C=C4)CC[C@H]32)C=C1Cl	C43H44ClN7O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-OVTIBW	WO2021231927A1_27	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=CC=C4CN(CC(=O)N5CC6=CC7=C(C=C6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CCC4=C3)CC2)C=C1Cl	C40H37ClN6O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-NEVVR4	SCHEMBL24031528	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-7,8-dihydro-5H-pyrrolo[3,4-g]isoquinolin-6-yl]-2-oxoethyl]-3,4-dihydro-1H-isoquinoline-6-carboxamide	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=CC=C4CN(CC(=O)N5CCC6=CC7=C(C=C6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CCC4=C3)CC2)C=C1Cl	C41H39ClN6O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-6TAO0V	WO2021231927A1_29	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=CC=C4CCN(CC(=O)N5CCC6=CC7=C(C=C6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CCC4=C3)CC2)C=C1Cl	C42H41ClN6O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-Y6LOYZ	SCHEMBL26806922	N-[4-(3-chloro-4-cyano-N-methylanilino)cyclohexyl]-2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]acetyl]-3,4-dihydro-1H-isoquinoline-6-carboxamide	CN(C1=CC=C(C#N)C(Cl)=C1)[C@H]1CC[C@H](NC(=O)C2=CC3=C(C=C2)CN(C(=O)CN2CC4=CC5=C(C=C4C2)C(=O)N(C2CCC(=O)NC2=O)C5=O)CC3)CC1	C41H40ClN7O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-8CSAYW	SCHEMBL26807006	N-[4-(3-chloro-4-cyanoanilino)cyclohexyl]-2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]acetyl]-3,4-dihydro-1H-isoquinoline-6-carboxamide	N#CC1=CC=C(N[C@H]2CC[C@H](NC(=O)C3=CC4=C(C=C3)CN(C(=O)CN3CC5=CC6=C(C=C5C3)C(=O)N(C3CCC(=O)NC3=O)C6=O)CC4)CC2)C=C1Cl	C40H38ClN7O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-UQSCLA	SCHEMBL24031414	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]acetyl]-1,3-dihydroisoindole-5-carboxamide	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=CC4=C(C=C3)CN(C(=O)CN3CC5=CC6=C(C=C5C3)C(=O)N(C3CCC(=O)NC3=O)C6=O)C4)CC2)C=C1Cl	C39H35ClN6O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-LJ7HGR	WO2021231927A1_33	.	CN(C1=CC=C(C#N)C(Cl)=C1)[C@H]1CC[C@H](NC(=O)C2=CC3=C(C=C2)CN(C(=O)CN2CC4=CC5=C(C=C4C2)C(=O)N(C2CCC(=O)NC2=O)C5=O)C3)CC1	C40H38ClN7O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-8FJFQW	WO2021231927A1_35	.	CC1(C)[C@H](NC(=O)C2=CC=C(C#CC34CCC(CN5CC6=CC7=C(C=C6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)(CC3)CC4)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C48H48ClN5O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-B29L9I	SCHEMBL24031531	2-Chloro-4-[1-[[4-[2-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]-1-bicyclo[2.2.2]octanyl]ethynyl]phenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile	CC1=C(C)N(CC2=CC=C(C#CC34CCC(CN5CC6=CC7=C(C=C6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)(CC3)CC4)C=C2)N=C1C1=CC=C(C#N)C(Cl)=C1	C45H41ClN6O4	AR	P10275	CRBN	WO-2021231927-A1
TPD-OQVCFO	SCHEMBL24031532	2-Chloro-4-[[8-[4-[2-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]cyclohexyl]ethynyl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzonitrile	[H]C1(OC2=CC=C(C#N)C(Cl)=C2)CC2CCC(C1)N2C(=O)C1=CC=C(C#C[C@H]2CC[C@H](CN3CC4=CC5=C(C=C4C3)C(=O)N(C3CCC(=O)NC3=O)C5=O)CC2)C=C1	C45H42ClN5O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-WAY7JR	SCHEMBL24031626	2-Chloro-4-[[8-[4-[2-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]-1-bicyclo[2.2.2]octanyl]ethynyl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzonitrile	[H]C1(OC2=CC=C(C#N)C(Cl)=C2)CC2CCC(C1)N2C(=O)C1=CC=C(C#CC23CCC(CN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)(CC2)CC3)C=C1	C47H44ClN5O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-YT6E3N	SCHEMBL24031623	2-Chloro-4-[1-[4-[2-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]-1-bicyclo[2.2.2]octanyl]ethynyl]benzoyl]piperidin-4-yl]oxybenzonitrile	N#CC1=C(Cl)C=C(OC2CCN(C(=O)C3=CC=C(C#CC45CCC(CN6CC7=CC8=C(C=C7C6)C(=O)N(C6CCC(=O)NC6=O)C8=O)(CC4)CC5)C=C3)CC2)C=C1	C45H42ClN5O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-P7SJSH	SCHEMBL24031625	2-chloro-4-[1-[4-[2-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-7,8-dihydro-5H-pyrrolo[3,4-g]isoquinolin-6-yl]methyl]-1-bicyclo[2.2.2]octanyl]ethynyl]benzoyl]piperidin-4-yl]oxybenzonitrile	N#CC1=C(Cl)C=C(OC2CCN(C(=O)C3=CC=C(C#CC45CCC(CN6CCC7=CC8=C(C=C7C6)C(=O)N(C6CCC(=O)NC6=O)C8=O)(CC4)CC5)C=C3)CC2)C=C1	C46H44ClN5O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-KMWL2F	SCHEMBL24031627	2-Chloro-4-[1-[[4-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindole-6-carbonyl]cyclohexyl]ethynyl]phenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile	CC1=C(C)N(CC2=CC=C(C#C[C@H]3CC[C@H](C(=O)N4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=C2)N=C1C1=CC(Cl)=C(C#N)C=C1	C43H37ClN6O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-43PXDH	SCHEMBL24031635	2-chloro-4-[1-[[4-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-7,8-dihydro-5H-pyrrolo[3,4-g]isoquinoline-6-carbonyl]cyclohexyl]ethynyl]phenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile	CC1=C(C)N(CC2=CC=C(C#C[C@H]3CC[C@H](C(=O)N4CCC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=C2)N=C1C1=CC(Cl)=C(C#N)C=C1	C44H39ClN6O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-586T1C	SCHEMBL24031643	2-Chloro-4-[[8-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]piperidine-1-carbonyl]phenyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzonitrile	[H]C1(OC2=CC=C(C#N)C(Cl)=C2)CC2CCC(C1)N2C1=CC=C(C(=O)N2CCC(N3CC4=CC5=C(C=C4C3)C(=O)N(C3CCC(=O)NC3=O)C5=O)CC2)C=C1	C41H39ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-UHGR9J	SCHEMBL24031632	2-Chloro-4-[[8-[4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidine-1-carbonyl]phenyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzonitrile	[H]C1(OC2=CC=C(C#N)C(Cl)=C2)CC2CCC(C1)N2C1=CC=C(C(=O)N2CCC(CN3CC4=CC5=C(C=C4C3)C(=O)N(C3CCC(=O)NC3=O)C5=O)CC2)C=C1	C42H41ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-9A3847	SCHEMBL24031633	2-chloro-4-[1-[4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-7,8-dihydro-5H-pyrrolo[3,4-g]isoquinolin-6-yl]methyl]piperidine-1-carbonyl]phenyl]piperidin-4-yl]oxybenzonitrile	N#CC1=CC=C(OC2CCN(C3=CC=C(C(=O)N4CCC(CN5CCC6=CC7=C(C=C6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)C=C3)CC2)C=C1Cl	C41H41ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-A4O36O	SCHEMBL24031943	2-Chloro-4-[1-[[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]piperidine-1-carbonyl]phenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile	CC1=C(C)N(CC2=CC=C(C(=O)N3CCC(N4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)N=C1C1=CC(Cl)=C(C#N)C=C1	C40H36ClN7O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-NCFB3R	SCHEMBL24031944	2-Chloro-4-[1-[[4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidine-1-carbonyl]phenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile	CC1=C(C)N(CC2=CC=C(C(=O)N3CCC(CN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)N=C1C1=CC(Cl)=C(C#N)C=C1	C41H38ClN7O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-U7ZS6X	SCHEMBL24031942	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-6-yl]methyl]piperidine-1-carbonyl]benzamide	CC1(C)[C@H](NC(=O)C2=CC=C(C(=O)N3CCC(CN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C44H47ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-VHBV1G	WO2021231927A1_49	.	CC1(C)[C@H](NC(=O)C2=CC=C(C(=O)N3CC4(CC(CN5CC6=CC7=C(C=C6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C4)C3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C45H45ClN6O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-QSAK5C	SCHEMBL24031817	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[3-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]azetidine-1-carbonyl]benzamide	CC1(C)[C@H](NC(=O)C2=CC=C(C(=O)N3CC(CN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)C3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C42H41ClN6O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-2D9N12	SCHEMBL24031355	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]benzamide	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(CN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C43H45ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-52P67D	SCHEMBL24031947	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]ethyl]piperidin-1-yl]benzamide	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(CCN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C44H47ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-TZ3ECS	WO2021231927A1_53	.	CC1(C)[C@H](NC2=CC=C(C(=O)N3CCC(N4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C42H43ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-J68VB6	WO2021231927A1_54	.	CC1(C)[C@H](NC2=CC=C(C(=O)N3CCC(CN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C43H45ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-D6D48I	SCHEMBL24031946	2-Chloro-4-[1-[[4-[4-[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]azetidin-1-yl]piperidine-1-carbonyl]phenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile	CC1=C(C)N(CC2=CC=C(C(=O)N3CCC(N4CC(N5CC6=CC7=C(C=C6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C4)CC3)C=C2)N=C1C1=CC(Cl)=C(C#N)C=C1	C43H41ClN8O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-1PZ2BQ	SCHEMBL24031448	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]azetidin-1-yl]piperidin-1-yl]benzamide	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(N4CC(N5CC6=CC7=C(C=C6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C4)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C45H48ClN7O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-F4VHIP	SCHEMBL24031454	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]piperidin-1-yl]benzamide; SCHEMBL26667226	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(N4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C42H43ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-Q7GVGS	SCHEMBL24031449	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-6-yl]piperidin-1-yl]benzamide	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(N4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C42H45ClN6O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-B26S1E	SCHEMBL24031459	N-[3-(3-chloro-4-cyanophenoxy)cyclobutyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidine-1-carbonyl]benzamide	N#CC1=CC=C(O[C@H]2C[C@H](NC(=O)C3=CC=C(C(=O)N4CCC(CN5CC6=CC7=C(C=C6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)C=C3)C2)C=C1Cl	C40H37ClN6O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-A6YSB5	SCHEMBL24031456	N-[3-(3-chloro-4-cyanophenoxy)cyclobutyl]-4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]piperidin-1-yl]benzamide	N#CC1=CC=C(O[C@H]2C[C@H](NC(=O)C3=CC=C(N4CCC(N5CC6=CC7=C(C=C6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)C=C3)C2)C=C1Cl	C38H35ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-I8CRXU	SCHEMBL24031460	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidine-1-carbonyl]bicyclo[2.2.2]octane-1-carboxamide; SCHEMBL26667221	CC1(C)[C@H](NC(=O)C23CCC(C(=O)N4CCC(CN5CC6=CC7=C(C=C6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)(CC2)CC3)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C46H53ClN6O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-NHNJL4	SCHEMBL24031451	2-chloro-4-[(3R)-1-[4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidine-1-carbonyl]benzoyl]-2,2-dimethylazetidin-3-yl]oxybenzonitrile	CC1(C)[C@H](OC2=CC(Cl)=C(C#N)C=C2)CN1C(=O)C1=CC=C(C(=O)N2CCC(CN3CC4=CC5=C(C=C4C3)C(=O)N(C3CCC(=O)NC3=O)C5=O)CC2)C=C1	C41H39ClN6O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-DUJA1L	SCHEMBL24031453	2-chloro-4-[(3S)-1-[4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidine-1-carbonyl]benzoyl]-2,2-dimethylazetidin-3-yl]oxybenzonitrile	CC1(C)[C@@H](OC2=CC(Cl)=C(C#N)C=C2)CN1C(=O)C1=CC=C(C(=O)N2CCC(CN3CC4=CC5=C(C=C4C3)C(=O)N(C3CCC(=O)NC3=O)C5=O)CC2)C=C1	C41H39ClN6O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-JRZLL5	SCHEMBL24031457	2-chloro-4-[(3R)-1-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]piperidin-1-yl]benzoyl]-2,2-dimethylazetidin-3-yl]oxybenzonitrile	CC1(C)[C@H](OC2=CC(Cl)=C(C#N)C=C2)CN1C(=O)C1=CC=C(N2CCC(N3CC4=CC5=C(C=C4C3)C(=O)N(C3CCC(=O)NC3=O)C5=O)CC2)C=C1	C39H37ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-88JFCT	SCHEMBL24031458	2-chloro-4-[(3S)-1-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]piperidin-1-yl]benzoyl]-2,2-dimethylazetidin-3-yl]oxybenzonitrile	CC1(C)[C@@H](OC2=CC(Cl)=C(C#N)C=C2)CN1C(=O)C1=CC=C(N2CCC(N3CC4=CC5=C(C=C4C3)C(=O)N(C3CCC(=O)NC3=O)C5=O)CC2)C=C1	C39H37ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-PKH1SZ	WO2021231927A1_66	.	N#CC1=CC=C(O[C@H]2C[C@H](NC(=O)C3=CC=C(N4CCC(CN5CC6=CC7=C(C=C6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)C=C3)C2)C=C1Cl	C39H37ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-W4WZPJ	WO2021231927A1_67	.	N#CC1=CC=C(O[C@H]2C[C@H](NC(=O)C3=CC=C(N4CCC(CN5CC6=CC7=C(C=C6C5)C(=O)N(C5CCC(=O)NC5=O)C7)CC4)C=C3)C2)C=C1Cl	C39H39ClN6O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-7WURW6	SCHEMBL24031758	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]benzamide; SCHEMBL26667219	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(CN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C43H47ClN6O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-979398	SCHEMBL24031293	2-chloro-4-[(3S)-1-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-6-yl]piperidin-1-yl]benzoyl]-2,2-dimethylazetidin-3-yl]oxybenzonitrile	CC1(C)[C@@H](OC2=CC(Cl)=C(C#N)C=C2)CN1C(=O)C1=CC=C(N2CCC(N3CC4=CC5=C(C=C4C3)C(=O)N(C3CCC(=O)NC3=O)C5)CC2)C=C1	C39H39ClN6O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-XSBODQ	SCHEMBL24031290	2-chloro-4-[(3S)-1-[4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]benzoyl]-2,2-dimethylazetidin-3-yl]oxybenzonitrile	CC1(C)[C@@H](OC2=CC(Cl)=C(C#N)C=C2)CN1C(=O)C1=CC=C(N2CCC(CN3CC4=CC5=C(C=C4C3)C(=O)N(C3CCC(=O)NC3=O)C5)CC2)C=C1	C40H41ClN6O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-L133E4	SCHEMBL24031617	2-chloro-4-[(3S)-1-[4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]benzoyl]-2,2-dimethylazetidin-3-yl]oxybenzonitrile	CC1(C)[C@@H](OC2=CC(Cl)=C(C#N)C=C2)CN1C(=O)C1=CC=C(N2CCC(CN3CC4=CC5=C(C=C4C3)C(=O)N(C3CCC(=O)NC3=O)C5=O)CC2)C=C1	C40H39ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-09V8S4	WO2021231927A1_72	.	CC1(C)[C@H](NC(=O)C23CCC(C(=O)N4CCC(CN5CC6=CC7=C(C=C6C5)C(=O)N(C5CCC(=O)NC5=O)C7)CC4)(CC2)CC3)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C46H55ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-5R75SZ	SCHEMBL24031295	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]piperidine-1-carbonyl]bicyclo[2.2.2]octane-1-carboxamide	CC1(C)[C@H](NC(=O)C23CCC(C(=O)N4CCC(N5CC6=CC7=C(C=C6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)(CC2)CC3)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C45H51ClN6O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-059Y5D	SCHEMBL24031292	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-6-yl]piperidine-1-carbonyl]bicyclo[2.2.2]octane-1-carboxamide	CC1(C)[C@H](NC(=O)C23CCC(C(=O)N4CCC(N5CC6=CC7=C(C=C6C5)C(=O)N(C5CCC(=O)NC5=O)C7)CC4)(CC2)CC3)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C45H53ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-WC2976	SCHEMBL24031926	2-Chloro-4-[3-[[4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidine-1-carbonyl]cyclohexyl]amino]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](N[C@H]2CC[C@H](C(=O)N3CCC(CN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)CC2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C43H51ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-CZ49WH	SCHEMBL24031925	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]cyclohexane-1-carboxamide	CC1(C)[C@H](NC(=O)[C@H]2CC[C@H](N3CCC(CN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)CC2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C43H51ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-6N4DOH	SCHEMBL24031615	N-[(1S,3S)-3-(3-chloro-4-cyanophenoxy)-2,2-dimethylcyclobutyl]-4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]piperidin-1-yl]benzamide	CC1(C)[C@@H](NC(=O)C2=CC=C(N3CCC(N4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C[C@@H]1OC1=CC=C(C#N)C(Cl)=C1	C40H39ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-O6UTMW	SCHEMBL24031844	N-[(1S,3S)-3-(3-chloro-4-cyanophenoxy)-2,2-dimethylcyclobutyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]benzamide	CC1(C)[C@@H](NC(=O)C2=CC=C(N3CCC(CN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C[C@@H]1OC1=CC=C(C#N)C(Cl)=C1	C41H41ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-FDCWNM	SCHEMBL24031927	N-[(1S,3S)-3-(3-chloro-4-cyanophenoxy)-2,2-dimethylcyclobutyl]-4-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-6-yl]piperidin-1-yl]benzamide	CC1(C)[C@@H](NC(=O)C2=CC=C(N3CCC(N4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6)CC3)C=C2)C[C@@H]1OC1=CC=C(C#N)C(Cl)=C1	C40H41ClN6O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-YJAE8Q	WO2021231927A1_80	N-[(1S,3S)-3-(3-chloro-4-cyanophenoxy)-2,2-dimethylcyclobutyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]benzamide	CC1(C)[C@@H](NC(=O)C2=CC=C(N3CCC(CN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6)CC3)C=C2)C[C@@H]1OC1=CC=C(C#N)C(Cl)=C1	C41H43ClN6O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-AYPOQT	WO2021231927A1_81	.	CC1(C)[C@H](OC2=CC=C(C(=O)N3CCC(CN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C43H44ClN5O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-KGXDQS	WO2021231927A1_82	.	CC1(C)[C@H](OC2=CC=C(C(=O)N3CCC(N4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C42H42ClN5O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-EXL9LW	WO2021231927A1_83	2-chloro-4-[(1S,3S)-3-[4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidine-1-carbonyl]phenoxy]-2,2-dimethylcyclobutyl]oxybenzonitrile	CC1(C)[C@@H](OC2=CC=C(C(=O)N3CCC(CN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C[C@@H]1OC1=CC=C(C#N)C(Cl)=C1	C41H40ClN5O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-IEAPRZ	WO2021231927A1_84	2-chloro-4-[(1S,3S)-3-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]piperidine-1-carbonyl]phenoxy]-2,2-dimethylcyclobutyl]oxybenzonitrile	CC1(C)[C@@H](OC2=CC=C(C(=O)N3CCC(N4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C[C@@H]1OC1=CC=C(C#N)C(Cl)=C1	C40H38ClN5O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-W8WLG6	SCHEMBL24031604	N-[(1S,3S)-3-(3-chloro-4-cyanophenoxy)cyclopentyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]benzamide	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=CC=C(N4CCC(CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C3)C2)C=C1Cl	C40H39ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-HBZCPV	SCHEMBL24031722	N-[(1R,3R)-3-(3-chloro-4-cyanophenoxy)cyclopentyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]benzamide	N#CC1=CC=C(O[C@@H]2CC[C@@H](NC(=O)C3=CC=C(N4CCC(CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C3)C2)C=C1Cl	C40H39ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-Z5VMPX	SCHEMBL24031723	N-[(1S,3S)-3-(3-chloro-4-cyanophenoxy)cyclohexyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]benzamide	N#CC1=CC=C(O[C@H]2CCC[C@H](NC(=O)C3=CC=C(N4CCC(CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C3)C2)C=C1Cl	C41H41ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-KM5RS8	SCHEMBL24031724	N-[(1R,3R)-3-(3-chloro-4-cyanophenoxy)cyclohexyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]benzamide	N#CC1=CC=C(O[C@@H]2CCC[C@@H](NC(=O)C3=CC=C(N4CCC(CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C3)C2)C=C1Cl	C41H41ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-ANGGXN	SCHEMBL23051611	N-[4-(3-chloro-4-cyanophenoxy)-1-bicyclo[2.2.2]octanyl]-4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]piperidin-1-yl]benzamide; SCHEMBL29707028	N#CC1=CC=C(OC23CCC(NC(=O)C4=CC=C(N5CCC(N6CC7=C(C=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)C6)CC5)C=C4)(CC2)CC3)C=C1Cl	C42H41ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-W8QDAR	SCHEMBL24031725	N-[4-(3-chloro-4-cyanophenoxy)-1-bicyclo[2.2.1]heptanyl]-4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]piperidin-1-yl]benzamide	N#CC1=CC=C(OC23CCC(NC(=O)C4=CC=C(N5CCC(N6CC7=C(C=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)C6)CC5)C=C4)(CC2)C3)C=C1Cl	C41H39ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-IM8HJR	SCHEMBL24031721	N-[4-(3-chloro-4-cyanophenoxy)-1-bicyclo[2.2.1]heptanyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]benzamide	N#CC1=CC=C(OC23CCC(NC(=O)C4=CC=C(N5CCC(CN6CC7=C(C=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)C6)CC5)C=C4)(CC2)C3)C=C1Cl	C42H41ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-MCNNXX	SCHEMBL24031727	N-[(1S,3R)-3-(3-chloro-4-cyanophenoxy)cyclopentyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]benzamide	N#CC1=CC=C(O[C@@H]2CC[C@H](NC(=O)C3=CC=C(N4CCC(CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C3)C2)C=C1Cl	C40H39ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-Q49AM4	WO2021231927A1_93	N-[(1R,3S)-3-(3-chloro-4-cyanophenoxy)cyclopentyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]benzamide	N#CC1=CC=C(O[C@H]2CC[C@@H](NC(=O)C3=CC=C(N4CCC(CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C3)C2)C=C1Cl	C40H39ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-IPAMX5	WO2021231927A1_94	.	[H]C1(OC2=CC=C(C#N)C(Cl)=C2)CC2CCC(C1)N2C(=O)C1=CC=C(N2CCC(N3CC4=C(C=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)C3)CC2)C=C1	C41H39ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-AW5KVI	SCHEMBL24031699	2-Chloro-4-[[8-[4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzonitrile	[H]C1(OC2=CC=C(C#N)C(Cl)=C2)CC2CCC(C1)N2C(=O)C1=CC=C(N2CCC(CN3CC4=C(C=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)C3)CC2)C=C1	C42H41ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-CRCVP3	WO2021231927A1_96	2-Chloro-4-[1-[[4-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]ethyl]piperidine-1-carbonyl]phenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile	CC1=C(C)N(CC2=CC=C(C(=O)N3CCC(CCN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)N=C1C1=CC(Cl)=C(C#N)C=C1	C42H40ClN7O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-VMNY8Z	SCHEMBL24031657	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-3-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]piperidine-1-carbonyl]bicyclo[1.1.1]pentane-1-carboxamide	CC1(C)[C@H](NC(=O)C23CC(C(=O)N4CCC(N5CC6=CC7=C(C=C6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)(C2)C3)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C42H45ClN6O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-GQZ0G0	SCHEMBL24031660	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-3-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidine-1-carbonyl]bicyclo[1.1.1]pentane-1-carboxamide	CC1(C)[C@H](NC(=O)C23CC(C(=O)N4CCC(CN5CC6=CC7=C(C=C6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)(C2)C3)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C43H47ClN6O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-0BC6IR	WO2021231927A1_99	.	CC1=CC(N2C[C@H](NC(=O)C3=CC=C(N4CCC(N5CC6=CC7=C(C=C6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)C=C3)C[C@@H]2C)=CC=C1C#N	C40H41N7O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-875NIS	WO2021231927A1_100	.	CC1=CC(N2C[C@@H](NC(=O)C3=CC=C(N4CCC(N5CC6=CC7=C(C=C6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)C=C3)C[C@@H]2C)=CC=C1C#N	C40H41N7O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-10EUHT	SCHEMBL24031667	2-Chloro-4-[1-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]piperidin-1-yl]benzoyl]piperidin-4-yl]oxybenzonitrile	N#CC1=CC=C(OC2CCN(C(=O)C3=CC=C(N4CCC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C3)CC2)C=C1Cl	C39H37ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-M09Q78	SCHEMBL24031661	2-Chloro-4-[1-[4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]benzoyl]piperidin-4-yl]oxybenzonitrile	N#CC1=CC=C(OC2CCN(C(=O)C3=CC=C(N4CCC(CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C3)CC2)C=C1Cl	C40H39ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-FEL2HF	SCHEMBL24031668	N-[(3R,5S)-1-(3-chloro-4-cyanophenyl)-5-methylpyrrolidin-3-yl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]benzamide	C[C@H]1C[C@@H](NC(=O)C2=CC=C(N3CCC(CN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)CN1C1=CC=C(C#N)C(Cl)=C1	C40H40ClN7O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-3MDJL5	SCHEMBL24031812	N-[(3S,5S)-1-(3-chloro-4-cyanophenyl)-5-methylpyrrolidin-3-yl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]benzamide	C[C@H]1C[C@H](NC(=O)C2=CC=C(N3CCC(CN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)CN1C1=CC=C(C#N)C(Cl)=C1	C40H40ClN7O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-QPDIQ8	SCHEMBL26802005	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]azetidine-1-carbonyl]benzamide	CC1(C)[C@H](NC(=O)C2=CC=C(C(=O)N3CC(N4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)C3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C41H39ClN6O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-ZGLYQA	SCHEMBL24031818	2-chloro-4-[(3R)-3-[4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidine-1-carbonyl]phenoxy]-2,2-dimethylazetidin-1-yl]benzonitrile	CC1(C)[C@H](OC2=CC=C(C(=O)N3CCC(CN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)CN1C1=CC(Cl)=C(C#N)C=C1	C40H39ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-OVIUXF	SCHEMBL24031820	2-chloro-4-[(3S)-3-[4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidine-1-carbonyl]phenoxy]-2,2-dimethylazetidin-1-yl]benzonitrile	CC1(C)[C@@H](OC2=CC=C(C(=O)N3CCC(CN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)CN1C1=CC(Cl)=C(C#N)C=C1	C40H39ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-71E043	SCHEMBL24031805	2-chloro-4-[(3R)-3-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]piperidine-1-carbonyl]phenoxy]-2,2-dimethylazetidin-1-yl]benzonitrile	CC1(C)[C@H](OC2=CC=C(C(=O)N3CCC(N4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)CN1C1=CC(Cl)=C(C#N)C=C1	C39H37ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-P2RKYW	SCHEMBL24031806	2-chloro-4-[(3S)-3-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]piperidine-1-carbonyl]phenoxy]-2,2-dimethylazetidin-1-yl]benzonitrile	CC1(C)[C@@H](OC2=CC=C(C(=O)N3CCC(N4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)CN1C1=CC(Cl)=C(C#N)C=C1	C39H37ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-X6YEGE	SCHEMBL24031807	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-6,7-dihydro-5H-cyclopenta[f]isoindol-6-yl]piperazin-1-yl]benzamide	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCN(C4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C42H43ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-MEKZAI	SCHEMBL24031821	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-6,7-dihydro-5H-cyclopenta[f]isoindol-6-yl]methyl]piperazin-1-yl]benzamide	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCN(CC4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C43H45ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-MH0OER	SCHEMBL24031718	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-6,7-dihydro-5H-cyclopenta[f]isoindole-6-carbonyl]piperazin-1-yl]benzamide	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCN(C(=O)C4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C43H43ClN6O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-23NF0R	SCHEMBL24031717	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-6,7-dihydro-5H-cyclopenta[f]isoindol-6-yl]acetyl]piperazin-1-yl]benzamide	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCN(C(=O)CC4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C44H45ClN6O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-FVS7QD	SCHEMBL24031715	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxospiro[5,7-dihydrocyclopenta[f]isoindole-6,3'-azetidine]-1'-yl]piperidin-1-yl]benzamide	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(N4CC5(CC6=CC7=C(C=C6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C4)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C45H47ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-PWLZHW	SCHEMBL26802019	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxospiro[5,7-dihydrocyclopenta[f]isoindole-6,3'-azetidine]-1'-yl]methyl]piperidin-1-yl]benzamide	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(CN4CC5(CC6=CC7=C(C=C6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C4)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C46H49ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-XUQBDW	SCHEMBL24031719	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxospiro[5,7-dihydrocyclopenta[f]isoindole-6,4'-piperidine]-1'-yl]piperidin-1-yl]benzamide	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(N4CCC5(CC4)CC4=CC6=C(C=C4C5)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C47H51ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-1KWB55	SCHEMBL24031713	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxospiro[5,7-dihydrocyclopenta[f]isoindole-6,4'-piperidine]-1'-yl]methyl]piperidin-1-yl]benzamide	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(CN4CCC5(CC4)CC4=CC6=C(C=C4C5)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C48H53ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-LTL5WL	SCHEMBL26802029	2-chloro-4-[(7S)-4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]piperidine-1-carbonyl]phenyl]-7-methyl-1,4-diazepan-1-yl]benzonitrile	C[C@H]1CCN(C2=CC=C(C(=O)N3CCC(N4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)CCN1C1=CC(Cl)=C(C#N)C=C1	C40H40ClN7O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-VRAANV	SCHEMBL24031716	2-chloro-4-[(7S)-4-[4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidine-1-carbonyl]phenyl]-7-methyl-1,4-diazepan-1-yl]benzonitrile	C[C@H]1CCN(C2=CC=C(C(=O)N3CCC(CN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)CCN1C1=CC(Cl)=C(C#N)C=C1	C41H42ClN7O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-KHCDF0	SCHEMBL26802032	2-chloro-4-[(3S,4R)-1-[4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]benzoyl]-4-methylpiperidin-3-yl]oxybenzonitrile	C[C@@H]1CCN(C(=O)C2=CC=C(N3CCC(CN4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=C2)C[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C41H41ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-2PFK0Z	SCHEMBL26802035	2-chloro-4-[(3S,4R)-1-[4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]benzoyl]-4-methylpyrrolidin-3-yl]oxybenzonitrile	C[C@@H]1CN(C(=O)C2=CC=C(N3CCC(CN4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=C2)C[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C40H39ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-7LMVL2	SCHEMBL24031350	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-7,8-dihydro-5H-pyrrolo[3,4-g]isoquinolin-6-yl]methyl]piperidin-1-yl]benzamide	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(CN4CCC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C44H47ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-9UDHEL	SCHEMBL26802041	N-[2-(3-chloro-4-cyanophenoxy)spiro[3.3]heptan-6-yl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]benzamide	N#CC1=CC=C(OC2CC3(CC(NC(=O)C4=CC=C(N5CCC(CN6CC7=C(C=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)C6)CC5)C=C4)C3)C2)C=C1Cl	C42H41ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-VKB8MH	SCHEMBL26802043	N-[7-(3-chloro-4-cyanophenoxy)spiro[3.5]nonan-2-yl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]benzamide	N#CC1=CC=C(OC2CCC3(CC2)CC(NC(=O)C2=CC=C(N4CCC(CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C2)C3)C=C1Cl	C44H45ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-PDSUCS	SCHEMBL26802045	N-[2-(3-chloro-4-cyanophenoxy)spiro[3.5]nonan-7-yl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]benzamide	N#CC1=CC=C(OC2CC3(CCC(NC(=O)C4=CC=C(N5CCC(CN6CC7=C(C=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)C6)CC5)C=C4)CC3)C2)C=C1Cl	C44H45ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-QA71G9	SCHEMBL24031342	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-7,8-dihydro-5H-pyrrolo[3,4-g]isoquinolin-6-yl]piperidin-1-yl]benzamide	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(N4CCC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C43H45ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-31B55T	SCHEMBL24031344	N-[(1S,3S)-3-(3-chloro-4-cyanophenoxy)-2,2-dimethylcyclobutyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-7,8-dihydro-5H-pyrrolo[3,4-g]isoquinolin-6-yl]methyl]piperidin-1-yl]benzamide	CC1(C)[C@@H](NC(=O)C2=CC=C(N3CCC(CN4CCC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=C2)C[C@@H]1OC1=CC=C(C#N)C(Cl)=C1	C42H43ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-JB75F9	SCHEMBL26802048	N-[(1S,3S)-3-(3-chloro-4-cyanophenoxy)-2,2-dimethylcyclobutyl]-4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-7,8-dihydro-5H-pyrrolo[3,4-g]isoquinolin-6-yl]piperidin-1-yl]benzamide	CC1(C)[C@@H](NC(=O)C2=CC=C(N3CCC(N4CCC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=C2)C[C@@H]1OC1=CC=C(C#N)C(Cl)=C1	C41H41ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-7Q630G	SCHEMBL24031830	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-7,8-dihydro-5H-pyrrolo[3,4-g]isoquinolin-6-yl]methyl]piperidin-1-yl]benzamide	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=CC=C(N4CCC(CN5CCC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C3)CC2)C=C1Cl	C42H43ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-FXJH4V	SCHEMBL26802053	[4-[4-[[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidine-1-carbonyl]phenyl] 4-(3-chloro-4-cyanophenoxy)piperidine-1-carboxylate	N#CC1=CC=C(OC2CCN(C(=O)OC3=CC=C(C(=O)N4CCC(CN5CC6=CC7=C(C=C6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)C=C3)CC2)C=C1Cl	C41H39ClN6O8	AR	P10275	CRBN	WO-2021231927-A1
TPD-G04ODZ	SCHEMBL24031831	4-(3-chloro-4-cyanophenoxy)-N-[4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidine-1-carbonyl]phenyl]piperidine-1-carboxamide	N#CC1=CC=C(OC2CCN(C(=O)NC3=CC=C(C(=O)N4CCC(CN5CC6=CC7=C(C=C6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)C=C3)CC2)C=C1Cl	C41H40ClN7O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-L2H4JM	SCHEMBL24031828	5-[3-[6-[2-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]cyclohexyl]ethynyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxy-3-(trifluoromethyl)pyridine-2-carbonitrile	CC1(C)[C@H](OC2=CN=C(C#N)C(C(F)(F)F)=C2)C(C)(C)[C@H]1N1CC2=CC(C#C[C@H]3CC[C@H](CN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)=CC=C2C1=O	C47H45F3N6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-85ILV5	SCHEMBL26810961	2-chloro-4-[4-[6-[2-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]cyclohexyl]ethynyl]-3-oxo-1H-isoindol-2-yl]cyclohexyl]oxybenzonitrile	N#CC1=CC=C(O[C@H]2CC[C@H](N3CC4=CC(C#C[C@H]5CC[C@H](CN6CC7=CC8=C(C=C7C6)C(=O)N(C6CCC(=O)NC6=O)C8=O)CC5)=CC=C4C3=O)CC2)C=C1Cl	C45H42ClN5O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-4DZGK8	SCHEMBL24031829	2-chloro-4-[4-[6-[2-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-7,8-dihydro-5H-pyrrolo[3,4-g]isoquinolin-6-yl]methyl]cyclohexyl]ethynyl]-3-oxo-1H-isoindol-2-yl]cyclohexyl]oxybenzonitrile	N#CC1=CC=C(O[C@H]2CC[C@H](N3CC4=CC(C#C[C@H]5CC[C@H](CN6CCC7=CC8=C(C=C7C6)C(=O)N(C6CCC(=O)NC6=O)C8=O)CC5)=CC=C4C3=O)CC2)C=C1Cl	C46H44ClN5O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-BKY8FB	SCHEMBL24031832	2-chloro-4-[3-[6-[2-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]cyclohexyl]ethynyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@H]1N1CC2=CC(C#C[C@H]3CC[C@H](CN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)=CC=C2C1=O	C47H46ClN5O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-ITB2VU	SCHEMBL26802062	2-chloro-4-[3-[6-[2-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-7,8-dihydro-5H-pyrrolo[3,4-g]isoquinolin-6-yl]methyl]cyclohexyl]ethynyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@H]1N1CC2=CC(C#C[C@H]3CC[C@H](CN4CCC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)=CC=C2C1=O	C48H48ClN5O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-TZSNVM	SCHEMBL26802063	2-chloro-4-[3-[6-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]cyclohexyl]ethynyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@H]1N1CC2=CC(C#CC3CCC(N4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)=CC=C2C1=O	C46H44ClN5O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-J8QGJ2	SCHEMBL24031922	2-chloro-4-[3-[6-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-7,8-dihydro-5H-pyrrolo[3,4-g]isoquinolin-6-yl]cyclohexyl]ethynyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@H]1N1CC2=CC(C#CC3CCC(N4CCC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)=CC=C2C1=O	C47H46ClN5O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-EPTD2E	SCHEMBL24031923	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]piperidine-1-carbonyl]benzamide	CC1(C)[C@H](NC(=O)C2=CC=C(C(=O)N3CCC(N4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C43H43ClN6O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-URW6IV	SCHEMBL26802070	2-chloro-4-[3-[6-[4-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-6-yl]methyl]piperidine-1-carbonyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC(Cl)=C(C#N)C=C2)C(C)(C)[C@H]1N1CC2=CC(C(=O)N3CCC(CN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6)CC3)=CC=C2C1=O	C45H47ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-AEUQOT	SCHEMBL26811431	2-chloro-4-[3-[6-[6-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]-2-azaspiro[3.3]heptane-2-carbonyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC(Cl)=C(C#N)C=C2)C(C)(C)[C@H]1N1CC2=CC(C(=O)N3CC4(CC(CN5CC6=CC7=C(C=C6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C4)C3)=CC=C2C1=O	C46H45ClN6O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-EWKN8W	SCHEMBL24031919	2-chloro-4-[3-[6-[3-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]azetidine-1-carbonyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC(Cl)=C(C#N)C=C2)C(C)(C)[C@H]1N1CC2=CC(C(=O)N3CC(CN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)C3)=CC=C2C1=O	C43H41ClN6O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-XNV3ZY	SCHEMBL26667225	2-chloro-4-[3-[6-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindole-6-carbonyl]cyclohexyl]ethynyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile; SCHEMBL26811534	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@H]1N1CC2=CC(C#C[C@H]3CC[C@H](C(=O)N4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)=CC=C2C1=O	C47H44ClN5O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-7D0BSK	WO2021231927A1_147	.	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@H]1N1CC2=CC(C#CC3CCC(C(=O)N4CCC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)=CC=C2C1=O	C48H46ClN5O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-VD3T30	SCHEMBL24031755	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-3-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]-2-oxoethyl]-1,2,4,5-tetrahydro-3-benzazepine-7-carboxamide	CC1(C)[C@H](NC(=O)C2=CC=C3CCN(CC(=O)N4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CCC3=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C43H43ClN6O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-22TXMI	SCHEMBL26802094	2-chloro-4-[3-[6-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@H]1N1CC2=CC(N3CCC(CN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)=CC=C2C1=O	C44H45ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-GABO5J	SCHEMBL26802079	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-3-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]acetyl]-1,2,4,5-tetrahydro-3-benzazepine-7-carboxamide	CC1(C)[C@H](NC(=O)C2=CC=C3CCN(C(=O)CN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CCC3=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C43H43ClN6O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-6ZG40R	WO2021231927A1_151	.	CC1(C)[C@H](NC(=O)C2=CC=C3CN(C(=O)CN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C41H39ClN6O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-CYXFCA	WO2021231927A1_152	.	CC1(C)[C@H](NC(=O)C2=CC=C3CN(CC(=O)N4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C41H39ClN6O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-3F1R48	SCHEMBL26802080	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]acetyl]-3,4-dihydro-1H-isoquinoline-6-carboxamide	CC1(C)[C@H](NC(=O)C2=CC=C3CN(C(=O)CN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CCC3=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C42H41ClN6O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-Y07VJN	SCHEMBL26802082	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]-2-oxoethyl]-3,4-dihydro-1H-isoquinoline-6-carboxamide	CC1(C)[C@H](NC(=O)C2=CC=C3CN(CC(=O)N4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CCC3=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C42H41ClN6O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-E6W96M	SCHEMBL24031800	N-[(3R,5S)-1-(3-chloro-4-cyanophenyl)-5-methylpyrrolidin-3-yl]-2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]acetyl]-1,3-dihydroisoindole-5-carboxamide	C[C@H]1C[C@@H](NC(=O)C2=CC=C3CN(C(=O)CN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3=C2)CN1C1=CC=C(C#N)C(Cl)=C1	C38H34ClN7O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-7GYHH6	SCHEMBL24031801	N-[(3R,5S)-1-(3-chloro-4-cyanophenyl)-5-methylpyrrolidin-3-yl]-2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]acetyl]-3,4-dihydro-1H-isoquinoline-6-carboxamide	C[C@H]1C[C@@H](NC(=O)C2=CC=C3CN(C(=O)CN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CCC3=C2)CN1C1=CC=C(C#N)C(Cl)=C1	C39H36ClN7O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-UH0AXH	SCHEMBL24031795	N-[(1S,3S)-3-(3-chloro-4-cyanophenoxy)-2,2-dimethylcyclobutyl]-2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]acetyl]-1,3-dihydroisoindole-5-carboxamide	CC1(C)[C@@H](NC(=O)C2=CC=C3CN(C(=O)CN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3=C2)C[C@@H]1OC1=CC=C(C#N)C(Cl)=C1	C39H35ClN6O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-TS8B3G	WO2021231927A1_158	N-[(1S,3S)-3-(3-chloro-4-cyanophenoxy)-2,2-dimethylcyclobutyl]-2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]acetyl]-3,4-dihydro-1H-isoquinoline-6-carboxamide	CC1(C)[C@@H](NC(=O)C2=CC=C3CN(C(=O)CN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CCC3=C2)C[C@@H]1OC1=CC=C(C#N)C(Cl)=C1	C40H37ClN6O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-Z5KNFI	SCHEMBL26802098	2-chloro-4-[3-[6-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@H]1N1CC2=CC(N3CCC(N4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)=CC=C2C1=O	C43H43ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-1R0M4Q	SCHEMBL24031563	2-chloro-4-[3-[6-[3-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]azetidin-1-yl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@H]1N1CC2=CC(N3CC(CN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)C3)=CC=C2C1=O	C42H41ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-FD8BM9	SCHEMBL24031562	2-chloro-4-[3-[6-[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]azetidin-1-yl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@H]1N1CC2=CC(N3CC(N4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)C3)=CC=C2C1=O	C41H39ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-FSVTE0	SCHEMBL24031564	2-chloro-4-[3-[6-[4-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@H]1N1CC2=CC(N3CCC(CN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6)CC3)=CC=C2C1=O	C44H47ClN6O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-SV29YE	SCHEMBL24031565	2-chloro-4-[3-[6-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-6-yl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile; SCHEMBL26667227	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@H]1N1CC2=CC(N3CCC(N4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6)CC3)=CC=C2C1=O	C43H45ClN6O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-S0HEBM	SCHEMBL26802101	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-2-[1-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]acetyl]azetidin-3-yl]-3,4-dihydro-1H-isoquinoline-6-carboxamide	CC1(C)[C@H](NC(=O)C2=CC=C3CN(C4CN(C(=O)CN5CC6=CC7=C(C=C6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C4)CCC3=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C45H46ClN7O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-KLQH3T	SCHEMBL24031561	2-chloro-4-[1-[[4-[2-[1-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-7,8-dihydro-5H-pyrrolo[3,4-g]isoquinolin-6-yl]-2-oxoethyl]piperidin-4-yl]ethynyl]phenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile	CC1=C(C)N(CC2=CC=C(C#CC3CCN(CC(=O)N4CCC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)N=C1C1=CC(Cl)=C(C#N)C=C1	C44H40ClN7O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-5LOH20	SCHEMBL24031325	2-chloro-4-[1-[[4-[2-[1-[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-7,8-dihydro-5H-pyrrolo[3,4-g]isoquinolin-6-yl]-3-oxopropyl]piperidin-4-yl]ethynyl]phenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile	CC1=C(C)N(CC2=CC=C(C#CC3CCN(CCC(=O)N4CCC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)N=C1C1=CC(Cl)=C(C#N)C=C1	C45H42ClN7O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-86U3A7	SCHEMBL24031328	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-7,8-dihydro-5H-pyrrolo[3,4-g]isoquinolin-6-yl]piperidin-1-yl]benzamide	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=CC=C(N4CCC(N5CCC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C3)CC2)C=C1Cl	C41H41ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-UPSP3R	SCHEMBL24031329	N-[4-(3-chloro-4-cyanoanilino)cyclohexyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-7,8-dihydro-5H-pyrrolo[3,4-g]isoquinolin-6-yl]methyl]piperidin-1-yl]benzamide	N#CC1=CC=C(N[C@H]2CC[C@H](NC(=O)C3=CC=C(N4CCC(CN5CCC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C3)CC2)C=C1Cl	C42H44ClN7O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-ZTC9SW	SCHEMBL24031346	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[2-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-7,8-dihydro-5H-pyrrolo[3,4-g]isoquinolin-6-yl]methyl]cyclohexyl]ethynyl]benzamide	CC1(C)[C@H](NC(=O)C2=CC=C(C#CC3CCC(CN4CCC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C47H48ClN5O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-IRNHNX	SCHEMBL24031349	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[2-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]cyclohexyl]ethynyl]benzamide	CC1(C)[C@H](NC(=O)C2=CC=C(C#CC3CCC(CN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C46H46ClN5O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-S7NUNW	SCHEMBL24031336	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-4-[2-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-7,8-dihydro-5H-pyrrolo[3,4-g]isoquinolin-6-yl]methyl]cyclohexyl]ethynyl]benzamide	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=CC=C(C#CC4CCC(CN5CCC6=CC7=C(C=C6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)C=C3)CC2)C=C1Cl	C45H44ClN5O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-JU8J0J	SCHEMBL24031316	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-4-[2-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]cyclohexyl]ethynyl]benzamide	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=CC=C(C#CC4CCC(CN5CC6=CC7=C(C=C6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)C=C3)CC2)C=C1Cl	C44H42ClN5O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-FU92EU	SCHEMBL24031351	2-chloro-4-[4-[6-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]piperidine-1-carbonyl]-3-oxo-1H-isoindol-2-yl]cyclohexyl]oxybenzonitrile	N#CC1=CC=C(O[C@H]2CC[C@H](N3CC4=C(C=CC(C(=O)N5CCC(N6CC7=CC8=C(C=C7C6)C(=O)N(C6CCC(=O)NC6=O)C8=O)CC5)=C4)C3=O)CC2)C=C1Cl	C42H39ClN6O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-RUVTG7	SCHEMBL24031332	2-chloro-4-[4-[6-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidine-1-carbonyl]-3-oxo-1H-isoindol-2-yl]cyclohexyl]oxybenzonitrile	N#CC1=CC=C(O[C@H]2CC[C@H](N3CC4=C(C=CC(C(=O)N5CCC(CN6CC7=CC8=C(C=C7C6)C(=O)N(C6CCC(=O)NC6=O)C8=O)CC5)=C4)C3=O)CC2)C=C1Cl	C43H41ClN6O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-39HCP1	WO2021231927A1_175	.	CC1(C)C(NC2=CC=C(C(=O)N3CCC(CN4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=C2)C(C)(C)C1OC1=CC=C(C#N)C(Cl)=C1	C43H45ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-IWRY4C	WO2021231927A1_176	.	CC1(C)C(NC2=CC=C(C(=O)N3CCC(N4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=C2)C(C)(C)C1OC1=CC=C(C#N)C(Cl)=C1	C42H43ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-EM29U9	SCHEMBL24031333	N-[4-(3-chloro-4-cyanoanilino)cyclohexyl]-4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-7,8-dihydro-5H-pyrrolo[3,4-g]isoquinolin-6-yl]piperidin-1-yl]benzamide	N#CC1=CC=C(N[C@H]2CC[C@H](NC(=O)C3=CC=C(N4CCC(N5CCC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C3)CC2)C=C1Cl	C41H42ClN7O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-4N5W3I	SCHEMBL24031313	N-[4-(3-chloro-4-cyano-N-methylanilino)cyclohexyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-7,8-dihydro-5H-pyrrolo[3,4-g]isoquinolin-6-yl]methyl]piperidin-1-yl]benzamide	CN(C1=CC=C(C#N)C(Cl)=C1)[C@H]1CC[C@H](NC(=O)C2=CC=C(N3CCC(CN4CCC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=C2)CC1	C43H46ClN7O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-KSWXNC	SCHEMBL24031317	N-[4-(3-chloro-4-cyano-N-methylanilino)cyclohexyl]-4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-7,8-dihydro-5H-pyrrolo[3,4-g]isoquinolin-6-yl]piperidin-1-yl]benzamide	CN(C1=CC=C(C#N)C(Cl)=C1)[C@H]1CC[C@H](NC(=O)C2=CC=C(N3CCC(N4CCC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=C2)CC1	C42H44ClN7O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-5XVCWD	SCHEMBL24031326	2-chloro-4-[3-[6-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-7,8-dihydro-5H-pyrrolo[3,4-g]isoquinolin-6-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@H]1N1CC2=CC(N3CCC(CN4CCC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)=CC=C2C1=O	C45H47ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-DBSS89	SCHEMBL24031337	2-chloro-4-[3-[6-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-7,8-dihydro-5H-pyrrolo[3,4-g]isoquinolin-6-yl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@H]1N1CC2=CC(N3CCC(N4CCC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)=CC=C2C1=O	C44H45ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-PX47TB	SCHEMBL24031839	2-chloro-4-[4-[6-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-7,8-dihydro-5H-pyrrolo[3,4-g]isoquinolin-6-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]cyclohexyl]oxybenzonitrile	N#CC1=CC=C(O[C@H]2CC[C@H](N3CC4=CC(N5CCC(CN6CCC7=C(C=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)C6)CC5)=CC=C4C3=O)CC2)C=C1Cl	C43H43ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-Z6GMFL	SCHEMBL24031836	N-[3-(3-chloro-4-cyanoanilino)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]benzamide	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(CN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1NC1=CC=C(C#N)C(Cl)=C1	C43H46ClN7O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-LRSH7T	SCHEMBL24031837	N-[3-(3-chloro-4-cyano-N-methylanilino)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]benzamide	CN(C1=CC=C(C#N)C(Cl)=C1)[C@H]1C(C)(C)[C@H](NC(=O)C2=CC=C(N3CCC(CN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C1(C)C	C44H48ClN7O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-7UJHZ4	SCHEMBL24031834	N-[3-(3-chloro-4-cyanoanilino)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]piperidin-1-yl]benzamide	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(N4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1NC1=CC=C(C#N)C(Cl)=C1	C42H44ClN7O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-DSETOW	SCHEMBL24031842	N-[3-(3-chloro-4-cyano-N-methylanilino)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]piperidin-1-yl]benzamide	CN(C1=CC=C(C#N)C(Cl)=C1)[C@H]1C(C)(C)[C@H](NC(=O)C2=CC=C(N3CCC(N4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C1(C)C	C43H46ClN7O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-MMYOPV	SCHEMBL24031835	N-[3-[4-cyano-3-(trifluoromethyl)phenoxy]-2,2,4,4-tetramethylcyclobutyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]benzamide	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(CN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(C(F)(F)F)=C1	C44H45F3N6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-M6NUG3	SCHEMBL24031840	N-[3-[6-cyano-5-(trifluoromethyl)pyridin-3-yl]oxy-2,2,4,4-tetramethylcyclobutyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]benzamide	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(CN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CN=C(C#N)C(C(F)(F)F)=C1	C43H44F3N7O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-7LF4NG	SCHEMBL24031833	N-[3-(3-chloro-4-cyano-2-methylphenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]benzamide	CC1=C(Cl)C(C#N)=CC=C1O[C@H]1C(C)(C)[C@H](NC(=O)C2=CC=C(N3CCC(CN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C1(C)C	C44H47ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-2JA1XV	SCHEMBL24031838	N-[3-(4-cyano-3-fluorophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]benzamide	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(CN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(F)=C1	C43H45FN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-4358WI	SCHEMBL24031959	N-[3-(4-cyano-3-fluoro-2-methylphenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]benzamide	CC1=C(F)C(C#N)=CC=C1O[C@H]1C(C)(C)[C@H](NC(=O)C2=CC=C(N3CCC(CN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C1(C)C	C44H47FN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-IY6XPU	SCHEMBL24031958	N-[3-(4-cyano-3-methylphenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]benzamide	CC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(CN5CC6=CC7=C(C=C6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)C=C3)C2(C)C)=CC=C1C#N	C44H48N6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-HUVVNA	SCHEMBL24031937	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[[2-(1-methyl-2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]benzamide	CN1C(=O)CCC(N2C(=O)C3=C(C=C4CN(CC5CCN(C6=CC=C(C(=O)N[C@H]7C(C)(C)[C@H](OC8=CC=C(C#N)C(Cl)=C8)C7(C)C)C=C6)CC5)CC4=C3)C2=O)C1=O	C44H47ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-68Q8RS	SCHEMBL24031962	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]-2-fluorobenzamide	CC1(C)[C@H](NC(=O)C2=C(F)C=C(N3CCC(CN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C43H44ClFN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-WPEKJO	SCHEMBL24031968	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]-3-fluorobenzamide	CC1(C)[C@H](NC(=O)C2=CC(F)=C(N3CCC(CN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C43H44ClFN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-AEMX3H	SCHEMBL24031965	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-5-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]pyridine-2-carboxamide	CC1(C)[C@H](NC(=O)C2=NC=C(N3CCC(CN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C42H44ClN7O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-U3L0RE	SCHEMBL24031966	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]pyridine-3-carboxamide	CC1(C)[C@H](NC(=O)C2=CN=C(N3CCC(CN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C42H44ClN7O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-B3NMTW	SCHEMBL24031960	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide	CC1(C)[C@H](NC(=O)C2=NN=C(N3CCC(CN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C41H43ClN8O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-JAIJX9	SCHEMBL24031969	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-2-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]pyrimidine-5-carboxamide	CC1(C)[C@H](NC(=O)C2=CN=C(N3CCC(CN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)N=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C41H43ClN8O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-HWH0WU	SCHEMBL24031783	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]-4-methylpiperidin-1-yl]benzamide	CC1(CN2CC3=CC4=C(C=C3C2)C(=O)N(C2CCC(=O)NC2=O)C4=O)CCN(C2=CC=C(C(=O)N[C@H]3C(C)(C)[C@H](OC4=CC=C(C#N)C(Cl)=C4)C3(C)C)C=C2)CC1	C44H47ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-D5GAH1	SCHEMBL24031781	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]-4-fluoropiperidin-1-yl]benzamide	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(F)(CN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C43H44ClFN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-OKZATW	SCHEMBL24031787	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-chloro-4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]benzamide	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(Cl)(CN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C43H44Cl2N6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-QB6T2L	SCHEMBL24031782	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]-4-methoxypiperidin-1-yl]benzamide	COC1(CN2CC3=CC4=C(C=C3C2)C(=O)N(C2CCC(=O)NC2=O)C4=O)CCN(C2=CC=C(C(=O)N[C@H]3C(C)(C)[C@H](OC4=CC=C(C#N)C(Cl)=C4)C3(C)C)C=C2)CC1	C44H47ClN6O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-DXJYNW	SCHEMBL24031780	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]-4-ethoxypiperidin-1-yl]benzamide	CCOC1(CN2CC3=CC4=C(C=C3C2)C(=O)N(C2CCC(=O)NC2=O)C4=O)CCN(C2=CC=C(C(=O)N[C@H]3C(C)(C)[C@H](OC4=CC=C(C#N)C(Cl)=C4)C3(C)C)C=C2)CC1	C45H49ClN6O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-3V0TAZ	SCHEMBL24031785	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]-4-hydroxypiperidin-1-yl]benzamide	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(O)(CN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C43H45ClN6O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-Q0KU8K	SCHEMBL24031784	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-cyano-4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]benzamide	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(C#N)(CN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C44H44ClN7O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-81OKBA	SCHEMBL24031786	N-[3-(3-chloro-4-cyano-2-methylphenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]piperidin-1-yl]benzamide	CC1=C(Cl)C(C#N)=CC=C1O[C@H]1C(C)(C)[C@H](NC(=O)C2=CC=C(N3CCC(N4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C1(C)C	C43H45ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-1EO693	SCHEMBL24031335	N-[3-[4-cyano-3-(trifluoromethyl)phenoxy]-2,2,4,4-tetramethylcyclobutyl]-4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]piperidin-1-yl]benzamide	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(N4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(C(F)(F)F)=C1	C43H43F3N6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-VD8RM4	SCHEMBL24031320	N-[3-[6-cyano-5-(trifluoromethyl)pyridin-3-yl]oxy-2,2,4,4-tetramethylcyclobutyl]-4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]piperidin-1-yl]benzamide	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(N4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CN=C(C#N)C(C(F)(F)F)=C1	C42H42F3N7O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-DBM02W	SCHEMBL24031321	N-[3-(4-cyano-3-fluorophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]piperidin-1-yl]benzamide	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(N4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(F)=C1	C42H43FN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-RUKK2C	SCHEMBL24031327	N-[3-(4-cyano-3-fluoro-2-methylphenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]piperidin-1-yl]benzamide	CC1=C(F)C(C#N)=CC=C1O[C@H]1C(C)(C)[C@H](NC(=O)C2=CC=C(N3CCC(N4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C1(C)C	C43H45FN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-719UVQ	SCHEMBL24031340	N-[3-(4-cyano-3-methylphenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]piperidin-1-yl]benzamide	CC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(N5CC6=CC7=C(C=C6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)C=C3)C2(C)C)=CC=C1C#N	C43H46N6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-56JZWA	SCHEMBL24031343	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-5-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]piperidin-1-yl]pyridine-2-carboxamide	CC1(C)[C@H](NC(=O)C2=NC=C(N3CCC(N4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C41H42ClN7O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-UYTVZ4	SCHEMBL24031322	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]piperidin-1-yl]pyridine-3-carboxamide	CC1(C)[C@H](NC(=O)C2=CN=C(N3CCC(N4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C41H42ClN7O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-9B8D5Q	SCHEMBL24031323	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]piperidin-1-yl]pyridazine-3-carboxamide	CC1(C)[C@H](NC(=O)C2=NN=C(N3CCC(N4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C40H41ClN8O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-AUKD1H	SCHEMBL24031324	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-2-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]piperidin-1-yl]pyrimidine-5-carboxamide	CC1(C)[C@H](NC(=O)C2=CN=C(N3CCC(N4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)N=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C40H41ClN8O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-7OD9C7	SCHEMBL24031952	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]piperidin-1-yl]-2-fluorobenzamide	CC1(C)[C@H](NC(=O)C2=C(F)C=C(N3CCC(N4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C42H42ClFN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-8FSDJZ	SCHEMBL24031954	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]piperidin-1-yl]-3-fluorobenzamide	CC1(C)[C@H](NC(=O)C2=CC(F)=C(N3CCC(N4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C42H42ClFN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-KSG2DF	SCHEMBL24031951	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]-2-oxoethyl]piperazin-1-yl]pyridine-3-carboxamide	CC1(C)[C@H](NC(=O)C2=CN=C(N3CCN(CC(=O)N4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C42H43ClN8O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-LBIWQD	SCHEMBL24031956	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]acetyl]piperazin-1-yl]pyridine-3-carboxamide	CC1(C)[C@H](NC(=O)C2=CN=C(N3CCN(C(=O)CN4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C42H43ClN8O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-O254W7	SCHEMBL24031953	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-2-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]-2-oxoethyl]piperazin-1-yl]pyrimidine-5-carboxamide	CC1(C)[C@H](NC(=O)C2=CN=C(N3CCN(CC(=O)N4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)N=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C41H42ClN9O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-DYHOW4	SCHEMBL24031957	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-2-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]acetyl]piperazin-1-yl]pyrimidine-5-carboxamide	CC1(C)[C@H](NC(=O)C2=CN=C(N3CCN(C(=O)CN4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)N=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C41H42ClN9O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-HNW2WL	SCHEMBL24031955	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-5-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]-2-oxoethyl]piperazin-1-yl]pyridine-2-carboxamide	CC1(C)[C@H](NC(=O)C2=NC=C(N3CCN(CC(=O)N4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C42H43ClN8O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-ZG2GW7	SCHEMBL24031950	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-5-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]acetyl]piperazin-1-yl]pyridine-2-carboxamide	CC1(C)[C@H](NC(=O)C2=NC=C(N3CCN(C(=O)CN4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C42H43ClN8O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-VYQ0JM	WO2021231927A1_225	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCN(CC(=O)N4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)N=N2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C41H42ClN9O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-YQMTN4	SCHEMBL24031746	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]acetyl]piperazin-1-yl]pyridazine-3-carboxamide	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCN(C(=O)CN4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)N=N2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C41H42ClN9O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-08TWRS	SCHEMBL24031747	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]-2-oxoethyl]piperazin-1-yl]-2-fluorobenzamide	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCN(CC(=O)N4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=C2F)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C43H43ClFN7O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-RWPFA2	SCHEMBL24031748	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]acetyl]piperazin-1-yl]-2-fluorobenzamide	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCN(C(=O)CN4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=C2F)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C43H43ClFN7O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-W8TTJQ	SCHEMBL24031750	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]-2-oxoethyl]piperazin-1-yl]-3-fluorobenzamide	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCN(CC(=O)N4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C(F)=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C43H43ClFN7O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-9V9LVZ	SCHEMBL24031742	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]acetyl]piperazin-1-yl]-3-fluorobenzamide	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCN(C(=O)CN4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C(F)=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C43H43ClFN7O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-HDW9WG	WO2021231927A1_231	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=CN=C(N4CCC(CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C3)CC2)C=C1Cl	C40H40ClN7O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-0O2P95	WO2021231927A1_232	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=CN=C(N4CCC(CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)N=C3)CC2)C=C1Cl	C39H39ClN8O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-GT9R1D	WO2021231927A1_233	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=CC=C(N4CCC(CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)N=N3)CC2)C=C1Cl	C39H39ClN8O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-RKYXRH	WO2021231927A1_234	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=CN=C(N4CCN(CC(=O)N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C3)CC2)C=C1Cl	C40H39ClN8O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-NHWHQT	WO2021231927A1_235	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=CN=C(N4CCN(C(=O)CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C3)CC2)C=C1Cl	C40H39ClN8O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-UV5TZL	WO2021231927A1_236	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=CN=C(N4CCN(CC(=O)N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)N=C3)CC2)C=C1Cl	C39H38ClN9O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-LVGC2R	WO2021231927A1_237	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=CN=C(N4CCN(C(=O)CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)N=C3)CC2)C=C1Cl	C39H38ClN9O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-Q9SC7B	SCHEMBL24031916	N-[4-(3-chloro-4-cyano-N-methylanilino)cyclohexyl]-6-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]pyridine-3-carboxamide	CN(C1=CC=C(C#N)C(Cl)=C1)[C@H]1CC[C@H](NC(=O)C2=CN=C(N3CCC(CN4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=C2)CC1	C41H43ClN8O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-PPN142	SCHEMBL24031921	N-[4-(3-chloro-4-cyano-N-ethylanilino)cyclohexyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]benzamide	CCN(C1=CC=C(C#N)C(Cl)=C1)[C@H]1CC[C@H](NC(=O)C2=CC=C(N3CCC(CN4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=C2)CC1	C43H46ClN7O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-ZYL2KH	SCHEMBL24031733	N-[4-(3-chloro-4-cyano-N-methylanilino)cyclohexyl]-2-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]pyrimidine-5-carboxamide	CN(C1=CC=C(C#N)C(Cl)=C1)[C@H]1CC[C@H](NC(=O)C2=CN=C(N3CCC(CN4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)N=C2)CC1	C40H42ClN9O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-RMEI74	SCHEMBL24031736	N-[4-(3-chloro-4-cyano-N-propan-2-ylanilino)cyclohexyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]benzamide	CC(C)N(C1=CC=C(C#N)C(Cl)=C1)[C@H]1CC[C@H](NC(=O)C2=CC=C(N3CCC(CN4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=C2)CC1	C44H48ClN7O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-YME6DU	SCHEMBL24031357	N-[4-(3-chloro-4-cyano-N-methylanilino)cyclohexyl]-6-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide	CN(C1=CC=C(C#N)C(Cl)=C1)[C@H]1CC[C@H](NC(=O)C2=CC=C(N3CCC(CN4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)N=N2)CC1	C40H42ClN9O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-AGO3JT	SCHEMBL24031734	N-[4-(3-chloro-4-cyano-N-cyclopropylanilino)cyclohexyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]benzamide	N#CC1=CC=C(N(C2CC2)[C@H]2CC[C@H](NC(=O)C3=CC=C(N4CCC(CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C3)CC2)C=C1Cl	C44H46ClN7O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-KZH2VS	SCHEMBL24031735	N-[(4aR,6R,8aR)-1-(3-chloro-4-cyanophenyl)-3,4,4a,5,6,7,8,8a-octahydro-2H-quinolin-6-yl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]benzamide	N#CC1=CC=C(N2CCC[C@@H]3C[C@H](NC(=O)C4=CC=C(N5CCC(CN6CC7=C(C=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)C6)CC5)C=C4)CC[C@H]32)C=C1Cl	C44H46ClN7O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-M979RI	SCHEMBL24031737	N-[(4aR,7R,8aR)-4-(3-chloro-4-cyanophenyl)-2,3,4a,5,6,7,8,8a-octahydrobenzo[b][1,4]oxazin-7-yl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]benzamide	N#CC1=CC=C(N2CCO[C@@H]3C[C@H](NC(=O)C4=CC=C(N5CCC(CN6CC7=C(C=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)C6)CC5)C=C4)CC[C@H]32)C=C1Cl	C43H44ClN7O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-GRC8Y7	WO2021231927A1_246	.	N#CC1=CC=C(N2CCC[C@H]3C[C@H](NC(=O)C4=CC=C(N5CCC(CN6CC7=C(C=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)C6)CC5)C=C4)CC[C@H]32)C=C1Cl	C44H46ClN7O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-O40FAA	WO2021231927A1_247	.	N#CC1=CC=C(N2CCO[C@H]3C[C@H](NC(=O)C4=CC=C(N5CCC(CN6CC7=C(C=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)C6)CC5)C=C4)CC[C@H]32)C=C1Cl	C43H44ClN7O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-V7QKVO	SCHEMBL24031932	N-[4-(4-chloro-5-cyano-2,3-dihydroindol-1-yl)cyclohexyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]benzamide	N#CC1=CC=C2C(=C1Cl)CCN2[C@H]1CC[C@H](NC(=O)C2=CC=C(N3CCC(CN4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=C2)CC1	C43H44ClN7O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-3N9DMY	SCHEMBL24031933	N-[4-[(2S)-4-chloro-5-cyano-2-methyl-2,3-dihydroindol-1-yl]cyclohexyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]benzamide	C[C@H]1CC2=C(Cl)C(C#N)=CC=C2N1[C@H]1CC[C@H](NC(=O)C2=CC=C(N3CCC(CN4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=C2)CC1	C44H46ClN7O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-CBY224	SCHEMBL26815525	N-[4-(6-chloro-5-cyano-2,3-dihydroindol-1-yl)cyclohexyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]benzamide	N#CC1=CC2=C(C=C1Cl)N([C@H]1CC[C@H](NC(=O)C3=CC=C(N4CCC(CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C3)CC1)CC2	C43H44ClN7O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-7ZP27A	SCHEMBL24031939	N-[4-[(2R)-6-chloro-5-cyano-2-methyl-2,3-dihydroindol-1-yl]cyclohexyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]benzamide	C[C@@H]1CC2=C(C=C(Cl)C(C#N)=C2)N1[C@H]1CC[C@H](NC(=O)C2=CC=C(N3CCC(CN4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=C2)CC1	C44H46ClN7O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-B30RRD	SCHEMBL24031940	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]-4-fluoropiperidin-1-yl]benzamide	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=CC=C(N4CCC(F)(CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C3)CC2)C=C1Cl	C41H40ClFN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-1N9N7F	SCHEMBL24031935	N-[4-(3-chloro-4-cyano-N-methylanilino)cyclohexyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]-4-fluoropiperidin-1-yl]benzamide	CN(C1=CC=C(C#N)C(Cl)=C1)[C@H]1CC[C@H](NC(=O)C2=CC=C(N3CCC(F)(CN4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=C2)CC1	C42H43ClFN7O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-STUJYJ	SCHEMBL24031679	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]-4-methoxypiperidin-1-yl]benzamide	COC1(CN2CC3=C(C=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)C2)CCN(C2=CC=C(C(=O)N[C@H]3CC[C@H](OC4=CC=C(C#N)C(Cl)=C4)CC3)C=C2)CC1	C42H43ClN6O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-5LEFFW	SCHEMBL24031678	N-[4-(3-chloro-4-cyano-N-methylanilino)cyclohexyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]-4-methoxypiperidin-1-yl]benzamide	COC1(CN2CC3=C(C=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)C2)CCN(C2=CC=C(C(=O)N[C@H]3CC[C@H](N(C)C4=CC=C(C#N)C(Cl)=C4)CC3)C=C2)CC1	C43H46ClN7O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-A3HL26	SCHEMBL24031681	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]-4-methylpiperidin-1-yl]benzamide	CC1(CN2CC3=C(C=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)C2)CCN(C2=CC=C(C(=O)N[C@H]3CC[C@H](OC4=CC=C(C#N)C(Cl)=C4)CC3)C=C2)CC1	C42H43ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-2CYU0O	SCHEMBL24031680	N-[4-(3-chloro-4-cyano-N-methylanilino)cyclohexyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]-4-methylpiperidin-1-yl]benzamide	CN(C1=CC=C(C#N)C(Cl)=C1)[C@H]1CC[C@H](NC(=O)C2=CC=C(N3CCC(C)(CN4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=C2)CC1	C43H46ClN7O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-X7KQLY	SCHEMBL24031682	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]-4-hydroxypiperidin-1-yl]benzamide	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=CC=C(N4CCC(O)(CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C3)CC2)C=C1Cl	C41H41ClN6O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-7F4U3L	SCHEMBL24031683	N-[4-(3-chloro-4-cyano-N-methylanilino)cyclohexyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]-4-hydroxypiperidin-1-yl]benzamide	CN(C1=CC=C(C#N)C(Cl)=C1)[C@H]1CC[C@H](NC(=O)C2=CC=C(N3CCC(O)(CN4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=C2)CC1	C42H44ClN7O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-146A32	WO2021231927A1_260	.	N#CC1=CC=C(O[C@@H]2CCC3=C(C2)N=C(C2=CC=C(N4CCC(CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C2)N3)C=C1Cl	C41H38ClN7O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-4I2P0K	SCHEMBL24031849	2-chloro-4-[[(5R)-2-[4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]phenyl]-4,5,6,7-tetrahydro-3H-benzimidazol-5-yl]-methylamino]benzonitrile	CN(C1=CC=C(C#N)C(Cl)=C1)[C@@H]1CCC2=C(C1)N=C(C1=CC=C(N3CCC(CN4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=C1)N2	C42H41ClN8O4	AR	P10275	CRBN	WO-2021231927-A1
TPD-FFCZO6	SCHEMBL24031850	2-chloro-4-[[(5R)-2-[4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]phenyl]-4,5,6,7-tetrahydro-1,3-benzoxazol-5-yl]oxy]benzonitrile	N#CC1=CC=C(O[C@@H]2CCC3=C(C2)N=C(C2=CC=C(N4CCC(CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C2)O3)C=C1Cl	C41H37ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-H8VF2T	SCHEMBL24031852	2-chloro-4-[[(5R)-2-[4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]phenyl]-4,5,6,7-tetrahydro-1,3-benzoxazol-5-yl]-methylamino]benzonitrile	CN(C1=CC=C(C#N)C(Cl)=C1)[C@@H]1CCC2=C(C1)N=C(C1=CC=C(N3CCC(CN4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=C1)O2	C42H40ClN7O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-7G0MKI	WO2021231927A1_264	.	N#CC1=NC=C(O[C@H]2CC[C@H](NC(=O)C3=CC=C(N4CCC(CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C3)CC2)C=C1C(F)(F)F	C41H40F3N7O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-S9SUSV	SCHEMBL24031853	N-[4-[[6-cyano-5-(trifluoromethyl)pyridin-3-yl]-methylamino]cyclohexyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]benzamide	CN(C1=CN=C(C#N)C(C(F)(F)F)=C1)[C@H]1CC[C@H](NC(=O)C2=CC=C(N3CCC(CN4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=C2)CC1	C42H43F3N8O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-2CIWUG	WO2021231927A1_266	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=CC=C(N4CCC(CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C3)CC2)C=C1C(F)(F)F	C42H41F3N6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-KM83B7	WO2021231927A1_267	.	CN(C1=CC=C(C#N)C(C(F)(F)F)=C1)[C@H]1CC[C@H](NC(=O)C2=CC=C(N3CCC(CN4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=C2)CC1	C43H44F3N7O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-FC34HC	SCHEMBL24031858	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidine-1-carbonyl]benzamide; SCHEMBL26667224	CC1(C)[C@H](NC(=O)C2=CC=C(C(=O)N3CCC(CN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C44H45ClN6O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-295PQO	SCHEMBL23051613	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]piperidin-1-yl]benzamide; SCHEMBL29707058	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=CC=C(N4CCC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C3)CC2)C=C1Cl	C40H39ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-ZDV7S1	SCHEMBL24031555	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxopyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]benzamide	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(CN4C=C5C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC5=C4)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C43H43ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-4GUZLS	SCHEMBL24031556	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxopyrrolo[3,4-f]isoindol-6-yl]piperidin-1-yl]benzamide	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(N4C=C5C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC5=C4)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C42H41ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-W49J16	WO2021231927A1_272	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=CC=C(N4CCC(CN5C=C6C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC6=C5)CC4)C=C3)CC2)C=C1Cl	C41H39ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-E42UDQ	SCHEMBL24031559	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxopyrrolo[3,4-f]isoindol-6-yl]piperidin-1-yl]benzamide	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=CC=C(N4CCC(N5C=C6C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC6=C5)CC4)C=C3)CC2)C=C1Cl	C40H37ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-V6REZV	SCHEMBL26816557	N-[4-(3-chloro-4-cyano-N-methylanilino)cyclohexyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxopyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]benzamide	CN(C1=CC=C(C#N)C(Cl)=C1)[C@H]1CC[C@H](NC(=O)C2=CC=C(N3CCC(CN4C=C5C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC5=C4)CC3)C=C2)CC1	C42H42ClN7O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-KXVYUJ	SCHEMBL24031548	N-[4-(3-chloro-4-cyano-N-methylanilino)cyclohexyl]-4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxopyrrolo[3,4-f]isoindol-6-yl]piperidin-1-yl]benzamide	CN(C1=CC=C(C#N)C(Cl)=C1)[C@H]1CC[C@H](NC(=O)C2=CC=C(N3CCC(N4C=C5C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC5=C4)CC3)C=C2)CC1	C41H40ClN7O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-LV9161	SCHEMBL24031551	2-chloro-4-[4-[6-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-7,8-dihydro-5H-pyrrolo[3,4-g]isoquinolin-6-yl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]cyclohexyl]oxybenzonitrile	N#CC1=CC=C(O[C@H]2CC[C@H](N3CC4=CC(N5CCC(N6CCC7=C(C=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)C6)CC5)=CC=C4C3=O)CC2)C=C1Cl	C42H41ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-CPK4MR	SCHEMBL24031549	N-[4-(3-chloro-4-cyano-N-ethylanilino)cyclohexyl]-4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]piperidin-1-yl]benzamide	CCN(C1=CC(Cl)=C(C#N)C=C1)[C@H]1CC[C@H](NC(=O)C2=CC=C(N3CCC(N4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)CC1	C42H44ClN7O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-EIFGU4	SCHEMBL24031544	N-[4-(3-chloro-4-cyano-N-methylanilino)cyclohexyl]-4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]piperidin-1-yl]methyl]benzamide	CN(C1=CC=C(C#N)C(Cl)=C1)[C@H]1CC[C@H](NC(=O)C2=CC=C(CN3CCC(N4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=C2)CC1	C42H44ClN7O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-MW6WQ7	SCHEMBL24031545	N-[4-(3-chloro-4-cyano-N-methylanilino)cyclohexyl]-6-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]cyclohexyl]pyridine-3-carboxamide	CN(C1=CC=C(C#N)C(Cl)=C1)[C@H]1CC[C@H](NC(=O)C2=CC=C([C@H]3CC[C@H](CN4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)N=C2)CC1	C42H44ClN7O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-KNZLME	SCHEMBL24031707	N-[4-(3-chloro-4-cyano-N-methylanilino)cyclohexyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]cyclohexyl]benzamide	CN(C1=CC=C(C#N)C(Cl)=C1)[C@H]1CC[C@H](NC(=O)C2=CC=C([C@H]3CC[C@H](CN4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=C2)CC1	C43H45ClN6O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-OMQQD6	SCHEMBL24031331	N-[4-(3-chloro-4-cyano-N-methylanilino)cyclohexyl]-4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]cyclohexyl]oxybenzamide; SCHEMBL26667229; SCHEMBL26667235	CN(C1=CC=C(C#N)C(Cl)=C1)[C@H]1CC[C@H](NC(=O)C2=CC=C(O[C@H]3CC[C@H](N4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=C2)CC1	C42H43ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-OAEAIU	WO2021231927A1_282	.	CN(C1=CC=C(C#N)C(Cl)=C1)[C@H]1CC[C@H](NC(=O)C2=CC=C(O[C@H]3CC[C@H](N4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)N=C2)CC1	C41H42ClN7O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-O2UWP4	SCHEMBL26802294	N-[4-(3-chloro-4-cyano-N-methylanilino)cyclohexyl]-5-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]piperidin-1-yl]methyl]pyridine-2-carboxamide	CN(C1=CC=C(C#N)C(Cl)=C1)[C@H]1CC[C@H](NC(=O)C2=CC=C(CN3CCC(N4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=N2)CC1	C41H43ClN8O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-6DA7W5	SCHEMBL24031709	N-[4-(3-chloro-4-cyano-N-methylanilino)cyclohexyl]-2-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]piperidin-1-yl]methyl]pyrimidine-5-carboxamide	CN(C1=CC=C(C#N)C(Cl)=C1)[C@H]1CC[C@H](NC(=O)C2=CN=C(CN3CCC(N4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)N=C2)CC1	C40H42ClN9O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-2WZDRK	SCHEMBL24031793	N-[4-(3-chloro-4-cyano-N-methylanilino)cyclohexyl]-6-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]piperidin-1-yl]methyl]pyridazine-3-carboxamide	CN(C1=CC=C(C#N)C(Cl)=C1)[C@H]1CC[C@H](NC(=O)C2=CC=C(CN3CCC(N4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)N=N2)CC1	C40H42ClN9O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-JLI5C0	SCHEMBL24031796	N-[4-(3-chloro-4-cyano-N-methylanilino)cyclohexyl]-5-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]cyclohexyl]pyridine-2-carboxamide	CN(C1=CC=C(C#N)C(Cl)=C1)[C@H]1CC[C@H](NC(=O)C2=CC=C([C@H]3CC[C@H](CN4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=N2)CC1	C42H44ClN7O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-JPLV3G	SCHEMBL24031798	N-[4-(3-chloro-4-cyano-N-methylanilino)cyclohexyl]-6-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]cyclohexyl]pyridazine-3-carboxamide	CN(C1=CC=C(C#N)C(Cl)=C1)[C@H]1CC[C@H](NC(=O)C2=CC=C([C@H]3CC[C@H](CN4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)N=N2)CC1	C41H43ClN8O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-INV193	SCHEMBL24031791	N-[4-(3-chloro-4-cyano-N-methylanilino)cyclohexyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]cyclohexyl]oxybenzamide	CN(C1=CC=C(C#N)C(Cl)=C1)[C@H]1CC[C@H](NC(=O)C2=CC=C(O[C@H]3CC[C@H](CN4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=C2)CC1	C43H45ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-7X39IP	SCHEMBL24031797	N-[4-(3-chloro-4-cyano-N-methylanilino)cyclohexyl]-6-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]cyclohexyl]oxypyridine-3-carboxamide	CN(C1=CC=C(C#N)C(Cl)=C1)[C@H]1CC[C@H](NC(=O)C2=CC=C(O[C@H]3CC[C@H](CN4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)N=C2)CC1	C42H44ClN7O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-Z5FMUU	SCHEMBL24031792	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]piperidin-1-yl]methyl]benzamide	CC1(C)[C@H](NC(=O)C2=CC=C(CN3CCC(N4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C43H45ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-PR8K6A	SCHEMBL24031975	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]cyclohexyl]-methylamino]benzamide	CN(C1=CC=C(C(=O)N[C@H]2C(C)(C)[C@H](OC3=CC=C(C#N)C(Cl)=C3)C2(C)C)C=C1)[C@H]1CC[C@H](N2CC3=CC4=C(C=C3C2)C(=O)N(C2CCC(=O)NC2=O)C4=O)CC1	C44H47ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-UEBVUC	SCHEMBL24031973	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]cyclohexyl]amino]benzamide	CC1(C)[C@H](NC(=O)C2=CC=C(N[C@H]3CC[C@H](N4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C43H45ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-EYLYXB	SCHEMBL24031974	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]cyclohexyl]pyridine-3-carboxamide	CC1(C)[C@H](NC(=O)C2=CN=C([C@H]3CC[C@H](CN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C43H45ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-1VKB4T	SCHEMBL24031971	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-5-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]cyclohexyl]pyridine-2-carboxamide	CC1(C)[C@H](NC(=O)C2=NC=C([C@H]3CC[C@H](CN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C43H45ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-YNC6V5	SCHEMBL24031978	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-2-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]cyclohexyl]pyrimidine-5-carboxamide	CC1(C)[C@H](NC(=O)C2=CN=C([C@H]3CC[C@H](CN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)N=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C42H44ClN7O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-ZNE459	SCHEMBL24031976	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]cyclohexyl]pyridazine-3-carboxamide	CC1(C)[C@H](NC(=O)C2=NN=C([C@H]3CC[C@H](CN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C42H44ClN7O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-J2SPF5	SCHEMBL24031815	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]cyclohexyl]oxypyridine-3-carboxamide	CC1(C)[C@H](NC(=O)C2=CN=C(O[C@H]3CC[C@H](N4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C42H43ClN6O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-D7H63X	SCHEMBL24031823	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-5-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]cyclohexyl]oxypyridine-2-carboxamide	CC1(C)[C@H](NC(=O)C2=NC=C(O[C@H]3CC[C@H](N4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C42H43ClN6O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-WSIS32	SCHEMBL24031811	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-2-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]cyclohexyl]oxypyrimidine-5-carboxamide	CC1(C)[C@H](NC(=O)C2=CN=C(O[C@H]3CC[C@H](N4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)N=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C41H42ClN7O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-24OZSM	SCHEMBL24031813	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]cyclohexyl]oxypyridazine-3-carboxamide	CC1(C)[C@H](NC(=O)C2=NN=C(O[C@H]3CC[C@H](N4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C41H42ClN7O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-FWVVBZ	SCHEMBL24031810	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[[8-(2,6-dioxopiperidin-3-yl)-7,9-dioxo-3,5-dihydro-2H-pyrrolo[3,4-h][1,4]benzoxazepin-4-yl]methyl]piperidin-1-yl]benzamide	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(CN4CCOC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C44H47ClN6O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-SGUMAU	SCHEMBL24031816	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[8-(2,6-dioxopiperidin-3-yl)-7,9-dioxo-3,5-dihydro-2H-pyrrolo[3,4-h][1,4]benzoxazepin-4-yl]piperidin-1-yl]benzamide	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(N4CCOC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C43H45ClN6O7	AR	P10275	CRBN	WO-2021231927-A1
TPD-SYTU1S	WO2021231927A1_303	.	C=NC1=CC=C(N(C)[C@H]2CC[C@H](NC(=O)C3=CC=C(N4CCC(CN5CCOC6=CC7=C(C=C6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)C=C3)CC2)C=C1Cl	C43H48ClN7O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-FYCGIP	SCHEMBL24031928	N-[4-(3-chloro-4-cyano-N-methylanilino)cyclohexyl]-4-[4-[8-(2,6-dioxopiperidin-3-yl)-7,9-dioxo-3,5-dihydro-2H-pyrrolo[3,4-h][1,4]benzoxazepin-4-yl]piperidin-1-yl]benzamide	CN(C1=CC=C(C#N)C(Cl)=C1)[C@H]1CC[C@H](NC(=O)C2=CC=C(N3CCC(N4CCOC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)CC1	C42H44ClN7O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-FSMYC4	SCHEMBL24031931	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,6,8,9-tetrahydropyrrolo[3,4-h][3]benzazepin-7-yl]methyl]piperidin-1-yl]benzamide	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(CN4CCC5=CC6=C(C=C5CC4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C45H49ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-TFIJ30	SCHEMBL24031934	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7,8,9-tetrahydropyrrolo[3,4-h][2]benzazepin-6-yl]methyl]piperidin-1-yl]benzamide	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(CN4CCCC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C45H49ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-LI96BN	SCHEMBL24031938	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]propyl]piperidin-1-yl]benzamide	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(CCCN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C45H49ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-2OIS7P	SCHEMBL24031929	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]piperidin-1-yl]piperidin-1-yl]benzamide	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(N4CCC(N5CC6=CC7=C(C=C6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C47H52ClN7O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-ULNZHK	SCHEMBL24031930	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]methyl]benzamide	CC1(C)[C@H](NC(=O)C2=CC=C(CN3CCC(CN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C44H47ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-OJTEN3	SCHEMBL24031566	N-[4-(3-chloro-4-cyano-N-methylanilino)cyclohexyl]-6-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]piperidin-1-yl]methyl]pyridine-3-carboxamide	CN(C1=CC=C(C#N)C(Cl)=C1)[C@H]1CC[C@H](NC(=O)C2=CC=C(CN3CCC(N4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)N=C2)CC1	C41H43ClN8O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-2VNOA4	SCHEMBL24031970	N-[4-(3-chloro-4-cyano-N-methylanilino)cyclohexyl]-4-[4-[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]azetidin-1-yl]piperidin-1-yl]benzamide	CN(C1=CC=C(C#N)C(Cl)=C1)[C@H]1CC[C@H](NC(=O)C2=CC=C(N3CCC(N4CC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)C4)CC3)C=C2)CC1	C44H47ClN8O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-B79RFZ	SCHEMBL26802302	N-[4-(3-chloro-4-cyano-N-methylanilino)cyclohexyl]-4-[4-[3-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]azetidin-1-yl]piperidin-1-yl]benzamide	CN(C1=CC=C(C#N)C(Cl)=C1)[C@H]1CC[C@H](NC(=O)C2=CC=C(N3CCC(N4CC(CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)C4)CC3)C=C2)CC1	C45H49ClN8O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-03BV6S	SCHEMBL24031979	N-[4-(3-chloro-4-cyano-N-methylanilino)cyclohexyl]-4-[4-[[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]azetidin-1-yl]methyl]piperidin-1-yl]benzamide; SCHEMBL26802306	CN(C1=CC=C(C#N)C(Cl)=C1)[C@H]1CC[C@H](NC(=O)C2=CC=C(N3CCC(CN4CC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)C4)CC3)C=C2)CC1	C45H49ClN8O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-EZ2Y6P	SCHEMBL26802313	N-[4-(3-chloro-4-cyano-N-methylanilino)cyclohexyl]-5-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]pyridine-2-carboxamide	CN(C1=CC=C(C#N)C(Cl)=C1)[C@H]1CC[C@H](NC(=O)C2=CC=C(N3CCC(CN4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=N2)CC1	C41H43ClN8O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-L4PQHY	SCHEMBL24031362	N-[4-(3-chloro-4-cyano-N-methylanilino)cyclohexyl]-4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindole-6-carbonyl]piperidin-1-yl]methyl]benzamide	CN(C1=CC(Cl)=C(C#N)C=C1)[C@H]1CC[C@H](NC(=O)C2=CC=C(CN3CCC(C(=O)N4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6)CC3)C=C2)CC1	C43H46ClN7O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-DVZUVT	SCHEMBL24031360	N-[4-(3-chloro-4-cyano-N-methylanilino)cyclohexyl]-4-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-6-yl]-2-oxoethyl]piperazin-1-yl]benzamide; SCHEMBL26667244	CN(C1=CC(Cl)=C(C#N)C=C1)[C@H]1CC[C@H](NC(=O)C2=CC=C(N3CCN(CC(=O)N4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6)CC3)C=C2)CC1	C42H45ClN8O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-RLNUHD	SCHEMBL24031361	N-[4-(3-chloro-4-cyano-N-methylanilino)cyclohexyl]-4-[1-[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-6-yl]-2-oxoethyl]piperidin-4-yl]benzamide; SCHEMBL26667222	CN(C1=CC(Cl)=C(C#N)C=C1)[C@H]1CC[C@H](NC(=O)C2=CC=C(C3CCN(CC(=O)N4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6)CC3)C=C2)CC1	C43H46ClN7O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-HS9I20	SCHEMBL24031372	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-4-[4-[[2-[(3R)-2,6-dioxopiperidin-3-yl]-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]benzamide	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=CC=C(N4CCC(CN5CC6=C(C=C7C(=O)N([C@@H]8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C3)CC2)C=C1Cl	C41H41ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-FNTJ80	SCHEMBL24031363	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-4-[4-[[2-[(3S)-2,6-dioxopiperidin-3-yl]-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]benzamide	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=CC=C(N4CCC(CN5CC6=C(C=C7C(=O)N([C@H]8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C3)CC2)C=C1Cl	C41H41ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-YO4SQ0	SCHEMBL24031364	N-[4-(3-chloro-4-cyano-N-methylanilino)cyclohexyl]-4-[4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]piperidin-1-yl]benzamide	CN(C1=CC=C(C#N)C(Cl)=C1)[C@H]1CC[C@H](NC(=O)C2=CC=C(N3CCC(N4CC5=C(C=C6C(=O)N([C@H]7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=C2)CC1	C41H42ClN7O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-I7OD6N	SCHEMBL24031654	N-[4-(3-chloro-4-cyano-N-methylanilino)cyclohexyl]-4-[4-[2-[(3R)-2,6-dioxopiperidin-3-yl]-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]piperidin-1-yl]benzamide	CN(C1=CC=C(C#N)C(Cl)=C1)[C@H]1CC[C@H](NC(=O)C2=CC=C(N3CCC(N4CC5=C(C=C6C(=O)N([C@@H]7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=C2)CC1	C41H42ClN7O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-DOQ6RG	SCHEMBL24031411	N-[4-(3-chloro-4-cyano-N-methylanilino)cyclohexyl]-4-[4-[[2-[(3S)-2,6-dioxopiperidin-3-yl]-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]benzamide	CN(C1=CC=C(C#N)C(Cl)=C1)[C@H]1CC[C@H](NC(=O)C2=CC=C(N3CCC(CN4CC5=C(C=C6C(=O)N([C@H]7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=C2)CC1	C42H44ClN7O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-X5CBLB	SCHEMBL24031648	N-[4-(3-chloro-4-cyano-N-methylanilino)cyclohexyl]-4-[4-[[2-[(3R)-2,6-dioxopiperidin-3-yl]-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]benzamide	CN(C1=CC=C(C#N)C(Cl)=C1)[C@H]1CC[C@H](NC(=O)C2=CC=C(N3CCC(CN4CC5=C(C=C6C(=O)N([C@@H]7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=C2)CC1	C42H44ClN7O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-84GDIN	SCHEMBL24031670	N-[4-(3-chloro-4-cyano-N-ethylanilino)cyclohexyl]-4-[4-[[2-[(3S)-2,6-dioxopiperidin-3-yl]-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]benzamide	CCN(C1=CC=C(C#N)C(Cl)=C1)[C@H]1CC[C@H](NC(=O)C2=CC=C(N3CCC(CN4CC5=C(C=C6C(=O)N([C@H]7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=C2)CC1	C43H46ClN7O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-XF4RUC	SCHEMBL24031655	N-[4-(3-chloro-4-cyano-N-ethylanilino)cyclohexyl]-4-[4-[[2-[(3R)-2,6-dioxopiperidin-3-yl]-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]benzamide	CCN(C1=CC=C(C#N)C(Cl)=C1)[C@H]1CC[C@H](NC(=O)C2=CC=C(N3CCC(CN4CC5=C(C=C6C(=O)N([C@@H]7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=C2)CC1	C43H46ClN7O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-IFABDQ	SCHEMBL24031656	N-[4-(3-chloro-4-cyano-N-methylanilino)cyclohexyl]-4-[4-[[2-[(3S)-2,6-dioxopiperidin-3-yl]-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]cyclohexyl]benzamide	CN(C1=CC=C(C#N)C(Cl)=C1)[C@H]1CC[C@H](NC(=O)C2=CC=C([C@H]3CC[C@H](CN4CC5=C(C=C6C(=O)N([C@H]7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=C2)CC1	C43H45ClN6O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-CGSCQL	SCHEMBL24031669	N-[4-(3-chloro-4-cyano-N-methylanilino)cyclohexyl]-4-[4-[[2-[(3R)-2,6-dioxopiperidin-3-yl]-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]cyclohexyl]benzamide	CN(C1=CC=C(C#N)C(Cl)=C1)[C@H]1CC[C@H](NC(=O)C2=CC=C([C@H]3CC[C@H](CN4CC5=C(C=C6C(=O)N([C@@H]7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=C2)CC1	C43H45ClN6O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-XFHFSN	SCHEMBL24031663	N-[4-(3-chloro-4-cyano-N-methylanilino)cyclohexyl]-5-[4-[[2-[(3S)-2,6-dioxopiperidin-3-yl]-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]cyclohexyl]pyridine-2-carboxamide	CN(C1=CC=C(C#N)C(Cl)=C1)[C@H]1CC[C@H](NC(=O)C2=CC=C([C@H]3CC[C@H](CN4CC5=C(C=C6C(=O)N([C@H]7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=N2)CC1	C42H44ClN7O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-DE662K	SCHEMBL26819294	N-[4-(3-chloro-4-cyano-N-methylanilino)cyclohexyl]-5-[4-[[2-[(3R)-2,6-dioxopiperidin-3-yl]-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]cyclohexyl]pyridine-2-carboxamide	CN(C1=CC=C(C#N)C(Cl)=C1)[C@H]1CC[C@H](NC(=O)C2=CC=C([C@H]3CC[C@H](CN4CC5=C(C=C6C(=O)N([C@@H]7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=N2)CC1	C42H44ClN7O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-8NG78A	SCHEMBL24031652	N-[4-(3-chloro-4-cyano-N-methylanilino)cyclohexyl]-4-[4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]cyclohexyl]oxybenzamide	CN(C1=CC=C(C#N)C(Cl)=C1)[C@H]1CC[C@H](NC(=O)C2=CC=C(O[C@H]3CC[C@H](N4CC5=C(C=C6C(=O)N([C@H]7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=C2)CC1	C42H43ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-7ZEH5L	SCHEMBL24031653	N-[4-(3-chloro-4-cyano-N-methylanilino)cyclohexyl]-4-[4-[2-[(3R)-2,6-dioxopiperidin-3-yl]-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]cyclohexyl]oxybenzamide	CN(C1=CC=C(C#N)C(Cl)=C1)[C@H]1CC[C@H](NC(=O)C2=CC=C(O[C@H]3CC[C@H](N4CC5=C(C=C6C(=O)N([C@@H]7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=C2)CC1	C42H43ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-93414Z	SCHEMBL24031664	N-[4-(3-chloro-4-cyano-N-methylanilino)cyclohexyl]-4-[[4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindole-6-carbonyl]piperidin-1-yl]methyl]benzamide	CN(C1=CC(Cl)=C(C#N)C=C1)[C@H]1CC[C@H](NC(=O)C2=CC=C(CN3CCC(C(=O)N4CC5=CC6=C(C=C5C4)C(=O)N([C@H]4CCC(=O)NC4=O)C6)CC3)C=C2)CC1	C43H46ClN7O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-2AC4NY	SCHEMBL24031368	N-[4-(3-chloro-4-cyano-N-methylanilino)cyclohexyl]-4-[[4-[2-[(3R)-2,6-dioxopiperidin-3-yl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindole-6-carbonyl]piperidin-1-yl]methyl]benzamide	CN(C1=CC(Cl)=C(C#N)C=C1)[C@H]1CC[C@H](NC(=O)C2=CC=C(CN3CCC(C(=O)N4CC5=CC6=C(C=C5C4)C(=O)N([C@@H]4CCC(=O)NC4=O)C6)CC3)C=C2)CC1	C43H46ClN7O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-EO7904	SCHEMBL24031356	N-[4-(3-chloro-4-cyano-N-methylanilino)cyclohexyl]-4-[4-[2-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-6-yl]-2-oxoethyl]piperazin-1-yl]benzamide	CN(C1=CC(Cl)=C(C#N)C=C1)[C@H]1CC[C@H](NC(=O)C2=CC=C(N3CCN(CC(=O)N4CC5=CC6=C(C=C5C4)C(=O)N([C@H]4CCC(=O)NC4=O)C6)CC3)C=C2)CC1	C42H45ClN8O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-IPGYBI	SCHEMBL24031367	N-[4-(3-chloro-4-cyano-N-methylanilino)cyclohexyl]-4-[4-[2-[2-[(3R)-2,6-dioxopiperidin-3-yl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-6-yl]-2-oxoethyl]piperazin-1-yl]benzamide	CN(C1=CC(Cl)=C(C#N)C=C1)[C@H]1CC[C@H](NC(=O)C2=CC=C(N3CCN(CC(=O)N4CC5=CC6=C(C=C5C4)C(=O)N([C@@H]4CCC(=O)NC4=O)C6)CC3)C=C2)CC1	C42H45ClN8O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-U1M56I	SCHEMBL24031370	N-[4-(3-chloro-4-cyano-N-methylanilino)cyclohexyl]-4-[[4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]piperidin-1-yl]methyl]benzamide	CN(C1=CC=C(C#N)C(Cl)=C1)[C@H]1CC[C@H](NC(=O)C2=CC=C(CN3CCC(N4CC5=C(C=C6C(=O)N([C@H]7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=C2)CC1	C42H44ClN7O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-TEJAQA	SCHEMBL24031358	N-[4-(3-chloro-4-cyano-N-methylanilino)cyclohexyl]-4-[[4-[2-[(3R)-2,6-dioxopiperidin-3-yl]-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]piperidin-1-yl]methyl]benzamide	CN(C1=CC=C(C#N)C(Cl)=C1)[C@H]1CC[C@H](NC(=O)C2=CC=C(CN3CCC(N4CC5=C(C=C6C(=O)N([C@@H]7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=C2)CC1	C42H44ClN7O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-XHFODU	WO2021231927A1_349	.	[H]C1(OC2=CC=C(C#N)C(Cl)=C2)CC2CCC(C1)N2C1=CC=C(C(=O)N2CCC(CN3CC4=CC5=C(C=C4C3)C(=O)N([C@@H]3CCC(=O)NC3=O)C5=O)CC2)C=C1	C42H41ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-F480F0	SCHEMBL24031371	2-chloro-4-[[8-[4-[4-[[2-[(3S)-2,6-dioxopiperidin-3-yl]-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidine-1-carbonyl]phenyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzonitrile	[H]C1(OC2=CC=C(C#N)C(Cl)=C2)CC2CCC(C1)N2C1=CC=C(C(=O)N2CCC(CN3CC4=CC5=C(C=C4C3)C(=O)N([C@H]3CCC(=O)NC3=O)C5=O)CC2)C=C1	C42H41ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-WCTILD	SCHEMBL24031645	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[[2-[(3R)-2,6-dioxopiperidin-3-yl]-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]benzamide	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(CN4CC5=CC6=C(C=C5C4)C(=O)N([C@@H]4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C43H45ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-NM7T89	SCHEMBL24031629	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[[2-[(3S)-2,6-dioxopiperidin-3-yl]-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]benzamide	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(CN4CC5=CC6=C(C=C5C4)C(=O)N([C@H]4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C43H45ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-L5DH6N	SCHEMBL24031630	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[2-[2-[(3R)-2,6-dioxopiperidin-3-yl]-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]ethyl]piperidin-1-yl]benzamide	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(CCN4CC5=CC6=C(C=C5C4)C(=O)N([C@@H]4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C44H47ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-3KS3Q4	SCHEMBL24031636	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[2-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]ethyl]piperidin-1-yl]benzamide	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(CCN4CC5=CC6=C(C=C5C4)C(=O)N([C@H]4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C44H47ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-VZYBFB	SCHEMBL24031637	2-chloro-4-[3-[4-[4-[2-[(3R)-2,6-dioxopiperidin-3-yl]-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]piperidine-1-carbonyl]anilino]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](NC2=CC=C(C(=O)N3CCC(N4CC5=CC6=C(C=C5C4)C(=O)N([C@@H]4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C42H43ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-AC9Y5I	SCHEMBL24031631	2-chloro-4-[3-[4-[4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]piperidine-1-carbonyl]anilino]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](NC2=CC=C(C(=O)N3CCC(N4CC5=CC6=C(C=C5C4)C(=O)N([C@H]4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C42H43ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-CA7APV	SCHEMBL24031639	2-chloro-4-[3-[4-[4-[[2-[(3R)-2,6-dioxopiperidin-3-yl]-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidine-1-carbonyl]anilino]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](NC2=CC=C(C(=O)N3CCC(CN4CC5=CC6=C(C=C5C4)C(=O)N([C@@H]4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C43H45ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-EBZZM5	SCHEMBL24031641	2-chloro-4-[3-[4-[4-[[2-[(3S)-2,6-dioxopiperidin-3-yl]-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidine-1-carbonyl]anilino]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](NC2=CC=C(C(=O)N3CCC(CN4CC5=CC6=C(C=C5C4)C(=O)N([C@H]4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C43H45ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-AGPU3O	SCHEMBL24031574	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[[2-[(3R)-2,6-dioxopiperidin-3-yl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]benzamide	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(CN4CC5=CC6=C(C=C5C4)C(=O)N([C@@H]4CCC(=O)NC4=O)C6)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C43H47ClN6O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-XJX273	SCHEMBL24031593	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]benzamide	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(CN4CC5=CC6=C(C=C5C4)C(=O)N([C@H]4CCC(=O)NC4=O)C6)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C43H47ClN6O5	AR	P10275	CRBN	WO-2021231927-A1
TPD-LAPUIW	SCHEMBL24031576	N-[(1S,3S)-3-(3-chloro-4-cyanophenoxy)-2,2-dimethylcyclobutyl]-4-[4-[[2-[(3R)-2,6-dioxopiperidin-3-yl]-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]benzamide	CC1(C)[C@@H](NC(=O)C2=CC=C(N3CCC(CN4CC5=CC6=C(C=C5C4)C(=O)N([C@@H]4CCC(=O)NC4=O)C6=O)CC3)C=C2)C[C@@H]1OC1=CC=C(C#N)C(Cl)=C1	C41H41ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-M412GS	SCHEMBL24031581	N-[(1S,3S)-3-(3-chloro-4-cyanophenoxy)-2,2-dimethylcyclobutyl]-4-[4-[[2-[(3S)-2,6-dioxopiperidin-3-yl]-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]benzamide	CC1(C)[C@@H](NC(=O)C2=CC=C(N3CCC(CN4CC5=CC6=C(C=C5C4)C(=O)N([C@H]4CCC(=O)NC4=O)C6=O)CC3)C=C2)C[C@@H]1OC1=CC=C(C#N)C(Cl)=C1	C41H41ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-74VIXA	SCHEMBL24031577	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[[2-[(3R)-2,6-dioxopiperidin-3-yl]-1,3-dioxo-6,7-dihydro-5H-cyclopenta[f]isoindol-6-yl]methyl]piperazin-1-yl]benzamide	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCN(CC4CC5=CC6=C(C=C5C4)C(=O)N([C@@H]4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C43H45ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-3FRZT9	SCHEMBL24031586	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[[2-[(3S)-2,6-dioxopiperidin-3-yl]-1,3-dioxo-6,7-dihydro-5H-cyclopenta[f]isoindol-6-yl]methyl]piperazin-1-yl]benzamide	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCN(CC4CC5=CC6=C(C=C5C4)C(=O)N([C@H]4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C43H45ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-E5MX3F	SCHEMBL24031583	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[3-[2-[(3R)-2,6-dioxopiperidin-3-yl]-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]propyl]piperidin-1-yl]benzamide	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(CCCN4CC5=CC6=C(C=C5C4)C(=O)N([C@@H]4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C45H49ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-GTGJ12	SCHEMBL24031594	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[3-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]propyl]piperidin-1-yl]benzamide	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(CCCN4CC5=CC6=C(C=C5C4)C(=O)N([C@H]4CCC(=O)NC4=O)C6=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C45H49ClN6O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-21RSM9	SCHEMBL24031310	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[4-[2-[(3R)-2,6-dioxopiperidin-3-yl]-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]piperidin-1-yl]piperidin-1-yl]benzamide	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(N4CCC(N5CC6=CC7=C(C=C6C5)C(=O)N([C@@H]5CCC(=O)NC5=O)C7=O)CC4)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C47H52ClN7O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-1KI6KC	SCHEMBL24031311	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]piperidin-1-yl]piperidin-1-yl]benzamide	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(N4CCC(N5CC6=CC7=C(C=C6C5)C(=O)N([C@H]5CCC(=O)NC5=O)C7=O)CC4)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C47H52ClN7O6	AR	P10275	CRBN	WO-2021231927-A1
TPD-XWJB3G	SCHEMBL24142007	(2S)-2-[[4-[(2,4-diaminopteridin-6-yl)methyl-methylamino]benzoyl]amino]-5-[2-[2-[2-[2-[2-[[1-[(4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]ethoxy]ethoxy]ethoxy]ethylamino]-5-oxopentanoic acid	Cc1ncsc1-c1ccc(CNC(=O)C2C[C@@H](O)CN2C(=O)C(NC(=O)COCCOCCOCCOCCNC(=O)CC[C@H](NC(=O)c2ccc(N(C)Cc3cnc4nc(N)nc(N)c4n3)cc2)C(=O)O)C(C)(C)C)cc1	C52H69N13O12S	DHFR	P00374	VHL	WO-2021262693-A1
TPD-84QPRR	SCHEMBL24142016	(2S)-2-[[4-[(2,4-diaminopteridin-6-yl)methyl-methylamino]benzoyl]amino]-5-[2-[2-[2-[[1-[(4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]ethoxy]ethylamino]-5-oxopentanoic acid	Cc1ncsc1-c1ccc(CNC(=O)C2C[C@@H](O)CN2C(=O)C(NC(=O)COCCOCCNC(=O)CC[C@H](NC(=O)c2ccc(N(C)Cc3cnc4nc(N)nc(N)c4n3)cc2)C(=O)O)C(C)(C)C)cc1	C48H61N13O10S	DHFR	P00374	VHL	WO-2021262693-A1
TPD-LA1P12	SCHEMBL24142052	(2S)-2-[[4-[(2,4-diaminopteridin-6-yl)methyl-methylamino]benzoyl]amino]-5-[6-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]hexylamino]-5-oxopentanoic acid	CN(Cc1cnc2nc(N)nc(N)c2n1)c1ccc(C(=O)N[C@@H](CCC(=O)NCCCCCCNc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)C(=O)O)cc1	C39H44N12O8	DHFR	P00374	CRBN	WO-2021262693-A1
TPD-MRQIB7	SCHEMBL24142027	(2S)-2-[[4-[(2,4-diaminopteridin-6-yl)methyl-methylamino]benzoyl]amino]-5-[4-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]acetyl]amino]butylamino]-5-oxopentanoic acid; SCHEMBL30638283	CN(Cc1cnc2nc(N)nc(N)c2n1)c1ccc(C(=O)N[C@@H](CCC(=O)NCCCCNC(=O)CNc2cccc3c2CN(C2CCC(=O)NC2=O)C3=O)C(=O)O)cc1	C39H45N13O8	DHFR	P00374	CRBN	WO-2021262693-A1
TPD-UYDM8J	SCHEMBL24142053	(2S)-2-[[4-[(2,4-diaminopteridin-6-yl)methyl-methylamino]benzoyl]amino]-5-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]butylamino]-5-oxopentanoic acid; SCHEMBL30638288	CN(Cc1cnc2nc(N)nc(N)c2n1)c1ccc(C(=O)N[C@@H](CCC(=O)NCCCCc2cccc3c2CN(C2CCC(=O)NC2=O)C3=O)C(=O)O)cc1	C37H41N11O7	DHFR	P00374	CRBN	WO-2021262693-A1
TPD-B31OLW	WO2021262693A1_NCGC00687472	.	COC(O)[C@H](CCC(=O)NCCCCCCCCNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O)NC(=O)c1ccc(N(C)Cc2cnc3nc(N)nc(N)c3n2)cc1	C42H52N12O8	DHFR	P00374	CRBN	WO-2021262693-A1
TPD-8R4P16	SCHEMBL24141981	(2S)-2-[[4-[(2,4-diaminopteridin-6-yl)methyl-methylamino]benzoyl]amino]-5-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethylamino]-5-oxopentanoic acid	CN(Cc1cnc2nc(N)nc(N)c2n1)c1ccc(C(=O)N[C@@H](CCC(=O)NCCOCCOCCNc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)C(=O)O)cc1	C39H44N12O10	DHFR	P00374	CRBN	WO-2021262693-A1
TPD-DCCMC2	WO2021262693A1_NCGC00687569	.	COC(=O)[C@H](CCC(=O)NCCCCCCCCNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O)NC(=O)CC[C@H](NC(=O)c1ccc(N(C)CC2=NC3=C(N)N=C(N)NC3N=C2)cc1)C(=O)OC	C48H61N13O11	DHFR	P00374	CRBN	WO-2021262693-A1
TPD-FT2W3S	SCHEMBL24141992	(2S)-2-[[4-[(2,4-diaminopteridin-6-yl)methyl-methylamino]benzoyl]amino]-5-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethylamino]-5-oxopentanoic acid; SCHEMBL30638296	CN(Cc1cnc2nc(N)nc(N)c2n1)c1ccc(C(=O)N[C@@H](CCC(=O)NCCOCCNc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)C(=O)O)cc1	C37H40N12O9	DHFR	P00374	CRBN	WO-2021262693-A1
TPD-8NH545	SCHEMBL24142029	(2S)-2-[[4-[(2,4-diaminopteridin-6-yl)methyl-methylamino]benzoyl]amino]-5-[[(2S)-5-[8-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]octylamino]-1-methoxy-1,5-dioxopentan-2-yl]amino]-5-oxopentanoic acid	COC(=O)[C@H](CCC(=O)NCCCCCCCCNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O)NC(=O)CC[C@H](NC(=O)c1ccc(N(C)Cc2cnc3nc(N)nc(N)c3n2)cc1)C(=O)O	C47H57N13O11	DHFR	P00374	CRBN	WO-2021262693-A1
TPD-3E8CIR	SCHEMBL26966103	(2S)-2-[[4-[(2,4-diaminopteridin-6-yl)methyl-methylamino]benzoyl]amino]-5-[[(2S)-5-[[(2S)-5-[[(2S)-5-[8-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]octylamino]-1-methoxy-1,5-dioxopentan-2-yl]amino]-1-methoxy-1,5-dioxopentan-2-yl]amino]-1-methoxy-1,5-dioxopentan-2-yl]amino]-5-oxopentanoic acid	COC(=O)[C@H](CCC(=O)NCCCCCCCCNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O)NC(=O)CC[C@H](NC(=O)CC[C@H](NC(=O)CC[C@H](NC(=O)c1ccc(N(C)Cc2cnc3nc(N)nc(N)c3n2)cc1)C(=O)O)C(=O)OC)C(=O)OC	C59H75N15O17	DHFR	P00374	CRBN	WO-2021262693-A1
TPD-H7G62Z	WO2021262693A1_NCGC00687811	.	COC(=O)C(CCC(=O)NCCCCCCCCNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O)NC(=O)CC[C@H](NC(=O)CC[C@H](NC(=O)CC[C@H](NC(=O)CC[C@H](NC(=O)c1ccc(N(C)Cc2cnc3nc(N)nc(N)c3n2)cc1)C(=O)O)C(=O)OC)C(=O)OC)C(=O)OC	C65H84N16O20	DHFR	P00374	CRBN	WO-2021262693-A1
TPD-N6YRRL	SCHEMBL24142094	(2S)-2-[[4-[2-(2-amino-4-oxo-3,7-dihydropyrrolo[2,3-d]pyrimidin-5-yl)ethyl]benzoyl]amino]-5-[8-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]octylamino]-5-oxopentanoic acid	Nc1nc2[nH]cc(CCc3ccc(C(=O)N[C@@H](CCC(=O)NCCCCCCCCNc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)C(=O)O)cc3)c2c(=O)[nH]1	C41H47N9O9	DHFR	P00374	CRBN	WO-2021262693-A1
TPD-674EMH	SCHEMBL24142092	(2S)-2-[[4-[2-(2-amino-4-oxo-3,7-dihydropyrrolo[2,3-d]pyrimidin-5-yl)ethyl]benzoyl]amino]-5-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethylamino]-5-oxopentanoic acid	Nc1nc2[nH]cc(CCc3ccc(C(=O)N[C@@H](CCC(=O)NCCOCCOCCNc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)C(=O)O)cc3)c2c(=O)[nH]1	C39H43N9O11	DHFR	P00374	CRBN	WO-2021262693-A1
TPD-QP8AAV	SCHEMBL24142011	(2S)-2-[[4-[2-(2-amino-4-oxo-3,7-dihydropyrrolo[2,3-d]pyrimidin-5-yl)ethyl]benzoyl]amino]-5-[2-[2-[2-[2-[[1-[(4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]ethoxy]ethoxy]ethylamino]-5-oxopentanoic acid	Cc1ncsc1-c1ccc(CNC(=O)C2C[C@@H](O)CN2C(=O)C(NC(=O)COCCOCCOCCNC(=O)CC[C@H](NC(=O)c2ccc(CCc3c[nH]c4nc(N)[nH]c(=O)c34)cc2)C(=O)O)C(C)(C)C)cc1	C50H64N10O12S	DHFR	P00374	VHL	WO-2021262693-A1
TPD-ZZO60O	SCHEMBL24142012	(2S)-2-[[4-[2-(2-amino-4-oxo-3,7-dihydropyrrolo[2,3-d]pyrimidin-5-yl)ethyl]benzoyl]amino]-5-[2-[2-[2-[[1-[(4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]ethoxy]ethylamino]-5-oxopentanoic acid	Cc1ncsc1-c1ccc(CNC(=O)C2C[C@@H](O)CN2C(=O)C(NC(=O)COCCOCCNC(=O)CC[C@H](NC(=O)c2ccc(CCc3c[nH]c4nc(N)[nH]c(=O)c34)cc2)C(=O)O)C(C)(C)C)cc1	C48H60N10O11S	DHFR	P00374	VHL	WO-2021262693-A1
TPD-3GMSYH	WO2021262693A1_NCGC00690075	.	Nc1nc(N)c2nc(CNc3ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)NCCCCCCCCNc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)cc3)cnc2n1	C40H46N12O8	DHFR	P00374	CRBN	WO-2021262693-A1
TPD-R8KG82	SCHEMBL24142051	(2S)-2-[[4-[(2,4-diaminopteridin-6-yl)methyl-[6-[3-[2-[2-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]propanoylamino]hexyl]amino]benzoyl]amino]pentanedioic acid	Nc1nc(N)c2nc(CN(CCCCCCNC(=O)CCOCCOCCOCCOCCOc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)c3ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)cc3)cnc2n1	C49H61N11O15	DHFR	P00374	CRBN	WO-2021262693-A1
TPD-H1WY6M	SCHEMBL24142050	(2S)-2-[[4-[(2,4-diaminopteridin-6-yl)methyl-[6-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyacetyl]amino]hexyl]amino]benzoyl]amino]pentanedioic acid	Nc1nc(N)c2nc(CN(CCCCCCNC(=O)COc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)c3ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)cc3)cnc2n1	C40H43N11O11	DHFR	P00374	CRBN	WO-2021262693-A1
TPD-8V7JU0	SCHEMBL24142117	(2S)-2-[[4-[(2,4-diaminopteridin-6-yl)methyl-[6-[3-[2-[2-[2-[3-[[1-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-3-oxopropoxy]ethoxy]ethoxy]ethoxy]propanoylamino]hexyl]amino]benzoyl]amino]pentanedioic acid	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)C(NC(=O)CCOCCOCCOCCOCCC(=O)NCCCCCCN(Cc2cnc3nc(N)nc(N)c3n2)c2ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)cc2)C(C)(C)C)cc1	C59H81N13O14S	DHFR	P00374	VHL	WO-2021262693-A1
TPD-683GYG	SCHEMBL24142009	(4S)-4-[[4-[(2,4-diaminopteridin-6-yl)methyl-methylamino]benzoyl]amino]-5-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethylamino]-5-oxopentanoic acid	CN(Cc1cnc2nc(N)nc(N)c2n1)c1ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)NCCOCCOCCNc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)cc1	C39H44N12O10	DHFR	P00374	CRBN	WO-2021262693-A1
TPD-L34ZCR	SCHEMBL26966101	(4S)-4-[[4-[(2,4-diaminopteridin-6-yl)methyl-methylamino]benzoyl]amino]-5-[3-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]propylamino]-5-oxopentanoic acid	CN(Cc1cnc2nc(N)nc(N)c2n1)c1ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)NCCCNc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)cc1	C36H38N12O8	DHFR	P00374	CRBN	WO-2021262693-A1
TPD-O8HUYZ	SCHEMBL26966106	(2S)-2-[[4-[(2,4-diaminopteridin-6-yl)methyl-[6-[3-[2-[3-[[1-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-3-oxopropoxy]ethoxy]propanoylamino]hexyl]amino]benzoyl]amino]pentanedioic acid	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)C(NC(=O)CCOCCOCCC(=O)NCCCCCCN(Cc2cnc3nc(N)nc(N)c3n2)c2ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)cc2)C(C)(C)C)cc1	C55H73N13O12S	DHFR	P00374	CRBN	WO-2021262693-A1
TPD-BAIIQC	SCHEMBL24142093	(2S)-2-[[4-[(2,4-diaminopteridin-6-yl)methyl-methylamino]benzoyl]amino]-5-[8-[[2-(1-methyl-2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]octylamino]-5-oxopentanoic acid	CN1C(=O)CCC(N2C(=O)c3cccc(NCCCCCCCCNC(=O)CC[C@H](NC(=O)c4ccc(N(C)Cc5cnc6nc(N)nc(N)c6n5)cc4)C(=O)O)c3C2=O)C1=O	C42H50N12O8	DHFR	P00374	CRBN	WO-2021262693-A1
TPD-T9RQLN	SCHEMBL24141947	(2S)-2-[[4-[(2,4-diaminopteridin-6-yl)methyl-methylamino]benzoyl]amino]-5-[2-[2-[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]prop-2-ynoxy]ethoxy]ethylamino]-5-oxopentanoic acid	CN(Cc1cnc2nc(N)nc(N)c2n1)c1ccc(C(=O)N[C@@H](CCC(=O)NCCOCCOCC#Cc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)C(=O)O)cc1	C40H41N11O10	DHFR	P00374	CRBN	WO-2021262693-A1
TPD-FB3Z8S	WO2021262693A1_NCGC00842343	.	C/C(N)=N\C(N)=C1\N=C(CN(C)c2ccc(C(=O)N[C@@H](CCC(=O)NCCOCCOCCOCC#Cc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)C(=O)O)cc2)C=NC1=N	C43H49N11O11	DHFR	P00374	CRBN	WO-2021262693-A1
TPD-K8984V	WO2021262693A1_NCGC00842344	.	CC(Cc1cnc2nc(N)nc(N)c2n1)c1ccc(C(=O)N[C@@H](CCC(=O)NCCCCCCCCNc2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)C(=O)O)cc1	C42H49N11O8	DHFR	P00374	CRBN	WO-2021262693-A1
TPD-ZA304K	SCHEMBL24141994	(2S)-2-[[4-[(2,4-diaminopteridin-6-yl)methyl-methylamino]benzoyl]amino]-5-[2-[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]prop-2-ynoxy]ethylamino]-5-oxopentanoic acid; SCHEMBL30638307	CN(Cc1cnc2nc(N)nc(N)c2n1)c1ccc(C(=O)N[C@@H](CCC(=O)NCCOCC#Cc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)C(=O)O)cc1	C38H37N11O9	DHFR	P00374	CRBN	WO-2021262693-A1
TPD-92GWMF	WO2021262693A1_NCGC00842349	.	CN(Cc1cnc2nc(N)nc(N)c2n1)c1ccc(C(=O)N[C@@H](CCC(=O)NCCOCCOCCOCCNC(=O)COc2ccc(C=O)c(C(=O)N(C)C3CCC(=O)NC3=O)c2)C(=O)O)cc1	C44H54N12O13	DHFR	P00374	CRBN	WO-2021262693-A1
TPD-840W69	SCHEMBL24142113	(2S)-2-[[4-[(2,4-diaminopteridin-6-yl)methyl-methylamino]benzoyl]amino]-5-[4-[1-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyacetyl]piperidin-4-yl]piperidin-1-yl]-5-oxopentanoic acid	CN(Cc1cnc2nc(N)nc(N)c2n1)c1ccc(C(=O)N[C@@H](CCC(=O)N2CCC(C3CCN(C(=O)COc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)C(=O)O)cc1	C45H50N12O10	DHFR	P00374	CRBN	WO-2021262693-A1
TPD-OR5CCZ	SCHEMBL24141995	(2S)-2-[[4-[(2,4-diaminopteridin-6-yl)methyl-methylamino]benzoyl]amino]-5-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperidin-1-yl]-5-oxopentanoic acid	CN(Cc1cnc2nc(N)nc(N)c2n1)c1ccc(C(=O)N[C@@H](CCC(=O)N2CCC(C3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)C(=O)O)cc1	C43H48N12O8	DHFR	P00374	CRBN	WO-2021262693-A1
TPD-935WJU	SCHEMBL24142308	(2S)-2-[[4-[(2,4-diaminopteridin-6-yl)methyl-methylamino]benzoyl]amino]-5-[2-[2-[2-[2-[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]prop-2-ynoxy]ethoxy]ethoxy]ethoxy]ethylamino]-5-oxopentanoic acid	CN(Cc1cnc2nc(N)nc(N)c2n1)c1ccc(C(=O)N[C@@H](CCC(=O)NCCOCCOCCOCCOCC#Cc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)C(=O)O)cc1	C44H49N11O12	DHFR	P00374	CRBN	WO-2021262693-A1
TPD-842Q9V	WO2021262693A1_NCGC00842358	.	C=C1c2c(OCC(=O)NCCOCCOCCOCCNC(=O)CC[C@H](NC(=O)c3ccc(N(C)Cc4cnc5nc(N)nc(N)c5n4)cc3)C(=O)O)cccc2C(=O)N1C1CCC(=O)N(C)C1=O	C45H54N12O12	DHFR	P00374	CRBN	WO-2021262693-A1
TPD-CPRT7E	SCHEMBL24142056	methyl (2S)-2-[[4-[(2,4-diaminopteridin-6-yl)methyl-methylamino]benzoyl]amino]-5-[2-[2-[2-[2-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyacetyl]amino]ethoxy]ethoxy]ethoxy]ethylamino]-5-oxopentanoate; SCHEMBL30638300	COC(=O)[C@H](CCC(=O)NCCOCCOCCOCCNC(=O)COc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O)NC(=O)c1ccc(N(C)Cc2cnc3nc(N)nc(N)c3n2)cc1	C44H52N12O13	DHFR	P00374	CRBN	WO-2021262693-A1
TPD-D378SP	SCHEMBL24141993	(2S)-2-[[4-[(2,4-diaminopteridin-6-yl)methyl-methylamino]benzoyl]amino]-5-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethylamino]-5-oxopentanoic acid	CN(Cc1cnc2nc(N)nc(N)c2n1)c1ccc(C(=O)N[C@@H](CCC(=O)NCCOCCOCCOCCNc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)C(=O)O)cc1	C41H48N12O11	DHFR	P00374	CRBN	WO-2021262693-A1
TPD-UEGHZ3	SCHEMBL24142127	(2S)-2-[[4-[(2,4-diaminopteridin-6-yl)methyl-methylamino]benzoyl]amino]-5-[3-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]propylamino]-5-oxopentanoic acid	CN(Cc1cnc2nc(N)nc(N)c2n1)c1ccc(C(=O)N[C@@H](CCC(=O)NCCCNc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)C(=O)O)cc1	C36H38N12O8	DHFR	P00374	CRBN	WO-2021262693-A1
TPD-ML6OWE	SCHEMBL24185858	2-[4-[1-[(3aS,6aR)-2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-3,3a,4,5,6,6a-hexahydro-1H-cyclopenta[c]pyrrol-5-yl]piperidin-4-yl]pyrazol-1-yl]-N-[4-cyano-3-(trifluoromethyl)phenyl]-2-methylpropanamide; SCHEMBL30634958	CC(C)(C(=O)Nc1ccc(C#N)c(C(F)(F)F)c1)n1cc(C2CCN(C3C[C@@H]4CN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C[C@@H]4C3)CC2)cn1	C40H41F3N8O5	AR	P10275	CRBN	WO-2022007903-A1
TPD-2LG5SX	SCHEMBL24185094	N-[4-cyano-3-(trifluoromethyl)phenyl]-2-[4-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]pyrrolidin-3-yl]methyl]piperidin-4-yl]pyrazol-1-yl]-2-methylpropanamide	CC(C)(C(=O)Nc1ccc(C#N)c(C(F)(F)F)c1)n1cc(C2CCN(CC3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)CC2)cn1	C38H39F3N8O5	AR	P10275	CRBN	WO-2022007903-A1
TPD-Z8RFTC	SCHEMBL24185118	N-[4-cyano-3-(trifluoromethyl)phenyl]-2-[4-[1-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-2-azaspiro[3.5]nonan-7-yl]piperidin-4-yl]pyrazol-1-yl]-2-methylpropanamide; SCHEMBL30173710	CC(C)(C(=O)Nc1ccc(C#N)c(C(F)(F)F)c1)n1cc(C2CCN(C3CCC4(CC3)CN(c3ccc5c(c3)C(=O)N(C3CCC(=O)NC3=O)C5=O)C4)CC2)cn1	C41H43F3N8O5	AR	P10275	CRBN	WO-2022007903-A1
TPD-GQ2RRS	SCHEMBL25208448	N-[4-cyano-3-(trifluoromethyl)phenyl]-1-[4-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]pyrrolidin-3-yl]methyl]piperidin-4-yl]pyrazol-1-yl]cyclobutane-1-carboxamide	N#Cc1ccc(NC(=O)C2(n3cc(C4CCN(CC5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cn3)CCC2)cc1C(F)(F)F	C39H39F3N8O5	AR	P10275	CRBN	WO-2022007903-A1
TPD-HIYMT5	SCHEMBL24185154	N-[4-cyano-3-(trifluoromethyl)phenyl]-2-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]pyrazol-1-yl]-2-methylpropanamide	CC(C)(C(=O)Nc1ccc(C#N)c(C(F)(F)F)c1)n1cc(C2CCN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)cn1	C33H30F3N7O5	AR	P10275	CRBN	WO-2022007903-A1
TPD-B3QMH2	SCHEMBL25200182	N-[4-cyano-3-(trifluoromethyl)phenyl]-1-[4-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]cyclobutane-1-carboxamide	N#Cc1ccc(NC(=O)C2(n3cc(C#CC4CN(C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)C4)cn3)CCC2)cc1C(F)(F)F	C37H31F3N8O5	AR	P10275	CRBN	WO-2022007903-A1
TPD-L0PC5I	SCHEMBL24185150	N-[4-cyano-3-(trifluoromethyl)phenyl]-1-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]cyclobutane-1-carboxamide	N#Cc1ccc(NC(=O)C2(n3cc(C#CC4CN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)cn3)CCC2)cc1C(F)(F)F	C34H26F3N7O5	AR	P10275	CRBN	WO-2022007903-A1
TPD-PEWHFN	SCHEMBL24185053	N-[4-cyano-3-(trifluoromethyl)phenyl]-2-[4-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide	CC(C)(C(=O)Nc1ccc(C#N)c(C(F)(F)F)c1)n1cc(C#CC2CN(C3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)C2)cn1	C36H31F3N8O5	AR	P10275	CRBN	WO-2022007903-A1
TPD-UGQYOC	SCHEMBL24185186	N-[4-cyano-3-(trifluoromethyl)phenyl]-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide; SCHEMBL30137234	CC(C)(C(=O)Nc1ccc(C#N)c(C(F)(F)F)c1)n1cc(C#CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)cn1	C33H26F3N7O5	AR	P10275	CRBN	WO-2022007903-A1
TPD-VNF1WU	SCHEMBL24185225	N-[4-cyano-3-(trifluoromethyl)phenyl]-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]ethynyl]pyrazol-1-yl]-2-methylpropanamide	CC(C)(C(=O)Nc1ccc(C#N)c(C(F)(F)F)c1)n1cc(C#CC2CCN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)cn1	C35H30F3N7O5	AR	P10275	CRBN	WO-2022007903-A1
TPD-F7MKXX	WO2022011204A1_1	.	N#CC1=CC=C(OC2CC3CC(C2)N3C(=O)C2=CC=C(N3CCC(CN4CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)C=C2)C=C1Cl	C43H44ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-8FQZOO	SCHEMBL24186794	2-Chloro-4-[[8-[6-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]pyridine-3-carbonyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzonitrile	N#CC1=CC=C(OC2CC3CCC(C2)N3C(=O)C2=CN=C(N3CCN(CC4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)C=C2)C=C1Cl	C43H45ClN8O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-CNX1KK	SCHEMBL24186795	2-Chloro-4-[[8-[6-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperidin-4-yl]methyl]piperazin-1-yl]pyridine-3-carbonyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzonitrile	N#CC1=CC=C(OC2CC3CCC(C2)N3C(=O)C2=CC=C(N3CCN(CC4CCN(C5=CC=CC6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)N=C2)C=C1Cl	C43H45ClN8O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-D5CRKI	SCHEMBL24186791	2-Chloro-4-[[8-[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]methyl]piperazin-1-yl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzonitrile	N#CC1=CC=C(OC2CC3CCC(C2)N3C(=O)C2=CC=C(N3CCN(CC4CN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=C2)C=C1Cl	C42H42ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-CM433C	SCHEMBL24186991	2-Chloro-4-[[8-[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]azetidin-3-yl]methyl]piperazin-1-yl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzonitrile	N#CC1=CC=C(OC2CC3CCC(C2)N3C(=O)C2=CC=C(N3CCN(CC4CN(C5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)C4)CC3)C=C2)C=C1Cl	C42H42ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-FVBGS6	SCHEMBL24186989	4-[[8-[4-[4-[[1-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]-2-(trifluoromethyl)benzonitrile	N#CC1=CC=C(OC2CC3CCC(C2)N3C(=O)C2=CC=C(N3CCN(CC4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)C=C2)C=C1C(F)(F)F	C45H46F3N7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-H59MXO	SCHEMBL24186994	5-[[8-[4-[4-[[1-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]-3-(trifluoromethyl)pyridine-2-carbonitrile	N#CC1=NC=C(OC2CC3CCC(C2)N3C(=O)C2=CC=C(N3CCN(CC4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)C=C2)C=C1C(F)(F)F	C44H45F3N8O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-OVCQMY	SCHEMBL24186993	2-Chloro-4-[[8-[4-[4-[7-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-7-azaspiro[3.5]nonan-2-yl]piperazin-1-yl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzonitrile	N#CC1=CC=C(OC2CC3CCC(C2)N3C(=O)C2=CC=C(N3CCN(C4CC5(CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)C4)CC3)C=C2)C=C1Cl	C46H48ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-Y286NQ	SCHEMBL24186990	2-Chloro-4-[[8-[4-[4-[7-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]-7-azaspiro[3.5]nonan-2-yl]piperazin-1-yl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzonitrile	N#CC1=CC=C(OC2CC3CCC(C2)N3C(=O)C2=CC=C(N3CCN(C4CC5(CCN(C6=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)CC5)C4)CC3)C=C2)C=C1Cl	C46H48ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-ROPLSM	SCHEMBL24186992	2-Chloro-4-[[8-[4-[7-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]-2,7-diazaspiro[3.5]nonan-2-yl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzonitrile	N#CC1=CC=C(OC2CC3CCC(C2)N3C(=O)C2=CC=C(N3CC4(CCN(C5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C3)C=C2)C=C1Cl	C46H48ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-F070EJ	SCHEMBL24186931	2-Chloro-4-[[8-[4-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperazine-1-carbonyl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzonitrile	N#CC1=CC=C(OC2CC3CCC(C2)N3C(=O)C2=CC=C(C(=O)N3CCN(C4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)C=C2)C=C1Cl	C44H44ClN7O7	AR	P10275	CRBN	WO-2022011204-A1
TPD-9TJW35	SCHEMBL24186933	2-Chloro-4-[[8-[4-[7-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]-2,7-diazaspiro[3.5]nonan-2-yl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzonitrile	N#CC1=CC=C(OC2CC3CCC(C2)N3C(=O)C2=CC=C(N3CC4(CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C3)C=C2)C=C1Cl	C47H50ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-AH334W	SCHEMBL24186932	2-Chloro-4-[[8-[4-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperidin-4-yl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzonitrile	N#CC1=CC=C(OC2CC3CCC(C2)N3C(=O)C2=CC=C(C3CCN(CC4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)C=C2)C=C1Cl	C45H47ClN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-NKZL4M	WO2022011204A1_17	.	[2H]C1(OC2=CC=C(C#N)C(Cl)=C2)CC2CCC(C1)N2C(=O)C1=CC=C(OC2CCN(CC3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)C=C1	C45H47ClN6O7	AR	P10275	CRBN	WO-2022011204-A1
TPD-XWV3XR	WO2022011204A1_18	.	N#CC1=CC=C(OC2CC3CCC(C2)N3C(=O)C2=CCC(OC3CCN(C4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)C=C2)C=C1Cl	C44H47ClN6O7	AR	P10275	CRBN	WO-2022011204-A1
TPD-NQV7JR	SCHEMBL24186934	2-Chloro-4-[[8-[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]benzoyl]-3-methyl-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzonitrile	CC1(OC2=CC=C(C#N)C(Cl)=C2)CC2CCC(C1)N2C(=O)C1=CC=C(N2CCN(CC3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)C=C1	C45H48ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-MPDS6P	SCHEMBL24186926	2-Chloro-4-[[8-[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]-3-fluorobenzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzonitrile	N#CC1=CC=C(OC2CC3CCC(C2)N3C(=O)C2=CC=C(N3CCN(CC4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)C(F)=C2)C=C1Cl	C44H45ClFN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-NFK2HR	WO2022011204A1_21	.	N#CC1=CC=C(OC2CC3CCC(C2)N3C(=O)C2=CC=C(N3CC4(C3)CN(C3CCC(N5CC6=C(C5)C5=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C5=O)CC3)C4)C=C2)C=C1Cl	C47H48ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-YMRMU4	WO2022011204A1_23	2-Chloro-4-[[8-[4-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-2-azaspiro[3.3]heptane-6-carbonyl]piperazin-1-yl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzonitrile	N#CC1=CC=C(OC2CC3CCC(C2)N3C(=O)C2=CC=C(N3CCN(C(=O)C4CC5(C4)CN(C4=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C4)C5)CC3)C=C2)C=C1Cl	C45H44ClN7O7	AR	P10275	CRBN	WO-2022011204-A1
TPD-62ZUS5	WO2022011204A1_24	2-Chloro-4-[[8-[4-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-2-azaspiro[3.3]heptan-6-yl]methyl]piperazin-1-yl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzonitrile	N#CC1=CC=C(OC2CC3CCC(C2)N3C(=O)C2=CC=C(N3CCN(CC4CC5(C4)CN(C4=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C4)C5)CC3)C=C2)C=C1Cl	C45H46ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-80AWPB	SCHEMBL26211772	2-Chloro-4-[[8-[4-[6-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]-2,6-diazaspiro[3.3]heptan-2-yl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzonitrile	N#CC1=CC=C(OC2CC3CCC(C2)N3C(=O)C2=CC=C(N3CC4(CN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)C4)C3)C=C2)C=C1Cl	C45H46ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-LCY30T	SCHEMBL24186781	6-[[8-[4-[4-[[1-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]-4-(trifluoromethyl)pyridine-3-carbonitrile	N#CC1=CN=C(OC2CC3CCC(C2)N3C(=O)C2=CC=C(N3CCN(CC4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)C=C2)C=C1C(F)(F)F	C44H45F3N8O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-KB1LZH	WO2022011204A1_27	.	[2H]C1(OC2=CC=C(C#N)C(Cl)=C2C)CC2CCC(C1)N2C(=O)C1=CC=C(C2CCN(CC3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)C=C1	C46H49ClN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-K26XAK	SCHEMBL25385633	2-Chloro-4-[1-[4-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperazin-1-yl]benzoyl]piperidin-4-yl]oxybenzonitrile	N#CC1=C(Cl)C=C(OC2CCN(C(=O)C3=CC=C(N4CCN(C5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C=C3)CC2)C=C1	C41H42ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-1N8XOW	SCHEMBL24186782	2-Chloro-4-[[8-[4-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperazin-1-yl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzonitrile	N#CC1=CC=C(OC2CC3CCC(C2)N3C(=O)C2=CC=C(N3CCN(C4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)C=C2)C=C1Cl	C43H44ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-4EJSY6	SCHEMBL24187131	2-Chloro-4-[[8-[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]-3-methylbenzonitrile	CC1=C(Cl)C(C#N)=CC=C1OC1CC2CCC(C1)N2C(=O)C1=CC=C(N2CCN(CC3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)C=C1	C45H48ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-TXVF0K	SCHEMBL24187130	2-Chloro-4-[1-[[4-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperidin-4-yl]ethynyl]-3-fluorophenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile	CC1=C(C)N(CC2=CC=C(C#CC3CCN(C4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)C(F)=C2)N=C1C1=CC(Cl)=C(C#N)C=C1	C44H41ClFN7O4	AR	P10275	CRBN	WO-2022011204-A1
TPD-ROQUZ3	SCHEMBL25386888	2-Chloro-4-[1-[[4-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperidin-4-yl]ethynyl]-2-fluorophenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile	CC1=C(C)N(CC2=CC=C(C#CC3CCN(C4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)C=C2F)N=C1C1=CC(Cl)=C(C#N)C=C1	C44H41ClFN7O4	AR	P10275	CRBN	WO-2022011204-A1
TPD-R625TN	SCHEMBL25385432	2-chloro-4-[1-[[4-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperidin-4-yl]ethynyl]phenyl]methyl]-5,6-dihydro-4H-cyclopenta[c]pyrazol-3-yl]benzonitrile	N#CC1=C(Cl)C=C(C2=NN(CC3=CC=C(C#CC4CCN(C5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C=C3)C3=C2CCC3)C=C1	C45H42ClN7O4	AR	P10275	CRBN	WO-2022011204-A1
TPD-DGQSTR	SCHEMBL24187137	2-Chloro-4-[1-[[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazine-1-carbonyl]phenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile	CC1=C(C)N(CC2=CC=C(C(=O)N3CCN(CC4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)C=C2)N=C1C1=CC(Cl)=C(C#N)C=C1	C43H43ClN8O5	AR	P10275	CRBN	WO-2022011204-A1
TPD-OYWGPM	SCHEMBL24186820	2-Chloro-4-[1-[[4-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperazine-1-carbonyl]phenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile	CC1=C(C)N(CC2=CC=C(C(=O)N3CCN(C4CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)C=C2)N=C1C1=CC(Cl)=C(C#N)C=C1	C42H41ClN8O5	AR	P10275	CRBN	WO-2022011204-A1
TPD-UVGFM2	SCHEMBL22565546	2-chloro-4-[3-[6-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperidin-4-yl]ethynyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile; SCHEMBL28484224	CC1(C)[C@H](OC2=CC(Cl)=C(C#N)C=C2)C(C)(C)[C@H]1N1CC2=CC(C#CC3CCN(C4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)=CC=C2C1=O	C48H49ClN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-JVS0YM	WO2022011204A1_37	.	N#CC1=C(Cl)C=C(OC2CCC(N3CC4=CC(C#CC5CCN(C6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)CC5)=CC=C4C3=O)CC2)C=C1	C46H45ClN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-2FYBMH	SCHEMBL24187133	2-chloro-4-[3-[6-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile; SCHEMBL25385351	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@@H]1N1CC2=CC(N3CCN(C4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)=CC=C2C1=O	C45H48ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-JXZ5C0	SCHEMBL24186768	2-chloro-4-[3-[6-[4-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]azetidin-3-yl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile; SCHEMBL25385375	CC1(C)[C@H](OC2=CC(Cl)=C(C#N)C=C2)C(C)(C)[C@@H]1N1CC2=CC(N3CCN(C4CN(C5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)C4)CC3)=CC=C2C1=O	C48H53ClN8O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-E47LAJ	SCHEMBL25383774	2-chloro-4-[3-[5-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperidin-4-yl]ethynyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC(Cl)=C(C#N)C=C2)C(C)(C)[C@@H]1N1CC2=CC=C(C#CC3CCN(C4CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)C=C2C1=O	C48H49ClN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-L67O7W	SCHEMBL25388119	2-chloro-4-[3-[6-[2-[1-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-2-azaspiro[3.3]heptan-6-yl]piperidin-4-yl]ethynyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile; SCHEMBL25388129	CC1(C)[C@H](OC2=CC(Cl)=C(C#N)C=C2)C(C)(C)[C@H]1N1CC2=CC(C#CC3CCN(C4CC5(C4)CN(C4=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C4)C5)CC3)=CC=C2C1=O	C49H49ClN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-07SPWM	SCHEMBL25383813	2-chloro-4-[3-[6-[2-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]cyclohexyl]ethynyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile; SCHEMBL25383818	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@@H]1N1CC2=CC(C#CC3CCC(N4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)=CC=C2C1=O	C48H49ClN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-TLZCC7	SCHEMBL25386155	2-Chloro-4-[1-[[4-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperidin-4-yl]ethynyl]phenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile	CC1=C(C)N(CC2=CC=C(C#CC3CCN(C4CCN(C5=C(F)C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)C=C2)N=C1C1=CC(Cl)=C(C#N)C=C1	C44H41ClFN7O4	AR	P10275	CRBN	WO-2022011204-A1
TPD-ZHW0IM	SCHEMBL25386438	2-Chloro-4-[1-[[4-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperidin-4-yl]ethynyl]phenyl]methyl]-4,5,6,7-tetrahydroindazol-3-yl]benzonitrile	N#CC1=C(Cl)C=C(C2=NN(CC3=CC=C(C#CC4CCN(C5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C=C3)C3=C2CCCC3)C=C1	C46H44ClN7O4	AR	P10275	CRBN	WO-2022011204-A1
TPD-DYXCPP	SCHEMBL24186771	2-Chloro-4-[1-[[4-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperidin-4-yl]ethynyl]phenyl]methyl]-4-ethyl-5-methylpyrazol-3-yl]benzonitrile	CCC1=C(C)N(CC2=CC=C(C#CC3CCN(C4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)C=C2)N=C1C1=CC(Cl)=C(C#N)C=C1	C45H44ClN7O4	AR	P10275	CRBN	WO-2022011204-A1
TPD-31VQWN	SCHEMBL25386440	4-[1-[[4-[2-[1-[1-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperidin-4-yl]ethynyl]phenyl]methyl]-4,5-dimethylpyrazol-3-yl]-2-(trifluoromethyl)benzonitrile	CC1=C(C)N(CC2=CC=C(C#CC3CCN(C4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)C=C2)N=C1C1=CC(C(F)(F)F)=C(C#N)C=C1	C45H42F3N7O4	AR	P10275	CRBN	WO-2022011204-A1
TPD-A2U4MB	SCHEMBL24186772	2-chloro-4-[1-[[4-[2-[4-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-3-oxo-1H-isoindol-5-yl]ethynyl]piperidine-1-carbonyl]cyclohexyl]ethynyl]phenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile; SCHEMBL25385393	CC1=C(C)N(CC2=CC=C(C#CC3CCC(C(=O)N4CCC(C#CC5=CC=C6CN(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)C=C2)N=C1C1=CC(Cl)=C(C#N)C=C1	C48H45ClN6O4	AR	P10275	CRBN	WO-2022011204-A1
TPD-7LN9NN	SCHEMBL25386210	2-chloro-4-[3-[5-[2-[1-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-2-azaspiro[3.3]heptan-6-yl]piperidin-4-yl]ethynyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile; SCHEMBL25386217	CC1(C)[C@H](OC2=CC(Cl)=C(C#N)C=C2)C(C)(C)[C@H]1N1CC2=CC=C(C#CC3CCN(C4CC5(C4)CN(C4=CC6=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)C5)CC3)C=C2C1=O	C49H49ClN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-16QJUH	SCHEMBL24186809	2-chloro-4-[3-[6-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-2-azaspiro[3.3]heptan-6-yl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile; SCHEMBL25386750	CC1(C)[C@H](OC2=CC(Cl)=C(C#N)C=C2)C(C)(C)[C@@H]1N1CC2=CC(N3CCN(C4CC5(C4)CN(C4=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C4)C5)CC3)=CC=C2C1=O	C46H48ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-PJOHXF	SCHEMBL24186819	2-chloro-4-[4-[5-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperidin-4-yl]ethynyl]-3-oxo-1H-isoindol-2-yl]cyclohexyl]oxybenzonitrile	N#CC1=C(Cl)C=C(OC2CCC(N3CC4=CC=C(C#CC5CCN(C6CCN(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)C=C4C3=O)CC2)C=C1	C46H45ClN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-GX2YEG	SCHEMBL25385372	2-chloro-4-[4-[5-[2-[1-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-2-azaspiro[3.3]heptan-6-yl]piperidin-4-yl]ethynyl]-3-oxo-1H-isoindol-2-yl]cyclohexyl]oxybenzonitrile; SCHEMBL25385381	N#CC1=CC=C(OC2CCC(N3CC4=CC=C(C#CC5CCN(C6CC7(C6)CN(C6=CC8=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C8=O)C7)CC5)C=C4C3=O)CC2)C=C1Cl	C47H45ClN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-JKKKVL	SCHEMBL25386724	2-Chloro-4-[1-[[4-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-2-azaspiro[3.3]heptan-6-yl]piperazine-1-carbonyl]phenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile	CC1=C(C)N(CC2=CC=C(C(=O)N3CCN(C4CC5(C4)CN(C4=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C4)C5)CC3)C=C2)N=C1C1=CC(Cl)=C(C#N)C=C1	C43H41ClN8O5	AR	P10275	CRBN	WO-2022011204-A1
TPD-Y49SGT	WO2022011204A1_54	.	N#CC1=CC=C(OC2CC3CC(C2)N3C2=CC=C(C(=O)N3CCN(CC4CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)C=C2)C=C1Cl	C43H44ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-NGXX26	WO2022011204A1_55	.	N#CC1=CC=C(OC2CC3CCC(C2)N3C2=CC=C(C(=O)N3CCN(C4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)C=C2)C=C1Cl	C43H44ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-LUXO0O	SCHEMBL25383928	2-Chloro-4-[1-[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazine-1-carbonyl]phenyl]piperidin-4-yl]oxybenzonitrile	N#CC1=CC=C(OC2CCN(C3=CC=C(C(=O)N4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C=C3)CC2)C=C1Cl	C42H44ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-35DUVL	SCHEMBL25385119	2-Chloro-4-[1-[4-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperazine-1-carbonyl]phenyl]piperidin-4-yl]oxybenzonitrile	N#CC1=CC=C(OC2CCN(C3=CC=C(C(=O)N4CCN(C5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C=C3)CC2)C=C1Cl	C41H42ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-EA9915	SCHEMBL24186922	2-chloro-4-[4-[6-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperazine-1-carbonyl]-3-oxo-1H-isoindol-2-yl]cyclohexyl]oxybenzonitrile	N#CC1=CC=C(O[C@H]2CC[C@@H](N3CC4=C(C=CC(C(=O)N5CCN(C6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)CC5)=C4)C3=O)CC2)C=C1Cl	C44H44ClN7O7	AR	P10275	CRBN	WO-2022011204-A1
TPD-XES8LN	SCHEMBL24186923	2-chloro-4-[4-[6-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazine-1-carbonyl]-3-oxo-1H-isoindol-2-yl]cyclohexyl]oxybenzonitrile	N#CC1=CC=C(OC2CCC(N3CC4=C(C=CC(C(=O)N5CCN(CC6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)CC5)=C4)C3=O)CC2)C=C1Cl	C45H46ClN7O7	AR	P10275	CRBN	WO-2022011204-A1
TPD-3FDLXK	SCHEMBL26212141	2-chloro-4-[4-[6-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-2-azaspiro[3.3]heptan-6-yl]piperazine-1-carbonyl]-3-oxo-1H-isoindol-2-yl]cyclohexyl]oxybenzonitrile	N#CC1=CC=C(O[C@H]2CC[C@H](N3CC4=C(C=CC(C(=O)N5CCN(C6CC7(C6)CN(C6=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C6)C7)CC5)=C4)C3=O)CC2)C=C1Cl	C45H44ClN7O7	AR	P10275	CRBN	WO-2022011204-A1
TPD-3OHMNK	SCHEMBL24186946	2-chloro-4-[4-[6-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]methyl]piperazine-1-carbonyl]-3-oxo-1H-isoindol-2-yl]cyclohexyl]oxybenzonitrile	N#CC1=CC=C(O[C@H]2CC[C@H](N3CC4=C(C=CC(C(=O)N5CCN(CC6CN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)C6)CC5)=C4)C3=O)CC2)C=C1Cl	C43H42ClN7O7	AR	P10275	CRBN	WO-2022011204-A1
TPD-L4MVGG	WO2022011204A1_62	.	CC1(C)CN(C(=O)C2=CC=C(N3CCN(C4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)C=C2)CC[C@H]1OC1=CC(Cl)=C(C#N)C=C1	C43H46ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-42ESG4	SCHEMBL24186937	2-chloro-4-[1-[4-[4-[3-[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]ethynyl]azetidin-1-yl]piperidin-1-yl]benzoyl]piperidin-4-yl]oxybenzonitrile	N#CC1=CC=C(OC2CCN(C(=O)C3=CC=C(N4CCC(N5CC(C#CC6=C7CN(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)C5)CC4)C=C3)CC2)C=C1Cl	C42H41ClN6O5	AR	P10275	CRBN	WO-2022011204-A1
TPD-D08IIJ	SCHEMBL24186929	2-chloro-4-[1-[4-[4-[3-[2-[2-(2,6-dioxopiperidin-3-yl)-3-oxo-1H-isoindol-5-yl]ethynyl]azetidin-1-yl]piperidin-1-yl]benzoyl]piperidin-4-yl]oxybenzonitrile	N#CC1=CC=C(OC2CCN(C(=O)C3=CC=C(N4CCC(N5CC(C#CC6=CC=C7CN(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C3)CC2)C=C1Cl	C42H41ClN6O5	AR	P10275	CRBN	WO-2022011204-A1
TPD-SYVNMU	SCHEMBL26212188	2-chloro-4-[1-[4-[4-[3-[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]ethynyl]azetidin-1-yl]piperidin-1-yl]benzoyl]piperidin-4-yl]oxybenzonitrile	N#CC1=CC=C(OC2CCN(C(=O)C3=CC=C(N4CCC(N5CC(C#CC6=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)C5)CC4)C=C3)CC2)C=C1Cl	C42H41ClN6O5	AR	P10275	CRBN	WO-2022011204-A1
TPD-RROGMK	SCHEMBL24187139	2-chloro-4-[1-[4-[4-[[3-[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]ethynyl]azetidin-1-yl]methyl]piperidin-1-yl]benzoyl]piperidin-4-yl]oxybenzonitrile	N#CC1=CC=C(OC2CCN(C(=O)C3=CC=C(N4CCC(CN5CC(C#CC6=C7CN(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)C5)CC4)C=C3)CC2)C=C1Cl	C43H43ClN6O5	AR	P10275	CRBN	WO-2022011204-A1
TPD-I9DKL8	SCHEMBL24187141	2-chloro-4-[1-[4-[4-[[3-[2-[2-(2,6-dioxopiperidin-3-yl)-3-oxo-1H-isoindol-5-yl]ethynyl]azetidin-1-yl]methyl]piperidin-1-yl]benzoyl]piperidin-4-yl]oxybenzonitrile	N#CC1=CC=C(OC2CCN(C(=O)C3=CC=C(N4CCC(CN5CC(C#CC6=CC=C7CN(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C3)CC2)C=C1Cl	C43H43ClN6O5	AR	P10275	CRBN	WO-2022011204-A1
TPD-ITNT9D	SCHEMBL24187145	2-chloro-4-[1-[4-[4-[[3-[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]ethynyl]azetidin-1-yl]methyl]piperidin-1-yl]benzoyl]piperidin-4-yl]oxybenzonitrile	N#CC1=CC=C(OC2CCN(C(=O)C3=CC=C(N4CCC(CN5CC(C#CC6=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)C5)CC4)C=C3)CC2)C=C1Cl	C43H43ClN6O5	AR	P10275	CRBN	WO-2022011204-A1
TPD-Y5WJK8	SCHEMBL24187140	2-Chloro-4-[1-[4-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperidin-4-yl]benzoyl]piperidin-4-yl]oxy-3-methylbenzonitrile	CC1=C(OC2CCN(C(=O)C3=CC=C(C4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C=C3)CC2)C=CC(C#N)=C1Cl	C44H47ClN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-B02D15	SCHEMBL24187033	2-Chloro-4-[1-[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]benzoyl]piperidin-4-yl]oxy-3-methylbenzonitrile	CC1=C(OC2CCN(C(=O)C3=CC=C(N4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C=C3)CC2)C=CC(C#N)=C1Cl	C43H46ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-URGQ98	SCHEMBL26212235	2-Chloro-4-[1-[4-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperidin-4-yl]benzoyl]-3,3,5,5-tetramethylpiperidin-4-yl]oxybenzonitrile	CC1(C)CN(C(=O)C2=CC=C(C3CCN(CC4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)C=C2)CC(C)(C)C1OC1=CC=C(C#N)C(Cl)=C1	C47H53ClN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-W5HZ6L	SCHEMBL24187142	2-Chloro-4-[1-[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]benzoyl]-3,3,5,5-tetramethylpiperidin-4-yl]oxybenzonitrile	CC1(C)CN(C(=O)C2=CC=C(N3CCN(CC4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)C=C2)CC(C)(C)C1OC1=CC(Cl)=C(C#N)C=C1	C46H52ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-XK5WXE	SCHEMBL24187034	4-[[(3aR,6aS)-2-[4-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperidin-4-yl]benzoyl]-3,3a,4,5,6,6a-hexahydro-1H-cyclopenta[c]pyrrol-5-yl]oxy]-2-chlorobenzonitrile; SCHEMBL26209799	N#CC1=C(Cl)C=C(O[C@H]2C[C@@H]3CN(C(=O)C4=CC=C(C5CCN(CC6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)CC5)C=C4)C[C@@H]3C2)C=C1	C45H47ClN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-HQKKW7	SCHEMBL26209810	2-Chloro-4-[1-[4-[1-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-2-azaspiro[3.3]heptan-6-yl]methyl]piperidin-4-yl]benzoyl]piperidin-4-yl]oxybenzonitrile	N#CC1=C(Cl)C=C(OC2CCN(C(=O)C3=CC=C(C4CCN(CC5CC6(C5)CN(C5=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C5)C6)CC4)C=C3)CC2)C=C1	C44H45ClN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-MTUBIH	SCHEMBL26209812	2-Chloro-4-[1-[4-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-2-azaspiro[3.3]heptan-6-yl]methyl]piperazin-1-yl]benzoyl]piperidin-4-yl]oxybenzonitrile	N#CC1=C(Cl)C=C(OC2CCN(C(=O)C3=CC=C(N4CCN(CC5CC6(C5)CN(C5=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C5)C6)CC4)C=C3)CC2)C=C1	C43H44ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-H7VVGR	SCHEMBL24187036	N-[(3aR,6aS)-5-(3-chloro-4-cyanophenoxy)-1,2,3,3a,4,5,6,6a-octahydropentalen-2-yl]-4-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperidin-4-yl]benzamide	N#CC1=CC=C(O[C@@H]2C[C@H]3C[C@H](NC(=O)C4=CC=C(C5CCN(CC6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)CC5)C=C4)C[C@H]3C2)C=C1Cl	C46H49ClN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-A1D40N	SCHEMBL24187038	N-[(3aR,6aS)-5-(3-chloro-4-cyanophenoxy)-1,2,3,3a,4,5,6,6a-octahydropentalen-2-yl]-4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]benzamide	N#CC1=CC=C(O[C@H]2C[C@H]3C[C@@H](NC(=O)C4=CC=C(N5CCN(CC6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)CC5)C=C4)C[C@H]3C2)C=C1Cl	C45H48ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-73VTC0	SCHEMBL24187039	2-Chloro-4-[1-[4-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidine-4-carbonyl]piperazin-1-yl]benzoyl]piperidin-4-yl]oxybenzonitrile	N#CC1=C(Cl)C=C(OC2CCN(C(=O)C3=CC=C(N4CCN(C(=O)C5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C=C3)CC2)C=C1	C42H42ClN7O7	AR	P10275	CRBN	WO-2022011204-A1
TPD-557YNP	SCHEMBL24187047	2-Chloro-4-[1-[4-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidine-4-carbonyl]piperidin-4-yl]benzoyl]piperidin-4-yl]oxybenzonitrile	N#CC1=C(Cl)C=C(OC2CCN(C(=O)C3=CC=C(C4CCN(C(=O)C5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C=C3)CC2)C=C1	C43H43ClN6O7	AR	P10275	CRBN	WO-2022011204-A1
TPD-T1J9OG	SCHEMBL24186975	2-Chloro-4-[1-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]benzoyl]piperidin-4-yl]oxybenzonitrile	N#CC1=C(Cl)C=C(OC2CCN(C(=O)C3=CC=C(N4CCC(CN5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C=C3)CC2)C=C1	C42H44ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-24MJP6	SCHEMBL26209814	2-Chloro-4-[1-[4-[6-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]-2,6-diazaspiro[3.3]heptan-2-yl]benzoyl]piperidin-4-yl]oxy-3-methylbenzonitrile	CC1=C(OC2CCN(C(=O)C3=CC=C(N4CC5(CN(CC6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)C5)C4)C=C3)CC2)C=CC(C#N)=C1Cl	C44H46ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-WVQ3WO	SCHEMBL24187035	2-Chloro-4-[1-[4-[2-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-5-yl]benzoyl]piperidin-4-yl]oxy-3-methylbenzonitrile	CC1=C(OC2CCN(C(=O)C3=CC=C(N4CC5CN(CC6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)CC5C4)C=C3)CC2)C=CC(C#N)=C1Cl	C45H48ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-6FA8UV	SCHEMBL24187006	5-[4-[4-[4-[[1-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]phenoxy]piperidin-1-yl]-3-(trifluoromethyl)pyridine-2-carbonitrile	N#CC1=C(C(F)(F)F)C=C(N2CCC(OC3=CC=C(N4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C=C3)CC2)C=N1	C41H43F3N8O5	AR	P10275	CRBN	WO-2022011204-A1
TPD-RGZ34T	SCHEMBL24187007	[4-[4-[[1-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]phenyl] 4-(3-chloro-4-cyanophenoxy)piperidine-1-carboxylate	N#CC1=CC=C(OC2CCN(C(=O)OC3=CC=C(N4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C=C3)CC2)C=C1Cl	C42H44ClN7O7	AR	P10275	CRBN	WO-2022011204-A1
TPD-X85W0C	WO2022011204A1_86	[4-[4-[[1-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]phenyl] 2-(3-chloro-4-cyanophenoxy)-7-azabicyclo[2.2.1]heptane-7-carboxylate	N#CC1=CC=C(OC2CC3CCC2N3C(=O)OC2=CC=C(N3CCN(CC4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)C=C2)C=C1Cl	C43H44ClN7O7	AR	P10275	CRBN	WO-2022011204-A1
TPD-SO82IG	SCHEMBL24187005	[4-[4-[[1-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]phenyl] 4-(3-chloro-4-cyanophenyl)piperazine-1-carboxylate	N#CC1=CC=C(N2CCN(C(=O)OC3=CC=C(N4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C=C3)CC2)C=C1Cl	C41H43ClN8O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-RDJ3PF	SCHEMBL24186765	2-chloro-4-[4-[6-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]cyclohexyl]oxybenzonitrile; SCHEMBL25384869	N#CC1=CC=C(O[C@H]2CC[C@@H](N3CC4=C(C=CC(N5CCN(CC6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)CC5)=C4)C3=O)CC2)C=C1Cl	C44H46ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-D5D2S8	SCHEMBL24186874	2-chloro-4-[3-[6-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile; SCHEMBL25385621	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@@H]1N1CC2=C(C=CC(N3CCN(CC4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)=C2)C1=O	C46H50ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-5LM36G	SCHEMBL24187009	2-Chloro-4-[1-[[4-[2-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperidin-4-yl]ethynyl]phenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile	CC1=C(C)N(CC2=CC=C(C#CC3CCN(CC4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)C=C2)N=C1C1=CC(Cl)=C(C#N)C=C1	C45H44ClN7O4	AR	P10275	CRBN	WO-2022011204-A1
TPD-8RSS4T	WO2022011204A1_91	.	C=C1C(=O)N(C2CCC(=O)NC2=O)C(=O)/C1=C/C(=C)N(C)CCC(C)N(C)CCC(C)C#CC1=CC=C(CN2N=C(C3=CC(Cl)=C(C#N)C=C3)C(C)=C2C)C=C1	C44H48ClN7O4	AR	P10275	CRBN	WO-2022011204-A1
TPD-AY8EVA	SCHEMBL26209827	2-chloro-4-[3-[6-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-4-methoxypiperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	COC1(CN2CCN(C3=CC4=C(C=C3)C(=O)N([C@H]3C(C)(C)[C@@H](OC5=CC=C(C#N)C(Cl)=C5)C3(C)C)C4)CC2)CCN(C2=CC=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=C2)CC1	C47H52ClN7O7	AR	P10275	CRBN	WO-2022011204-A1
TPD-5FWPPW	SCHEMBL24186813	2-chloro-4-[4-[6-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-4-methoxypiperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]cyclohexyl]oxybenzonitrile	COC1(CN2CCN(C3=CC4=C(C=C3)C(=O)N([C@H]3CC[C@H](OC5=CC(Cl)=C(C#N)C=C5)CC3)C4)CC2)CCN(C2=CC=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=C2)CC1	C45H48ClN7O7	AR	P10275	CRBN	WO-2022011204-A1
TPD-4DWUDW	SCHEMBL24186815	2-chloro-4-[3-[6-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-4-fluoropiperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@@H]1N1CC2=C(C=CC(N3CCN(CC4(F)CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)=C2)C1=O	C46H49ClFN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-AMOFZC	SCHEMBL24186817	2-chloro-4-[4-[6-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-4-fluoropiperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]cyclohexyl]oxybenzonitrile	N#CC1=CC=C(O[C@H]2CC[C@@H](N3CC4=C(C=CC(N5CCN(CC6(F)CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)CC5)=C4)C3=O)CC2)C=C1Cl	C44H45ClFN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-5Z3LSH	SCHEMBL24186822	2-chloro-4-[4-[6-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]cyclohexyl]oxybenzonitrile	N#CC1=CC=C(O[C@H]2CC[C@@H](N3CC4=C(C=CC(N5CCN(CC6CN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)C6)CC5)=C4)C3=O)CC2)C=C1Cl	C42H42ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-VTUA02	SCHEMBL24186918	2-chloro-4-[3-[6-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@@H]1N1CC2=C(C=CC(N3CCN(CC4CN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)=C2)C1=O	C44H46ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-SVRWLW	SCHEMBL24186831	2-chloro-4-[3-[6-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@@H]1N1CC2=C(C=CC(N3CCN(CC4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)CC6=C5)CC4)CC3)=C2)C1=O	C46H52ClN7O5	AR	P10275	CRBN	WO-2022011204-A1
TPD-XAHJOI	SCHEMBL24186919	5-[4-[6-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]cyclohexyl]oxy-3-(trifluoromethyl)pyridine-2-carbonitrile	N#CC1=C(C(F)(F)F)C=C(O[C@H]2CC[C@@H](N3CC4=C(C=CC(N5CCN(CC6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)CC5)=C4)C3=O)CC2)C=N1	C44H45F3N8O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-1BN8YW	SCHEMBL26209832	5-[3-[6-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-4-fluoropiperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxy-3-(trifluoromethyl)pyridine-2-carbonitrile	CC1(C)[C@H](OC2=CC(C(F)(F)F)=C(C#N)N=C2)C(C)(C)[C@@H]1N1CC2=C(C=CC(N3CCN(CC4(F)CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)=C2)C1=O	C46H48F4N8O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-3N77SW	SCHEMBL24186917	5-[4-[6-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-4-fluoropiperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]cyclohexyl]oxy-3-(trifluoromethyl)pyridine-2-carbonitrile; SCHEMBL26209834	N#CC1=C(C(F)(F)F)C=C(O[C@H]2CC[C@H](N3CC4=C(C=CC(N5CCN(CC6(F)CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)CC5)=C4)C3=O)CC2)C=N1	C44H44F4N8O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-R9TITU	SCHEMBL24187080	2-chloro-4-[3-[6-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-4-hydroxypiperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@@H]1N1CC2=C(C=CC(N3CCN(CC4(O)CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)=C2)C1=O	C46H50ClN7O7	AR	P10275	CRBN	WO-2022011204-A1
TPD-CPQJGX	SCHEMBL24187083	2-chloro-4-[3-[6-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-4-methylpiperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(CN2CCN(C3=CC4=C(C=C3)C(=O)N([C@H]3C(C)(C)[C@@H](OC5=CC=C(C#N)C(Cl)=C5)C3(C)C)C4)CC2)CCN(C2=CC=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=C2)CC1	C47H52ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-HQDK1D	SCHEMBL24187075	5-[3-[6-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-4-methylpiperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxy-3-(trifluoromethyl)pyridine-2-carbonitrile	CC1(CN2CCN(C3=CC4=C(C=C3)C(=O)N([C@H]3C(C)(C)[C@@H](OC5=CC(C(F)(F)F)=C(C#N)N=C5)C3(C)C)C4)CC2)CCN(C2=CC=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=C2)CC1	C47H51F3N8O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-2B79AH	SCHEMBL24187094	5-[4-[6-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-4-methylpiperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]cyclohexyl]oxy-3-(trifluoromethyl)pyridine-2-carbonitrile	CC1(CN2CCN(C3=CC4=C(C=C3)C(=O)N([C@H]3CC[C@H](OC5=CC(C(F)(F)F)=C(C#N)N=C5)CC3)C4)CC2)CCN(C2=CC=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=C2)CC1	C45H47F3N8O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-NQWLUH	SCHEMBL24187074	2-chloro-4-[3-[6-[4-[[(3S)-1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]pyrrolidin-3-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC(Cl)=C(C#N)C=C2)C(C)(C)[C@H]1N1CC2=C(C=CC(N3CCN(C[C@@H]4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)=C2)C1=O	C45H48ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-5I8XPJ	SCHEMBL24186753	2-chloro-4-[3-[6-[4-[[(3R)-1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]pyrrolidin-3-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC(Cl)=C(C#N)C=C2)C(C)(C)[C@H]1N1CC2=C(C=CC(N3CCN(C[C@H]4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)=C2)C1=O	C45H48ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-2VWTRU	WO2022011204A1_108	.	N#CC1=CC=C(O[C@H]2CC[C@@H](N3CC4=C(C=CC(N5CCN(C[C@@H]6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)C6)CC5)=C4)C3=O)CC2)C=C1Cl	C43H44ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-58XF1S	WO2022011204A1_109	.	N#CC1=CC=C(O[C@H]2CC[C@@H](N3CC4=C(C=CC(N5CCN(C[C@H]6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)C6)CC5)=C4)C3=O)CC2)C=C1Cl	C43H44ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-CML1VP	SCHEMBL24186751	2-chloro-4-[3-[6-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]-4-fluoro-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC(Cl)=C(C#N)C=C2)C(C)(C)[C@@H]1N1CC2=C(C1=O)C(F)=CC(N1CCN(CC3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC1)=C2	C46H49ClFN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-4CJL6F	SCHEMBL24186752	2-chloro-4-[(1R,3R)-3-[6-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]cyclopentyl]oxybenzonitrile	N#CC1=CC=C(O[C@@H]2CC[C@@H](N3CC4=C(C=CC(N5CCN(CC6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)CC5)=C4)C3=O)C2)C=C1Cl	C43H44ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-YIDES9	SCHEMBL26209844	2-chloro-4-[4-[6-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]cyclohexyl]oxybenzonitrile	N#CC1=CC=C(O[C@H]2CC[C@@H](N3CC4=C(C=CC(N5CCN(CC6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7)CC6)CC5)=C4)C3=O)CC2)C=C1Cl	C44H48ClN7O5	AR	P10275	CRBN	WO-2022011204-A1
TPD-0FMIDP	SCHEMBL24186829	2-chloro-4-[3-[6-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperazine-1-carbonyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile; SCHEMBL25385636	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@@H]1N1CC2=CC(C(=O)N3CCN(C4CN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)=CC=C2C1=O	C44H44ClN7O7	AR	P10275	CRBN	WO-2022011204-A1
TPD-P6E9V3	SCHEMBL24186832	2-chloro-4-[3-[6-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidine-4-carbonyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC(Cl)=C(C#N)C=C2)C(C)(C)[C@@H]1N1CC2=C(C=CC(N3CCN(C(=O)C4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)=C2)C1=O	C46H48ClN7O7	AR	P10275	CRBN	WO-2022011204-A1
TPD-W2P4LP	SCHEMBL26212748	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]benzenesulfonamide	CC1(C)[C@H](NS(=O)(=O)C2=CC=C(N3CCN(CC4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)C=C2)C(C)(C)[C@@H]1OC1=CC=C(C#N)C(Cl)=C1	C44H50ClN7O7S	AR	P10275	CRBN	WO-2022011204-A1
TPD-AB89VQ	SCHEMBL26209852	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]benzenesulfonamide	N#CC1=CC=C(O[C@H]2CC[C@H](NS(=O)(=O)C3=CC=C(N4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C=C3)CC2)C=C1Cl	C42H46ClN7O7S	AR	P10275	CRBN	WO-2022011204-A1
TPD-IYZWCR	WO2022011204A1_118	.	C=C1C(=O)N(C2C(C)(C)C(OC3=CC(Cl)=C(C#N)C=C3)C2(C)C)C/C1=C/C(=C)N(C)CCN(C)C1CC2CN(C3=CC4=C(CC3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2C1	C47H56ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-3W1I2W	SCHEMBL24186915	2-chloro-4-[3-[2-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]-5-oxo-7H-pyrrolo[3,4-b]pyridin-6-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@@H]1N1CC2=C(C=CC(N3CCN(CC4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)=N2)C1=O	C45H49ClN8O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-82MW9L	SCHEMBL26209854	2-chloro-4-[4-[2-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]-5-oxo-7H-pyrrolo[3,4-b]pyridin-6-yl]cyclohexyl]oxybenzonitrile	N#CC1=CC=C(O[C@H]2CC[C@@H](N3CC4=C(C=CC(N5CCN(CC6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)CC5)=N4)C3=O)CC2)C=C1Cl	C43H45ClN8O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-RIXIHP	SCHEMBL24186912	2-chloro-4-[3-[6-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperazine-1-carbonyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile; SCHEMBL25384593	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@@H]1N1CC2=CC(C(=O)N3CCN(C4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)=CC=C2C1=O	C46H48ClN7O7	AR	P10275	CRBN	WO-2022011204-A1
TPD-6VJVRY	WO2022011204A1_122	.	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@@H]1N1CC2=CC(C(=O)N3CCN(CC4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)=CC=C2C1=O	C47H50ClN7O7	AR	P10275	CRBN	WO-2022011204-A1
TPD-8QLHPU	SCHEMBL26212832	2-chloro-4-[3-[6-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-2-azaspiro[3.3]heptan-6-yl]piperazine-1-carbonyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@@H]1N1CC2=CC(C(=O)N3CCN(C4CC5(C4)CN(C4=CC6=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)C5)CC3)=CC=C2C1=O	C47H48ClN7O7	AR	P10275	CRBN	WO-2022011204-A1
TPD-KJFRCR	SCHEMBL24187066	2-chloro-4-[(7S)-4-[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazine-1-carbonyl]phenyl]-7-methyl-1,4-diazepan-1-yl]benzonitrile	C[C@H]1CCN(C2=CC=C(C(=O)N3CCN(CC4CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)C=C2)CCN1C1=CC=C(C#N)C(Cl)=C1	C43H47ClN8O5	AR	P10275	CRBN	WO-2022011204-A1
TPD-URWP48	WO2022011204A1_125	.	C[C@@H]1CCN(C2=CC=C(C(=O)N3CCN(C4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)C=C2)CCN1C1=CC=C(C#N)C=C1	C42H46N8O5	AR	P10275	CRBN	WO-2022011204-A1
TPD-PO9KEU	WO2022011204A1_126	.	C[C@H]1CCN(C2=CC=C(C(=O)N3CCN(C4CN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=C2)CCN1C1=CC=C(C#N)C=C1	C40H42N8O5	AR	P10275	CRBN	WO-2022011204-A1
TPD-JE0JZ3	SCHEMBL24187065	2-Chloro-4-[1-[4-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperazine-1-carbonyl]phenyl]piperidin-4-yl]oxybenzonitrile	N#CC1=C(Cl)C=C(OC2CCN(C3=CC=C(C(=O)N4CCN(C5CN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C3)CC2)C=C1	C39H38ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-QZ903D	SCHEMBL24187069	2-chloro-4-[4-[6-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]cyclohexyl]oxybenzonitrile	N#CC1=CC=C(O[C@H]2CC[C@@H](N3CC4=C(C=CC(N5CCN(C6CN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)C6)CC5)=C4)C3=O)CC2)C=C1Cl	C41H40ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-17AWXI	SCHEMBL25385894	2-Chloro-4-[[6-[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]benzoyl]-6-azaspiro[3.5]nonan-9-yl]oxy]benzonitrile	N#CC1=CC=C(OC2CCN(C(=O)C3=CC=C(N4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C=C3)CC23CCC3)C=C1Cl	C45H48ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-QFAUIU	SCHEMBL25387092	2-Chloro-4-[[6-[4-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperazin-1-yl]benzoyl]-6-azaspiro[3.5]nonan-9-yl]oxy]benzonitrile	N#CC1=CC=C(OC2CCN(C(=O)C3=CC=C(N4CCN(C5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C=C3)CC23CCC3)C=C1Cl	C44H46ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-SLTSPZ	SCHEMBL24187054	2-Chloro-4-[1-[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]benzoyl]piperidin-4-yl]oxybenzonitrile	N#CC1=CC=C(OC2CCN(C(=O)C3=CC=C(N4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C=C3)CC2)C=C1Cl	C42H44ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-528HCM	SCHEMBL25385606	2-Chloro-4-[[5-[4-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperazin-1-yl]benzoyl]-5-azaspiro[2.5]octan-8-yl]oxy]benzonitrile	N#CC1=CC=C(OC2CCN(C(=O)C3=CC=C(N4CCN(C5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C=C3)CC23CC3)C=C1Cl	C43H44ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-62239N	SCHEMBL25386060	2-Chloro-4-[[3-[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]benzoyl]-3-azabicyclo[3.2.1]octan-8-yl]oxy]benzonitrile	N#CC1=CC=C(OC2C3CCC2CN(C(=O)C2=CC=C(N4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C=C2)C3)C=C1Cl	C44H46ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-E8UBDY	SCHEMBL25382944	2-Chloro-4-[[7-[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]benzoyl]-3-oxa-7-azabicyclo[3.3.1]nonan-9-yl]oxy]benzonitrile	N#CC1=CC=C(OC2C3COCC2CN(C(=O)C2=CC=C(N4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C=C2)C3)C=C1Cl	C44H46ClN7O7	AR	P10275	CRBN	WO-2022011204-A1
TPD-OEFOKD	WO2022011204A1_135	.	N#CC1=CC=C(OC2CC3CN(C(=O)C4=CC=C(N5CCN(C6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)CC5)C=C4)CC2O3)C=C1Cl	C42H42ClN7O7	AR	P10275	CRBN	WO-2022011204-A1
TPD-RDLOC4	SCHEMBL25383239	2-Chloro-4-[[3-[4-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperazin-1-yl]benzoyl]-3-azabicyclo[3.2.1]octan-8-yl]oxy]benzonitrile	N#CC1=CC=C(OC2C3CCC2CN(C(=O)C2=CC=C(N4CCN(C5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C=C2)C3)C=C1Cl	C43H44ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-P9HFLQ	SCHEMBL25385619	2-Chloro-4-[1-[[4-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperazine-1-carbonyl]phenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile	CC1=C(C)N(CC2=CC=C(C(=O)N3CCN(C4CN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)CC3)C=C2)N=C1C1=CC=C(C#N)C(Cl)=C1	C40H37ClN8O5	AR	P10275	CRBN	WO-2022011204-A1
TPD-B8208B	SCHEMBL24187127	2-Chloro-4-[1-[[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]methyl]piperazine-1-carbonyl]phenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile	CC1=C(C)N(CC2=CC=C(C(=O)N3CCN(CC4CN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=C2)N=C1C1=CC=C(C#N)C(Cl)=C1	C41H39ClN8O5	AR	P10275	CRBN	WO-2022011204-A1
TPD-FILG0P	SCHEMBL24187129	2-chloro-4-[1-[[4-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-3-oxo-1H-isoindol-5-yl]azetidin-3-yl]piperazine-1-carbonyl]phenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile	CC1=C(C)N(CC2=CC=C(C(=O)N3CCN(C4CN(C5=CC6=C(C=C5)CN(C5CCC(=O)NC5=O)C6=O)C4)CC3)C=C2)N=C1C1=CC=C(C#N)C(Cl)=C1	C40H39ClN8O4	AR	P10275	CRBN	WO-2022011204-A1
TPD-7MZG9H	SCHEMBL22565547	2-chloro-4-[3-[6-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperidin-4-yl]ethynyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile; SCHEMBL25387165	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@H]1N1CC2=CC(C#CC3CCN(C4CN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)=CC=C2C1=O	C46H45ClN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-SF78L7	WO2022011204A1_143	.	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@H]1N1CC2=CC(C(=O)N3CCN(CC4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)=CC=C2C1=O	C47H50ClN7O7	AR	P10275	CRBN	WO-2022011204-A1
TPD-Y54EPA	SCHEMBL24186965	2-chloro-4-[3-[6-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]methyl]piperazine-1-carbonyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile; SCHEMBL25383932	CC1(C)[C@H](OC2=CC(Cl)=C(C#N)C=C2)C(C)(C)[C@@H]1N1CC2=CC(C(=O)N3CCN(CC4CN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)=CC=C2C1=O	C45H46ClN7O7	AR	P10275	CRBN	WO-2022011204-A1
TPD-SCFGPI	SCHEMBL24187070	2-chloro-4-[3-[6-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile; SCHEMBL25384234	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@@H]1N1CC2=CC(N3CCN(C4CN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)=CC=C2C1=O	C43H44ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-66V7NU	SCHEMBL25384790	2-chloro-4-[3-[6-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-2-azaspiro[3.3]heptan-6-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile; SCHEMBL25384794	CC1(C)[C@H](OC2=CC(Cl)=C(C#N)C=C2)C(C)(C)[C@@H]1N1CC2=CC(N3CCN(CC4CC5(C4)CN(C4=CC6=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)C5)CC3)=CC=C2C1=O	C47H50ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-NNW6XZ	SCHEMBL24187073	2-chloro-4-[3-[6-[4-[6-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-6-azaspiro[3.4]octan-2-yl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile; SCHEMBL25385623	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@@H]1N1CC2=CC(N3CCN(C4CC5(CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)C4)CC3)=CC=C2C1=O	C47H50ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-EDQ1C2	SCHEMBL24187079	2-chloro-4-[3-[6-[4-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]azetidin-3-yl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@@H]1N1CC2=CC(N3CCN(C4CN(C5CN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)C4)CC3)=CC=C2C1=O	C46H49ClN8O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-5PJ034	SCHEMBL24187091	2-chloro-4-[3-[6-[4-[7-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-7-azaspiro[3.5]nonan-2-yl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile; SCHEMBL25385143	CC1(C)[C@H](OC2=CC(Cl)=C(C#N)C=C2)C(C)(C)[C@H]1N1CC2=CC(N3CCN(C4CC5(CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)C4)CC3)=CC=C2C1=O	C48H52ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-Q8JZ8D	SCHEMBL24187138	2-chloro-4-[3-[6-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]azetidin-3-yl]ethynyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile; SCHEMBL25386055	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@H]1N1CC2=CC(C#CC3CN(C4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)C3)=CC=C2C1=O	C46H45ClN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-6W4I83	SCHEMBL25386115	2-chloro-4-[3-[6-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-1-azaspiro[3.3]heptan-6-yl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile; SCHEMBL25386118	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@@H]1N1CC2=CC(N3CCN(C4CC5(CCN5C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)CC3)=CC=C2C1=O	C46H48ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-9RMFEE	SCHEMBL24187148	2-chloro-4-[3-[6-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-2-azaspiro[3.5]nonan-7-yl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile; SCHEMBL25387156	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@@H]1N1CC2=CC(N3CCN(C4CCC5(CC4)CN(C4=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C4)C5)CC3)=CC=C2C1=O	C48H52ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-UJI01B	SCHEMBL25386836	2-chloro-4-[3-[6-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-1-azaspiro[3.3]heptan-6-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile; SCHEMBL25386839	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@H]1N1CC2=CC(N3CCN(CC4CC5(CCN5C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)CC3)=CC=C2C1=O	C47H50ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-WMZCFH	SCHEMBL24187153	2-chloro-4-[3-[6-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]azetidin-3-yl]ethynyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@H]1N1CC2=CC(C#CC3CN(C4CN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)C3)=CC=C2C1=O	C44H41ClN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-HE6MB6	SCHEMBL24187154	2-chloro-4-[3-[6-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]ethynyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile; SCHEMBL25317825	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@@H]1N1CC2=CC(C#CC3CCN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)=CC=C2C1=O	C43H40ClN5O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-PGLO4Q	SCHEMBL25315729	2-chloro-4-[3-[6-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile; SCHEMBL25315732	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@H]1N1CC2=CC(C#CC3CN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)C3)=CC=C2C1=O	C41H36ClN5O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-5AWQG5	SCHEMBL25317598	2-chloro-4-[3-[6-[2-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]-2-azaspiro[3.3]heptan-6-yl]ethynyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile; SCHEMBL25317605	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@H]1N1CC2=CC(C#CC3CC4(C3)CN(C3CN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C3)C4)=CC=C2C1=O	C47H45ClN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-16T9CT	SCHEMBL25387013	2-chloro-4-[3-[6-[2-[6-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]-6-azaspiro[3.4]octan-2-yl]ethynyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile; SCHEMBL25387017	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@H]1N1CC2=CC(C#CC3CC4(CCN(C5CN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)C4)C3)=CC=C2C1=O	C48H47ClN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-AA73KV	SCHEMBL25317793	2-chloro-4-[3-[6-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-2-azaspiro[3.3]heptan-6-yl]ethynyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile; SCHEMBL25317798	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@@H]1N1CC2=CC(C#CC3CC4(C3)CN(C3=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C3)C4)=CC=C2C1=O	C44H40ClN5O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-25RVYG	SCHEMBL25319278	2-chloro-4-[3-[6-[2-[6-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-6-azaspiro[3.4]octan-2-yl]ethynyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile; SCHEMBL25319282	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@H]1N1CC2=CC(C#CC3CC4(CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)C3)=CC=C2C1=O	C45H42ClN5O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-9EVMN8	SCHEMBL25318384	2-chloro-4-[3-[6-[2-[1-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-2-azaspiro[3.3]heptan-6-yl]azetidin-3-yl]ethynyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile; SCHEMBL25318390	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@H]1N1CC2=CC(C#CC3CN(C4CC5(C4)CN(C4=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C4)C5)C3)=CC=C2C1=O	C47H45ClN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-XILTZW	SCHEMBL25384717	2-chloro-4-[4-[6-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperidin-4-yl]ethynyl]-3-oxo-1H-isoindol-2-yl]cyclohexyl]oxybenzonitrile; SCHEMBL25384721	N#CC1=C(Cl)C=C(OC2CCC(N3CC4=CC(C#CC5CCN(C6CN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)C6)CC5)=CC=C4C3=O)CC2)C=C1	C44H41ClN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-MRPOZH	SCHEMBL25385818	2-chloro-4-[4-[6-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]azetidin-3-yl]ethynyl]-3-oxo-1H-isoindol-2-yl]cyclohexyl]oxybenzonitrile; SCHEMBL25385819	N#CC1=C(Cl)C=C(OC2CCC(N3CC4=CC(C#CC5CN(C6CCN(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)C5)=CC=C4C3=O)CC2)C=C1	C44H41ClN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-BSMWQR	SCHEMBL26213817	2-chloro-4-[4-[6-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]azetidin-3-yl]ethynyl]-3-oxo-1H-isoindol-2-yl]cyclohexyl]oxybenzonitrile	N#CC1=C(Cl)C=C(OC2CCC(N3CC4=CC(C#CC5CN(C6CN(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8=O)C6)C5)=CC=C4C3=O)CC2)C=C1	C42H37ClN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-82KK3X	SCHEMBL24187150	2-chloro-4-[1-[[4-[4-[7-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]hept-6-ynoyl]piperazin-1-yl]phenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile	CC1=C(C)N(CC2=CC=C(N3CCN(C(=O)CCCCC#CC4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5)CC3)C=C2)N=C1C1=CC=C(C#N)C(Cl)=C1	C43H42ClN7O4	AR	P10275	CRBN	WO-2022011204-A1
TPD-6KD9Y7	SCHEMBL24187149	2-Chloro-4-[1-[[4-[2-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperazin-1-yl]piperidine-1-carbonyl]cyclohexyl]ethynyl]phenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile; SCHEMBL25385907	CC1=C(C)N(CC2=CC=C(C#CC3CCC(C(=O)N4CCC(N5CCN(C6=CC=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)CC3)C=C2)N=C1C1=CC=C(C#N)C(Cl)=C1	C50H51ClN8O5	AR	P10275	CRBN	WO-2022011204-A1
TPD-U8O5MB	SCHEMBL24186807	4-[3-[6-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]azetidin-3-yl]ethynyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxy-2-(trifluoromethyl)benzonitrile	CC1(C)[C@H](OC2=CC=C(C#N)C(C(F)(F)F)=C2)C(C)(C)[C@@H]1N1CC2=CC(C#CC3CN(C4CN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)C3)=CC=C2C1=O	C45H41F3N6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-0G4JPG	SCHEMBL26213872	5-[3-[6-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]azetidin-3-yl]ethynyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxy-3-(trifluoromethyl)pyridine-2-carbonitrile	CC1(C)[C@H](OC2=CN=C(C#N)C(C(F)(F)F)=C2)C(C)(C)[C@@H]1N1CC2=CC(C#CC3CN(C4CN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)C3)=CC=C2C1=O	C44H40F3N7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-Z6MWZ2	SCHEMBL25385969	2-chloro-4-[3-[6-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]azetidin-3-yl]ethynyl]-7-fluoro-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@H]1N1CC2=C(F)C(C#CC3CN(C4CN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)C3)=CC=C2C1=O	C44H40ClFN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-2J2GQF	SCHEMBL25387202	2-chloro-4-[3-[6-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]azetidin-3-yl]ethynyl]-5-fluoro-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@H]1N1CC2=CC(C#CC3CN(C4CN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)C3)=C(F)C=C2C1=O	C44H40ClFN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-VIENC9	SCHEMBL24186810	2-chloro-4-[3-[6-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]azetidin-3-yl]ethynyl]-4-fluoro-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@H]1N1CC2=CC(C#CC3CN(C4CN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)C3)=CC(F)=C2C1=O	C44H40ClFN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-O9WYEX	SCHEMBL24186814	2-chloro-4-[3-[6-[2-[1-[2-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]-2-azaspiro[3.3]heptan-6-yl]azetidin-3-yl]ethynyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@H]1N1CC2=CC(C#CC3CN(C4CC5(C4)CN(C4=CC6=C(C=C4F)C(=O)N(C4CCC(=O)NC4=O)C6=O)C5)C3)=CC=C2C1=O	C47H44ClFN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-DZSWCV	SCHEMBL26213937	2-chloro-4-[3-[6-[2-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]azetidin-3-yl]-2-azaspiro[3.3]heptan-6-yl]ethynyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@H]1N1CC2=CC(C#CC3CC4(C3)CN(C3CN(C5=CC6=C(C=C5F)C(=O)N(C5CCC(=O)NC5=O)C6=O)C3)C4)=CC=C2C1=O	C47H44ClFN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-53ALKL	SCHEMBL26213948	2-chloro-4-[3-[6-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]-2-azaspiro[3.3]heptan-6-yl]ethynyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@@H]1N1CC2=CC(C#CC3CC4(C3)CN(C3=CC5=C(C=C3F)C(=O)N(C3CCC(=O)NC3=O)C5=O)C4)=CC=C2C1=O	C44H39ClFN5O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-O127BP	SCHEMBL26213959	2-chloro-4-[3-[6-[2-[6-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]-6-azaspiro[3.4]octan-2-yl]ethynyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@@H]1N1CC2=CC(C#CC3CC4(CCN(C5=CC6=C(C=C5F)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)C3)=CC=C2C1=O	C45H41ClFN5O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-T94XZO	SCHEMBL24186849	2-chloro-4-[3-[6-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]azetidin-3-yl]ethynyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@H]1N1CC2=CC(C#CC3CN(C4=CC5=C(C=C4F)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)=CC=C2C1=O	C41H35ClFN5O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-C4S9CQ	WO2022011204A1_177	.	CC1=C(C)N(CC2=CC=C(C#CC3CCC(C(=O)NCCN(C)CCN(C)C4=CC=CC5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)C=C2)N=C1C1=CC=C(C#N)C(Cl)=C1	C47H49ClN8O5	AR	P10275	CRBN	WO-2022011204-A1
TPD-QKJFU1	SCHEMBL26213951	2-chloro-4-[3-[6-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperidin-4-yl]ethynyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@@H]1N1CC2=CC(C#CC3CCN(C4=CC5=C(C=C4F)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)=CC=C2C1=O	C43H39ClFN5O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-BQXT8U	WO2022011204A1_179	.	CC1=C(C)N(CC2=CC=C(N3CCN(CCN(C)CCN(C)C4=CC=CC5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)C=C2)N=C1C1=CC=C(C#N)C(Cl)=C1	C42H46ClN9O4	AR	P10275	CRBN	WO-2022011204-A1
TPD-HINEIB	WO2022011204A1_180	.	CC1=C(C)N(CC2=CC=C(C#CC3CCC(C(=O)N4CCN(C5CCN(C6=CC=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)CC3)C=C2)N=C1C1=CC=C(C#N)C(Cl)=C1	C50H51ClN8O5	AR	P10275	CRBN	WO-2022011204-A1
TPD-X3W6DB	SCHEMBL25385828	2-Chloro-4-[1-[[4-[2-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperazine-1-carbonyl]cyclohexyl]ethynyl]phenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile; SCHEMBL25385836	CC1=C(C)N(CC2=CC=C(C#CC3CCC(C(=O)N4CCN(C5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)CC4)CC3)C=C2)N=C1C1=CC=C(C#N)C(Cl)=C1	C45H42ClN7O5	AR	P10275	CRBN	WO-2022011204-A1
TPD-K0HFY5	SCHEMBL24186855	2-Chloro-4-[1-[[4-[2-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]piperidine-1-carbonyl]cyclohexyl]ethynyl]phenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile; SCHEMBL25383386	CC1=C(C)N(CC2=CC=C(C#CC3CCC(C(=O)N4CCC(N5CCN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)CC3)C=C2)N=C1C1=CC=C(C#N)C(Cl)=C1	C50H51ClN8O5	AR	P10275	CRBN	WO-2022011204-A1
TPD-EO0Z0X	SCHEMBL24187158	2-Chloro-4-[1-[[4-[2-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazine-1-carbonyl]cyclohexyl]ethynyl]phenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile; SCHEMBL25385946	CC1=C(C)N(CC2=CC=C(C#CC3CCC(C(=O)N4CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)C=C2)N=C1C1=CC=C(C#N)C(Cl)=C1	C45H42ClN7O5	AR	P10275	CRBN	WO-2022011204-A1
TPD-W6TGSE	SCHEMBL24187161	2-chloro-4-[1-[[4-[2-[4-[[3-[2-[6-(2,6-dioxopiperidin-3-yl)-5-oxo-7H-pyrrolo[3,4-b]pyridin-3-yl]ethynyl]azetidin-1-yl]methyl]-1-bicyclo[2.2.2]octanyl]ethynyl]phenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile	CC1=C(C)N(CC2=CC=C(C#CC34CCC(CN5CC(C#CC6=CC7=C(CN(C8CCC(=O)NC8=O)C7=O)N=C6)C5)(CC3)CC4)C=C2)N=C1C1=CC=C(C#N)C(Cl)=C1	C47H44ClN7O3	AR	P10275	CRBN	WO-2022011204-A1
TPD-JC4C9G	SCHEMBL25385604	2-Chloro-4-[1-[[4-[2-[4-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperazine-1-carbonyl]cyclohexyl]ethynyl]phenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile; SCHEMBL25385609	CC1=C(C)N(CC2=CC=C(C#CC3CCC(C(=O)N4CCN(C5CCN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)CC3)C=C2)N=C1C1=CC=C(C#N)C(Cl)=C1	C50H51ClN8O5	AR	P10275	CRBN	WO-2022011204-A1
TPD-T1XWO8	SCHEMBL24187008	2-Chloro-4-[1-[[4-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperidin-4-yl]ethynyl]phenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile	CC1=C(C)N(CC2=CC=C(C#CC3CCN(C4CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)C=C2)N=C1C1=CC=C(C#N)C(Cl)=C1	C44H42ClN7O4	AR	P10275	CRBN	WO-2022011204-A1
TPD-FHFRN5	SCHEMBL25385689	2-Chloro-4-[1-[[4-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperidin-4-yl]ethyl]piperazin-1-yl]phenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile	CC1=C(C)N(CC2=CC=C(N3CCN(CCC4CCN(C5=CC=CC6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)C=C2)N=C1C1=CC=C(C#N)C(Cl)=C1	C43H45ClN8O4	AR	P10275	CRBN	WO-2022011204-A1
TPD-SMRUYK	SCHEMBL24186793	2-Chloro-4-[[8-[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzonitrile	N#CC1=CC=C(OC2CC3CCC(C2)N3C(=O)C2=CC=C(N3CCN(CC4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)C=C2)C=C1Cl	C44H46ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-SW9AFK	SCHEMBL24187160	2-Chloro-4-[[8-[4-[2-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperidin-4-yl]ethynyl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzonitrile	N#CC1=CC=C(OC2CC3CCC(C2)N3C(=O)C2=CC=C(C#CC3CCN(CC4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)C=C2)C=C1Cl	C47H47ClN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-86A0CN	WO2022011204A1_192	.	CN(CCN1CCN(C2=CC=C(C(=O)N3C4CCC3CC(OC3=CC=C(C#N)C(Cl)=C3)C4)C=C2)CC1)CCN(C)C1=CC2=C(CC1)C(=O)N(C1CCC(=O)NC1=O)C2=O	C44H51ClN8O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-YZCZEW	SCHEMBL24187023	2-Chloro-4-[1-[[4-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]ethyl]piperazin-1-yl]phenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile	CC1=C(C)N(CC2=CC=C(N3CCN(CCC4CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)C=C2)N=C1C1=CC=C(C#N)C(Cl)=C1	C43H45ClN8O4	AR	P10275	CRBN	WO-2022011204-A1
TPD-ZYNKPU	SCHEMBL26214186	2-Chloro-4-[[8-[4-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperidin-4-yl]piperidin-4-yl]ethynyl]benzoyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzonitrile	N#CC1=CC=C(OC2CC3CCC(C2)N3C(=O)C2=CC=C(C#CC3CCN(C4CCN(C5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)CC4)CC3)C=C2)C=C1Cl	C46H45ClN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-42SCBM	SCHEMBL26214240	2-chloro-4-[1-[[4-[2-[4-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]ethynyl]piperidine-1-carbonyl]cyclohexyl]ethynyl]phenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile	CC1=C(C)N(CC2=CC=C(C#CC3CCC(C(=O)N4CCC(C#CC5=CC=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)CC3)C=C2)N=C1C1=CC(Cl)=C(C#N)C=C1	C48H45ClN6O4	AR	P10275	CRBN	WO-2022011204-A1
TPD-0R3KF3	SCHEMBL26214249	2-chloro-4-[1-[[4-[5-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]ethynyl]piperidin-1-yl]-5-oxopent-1-ynyl]phenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile	CC1=C(C)N(CC2=CC=C(C#CCCC(=O)N3CCC(C#CC4=CC=CC5=C4CN(C4CCC(=O)NC4=O)C5=O)CC3)C=C2)N=C1C1=CC(Cl)=C(C#N)C=C1	C44H39ClN6O4	AR	P10275	CRBN	WO-2022011204-A1
TPD-UNB6PX	WO2022011204A1_200	.	CC1=C(C)N(CC2=CC=C(C#CC3CCN(CCC#CC4=CC=CC5=C4CN(C4CCC(=O)NC4=O)C5=O)CC3)C=C2)N=C1C1=CC(Cl)=C(C#N)C=C1	C43H39ClN6O3	AR	P10275	CRBN	WO-2022011204-A1
TPD-4ZF21X	SCHEMBL26209916	2-chloro-4-[1-[[4-[2-[1-[5-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]pent-4-ynyl]piperidin-4-yl]ethynyl]phenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile	CC1=C(C)N(CC2=CC=C(C#CC3CCN(CCCC#CC4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5)CC3)C=C2)N=C1C1=CC(Cl)=C(C#N)C=C1	C44H41ClN6O3	AR	P10275	CRBN	WO-2022011204-A1
TPD-EUDANG	SCHEMBL26209917	2-chloro-4-[1-[[4-[2-[1-[5-[2-(2,6-dioxopiperidin-3-yl)-3-oxo-1H-isoindol-5-yl]pent-4-ynyl]piperidin-4-yl]ethynyl]phenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile	CC1=C(C)N(CC2=CC=C(C#CC3CCN(CCCC#CC4=CC5=C(C=C4)CN(C4CCC(=O)NC4=O)C5=O)CC3)C=C2)N=C1C1=CC(Cl)=C(C#N)C=C1	C44H41ClN6O3	AR	P10275	CRBN	WO-2022011204-A1
TPD-E9RD8U	WO2022011204A1_203	.	C=C(C#CC1CCC(N2CC(C#CC3=CC=CC4=C3CN(C3CCC(=O)NC3=O)C4=O)C2)CC1)/C=C\C(=C)CN1N=C(C2=CC(Cl)=C(C#N)C=C2)C(C)=C1C	C45H43ClN6O3	AR	P10275	CRBN	WO-2022011204-A1
TPD-D7WU6U	WO2022011204A1_204	.	C=C(C#CC1CCC(N2CC(C#CC3=CC=C4C(=O)N(C5CCC(=O)NC5=O)CC4=C3)C2)CC1)/C=C\C(=C)CN1N=C(C2=CC(Cl)=C(C#N)C=C2)C(C)=C1C	C45H43ClN6O3	AR	P10275	CRBN	WO-2022011204-A1
TPD-CLBYGU	SCHEMBL26209921	2-chloro-4-[1-[[4-[2-[4-[3-[2-[2-(2,6-dioxopiperidin-3-yl)-3-oxo-1H-isoindol-5-yl]ethynyl]azetidin-1-yl]cyclohexyl]ethynyl]phenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile	CC1=C(C)N(CC2=CC=C(C#CC3CCC(N4CC(C#CC5=CC6=C(C=C5)CN(C5CCC(=O)NC5=O)C6=O)C4)CC3)C=C2)N=C1C1=CC(Cl)=C(C#N)C=C1	C45H41ClN6O3	AR	P10275	CRBN	WO-2022011204-A1
TPD-WR7D5K	WO2022011204A1_206	.	C=C(C#CC1=CC=C(CN2CC(C#CC3=CC=CC4=C3CN(C3CCC(=O)NC3=O)C4=O)C2)C=C1)/C=C\C(=C)CN1N=C(C2=CC(Cl)=C(C#N)C=C2)C(C)=C1C	C46H39ClN6O3	AR	P10275	CRBN	WO-2022011204-A1
TPD-TWJ0YY	WO2022011204A1_207	.	C=C(C#CC1=CC=C(CN2CC(C#CC3=CC=C4C(=O)N(C5CCC(=O)NC5=O)CC4=C3)C2)C=C1)/C=C\C(=C)CN1N=C(C2=CC(Cl)=C(C#N)C=C2)C(C)=C1C	C46H39ClN6O3	AR	P10275	CRBN	WO-2022011204-A1
TPD-CH6TU7	SCHEMBL26209925	2-chloro-4-[1-[[4-[2-[4-[[3-[2-[2-(2,6-dioxopiperidin-3-yl)-3-oxo-1H-isoindol-5-yl]ethynyl]azetidin-1-yl]methyl]phenyl]ethynyl]phenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile	CC1=C(C)N(CC2=CC=C(C#CC3=CC=C(CN4CC(C#CC5=CC6=C(C=C5)CN(C5CCC(=O)NC5=O)C6=O)C4)C=C3)C=C2)N=C1C1=CC(Cl)=C(C#N)C=C1	C46H37ClN6O3	AR	P10275	CRBN	WO-2022011204-A1
TPD-TSPVGO	SCHEMBL26209926	2-chloro-4-[1-[[4-[2-[4-[[3-[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]ethynyl]azetidin-1-yl]methyl]cyclohexyl]ethynyl]phenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile	CC1=C(C)N(CC2=CC=C(C#CC3CCC(CN4CC(C#CC5=CC=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)C4)CC3)C=C2)N=C1C1=CC(Cl)=C(C#N)C=C1	C46H43ClN6O3	AR	P10275	CRBN	WO-2022011204-A1
TPD-WJ4G8B	WO2022011204A1_210	.	C=C(C#CC1CCC(CN2CC(C#CC3=CC=C4C(=O)N(C5CCC(=O)NC5=O)CC4=C3)C2)CC1)C=CC(=C)CN1N=C(C2=CC(Cl)=C(C#N)C=C2)C(C)=C1C	C46H45ClN6O3	AR	P10275	CRBN	WO-2022011204-A1
TPD-KT3I4M	SCHEMBL26209931	2-chloro-4-[1-[[4-[2-[4-[[3-[2-[2-(2,6-dioxopiperidin-3-yl)-3-oxo-1H-isoindol-5-yl]ethynyl]azetidin-1-yl]methyl]cyclohexyl]ethynyl]phenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile	CC1=C(C)N(CC2=CC=C(C#CC3CCC(CN4CC(C#CC5=CC6=C(C=C5)CN(C5CCC(=O)NC5=O)C6=O)C4)CC3)C=C2)N=C1C1=CC(Cl)=C(C#N)C=C1	C46H43ClN6O3	AR	P10275	CRBN	WO-2022011204-A1
TPD-M9VI1N	WO2022011204A1_212	.	C=C(C#CC1CCC(CN2CCC(C#CC3=CC=CC4=C3CN(C3CCC(=O)NC3=O)C4=O)CC2)CC1)/C=C\C(=C)CN1N=C(C2=CC(Cl)=C(C#N)C=C2)C(C)=C1C	C48H49ClN6O3	AR	P10275	CRBN	WO-2022011204-A1
TPD-3J1IL7	WO2022011204A1_213	.	C=C(C#CC1CCC(CN2CCC(C#CC3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4)CC2)CC1)/C=C/C(=C)CN1N=C(C2=CC(Cl)=C(C#N)C=C2)C(C)=C1C	C48H49ClN6O3	AR	P10275	CRBN	WO-2022011204-A1
TPD-LDB71M	SCHEMBL26209941	2-chloro-4-[1-[[4-[2-[4-[[4-[2-[2-(2,6-dioxopiperidin-3-yl)-3-oxo-1H-isoindol-5-yl]ethynyl]piperidin-1-yl]methyl]cyclohexyl]ethynyl]phenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile; SCHEMBL26209974	CC1=C(C)N(CC2=CC=C(C#CC3CCC(CN4CCC(C#CC5=CC6=C(C=C5)CN(C5CCC(=O)NC5=O)C6=O)CC4)CC3)C=C2)N=C1C1=CC(Cl)=C(C#N)C=C1	C48H47ClN6O3	AR	P10275	CRBN	WO-2022011204-A1
TPD-K5AFTO	WO2022011204A1_215	.	C=C(C#CC(C)CCN(C)C1=CC=CC2=C1CN(C1CCC(=O)NC1=O)C2=O)/C=C\C(=C)CN1N=C(C2=CC(Cl)=C(C#N)C=C2)C(C)=C1C	C39H39ClN6O3	AR	P10275	CRBN	WO-2022011204-A1
TPD-LWL38I	WO2022011204A1_216	.	CC1=C(C)N(CC2=CC=C(C#CC(C)CCN(C)C3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4)C=C2)N=C1C1=CC(Cl)=C(C#N)C=C1	C39H37ClN6O3	AR	P10275	CRBN	WO-2022011204-A1
TPD-2AM12Q	SCHEMBL24187164	2-chloro-4-[1-[[4-[2-[4-[3-[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]ethynyl]azetidine-1-carbonyl]cyclohexyl]ethynyl]phenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile	CC1=C(C)N(CC2=CC=C(C#CC3CCC(C(=O)N4CC(C#CC5=CC=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)C4)CC3)C=C2)N=C1C1=CC(Cl)=C(C#N)C=C1	C46H41ClN6O4	AR	P10275	CRBN	WO-2022011204-A1
TPD-TJHD3U	SCHEMBL26209949	2-chloro-4-[1-[[4-[2-[4-[3-[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]ethynyl]azetidine-1-carbonyl]cyclohexyl]ethynyl]phenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile	CC1=C(C)N(CC2=CC=C(C#CC3CCC(C(=O)N4CC(C#CC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6)C4)CC3)C=C2)N=C1C1=CC(Cl)=C(C#N)C=C1	C46H41ClN6O4	AR	P10275	CRBN	WO-2022011204-A1
TPD-VFL2SZ	SCHEMBL24186896	2-chloro-4-[1-[[4-[2-[4-[3-[2-[2-(2,6-dioxopiperidin-3-yl)-3-oxo-1H-isoindol-5-yl]ethynyl]azetidine-1-carbonyl]cyclohexyl]ethynyl]phenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile	CC1=C(C)N(CC2=CC=C(C#CC3CCC(C(=O)N4CC(C#CC5=CC6=C(C=C5)CN(C5CCC(=O)NC5=O)C6=O)C4)CC3)C=C2)N=C1C1=CC(Cl)=C(C#N)C=C1	C46H41ClN6O4	AR	P10275	CRBN	WO-2022011204-A1
TPD-A4Q4R6	SCHEMBL26209950	2-chloro-4-[1-[[4-[2-[4-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]ethynyl]piperidine-1-carbonyl]cyclohexyl]ethynyl]phenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile	CC1=C(C)N(CC2=CC=C(C#CC3CCC(C(=O)N4CCC(C#CC5=CC=C6C(=O)N(C7CCC(=O)NC7=O)CC6=C5)CC4)CC3)C=C2)N=C1C1=CC(Cl)=C(C#N)C=C1	C48H45ClN6O4	AR	P10275	CRBN	WO-2022011204-A1
TPD-J96NZF	WO2022011204A1_222	.	C=C(C#CC1CCN(CC2CCC(C#CC3=CC=CC4=C3CN(C3CCC(=O)NC3=O)C4=O)CC2)CC1)C=CC(=C)CN1N=C(C2=CC(Cl)=C(C#N)C=C2)C(C)=C1C	C48H49ClN6O3	AR	P10275	CRBN	WO-2022011204-A1
TPD-576XBX	WO2022011204A1_223	.	C=C(C#CC1CCN(CC2CCC(C#CC3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4)CC2)CC1)C=CC(=C)CN1N=C(C2=CC(Cl)=C(C#N)C=C2)C(C)=C1C	C48H49ClN6O3	AR	P10275	CRBN	WO-2022011204-A1
TPD-U1LUIV	SCHEMBL26209955	2-chloro-4-[1-[[4-[2-[1-[[4-[2-[2-(2,6-dioxopiperidin-3-yl)-3-oxo-1H-isoindol-5-yl]ethynyl]cyclohexyl]methyl]piperidin-4-yl]ethynyl]phenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile	CC1=C(C)N(CC2=CC=C(C#CC3CCN(CC4CCC(C#CC5=CC6=C(C=C5)CN(C5CCC(=O)NC5=O)C6=O)CC4)CC3)C=C2)N=C1C1=CC(Cl)=C(C#N)C=C1	C48H47ClN6O3	AR	P10275	CRBN	WO-2022011204-A1
TPD-MUA3T2	SCHEMBL24186898	2-chloro-4-[1-[[4-[2-[1-[[4-[2-[2-(2,6-dioxopiperidin-3-yl)-3-oxo-1H-isoindol-5-yl]ethynyl]cyclohexyl]methyl]azetidin-3-yl]ethynyl]phenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile	CC1=C(C)N(CC2=CC=C(C#CC3CN(CC4CCC(C#CC5=CC6=C(C=C5)CN(C5CCC(=O)NC5=O)C6=O)CC4)C3)C=C2)N=C1C1=CC(Cl)=C(C#N)C=C1	C46H43ClN6O3	AR	P10275	CRBN	WO-2022011204-A1
TPD-U5PL2H	SCHEMBL24187101	2-chloro-4-[1-[[4-[2-[1-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]ethynyl]cyclohexanecarbonyl]piperidin-4-yl]ethynyl]phenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile	CC1=C(C)N(CC2=CC=C(C#CC3CCN(C(=O)C4CCC(C#CC5=CC=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)CC3)C=C2)N=C1C1=CC(Cl)=C(C#N)C=C1	C48H45ClN6O4	AR	P10275	CRBN	WO-2022011204-A1
TPD-9MPCBR	SCHEMBL24187103	2-chloro-4-[1-[[4-[2-[1-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-3-oxo-1H-isoindol-5-yl]ethynyl]cyclohexanecarbonyl]piperidin-4-yl]ethynyl]phenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile	CC1=C(C)N(CC2=CC=C(C#CC3CCN(C(=O)C4CCC(C#CC5=CC6=C(C=C5)CN(C5CCC(=O)NC5=O)C6=O)CC4)CC3)C=C2)N=C1C1=CC(Cl)=C(C#N)C=C1	C48H45ClN6O4	AR	P10275	CRBN	WO-2022011204-A1
TPD-JUQN8G	SCHEMBL24187105	2-chloro-4-[1-[[4-[2-[1-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-3-oxo-1H-isoindol-5-yl]ethynyl]cyclohexanecarbonyl]azetidin-3-yl]ethynyl]phenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile	CC1=C(C)N(CC2=CC=C(C#CC3CN(C(=O)C4CCC(C#CC5=CC6=C(C=C5)CN(C5CCC(=O)NC5=O)C6=O)CC4)C3)C=C2)N=C1C1=CC(Cl)=C(C#N)C=C1	C46H41ClN6O4	AR	P10275	CRBN	WO-2022011204-A1
TPD-S1VBGN	SCHEMBL26209958	2-Chloro-4-[1-[[4-[2-[4-[[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]-3,9-diazaspiro[5.5]undecan-9-yl]methyl]cyclohexyl]ethynyl]phenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile	CC1=C(C)N(CC2=CC=C(C#C[C@H]3CC[C@H](CN4CCC5(CC4)CCN(C4=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C4)CC5)CC3)C=C2)N=C1C1=CC(Cl)=C(C#N)C=C1	C50H52ClN7O4	AR	P10275	CRBN	WO-2022011204-A1
TPD-IPR07B	SCHEMBL26209960	2-Chloro-4-[1-[[4-[2-[4-[[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-3,9-diazaspiro[5.5]undecan-9-yl]methyl]cyclohexyl]ethynyl]phenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile	CC1=C(C)N(CC2=CC=C(C#CC3CCC(CN4CCC5(CC4)CCN(C4=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C4)CC5)CC3)C=C2)N=C1C1=CC(Cl)=C(C#N)C=C1	C50H52ClN7O4	AR	P10275	CRBN	WO-2022011204-A1
TPD-74GE03	SCHEMBL24187093	2-chloro-4-[1-[[4-[2-[4-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-3-oxo-1H-isoindol-5-yl]ethynyl]piperidin-1-yl]cyclohexyl]ethynyl]phenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile	CC1=C(C)N(CC2=CC=C(C#CC3CCC(N4CCC(C#CC5=CC6=C(C=C5)CN(C5CCC(=O)NC5=O)C6=O)CC4)CC3)C=C2)N=C1C1=CC(Cl)=C(C#N)C=C1	C47H45ClN6O3	AR	P10275	CRBN	WO-2022011204-A1
TPD-WXFTM3	SCHEMBL26209961	2-chloro-4-[1-[[4-[2-[2-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-3-oxo-1H-isoindol-5-yl]ethynyl]cyclohexyl]-2-azaspiro[3.5]nonan-7-yl]ethynyl]phenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile	CC1=C(C)N(CC2=CC=C(C#CC3CCC4(CC3)CN(C3CCC(C#CC5=CC6=C(C=C5)CN(C5CCC(=O)NC5=O)C6=O)CC3)C4)C=C2)N=C1C1=CC(Cl)=C(C#N)C=C1	C50H49ClN6O3	AR	P10275	CRBN	WO-2022011204-A1
TPD-W9M4UF	SCHEMBL26209962	2-chloro-4-[1-[[4-[2-[4-[[3-[2-[2-(2,6-dioxopiperidin-3-yl)-3-oxo-1H-isoindol-5-yl]ethynyl]azetidin-1-yl]methyl]-1-bicyclo[2.2.2]octanyl]ethynyl]phenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile	CC1=C(C)N(CC2=CC=C(C#CC34CCC(CN5CC(C#CC6=CC=C7CN(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)(CC3)CC4)C=C2)N=C1C1=CC(Cl)=C(C#N)C=C1	C48H45ClN6O3	AR	P10275	CRBN	WO-2022011204-A1
TPD-1EY8OA	SCHEMBL26209964	2-chloro-4-[1-[[4-[2-[4-[[3-[2-[2-(2,6-dioxopiperidin-3-yl)-3-oxo-1H-isoindol-5-yl]ethynyl]piperidin-1-yl]methyl]cyclohexyl]ethynyl]phenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile	CC1=C(C)N(CC2=CC=C(C#CC3CCC(CN4CCCC(C#CC5=CC6=C(C=C5)CN(C5CCC(=O)NC5=O)C6=O)C4)CC3)C=C2)N=C1C1=CC(Cl)=C(C#N)C=C1	C48H47ClN6O3	AR	P10275	CRBN	WO-2022011204-A1
TPD-JPRAFE	SCHEMBL26209968	2-chloro-4-[1-[[4-[2-[4-[[3-[2-[2-(2,6-dioxopiperidin-3-yl)-3-oxo-1H-isoindol-5-yl]ethynyl]pyrrolidin-1-yl]methyl]cyclohexyl]ethynyl]phenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile	CC1=C(C)N(CC2=CC=C(C#CC3CCC(CN4CCC(C#CC5=CC6=C(C=C5)CN(C5CCC(=O)NC5=O)C6=O)C4)CC3)C=C2)N=C1C1=CC(Cl)=C(C#N)C=C1	C47H45ClN6O3	AR	P10275	CRBN	WO-2022011204-A1
TPD-BUWRCI	WO2022011204A1_236	.	CC1=C(C2=NN(CC3=CC=C(C#CC4CCC(CN5CCC(C#CC6=CC7=C(C=C6)CN(C6CCC(=O)NC6=O)C7=O)CC5)CC4)C=C3)C(C)=C2C)C=CC(C#N)=C1Cl	C49H49ClN6O3	AR	P10275	CRBN	WO-2022011204-A1
TPD-HHSAZC	WO2022011204A1_237	.	CC1=C(C2=NN(CC3=CC=C(C#CC4CCC(CN5CC(C#CC6=CC7=C(C=C6)CN(C6CCC(=O)NC6=O)C7=O)C5)CC4)C=C3)C(C)=C2C)C=CC(C#N)=C1Cl	C47H45ClN6O3	AR	P10275	CRBN	WO-2022011204-A1
TPD-OJJMKK	WO2022011204A1_238	.	C=C(C#CC1CCC(CN2CC(C#CC3=CC=C(C(=O)NC4CCC(=O)NC4=O)C=C3)C2)CC1)/C=C/C(=C)CN1N=C(C2=CC(Cl)=C(C#N)C=C2)C(C)=C1C	C45H45ClN6O3	AR	P10275	CRBN	WO-2022011204-A1
TPD-XL708D	SCHEMBL26209987	2-chloro-4-[1-[[4-[2-[4-[[4-[[2-(2,6-dioxopiperidin-3-yl)-3-oxo-1H-isoindol-5-yl]oxy]piperidin-1-yl]methyl]cyclohexyl]ethynyl]phenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile	CC1=C(C)N(CC2=CC=C(C#CC3CCC(CN4CCC(OC5=CC6=C(C=C5)CN(C5CCC(=O)NC5=O)C6=O)CC4)CC3)C=C2)N=C1C1=CC(Cl)=C(C#N)C=C1	C46H47ClN6O4	AR	P10275	CRBN	WO-2022011204-A1
TPD-EX6FM4	SCHEMBL24186987	2-chloro-4-[1-[[4-[2-[4-[[4-[[2-(2,6-dioxopiperidin-3-yl)-3-oxo-1H-isoindol-5-yl]oxy]piperidin-1-yl]methyl]cyclohexyl]ethynyl]phenyl]methyl]-5,6-dihydro-4H-cyclopenta[c]pyrazol-3-yl]-3-methylbenzonitrile	CC1=C(C2=NN(CC3=CC=C(C#CC4CCC(CN5CCC(OC6=CC7=C(C=C6)CN(C6CCC(=O)NC6=O)C7=O)CC5)CC4)C=C3)C3=C2CCC3)C=CC(C#N)=C1Cl	C48H49ClN6O4	AR	P10275	CRBN	WO-2022011204-A1
TPD-0OJC2T	SCHEMBL24187060	2-chloro-4-[1-[[4-[2-[4-[[3-[2-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-3-oxo-1H-isoindol-5-yl]ethynyl]azetidin-1-yl]methyl]cyclohexyl]ethynyl]phenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile	CC1=C(C)N(CC2=CC=C(C#CC3CCC(CN4CC(C#CC5=CC6=C(C=C5F)CN(C5CCC(=O)NC5=O)C6=O)C4)CC3)C=C2)N=C1C1=CC(Cl)=C(C#N)C=C1	C46H42ClFN6O3	AR	P10275	CRBN	WO-2022011204-A1
TPD-K3UIXG	WO2022011204A1_242	.	N#CC1=CC=C(OC2C3CCC2CN(C(=O)C2=CC=C(C#CC4CCN(C5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C=C2)C3)C=C1Cl	C46H45ClN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-1XJ60L	SCHEMBL26214799	2-Chloro-4-[[2-[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperidin-4-yl]methyl]piperazin-1-yl]benzoyl]-2-azabicyclo[2.2.1]heptan-7-yl]oxy]benzonitrile	N#CC1=CC=C(OC2C3CCC2N(C(=O)C2=CC=C(N4CCN(CC5CCN(C6=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)CC5)CC4)C=C2)C3)C=C1Cl	C43H44ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-M040VP	SCHEMBL26214826	2-Chloro-4-[[2-[4-[2-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperidin-4-yl]methyl]piperidin-4-yl]ethynyl]benzoyl]-2-azabicyclo[2.2.1]heptan-7-yl]oxy]benzonitrile	N#CC1=CC=C(OC2C3CCC2N(C(=O)C2=CC=C(C#CC4CCN(CC5CCN(C6=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)CC5)CC4)C=C2)C3)C=C1Cl	C46H45ClN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-1EWCRY	SCHEMBL26214839	2-Chloro-4-[[2-[4-[2-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperidin-4-yl]ethynyl]benzoyl]-2-azabicyclo[2.2.1]heptan-7-yl]oxy]benzonitrile	N#CC1=CC=C(OC2C3CCC2N(C(=O)C2=CC=C(C#CC4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C=C2)C3)C=C1Cl	C46H45ClN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-FSAPQN	SCHEMBL26214856	2-Chloro-4-[[2-[4-[2-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]azetidin-3-yl]methyl]piperidin-4-yl]ethynyl]benzoyl]-2-azabicyclo[2.2.1]heptan-7-yl]oxy]benzonitrile	N#CC1=CC=C(OC2C3CCC2N(C(=O)C2=CC=C(C#CC4CCN(CC5CN(C6=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)C5)CC4)C=C2)C3)C=C1Cl	C44H41ClN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-HT89V9	SCHEMBL26214863	2-Chloro-4-[[2-[4-[2-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]methyl]piperidin-4-yl]ethynyl]benzoyl]-2-azabicyclo[2.2.1]heptan-7-yl]oxy]benzonitrile	N#CC1=CC=C(OC2C3CCC2N(C(=O)C2=CC=C(C#CC4CCN(CC5CN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C2)C3)C=C1Cl	C44H41ClN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-CMGNPU	SCHEMBL24186839	2-Chloro-4-[4-[4-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperidin-4-yl]methyl]piperidin-4-yl]phenoxy]piperidin-1-yl]benzonitrile	N#CC1=C(Cl)C=C(N2CCC(OC3=CC=C(C4CCN(CC5CCN(C6=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)CC5)CC4)C=C3)CC2)C=C1	C42H45ClN6O5	AR	P10275	CRBN	WO-2022011204-A1
TPD-78RWKC	SCHEMBL24187191	2-Chloro-4-[4-[4-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperidin-4-yl]phenoxy]piperidin-1-yl]benzonitrile	N#CC1=C(Cl)C=C(N2CCC(OC3=CC=C(C4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C=C3)CC2)C=C1	C42H45ClN6O5	AR	P10275	CRBN	WO-2022011204-A1
TPD-XYUHVS	SCHEMBL24186840	2-Chloro-4-[1-[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperidin-4-yl]methyl]piperazin-1-yl]benzoyl]azepan-4-yl]oxybenzonitrile	N#CC1=C(Cl)C=C(OC2CCCN(C(=O)C3=CC=C(N4CCN(CC5CCN(C6=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)CC5)CC4)C=C3)CC2)C=C1	C43H46ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-YNWQW2	SCHEMBL24186847	2-Chloro-4-[1-[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]benzoyl]azepan-4-yl]oxybenzonitrile	N#CC1=C(Cl)C=C(OC2CCCN(C(=O)C3=CC=C(N4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C=C3)CC2)C=C1	C43H46ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-Y4TQDS	SCHEMBL24187020	2-Chloro-4-[1-[4-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperidin-4-yl]methyl]piperidin-4-yl]benzoyl]piperidin-4-yl]oxybenzonitrile	N#CC1=C(Cl)C=C(OC2CCN(C(=O)C3=CC=C(C4CCN(CC5CCN(C6=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)CC5)CC4)C=C3)CC2)C=C1	C43H45ClN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-9MGQOX	SCHEMBL23138838	2-Chloro-4-[1-[4-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperidin-4-yl]benzoyl]piperidin-4-yl]oxybenzonitrile	N#CC1=C(Cl)C=C(OC2CCN(C(=O)C3=CC=C(C4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C=C3)CC2)C=C1	C43H45ClN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-AUZ6AU	WO2022011204A1_260	.	N#CC1=C(Cl)C=C(N2CCC(OC3=CC=C(C4CCN(CCC5CCN(C6=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)CC5)CC4)C=C3)CC2)C=C1	C43H47ClN6O5	AR	P10275	CRBN	WO-2022011204-A1
TPD-J3OUDR	SCHEMBL26215085	2-Chloro-4-[4-[4-[1-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]ethyl]piperidin-4-yl]phenoxy]piperidin-1-yl]benzonitrile	N#CC1=C(Cl)C=C(N2CCC(OC3=CC=C(C4CCN(CCC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C=C3)CC2)C=C1	C43H47ClN6O5	AR	P10275	CRBN	WO-2022011204-A1
TPD-T5JBC3	SCHEMBL26215103	2-Chloro-4-[1-[[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]phenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile	CC1=C(C)N(CC2=CC=C(N3CCN(CC4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)C=C2)N=C1C1=CC=C(C#N)C(Cl)=C1	C42H43ClN8O4	AR	P10275	CRBN	WO-2022011204-A1
TPD-7EFUJV	SCHEMBL26215130	2-Chloro-4-[1-[[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperidin-4-yl]methyl]piperazin-1-yl]phenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile	CC1=C(C)N(CC2=CC=C(N3CCN(CC4CCN(C5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)CC4)CC3)C=C2)N=C1C1=CC=C(C#N)C(Cl)=C1	C42H43ClN8O4	AR	P10275	CRBN	WO-2022011204-A1
TPD-P6RDQP	SCHEMBL26215162	2-chloro-4-[1-[[4-[4-[[4-[2-[2-(2,6-dioxopiperidin-3-yl)-3-oxo-1H-isoindol-4-yl]ethynyl]piperidin-1-yl]methyl]piperidine-1-carbonyl]phenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile	CC1=C(C)N(CC2=CC=C(C(=O)N3CCC(CN4CCC(C#CC5=C6C(=O)N(C7CCC(=O)NC7=O)CC6=CC=C5)CC4)CC3)C=C2)N=C1C1=CC=C(C#N)C(Cl)=C1	C46H46ClN7O4	AR	P10275	CRBN	WO-2022011204-A1
TPD-TCTT6A	SCHEMBL26215187	4-[[3-(3-chloro-4-cyanophenyl)-4,5-dimethylpyrazol-1-yl]methyl]-N-[1-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-3-oxo-1H-isoindol-4-yl]ethynyl]cyclohexyl]piperidin-4-yl]benzamide	CC1=C(C)N(CC2=CC=C(C(=O)NC3CCN(C4CCC(C#CC5=C6C(=O)N(C7CCC(=O)NC7=O)CC6=CC=C5)CC4)CC3)C=C2)N=C1C1=CC=C(C#N)C(Cl)=C1	C46H46ClN7O4	AR	P10275	CRBN	WO-2022011204-A1
TPD-WEYEY2	SCHEMBL24187171	2-chloro-4-[(3R)-1-[4-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperidin-4-yl]ethynyl]benzoyl]-4,4-dimethylpyrrolidin-3-yl]oxybenzonitrile	CC1(C)CN(C(=O)C2=CC=C(C#CC3CCN(C4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)C=C2)C[C@@H]1OC1=CC=C(C#N)C(Cl)=C1	C45H45ClN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-44WOLR	SCHEMBL24187177	2-chloro-4-[(3R)-1-[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]benzoyl]-4,4-dimethylpyrrolidin-3-yl]oxybenzonitrile	CC1(C)CN(C(=O)C2=CC=C(N3CCN(CC4CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)C=C2)C[C@@H]1OC1=CC=C(C#N)C(Cl)=C1	C43H46ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-UXHFFS	SCHEMBL24187173	2-chloro-4-[(3R)-1-[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperidin-4-yl]methyl]piperazin-1-yl]benzoyl]-4,4-dimethylpyrrolidin-3-yl]oxybenzonitrile	CC1(C)CN(C(=O)C2=CC=C(N3CCN(CC4CCN(C5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)CC4)CC3)C=C2)C[C@@H]1OC1=CC=C(C#N)C(Cl)=C1	C43H46ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-FNHVUJ	SCHEMBL24187179	2-Chloro-4-[1-[4-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperidin-4-yl]ethynyl]benzoyl]piperidin-3-yl]oxybenzonitrile	N#CC1=CC=C(OC2CCCN(C(=O)C3=CC=C(C#CC4CCN(C5CCN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)C=C3)C2)C=C1Cl	C44H43ClN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-NR5P2Z	SCHEMBL26215271	2-Chloro-4-[1-[4-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperidin-4-yl]piperidin-4-yl]ethynyl]benzoyl]piperidin-3-yl]oxybenzonitrile	N#CC1=CC=C(OC2CCCN(C(=O)C3=CC=C(C#CC4CCN(C5CCN(C6=CC=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)C=C3)C2)C=C1Cl	C44H43ClN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-BF77HS	SCHEMBL26215292	2-Chloro-4-[1-[4-[2-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperidin-4-yl]methyl]piperidin-4-yl]ethynyl]benzoyl]piperidin-3-yl]oxybenzonitrile	N#CC1=CC=C(OC2CCCN(C(=O)C3=CC=C(C#CC4CCN(CC5CCN(C6=CC=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)C=C3)C2)C=C1Cl	C45H45ClN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-JUYVQ5	WO2022011204A1_273	.	N#CC1=CC=C(OC2CCCN(C(=O)C3=CC=C(C#CC4CCN(CC5CCN(C6=CC7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7C=C6)CC5)CC4)C=C3)C2)C=C1Cl	C45H47ClN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-S93RH6	SCHEMBL24187180	2-Chloro-4-[1-[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperidin-4-yl]methyl]piperazin-1-yl]benzoyl]piperidin-3-yl]oxybenzonitrile	N#CC1=CC=C(OC2CCCN(C(=O)C3=CC=C(N4CCN(CC5CCN(C6=CC=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)C=C3)C2)C=C1Cl	C42H44ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-GXLNUV	SCHEMBL24187170	2-Chloro-4-[1-[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]benzoyl]piperidin-3-yl]oxybenzonitrile	N#CC1=CC=C(OC2CCCN(C(=O)C3=CC=C(N4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C=C3)C2)C=C1Cl	C42H44ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-I7RCXT	SCHEMBL24186928	2-Chloro-4-[[8-[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperidin-4-yl]methyl]piperazin-1-yl]phenyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzonitrile	N#CC1=CC=C(OC2CC3CCC(C2)N3C2=CC=C(N3CCN(CC4CCN(C5=CC=CC6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)C=C2)C=C1Cl	C43H46ClN7O5	AR	P10275	CRBN	WO-2022011204-A1
TPD-0O1TVU	SCHEMBL24186947	2-Chloro-4-[[8-[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]phenyl]-8-azabicyclo[3.2.1]octan-3-yl]oxy]benzonitrile	N#CC1=CC=C(OC2CC3CCC(C2)N3C2=CC=C(N3CCN(CC4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)C=C2)C=C1Cl	C43H46ClN7O5	AR	P10275	CRBN	WO-2022011204-A1
TPD-MICMW5	WO2022011204A1_278	.	CC1(C)CN(C(=O)C2=CC=C(N3CCN(CC4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)C=C2)CC[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C44H48ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-LKR1T7	SCHEMBL24186945	2-Chloro-4-[1-[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperidin-4-yl]methyl]piperazin-1-yl]benzoyl]-3,3-dimethylpiperidin-4-yl]oxybenzonitrile	CC1(C)CN(C(=O)C2=CC=C(N3CCN(CC4CCN(C5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)CC4)CC3)C=C2)CCC1OC1=CC=C(C#N)C(Cl)=C1	C44H48ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-MRI21Z	SCHEMBL24186938	2-Chloro-4-[1-[4-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperidin-4-yl]ethynyl]benzoyl]-3,3-dimethylpiperidin-4-yl]oxybenzonitrile	CC1(C)CN(C(=O)C2=CC=C(C#CC3CCN(C4CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)C=C2)CCC1OC1=CC=C(C#N)C(Cl)=C1	C46H47ClN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-VU093B	SCHEMBL24186949	2-Chloro-4-[1-[4-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperidin-4-yl]piperidin-4-yl]ethynyl]benzoyl]-3,3-dimethylpiperidin-4-yl]oxybenzonitrile	CC1(C)CN(C(=O)C2=CC=C(C#CC3CCN(C4CCN(C5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)CC4)CC3)C=C2)CCC1OC1=CC=C(C#N)C(Cl)=C1	C46H47ClN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-4QBAA1	SCHEMBL24186939	2-Chloro-4-[1-[4-[4-[7-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-7-azaspiro[3.5]nonan-2-yl]piperazin-1-yl]benzoyl]piperidin-4-yl]oxybenzonitrile	N#CC1=CC=C(OC2CCN(C(=O)C3=CC=C(N4CCN(C5CC6(CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)C5)CC4)C=C3)CC2)C=C1Cl	C44H46ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-VESFJC	SCHEMBL24186940	2-Chloro-4-[1-[4-[4-[7-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]-7-azaspiro[3.5]nonan-2-yl]piperazin-1-yl]benzoyl]piperidin-4-yl]oxybenzonitrile	N#CC1=CC=C(OC2CCN(C(=O)C3=CC=C(N4CCN(C5CC6(CCN(C7=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=CC=C7)CC6)C5)CC4)C=C3)CC2)C=C1Cl	C44H46ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-KYCXPZ	SCHEMBL26215456	2-Chloro-4-[1-[4-[2-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]-2,7-diazaspiro[3.5]nonan-7-yl]benzoyl]piperidin-4-yl]oxybenzonitrile	N#CC1=CC=C(OC2CCN(C(=O)C3=CC=C(N4CCC5(CC4)CN(CC4CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC4)C5)C=C3)CC2)C=C1Cl	C45H48ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-BI5HUO	SCHEMBL26215473	2-Chloro-4-[1-[4-[2-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperidin-4-yl]methyl]-2,7-diazaspiro[3.5]nonan-7-yl]benzoyl]piperidin-4-yl]oxybenzonitrile	N#CC1=CC=C(OC2CCN(C(=O)C3=CC=C(N4CCC5(CC4)CN(CC4CCN(C6=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)CC4)C5)C=C3)CC2)C=C1Cl	C45H48ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-I4J6I5	SCHEMBL24186865	2-Chloro-4-[1-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]-2,7-diazaspiro[3.5]nonan-7-yl]benzoyl]piperidin-4-yl]oxybenzonitrile	N#CC1=CC=C(OC2CCN(C(=O)C3=CC=C(N4CCC5(CC4)CN(C4CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC4)C5)C=C3)CC2)C=C1Cl	C44H46ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-6SYX7K	SCHEMBL24186867	2-Chloro-4-[1-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperidin-4-yl]-2,7-diazaspiro[3.5]nonan-7-yl]benzoyl]piperidin-4-yl]oxybenzonitrile	N#CC1=CC=C(OC2CCN(C(=O)C3=CC=C(N4CCC5(CC4)CN(C4CCN(C6=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)CC4)C5)C=C3)CC2)C=C1Cl	C44H46ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-L3DEVA	SCHEMBL24186860	2-Chloro-4-[1-[4-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]azetidin-3-yl]benzoyl]piperidin-4-yl]oxybenzonitrile	N#CC1=CC=C(OC2CCN(C(=O)C3=CC=C(C4CN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)C4)C=C3)CC2)C=C1Cl	C41H41ClN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-MBDEJB	WO2022011204A1_289	.	N#CC1=CC=C(OC2CCN(C(=O)C3=CC=C(C4CN(CC5CCN(C6=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)CC5)C4)C=C3)CC2)C=C1Cl	C41H41ClN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-FUCLGS	SCHEMBL24186871	2-Chloro-4-[1-[4-[1-[7-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-7-azaspiro[3.5]nonan-2-yl]azetidin-3-yl]benzoyl]piperidin-4-yl]oxybenzonitrile	N#CC1=CC=C(OC2CCN(C(=O)C3=CC=C(C4CN(C5CC6(CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)C5)C4)C=C3)CC2)C=C1Cl	C43H43ClN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-NHC4E5	SCHEMBL24187102	2-Chloro-4-[1-[4-[1-[7-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]-7-azaspiro[3.5]nonan-2-yl]azetidin-3-yl]benzoyl]piperidin-4-yl]oxybenzonitrile	N#CC1=CC=C(OC2CCN(C(=O)C3=CC=C(C4CN(C5CC6(CCN(C7=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=CC=C7)CC6)C5)C4)C=C3)CC2)C=C1Cl	C43H43ClN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-038VWZ	SCHEMBL26215548	4-[3-[6-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperidin-4-yl]ethynyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxy-2-methylbenzonitrile	CC1=CC(O[C@H]2C(C)(C)[C@@H](N3CC4=CC(C#CC5CCN(C6CN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)C6)CC5)=CC=C4C3=O)C2(C)C)=CC=C1C#N	C47H48N6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-AESI65	SCHEMBL26215556	4-[3-[6-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperidin-4-yl]ethynyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxy-2-(trifluoromethyl)benzonitrile	CC1(C)[C@H](OC2=CC=C(C#N)C(C(F)(F)F)=C2)C(C)(C)[C@@H]1N1CC2=CC(C#CC3CCN(C4CN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)=CC=C2C1=O	C47H45F3N6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-971GQJ	SCHEMBL26215567	5-[3-[6-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperidin-4-yl]ethynyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxy-3-(trifluoromethyl)pyridine-2-carbonitrile	CC1(C)[C@H](OC2=CN=C(C#N)C(C(F)(F)F)=C2)C(C)(C)[C@H]1N1CC2=CC(C#CC3CCN(C4CN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)=CC=C2C1=O	C46H44F3N7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-071Y55	SCHEMBL24187096	2-chloro-4-[3-[6-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperidin-4-yl]ethynyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxy-3-methylbenzonitrile	CC1=C(Cl)C(C#N)=CC=C1O[C@H]1C(C)(C)[C@H](N2CC3=CC(C#CC4CCN(C5CN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)=CC=C3C2=O)C1(C)C	C47H47ClN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-YUTFNU	SCHEMBL24187090	4-[3-[6-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperidin-4-yl]ethynyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxy-2-fluorobenzonitrile	CC1(C)[C@H](OC2=CC=C(C#N)C(F)=C2)C(C)(C)[C@H]1N1CC2=CC(C#CC3CCN(C4CN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)=CC=C2C1=O	C46H45FN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-2D8NH5	SCHEMBL26215623	4-[3-[6-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperidin-4-yl]ethynyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxy-2-fluoro-3-methylbenzonitrile	CC1=C(F)C(C#N)=CC=C1O[C@H]1C(C)(C)[C@H](N2CC3=CC(C#CC4CCN(C5CN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)=CC=C3C2=O)C1(C)C	C47H47FN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-KYM5QK	SCHEMBL24187178	2-chloro-4-[3-[6-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperidin-4-yl]ethynyl]-7-fluoro-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@H]1N1CC2=C(F)C(C#CC3CCN(C4CN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)=CC=C2C1=O	C46H44ClFN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-C5ERRF	SCHEMBL24187181	2-chloro-4-[3-[6-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperidin-4-yl]ethynyl]-5-fluoro-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@H]1N1CC2=CC(C#CC3CCN(C4CN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)=C(F)C=C2C1=O	C46H44ClFN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-N288JK	SCHEMBL26215652	2-chloro-4-[3-[6-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperidin-4-yl]ethynyl]-4-fluoro-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@H]1N1CC2=CC(C#CC3CCN(C4CN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)=CC(F)=C2C1=O	C46H44ClFN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-4G9UKZ	SCHEMBL22565065	2-chloro-4-[3-[2-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperidin-4-yl]ethynyl]-5-oxo-7H-pyrrolo[3,4-b]pyridin-6-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@H]1N1CC2=NC(C#CC3CCN(C4CN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)=CC=C2C1=O	C45H44ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-HUOF1R	SCHEMBL26215678	2-chloro-4-[3-[6-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperidin-4-yl]ethynyl]-3-oxo-1H-pyrrolo[3,4-c]pyridin-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@H]1N1CC2=CC(C#CC3CCN(C4CN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)=NC=C2C1=O	C45H44ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-505NDD	SCHEMBL24187172	2-chloro-4-[3-[3-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperidin-4-yl]ethynyl]-7-oxo-5H-pyrrolo[3,4-b]pyridin-6-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@H]1N1CC2=CC(C#CC3CCN(C4CN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)=CN=C2C1=O	C45H44ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-INX3EZ	SCHEMBL24187175	2-chloro-4-[3-[6-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperidin-4-yl]ethynyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@H]1N1CC2=CC(C#CC3CCN(C4CN(C5=CC6=C(C=C5F)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)CC3)=CC=C2C1=O	C46H44ClFN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-HPRW6E	SCHEMBL24186925	2-chloro-4-[3-[6-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxopyrrolo[3,4-c]pyridin-6-yl]azetidin-3-yl]piperidin-4-yl]ethynyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@H]1N1CC2=CC(C#CC3CCN(C4CN(C5=CC6=C(C=N5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)CC3)=CC=C2C1=O	C45H44ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-X2RO3W	SCHEMBL24186948	2-chloro-4-[3-[6-[2-[1-[1-[6-(2,6-dioxopiperidin-3-yl)-5,7-dioxopyrrolo[3,4-b]pyridin-3-yl]azetidin-3-yl]piperidin-4-yl]ethynyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@H]1N1CC2=CC(C#CC3CCN(C4CN(C5=CC6=C(N=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)CC3)=CC=C2C1=O	C45H44ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-PVB0DI	SCHEMBL26215760	2-chloro-4-[3-[6-[2-[1-[1-[6-(2,6-dioxopiperidin-3-yl)-5,7-dioxopyrrolo[3,4-b]pyrazin-3-yl]azetidin-3-yl]piperidin-4-yl]ethynyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@H]1N1CC2=CC(C#CC3CCN(C4CN(C5=NC6=C(N=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)CC3)=CC=C2C1=O	C44H43ClN8O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-2SYTLB	SCHEMBL24186942	2-chloro-4-[3-[6-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]azetidin-3-yl]piperidin-4-yl]ethynyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@H]1N1CC2=CC(C#CC3CCN(C4CN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6)C4)CC3)=CC=C2C1=O	C46H47ClN6O5	AR	P10275	CRBN	WO-2022011204-A1
TPD-M428I7	SCHEMBL26215775	2-chloro-4-[2,2,4,4-tetramethyl-3-[6-[2-[1-[1-[2-(1-methyl-2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperidin-4-yl]ethynyl]-3-oxo-1H-isoindol-2-yl]cyclobutyl]oxybenzonitrile	CN1C(=O)CCC(N2C(=O)C3=CC=C(N4CC(N5CCC(C#CC6=CC=C7C(=O)N([C@H]8C(C)(C)[C@H](OC9=CC=C(C#N)C(Cl)=C9)C8(C)C)CC7=C6)CC5)C4)C=C3C2=O)C1=O	C47H47ClN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-WD755K	SCHEMBL26215785	2-chloro-4-[3-[6-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperidin-4-yl]ethynyl]-7-fluoro-3-oxo-1H-pyrrolo[3,4-c]pyridin-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@H]1N1CC2=C(F)C(C#CC3CCN(C4CN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)=NC=C2C1=O	C45H43ClFN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-7JQUUB	SCHEMBL26215798	2-chloro-4-[3-[3-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperidin-4-yl]ethynyl]-7-oxo-5H-pyrrolo[3,4-b]pyrazin-6-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@H]1N1CC2=NC(C#CC3CCN(C4CN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)=CN=C2C1=O	C44H43ClN8O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-JFZ9YN	SCHEMBL24186833	2-chloro-4-[3-[6-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-3-oxo-1H-isoindol-5-yl]azetidin-3-yl]piperidin-4-yl]ethynyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@H]1N1CC2=CC(C#CC3CCN(C4CN(C5=CC=C6CN(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)=CC=C2C1=O	C46H47ClN6O5	AR	P10275	CRBN	WO-2022011204-A1
TPD-XUQECT	SCHEMBL26215835	2-chloro-4-[3-[6-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]azetidin-3-yl]piperidin-4-yl]ethynyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@H]1N1CC2=CC(C#CC3CCN(C4CN(C5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)C4)CC3)=CC=C2C1=O	C46H45ClN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-XRATQU	SCHEMBL26215877	2-chloro-4-[3-[6-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]azetidin-3-yl]ethynyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxy-3-methylbenzonitrile	CC1=C(Cl)C(C#N)=CC=C1O[C@H]1C(C)(C)[C@H](N2CC3=CC(C#CC4CN(C5CN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)C4)=CC=C3C2=O)C1(C)C	C45H43ClN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-H9WP47	SCHEMBL26215888	4-[3-[6-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]azetidin-3-yl]ethynyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxy-2-fluorobenzonitrile	CC1(C)[C@H](OC2=CC=C(C#N)C(F)=C2)C(C)(C)[C@H]1N1CC2=CC(C#CC3CN(C4CN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)C3)=CC=C2C1=O	C44H41FN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-TN9U46	SCHEMBL26215903	4-[3-[6-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]azetidin-3-yl]ethynyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxy-2-fluoro-3-methylbenzonitrile	CC1=C(F)C(C#N)=CC=C1O[C@H]1C(C)(C)[C@H](N2CC3=CC(C#CC4CN(C5CN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)C4)=CC=C3C2=O)C1(C)C	C45H43FN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-TBYZ7O	SCHEMBL26215911	4-[3-[6-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]azetidin-3-yl]ethynyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxy-2-methylbenzonitrile	CC1=CC(O[C@H]2C(C)(C)[C@H](N3CC4=CC(C#CC5CN(C6CN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)C6)C5)=CC=C4C3=O)C2(C)C)=CC=C1C#N	C45H44N6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-GCHJZS	SCHEMBL22565054	2-chloro-4-[3-[2-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]azetidin-3-yl]ethynyl]-5-oxo-7H-pyrrolo[3,4-b]pyridin-6-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@H]1N1CC2=NC(C#CC3CN(C4CN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)C3)=CC=C2C1=O	C43H40ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-GZZNNQ	SCHEMBL26215932	2-chloro-4-[3-[6-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]azetidin-3-yl]ethynyl]-3-oxo-1H-pyrrolo[3,4-c]pyridin-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@H]1N1CC2=CC(C#CC3CN(C4CN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)C3)=NC=C2C1=O	C43H40ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-Y37WXC	SCHEMBL26215937	2-chloro-4-[3-[3-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]azetidin-3-yl]ethynyl]-7-oxo-5H-pyrrolo[3,4-b]pyridin-6-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@H]1N1CC2=CC(C#CC3CN(C4CN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)C3)=CN=C2C1=O	C43H40ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-D6DMEZ	SCHEMBL26215957	2-chloro-4-[3-[6-[2-[1-[1-[6-(2,6-dioxopiperidin-3-yl)-5,7-dioxopyrrolo[3,4-b]pyridin-3-yl]azetidin-3-yl]azetidin-3-yl]ethynyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@H]1N1CC2=CC(C#CC3CN(C4CN(C5=CC6=C(N=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)C3)=CC=C2C1=O	C43H40ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-A49ZOO	SCHEMBL26215971	2-chloro-4-[3-[6-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxopyrrolo[3,4-c]pyridin-6-yl]azetidin-3-yl]azetidin-3-yl]ethynyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@H]1N1CC2=CC(C#CC3CN(C4CN(C5=CC6=C(C=N5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)C3)=CC=C2C1=O	C43H40ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-JW7NQR	SCHEMBL26215980	2-chloro-4-[3-[6-[2-[1-[1-[6-(2,6-dioxopiperidin-3-yl)-5,7-dioxopyrrolo[3,4-b]pyridin-2-yl]azetidin-3-yl]azetidin-3-yl]ethynyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@H]1N1CC2=CC(C#CC3CN(C4CN(C5=NC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)C3)=CC=C2C1=O	C43H40ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-RCDS57	SCHEMBL26215992	2-chloro-4-[3-[6-[2-[1-[1-[6-(2,6-dioxopiperidin-3-yl)-5,7-dioxopyrrolo[3,4-b]pyrazin-3-yl]azetidin-3-yl]azetidin-3-yl]ethynyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@H]1N1CC2=CC(C#CC3CN(C4CN(C5=NC6=C(N=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)C3)=CC=C2C1=O	C42H39ClN8O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-AASA6M	SCHEMBL26213915	2-chloro-4-[3-[6-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]azetidin-3-yl]azetidin-3-yl]ethynyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@H]1N1CC2=CC(C#CC3CN(C4CN(C5=CC6=C(C=C5F)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)C3)=CC=C2C1=O	C44H40ClFN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-9H0796	WO2022011204A1_329	.	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@H]1N1CC2=CC(C#CC3CN(C4CN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6)C4)C3)=CC=C2C1=O	C44H43ClN6O5	AR	P10275	CRBN	WO-2022011204-A1
TPD-CAJ0PG	SCHEMBL26216027	2-chloro-4-[3-[6-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]azetidin-3-yl]azetidin-3-yl]ethynyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@H]1N1CC2=CC(C#CC3CN(C4CN(C5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)C4)C3)=CC=C2C1=O	C44H41ClN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-LXN3ED	SCHEMBL26216038	2-chloro-4-[2,2,4,4-tetramethyl-3-[6-[2-[1-[1-[2-(1-methyl-2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]azetidin-3-yl]ethynyl]-3-oxo-1H-isoindol-2-yl]cyclobutyl]oxybenzonitrile	CN1C(=O)CCC(N2C(=O)C3=CC=C(N4CC(N5CC(C#CC6=CC=C7C(=O)N([C@H]8C(C)(C)[C@H](OC9=CC=C(C#N)C(Cl)=C9)C8(C)C)CC7=C6)C5)C4)C=C3C2=O)C1=O	C45H43ClN6O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-7NWFM5	SCHEMBL26216070	2-chloro-4-[3-[3-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]azetidin-3-yl]ethynyl]-4-fluoro-7-oxo-5H-pyrrolo[3,4-b]pyridin-6-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@H]1N1CC2=C(F)C(C#CC3CN(C4CN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)C3)=CN=C2C1=O	C43H39ClFN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-11116F	SCHEMBL26216081	2-chloro-4-[3-[6-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-3-oxo-1H-isoindol-5-yl]azetidin-3-yl]azetidin-3-yl]ethynyl]-3-oxo-1H-isoindol-2-yl]-2,2,4,4-tetramethylcyclobutyl]oxybenzonitrile	CC1(C)[C@H](OC2=CC=C(C#N)C(Cl)=C2)C(C)(C)[C@H]1N1CC2=CC(C#CC3CN(C4CN(C5=CC6=C(C=C5)CN(C5CCC(=O)NC5=O)C6=O)C4)C3)=CC=C2C1=O	C44H43ClN6O5	AR	P10275	CRBN	WO-2022011204-A1
TPD-P2KCUV	SCHEMBL24187185	2-Chloro-4-[1-[[4-[2-[4-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]ethynyl]piperidine-1-carbonyl]cyclohexyl]ethynyl]phenyl]methyl]-4,5-dimethylpyrazol-3-yl]benzonitrile	CC1=C(C)N(CC2=CC=C(C#CC3CCC(C(=O)N4CCC(C#CC5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)C=C2)N=C1C1=CC(Cl)=C(C#N)C=C1	C48H43ClN6O5	AR	P10275	CRBN	WO-2022011204-A1
TPD-46A4Q3	CHEMBL4875549	2-Chloro-4-[1-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]piperidin-1-yl]benzoyl]piperidin-4-yl]oxybenzonitrile; SCHEMBL24187026; PD172468	N#CC1=C(Cl)C=C(OC2CCN(C(=O)C3=CC=C(N4CCC(N5CCN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)C=C3)CC2)C=C1	C41H42ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-CZEP6W	SCHEMBL24187024	2-Chloro-4-[1-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]piperidin-1-yl]benzoyl]azepan-4-yl]oxybenzonitrile; PD172469	N#CC1=CC=C(OC2CCCN(C(=O)C3=CC=C(N4CCC(N5CCN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)C=C3)CC2)C=C1Cl	C42H44ClN7O6	AR	P10275	CRBN	WO-2022011204-A1
TPD-9L48LU	SCHEMBL24187027	2-Chloro-4-[1-[[4-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperazine-1-carbonyl]phenyl]methyl]pyrazol-3-yl]benzonitrile	N#CC1=C(Cl)C=C(C2=NN(CC3=CC=C(C(=O)N4CCN(C5CCN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)C=C3)C=C2)C=C1	C40H37ClN8O5	AR	P10275	CRBN	WO-2022011204-A1
TPD-1JLVPJ	PD216410	2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]-N-[2-[2-[2-[4-[4-[[4-[[2-[methyl(methylsulfonyl)amino]phenyl]methylamino]-5-(trifluoromethyl)pyrimidin-2-yl]amino]phenyl]piperazin-1-yl]ethoxy]ethoxy]ethyl]acetamide	CN(c1ccccc1CNc1nc(Nc2ccc(N3CCN(CCOCCOCCNC(=O)CNc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)cc2)ncc1C(F)(F)F)S(C)(=O)=O	C45H52F3N11O9S	FAK	Q05397	CRBN	WO-2022028372-A1
TPD-VC3TIJ	WO2022028372A1_2	N-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethyl]-3-[3-[4-[4-[[4-[[2-[methyl(methylsulfonyl)amino]phenyl]methylamino]-5-(trifluoromethyl)pyrimidin-2-yl]amino]phenyl]piperazin-1-yl]propoxy]propanamide	CN(c1ccccc1CNc1nc(Nc2ccc(N3CCN(CCCOCCC(=O)NCCNc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)cc2)ncc1C(F)(F)F)S(C)(=O)=O	C45H52F3N11O8S	FAK	Q05397	CRBN	WO-2022028372-A1
TPD-ODP374	WO2022028372A1_3	N-[2-[[[2-[4-[4-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethyl]piperazin-1-yl]anilino]-5-(trifluoromethyl)pyrimidin-4-yl]amino]methyl]phenyl]-N-methylmethanesulfonamide	CN(c1ccccc1CNc1nc(Nc2ccc(N3CCN(CCOCCOCCNc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)cc2)ncc1C(F)(F)F)S(C)(=O)=O	C43H49F3N10O8S	FAK	Q05397	CRBN	WO-2022028372-A1
TPD-BLRXD4	WO2022028372A1_4	.	CN(c1ccccc1CNc1nc(Nc2ccc(N3CCN(CCOCCOCCOCCNc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)cc2)ncc1C(F)(F)F)S(C)(=O)=O	C45H53F3N10O9S	FAK	Q05397	CRBN	WO-2022028372-A1
TPD-MMSLCE	WO2022028372A1_5	.	CN(c1ccccc1CNc1nc(Nc2ccc(N3CCN(CCCCC(=O)Nc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)cc2)ncc1C(F)(F)F)S(C)(=O)=O	C42H45F3N10O7S	FAK	Q05397	CRBN	WO-2022028372-A1
TPD-O1AWLL	PD216411	N-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]-6-[4-[4-[[4-[[2-[methyl(methylsulfonyl)amino]phenyl]methylamino]-5-(trifluoromethyl)pyrimidin-2-yl]amino]phenyl]piperazin-1-yl]hexanamide	CN(c1ccccc1CNc1nc(Nc2ccc(N3CCN(CCCCCC(=O)Nc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)cc2)ncc1C(F)(F)F)S(C)(=O)=O	C43H47F3N10O7S	FAK	Q05397	CRBN	WO-2022028372-A1
TPD-KQRGYR	WO2022028372A1_7	.	CN(c1ccccc1CNc1nc(Nc2ccc(N3CCN(CCCCCCC(=O)Nc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)cc2)ncc1C(F)(F)F)S(C)(=O)=O	C44H49F3N10O7S	FAK	Q05397	CRBN	WO-2022028372-A1
TPD-33WCRB	WO2022028372A1_8	.	CN(c1ccccc1CNc1nc(Nc2ccc(N3CCN(CCCCCCCC(=O)Nc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)cc2)ncc1C(F)(F)F)S(C)(=O)=O	C45H51F3N10O7S	FAK	Q05397	CRBN	WO-2022028372-A1
TPD-R50IEH	WO2022028372A1_9	.	CN(c1ccccc1CNc1nc(Nc2ccc(N3CCN(CCCCCCCCC(=O)Nc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)cc2)ncc1C(F)(F)F)S(C)(=O)=O	C46H53F3N10O7S	FAK	Q05397	CRBN	WO-2022028372-A1
TPD-PUNKL2	WO2022028372A1_10	.	CN(c1ccccc1CNc1nc(Nc2ccc(N3CCN(CCCCCCCCCC(=O)Nc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)cc2)ncc1C(F)(F)F)S(C)(=O)=O	C47H55F3N10O7S	FAK	Q05397	CRBN	WO-2022028372-A1
TPD-7EC9VZ	WO2022028372A1_11	.	CN(c1ccccc1CNc1nc(Nc2ccc(N3CCN(CCCCC(=O)NCCNc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)cc2)ncc1C(F)(F)F)S(C)(=O)=O	C44H50F3N11O7S	FAK	Q05397	CRBN	WO-2022028372-A1
TPD-8B2QVM	WO2022028372A1_12	N-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethyl]-6-[4-[4-[[4-[[2-[methyl(methylsulfonyl)amino]phenyl]methylamino]-5-(trifluoromethyl)pyrimidin-2-yl]amino]phenyl]piperazin-1-yl]hexanamide	CN(c1ccccc1CNc1nc(Nc2ccc(N3CCN(CCCCCC(=O)NCCNc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)cc2)ncc1C(F)(F)F)S(C)(=O)=O	C45H52F3N11O7S	FAK	Q05397	CRBN	WO-2022028372-A1
TPD-QYLL59	PD216412	N-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethyl]-7-[4-[4-[[4-[[2-[methyl(methylsulfonyl)amino]phenyl]methylamino]-5-(trifluoromethyl)pyrimidin-2-yl]amino]phenyl]piperazin-1-yl]heptanamide	CN(c1ccccc1CNc1nc(Nc2ccc(N3CCN(CCCCCCC(=O)NCCNc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)cc2)ncc1C(F)(F)F)S(C)(=O)=O	C46H54F3N11O7S	FAK	Q05397	CRBN	WO-2022028372-A1
TPD-VM6FJ6	WO2022028372A1_14	.	CN(c1ccccc1CNc1nc(Nc2ccc(N3CCN(CCCCCCCC(=O)NCCNc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)cc2)ncc1C(F)(F)F)S(C)(=O)=O	C47H56F3N11O7S	FAK	Q05397	CRBN	WO-2022028372-A1
TPD-5XP6ZK	WO2022028372A1_15	.	CN(c1ccccc1CNc1nc(Nc2ccc(N3CCN(CCCCCCCCCC(=O)NCCNc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)cc2)ncc1C(F)(F)F)S(C)(=O)=O	C49H60F3N11O7S	FAK	Q05397	CRBN	WO-2022028372-A1
TPD-DXJGG8	WO2022028372A1_16	.	CN(c1ccccc1CNc1nc(Nc2ccc(N3CCN(CCCCC(=O)Nc4cccc5c4CN(C4CCC(=O)NC4=O)C5=O)CC3)cc2)ncc1C(F)(F)F)S(C)(=O)=O	C42H47F3N10O6S	FAK	Q05397	CRBN	WO-2022028372-A1
TPD-5OY23U	WO2022028372A1_17	.	CN(c1ccccc1CNc1nc(Nc2ccc(N3CCN(CCCCCC(=O)Nc4cccc5c4CN(C4CCC(=O)NC4=O)C5=O)CC3)cc2)ncc1C(F)(F)F)S(C)(=O)=O	C43H49F3N10O6S	FAK	Q05397	CRBN	WO-2022028372-A1
TPD-JPFNUO	WO2022028372A1_18	.	CN(c1ccccc1CNc1nc(Nc2ccc(N3CCN(CCCCCCCC(=O)Nc4cccc5c4CN(C4CCC(=O)NC4=O)C5=O)CC3)cc2)ncc1C(F)(F)F)S(C)(=O)=O	C45H53F3N10O6S	FAK	Q05397	CRBN	WO-2022028372-A1
TPD-SGYGVR	WO2022028372A1_19	N-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]-10-[4-[4-[[4-[[2-[methyl(methylsulfonyl)amino]phenyl]methylamino]-5-(trifluoromethyl)pyrimidin-2-yl]amino]phenyl]piperazin-1-yl]decanamide	CN(c1ccccc1CNc1nc(Nc2ccc(N3CCN(CCCCCCCCCC(=O)Nc4cccc5c4CN(C4CCC(=O)NC4=O)C5=O)CC3)cc2)ncc1C(F)(F)F)S(C)(=O)=O	C47H57F3N10O6S	FAK	Q05397	CRBN	WO-2022028372-A1
TPD-0DH2IM	WO2022028372A1_20	N-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-5-[4-[4-[[4-[[2-[methyl(methylsulfonyl)amino]phenyl]methylamino]-5-(trifluoromethyl)pyrimidin-2-yl]amino]phenyl]piperazin-1-yl]pentanamide	CN(c1ccccc1CNc1nc(Nc2ccc(N3CCN(CCCCC(=O)Nc4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)cc2)ncc1C(F)(F)F)S(C)(=O)=O	C42H45F3N10O7S	FAK	Q05397	CRBN	WO-2022028372-A1
TPD-E32X00	WO2022028372A1_21	.	CN(c1ccccc1CNc1nc(Nc2ccc(N3CCN(CCCCCC(=O)Nc4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)cc2)ncc1C(F)(F)F)S(C)(=O)=O	C43H47F3N10O7S	FAK	Q05397	CRBN	WO-2022028372-A1
TPD-A9S5E0	WO2022028372A1_22	.	CN(c1ccccc1CNc1nc(Nc2ccc(N3CCN(CCCCCCCC(=O)Nc4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)cc2)ncc1C(F)(F)F)S(C)(=O)=O	C45H51F3N10O7S	FAK	Q05397	CRBN	WO-2022028372-A1
TPD-Z7KBNN	WO2022028372A1_23	.	CN(c1ccccc1CNc1nc(Nc2ccc(N3CCN(CCCCCCCCCC(=O)Nc4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)cc2)ncc1C(F)(F)F)S(C)(=O)=O	C47H55F3N10O7S	FAK	Q05397	CRBN	WO-2022028372-A1
TPD-I55RNW	SCHEMBL30253819	(3R)-N-[3-[5-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-2-azaspiro[3.3]heptan-6-yl]oxy]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide; SCHEMBL30253825	O=C1CCC(N2CC3=CC(N4CC5(CC(OC6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6)C5)C4)=CC=C3C2=O)C(=O)N1	C43H38F3N7O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-O90BC2	WO2022047145A1_2	.	C[C@@]12CN(CC3CCC(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)CC5=C4)CC3)C[C@]1(C)CN(C1=CC=C(C3=CC4=C(N=C3)NC=C4C(=O)C3=C(F)C=CC(CS(=O)(=O)C4CC[C@@H](F)C4)=C3F)C=C1)C2	C54H57F3N6O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-CHXBY6	SCHEMBL30254045	(3R)-N-[3-[5-[4-[(3aR,7aS)-2-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]-3,3a,4,6,7,7a-hexahydro-1H-pyrrolo[3,4-c]pyridin-5-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	[H][C@]12CCN(C3=CC=C(C4=CC5=C(N=C4)NC=C5C(=O)C4=C(F)C=CC(NS(=O)(=O)N5CC[C@@H](F)C5)=C4F)C=C3)C[C@@]1([H])CN(CC1CCN(C3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4)CC1)C2	C50H52F3N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-WAWD7S	WO2022047145A1_4	.	O=C1CCC(N2CC3=CC(N4CC5(CCN(CC#CC6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)C8CC[C@@H](F)C8)=C7F)C=C6)C5)C4)=CC=C3C2=O)C(=O)N1	C47H42F3N7O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-RYRYJ6	SCHEMBL24319499	(3R)-N-[3-[5-[4-[(1R,4R)-5-[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]azetidin-3-yl]-2,5-diazabicyclo[2.2.1]heptan-2-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide; SCHEMBL30253690	O=C1CCC(N2CC3=C(C=CC(N4CC(N5C[C@H]6C[C@@H]5CN6C5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)C4)=C3)C2=O)C(=O)N1	C45H42F3N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-9TOOGR	CHEMBL5173366	(3R)-N-[3-[5-[4-[9-[[1-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]-3,9-diazaspiro[5.5]undecan-3-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide; SCHEMBL24319496; SCHEMBL30253919	COC1=C2C(=O)N(C3CCC(=O)NC3=O)CC2=CC(N2CCC(CN3CCC4(CC3)CCN(C3=CC=C(C5=CC6=C(N=C5)NC=C6C(=O)C5=C(F)C=CC(NS(=O)(=O)N6CC[C@@H](F)C6)=C5F)C=C3)CC4)CC2)=C1	C53H58F3N9O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-WUW2CA	SCHEMBL24319497	(3R)-N-[3-[5-[4-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]azetidin-3-yl]methyl]piperidin-4-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide; SCHEMBL30253844	O=C1CCC(N2CC3=CC(N4CC(CN5CCC(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6)CC5)C4)=CC=C3C2=O)C(=O)N1	C46H45F3N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-67S960	SCHEMBL30254115	(3R)-N-[3-[5-[2-[[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-2-azaspiro[3.3]heptan-6-yl]methyl]-3,4-dihydro-1H-isoquinolin-6-yl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(N4CC5(CC(CN6CCC7=C(C=CC(C8=CC9=C(N=C8)NC=C9C(=O)C8=C(F)C=CC(NS(=O)(=O)N9CC[C@@H](F)C9)=C8F)=C7)C6)C5)C4)=CC=C3C2=O)C(=O)N1	C47H45F3N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-ITEVY0	SCHEMBL29482961	(3R)-N-[3-[5-[4-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]-1,6-diazaspiro[3.3]heptan-6-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(N4CCC(N5CCC56CN(C5=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C5)C6)CC4)=CC=C3C2=O)C(=O)N1	C47H46F3N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-J7WTTQ	SCHEMBL30253665	(3R)-N-[3-[5-[4-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-2,8-diazaspiro[4.5]decan-8-yl]ethyl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=C(C=CC(N4CCC5(CCN(CCC6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6)CC5)C4)=C3)C2=O)C(=O)N1	C47H47F3N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-3XH687	SCHEMBL24021726	(3R)-N-[3-[5-[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]-3-fluorophenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide; SCHEMBL30253834	O=C1CCC(N2CC3=CC(N4CCC(CN5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6F)CC5)CC4)=CC=C3C2=O)C(=O)N1	C47H47F4N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-BDNZ9G	SCHEMBL30253646	(3R)-N-[3-[5-[4-[4-[[(3S)-6-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-5-yl]-3-methyl-2,6-diazaspiro[3.3]heptan-2-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	COC1=CC(N2CC3(C2)CN(CC2CCN(C4=CC=C(C5=CC6=C(N=C5)NC=C6C(=O)C5=C(F)C=CC(NS(=O)(=O)N6CC[C@@H](F)C6)=C5F)C=C4)CC2)[C@H]3C)=CC2=C1C(=O)N(C1CCC(=O)NC1=O)C2	C50H52F3N9O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-HFO48G	SCHEMBL24319918	(3R)-N-[3-[5-[4-[4-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]oxy]-8-oxa-5-azaspiro[3.5]nonan-5-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide; SCHEMBL24319919; SCHEMBL30254251	O=C1CCC(N2CC3=C(C=CC(O[C@H]4C[C@@]5(COCCN5CC5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6)CC5)C4)=C3)C2=O)C(=O)N1	C50H51F3N8O8S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-VDEZFK	WO2022047145A1_14	.	O=C1CCC(N2CC3=C(C=CC(O[C@H]4C[C@]5(COCCN5CC5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)C7F)C=C6)CC5)C4)=C3)C2=O)C(=O)N1	C50H53F3N8O8S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-ZXW5EU	SCHEMBL24319922	(3R)-N-[3-[5-[4-[[(2R)-1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]azetidin-2-yl]methoxy]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide; SCHEMBL30253808	O=C1CCC(N2CC3=CC(N4CC[C@@H]4COC4=CC=C(C5=CC6=C(N=C5)NC=C6C(=O)C5=C(F)C=CC(NS(=O)(=O)N6CC[C@@H](F)C6)=C5F)C=C4)=CC=C3C2=O)C(=O)N1	C41H36F3N7O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-QK8P02	WO2022047145A1_16	.	O=C1CCC(N2CC3C=C(N4CCC(N5C[C@@H]6C[C@H]5CN(C5=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C5)C6)CC4)C=CC3C2=O)C(=O)N1	C48H50F3N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-ARXOLI	SCHEMBL24319484	(3R)-N-[3-[5-[4-[(2S)-2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]oxymethyl]azetidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide; SCHEMBL30253645	O=C1CCC(N2CC3=CC(OC[C@@H]4CCN4C4=CC=C(C5=CC6=C(N=C5)NC=C6C(=O)C5=C(F)C=CC(NS(=O)(=O)N6CC[C@@H](F)C6)=C5F)C=C4)=CC=C3C2=O)C(=O)N1	C41H36F3N7O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-6MS986	SCHEMBL24319485	(3R)-N-[3-[5-[2-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]pyrimidin-5-yl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide; SCHEMBL30254180	O=C1CCC(N2CC3=CC(N4CCC(CN5CCN(C6=NC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=N6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C45H46F3N11O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-XIQVJI	WO2022047145A1_19	.	O=C1CCC(N2CC3=C(C=CC(N4CCC(F)(CN5CC6(C5)CN(C5=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)C8CC[C@@H](F)C8)=C7F)C=C5)C6)CC4)=C3)C2=O)C(=O)N1	C49H48F4N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-5BWSDF	SCHEMBL30254103	(3R)-N-[3-[5-[4-[4-[[(3R)-6-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-5-yl]-3-methyl-2,6-diazaspiro[3.3]heptan-2-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	COC1=CC(N2CC3(C2)CN(CC2CCN(C4=CC=C(C5=CC6=C(N=C5)NC=C6C(=O)C5=C(F)C=CC(NS(=O)(=O)N6CC[C@@H](F)C6)=C5F)C=C4)CC2)[C@@H]3C)=CC2=C1C(=O)N(C1CCC(=O)NC1=O)C2	C50H52F3N9O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-OS66S1	SCHEMBL30253858	(3R)-N-[3-[5-[4-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-5-yl]-2,6-diazaspiro[3.3]heptan-6-yl]ethyl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	COC1=C2C(=O)N(C3CCC(=O)NC3=O)CC2=CC(N2CC3(CN(CCC4=CC=C(C5=CC6=C(N=C5)NC=C6C(=O)C5=C(F)C=CC(NS(=O)(=O)N6CC[C@@H](F)C6)=C5F)C=C4)C3)C2)=C1	C45H43F3N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-NQW3A6	SCHEMBL30254144	(3R)-N-[3-[5-[4-[6-[3-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-5-yl]propyl]-2,6-diazaspiro[3.3]heptan-2-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	COC1=CC(CCCN2CC3(C2)CN(C2=CC=C(C4=CC5=C(N=C4)NC=C5C(=O)C4=C(F)C=CC(NS(=O)(=O)N5CC[C@@H](F)C5)=C4F)C=C2)C3)=CC2=C1C(=O)N(C1CCC(=O)NC1=O)C2	C46H45F3N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-RYDMXD	SCHEMBL30253807	(3R)-N-[3-[5-[4-[[(2S)-1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]azetidin-2-yl]methoxy]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(N4CC[C@H]4COC4=CC=C(C5=CC6=C(N=C5)NC=C6C(=O)C5=C(F)C=CC(NS(=O)(=O)N6CC[C@@H](F)C6)=C5F)C=C4)=CC=C3C2=O)C(=O)N1	C41H36F3N7O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-ENF6KY	SCHEMBL30254001	(3R)-N-[3-[5-[6-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridin-3-yl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(C4CCN(CC5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=N6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C47H48F3N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-RM5CP7	SCHEMBL24021882	(3R)-N-[3-[5-[6-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-3-yl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide; SCHEMBL30253929	O=C1CCC(N2CC3=CC(N4CCC(CN5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=N6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C46H47F3N10O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-A4F04V	SCHEMBL30253924	(3R)-N-[3-[5-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-2,6-diazaspiro[3.3]heptan-6-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(N4CC5(CN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6)C5)C4)=CC=C3C2=O)C(=O)N1	C42H37F3N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-QXQQIK	SCHEMBL24319445	4-[4-[2-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]ethyl]piperazin-1-yl]-N-[(3S)-2,6-dioxopiperidin-3-yl]-2-fluorobenzamide; SCHEMBL30254276	O=C1CC[C@H](NC(=O)C2=CC=C(N3CCN(CCC4=CC=C(C5=CC6=C(N=C5)NC=C6C(=O)C5=C(F)C=CC(NS(=O)(=O)N6CC[C@@H](F)C6)=C5F)C=C4)CC3)C=C2F)C(=O)N1	C42H40F4N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-N3MN30	WO2022047145A1_28	.	O=C1CC[C@@H](NC(=O)C2=CC=C(N3CCN(CCC4=CC=C(C5=CC6=C(N=C5)NC=C6C(=O)C5=C(F)C=CC(NS(=O)(=O)N6CC[C@@H](F)C6)C5F)C=C4)CC3)C=C2F)C(=O)N1	C42H42F4N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-29UVEN	SCHEMBL30253573	4-[4-[[2-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]-2,6-diazaspiro[3.3]heptan-6-yl]methyl]piperidin-1-yl]-N-[(3S)-2,6-dioxopiperidin-3-yl]-2-fluorobenzamide	O=C1CC[C@H](NC(=O)C2=CC=C(N3CCC(CN4CC5(C4)CN(C4=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C4)C5)CC3)C=C2F)C(=O)N1	C47H47F4N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-FITZE7	SCHEMBL30254360	4-[4-[[2-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]-2,6-diazaspiro[3.3]heptan-6-yl]methyl]piperidin-1-yl]-N-[(3R)-2,6-dioxopiperidin-3-yl]-2-fluorobenzamide	O=C1CC[C@@H](NC(=O)C2=CC=C(N3CCC(CN4CC5(C4)CN(C4=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C4)C5)CC3)C=C2F)C(=O)N1	C47H47F4N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-DHWJUT	SCHEMBL30254347	4-[6-[[1-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]piperidin-4-yl]methyl]-2,6-diazaspiro[3.3]heptan-2-yl]-N-[(3S)-2,6-dioxopiperidin-3-yl]-2-fluorobenzamide	O=C1CC[C@H](NC(=O)C2=CC=C(N3CC4(CN(CC5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6)CC5)C4)C3)C=C2F)C(=O)N1	C47H47F4N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-HHNFMG	SCHEMBL30253884	(3R)-N-[3-[5-[4-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-2-hydroxyethyl]piperazin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=C(C=CC(C(O)CN4CCN(C5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)CC4)=C3)C2=O)C(=O)N1	C43H41F3N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-WNINYV	SCHEMBL30253700	4-[1-[[1-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]piperidin-4-yl]methyl]piperidin-4-yl]-N-[(3S)-2,6-dioxopiperidin-3-yl]-2-fluorobenzamide	O=C1CC[C@H](NC(=O)C2=CC=C(C3CCN(CC4CCN(C5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)CC4)CC3)C=C2F)C(=O)N1	C47H48F4N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-MKICTL	WO2022047145A1_34	.	O=C1CC[C@H](N2CC3CC(N4CCC(OC5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C47H49F3N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-99OHQG	SCHEMBL30254133	(3R)-N-[3-[5-[4-[4-[1-[2-[(3R)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]oxypiperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CC[C@@H](N2CC3=CC(N4CCC(OC5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C47H47F3N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-OXU8VU	SCHEMBL24319561	(3R)-N-[3-[5-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]-3-fluorophenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide; SCHEMBL29482878	O=C1CCC(N2CC3=CC(C4CCN(CC5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6F)CC5)CC4)=CC=C3C2=O)C(=O)N1	C48H48F4N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-SE63FV	SCHEMBL30253728	4-[6-[[1-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]piperidin-4-yl]methyl]-2,6-diazaspiro[3.3]heptan-2-yl]-N-[(3R)-2,6-dioxopiperidin-3-yl]-2-fluorobenzamide	O=C1CC[C@@H](NC(=O)C2=CC=C(N3CC4(CN(CC5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6)CC5)C4)C3)C=C2F)C(=O)N1	C47H47F4N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-NUY345	SCHEMBL30253961	(3R)-N-[3-[5-[4-[6-[(E)-3-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]prop-2-enyl]-2,6-diazaspiro[3.3]heptan-2-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CC[C@H](N2CC3=CC(/C=C/CN4CC5(C4)CN(C4=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C4)C5)=CC=C3C2=O)C(=O)N1	C45H41F3N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-5PD3EI	SCHEMBL30254240	(3R)-N-[3-[5-[4-[6-[(E)-3-[2-[(3R)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]prop-2-enyl]-2,6-diazaspiro[3.3]heptan-2-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CC[C@@H](N2CC3=CC(/C=C/CN4CC5(C4)CN(C4=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C4)C5)=CC=C3C2=O)C(=O)N1	C45H41F3N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-YGT4YS	SCHEMBL30253811	(3R)-N-[3-[5-[4-[4-[[1-[2-[(3S)-2,6-dioxopiperidin-3-yl]-6-fluoro-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CC[C@H](N2CC3=CC(N4CCC(CN5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6)CC5)CC4)=C(F)C=C3C2=O)C(=O)N1	C47H47F4N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-QM594M	SCHEMBL30254023	(3R)-N-[3-[5-[4-[4-[[1-[2-[(3R)-2,6-dioxopiperidin-3-yl]-6-fluoro-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CC[C@@H](N2CC3=CC(N4CCC(CN5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6)CC5)CC4)=C(F)C=C3C2=O)C(=O)N1	C47H47F4N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-ZC3FGK	SCHEMBL30253928	(3R)-N-[3-[5-[4-[3-[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-2,6-diazaspiro[3.3]heptan-6-yl]prop-1-ynyl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(N4CC5(CN(CC#CC6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6)C5)C4)=CC=C3C2=O)C(=O)N1	C45H39F3N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-AQXLC3	SCHEMBL30253691	(3R)-N-[3-[5-[4-[6-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]oxy]-2-azaspiro[3.3]heptan-2-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(OC4CC5(C4)CN(C4=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C4)C5)=CC=C3C2=O)C(=O)N1	C43H38F3N7O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-X0XT4E	SCHEMBL30253827	(3R)-N-[3-[5-[4-[2-[4-[2-[[2-[(3S)-2,6-dioxopiperidin-3-yl]-7-methoxy-1-oxo-3H-isoindol-5-yl]oxy]ethyl]piperazin-1-yl]ethoxy]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	COC1=CC(OCCN2CCN(CCOC3=CC=C(C4=CC5=C(N=C4)NC=C5C(=O)C4=C(F)C=CC(NS(=O)(=O)N5CC[C@@H](F)C5)=C4F)C=C3)CC2)=CC2=C1C(=O)N([C@H]1CCC(=O)NC1=O)C2	C46H47F3N8O9S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-WRR0LP	SCHEMBL30253863	(3R)-N-[3-[5-[4-[2-[4-[2-[[2-[(3R)-2,6-dioxopiperidin-3-yl]-7-methoxy-1-oxo-3H-isoindol-5-yl]oxy]ethyl]piperazin-1-yl]ethoxy]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	COC1=CC(OCCN2CCN(CCOC3=CC=C(C4=CC5=C(N=C4)NC=C5C(=O)C4=C(F)C=CC(NS(=O)(=O)N5CC[C@@H](F)C5)=C4F)C=C3)CC2)=CC2=C1C(=O)N([C@@H]1CCC(=O)NC1=O)C2	C46H47F3N8O9S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-P60KCI	SCHEMBL30254148	(3R)-N-[3-[5-[2-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyrimidin-5-yl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(C4CCN(CC5CCN(C6=NC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=N6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C46H47F3N10O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-8I4355	SCHEMBL30254024	(3R)-N-[3-[5-[1-[[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-2-azaspiro[3.3]heptan-6-yl]methyl]-3,4-dihydro-2H-quinolin-6-yl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(N4CC5(CC(CN6CCCC7=C6C=CC(C6=CC8=C(N=C6)NC=C8C(=O)C6=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C6F)=C7)C5)C4)=CC=C3C2=O)C(=O)N1	C47H45F3N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-LJOVJ9	SCHEMBL30253886	4-[1-[[1-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]piperidin-4-yl]methyl]piperidin-4-yl]-N-[(3R)-2,6-dioxopiperidin-3-yl]-2-fluorobenzamide	O=C1CC[C@@H](NC(=O)C2=CC=C(C3CCN(CC4CCN(C5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)CC4)CC3)C=C2F)C(=O)N1	C47H48F4N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-RJCZ8X	SCHEMBL24319926	(3R)-N-[3-[5-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]propyl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide; SCHEMBL30254253	O=C1CCC(N2CC3=C(C=CC(C4CCN(CCCC5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)CC4)=C3)C2=O)C(=O)N1	C45H44F3N7O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-IEK561	SCHEMBL30254034	(3R)-N-[3-[5-[4-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-2,6-diazaspiro[3.3]heptan-6-yl]ethoxy]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(N4CC5(CN(CCOC6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6)C5)C4)=CC=C3C2=O)C(=O)N1	C44H41F3N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-CF5XM0	SCHEMBL30253806	(3R)-N-[3-[5-[4-[(3aS,6aR)-2-[[1-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]-3a-methyl-3,4,6,6a-tetrahydro-1H-pyrrolo[3,4-c]pyrrol-5-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	[H][C@]12CN(CC3CCN(C4=CC=C5C(=O)N([C@H]6CCC(=O)NC6=O)CC5=C4)CC3)C[C@@]1(C)CN(C1=CC=C(C3=CC4=C(N=C3)NC=C4C(=O)C3=C(F)C=CC(NS(=O)(=O)N4CC[C@@H](F)C4)=C3F)C=C1)C2	C50H52F3N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-14WLMV	SCHEMBL30253594	(3R)-N-[3-[5-[4-[(3aS,6aR)-2-[[1-[2-[(3R)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]-3a-methyl-3,4,6,6a-tetrahydro-1H-pyrrolo[3,4-c]pyrrol-5-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	[H][C@]12CN(CC3CCN(C4=CC=C5C(=O)N([C@@H]6CCC(=O)NC6=O)CC5=C4)CC3)C[C@@]1(C)CN(C1=CC=C(C3=CC4=C(N=C3)NC=C4C(=O)C3=C(F)C=CC(NS(=O)(=O)N4CC[C@@H](F)C4)=C3F)C=C1)C2	C50H52F3N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-3V4NV2	SCHEMBL30254371	(3R)-N-[3-[5-[4-[(3S,5R)-4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]azetidin-3-yl]methyl]-3,5-dimethylpiperazin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	C[C@@H]1CN(C2=CC=C(C3=CC4=C(N=C3)NC=C4C(=O)C3=C(F)C=CC(NS(=O)(=O)N4CC[C@@H](F)C4)=C3F)C=C2)C[C@H](C)N1CC1CN(C2=CC=C3C(=O)N(C4CCC(=O)NC4=O)CC3=C2)C1	C47H48F3N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-U8Y89C	SCHEMBL30253935	(3R)-N-[3-[5-[4-[6-[[4-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]-2-azaspiro[3.3]heptan-2-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	COC1=CC(C2CCN(CC3CC4(C3)CN(C3=CC=C(C5=CC6=C(N=C5)NC=C6C(=O)C5=C(F)C=CC(NS(=O)(=O)N6CC[C@@H](F)C6)=C5F)C=C3)C4)CC2)=CC2=C1C(=O)N(C1CCC(=O)NC1=O)C2	C50H51F3N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-LVDNZT	SCHEMBL30253992	(3R)-N-[3-[5-[4-[6-[[1-[2-[(3S)-2,6-dioxopiperidin-3-yl]-6-fluoro-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]-2,6-diazaspiro[3.3]heptan-2-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CC[C@H](N2CC3=CC(N4CCC(CN5CC6(C5)CN(C5=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C5)C6)CC4)=C(F)C=C3C2=O)C(=O)N1	C48H47F4N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-PN30G6	SCHEMBL30254303	(3R)-N-[3-[5-[4-[6-[[1-[2-[(3R)-2,6-dioxopiperidin-3-yl]-6-fluoro-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]-2,6-diazaspiro[3.3]heptan-2-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CC[C@@H](N2CC3=CC(N4CCC(CN5CC6(C5)CN(C5=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C5)C6)CC4)=C(F)C=C3C2=O)C(=O)N1	C48H47F4N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-3R5OEO	SCHEMBL30254008	(3R)-N-[3-[5-[4-[4-[[(3aS,6aR)-5-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-2-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	[H][C@@]12CN(CC3CCN(C4=CC=C(C5=CC6=C(N=C5)NC=C6C(=O)C5=C(F)C=CC(NS(=O)(=O)N6CC[C@@H](F)C6)=C5F)C=C4)CC3)C[C@]1([H])CN(C1=CC=C3C(=O)N([C@H]4CCC(=O)NC4=O)CC3=C1)C2	C49H50F3N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-BPZ4L5	SCHEMBL30253999	(3R)-N-[3-[5-[4-[4-[[(3aS,6aR)-5-[2-[(3R)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-2-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	[H][C@@]12CN(CC3CCN(C4=CC=C(C5=CC6=C(N=C5)NC=C6C(=O)C5=C(F)C=CC(NS(=O)(=O)N6CC[C@@H](F)C6)=C5F)C=C4)CC3)C[C@]1([H])CN(C1=CC=C3C(=O)N([C@@H]4CCC(=O)NC4=O)CC3=C1)C2	C49H50F3N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-3IQVPH	SCHEMBL30254157	(3R)-N-[3-[5-[4-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-5-yl]-2-azaspiro[3.3]heptan-6-yl]methyl]piperazin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	COC1=C2C(=O)N(C3CCC(=O)NC3=O)CC2=CC(N2CC3(CC(CN4CCN(C5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)CC4)C3)C2)=C1	C49H50F3N9O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-2R3SQJ	SCHEMBL30253673	(3R)-N-[3-[5-[4-[4-[2-[6-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-2,6-diazaspiro[3.3]heptan-2-yl]propan-2-yl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	CC(C)(C1CCN(C2=CC=C(C3=CC4=C(N=C3)NC=C4C(=O)C3=C(F)C=CC(NS(=O)(=O)N4CC[C@@H](F)C4)=C3F)C=C2)CC1)N1CC2(CN(C3=CC=C4C(=O)N(C5CCC(=O)NC5=O)CC4=C3)C2)C1	C50H52F3N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-MOPP40	SCHEMBL30253932	(3R)-N-[3-[5-[4-[6-[3-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-3-hydroxypropyl]-2,6-diazaspiro[3.3]heptan-2-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(C(O)CCN4CC5(C4)CN(C4=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C4)C5)=CC=C3C2=O)C(=O)N1	C45H43F3N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-ZXMCDE	SCHEMBL30253951	(3R)-N-[3-[5-[4-[6-[4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]butyl]-2,6-diazaspiro[3.3]heptan-2-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CC[C@H](N2CC3=CC(CCCCN4CC5(C4)CN(C4=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C4)C5)=CC=C3C2=O)C(=O)N1	C46H45F3N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-KECEYQ	SCHEMBL30254112	(3R)-N-[3-[5-[4-[6-[4-[2-[(3R)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]butyl]-2,6-diazaspiro[3.3]heptan-2-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CC[C@@H](N2CC3=CC(CCCCN4CC5(C4)CN(C4=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C4)C5)=CC=C3C2=O)C(=O)N1	C46H45F3N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-RXAUAF	SCHEMBL30253893	(3R)-N-[3-[5-[4-[4-[5-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]pentyl]piperazin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=C(C=CC(CCCCCN4CCN(C5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)CC4)=C3)C2=O)C(=O)N1	C46H47F3N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-KCEB21	SCHEMBL24320649	(3R)-N-[3-[5-[4-[1-[5-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]pentyl]piperidin-4-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide; SCHEMBL30254410	O=C1CCC(N2CC3=CC(CCCCCN4CCC(C5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C47H48F3N7O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-Z99TA0	SCHEMBL24320650	(3R)-N-[3-[5-[4-[5-[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]-2,5-diazaspiro[3.4]octan-2-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide; SCHEMBL30253609	O=C1CCC(N2CC3=CC(N4CCC(N5CCCC56CN(C5=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C5)C6)CC4)=CC=C3C2=O)C(=O)N1	C48H48F3N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-CX3LZL	SCHEMBL24320648	(3R)-N-[3-[5-[4-[1-[(3R)-3-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]-3-hydroxypropyl]piperidin-4-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide; SCHEMBL29482998	O=C1CC[C@H](N2CC3=CC([C@H](O)CCN4CCC(C5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C45H44F3N7O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-YP5EDP	SCHEMBL24319860	(3R)-N-[3-[5-[4-[1-[(3R)-3-[2-[(3R)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]-3-hydroxypropyl]piperidin-4-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide; SCHEMBL29482913	O=C1CC[C@@H](N2CC3=CC([C@H](O)CCN4CCC(C5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C45H44F3N7O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-PMAXE4	SCHEMBL30253684	(3R)-N-[3-[5-[4-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]ethoxy]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(C4CCN(CCOC5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C44H42F3N7O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-TPGRBZ	SCHEMBL30254231	(3R)-N-[3-[5-[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-5-yl]azetidin-3-yl]methyl]piperazin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	COC1=CC(N2CC(CN3CCN(C4=CC=C(C5=CC6=C(N=C5)NC=C6C(=O)C5=C(F)C=CC(NS(=O)(=O)N6CC[C@@H](F)C6)=C5F)C=C4)CC3)C2)=CC2=C1C(=O)N(C1CCC(=O)NC1=O)C2	C46H46F3N9O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-V72TR8	SCHEMBL30254219	(3R)-N-[3-[5-[4-[1-[(3S)-3-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]-3-hydroxypropyl]piperidin-4-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CC[C@H](N2CC3=CC([C@@H](O)CCN4CCC(C5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C45H44F3N7O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-BLFOVS	SCHEMBL30253984	(3R)-N-[3-[5-[4-[1-[(3S)-3-[2-[(3R)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]-3-hydroxypropyl]piperidin-4-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CC[C@@H](N2CC3=CC([C@@H](O)CCN4CCC(C5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C45H44F3N7O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-H1D2MJ	SCHEMBL30254092	(3R)-N-[3-[5-[4-[4-[(2R)-3-[2-[(3R)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]-2-hydroxypropyl]piperazin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CC[C@@H](N2CC3=C(C=CC(C[C@@H](O)CN4CCN(C5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)CC4)=C3)C2=O)C(=O)N1	C44H43F3N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-E5BTQA	SCHEMBL24319213	(3R)-N-[3-[5-[4-[4-[(2S)-3-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]-2-hydroxypropyl]piperazin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide; SCHEMBL29482830	O=C1CC[C@H](N2CC3=C(C=CC(C[C@H](O)CN4CCN(C5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)CC4)=C3)C2=O)C(=O)N1	C44H43F3N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-7TF297	SCHEMBL30253921	(3R)-N-[3-[5-[4-[4-[(2S)-3-[2-[(3R)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]-2-hydroxypropyl]piperazin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CC[C@@H](N2CC3=C(C=CC(C[C@H](O)CN4CCN(C5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)CC4)=C3)C2=O)C(=O)N1	C44H43F3N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-LBHJC7	SCHEMBL30253757	(3R)-N-[3-[5-[4-[(3aR,6aS)-2-[[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]methyl]-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-5-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	[H][C@@]12CN(CC3=CC=C4C(=O)N([C@H]5CCC(=O)NC5=O)CC4=C3)C[C@]1([H])CN(C1=CC=C(C3=CC4=C(N=C3)NC=C4C(=O)C3=C(F)C=CC(NS(=O)(=O)N4CC[C@@H](F)C4)=C3F)C=C1)C2	C44H41F3N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-MHGEZ3	SCHEMBL30253849	(3R)-N-[3-[5-[4-[(3aR,6aS)-2-[[2-[(3R)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]methyl]-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-5-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	[H][C@@]12CN(CC3=CC=C4C(=O)N([C@@H]5CCC(=O)NC5=O)CC4=C3)C[C@]1([H])CN(C1=CC=C(C3=CC4=C(N=C3)NC=C4C(=O)C3=C(F)C=CC(NS(=O)(=O)N4CC[C@@H](F)C4)=C3F)C=C1)C2	C44H41F3N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-6KVH0I	SCHEMBL30254085	(3R)-N-[3-[5-[4-[(3R)-4-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]methyl]-3-(hydroxymethyl)piperazin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(CN4CCN(C5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)C[C@@H]4CO)=CC=C3C2=O)C(=O)N1	C43H41F3N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-FRUSA7	SCHEMBL24319527	(3R)-N-[3-[5-[4-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-5-yl]azetidin-3-yl]piperazin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide; SCHEMBL29482822	COC1=C2C(=O)N(C3CCC(=O)NC3=O)CC2=CC(N2CC(N3CCN(C4=CC=C(C5=CC6=C(N=C5)NC=C6C(=O)C5=C(F)C=CC(NS(=O)(=O)N6CC[C@@H](F)C6)=C5F)C=C4)CC3)C2)=C1	C45H44F3N9O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-I38YON	SCHEMBL30253789	(3R)-N-[3-[5-[4-[6-[3-[[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]oxy]propyl]-2,6-diazaspiro[3.3]heptan-2-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CC[C@H](N2CC3=CC(OCCCN4CC5(C4)CN(C4=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C4)C5)=CC=C3C2=O)C(=O)N1	C45H43F3N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-I5ERQP	SCHEMBL30254058	(3R)-N-[3-[5-[4-[6-[3-[[2-[(3R)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]oxy]propyl]-2,6-diazaspiro[3.3]heptan-2-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CC[C@@H](N2CC3=CC(OCCCN4CC5(C4)CN(C4=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C4)C5)=CC=C3C2=O)C(=O)N1	C45H43F3N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-J0ZKN3	SCHEMBL30254152	(3R)-N-[3-[5-[4-[4-[(2R)-3-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]-2-hydroxypropyl]piperazin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CC[C@H](N2CC3=C(C=CC(C[C@@H](O)CN4CCN(C5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)CC4)=C3)C2=O)C(=O)N1	C44H43F3N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-RAAY7U	SCHEMBL30253765	(3R)-N-[3-[5-[4-[4-[[3-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]azetidin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CC[C@H](N2CC3=C(C=CC(C4CN(CC5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6)CC5)C4)=C3)C2=O)C(=O)N1	C46H45F3N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-H93WDE	SCHEMBL30254261	(3R)-N-[3-[5-[4-[4-[[3-[2-[(3R)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]azetidin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CC[C@@H](N2CC3=C(C=CC(C4CN(CC5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6)CC5)C4)=C3)C2=O)C(=O)N1	C46H45F3N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-XEUIOF	SCHEMBL30253891	(3R)-N-[3-[5-[4-[(3aS,6aR)-2-[[1-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]azetidin-3-yl]methyl]-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-5-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	[H][C@@]12CN(CC3CN(C4=CC=C5C(=O)N([C@H]6CCC(=O)NC6=O)CC5=C4)C3)C[C@]1([H])CN(C1=CC=C(C3=CC4=C(N=C3)NC=C4C(=O)C3=C(F)C=CC(NS(=O)(=O)N4CC[C@@H](F)C4)=C3F)C=C1)C2	C47H46F3N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-4XKAWN	SCHEMBL30253653	(3R)-N-[3-[5-[4-[(3aS,6aR)-2-[[1-[2-[(3R)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]azetidin-3-yl]methyl]-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-5-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	[H][C@@]12CN(CC3CN(C4=CC=C5C(=O)N([C@@H]6CCC(=O)NC6=O)CC5=C4)C3)C[C@]1([H])CN(C1=CC=C(C3=CC4=C(N=C3)NC=C4C(=O)C3=C(F)C=CC(NS(=O)(=O)N4CC[C@@H](F)C4)=C3F)C=C1)C2	C47H46F3N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-CMBO9F	SCHEMBL30254255	(3R)-N-[3-[5-[4-[4-[[4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]-3-fluorophenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CC[C@H](N2CC3=CC(C4CCN(CC5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6F)CC5)CC4)=CC=C3C2=O)C(=O)N1	C48H48F4N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-INF49E	SCHEMBL30253579	(3R)-N-[3-[5-[4-[4-[[4-[2-[(3R)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]-3-fluorophenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CC[C@@H](N2CC3=CC(C4CCN(CC5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6F)CC5)CC4)=CC=C3C2=O)C(=O)N1	C48H48F4N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-XC9YRN	SCHEMBL30253913	(3R)-N-[3-[5-[4-[6-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]oxy]ethyl]-2,6-diazaspiro[3.3]heptan-2-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(OCCN4CC5(C4)CN(C4=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C4)C5)=CC=C3C2=O)C(=O)N1	C44H41F3N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-WCJPFQ	SCHEMBL24319856	(3R)-N-[3-[5-[4-[(2R)-3-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]-2-hydroxypropyl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide; SCHEMBL29482841	O=C1CCC(N2CC3=CC(N4CCN(C[C@H](O)CC5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C44H43F3N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-GIMYCF	SCHEMBL30253754	(3R)-N-[3-[5-[2-[3-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]azetidin-1-yl]pyrimidin-5-yl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(N4CCN(CC5CN(C6=NC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=N6)C5)CC4)=CC=C3C2=O)C(=O)N1	C43H42F3N11O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-08XGVB	SCHEMBL30253723	(3R)-N-[3-[5-[6-[2-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]-2,7-diazaspiro[3.4]octan-7-yl]pyridin-3-yl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(N4CCC(CN5CC6(CCN(C7=CC=C(C8=CC9=C(N=C8)NC=C9C(=O)C8=C(F)C=CC(NS(=O)(=O)N9CC[C@@H](F)C9)=C8F)C=N7)C6)C5)CC4)=CC=C3C2=O)C(=O)N1	C48H49F3N10O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-Q0J1NM	CHEMBL5180482	(3R)-N-[3-[5-[2-[2-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]-2,7-diazaspiro[3.4]octan-7-yl]pyrimidin-5-yl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(N4CCC(CN5CC6(CCN(C7=NC=C(C8=CC9=C(N=C8)NC=C9C(=O)C8=C(F)C=CC(NS(=O)(=O)N9CC[C@@H](F)C9)=C8F)C=N7)C6)C5)CC4)=CC=C3C2=O)C(=O)N1	C47H48F3N11O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-QMBA78	SCHEMBL30253739	(3R)-N-[3-[5-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]-3,5-difluorophenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(C4CCN(CC5CCN(C6=C(F)C=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6F)CC5)CC4)=CC=C3C2=O)C(=O)N1	C48H47F5N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-9HQUUA	SCHEMBL30253890	(3R)-N-[3-[5-[6-[2-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]-2,8-diazaspiro[4.5]decan-8-yl]pyridin-3-yl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(N4CCC(CN5CCC6(CCN(C7=CC=C(C8=CC9=C(N=C8)NC=C9C(=O)C8=C(F)C=CC(NS(=O)(=O)N9CC[C@@H](F)C9)=C8F)C=N7)CC6)C5)CC4)=CC=C3C2=O)C(=O)N1	C50H53F3N10O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-8EQ1S6	SCHEMBL30254349	(3R)-N-[3-[5-[2-[2-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]-2,8-diazaspiro[4.5]decan-8-yl]pyrimidin-5-yl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(N4CCC(CN5CCC6(CCN(C7=NC=C(C8=CC9=C(N=C8)NC=C9C(=O)C8=C(F)C=CC(NS(=O)(=O)N9CC[C@@H](F)C9)=C8F)C=N7)CC6)C5)CC4)=CC=C3C2=O)C(=O)N1	C49H52F3N11O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-ZVXV3W	SCHEMBL30253668	(3R)-N-[3-[5-[4-[4-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]propan-2-yl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	CC(C)(C1CCN(C2=CC=C(C3=CC4=C(N=C3)NC=C4C(=O)C3=C(F)C=CC(NS(=O)(=O)N4CC[C@@H](F)C4)=C3F)C=C2)CC1)N1CCN(C2=CC=C3C(=O)N(C4CCC(=O)NC4=O)CC3=C2)CC1	C49H52F3N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-AS3P5T	SCHEMBL30253894	(3R)-N-[3-[5-[4-[(2S)-3-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]-2-hydroxypropyl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(N4CCN(C[C@@H](O)CC5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C44H43F3N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-G7CMNA	SCHEMBL30253914	(3R)-N-[3-[5-[4-[6-[[3-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]azetidin-1-yl]methyl]-2-azaspiro[3.3]heptan-2-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CC[C@H](N2CC3=C(C=CC(C4CN(CC5CC6(C5)CN(C5=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C5)C6)C4)=C3)C2=O)C(=O)N1	C47H45F3N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-JWJQZA	SCHEMBL30254123	(3R)-N-[3-[5-[4-[6-[[3-[2-[(3R)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]azetidin-1-yl]methyl]-2-azaspiro[3.3]heptan-2-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CC[C@@H](N2CC3=C(C=CC(C4CN(CC5CC6(C5)CN(C5=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C5)C6)C4)=C3)C2=O)C(=O)N1	C47H45F3N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-0W4SWH	SCHEMBL30253710	(3R)-N-[3-[5-[6-[3-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]azetidin-1-yl]pyridin-3-yl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(N4CCN(CC5CN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=N6)C5)CC4)=CC=C3C2=O)C(=O)N1	C44H43F3N10O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-SL88HU	SCHEMBL30253689	(3R)-N-[3-[5-[4-[4-[[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-5-yl]methyl]piperazin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	COC1=C2C(=O)N(C3CCC(=O)NC3=O)CC2=CC(CN2CCN(C3=CC=C(C4=CC5=C(N=C4)NC=C5C(=O)C4=C(F)C=CC(NS(=O)(=O)N5CC[C@@H](F)C5)=C4F)C=C3)CC2)=C1	C43H41F3N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-LCCPT3	SCHEMBL30253972	(3R)-N-[3-[5-[6-[6-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]-2-azaspiro[3.3]heptan-2-yl]pyridin-3-yl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(C4CCN(CC5CC6(C5)CN(C5=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=N5)C6)CC4)=CC=C3C2=O)C(=O)N1	C48H48F3N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-C34QUA	SCHEMBL30253801	(3R)-N-[3-[5-[4-[2-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]-2,8-diazaspiro[4.5]decan-8-yl]-3-fluorophenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(N4CCC(CN5CCC6(CCN(C7=CC=C(C8=CC9=C(N=C8)NC=C9C(=O)C8=C(F)C=CC(NS(=O)(=O)N9CC[C@@H](F)C9)=C8F)C=C7F)CC6)C5)CC4)=CC=C3C2=O)C(=O)N1	C51H53F4N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-922BTG	WO2022047145A1_105	.	O=C1CC[C@H](N2CC3=CC([C@H](O)CCN4CC5(C4)CN(C4=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)C6F)C=C4)C5)=CC=C3C2=O)C(=O)N1	C45H45F3N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-4ZWBCU	WO2022047145A1_106	.	O=C1CC[C@H](N2CC3=CC([C@@H](O)CCN4CC5(C4)CN(C4=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)C6F)C=C4)C5)=CC=C3C2=O)C(=O)N1	C45H45F3N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-H2IDVO	WO2022047145A1_107	(3R)-N-[3-[5-[4-[1-[(2R)-3-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]-2-hydroxypropyl]piperidin-4-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CC[C@H](N2CC3=C(C=CC(C[C@@H](O)CN4CCC(C5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)CC4)=C3)C2=O)C(=O)N1	C45H44F3N7O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-NDFYBJ	SCHEMBL30254039	(3R)-N-[3-[5-[4-[1-[(2R)-3-[2-[(3R)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]-2-hydroxypropyl]piperidin-4-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CC[C@@H](N2CC3=C(C=CC(C[C@@H](O)CN4CCC(C5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)CC4)=C3)C2=O)C(=O)N1	C45H44F3N7O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-V7RFSC	SCHEMBL30253776	(3R)-N-[3-[5-[4-[1-[(2S)-3-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]-2-hydroxypropyl]piperidin-4-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CC[C@H](N2CC3=C(C=CC(C[C@H](O)CN4CCC(C5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)CC4)=C3)C2=O)C(=O)N1	C45H44F3N7O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-QNQBB0	SCHEMBL30254357	(3R)-N-[3-[5-[4-[(2R)-3-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]-2-hydroxypropyl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(C4CCN(C[C@H](O)CC5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C45H44F3N7O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-RB8XU5	SCHEMBL30253816	(3R)-N-[3-[5-[4-[2-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]-2,7-diazaspiro[3.4]octan-7-yl]-3-fluorophenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(N4CCC(CN5CC6(CCN(C7=CC=C(C8=CC9=C(N=C8)NC=C9C(=O)C8=C(F)C=CC(NS(=O)(=O)N9CC[C@@H](F)C9)=C8F)C=C7F)C6)C5)CC4)=CC=C3C2=O)C(=O)N1	C49H49F4N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-AXWXBG	SCHEMBL30253735	(3R)-N-[3-[5-[4-[(3S)-4-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]methyl]-3-(hydroxymethyl)piperazin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(CN4CCN(C5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)C[C@H]4CO)=CC=C3C2=O)C(=O)N1	C43H41F3N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-OO74BC	SCHEMBL30253618	(3R)-N-[3-[5-[4-[4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]oxy]butyl]piperazin-1-yl]-3-fluorophenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(OCCCCN4CCN(C5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5F)CC4)=CC=C3C2=O)C(=O)N1	C45H44F4N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-UN7HMJ	SCHEMBL30254018	(3R)-N-[3-[5-[4-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-2,6-diazaspiro[3.3]heptan-6-yl]ethoxy]-3-fluorophenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(N4CC5(CN(CCOC6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6F)C5)C4)=CC=C3C2=O)C(=O)N1	C44H40F4N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-CB6X3S	SCHEMBL24319413	(3R)-N-[3-[5-[4-[4-[6-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]pyrimidin-4-yl]piperazin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide; SCHEMBL29482857	O=C1CCC(N2CC3=CC(N4CCN(C5=CC(N6CCN(C7=CC=C(C8=CC9=C(N=C8)NC=C9C(=O)C8=C(F)C=CC(NS(=O)(=O)N9CC[C@@H](F)C9)=C8F)C=C7)CC6)=NC=N5)CC4)=CC=C3C2=O)C(=O)N1	C49H47F3N12O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-P1BYVK	SCHEMBL30253657	(3R)-N-[3-[5-[4-[1-[(2S)-3-[2-[(3R)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]-2-hydroxypropyl]piperidin-4-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CC[C@@H](N2CC3=C(C=CC(C[C@H](O)CN4CCC(C5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)CC4)=C3)C2=O)C(=O)N1	C45H44F3N7O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-ULXWNM	SCHEMBL30254102	(3R)-N-[3-[5-[2-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-2,6-diazaspiro[3.3]heptan-6-yl]ethoxy]pyrimidin-5-yl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(N4CC5(CN(CCOC6=NC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=N6)C5)C4)=CC=C3C2=O)C(=O)N1	C42H39F3N10O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-FDLUA6	SCHEMBL30253854	(3R)-N-[3-[5-[4-[(2S)-3-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]-2-hydroxypropyl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(C4CCN(C[C@@H](O)CC5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C45H44F3N7O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-SWZ44S	WO2022047145A1_119	.	O=C1CCC(N2CC3=CC(C4CCN(CC5(O)CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N=N1	C48H48F3N9O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-HZLIW6	SCHEMBL30254192	(3R)-N-[3-[5-[6-[4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]oxy]butyl]piperazin-1-yl]pyridin-3-yl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(OCCCCN4CCN(C5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=N5)CC4)=CC=C3C2=O)C(=O)N1	C44H44F3N9O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-SJLRLK	SCHEMBL30253706	(3R)-N-[3-[5-[2-[4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]oxy]butyl]piperazin-1-yl]pyrimidin-5-yl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(OCCCCN4CCN(C5=NC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=N5)CC4)=CC=C3C2=O)C(=O)N1	C43H43F3N10O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-QY73WV	SCHEMBL30253956	(3R)-N-[3-[5-[4-[6-[(2S)-3-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]oxy]-2-hydroxypropyl]-2,6-diazaspiro[3.3]heptan-2-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(OC[C@@H](O)CN4CC5(C4)CN(C4=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C4)C5)=CC=C3C2=O)C(=O)N1	C45H43F3N8O8S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-J61CIB	SCHEMBL29482946	(3R)-N-[3-[5-[4-[6-[(2R)-3-[[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]oxy]-2-hydroxypropyl]-2,6-diazaspiro[3.3]heptan-2-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CC[C@H](N2CC3=CC(OC[C@H](O)CN4CC5(C4)CN(C4=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C4)C5)=CC=C3C2=O)C(=O)N1	C45H43F3N8O8S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-38SLS6	SCHEMBL29482967	(3R)-N-[3-[5-[4-[6-[(2R)-3-[[2-[(3R)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]oxy]-2-hydroxypropyl]-2,6-diazaspiro[3.3]heptan-2-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CC[C@@H](N2CC3=CC(OC[C@H](O)CN4CC5(C4)CN(C4=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C4)C5)=CC=C3C2=O)C(=O)N1	C45H43F3N8O8S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-EBY0TS	SCHEMBL30253777	(3R)-N-[3-[5-[4-[(3R,4S)-4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]-3-fluoropiperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(C4CCN(C[C@@H]5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6)C[C@@H]5F)CC4)=CC=C3C2=O)C(=O)N1	C48H48F4N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-L7E53U	WO2022047145A1_126	(3R)-N-[3-[5-[4-[4-[2-[[3-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]oxy]cyclobutyl]-methylamino]ethyl]piperazin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	CN(CCN1CCN(C2=CC=C(C3=CC4=C(N=C3)NC=C4C(=O)C3=C(F)C=CC(NS(=O)(=O)N4CC[C@@H](F)C4)=C3F)C=C2)CC1)[C@H]1C[C@@H](OC2=CC3=C(C=C2)C(=O)N(C2CCC(=O)NC2=O)C3)C1	C48H50F3N9O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-932O6B	SCHEMBL30254212	(3R)-N-[3-[5-[4-[4-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]ethyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(C4CCN(CCC5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C49H51F3N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-9KAPEC	SCHEMBL30253991	(3R)-N-[3-[5-[4-[6-[(2R)-3-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]-2-hydroxypropyl]-2,6-diazaspiro[3.3]heptan-2-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CC[C@H](N2CC3=C(C=CC(C[C@@H](O)CN4CC5(C4)CN(C4=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C4)C5)=C3)C2=O)C(=O)N1	C45H43F3N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-V1PH58	SCHEMBL30253696	(3R)-N-[3-[5-[4-[6-[(2R)-3-[2-[(3R)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]-2-hydroxypropyl]-2,6-diazaspiro[3.3]heptan-2-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CC[C@@H](N2CC3=C(C=CC(C[C@@H](O)CN4CC5(C4)CN(C4=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C4)C5)=C3)C2=O)C(=O)N1	C45H43F3N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-MD1OPV	SCHEMBL30253832	(3R)-N-[3-[5-[4-[6-[(2S)-3-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-2-hydroxypropyl]-2,6-diazaspiro[3.3]heptan-2-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=C(C=CC(C[C@H](O)CN4CC5(C4)CN(C4=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C4)C5)=C3)C2=O)C(=O)N1	C45H43F3N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-RL4LU1	WO2022047145A1_131	.	O=C1CCC(N2CC3=CC(N4CCN(CC5CN(C6=CC=C(C7=CC8=C(C=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6F)C5)CC4)=CC=C3C2=O)C(=O)N1	C46H44F4N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-AMCVXQ	SCHEMBL30254078	(3R)-N-[3-[5-[4-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-5-yl]-2,6-diazaspiro[3.3]heptan-6-yl]methyl]piperidin-1-yl]-3-fluorophenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	COC1=C2C(=O)N(C3CCC(=O)NC3=O)CC2=CC(N2CC3(CN(CC4CCN(C5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5F)CC4)C3)C2)=C1	C49H49F4N9O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-GO3DA4	SCHEMBL30254290	(3R)-N-[3-[5-[6-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-5-yl]-2,6-diazaspiro[3.3]heptan-6-yl]methyl]piperidin-1-yl]pyridin-3-yl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	COC1=C2C(=O)N(C3CCC(=O)NC3=O)CC2=CC(N2CC3(CN(CC4CCN(C5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=N5)CC4)C3)C2)=C1	C48H49F3N10O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-OA68VO	WO2022047145A1_134	(3R)-N-[3-[5-[2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-5-yl]-2,6-diazaspiro[3.3]heptan-6-yl]methyl]piperidin-1-yl]pyrimidin-5-yl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	COC1=C2C(=O)N(C3CCC(=O)NC3=O)CC2=CC(N2CC3(CN(CC4CCN(C5=NC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=N5)CC4)C3)C2)=C1	C47H48F3N11O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-UF6N4F	WO2022047145A1_135	.	O=C1CCC(N2CC3=CC(N4CCN(CCCC5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=N6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C48H51F3N10O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-RNZ9CV	SCHEMBL30253934	(3R)-N-[3-[5-[4-[2-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)-3-fluorophenyl]piperazin-1-yl]ethyl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCN(C2=C(F)C=C(N3CCN(CCC4=CC=C(C5=CC6=C(N=C5)NC=C6C(=O)C5=C(F)C=CC(NS(=O)(=O)N6CC[C@@H](F)C6)=C5F)C=C4)CC3)C=C2)C(=O)N1	C40H38F4N8O5S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-UJO48Z	SCHEMBL30253798	(3R)-N-[3-[5-[4-[4-[3-[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]propyl]piperazin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(N4CCC(CCCN5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C49H52F3N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-SI3NZ4	SCHEMBL29482882	(3R)-N-[3-[5-[4-[6-[(2R)-2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-2-hydroxyethyl]-2,6-diazaspiro[3.3]heptan-2-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC([C@@H](O)CN4CC5(C4)CN(C4=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C4)C5)=CC=C3C2=O)C(=O)N1	C44H41F3N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-TR4N6Y	WO2022047145A1_139	.	O=C1CCC(N2CC3=CC(OCCCOC4CCN(C5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)CC4)=CCC3C2=O)C(=O)N1	C45H46F3N7O8S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-QR9ITC	SCHEMBL30253640	(3R)-N-[3-[5-[4-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)-3-fluorophenyl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCN(C2=CC=C(C3CCN(CC4CCN(C5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)CC4)CC3)C=C2F)C(=O)N1	C45H46F4N8O5S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-1TO3SN	SCHEMBL30253953	(3R)-N-[3-[5-[6-[6-[3-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]propyl]-2,6-diazaspiro[3.3]heptan-2-yl]pyridin-3-yl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(CCCN4CC5(C4)CN(C4=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=N4)C5)=CC=C3C2=O)C(=O)N1	C44H42F3N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-P6RC2B	SCHEMBL29482924	(3R)-N-[3-[5-[4-[6-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-4-hydroxypiperidin-4-yl]methyl]-2,6-diazaspiro[3.3]heptan-2-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(N4CCC(O)(CN5CC6(C5)CN(C5=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C5)C6)CC4)=CC=C3C2=O)C(=O)N1	C48H48F3N9O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-9UHL2C	SCHEMBL24319588	(3R)-N-[3-[5-[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methoxymethyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide; SCHEMBL29482856	O=C1CCC(N2CC3=CC(N4CCC(COCC5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C49H51F3N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-8DYJXS	SCHEMBL30254011	(3R)-N-[3-[5-[4-[3-[[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]piperazin-1-yl]methyl]azetidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=C(C=CC(N4CCC(N5CCN(CC6CN(C7=CC=C(C8=CC9=C(N=C8)NC=C9C(=O)C8=C(F)C=CC(NS(=O)(=O)N9CC[C@@H](F)C9)=C8F)C=C7)C6)CC5)CC4)=C3)C2=O)C(=O)N1	C50H53F3N10O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-QHD3L1	SCHEMBL30253659	(3R)-N-[3-[5-[4-[4-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]ethyl-methylamino]cyclohexyl]oxyphenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	CN(CCN1CCN(C2=CC3=C(C=C2)C(=O)N(C2CCC(=O)NC2=O)C3)CC1)[C@H]1CC[C@H](OC2=CC=C(C3=CC4=C(N=C3)NC=C4C(=O)C3=C(F)C=CC(NS(=O)(=O)N4CC[C@@H](F)C4)=C3F)C=C2)CC1	C50H54F3N9O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-ZMZY92	WO2022047145A1_146	.	C=C1CCC(N2CC3=CC(N4CCC(CN5CCN(CC6C=CC(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)=CC6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C49H54F3N9O5S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-4SV7E5	SCHEMBL30253930	(3R)-N-[3-[5-[2-[6-[3-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]propyl]-2,6-diazaspiro[3.3]heptan-2-yl]pyrimidin-5-yl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(CCCN4CC5(C4)CN(C4=NC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=N4)C5)=CC=C3C2=O)C(=O)N1	C43H41F3N10O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-LR5ZFA	SCHEMBL30254365	(3R)-N-[3-[5-[4-[4-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]ethoxy]ethyl]piperazin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=C(C=CC(CCOCCN4CCN(C5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)CC4)=C3)C2=O)C(=O)N1	C45H45F3N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-OA2TGI	SCHEMBL24319925	(3R)-N-[3-[5-[4-[2-[(2S)-4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-2-(hydroxymethyl)piperidin-1-yl]ethyl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide; SCHEMBL30253613	O=C1CCC(N2CC3=C(C=CC(C4CCN(CCC5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)[C@H](CO)C4)=C3)C2=O)C(=O)N1	C45H44F3N7O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-0NKCBG	WO2022047145A1_150	.	O=NC[C@H]1CC(C2=CC3=C(C=C2)C(=O)N(C2CCC(=O)NC2=O)C3)CCN1CCC1C=CC(C2=CC3=C(N=C2)NC=C3C(=O)C2=C(F)C=CC(NS(=O)(=O)N3CC[C@@H](F)C3)=C2F)=CC1	C45H45F3N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-20IX0B	SCHEMBL30253762	(3R)-N-[3-[5-[4-[1-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]ethoxy]ethyl]piperidin-4-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(CCOCCN4CCC(C5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C46H46F3N7O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-BI7ZDW	SCHEMBL30254017	(3R)-N-[3-[5-[4-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]ethyl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(N4CCN(CCC5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)CC4)=C(F)C=C3C2=O)C(=O)N1	C43H40F4N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-P05F9H	SCHEMBL30253869	(3R)-N-[3-[5-[2-[[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]methyl]pyrimidin-5-yl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(N4CCC(CN5CCN(CC6=NC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=N6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C46H48F3N11O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-OE7JP9	WO2022047145A1_154	.	O=C1CCC(N2CC3=CC(N4CCC(CN5CCC(CC6=NC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=N6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C47H49F3N10O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-IIUXRY	SCHEMBL24021782	(3R)-N-[3-[5-[4-[4-[[[3-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]oxy]cyclobutyl]-methylamino]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	CN(CC1CCN(C2=CC=C(C3=CC4=C(N=C3)NC=C4C(=O)C3=C(F)C=CC(NS(=O)(=O)N4CC[C@@H](F)C4)=C3F)C=C2)CC1)[C@H]1C[C@@H](OC2=CC3=C(C=C2)C(=O)N(C2CCC(=O)NC2=O)C3)C1	C48H49F3N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-QT51GP	SCHEMBL30254355	(3R)-N-[3-[5-[4-[6-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)-3-fluorophenyl]piperidin-4-yl]methyl]-2,6-diazaspiro[3.3]heptan-2-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCN(C2=CC=C(N3CCC(CN4CC5(C4)CN(C4=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C4)C5)CC3)C=C2F)C(=O)N1	C45H45F4N9O5S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-DTWDMT	SCHEMBL30253588	(3R)-N-[3-[5-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(C4CCN(CC5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6)CC5)CC4)=C(F)C=C3C2=O)C(=O)N1	C48H48F4N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-Q3UUOE	SCHEMBL30253911	(3R)-N-[3-[5-[6-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-2,6-diazaspiro[3.3]heptan-6-yl]ethoxy]pyridin-3-yl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(N4CC5(CN(CCOC6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=N6)C5)C4)=CC=C3C2=O)C(=O)N1	C43H40F3N9O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-K6UBU9	SCHEMBL30253826	(3R)-N-[3-[5-[4-[3-[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]azetidin-3-yl]azetidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(N4CC(C5CN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6)C5)C4)=CC=C3C2=O)C(=O)N1	C43H39F3N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-GUNAFB	SCHEMBL24319381	(3R)-N-[3-[5-[4-[4-[[4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide; SCHEMBL29482877	O=C1CC[C@H](N2CC3=C(C=CC(C4CCN(CC5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C48H49F3N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-FS4AD4	WO2022047145A1_161	(3R)-N-[3-[5-[4-[4-[[4-[2-[(3R)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CC[C@@H](N2CC3=C(C=CC(C4CCN(CC5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C48H49F3N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-YEMNT1	WO2022047145A1_162	.	O=C1CCC(N2CC3CC(N4CCC(CN5CCN(C6(C7=CC=C(C8=CC9=C(N=C8)NC=C9C(=O)C8=C(F)C=CC(NS(=O)(=O)N9CC[C@@H](F)C9)=C8F)C=C7)CC6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C50H54F3N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-QIXQSR	SCHEMBL30253748	(3R)-N-[3-[5-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]-3-fluorophenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	COC1=C2C(=O)N(C3CCC(=O)NC3=O)CC2=CC(C2CCN(CC3CCN(C4=CC=C(C5=CC6=C(N=C5)NC=C6C(=O)C5=C(F)C=CC(NS(=O)(=O)N6CC[C@@H](F)C6)=C5F)C=C4F)CC3)CC2)=C1	C49H50F4N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-I4RZ05	SCHEMBL30253907	(3R)-N-[3-[5-[6-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridin-3-yl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	COC1=C2C(=O)N(C3CCC(=O)NC3=O)CC2=CC(C2CCN(CC3CCN(C4=CC=C(C5=CC6=C(N=C5)NC=C6C(=O)C5=C(F)C=CC(NS(=O)(=O)N6CC[C@@H](F)C6)=C5F)C=N4)CC3)CC2)=C1	C48H50F3N9O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-AH4J0E	SCHEMBL30254173	(3R)-N-[3-[5-[4-[6-[(2S)-3-[[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]oxy]-2-hydroxypropyl]-2,6-diazaspiro[3.3]heptan-2-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CC[C@H](N2CC3=CC(OC[C@@H](O)CN4CC5(C4)CN(C4=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C4)C5)=CC=C3C2=O)C(=O)N1	C45H43F3N8O8S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-DA9X20	SCHEMBL30253916	(3R)-N-[3-[5-[4-[6-[(2S)-3-[[2-[(3R)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]oxy]-2-hydroxypropyl]-2,6-diazaspiro[3.3]heptan-2-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CC[C@@H](N2CC3=CC(OC[C@@H](O)CN4CC5(C4)CN(C4=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C4)C5)=CC=C3C2=O)C(=O)N1	C45H43F3N8O8S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-BPWWKB	WO2022047145A1_167	(3R)-N-[3-[5-[4-[3-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl-methylamino]cyclobutyl]oxyphenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	CN(CC1CCN(C2=CC3=C(C=C2)C(=O)N(C2CCC(=O)NC2=O)C3)CC1)[C@H]1C[C@@H](OC2=CC=C(C3=CC4=C(N=C3)NC=C4C(=O)C3=C(F)C=CC(NS(=O)(=O)N4CC[C@@H](F)C4)=C3F)C=C2)C1	C48H49F3N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-R66YMU	SCHEMBL30253782	(3R)-N-[3-[5-[4-[4-[[4-[4-(2,6-dioxopiperidin-3-yl)-3-fluorophenyl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(C2=C(F)C=C(C3CCN(CC4CCN(C5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)CC4)CC3)C=C2)C(=O)N1	C46H47F4N7O5S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-ZAY8BI	SCHEMBL30253726	(3R)-N-[2,4-difluoro-3-[5-[4-[4-[[4-[2-(1-methyl-2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]phenyl]-3-fluoropyrrolidine-1-sulfonamide	CN1C(=O)CCC(N2CC3=C(C=CC(C4CCN(CC5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6)CC5)CC4)=C3)C2=O)C1=O	C49H51F3N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-7W9DEN	SCHEMBL30254405	(3R)-N-[3-[5-[4-[6-[(2S)-3-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]-2-hydroxypropyl]-2,6-diazaspiro[3.3]heptan-2-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CC[C@H](N2CC3=C(C=CC(C[C@H](O)CN4CC5(C4)CN(C4=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C4)C5)=C3)C2=O)C(=O)N1	C45H43F3N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-YUZOGC	WO2022047145A1_171	(3R)-N-[3-[5-[4-[6-[(2S)-3-[2-[(3R)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]-2-hydroxypropyl]-2,6-diazaspiro[3.3]heptan-2-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CC[C@@H](N2CC3=C(C=CC(C[C@H](O)CN4CC5(C4)CN(C4=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C4)C5)=C3)C2=O)C(=O)N1	C45H43F3N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-T3N83Z	SCHEMBL29482809	(3R)-N-[3-[5-[4-[6-[(2S)-4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]-2-hydroxybutyl]-2,6-diazaspiro[3.3]heptan-2-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CC[C@H](N2CC3=CC(CC[C@H](O)CN4CC5(C4)CN(C4=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C4)C5)=CC=C3C2=O)C(=O)N1	C46H45F3N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-IPEN0P	SCHEMBL29482976	(3R)-N-[3-[5-[4-[6-[(2S)-4-[2-[(3R)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]-2-hydroxybutyl]-2,6-diazaspiro[3.3]heptan-2-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide; SCHEMBL29482979	O=C1CC[C@@H](N2CC3=CC(CC[C@H](O)CN4CC5(C4)CN(C4=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C4)C5)=CC=C3C2=O)C(=O)N1	C46H45F3N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-437PMO	SCHEMBL30253631	(3R)-N-[3-[5-[4-[1-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperidin-4-yl]cyclopropyl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(N4CCC(CN5CCC(C6(C7=CC=C(C8=CC9=C(N=C8)NC=C9C(=O)C8=C(F)C=CC(NS(=O)(=O)N9CC[C@@H](F)C9)=C8F)C=C7)CC6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C51H53F3N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-HKFOVO	SCHEMBL30254010	(3R)-N-[3-[5-[2-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyrimidin-5-yl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	COC1=C2C(=O)N(C3CCC(=O)NC3=O)CC2=CC(C2CCN(CC3CCN(C4=NC=C(C5=CC6=C(N=C5)NC=C6C(=O)C5=C(F)C=CC(NS(=O)(=O)N6CC[C@@H](F)C6)=C5F)C=N4)CC3)CC2)=C1	C47H49F3N10O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-3UX0DM	SCHEMBL30254200	(3R)-N-[2,4-difluoro-3-[5-[4-[4-[[4-[3-fluoro-4-(3-methyl-2,6-dioxopiperidin-3-yl)phenyl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]phenyl]-3-fluoropyrrolidine-1-sulfonamide	CC1(C2=C(F)C=C(C3CCN(CC4CCN(C5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)CC4)CC3)C=C2)CCC(=O)NC1=O	C47H49F4N7O5S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-GU7NVO	SCHEMBL24320700	N-[3-[5-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]pyrrolidine-1-sulfonamide; SCHEMBL30254047	O=C1CCC(N2CC3=C(C=CC(C4CCN(CC5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CCCC8)=C7F)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C48H50F2N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-87ELAB	SCHEMBL24319575	(3R)-N-[3-[5-[4-[4-[2-[4-[4-(2,6-dioxopiperidin-3-yl)-3-fluorophenyl]piperidin-1-yl]ethyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide; SCHEMBL29482912	O=C1CCC(C2=C(F)C=C(C3CCN(CCC4CCN(C5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)CC4)CC3)C=C2)C(=O)N1	C47H49F4N7O5S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-USYKYV	SCHEMBL24320701	(3R)-N-[3-[5-[4-[(1S,5R)-6-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]-3-azabicyclo[3.1.0]hexan-3-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide; SCHEMBL30253830	[H][C@@]12CN(C3=CC=C(C4=CC5=C(N=C4)NC=C5C(=O)C4=C(F)C=CC(NS(=O)(=O)N5CC[C@@H](F)C5)=C4F)C=C3)C[C@]1([H])[C@H]2CN1CCC(C2=CC=C3C(=O)N(C4CCC(=O)NC4=O)CC3=C2)CC1	C48H47F3N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-GME5DZ	WO2022047145A1_180	.	O=C1CCC(N2CC3=CC(C4CCN(C[C@@H]5C[C@H]6CC[C@@H](C5)N6C5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C50H51F3N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-EZ8EEE	WO2022047145A1_181	.	O=C1CCC(N2CC3=CC(N4CCC(CC5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)CC6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C48H51F3N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-YDOSC4	WO2022047145A1_182	(3R)-N-[3-[5-[4-[3-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]ethyl-methylamino]cyclobutyl]oxyphenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	CN(CCN1CCN(C2=CC3=C(C=C2)C(=O)N(C2CCC(=O)NC2=O)C3)CC1)[C@H]1C[C@@H](OC2=CC=C(C3=CC4=C(N=C3)NC=C4C(=O)C3=C(F)C=CC(NS(=O)(=O)N4CC[C@@H](F)C4)=C3F)C=C2)C1	C48H50F3N9O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-J0C31Q	SCHEMBL30254060	(3R)-N-[2,4-difluoro-3-[5-[4-[4-[[4-[2-(3-methyl-2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]phenyl]-3-fluoropyrrolidine-1-sulfonamide	CC1(N2CC3=C(C=CC(C4CCN(CC5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6)CC5)CC4)=C3)C2=O)CCC(=O)NC1=O	C49H51F3N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-KTY8ZI	SCHEMBL30253843	4-[1-[[1-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]piperidin-4-yl]methyl]piperidin-4-yl]-N-(2,6-dioxopiperidin-3-yl)-2-methoxybenzamide	COC1=C(C(=O)NC2CCC(=O)NC2=O)C=CC(C2CCN(CC3CCN(C4=CC=C(C5=CC6=C(N=C5)NC=C6C(=O)C5=C(F)C=CC(NS(=O)(=O)N6CC[C@@H](F)C6)=C5F)C=C4)CC3)CC2)=C1	C48H51F3N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-91Q75A	SCHEMBL30254279	(3R)-N-[3-[5-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-3-oxo-1H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=C(C=C(C4CCN(CC5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6)CC5)CC4)C=C3)C2=O)C(=O)N1	C48H49F3N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-Q8GTN4	SCHEMBL24320348	(3R)-N-[3-[5-[4-[4-[(3R)-3-[2-[(3S)-2,6-dioxopiperidin-3-yl]-7-methoxy-1-oxo-3H-isoindol-5-yl]-3-hydroxypropyl]piperazin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide; SCHEMBL29482806	COC1=C2C(=O)N([C@H]3CCC(=O)NC3=O)CC2=CC([C@H](O)CCN2CCN(C3=CC=C(C4=CC5=C(N=C4)NC=C5C(=O)C4=C(F)C=CC(NS(=O)(=O)N5CC[C@@H](F)C5)=C4F)C=C3)CC2)=C1	C45H45F3N8O8S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-X4IANI	SCHEMBL24319767	(3R)-N-[3-[5-[4-[4-[(3R)-3-[2-[(3R)-2,6-dioxopiperidin-3-yl]-7-methoxy-1-oxo-3H-isoindol-5-yl]-3-hydroxypropyl]piperazin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide; SCHEMBL29482838	COC1=C2C(=O)N([C@@H]3CCC(=O)NC3=O)CC2=CC([C@H](O)CCN2CCN(C3=CC=C(C4=CC5=C(N=C4)NC=C5C(=O)C4=C(F)C=CC(NS(=O)(=O)N5CC[C@@H](F)C5)=C4F)C=C3)CC2)=C1	C45H45F3N8O8S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-OVE87J	WO2022047145A1_188	.	O=C1CCC(N2CC3=CC(C4CCN(C[C@H]5C[C@H]6CC[C@@H](C5)N6C5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C50H51F3N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-SKZXCF	WO2022047145A1_189	.	C=C1CCC(C2=CC=C(C3CCN(CC4CCN(C5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)CC4)CC3)C=C2)C(=O)N1	C47H50F3N7O4S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-WPOT5U	SCHEMBL30253687	N-[3-[5-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3,3-difluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=C(C=CC(C4CCN(CC5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CCC(F)(F)C8)=C7F)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C48H48F4N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-CG0QKE	SCHEMBL30253759	5-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-3-[3-[[ethyl(methyl)sulfamoyl]amino]-2,6-difluorobenzoyl]-1H-pyrrolo[2,3-b]pyridine	CCN(C)S(=O)(=O)NC1=C(F)C(C(=O)C2=CNC3=C2C=C(C2=CC=C(N4CCC(CN5CCC(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)CC5)CC4)C=C2)C=N3)=C(F)C=C1	C47H50F2N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-TEVLNE	SCHEMBL30253965	(3R)-N-[3-[5-[4-[[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]azetidin-3-yl]methyl]piperazin-1-yl]methyl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=C(C=CC(N4CC(CN5CCN(CC6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6)CC5)C4)=C3)C2=O)C(=O)N1	C46H46F3N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-37WNWY	SCHEMBL30253769	(3R)-N-[3-[5-[2-[[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]azetidin-3-yl]methyl]piperazin-1-yl]methyl]pyrimidin-5-yl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=C(C=CC(N4CC(CN5CCN(CC6=NC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=N6)CC5)C4)=C3)C2=O)C(=O)N1	C44H44F3N11O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-ITNE6H	SCHEMBL30253654	(3R)-N-[3-[5-[2-[[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]azetidin-3-yl]methyl]piperidin-4-yl]methyl]pyrimidin-5-yl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=C(C=CC(N4CC(CN5CCC(CC6=NC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=N6)CC5)C4)=C3)C2=O)C(=O)N1	C45H45F3N10O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-E16NFL	SCHEMBL30254116	(3R)-N-[3-[5-[4-[4-[2-[[4-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]oxy]cyclohexyl]-methylamino]ethyl]piperazin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	CN(CCN1CCN(C2=CC=C(C3=CC4=C(N=C3)NC=C4C(=O)C3=C(F)C=CC(NS(=O)(=O)N4CC[C@@H](F)C4)=C3F)C=C2)CC1)[C@H]1CC[C@H](OC2=CC3=C(C=C2)C(=O)N(C2CCC(=O)NC2=O)C3)CC1	C50H54F3N9O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-V02171	SCHEMBL30253856	5-[1-[[1-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]piperidin-4-yl]methyl]piperidin-4-yl]-N-[(3S)-2,6-dioxopiperidin-3-yl]-2-fluorobenzamide	O=C1CC[C@H](NC(=O)C2=CC(C3CCN(CC4CCN(C5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)CC4)CC3)=CC=C2F)C(=O)N1	C47H48F4N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-P7F5MT	SCHEMBL24319945	5-[1-[[1-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]piperidin-4-yl]methyl]piperidin-4-yl]-N-[(3R)-2,6-dioxopiperidin-3-yl]-2-fluorobenzamide; SCHEMBL30254343	O=C1CC[C@@H](NC(=O)C2=CC(C3CCN(CC4CCN(C5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)CC4)CC3)=CC=C2F)C(=O)N1	C47H48F4N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-T5Q9IO	SCHEMBL24319944	(3R)-N-[3-[5-[4-[3-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]azetidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide; SCHEMBL30254325	O=C1CCC(N2CC3=CC(C4CCN(CC5CN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6)C5)CC4)=CC=C3C2=O)C(=O)N1	C46H45F3N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-QP6N0W	SCHEMBL24319418	(3R)-N-[3-[5-[4-[4-[2-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)-3-fluorophenyl]piperidin-1-yl]ethyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide; SCHEMBL29482957	O=C1CCN(C2=C(F)C=C(C3CCN(CCC4CCN(C5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)CC4)CC3)C=C2)C(=O)N1	C46H48F4N8O5S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-R0T2YA	SCHEMBL24319946	(3R)-N-[3-[5-[4-[1-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]azetidin-3-yl]methyl]piperazin-1-yl]cyclopropyl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide; SCHEMBL31302555	O=C1CCC(N2CC3=C(C=CC(N4CC(CN5CCN(C6(C7=CC=C(C8=CC9=C(N=C8)NC=C9C(=O)C8=C(F)C=CC(NS(=O)(=O)N9CC[C@@H](F)C9)=C8F)C=C7)CC6)CC5)C4)=C3)C2=O)C(=O)N1	C48H48F3N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-MU93LZ	SCHEMBL24319502	(3R)-N-[3-[5-[2-[1-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]cyclopropyl]pyrimidin-5-yl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide; SCHEMBL30253812	O=C1CCC(N2CC3=C(C=CC(N4CCC(CN5CCN(C6(C7=NC=C(C8=CC9=C(N=C8)NC=C9C(=O)C8=C(F)C=CC(NS(=O)(=O)N9CC[C@@H](F)C9)=C8F)C=N7)CC6)CC5)CC4)=C3)C2=O)C(=O)N1	C48H50F3N11O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-848T76	SCHEMBL24319504	(3R)-N-[3-[5-[2-[1-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]azetidin-3-yl]methyl]piperazin-1-yl]cyclopropyl]pyrimidin-5-yl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide; SCHEMBL30253795	O=C1CCC(N2CC3=C(C=CC(N4CC(CN5CCN(C6(C7=NC=C(C8=CC9=C(N=C8)NC=C9C(=O)C8=C(F)C=CC(NS(=O)(=O)N9CC[C@@H](F)C9)=C8F)C=N7)CC6)CC5)C4)=C3)C2=O)C(=O)N1	C46H46F3N11O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-RFN96P	SCHEMBL24319501	(3R)-N-[3-[5-[4-[4-[[4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2-ethyl-4-fluorophenyl]-3-fluoropyrrolidine-1-sulfonamide; SCHEMBL29482942	CCC1=C(NS(=O)(=O)N2CC[C@@H](F)C2)C=CC(F)=C1C(=O)C1=CNC2=C1C=C(C1=CC=C(N3CCC(CN4CCC(C5=CC=C6C(=O)N([C@H]7CCC(=O)NC7=O)CC6=C5)CC4)CC3)C=C1)C=N2	C50H54F2N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-60VTOM	SCHEMBL24319290	N-[3-[5-[4-[4-[[4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-2-methylpropane-1-sulfonamide; SCHEMBL29482938	CC(C)CS(=O)(=O)NC1=CC=C(F)C(C(=O)C2=CNC3=NC=C(C4=CC=C(N5CCC(CN6CCC(C7=CC=C8C(=O)N([C@H]9CCC(=O)NC9=O)CC8=C7)CC6)CC5)C=C4)C=C23)=C1F	C48H51F2N7O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-ILX3AZ	SCHEMBL24319507	(3R)-N-[3-[5-[3-cyano-4-[4-[[4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide; SCHEMBL29482917	N#CC1=C(N2CCC(CN3CCC(C4=CC=C5C(=O)N([C@H]6CCC(=O)NC6=O)CC5=C4)CC3)CC2)C=CC(C2=CC3=C(N=C2)NC=C3C(=O)C2=C(F)C=CC(NS(=O)(=O)N3CC[C@@H](F)C3)=C2F)=C1	C49H48F3N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-UKKT40	SCHEMBL24319272	1-cyclopropyl-N-[3-[5-[4-[4-[[4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]methanesulfonamide; SCHEMBL29482952	O=C1CC[C@H](N2CC3=CC(C4CCN(CC5CCN(C6=CC=C(C7=CN=C8NC=C(C(=O)C9=C(F)C(NS(=O)(=O)CC%10CC%10)=CC=C9F)C8=C7)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C48H49F2N7O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-8R68NB	SCHEMBL24319579	(3R)-N-[3-[5-[4-[4-[[4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-4-fluoro-2-methoxyphenyl]-3-fluoropyrrolidine-1-sulfonamide; SCHEMBL29482845	COC1=C(C(=O)C2=CNC3=NC=C(C4=CC=C(N5CCC(CN6CCC(C7=CC=C8C(=O)N([C@H]9CCC(=O)NC9=O)CC8=C7)CC6)CC5)C=C4)C=C23)C(F)=CC=C1NS(=O)(=O)N1CC[C@@H](F)C1	C49H52F2N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-USJ3TX	SCHEMBL24319510	3-[2,6-difluoro-3-[[methyl(propan-2-yl)sulfamoyl]amino]benzoyl]-5-[4-[4-[[4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine; SCHEMBL29482922	CC(C)N(C)S(=O)(=O)NC1=CC=C(F)C(C(=O)C2=CNC3=NC=C(C4=CC=C(N5CCC(CN6CCC(C7=CC=C8C(=O)N([C@H]9CCC(=O)NC9=O)CC8=C7)CC6)CC5)C=C4)C=C23)=C1F	C48H52F2N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-2MR3ZD	SCHEMBL24319523	(3R)-N-[3-[5-[4-[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]azetidin-3-yl]methyl]piperazin-1-yl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide; SCHEMBL29482868	O=C1CCC(N2CC3=CC(N4CC(CN5CCN(C6CCN(C7=CC=C(C8=CN=C9NC=C(C(=O)C%10=C(F)C(NS(=O)(=O)N%11CC[C@@H](F)C%11)=CC=C%10F)C9=C8)C=C7)CC6)CC5)C4)=CC=C3C2=O)C(=O)N1	C50H53F3N10O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-5G3Z56	SCHEMBL24319506	(3R)-N-[3-[5-[4-[4-[[4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]-3-(methylamino)phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide; SCHEMBL29482801	CNC1=C(N2CCC(CN3CCC(C4=CC=C5C(=O)N([C@H]6CCC(=O)NC6=O)CC5=C4)CC3)CC2)C=CC(C2=CC3=C(N=C2)NC=C3C(=O)C2=C(F)C=CC(NS(=O)(=O)N3CC[C@@H](F)C3)=C2F)=C1	C49H52F3N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-12JXK4	SCHEMBL24319534	(2S)-N-[3-[5-[4-[4-[[4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-2-methylpyrrolidine-1-sulfonamide; SCHEMBL29482888	C[C@H]1CCCN1S(=O)(=O)NC1=C(F)C(C(=O)C2=CNC3=C2C=C(C2=CC=C(N4CCC(CN5CCC(C6=CC=C7C(=O)N([C@H]8CCC(=O)NC8=O)CC7=C6)CC5)CC4)C=C2)C=N3)=C(F)C=C1	C49H52F2N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-S3NI0S	SCHEMBL24319543	(3R)-N-[3-[5-[4-[4-[[4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2-fluoro-4-methoxyphenyl]-3-fluoropyrrolidine-1-sulfonamide; SCHEMBL29482880	COC1=C(C(=O)C2=CNC3=C2C=C(C2=CC=C(N4CCC(CN5CCC(C6=CC=C7C(=O)N([C@H]8CCC(=O)NC8=O)CC7=C6)CC5)CC4)C=C2)C=N3)C(F)=C(NS(=O)(=O)N2CC[C@@H](F)C2)C=C1	C49H52F2N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-ZCBNXC	SCHEMBL24319659	3-[3-[[2,2-difluoroethyl(methyl)sulfamoyl]amino]-2,6-difluorobenzoyl]-5-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine; SCHEMBL30253632	CN(CC(F)F)S(=O)(=O)NC1=C(F)C(C(=O)C2=CNC3=C2C=C(C2=CC=C(N4CCC(CN5CCC(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)CC5)CC4)C=C2)C=N3)=C(F)C=C1	C47H48F4N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-4MNDEX	SCHEMBL24319660	(3R)-N-[3-[5-[4-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide; SCHEMBL30253562	O=C1CCC(N2CC3=CC(N4CCC(C5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C47H47F3N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-4KTWOK	SCHEMBL24319658	(3R)-N-[3-[5-[5-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyrimidin-2-yl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide; SCHEMBL30253868	O=C1CCC(N2CC3=CC(C4CCN(CC5CCN(C6=CN=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)N=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C46H47F3N10O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-5OQA6S	SCHEMBL30254297	(3R)-N-[3-[5-[4-[(3R)-3-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]ethyl]pyrrolidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(C4CCN(CC[C@@H]5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6)C5)CC4)=CC=C3C2=O)C(=O)N1	C48H49F3N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-YT5R9K	SCHEMBL30253681	(3R)-N-[3-[5-[4-[(3S)-3-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]ethyl]pyrrolidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(C4CCN(CC[C@H]5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6)C5)CC4)=CC=C3C2=O)C(=O)N1	C48H49F3N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-00Q82T	SCHEMBL30254109	(3R)-N-[3-[5-[4-[3-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]ethyl]azetidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(C4CCN(CCC5CN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6)C5)CC4)=CC=C3C2=O)C(=O)N1	C47H47F3N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-5BHJZE	SCHEMBL24319807	(3R)-N-[3-[5-[4-[4-[[4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide; SCHEMBL30254051	O=C1CC[C@H](N2CC3=C(C=CC(N4CCN(CC5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C47H48F3N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-HTM5QJ	SCHEMBL30254195	(3R)-N-[3-[5-[4-[4-[[4-[2-[(3R)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CC[C@@H](N2CC3=C(C=CC(N4CCN(CC5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C47H48F3N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-MZ00F9	SCHEMBL30253970	(3R)-N-[3-[5-[4-[4-[[2-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]-2,6-diazaspiro[3.3]heptan-6-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CC[C@H](N2CC3=C(C=CC(N4CC5(CN(CC6CCN(C7=CC=C(C8=CC9=C(N=C8)NC=C9C(=O)C8=C(F)C=CC(NS(=O)(=O)N9CC[C@@H](F)C9)=C8F)C=C7)CC6)C5)C4)=C3)C2=O)C(=O)N1	C48H48F3N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-I53Z9O	SCHEMBL30253638	(3R)-N-[3-[5-[4-[4-[[2-[2-[(3R)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]-2,6-diazaspiro[3.3]heptan-6-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CC[C@@H](N2CC3=C(C=CC(N4CC5(CN(CC6CCN(C7=CC=C(C8=CC9=C(N=C8)NC=C9C(=O)C8=C(F)C=CC(NS(=O)(=O)N9CC[C@@H](F)C9)=C8F)C=C7)CC6)C5)C4)=C3)C2=O)C(=O)N1	C48H48F3N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-ZHPX6B	SCHEMBL24021698	(3R)-N-[3-[5-[4-[4-[[1-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide; SCHEMBL30254036	O=C1CC[C@H](N2CC3=C(C=CC(N4CCC(CN5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C47H48F3N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-XQOWG7	SCHEMBL24021696	(3R)-N-[3-[5-[4-[4-[[1-[2-[(3R)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide; SCHEMBL30253699	O=C1CC[C@@H](N2CC3=C(C=CC(N4CCC(CN5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C47H48F3N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-50G3AP	SCHEMBL30253678	(3R)-N-[3-[5-[4-[6-[[1-[2-[(3R)-2,6-dioxopiperidin-3-yl]-7-methoxy-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]-2,6-diazaspiro[3.3]heptan-2-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	COC1=CC(N2CCC(CN3CC4(C3)CN(C3=CC=C(C5=CC6=C(N=C5)NC=C6C(=O)C5=C(F)C=CC(NS(=O)(=O)N6CC[C@@H](F)C6)=C5F)C=C3)C4)CC2)=CC2=C1C(=O)N([C@@H]1CCC(=O)NC1=O)C2	C49H50F3N9O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-QFB9I9	SCHEMBL30253752	(3R)-N-[3-[5-[4-[6-[[1-[2-[(3S)-2,6-dioxopiperidin-3-yl]-7-methoxy-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]-2,6-diazaspiro[3.3]heptan-2-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	COC1=CC(N2CCC(CN3CC4(C3)CN(C3=CC=C(C5=CC6=C(N=C5)NC=C6C(=O)C5=C(F)C=CC(NS(=O)(=O)N6CC[C@@H](F)C6)=C5F)C=C3)C4)CC2)=CC2=C1C(=O)N([C@H]1CCC(=O)NC1=O)C2	C49H50F3N9O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-PEIEC6	SCHEMBL30253982	(3R)-N-[3-[5-[4-[4-[[3-[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]azetidin-3-yl]azetidin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(N4CC(C5CN(CC6CCN(C7=CC=C(C8=CC9=C(N=C8)NC=C9C(=O)C8=C(F)C=CC(NS(=O)(=O)N9CC[C@@H](F)C9)=C8F)C=C7)CC6)C5)C4)=CC=C3C2=O)C(=O)N1	C49H50F3N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-O8NS5G	SCHEMBL30253943	N-[3-[5-[4-[4-[[2-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]-2,6-diazaspiro[3.3]heptan-6-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]propane-1-sulfonamide	CCCS(=O)(=O)NC1=C(F)C(C(=O)C2=CNC3=C2C=C(C2=CC=C(N4CCC(CN5CC6(C5)CN(C5=CC=C7C(=O)N([C@H]8CCC(=O)NC8=O)CC7=C5)C6)CC4)C=C2)C=N3)=C(F)C=C1	C47H48F2N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-5O3XY5	SCHEMBL30253889	N-[3-[5-[4-[4-[[2-[2-[(3R)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]-2,6-diazaspiro[3.3]heptan-6-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]propane-1-sulfonamide	CCCS(=O)(=O)NC1=C(F)C(C(=O)C2=CNC3=C2C=C(C2=CC=C(N4CCC(CN5CC6(C5)CN(C5=CC=C7C(=O)N([C@@H]8CCC(=O)NC8=O)CC7=C5)C6)CC4)C=C2)C=N3)=C(F)C=C1	C47H48F2N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-1RCJ6C	SCHEMBL24319931	N-[3-[5-[4-[4-[[4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]pyrrolidine-1-sulfonamide; SCHEMBL30254095	O=C1CC[C@H](N2CC3=C(C=CC(C4CCN(CC5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CCCC8)=C7F)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C48H50F2N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-OM9LYZ	SCHEMBL24319933	N-[3-[5-[4-[4-[[4-[2-[(3R)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]pyrrolidine-1-sulfonamide; SCHEMBL30253786	O=C1CC[C@@H](N2CC3=C(C=CC(C4CCN(CC5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CCCC8)=C7F)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C48H50F2N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-M8BFF7	SCHEMBL30253770	N-[3-[5-[4-[4-[[4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3,3-difluoropyrrolidine-1-sulfonamide	O=C1CC[C@H](N2CC3=C(C=CC(C4CCN(CC5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CCC(F)(F)C8)=C7F)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C48H48F4N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-6VVHLE	SCHEMBL30254386	N-[3-[5-[4-[4-[[4-[2-[(3R)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3,3-difluoropyrrolidine-1-sulfonamide	O=C1CC[C@@H](N2CC3=C(C=CC(C4CCN(CC5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CCC(F)(F)C8)=C7F)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C48H48F4N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-7VY5GZ	SCHEMBL30254012	N-[3-[5-[4-[4-[[4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]propane-1-sulfonamide	CCCS(=O)(=O)NC1=C(F)C(C(=O)C2=CNC3=C2C=C(C2=CC=C(N4CCC(CN5CCC(C6=CC=C7C(=O)N([C@H]8CCC(=O)NC8=O)CC7=C6)CC5)CC4)C=C2)C=N3)=C(F)C=C1	C47H49F2N7O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-7UC2O2	SCHEMBL30253804	N-[3-[5-[4-[4-[[4-[2-[(3R)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]propane-1-sulfonamide	CCCS(=O)(=O)NC1=C(F)C(C(=O)C2=CNC3=C2C=C(C2=CC=C(N4CCC(CN5CCC(C6=CC=C7C(=O)N([C@@H]8CCC(=O)NC8=O)CC7=C6)CC5)CC4)C=C2)C=N3)=C(F)C=C1	C47H49F2N7O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-QM4H3Y	SCHEMBL24319803	N-[3-[5-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]propane-1-sulfonamide; SCHEMBL30253979	CCCS(=O)(=O)NC1=C(F)C(C(=O)C2=CNC3=C2C=C(C2=CC=C(N4CCC(CN5CCC(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)CC5)CC4)C=C2)C=N3)=C(F)C=C1	C47H49F2N7O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-GEPJRN	WO2022047145A1_237	.	CCCS(=O)(=O)NC1=C(F)C(C(=O)C2=CNC3=C2C=C(C2=CC=C(N4CC5(CN(CN6CCC(C7=CC(OC)=C8C(=O)N([C@H]9CCC(=O)NC9=O)CC8=C7)CC6)C5)C4)C=C2)C=N3)=C(F)C=C1	C48H50F2N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-V811LN	WO2022047145A1_238	.	CCCS(=O)(=O)NC1=C(F)C(C(=O)C2=CNC3=C2C=C(C2=CC=C(N4CC5(CN(CN6CCC(C7=CC(OC)=C8C(=O)N([C@@H]9CCC(=O)NC9=O)CC8=C7)CC6)C5)C4)C=C2)C=N3)=C(F)C=C1	C48H50F2N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-65K8EB	SCHEMBL24319804	(3R)-N-[3-[5-[4-[(2S,4S)-4-[[4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]-2-methylpiperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide; SCHEMBL30253625	C[C@H]1C[C@@H](CN2CCC(C3=CC=C4C(=O)N([C@H]5CCC(=O)NC5=O)CC4=C3)CC2)CCN1C1=CC=C(C2=CC3=C(N=C2)NC=C3C(=O)C2=C(F)C=CC(NS(=O)(=O)N3CC[C@@H](F)C3)=C2F)C=C1	C49H51F3N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-T74HXU	SCHEMBL30253851	(3R)-N-[3-[5-[4-[(2S,4S)-4-[[4-[2-[(3R)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]-2-methylpiperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	C[C@H]1C[C@@H](CN2CCC(C3=CC=C4C(=O)N([C@@H]5CCC(=O)NC5=O)CC4=C3)CC2)CCN1C1=CC=C(C2=CC3=C(N=C2)NC=C3C(=O)C2=C(F)C=CC(NS(=O)(=O)N3CC[C@@H](F)C3)=C2F)C=C1	C49H51F3N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-X6KQ0N	SCHEMBL30253964	(3R)-N-[3-[5-[4-[(2R,4R)-4-[[4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]-2-methylpiperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	C[C@@H]1C[C@H](CN2CCC(C3=CC=C4C(=O)N([C@H]5CCC(=O)NC5=O)CC4=C3)CC2)CCN1C1=CC=C(C2=CC3=C(N=C2)NC=C3C(=O)C2=C(F)C=CC(NS(=O)(=O)N3CC[C@@H](F)C3)=C2F)C=C1	C49H51F3N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-4RM1BR	SCHEMBL30254197	(3R)-N-[3-[5-[4-[(2R,4R)-4-[[4-[2-[(3R)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]-2-methylpiperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	C[C@@H]1C[C@H](CN2CCC(C3=CC=C4C(=O)N([C@@H]5CCC(=O)NC5=O)CC4=C3)CC2)CCN1C1=CC=C(C2=CC3=C(N=C2)NC=C3C(=O)C2=C(F)C=CC(NS(=O)(=O)N3CC[C@@H](F)C3)=C2F)C=C1	C49H51F3N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-15ZHA9	SCHEMBL30254094	N-[3-[5-[4-[4-[[1-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]propane-1-sulfonamide	CCCS(=O)(=O)NC1=C(F)C(C(=O)C2=CNC3=C2C=C(C2=CC=C(N4CCN(CC5CCN(C6=CC=C7C(=O)N([C@H]8CCC(=O)NC8=O)CC7=C6)CC5)CC4)C=C2)C=N3)=C(F)C=C1	C46H48F2N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-E7HKFP	SCHEMBL30254048	N-[3-[5-[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]propane-1-sulfonamide	CCCS(=O)(=O)NC1=C(F)C(C(=O)C2=CNC3=C2C=C(C2=CC=C(N4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)CC5)CC4)C=C2)C=N3)=C(F)C=C1	C46H48F2N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-VWLQGZ	SCHEMBL24319932	N-[3-[5-[4-[4-[[4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]propane-1-sulfonamide; SCHEMBL30254028	CCCS(=O)(=O)NC1=C(F)C(C(=O)C2=CNC3=C2C=C(C2=CC=C(N4CCC(CN5CCN(C6=CC=C7C(=O)N([C@H]8CCC(=O)NC8=O)CC7=C6)CC5)CC4)C=C2)C=N3)=C(F)C=C1	C46H48F2N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-940ADT	SCHEMBL30253790	N-[3-[5-[4-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-2,6-diazaspiro[3.3]heptan-6-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3,3-difluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(N4CC5(CN(CC6CCN(C7=CC=C(C8=CC9=C(N=C8)NC=C9C(=O)C8=C(F)C=CC(NS(=O)(=O)N9CCC(F)(F)C9)=C8F)C=C7)CC6)C5)C4)=CC=C3C2=O)C(=O)N1	C48H47F4N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-I3LJZU	SCHEMBL30253712	N-[3-[5-[4-[6-[[1-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]-2,6-diazaspiro[3.3]heptan-2-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3,3-difluoropyrrolidine-1-sulfonamide; SCHEMBL30253713	COC1=C2C(=O)N(C3CCC(=O)NC3=O)CC2=CC(N2CCC(CN3CC4(C3)CN(C3=CC=C(C5=CC6=C(N=C5)NC=C6C(=O)C5=C(F)C=CC(NS(=O)(=O)N6CCC(F)(F)C6)=C5F)C=C3)C4)CC2)=C1	C49H49F4N9O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-6KSRQT	SCHEMBL30253623	N-[3-[5-[4-[6-[3-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]propyl]-2,6-diazaspiro[3.3]heptan-2-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3,3-difluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(CCCN4CC5(C4)CN(C4=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CCC(F)(F)C7)=C6F)C=C4)C5)=CC=C3C2=O)C(=O)N1	C45H42F4N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-M0T594	SCHEMBL30253692	(3R)-N-[3-[5-[4-[4-[[2-[2-[(3S)-2,6-dioxopiperidin-3-yl]-7-methoxy-1-oxo-3H-isoindol-5-yl]-2,6-diazaspiro[3.3]heptan-6-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	COC1=CC(N2CC3(CN(CC4CCN(C5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)CC4)C3)C2)=CC2=C1C(=O)N([C@H]1CCC(=O)NC1=O)C2	C49H50F3N9O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-6EUH77	SCHEMBL30253912	(3R)-N-[3-[5-[4-[4-[[2-[2-[(3R)-2,6-dioxopiperidin-3-yl]-7-methoxy-1-oxo-3H-isoindol-5-yl]-2,6-diazaspiro[3.3]heptan-6-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	COC1=CC(N2CC3(CN(CC4CCN(C5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)CC4)C3)C2)=CC2=C1C(=O)N([C@@H]1CCC(=O)NC1=O)C2	C49H50F3N9O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-4GWPGM	SCHEMBL30253744	N-[3-[5-[4-[4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]oxy]butyl]piperazin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3,3-difluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(OCCCCN4CCN(C5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CCC(F)(F)C7)=C6F)C=C5)CC4)=CC=C3C2=O)C(=O)N1	C45H44F4N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-OSCM4C	SCHEMBL30254188	(3R)-N-[2-chloro-3-[5-[4-[4-[[4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-4-fluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CC[C@H](N2CC3=CC(C4CCN(CC5CCN(C6=CC=C(C7=CN=C8NC=C(C(=O)C9=C(Cl)C(NS(=O)(=O)N%10CC[C@@H](F)C%10)=CC=C9F)C8=C7)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C48H49ClF2N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-IC6RXQ	SCHEMBL30253622	(3R)-N-[3-[5-[4-[4-[[4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-4-fluoro-2-methylphenyl]-3-fluoropyrrolidine-1-sulfonamide	CC1=C(C(=O)C2=CNC3=NC=C(C4=CC=C(N5CCC(CN6CCC(C7=CC=C8C(=O)N([C@H]9CCC(=O)NC9=O)CC8=C7)CC6)CC5)C=C4)C=C23)C(F)=CC=C1NS(=O)(=O)N1CC[C@@H](F)C1	C49H52F2N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-8ZYG1N	SCHEMBL30253839	(3S)-3-[6-[1-[[1-[4-[3-(3-amino-2,6-difluorobenzoyl)-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]piperidin-4-yl]methyl]piperidin-4-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	NC1=CC=C(F)C(C(=O)C2=CNC3=NC=C(C4=CC=C(N5CCC(CN6CCC(C7=CC=C8C(=O)N([C@H]9CCC(=O)NC9=O)CC8=C7)CC6)CC5)C=C4)C=C23)=C1F	C44H43F2N7O4	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-ED34PE	SCHEMBL30254159	(3R)-N-[3-[5-[3-cyano-4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	N#CC1=C(N2CCC(CN3CCC(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)CC5=C4)CC3)CC2)C=CC(C2=CC3=C(N=C2)NC=C3C(=O)C2=C(F)C=CC(NS(=O)(=O)N3CC[C@@H](F)C3)=C2F)=C1	C49H48F3N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-52OOP2	SCHEMBL30253901	(3R)-N-[3-[5-[4-[4-[[4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]-3-methoxyphenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	COC1=C(N2CCC(CN3CCC(C4=CC=C5C(=O)N([C@H]6CCC(=O)NC6=O)CC5=C4)CC3)CC2)C=CC(C2=CN=C3NC=C(C(=O)C4=C(F)C(NS(=O)(=O)N5CC[C@@H](F)C5)=CC=C4F)C3=C2)=C1	C49H51F3N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-JCFJKY	SCHEMBL30254142	(3R)-N-[3-[5-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]-3-(methylamino)phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	CNC1=C(N2CCC(CN3CCC(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)CC5=C4)CC3)CC2)C=CC(C2=CC3=C(N=C2)NC=C3C(=O)C2=C(F)C=CC(NS(=O)(=O)N3CC[C@@H](F)C3)=C2F)=C1	C49H52F3N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-S32N5V	SCHEMBL30254016	(3R)-N-[3-[5-[4-[2-[[1-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]-2,8-diazaspiro[4.5]decan-8-yl]-3-fluorophenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CC[C@H](N2CC3=CC(N4CCC(CN5CCC6(CCN(C7=CC=C(C8=CC9=C(N=C8)NC=C9C(=O)C8=C(F)C=CC(NS(=O)(=O)N9CC[C@@H](F)C9)=C8F)C=C7F)CC6)C5)CC4)=CC=C3C2=O)C(=O)N1	C51H53F4N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-UKHHVG	SCHEMBL30254223	(3R)-N-[3-[5-[4-[2-[[1-[2-[(3R)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]-2,8-diazaspiro[4.5]decan-8-yl]-3-fluorophenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CC[C@@H](N2CC3=CC(N4CCC(CN5CCC6(CCN(C7=CC=C(C8=CC9=C(N=C8)NC=C9C(=O)C8=C(F)C=CC(NS(=O)(=O)N9CC[C@@H](F)C9)=C8F)C=C7F)CC6)C5)CC4)=CC=C3C2=O)C(=O)N1	C51H53F4N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-Y28DUE	SCHEMBL30254319	(3R)-N-[3-[5-[3,5-dicyano-4-[4-[[4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	N#CC1=CC(C2=CC3=C(N=C2)NC=C3C(=O)C2=C(F)C=CC(NS(=O)(=O)N3CC[C@@H](F)C3)=C2F)=CC(C#N)=C1N1CCC(CN2CCC(C3=CC=C4C(=O)N([C@H]5CCC(=O)NC5=O)CC4=C3)CC2)CC1	C50H47F3N10O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-3CMALM	SCHEMBL30253694	(3R)-N-[3-[5-[3,5-dicyano-4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	N#CC1=CC(C2=CC3=C(N=C2)NC=C3C(=O)C2=C(F)C=CC(NS(=O)(=O)N3CC[C@@H](F)C3)=C2F)=CC(C#N)=C1N1CCC(CN2CCC(C3=CC=C4C(=O)N(C5CCC(=O)NC5=O)CC4=C3)CC2)CC1	C50H47F3N10O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-L9O8V2	SCHEMBL30253908	(2S,5S)-N-[3-[5-[4-[4-[[4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-2,5-dimethylpyrrolidine-1-sulfonamide	C[C@H]1CC[C@H](C)N1S(=O)(=O)NC1=C(F)C(C(=O)C2=CNC3=C2C=C(C2=CC=C(N4CCC(CN5CCC(C6=CC=C7C(=O)N([C@H]8CCC(=O)NC8=O)CC7=C6)CC5)CC4)C=C2)C=N3)=C(F)C=C1	C50H54F2N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-GEJWIT	SCHEMBL30253904	(2S,5S)-N-[3-[5-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-2,5-dimethylpyrrolidine-1-sulfonamide	C[C@H]1CC[C@H](C)N1S(=O)(=O)NC1=C(F)C(C(=O)C2=CNC3=C2C=C(C2=CC=C(N4CCC(CN5CCC(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)CC5)CC4)C=C2)C=N3)=C(F)C=C1	C50H54F2N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-5N4ABJ	SCHEMBL30253820	(2S)-N-[3-[5-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-2-methylpyrrolidine-1-sulfonamide	C[C@H]1CCCN1S(=O)(=O)NC1=C(F)C(C(=O)C2=CNC3=C2C=C(C2=CC=C(N4CCC(CN5CCC(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)CC5)CC4)C=C2)C=N3)=C(F)C=C1	C49H52F2N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-F11IP6	SCHEMBL30253835	(3R)-N-[3-[5-[4-[4-[[4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-4-ethyl-2-fluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	CCC1=C(C(=O)C2=CNC3=C2C=C(C2=CC=C(N4CCC(CN5CCC(C6=CC=C7C(=O)N([C@H]8CCC(=O)NC8=O)CC7=C6)CC5)CC4)C=C2)C=N3)C(F)=C(NS(=O)(=O)N2CC[C@@H](F)C2)C=C1	C50H54F2N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-9T0OFW	SCHEMBL30253764	(3R)-N-[2,4-dichloro-3-[5-[4-[4-[[4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]phenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CC[C@H](N2CC3=CC(C4CCN(CC5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(Cl)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7Cl)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C48H49Cl2FN8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-OT9P0L	SCHEMBL24319909	(3R)-N-[2,4-dichloro-3-[5-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]phenyl]-3-fluoropyrrolidine-1-sulfonamide; SCHEMBL30253702	O=C1CCC(N2CC3=CC(C4CCN(CC5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(Cl)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7Cl)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C48H49Cl2FN8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-4UB8S1	SCHEMBL30253605	(3R)-N-[3-[5-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2-fluoro-4-methoxyphenyl]-3-fluoropyrrolidine-1-sulfonamide	COC1=C(C(=O)C2=CNC3=C2C=C(C2=CC=C(N4CCC(CN5CCC(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)CC5)CC4)C=C2)C=N3)C(F)=C(NS(=O)(=O)N2CC[C@@H](F)C2)C=C1	C49H52F2N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-Y3XUA5	SCHEMBL30254169	(2S,3R)-N-[3-[5-[4-[4-[[4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoro-2-methylpyrrolidine-1-sulfonamide	C[C@H]1[C@H](F)CCN1S(=O)(=O)NC1=C(F)C(C(=O)C2=CNC3=C2C=C(C2=CC=C(N4CCC(CN5CCC(C6=CC=C7C(=O)N([C@H]8CCC(=O)NC8=O)CC7=C6)CC5)CC4)C=C2)C=N3)=C(F)C=C1	C49H51F3N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-KP3WCM	SCHEMBL24319908	(2S,3R)-N-[3-[5-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoro-2-methylpyrrolidine-1-sulfonamide; SCHEMBL30253936	C[C@H]1[C@H](F)CCN1S(=O)(=O)NC1=C(F)C(C(=O)C2=CNC3=C2C=C(C2=CC=C(N4CCC(CN5CCC(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)CC5)CC4)C=C2)C=N3)=C(F)C=C1	C49H51F3N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-XRJQ0Z	SCHEMBL30253917	(3R)-N-[3-[5-[4-[4-[[4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-4-fluoro-2-(trifluoromethyl)phenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CC[C@H](N2CC3=CC(C4CCN(CC5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7C(F)(F)F)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C49H49F5N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-M9GKJA	SCHEMBL30253821	(3R)-N-[3-[5-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-4-fluoro-2-(trifluoromethyl)phenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(C4CCN(CC5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7C(F)(F)F)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C49H49F5N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-U4VCTM	SCHEMBL30253857	(3R)-N-[3-[5-[4-[4-[[4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-dimethoxyphenyl]-3-fluoropyrrolidine-1-sulfonamide	COC1=C(C(=O)C2=CNC3=C2C=C(C2=CC=C(N4CCC(CN5CCC(C6=CC=C7C(=O)N([C@H]8CCC(=O)NC8=O)CC7=C6)CC5)CC4)C=C2)C=N3)C(OC)=C(NS(=O)(=O)N2CC[C@@H](F)C2)C=C1	C50H55FN8O8S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-YFJKH3	SCHEMBL30253731	(3R)-N-[3-[5-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-dimethoxyphenyl]-3-fluoropyrrolidine-1-sulfonamide	COC1=C(C(=O)C2=CNC3=C2C=C(C2=CC=C(N4CCC(CN5CCC(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)CC5)CC4)C=C2)C=N3)C(OC)=C(NS(=O)(=O)N2CC[C@@H](F)C2)C=C1	C50H55FN8O8S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-NNGDE0	SCHEMBL30254083	(3R)-N-[3-[5-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2-ethyl-4-fluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	CCC1=C(NS(=O)(=O)N2CC[C@@H](F)C2)C=CC(F)=C1C(=O)C1=CNC2=C1C=C(C1=CC=C(N3CCC(CN4CCC(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)CC6=C5)CC4)CC3)C=C1)C=N2	C50H54F2N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-QLS34J	SCHEMBL30253669	(2R,5R)-N-[3-[5-[4-[4-[[4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-2,5-dimethylpyrrolidine-1-sulfonamide	C[C@@H]1CC[C@@H](C)N1S(=O)(=O)NC1=C(F)C(C(=O)C2=CNC3=C2C=C(C2=CC=C(N4CCC(CN5CCC(C6=CC=C7C(=O)N([C@H]8CCC(=O)NC8=O)CC7=C6)CC5)CC4)C=C2)C=N3)=C(F)C=C1	C50H54F2N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-85AREF	SCHEMBL30253880	(3R)-N-[3-[5-[4-[4-[[4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-hydroxypyrrolidine-1-sulfonamide	O=C1CC[C@H](N2CC3=CC(C4CCN(CC5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](O)C8)=C7F)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C48H50F2N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-T8SDM3	SCHEMBL30254068	N-[3-[5-[4-[4-[[4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-hydroxyazetidine-1-sulfonamide	O=C1CC[C@H](N2CC3=CC(C4CCN(CC5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC(O)C8)=C7F)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C47H48F2N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-V408P6	SCHEMBL30253986	3-[2,6-difluoro-3-[[2-hydroxyethyl(methyl)sulfamoyl]amino]benzoyl]-5-[4-[4-[[4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine	CN(CCO)S(=O)(=O)NC1=C(F)C(C(=O)C2=CNC3=C2C=C(C2=CC=C(N4CCC(CN5CCC(C6=CC=C7C(=O)N([C@H]8CCC(=O)NC8=O)CC7=C6)CC5)CC4)C=C2)C=N3)=C(F)C=C1	C47H50F2N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-QLJKDZ	SCHEMBL30253550	3-[3-[[cyclopropyl(methyl)sulfamoyl]amino]-2,6-difluorobenzoyl]-5-[4-[4-[[4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine	CN(C1CC1)S(=O)(=O)NC1=C(F)C(C(=O)C2=CNC3=C2C=C(C2=CC=C(N4CCC(CN5CCC(C6=CC=C7C(=O)N([C@H]8CCC(=O)NC8=O)CC7=C6)CC5)CC4)C=C2)C=N3)=C(F)C=C1	C48H50F2N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-ORU5VG	SCHEMBL30253902	N-[3-[5-[4-[4-[[4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-2-hydroxyethanesulfonamide	O=C1CC[C@H](N2CC3=CC(C4CCN(CC5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)CCO)=C7F)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C46H47F2N7O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-SQLM5B	SCHEMBL30253838	(3R)-N-[3-[5-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-4-fluoro-2-methoxyphenyl]-3-fluoropyrrolidine-1-sulfonamide	COC1=C(NS(=O)(=O)N2CC[C@@H](F)C2)C=CC(F)=C1C(=O)C1=CNC2=C1C=C(C1=CC=C(N3CCC(CN4CCC(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)CC6=C5)CC4)CC3)C=C1)C=N2	C49H52F2N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-8XL0L8	SCHEMBL30254215	(3R)-N-[3-[5-[4-[4-[[4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]-3,5-bis(methylamino)phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	CNC1=CC(C2=CC3=C(N=C2)NC=C3C(=O)C2=C(F)C=CC(NS(=O)(=O)N3CC[C@@H](F)C3)=C2F)=CC(NC)=C1N1CCC(CN2CCC(C3=CC=C4C(=O)N([C@H]5CCC(=O)NC5=O)CC4=C3)CC2)CC1	C50H55F3N10O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-59LC0V	SCHEMBL30253655	(3R)-N-[3-[5-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]-3,5-bis(methylamino)phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	CNC1=CC(C2=CC3=C(N=C2)NC=C3C(=O)C2=C(F)C=CC(NS(=O)(=O)N3CC[C@@H](F)C3)=C2F)=CC(NC)=C1N1CCC(CN2CCC(C3=CC=C4C(=O)N(C5CCC(=O)NC5=O)CC4=C3)CC2)CC1	C50H55F3N10O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-XK3NGK	WO2022047145A1_286	.	O=C1CC[C@@H](N2CC3=C(C=CC(N4CC(CN5CCN(C6(C7=NC=C(C8=CC9=C(N=C8)NC=C9C(=O)C8=C(F)CCC(NS(=O)(=O)N9CC[C@@H](F)C9)=C8F)C=N7)CC6)CC5)C4)=C3)C2=O)C(=O)N1	C46H48F3N11O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-ESE1Z7	SCHEMBL30253608	(3R)-N-[3-[5-[2-[[1-[[1-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperidin-4-yl]-methylamino]pyrimidin-5-yl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	CN(C1=NC=C(C2=CC3=C(N=C2)NC=C3C(=O)C2=C(F)C=CC(NS(=O)(=O)N3CC[C@@H](F)C3)=C2F)C=N1)C1CCN(CC2CCN(C3=CC=C4C(=O)N([C@H]5CCC(=O)NC5=O)CC4=C3)CC2)CC1	C47H50F3N11O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-SAMUV2	SCHEMBL30253876	(3R)-N-[3-[5-[6-[1-[4-[[1-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]cyclopropyl]pyridin-3-yl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CC[C@H](N2CC3=CC(N4CCC(CN5CCN(C6(C7=NC=C(C8=CC9=C(N=C8)NC=C9C(=O)C8=C(F)C=CC(NS(=O)(=O)N9CC[C@@H](F)C9)=C8F)C=C7)CC6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C49H51F3N10O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-IN8SOC	SCHEMBL30253915	(3R)-N-[3-[5-[2-[(1S)-1-[4-[[1-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]ethyl]pyrimidin-5-yl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	C[C@@H](C1=NC=C(C2=CC3=C(N=C2)NC=C3C(=O)C2=C(F)C=CC(NS(=O)(=O)N3CC[C@@H](F)C3)=C2F)C=N1)N1CCN(CC2CCN(C3=CC=C4C(=O)N([C@H]5CCC(=O)NC5=O)CC4=C3)CC2)CC1	C47H50F3N11O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-3SGPJ4	SCHEMBL30253780	(3R)-N-[3-[5-[2-[(1R)-1-[4-[[1-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]ethyl]pyrimidin-5-yl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	C[C@H](C1=NC=C(C2=CC3=C(N=C2)NC=C3C(=O)C2=C(F)C=CC(NS(=O)(=O)N3CC[C@@H](F)C3)=C2F)C=N1)N1CCN(CC2CCN(C3=CC=C4C(=O)N([C@H]5CCC(=O)NC5=O)CC4=C3)CC2)CC1	C47H50F3N11O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-7C5MR4	SCHEMBL30253719	(3R)-N-[3-[5-[4-[4-[[4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-4-fluoro-2-propylphenyl]-3-fluoropyrrolidine-1-sulfonamide	CCCC1=C(C(=O)C2=CNC3=NC=C(C4=CC=C(N5CCC(CN6CCC(C7=CC=C8C(=O)N([C@H]9CCC(=O)NC9=O)CC8=C7)CC6)CC5)C=C4)C=C23)C(F)=CC=C1NS(=O)(=O)N1CC[C@@H](F)C1	C51H56F2N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-QE25XU	SCHEMBL30254262	(3R)-N-[3-[5-[2-[1-[4-[[1-[2-[(3R)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]cyclopropyl]pyrimidin-5-yl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CC[C@@H](N2CC3=CC(N4CCC(CN5CCN(C6(C7=NC=C(C8=CC9=C(N=C8)NC=C9C(=O)C8=C(F)C=CC(NS(=O)(=O)N9CC[C@@H](F)C9)=C8F)C=N7)CC6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C48H50F3N11O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-YMYSXI	SCHEMBL30254000	(3R)-N-[3-[5-[4-[3-[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]azetidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(N4CCC(C5CN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6)C5)CC4)=CC=C3C2=O)C(=O)N1	C45H43F3N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-LB2C9F	SCHEMBL30253855	(3R)-N-[3-[5-[4-[4-[3-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]propoxymethyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=C(C=CC(CCCOCC4CCN(C5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)CC4)=C3)C2=O)C(=O)N1	C46H46F3N7O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-616L3N	WO2022047145A1_297	.	O=C1CCC(N2CC3=CC(C4CCN(C[C@H]5CCN(C6=CC=C(C7=CC8=C(C=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6)C[C@H]5F)CC4)=CC=C3C2=O)C(=O)N1	C49H49F4N7O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-0OZC8O	SCHEMBL30254227	(3R)-N-[3-[5-[4-[6-[(2S)-2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-2-hydroxyethyl]-2,6-diazaspiro[3.3]heptan-2-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC([C@H](O)CN4CC5(C4)CN(C4=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C4)C5)=CC=C3C2=O)C(=O)N1	C44H41F3N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-EFMYCV	SCHEMBL30253866	(3R)-N-[3-[5-[4-[4-[(3S)-3-[2-[(3S)-2,6-dioxopiperidin-3-yl]-6-fluoro-1-oxo-3H-isoindol-5-yl]-3-hydroxypropyl]piperazin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CC[C@H](N2CC3=CC([C@@H](O)CCN4CCN(C5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)CC4)=C(F)C=C3C2=O)C(=O)N1	C44H42F4N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-SASNMO	SCHEMBL30254132	(3R)-N-[3-[5-[4-[4-[(3S)-3-[2-[(3R)-2,6-dioxopiperidin-3-yl]-6-fluoro-1-oxo-3H-isoindol-5-yl]-3-hydroxypropyl]piperazin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CC[C@@H](N2CC3=CC([C@@H](O)CCN4CCN(C5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)CC4)=C(F)C=C3C2=O)C(=O)N1	C44H42F4N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-1IHJF2	SCHEMBL30253873	(3R)-N-[3-[5-[4-[3-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]azetidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(N4CCC(CC5CN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6)C5)CC4)=CC=C3C2=O)C(=O)N1	C46H45F3N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-4E5HLV	SCHEMBL30253945	(3R)-N-[3-[5-[4-[[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]azetidin-3-yl]methyl]piperidin-4-yl]methyl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=C(C=CC(N4CC(CN5CCC(CC6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6)CC5)C4)=C3)C2=O)C(=O)N1	C47H47F3N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-I1OLD5	SCHEMBL24319683	(3R)-N-[3-[5-[4-[1-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]azetidin-3-yl]methyl]piperidin-4-yl]cyclopropyl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide; SCHEMBL30254308	O=C1CCC(N2CC3=C(C=CC(N4CC(CN5CCC(C6(C7=CC=C(C8=CC9=C(N=C8)NC=C9C(=O)C8=C(F)C=CC(NS(=O)(=O)N9CC[C@@H](F)C9)=C8F)C=C7)CC6)CC5)C4)=C3)C2=O)C(=O)N1	C49H49F3N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-YICM0P	SCHEMBL24319682	(3R)-N-[3-[5-[4-[[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]azetidin-3-yl]methyl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide; SCHEMBL30253738	O=C1CCC(N2CC3=C(C=CC(N4CCC(CN5CC(CC6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6)C5)CC4)=C3)C2=O)C(=O)N1	C47H47F3N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-OOZOGO	SCHEMBL30253641	(3R)-N-[3-[5-[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]azetidin-3-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(N4CC(CC5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6)CC5)C4)=CC=C3C2=O)C(=O)N1	C46H45F3N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-JLBIPT	SCHEMBL24319685	(3R)-N-[3-[5-[2-[[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]azetidin-3-yl]methyl]pyrimidin-5-yl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide; SCHEMBL30253753	O=C1CCC(N2CC3=CC(N4CCC(CN5CC(CC6=NC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=N6)C5)CC4)=CC=C3C2=O)C(=O)N1	C45H45F3N10O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-13R7PL	SCHEMBL24319684	(3R)-N-[3-[5-[4-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]ethyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide; SCHEMBL30253778	O=C1CCC(N2CC3=CC(N4CCC(CCC5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C49H51F3N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-4BNQC9	SCHEMBL31302556	(3R)-N-[3-[5-[4-[(3aS,7aS)-5-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]-3,3a,4,6,7,7a-hexahydro-1H-pyrrolo[3,4-c]pyridin-2-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	[H][C@@]12CN(CC3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)CC5=C4)CC3)CC[C@]1([H])CN(C1=CC=C(C3=CC4=C(N=C3)NC=C4C(=O)C3=C(F)C=CC(NS(=O)(=O)N4CC[C@@H](F)C4)=C3F)C=C1)C2	C50H52F3N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-LA9QND	WO2022047145A1_310	.	C=C1CCC(N2CC3=CC(CCCN4CC5(C4)CN(C4=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C4F)C5)=CC=C3C2=O)C(=O)N1	C46H44F4N8O5S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-XNSMPL	SCHEMBL30254029	(3R)-N-[3-[5-[4-[(1R,6R)-3-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]-3,7-diazabicyclo[4.2.0]octan-7-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	[H][C@]12CN(CC3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)CC5=C4)CC3)CC[C@@]1([H])N(C1=CC=C(C3=CC4=C(N=C3)NC=C4C(=O)C3=C(F)C=CC(NS(=O)(=O)N4CC[C@@H](F)C4)=C3F)C=C1)C2	C49H50F3N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-X1RMAK	SCHEMBL30253656	(3R)-N-[3-[5-[4-[(4R)-4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]-2-oxopiperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=C(C=CC(C4CCN(C[C@@H]5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6)C(=O)C5)CC4)=C3)C2=O)C(=O)N1	C48H47F3N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-Y4D30M	SCHEMBL30254035	(3R)-N-[3-[5-[4-[(3aR,7aR)-5-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]-3,3a,4,6,7,7a-hexahydro-1H-pyrrolo[3,4-c]pyridin-2-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	[H][C@@]12CCN(CC3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)CC5=C4)CC3)C[C@]1([H])CN(C1=CC=C(C3=CC4=C(N=C3)NC=C4C(=O)C3=C(F)C=CC(NS(=O)(=O)N4CC[C@@H](F)C4)=C3F)C=C1)C2	C50H52F3N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-AP2RMD	SCHEMBL30253938	(3R)-N-[3-[5-[4-[(4S)-4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]-2-oxopiperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=C(C=CC(C4CCN(C[C@H]5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6)C(=O)C5)CC4)=C3)C2=O)C(=O)N1	C48H47F3N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-JSEIGS	SCHEMBL30253900	(3R)-N-[3-[5-[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]-6,6-difluoro-1,4-diazepan-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(N4CCC(CN5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6)CC(F)(F)C5)CC4)=CC=C3C2=O)C(=O)N1	C48H48F5N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-XLIK41	SCHEMBL30254287	(3R)-N-[3-[5-[4-[1-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]azetidin-3-yl]cyclopropyl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(N4CCC(CN5CC(C6(C7=CC=C(C8=CC9=C(N=C8)NC=C9C(=O)C8=C(F)C=CC(NS(=O)(=O)N9CC[C@@H](F)C9)=C8F)C=C7)CC6)C5)CC4)=CC=C3C2=O)C(=O)N1	C49H49F3N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-T5X3WN	SCHEMBL30253730	(3R)-N-[3-[5-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]butyl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCCCC5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)CC4)=C3)C2=O)C(=O)N1	C45H45F3N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-ZNHRPG	SCHEMBL30253703	(3R)-N-[3-[5-[4-[5-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]pentyl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCCCCC5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)CC4)=C3)C2=O)C(=O)N1	C46H47F3N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-OD3A9R	SCHEMBL30254162	(3R)-N-[3-[5-[4-[6-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]methyl]-2-azaspiro[3.3]heptan-2-yl]-3-fluorophenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(C4CCN(CC5CC6(C5)CN(C5=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C5F)C6)CC4)=CC=C3C2=O)C(=O)N1	C49H48F4N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-ZW01Q7	WO2022047145A1_320	.	O=C1CCC(N2CC3=C(C=CC(N4CC(CN5CCN(C6(C7=NC=C(C8=CC9=C(N=C8)NC=C9C(=O)C8=C(F)C=CC(NS(=O)(=O)N9CC[C@@H](F)C9)=C8F)C=N7)CC6)CC5)C4)=C3)C2=O)C(=O)N=N1	C46H45F3N12O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-71TUL7	SCHEMBL30253910	(3R)-N-[3-[5-[4-[6-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]butyl]-2,6-diazaspiro[3.3]heptan-2-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=C(C=CC(CCCCN4CC5(C4)CN(C4=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C4)C5)=C3)C2=O)C(=O)N1	C46H45F3N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-SGIDT0	SCHEMBL30253862	(3R)-N-[3-[5-[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]-1,4-diazepan-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(N4CCC(CN5CCCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C48H50F3N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-052KAG	SCHEMBL30253950	(3R)-N-[3-[5-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2C(=O)C3=CC=C(C4CCN(CC5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C48H47F3N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-ONPTVB	WO2022047145A1_324	.	O=C1CCC(N2CC3=CC(N4CCCN(CC5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7C(F)=C(NS(=O)(=O)N8CC[C@@H](F)C8)C=CC7F)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C48H52F3N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-QXUAUK	SCHEMBL30253743	(3R)-N-[3-[5-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]butyl]piperazin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=C(C=CC(CCCCN4CCN(C5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)CC4)=C3)C2=O)C(=O)N1	C45H45F3N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-LSI37J	SCHEMBL30254257	(3R)-N-[3-[5-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(C4CCN(C5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C47H47F3N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-HYM7CJ	SCHEMBL30253771	(3R)-N-[3-[5-[4-[6-[(2R)-4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]-2-hydroxybutyl]-2,6-diazaspiro[3.3]heptan-2-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CC[C@H](N2CC3=CC(CC[C@@H](O)CN4CC5(C4)CN(C4=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C4)C5)=CC=C3C2=O)C(=O)N1	C46H45F3N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-AIR98V	SCHEMBL30253925	(3R)-N-[3-[5-[4-[6-[(2R)-4-[2-[(3R)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]-2-hydroxybutyl]-2,6-diazaspiro[3.3]heptan-2-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CC[C@@H](N2CC3=CC(CC[C@@H](O)CN4CC5(C4)CN(C4=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C4)C5)=CC=C3C2=O)C(=O)N1	C46H45F3N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-3RX50N	SCHEMBL30254037	(3R)-N-[3-[5-[4-[(1S,6S)-3-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]-3,7-diazabicyclo[4.2.0]octan-7-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	[H][C@@]12CN(CC3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)CC5=C4)CC3)CC[C@]1([H])N(C1=CC=C(C3=CC4=C(N=C3)NC=C4C(=O)C3=C(F)C=CC(NS(=O)(=O)N4CC[C@@H](F)C4)=C3F)C=C1)C2	C49H50F3N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-BDLPGF	SCHEMBL30253875	(3R)-N-[3-[5-[4-[3-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]azetidin-3-yl]azetidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(N4CCC(CN5CC(C6CN(C7=CC=C(C8=CC9=C(N=C8)NC=C9C(=O)C8=C(F)C=CC(NS(=O)(=O)N9CC[C@@H](F)C9)=C8F)C=C7)C6)C5)CC4)=CC=C3C2=O)C(=O)N1	C49H50F3N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-6EXETQ	SCHEMBL30253831	(3R)-N-[3-[5-[4-[4-[4-[[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-5-yl]oxy]butyl]piperazin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	COC1=CC(OCCCCN2CCN(C3=CC=C(C4=CC5=C(N=C4)NC=C5C(=O)C4=C(F)C=CC(NS(=O)(=O)N5CC[C@@H](F)C5)=C4F)C=C3)CC2)=CC2=C1C(=O)N(C1CCC(=O)NC1=O)C2	C46H47F3N8O8S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-77RIR0	SCHEMBL30253840	(3R)-N-[3-[5-[4-[1-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]butyl]piperidin-4-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=C(C=CC(CCCCN4CCC(C5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)CC4)=C3)C2=O)C(=O)N1	C46H46F3N7O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-GXHQ6J	SCHEMBL30253577	(3R)-N-[3-[5-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-6,6-difluoro-1,4-diazepan-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=CC(N4CCN(CC5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6)CC5)CC(F)(F)C4)=CC=C3C2=O)C(=O)N1	C48H48F5N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-XNC38A	SCHEMBL30254113	(3R)-N-[3-[5-[2-[1-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]azetidin-3-yl]methyl]piperidin-4-yl]cyclopropyl]pyrimidin-5-yl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(N2CC3=C(C=CC(N4CC(CN5CCC(C6(C7=NC=C(C8=CC9=C(N=C8)NC=C9C(=O)C8=C(F)C=CC(NS(=O)(=O)N9CC[C@@H](F)C9)=C8F)C=N7)CC6)CC5)C4)=C3)C2=O)C(=O)N1	C47H47F3N10O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-U3WHPE	SCHEMBL30253948	(3R)-N-[3-[5-[4-[[(3R)-1-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]pyrrolidin-3-yl]methoxy]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide; SCHEMBL30253960	O=C1CC[C@H](N2CC3=CC(N4CC[C@@H](COC5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)C4)=CC=C3C2=O)C(=O)N1	C42H38F3N7O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-16NHP5	SCHEMBL30253642	(3R)-N-[3-[5-[4-[[(3R)-1-[2-[(3R)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]pyrrolidin-3-yl]methoxy]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CC[C@@H](N2CC3=CC(N4CC[C@@H](COC5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)C4)=CC=C3C2=O)C(=O)N1	C42H38F3N7O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-BETOHM	SCHEMBL24319900	(3R)-N-[3-[5-[4-[4-[[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-4-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide; SCHEMBL29482816	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=CC(C3CCN(CC4CCN(C5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)CC4)CC3)=C21	C48H50F3N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-91FITD	SCHEMBL30253761	4-[4-[[4-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]piperazin-1-yl]methyl]piperidin-1-yl]-N-[(3S)-2,6-dioxopiperidin-3-yl]-2-fluorobenzamide	O=C1CC[C@H](NC(=O)C2=CC=C(N3CCC(CN4CCN(C5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)CC4)CC3)C=C2F)C(=O)N1	C46H47F4N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-XX6B1J	SCHEMBL30253899	4-[4-[[4-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]piperazin-1-yl]methyl]piperidin-1-yl]-N-[(3R)-2,6-dioxopiperidin-3-yl]-2-fluorobenzamide	O=C1CC[C@@H](NC(=O)C2=CC=C(N3CCC(CN4CCN(C5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)CC4)CC3)C=C2F)C(=O)N1	C46H47F4N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-VNLZX9	SCHEMBL30254084	4-[4-[[1-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-N-[(3S)-2,6-dioxopiperidin-3-yl]-2-fluorobenzamide	O=C1CC[C@H](NC(=O)C2=CC=C(N3CCN(CC4CCN(C5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)CC4)CC3)C=C2F)C(=O)N1	C46H47F4N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-LEB51Y	SCHEMBL30254003	4-[4-[[1-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-N-[(3R)-2,6-dioxopiperidin-3-yl]-2-fluorobenzamide	O=C1CC[C@@H](NC(=O)C2=CC=C(N3CCN(CC4CCN(C5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)CC4)CC3)C=C2F)C(=O)N1	C46H47F4N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-5HKWJD	SCHEMBL30253555	4-[6-[[1-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]piperidin-4-yl]methyl]-2,6-diazaspiro[3.3]heptan-2-yl]-N-[(3S)-2,6-dioxopiperidin-3-yl]-2-methoxybenzamide	COC1=CC(N2CC3(CN(CC4CCN(C5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)CC4)C3)C2)=CC=C1C(=O)N[C@H]1CCC(=O)NC1=O	C48H50F3N9O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-YH0DBK	SCHEMBL30253683	4-[6-[[1-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]piperidin-4-yl]methyl]-2,6-diazaspiro[3.3]heptan-2-yl]-N-[(3R)-2,6-dioxopiperidin-3-yl]-2-methoxybenzamide	COC1=CC(N2CC3(CN(CC4CCN(C5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)CC4)C3)C2)=CC=C1C(=O)N[C@@H]1CCC(=O)NC1=O	C48H50F3N9O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-MQLJKD	SCHEMBL30253867	5-[6-[[1-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]piperidin-4-yl]methyl]-2,6-diazaspiro[3.3]heptan-2-yl]-N-[(3S)-2,6-dioxopiperidin-3-yl]pyridine-2-carboxamide	O=C1CC[C@H](NC(=O)C2=CC=C(N3CC4(CN(CC5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6)CC5)C4)C3)C=N2)C(=O)N1	C46H47F3N10O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-BKUAK4	SCHEMBL30253666	5-[6-[[1-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]piperidin-4-yl]methyl]-2,6-diazaspiro[3.3]heptan-2-yl]-N-[(3R)-2,6-dioxopiperidin-3-yl]pyridine-2-carboxamide	O=C1CC[C@@H](NC(=O)C2=CC=C(N3CC4(CN(CC5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6)CC5)C4)C3)C=N2)C(=O)N1	C46H47F3N10O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-ZROFP9	SCHEMBL30253695	4-[6-[[1-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]piperidin-4-yl]methyl]-2,6-diazaspiro[3.3]heptan-2-yl]-N-[(3S)-2,6-dioxopiperidin-3-yl]-2-fluoro-6-methoxybenzamide	COC1=C(C(=O)N[C@H]2CCC(=O)NC2=O)C(F)=CC(N2CC3(CN(CC4CCN(C5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)CC4)C3)C2)=C1	C48H49F4N9O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-UCNC54	SCHEMBL30253940	4-[6-[[1-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]piperidin-4-yl]methyl]-2,6-diazaspiro[3.3]heptan-2-yl]-N-(2,6-dioxopiperidin-3-yl)-2-fluoro-6-methoxybenzamide	COC1=C(C(=O)NC2CCC(=O)NC2=O)C(F)=CC(N2CC3(CN(CC4CCN(C5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)CC4)C3)C2)=C1	C48H49F4N9O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-6R4STH	SCHEMBL30253751	4-[4-[4-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]piperazin-1-yl]butoxy]-N-[(3S)-2,6-dioxopiperidin-3-yl]-2-fluorobenzamide	O=C1CC[C@H](NC(=O)C2=CC=C(OCCCCN3CCN(C4=CC=C(C5=CC6=C(N=C5)NC=C6C(=O)C5=C(F)C=CC(NS(=O)(=O)N6CC[C@@H](F)C6)=C5F)C=C4)CC3)C=C2F)C(=O)N1	C44H44F4N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-QWNAVW	SCHEMBL30254190	4-[4-[4-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]piperazin-1-yl]butoxy]-N-(2,6-dioxopiperidin-3-yl)-2-fluorobenzamide	O=C1CCC(NC(=O)C2=CC=C(OCCCCN3CCN(C4=CC=C(C5=CC6=C(N=C5)NC=C6C(=O)C5=C(F)C=CC(NS(=O)(=O)N6CC[C@@H](F)C6)=C5F)C=C4)CC3)C=C2F)C(=O)N1	C44H44F4N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-GO323K	SCHEMBL30253672	4-[6-[[1-[4-[3-[3-[(3,3-difluoropyrrolidin-1-yl)sulfonylamino]-2,6-difluorobenzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]piperidin-4-yl]methyl]-2,6-diazaspiro[3.3]heptan-2-yl]-N-[(3S)-2,6-dioxopiperidin-3-yl]-2-fluorobenzamide	O=C1CC[C@H](NC(=O)C2=CC=C(N3CC4(CN(CC5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CCC(F)(F)C8)=C7F)C=C6)CC5)C4)C3)C=C2F)C(=O)N1	C47H46F5N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-4VCHT2	SCHEMBL30253784	4-[4-[[2-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]-2,6-diazaspiro[3.3]heptan-6-yl]methyl]piperidin-1-yl]-N-[(3S)-2,6-dioxopiperidin-3-yl]-2-methoxybenzamide	COC1=CC(N2CCC(CN3CC4(C3)CN(C3=CC=C(C5=CC6=C(N=C5)NC=C6C(=O)C5=C(F)C=CC(NS(=O)(=O)N6CC[C@@H](F)C6)=C5F)C=C3)C4)CC2)=CC=C1C(=O)N[C@H]1CCC(=O)NC1=O	C48H50F3N9O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-S2I4AZ	SCHEMBL30253783	5-[4-[[2-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]-2,6-diazaspiro[3.3]heptan-6-yl]methyl]piperidin-1-yl]-N-[(3S)-2,6-dioxopiperidin-3-yl]pyridine-2-carboxamide	O=C1CC[C@H](NC(=O)C2=CC=C(N3CCC(CN4CC5(C4)CN(C4=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C4)C5)CC3)C=N2)C(=O)N1	C46H47F3N10O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-MP2Z80	SCHEMBL30253704	5-[4-[[2-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]-2,6-diazaspiro[3.3]heptan-6-yl]methyl]piperidin-1-yl]-N-(2,6-dioxopiperidin-3-yl)pyridine-2-carboxamide	O=C1CCC(NC(=O)C2=CC=C(N3CCC(CN4CC5(C4)CN(C4=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C4)C5)CC3)C=N2)C(=O)N1	C46H47F3N10O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-DUSYPM	SCHEMBL30253746	4-[3-[2-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]-2,6-diazaspiro[3.3]heptan-6-yl]propyl]-N-[(3S)-2,6-dioxopiperidin-3-yl]-2-fluorobenzamide	O=C1CC[C@H](NC(=O)C2=CC=C(CCCN3CC4(C3)CN(C3=CC=C(C5=CC6=C(N=C5)NC=C6C(=O)C5=C(F)C=CC(NS(=O)(=O)N6CC[C@@H](F)C6)=C5F)C=C3)C4)C=C2F)C(=O)N1	C44H42F4N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-7QHY0Y	SCHEMBL30253747	4-[3-[2-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]-2,6-diazaspiro[3.3]heptan-6-yl]propyl]-N-(2,6-dioxopiperidin-3-yl)-2-fluorobenzamide	O=C1CCC(NC(=O)C2=CC=C(CCCN3CC4(C3)CN(C3=CC=C(C5=CC6=C(N=C5)NC=C6C(=O)C5=C(F)C=CC(NS(=O)(=O)N6CC[C@@H](F)C6)=C5F)C=C3)C4)C=C2F)C(=O)N1	C44H42F4N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-3GEQE5	SCHEMBL30254088	4-[4-[[4-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]piperazin-1-yl]methyl]piperidin-1-yl]-N-[(3S)-2,6-dioxopiperidin-3-yl]-2-methoxybenzamide	COC1=CC(N2CCC(CN3CCN(C4=CC=C(C5=CC6=C(N=C5)NC=C6C(=O)C5=C(F)C=CC(NS(=O)(=O)N6CC[C@@H](F)C6)=C5F)C=C4)CC3)CC2)=CC=C1C(=O)N[C@H]1CCC(=O)NC1=O	C47H50F3N9O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-5AGC1M	SCHEMBL30253969	4-[4-[[4-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]piperazin-1-yl]methyl]piperidin-1-yl]-N-(2,6-dioxopiperidin-3-yl)-2-methoxybenzamide	COC1=CC(N2CCC(CN3CCN(C4=CC=C(C5=CC6=C(N=C5)NC=C6C(=O)C5=C(F)C=CC(NS(=O)(=O)N6CC[C@@H](F)C6)=C5F)C=C4)CC3)CC2)=CC=C1C(=O)NC1CCC(=O)NC1=O	C47H50F3N9O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-LWVJXI	SCHEMBL30253859	4-[4-[[1-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-N-[(3S)-2,6-dioxopiperidin-3-yl]-2-methoxybenzamide	COC1=CC(N2CCN(CC3CCN(C4=CC=C(C5=CC6=C(N=C5)NC=C6C(=O)C5=C(F)C=CC(NS(=O)(=O)N6CC[C@@H](F)C6)=C5F)C=C4)CC3)CC2)=CC=C1C(=O)N[C@H]1CCC(=O)NC1=O	C47H50F3N9O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-C7WDFY	SCHEMBL21934201	4-[4-[[1-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-N-(2,6-dioxopiperidin-3-yl)-2-methoxybenzamide; SCHEMBL30253600	COC1=CC(N2CCN(CC3CCN(C4=CC=C(C5=CC6=C(N=C5)NC=C6C(=O)C5=C(F)C=CC(NS(=O)(=O)N6CC[C@@H](F)C6)=C5F)C=C4)CC3)CC2)=CC=C1C(=O)NC1CCC(=O)NC1=O	C47H50F3N9O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-ME1ITT	SCHEMBL30253996	4-[6-[2-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]ethyl]-2,6-diazaspiro[3.3]heptan-2-yl]-N-[(3S)-2,6-dioxopiperidin-3-yl]-2-methoxybenzamide	COC1=C(C(=O)N[C@H]2CCC(=O)NC2=O)C=CC(N2CC3(CN(CCC4=CC=C(C5=CC6=C(N=C5)NC=C6C(=O)C5=C(F)C=CC(NS(=O)(=O)N6CC[C@@H](F)C6)=C5F)C=C4)C3)C2)=C1	C44H43F3N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-VDZZ1Z	SCHEMBL30253676	4-[6-[2-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]ethyl]-2,6-diazaspiro[3.3]heptan-2-yl]-N-(2,6-dioxopiperidin-3-yl)-2-methoxybenzamide	COC1=C(C(=O)NC2CCC(=O)NC2=O)C=CC(N2CC3(CN(CCC4=CC=C(C5=CC6=C(N=C5)NC=C6C(=O)C5=C(F)C=CC(NS(=O)(=O)N6CC[C@@H](F)C6)=C5F)C=C4)C3)C2)=C1	C44H43F3N8O7S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-ULQMWB	SCHEMBL30254077	4-[6-[[1-[4-[3-(3-amino-2,6-difluorobenzoyl)-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]piperidin-4-yl]methyl]-2,6-diazaspiro[3.3]heptan-2-yl]-N-[(3S)-2,6-dioxopiperidin-3-yl]-2-fluorobenzamide	NC1=C(F)C(C(=O)C2=CNC3=C2C=C(C2=CC=C(N4CCC(CN5CC6(C5)CN(C5=CC=C(C(=O)N[C@H]7CCC(=O)NC7=O)C(F)=C5)C6)CC4)C=C2)C=N3)=C(F)C=C1	C43H41F3N8O4	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-O518GP	SCHEMBL30253824	5-[1-[[1-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]piperidin-4-yl]methyl]piperidin-4-yl]-N-(2,6-dioxopiperidin-3-yl)-3,4-dihydro-2H-1,8-naphthyridine-1-carboxamide	O=C1CCC(NC(=O)N2CCCC3=C2N=CC=C3C2CCN(CC3CCN(C4=CC=C(C5=CC6=C(N=C5)NC=C6C(=O)C5=C(F)C=CC(NS(=O)(=O)N6CC[C@@H](F)C6)=C5F)C=C4)CC3)CC2)C(=O)N1	C49H53F3N10O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-4I8S3I	SCHEMBL30253763	(3R)-N-[3-[5-[4-[4-[[4-[6-(2,6-dioxopiperidin-3-yl)pyridin-3-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(C2=NC=C(C3CCN(CC4CCN(C5=CC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)CC4)CC3)C=C2)C(=O)N1	C45H47F3N8O5S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-HWN2RM	SCHEMBL30254053	5-[1-[[1-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]piperidin-4-yl]methyl]piperidin-4-yl]-N-[(3S)-2,6-dioxopiperidin-3-yl]-3,4-dihydro-2H-1,8-naphthyridine-1-carboxamide	O=C1CC[C@H](NC(=O)N2CCCC3=C2N=CC=C3C2CCN(CC3CCN(C4=CC=C(C5=CC6=C(N=C5)NC=C6C(=O)C5=C(F)C=CC(NS(=O)(=O)N6CC[C@@H](F)C6)=C5F)C=C4)CC3)CC2)C(=O)N1	C49H53F3N10O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-CQ8VMU	SCHEMBL30253733	5-[1-[[1-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]piperidin-4-yl]methyl]piperidin-4-yl]-N-[(3R)-2,6-dioxopiperidin-3-yl]-3,4-dihydro-2H-1,8-naphthyridine-1-carboxamide	O=C1CC[C@@H](NC(=O)N2CCCC3=C2N=CC=C3C2CCN(CC3CCN(C4=CC=C(C5=CC6=C(N=C5)NC=C6C(=O)C5=C(F)C=CC(NS(=O)(=O)N6CC[C@@H](F)C6)=C5F)C=C4)CC3)CC2)C(=O)N1	C49H53F3N10O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-6E1MXC	SCHEMBL30254046	(3R)-N-[3-[5-[4-[4-[[2-[4-(2,6-dioxopiperidin-3-yl)phenyl]-2,6-diazaspiro[3.3]heptan-6-yl]methyl]piperidin-1-yl]phenyl]-1H-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]-3-fluoropyrrolidine-1-sulfonamide	O=C1CCC(C2=CC=C(N3CC4(CN(CC5CCN(C6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6)CC5)C4)C3)C=C2)C(=O)N1	C46H47F3N8O5S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-V8EC5M	SCHEMBL30253545	5-[4-[[1-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-N-[(3S)-2,6-dioxopiperidin-3-yl]-3,4-dihydro-2H-1,8-naphthyridine-1-carboxamide	O=C1CC[C@H](NC(=O)N2CCCC3=C2N=CC=C3N2CCN(CC3CCN(C4=CC=C(C5=CC6=C(N=C5)NC=C6C(=O)C5=C(F)C=CC(NS(=O)(=O)N6CC[C@@H](F)C6)=C5F)C=C4)CC3)CC2)C(=O)N1	C48H52F3N11O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-AWN2UO	SCHEMBL21934200	5-[4-[[1-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-N-(2,6-dioxopiperidin-3-yl)-3,4-dihydro-2H-1,8-naphthyridine-1-carboxamide; SCHEMBL30253799	O=C1CCC(NC(=O)N2CCCC3=C2N=CC=C3N2CCN(CC3CCN(C4=CC=C(C5=CC6=C(N=C5)NC=C6C(=O)C5=C(F)C=CC(NS(=O)(=O)N6CC[C@@H](F)C6)=C5F)C=C4)CC3)CC2)C(=O)N1	C48H52F3N11O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-CQI7QA	SCHEMBL30254007	5-[4-[[4-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]piperazin-1-yl]methyl]piperidin-1-yl]-N-[(3S)-2,6-dioxopiperidin-3-yl]-3,4-dihydro-2H-1,8-naphthyridine-1-carboxamide	O=C1CC[C@H](NC(=O)N2CCCC3=C2N=CC=C3N2CCC(CN3CCN(C4=CC=C(C5=CC6=C(N=C5)NC=C6C(=O)C5=C(F)C=CC(NS(=O)(=O)N6CC[C@@H](F)C6)=C5F)C=C4)CC3)CC2)C(=O)N1	C48H52F3N11O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-Q36QLA	SCHEMBL30253939	5-[4-[[4-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]piperazin-1-yl]methyl]piperidin-1-yl]-N-[(3R)-2,6-dioxopiperidin-3-yl]-3,4-dihydro-2H-1,8-naphthyridine-1-carboxamide	O=C1CC[C@@H](NC(=O)N2CCCC3=C2N=CC=C3N2CCC(CN3CCN(C4=CC=C(C5=CC6=C(N=C5)NC=C6C(=O)C5=C(F)C=CC(NS(=O)(=O)N6CC[C@@H](F)C6)=C5F)C=C4)CC3)CC2)C(=O)N1	C48H52F3N11O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-E2SOBR	WO2022047145A1_373	.	CC1=C(C(=O)C2=CNC3=C2C=C(C2=CC=C(CCN4CC5(C4)CN(C4=CC(F)=C(C(=O)N[C@H]6CCC(=O)NC6=O)C=C4)C5)C=C2)C=N3)C(F)=C(NS(=O)(=O)N2CC[C@@H](F)C2)C=C1	C44H43F3N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-9BCCJH	WO2022047145A1_374	.	CC1=C(C(=O)C2=CNC3=C2C=C(C2=CC=C(CCN4CC5(C4)CN(C4=CC(F)=C(C(=O)NC6CCC(=O)NC6=O)C=C4)C5)C=C2)C=N3)C(F)=C(NS(=O)(=O)N2CC[C@@H](F)C2)C=C1	C44H43F3N8O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-D26O26	SCHEMBL30253714	4-[1-[[1-[5-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]pyrimidin-2-yl]piperidin-4-yl]methyl]piperidin-4-yl]-N-[(3S)-2,6-dioxopiperidin-3-yl]-2-fluorobenzamide	O=C1CC[C@H](NC(=O)C2=C(F)C=C(C3CCN(CC4CCN(C5=NC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=N5)CC4)CC3)C=C2)C(=O)N1	C45H46F4N10O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-2UW5CV	SCHEMBL30254210	4-[1-[[1-[5-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]pyrimidin-2-yl]piperidin-4-yl]methyl]piperidin-4-yl]-N-(2,6-dioxopiperidin-3-yl)-2-fluorobenzamide	O=C1CCC(NC(=O)C2=C(F)C=C(C3CCN(CC4CCN(C5=NC=C(C6=CC7=C(N=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=N5)CC4)CC3)C=C2)C(=O)N1	C45H46F4N10O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-4JACEK	WO2022047145A1_377	.	O=C1CC[C@H](NC(=O)C2=C(F)C=C(N3CCN(CCN4CCN(C5=CC=C(C6=CC7=C(C=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)CC4)CC3)C=C2)C(=O)N1	C47H49F4N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-YWWZD7	WO2022047145A1_378	.	O=C1CCC(NC(=O)C2=C(F)C=C(N3CCN(CCN4CCN(C5=CC=C(C6=CC7=C(C=C6)NC=C7C(=O)C6=C(F)C=CC(NS(=O)(=O)N7CC[C@@H](F)C7)=C6F)C=C5)CC4)CC3)C=C2)C(=O)N1	C47H49F4N9O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-S91991	SCHEMBL30254117	5-[6-[2-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]ethyl]-2,6-diazaspiro[3.3]heptan-2-yl]-N-[(3S)-2,6-dioxopiperidin-3-yl]-3,4-dihydro-2H-1,8-naphthyridine-1-carboxamide	O=C1CC[C@H](NC(=O)N2CCCC3=C(N4CC5(CN(CCC6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6)C5)C4)C=CN=C32)C(=O)N1	C45H45F3N10O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-56YKDG	SCHEMBL30253680	5-[6-[2-[4-[3-[2,6-difluoro-3-[[(3R)-3-fluoropyrrolidin-1-yl]sulfonylamino]benzoyl]-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]ethyl]-2,6-diazaspiro[3.3]heptan-2-yl]-N-[(3R)-2,6-dioxopiperidin-3-yl]-3,4-dihydro-2H-1,8-naphthyridine-1-carboxamide	O=C1CC[C@@H](NC(=O)N2CCCC3=C(N4CC5(CN(CCC6=CC=C(C7=CC8=C(N=C7)NC=C8C(=O)C7=C(F)C=CC(NS(=O)(=O)N8CC[C@@H](F)C8)=C7F)C=C6)C5)C4)C=CN=C32)C(=O)N1	C45H45F3N10O6S	BRAF	P15056	CRBN	WO-2022047145-A1
TPD-5NA8Y9	Protac lzk-IN-1	PROTAC LZK-IN-1; orb2945715; SCHEMBL24278009; HY-170595; 2763268-64-8	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCC(=O)N2CCC(c3cc(Nc4cc(C#N)ccn4)nc(N4CCC(F)(F)C4)c3)CC2)C(C)(C)C)cc1	C51H64F2N10O5S	LZK	O43283	VHL	WO-2022051326-A1
TPD-S1FAOQ	SCHEMBL24278063	(2S,4R)-1-[(2S)-2-[[8-[4-[2-(3,3-difluoropyrrolidin-1-yl)-6-[[4-(trifluoromethyl)pyridin-2-yl]amino]pyridin-4-yl]piperidin-1-yl]-8-oxooctanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCC(=O)N2CCC(c3cc(Nc4cc(C(F)(F)F)ccn4)nc(N4CCC(F)(F)C4)c3)CC2)C(C)(C)C)cc1	C51H64F5N9O5S	LZK	O43283	VHL	WO-2022051326-A1
TPD-RVK6E1	SCHEMBL24278000	8-[4-[2-(3,3-difluoropyrrolidin-1-yl)-6-[[4-(trifluoromethyl)pyridin-2-yl]amino]pyridin-4-yl]piperidin-1-yl]-N-[4-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]acetyl]amino]butyl]-8-oxooctanamide	O=C(CCCCCCC(=O)N1CCC(c2cc(Nc3cc(C(F)(F)F)ccn3)nc(N3CCC(F)(F)C3)c2)CC1)NCCCCNC(=O)CNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O	C47H55F5N10O7	LZK	O43283	CRBN	WO-2022051326-A1
TPD-YTN256	SCHEMBL24278001	8-[4-[2-[(4-cyanopyridin-2-yl)amino]-6-(3,3-difluoropyrrolidin-1-yl)pyridin-4-yl]piperidin-1-yl]-N-[4-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]acetyl]amino]butyl]-8-oxooctanamide	N#Cc1ccnc(Nc2cc(C3CCN(C(=O)CCCCCCC(=O)NCCCCNC(=O)CNc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)cc(N3CCC(F)(F)C3)n2)c1	C47H55F2N11O7	LZK	O43283	CRBN	WO-2022051326-A1
TPD-O37VON	SCHEMBL24278012	5-[4-[2-[(4-cyanopyridin-2-yl)amino]-6-(3,3-difluoropyrrolidin-1-yl)pyridin-4-yl]piperidine-1-carbonyl]-N-[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]pyridine-3-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)c2cncc(C(=O)N3CCC(c4cc(Nc5cc(C#N)ccn5)nc(N5CCC(F)(F)C5)c4)CC3)c2)C(C)(C)C)cc1	C50H55F2N11O5S	LZK	O43283	VHL	WO-2022051326-A1
TPD-OWV711	SCHEMBL24278166	5-[4-[2-[(4-cyanopyridin-2-yl)amino]-6-(3,3-difluoropyrrolidin-1-yl)pyridin-4-yl]piperidine-1-carbonyl]-N-[4-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]acetyl]amino]butyl]pyridine-3-carboxamide	N#Cc1ccnc(Nc2cc(C3CCN(C(=O)c4cncc(C(=O)NCCCCNC(=O)CNc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6=O)c4)CC3)cc(N3CCC(F)(F)C3)n2)c1	C46H46F2N12O7	LZK	O43283	CRBN	WO-2022051326-A1
TPD-Z2O13V	SCHEMBL24278047	(2S,4R)-1-[(2S)-2-[[6-[[4-[2-[(4-cyanopyridin-2-yl)amino]-6-(3,3-difluoropyrrolidin-1-yl)pyridin-4-yl]piperidin-1-yl]methyl]pyridin-2-yl]methylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NCc2cccc(CN3CCC(c4cc(Nc5cc(C#N)ccn5)nc(N5CCC(F)(F)C5)c4)CC3)n2)C(C)(C)C)cc1	C50H59F2N11O3S	LZK	O43283	VHL	WO-2022051326-A1
TPD-WYHK0Z	SCHEMBL24278195	(2S,4R)-1-[(2S)-2-[[10-[4-[2-[(4-cyanopyridin-2-yl)amino]-6-(3,3-difluoropyrrolidin-1-yl)pyridin-4-yl]piperidin-1-yl]-10-oxodecanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCCCC(=O)N2CCC(c3cc(Nc4cc(C#N)ccn4)nc(N4CCC(F)(F)C4)c3)CC2)C(C)(C)C)cc1	C53H68F2N10O5S	LZK	O43283	VHL	WO-2022051326-A1
TPD-YHMZIR	SCHEMBL24278196	(2S,4R)-1-[(2S)-2-[[12-[4-[2-[(4-cyanopyridin-2-yl)amino]-6-(3,3-difluoropyrrolidin-1-yl)pyridin-4-yl]piperidin-1-yl]-12-oxododecanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCCCCCC(=O)N2CCC(c3cc(Nc4cc(C#N)ccn4)nc(N4CCC(F)(F)C4)c3)CC2)C(C)(C)C)cc1	C55H72F2N10O5S	LZK	O43283	VHL	WO-2022051326-A1
TPD-SDJPIZ	SCHEMBL24278008	(2S,4R)-1-[(2S)-2-[[6-[4-[2-[(4-cyanopyridin-2-yl)amino]-6-(3,3-difluoropyrrolidin-1-yl)pyridin-4-yl]piperidin-1-yl]-6-oxohexanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCC(=O)N2CCC(c3cc(Nc4cc(C#N)ccn4)nc(N4CCC(F)(F)C4)c3)CC2)C(C)(C)C)cc1	C49H60F2N10O5S	LZK	O43283	VHL	WO-2022051326-A1
TPD-ZQOZFE	SCHEMBL24278564	(2S,4R)-1-[(2S)-2-[[4-[4-[2-[(4-cyanopyridin-2-yl)amino]-6-(3,3-difluoropyrrolidin-1-yl)pyridin-4-yl]piperidine-1-carbonyl]phenyl]methylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NCc2ccc(C(=O)N3CCC(c4cc(Nc5cc(C#N)ccn5)nc(N5CCC(F)(F)C5)c4)CC3)cc2)C(C)(C)C)cc1	C51H58F2N10O4S	LZK	O43283	VHL	WO-2022051326-A1
TPD-K3M6TE	SCHEMBL24278592	(2S,4R)-1-[(2S)-2-[[4-[4-[2-[(4-cyanopyridin-2-yl)amino]-6-(3,3-difluoropyrrolidin-1-yl)pyridin-4-yl]piperidin-1-yl]-4-oxobutanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCC(=O)N2CCC(c3cc(Nc4cc(C#N)ccn4)nc(N4CCC(F)(F)C4)c3)CC2)C(C)(C)C)cc1	C47H56F2N10O5S	LZK	O43283	VHL	WO-2022051326-A1
TPD-3IJGT9	SCHEMBL24278088	(2S,4R)-1-[(2S)-2-[[4-[4-[2-[(4-cyanopyridin-2-yl)amino]-6-(3,3-difluoropyrrolidin-1-yl)pyridin-4-yl]piperidine-1-carbonyl]benzoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)c2ccc(C(=O)N3CCC(c4cc(Nc5cc(C#N)ccn5)nc(N5CCC(F)(F)C5)c4)CC3)cc2)C(C)(C)C)cc1	C51H56F2N10O5S	LZK	O43283	VHL	WO-2022051326-A1
TPD-NSJ3TK	SCHEMBL24278539	(2S,4R)-1-[(2S)-2-[[2-[[4-[4-[2-[(4-cyanopyridin-2-yl)amino]-6-(3,3-difluoropyrrolidin-1-yl)pyridin-4-yl]piperidin-1-yl]-4-oxobutanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C(CCCNC(=N)N)NC(=O)CCC(=O)N2CCC(c3cc(Nc4cc(C#N)ccn4)nc(N4CCC(F)(F)C4)c3)CC2)C(C)(C)C)cc1	C53H68F2N14O6S	LZK	O43283	VHL	WO-2022051326-A1
TPD-2770NX	WO2022051326A1_17	(2S,4R)-1-[(2S)-2-[[2-[[2-[[4-[4-[2-[(4-cyanopyridin-2-yl)amino]-6-(3,3-difluoropyrrolidin-1-yl)pyridin-4-yl]piperidin-1-yl]-4-oxobutanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C(CCCNC(=N)N)NC(=O)C(CCCNC(=N)N)NC(=O)CCC(=O)N2CCC(c3cc(Nc4cc(C#N)ccn4)nc(N4CCC(F)(F)C4)c3)CC2)C(C)(C)C)cc1	C59H80F2N18O7S	LZK	O43283	VHL	WO-2022051326-A1
TPD-EC18K1	SCHEMBL24278149	(2S,4R)-1-[(2S)-2-[[3-[4-[2-[(4-cyanopyridin-2-yl)amino]-6-(3,3-difluoropyrrolidin-1-yl)pyridin-4-yl]piperidine-1-carbonyl]phenyl]methylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NCc2cccc(C(=O)N3CCC(c4cc(Nc5cc(C#N)ccn5)nc(N5CCC(F)(F)C5)c4)CC3)c2)C(C)(C)C)cc1	C51H58F2N10O4S	LZK	O43283	VHL	WO-2022051326-A1
TPD-7B1BHB	SCHEMBL24278057	(2S,4R)-1-[(2S)-2-[[3-[4-[2-[(4-cyanopyridin-2-yl)amino]-6-(3,3-difluoropyrrolidin-1-yl)pyridin-4-yl]piperidine-1-carbonyl]benzoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)c2cccc(C(=O)N3CCC(c4cc(Nc5cc(C#N)ccn5)nc(N5CCC(F)(F)C5)c4)CC3)c2)C(C)(C)C)cc1	C51H56F2N10O5S	LZK	O43283	VHL	WO-2022051326-A1
TPD-I9AKDX	SCHEMBL24278146	6-[4-[2-[(4-cyanopyridin-2-yl)amino]-6-(3,3-difluoropyrrolidin-1-yl)pyridin-4-yl]piperidine-1-carbonyl]-N-[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]pyrimidine-4-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)c2cc(C(=O)N3CCC(c4cc(Nc5cc(C#N)ccn5)nc(N5CCC(F)(F)C5)c4)CC3)ncn2)C(C)(C)C)cc1	C49H54F2N12O5S	LZK	O43283	VHL	WO-2022051326-A1
TPD-W39JU8	SCHEMBL24278100	6-[4-[2-[(4-cyanopyridin-2-yl)amino]-6-(3,3-difluoropyrrolidin-1-yl)pyridin-4-yl]piperidine-1-carbonyl]-N-[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]pyridazine-3-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)c2ccc(C(=O)N3CCC(c4cc(Nc5cc(C#N)ccn5)nc(N5CCC(F)(F)C5)c4)CC3)nn2)C(C)(C)C)cc1	C49H54F2N12O5S	LZK	O43283	VHL	WO-2022051326-A1
TPD-FE5CSH	SCHEMBL24278055	6-[4-[2-[(4-cyanopyridin-2-yl)amino]-6-(3,3-difluoropyrrolidin-1-yl)pyridin-4-yl]piperidine-1-carbonyl]-N-[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]pyrazine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)c2cncc(C(=O)N3CCC(c4cc(Nc5cc(C#N)ccn5)nc(N5CCC(F)(F)C5)c4)CC3)n2)C(C)(C)C)cc1	C49H54F2N12O5S	LZK	O43283	VHL	WO-2022051326-A1
TPD-KHL9AA	SCHEMBL24278036	5-[4-[2-[(4-cyanopyridin-2-yl)amino]-6-(3,3-difluoropyrrolidin-1-yl)pyridin-4-yl]piperidine-1-carbonyl]-N-[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]pyrazine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)c2cnc(C(=O)N3CCC(c4cc(Nc5cc(C#N)ccn5)nc(N5CCC(F)(F)C5)c4)CC3)cn2)C(C)(C)C)cc1	C49H54F2N12O5S	LZK	O43283	VHL	WO-2022051326-A1
TPD-YGX9Q6	SCHEMBL24278148	(2S)-1-[(2S)-2-[[3-[4-[2-[(4-cyanopyridin-2-yl)amino]-6-(3,3-difluoropyrrolidin-1-yl)pyridin-4-yl]piperidine-1-carbonyl]cyclobutanecarbonyl]amino]-3,3-dimethylbutanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2CCCN2C(=O)[C@@H](NC(=O)[C@H]2C[C@H](C(=O)N3CCC(c4cc(Nc5cc(C#N)ccn5)nc(N5CCC(F)(F)C5)c4)CC3)C2)C(C)(C)C)cc1	C49H58F2N10O4S	LZK	O43283	VHL	WO-2022051326-A1
TPD-IA74PM	SCHEMBL24278045	(2S,4R)-1-[(2S)-2-[[(1S,2S)-2-[4-[2-[(4-cyanopyridin-2-yl)amino]-6-(3,3-difluoropyrrolidin-1-yl)pyridin-4-yl]piperidine-1-carbonyl]cyclobutanecarbonyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)[C@H]2CC[C@@H]2C(=O)N2CCC(c3cc(Nc4cc(C#N)ccn4)nc(N4CCC(F)(F)C4)c3)CC2)C(C)(C)C)cc1	C49H58F2N10O5S	LZK	O43283	VHL	WO-2022051326-A1
TPD-4ZSVRK	SCHEMBL24278117	(2S,4R)-1-[(2S)-2-[[(2R)-2-[4-[2-[(4-cyanopyridin-2-yl)amino]-6-(3,3-difluoropyrrolidin-1-yl)pyridin-4-yl]piperidine-1-carbonyl]cyclobutanecarbonyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CC[C@H]2C(=O)N2CCC(c3cc(Nc4cc(C#N)ccn4)nc(N4CCC(F)(F)C4)c3)CC2)C(C)(C)C)cc1	C49H58F2N10O5S	LZK	O43283	VHL	WO-2022051326-A1
TPD-TAES79	SCHEMBL24282124	4-[2-[(4-cyanopyridin-2-yl)amino]-6-(3,3-difluoropyrrolidin-1-yl)pyridin-4-yl]-N-[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]piperidine-1-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)N2CCC(c3cc(Nc4cc(C#N)ccn4)nc(N4CCC(F)(F)C4)c3)CC2)C(C)(C)C)cc1	C44H52F2N10O4S	LZK	O43283	VHL	WO-2022051326-A1
TPD-SVBN6H	WO2022051326A1_28	(2S,4R)-1-[(2S)-2-[[2-[4-[2-[(4-cyanopyridin-2-yl)amino]-6-(3,3-difluoropyrrolidin-1-yl)pyridin-4-yl]piperidin-1-yl]-2-oxoethyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NCC(=O)N2CCC(c3cc(Nc4cc(C#N)ccn4)nc(N4CCC(F)(F)C4)c3)CC2)C(C)(C)C)cc1	C45H54F2N10O4S	LZK	O43283	VHL	WO-2022051326-A1
TPD-5Q6MZY	WO2022051326A1_29	(2S,4R)-1-[(2S)-2-[[(2S)-2-[[2-amino-5-(diaminomethylideneamino)pentanoyl]amino]-5-[4-[2-[(4-cyanopyridin-2-yl)amino]-6-(3,3-difluoropyrrolidin-1-yl)pyridin-4-yl]piperidin-1-yl]-5-oxopentanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)[C@H](CCC(=O)N2CCC(c3cc(Nc4cc(C#N)ccn4)nc(N4CCC(F)(F)C4)c3)CC2)NC(=O)C(N)CCCNC(=N)N)C(C)(C)C)cc1	C54H71F2N15O6S	LZK	O43283	VHL	WO-2022051326-A1
TPD-QOFLI5	SCHEMBL24278122	tert-butyl N-[(2S)-1-[[(1S)-2-[(2S,4S)-4-[[8-[4-[2-[(4-cyanopyridin-2-yl)amino]-6-(3,3-difluoropyrrolidin-1-yl)pyridin-4-yl]piperidin-1-yl]-8-oxooctanoyl]amino]-2-[[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]carbamoyl]pyrrolidin-1-yl]-1-cyclohexyl-2-oxoethyl]amino]-1-oxopropan-2-yl]-N-methylcarbamate	C[C@@H](C(=O)N[C@H](C(=O)N1C[C@@H](NC(=O)CCCCCCC(=O)N2CCC(c3cc(Nc4cc(C#N)ccn4)nc(N4CCC(F)(F)C4)c3)CC2)C[C@H]1C(=O)N[C@@H]1CCCc2ccccc21)C1CCCCC1)N(C)C(=O)OC(C)(C)C	C60H81F2N11O7	LZK	O43283	VHL	WO-2022051326-A1
TPD-SE290N	SCHEMBL24278119	2-[4-[(4R,5S)-4,5-bis(4-chlorophenyl)-2-(4-methoxy-2-propan-2-yloxyphenyl)-4,5-dihydroimidazole-1-carbonyl]-2-oxopiperazin-1-yl]-N-[6-[4-[2-[(4-cyanopyridin-2-yl)amino]-6-(3,3-difluoropyrrolidin-1-yl)pyridin-4-yl]piperidin-1-yl]-6-oxohexyl]acetamide	COc1ccc(C2=N[C@H](c3ccc(Cl)cc3)[C@H](c3ccc(Cl)cc3)N2C(=O)N2CCN(CC(=O)NCCCCCC(=O)N3CCC(c4cc(Nc5cc(C#N)ccn5)nc(N5CCC(F)(F)C5)c4)CC3)C(=O)C2)c(OC(C)C)c1	C58H63Cl2F2N11O6	LZK	O43283	VHL	WO-2022051326-A1
TPD-QZP811	WO2022051326A1_32	.	Cc1ncsc1-c1ccc([C@@H](C)NC(=O)[C@H]2C[C@H](O)CN2C(=O)[C@H](NC(=O)CCCCCCCCCCCC(=O)NC23CC(n4cc(-c5cnc(N)c(OC(F)(F)F)c5)nc4C(O)C(C)C)(C2)C3)C(C)(C)C)cc1	C54H74F3N9O7S	LZK	O43283	VHL	WO-2022051326-A1
TPD-BBJT0G	SCHEMBL24278072	(2S,4R)-N-[[2-[4-[[4-[4-[2-[(4-cyanopyridin-2-yl)amino]-6-(3,3-difluoropyrrolidin-1-yl)pyridin-4-yl]piperidin-1-yl]-4-oxobutanoyl]amino]butoxy]-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-1-[(2S)-2-[(1-fluorocyclopropanecarbonyl)amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)C)c(OCCCCNC(=O)CCC(=O)N2CCC(c3cc(Nc4cc(C#N)ccn4)nc(N4CCC(F)(F)C4)c3)CC2)c1	C54H66F3N11O7S	LZK	O43283	VHL	WO-2022051326-A1
TPD-X6GXEJ	SCHEMBL24282183	(2S,4R)-1-[(2S)-2-[[3-[4-[2-(3,3-difluoropyrrolidin-1-yl)-6-(pyrazin-2-ylamino)pyridin-4-yl]piperidine-1-carbonyl]cyclobutanecarbonyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)[C@H]2C[C@H](C(=O)N3CCC(c4cc(Nc5cnccn5)nc(N5CCC(F)(F)C5)c4)CC3)C2)C(C)(C)C)cc1	C47H58F2N10O5S	LZK	O43283	VHL	WO-2022051326-A1
TPD-RYO35A	SCHEMBL24278136	5-[4-[2-(3,3-difluoropyrrolidin-1-yl)-6-(pyrazin-2-ylamino)pyridin-4-yl]piperidine-1-carbonyl]-N-[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]pyrazine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)c2cnc(C(=O)N3CCC(c4cc(Nc5cnccn5)nc(N5CCC(F)(F)C5)c4)CC3)cn2)C(C)(C)C)cc1	C47H54F2N12O5S	LZK	O43283	VHL	WO-2022051326-A1
TPD-P93K4Q	SCHEMBL24278061	(2S,4R)-1-[(2S)-2-[[8-[4-[2-(3,3-difluoropyrrolidin-1-yl)-6-(pyrazin-2-ylamino)pyridin-4-yl]piperidin-1-yl]-8-oxooctanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCC(=O)N2CCC(c3cc(Nc4cnccn4)nc(N4CCC(F)(F)C4)c3)CC2)C(C)(C)C)cc1	C49H64F2N10O5S	LZK	O43283	VHL	WO-2022051326-A1
TPD-UBGITJ	SCHEMBL24278144	2-N-[3-[4-[6-amino-5-(trifluoromethoxy)pyridin-3-yl]-2-(1-hydroxy-2-methylpropyl)imidazol-1-yl]-1-bicyclo[1.1.1]pentanyl]-5-N-[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]pyrazine-2,5-dicarboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)c2cnc(C(=O)NC34CC(n5cc(-c6cnc(N)c(OC(F)(F)F)c6)nc5C(O)C(C)C)(C3)C4)cn2)C(C)(C)C)cc1	C47H54F3N11O7S	LZK	O43283	VHL	WO-2022051326-A1
TPD-G7D5UO	WO2022051326A1_38	1-N-[3-[4-[6-amino-5-(trifluoromethoxy)pyridin-3-yl]-2-(1-hydroxy-2-methylpropyl)imidazol-1-yl]-1-bicyclo[1.1.1]pentanyl]-3-N-[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]cyclobutane-1,3-dicarboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CC(C(=O)NC34CC(n5cc(-c6cnc(N)c(OC(F)(F)F)c6)nc5C(O)C(C)C)(C3)C4)C2)C(C)(C)C)cc1	C47H58F3N9O7S	LZK	O43283	VHL	WO-2022051326-A1
TPD-HZT8RP	SCHEMBL24278135	3-[2-[2-[2-[3-[4-[2-(3,3-difluoropyrrolidin-1-yl)-6-[[4-(trifluoromethyl)pyridin-2-yl]amino]pyridin-4-yl]piperidin-1-yl]-3-oxopropoxy]ethoxy]ethoxy]ethoxy]-N-[4-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]acetyl]amino]butyl]propanamide	O=C(CCOCCOCCOCCOCCC(=O)N1CCC(c2cc(Nc3cc(C(F)(F)F)ccn3)nc(N3CCC(F)(F)C3)c2)CC1)NCCCCNC(=O)CNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O	C51H63F5N10O11	LZK	O43283	CRBN	WO-2022051326-A1
TPD-0XYZBU	SCHEMBL24278128	(2S,4R)-1-[(2S)-2-[3-[2-[2-[2-[3-[4-[2-(3,3-difluoropyrrolidin-1-yl)-6-[[4-(trifluoromethyl)pyridin-2-yl]amino]pyridin-4-yl]piperidin-1-yl]-3-oxopropoxy]ethoxy]ethoxy]ethoxy]propanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCOCCOCCOCCOCCC(=O)N2CCC(c3cc(Nc4cc(C(F)(F)F)ccn4)nc(N4CCC(F)(F)C4)c3)CC2)C(C)(C)C)cc1	C55H72F5N9O9S	LZK	O43283	VHL	WO-2022051326-A1
TPD-2C03KG	SCHEMBL24278191	(2S,4R)-1-[(2S)-2-[6-[4-[2-[(4-cyanopyridin-2-yl)amino]-6-(3,3-difluoropyrrolidin-1-yl)pyridin-4-yl]piperidin-1-yl]hexylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NCCCCCCN2CCC(c3cc(Nc4cc(C#N)ccn4)nc(N4CCC(F)(F)C4)c3)CC2)C(C)(C)C)cc1	C49H64F2N10O3S	LZK	O43283	VHL	WO-2022051326-A1
TPD-D9YJUA	SCHEMBL24278188	(2S,4R)-1-[(2S)-2-[[6-[4-[2-[(4-cyanopyridin-2-yl)amino]-6-(3,3-difluoropyrrolidin-1-yl)pyridin-4-yl]piperidin-1-yl]-6-oxohexyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NCCCCCC(=O)N2CCC(c3cc(Nc4cc(C#N)ccn4)nc(N4CCC(F)(F)C4)c3)CC2)C(C)(C)C)cc1	C49H62F2N10O4S	LZK	O43283	VHL	WO-2022051326-A1
TPD-6Y7UWE	SCHEMBL24278203	(2S,4R)-1-[(2S)-2-[[4-[4-[4-[2-[(4-cyanopyridin-2-yl)amino]-6-(3,3-difluoropyrrolidin-1-yl)pyridin-4-yl]piperidine-1-carbonyl]phenyl]benzoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)c2ccc(-c3ccc(C(=O)N4CCC(c5cc(Nc6cc(C#N)ccn6)nc(N6CCC(F)(F)C6)c5)CC4)cc3)cc2)C(C)(C)C)cc1	C57H60F2N10O5S	LZK	O43283	VHL	WO-2022051326-A1
TPD-OGW95E	SCHEMBL24278200	(2S,4R)-1-[(2S)-2-[[4-[4-[2-[(4-cyanopyridin-2-yl)amino]-6-(3,3-difluoropyrrolidin-1-yl)pyridin-4-yl]piperidine-1-carbonyl]bicyclo[1.1.1]pentane-2-carbonyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2C3CC2C3C(=O)N2CCC(c3cc(Nc4cc(C#N)ccn4)nc(N4CCC(F)(F)C4)c3)CC2)C(C)(C)C)cc1	C50H58F2N10O5S	LZK	O43283	VHL	WO-2022051326-A1
TPD-T28G76	SCHEMBL24278186	(2S,4R)-1-[(2S)-2-[[(1R,2R)-2-[4-[2-[(4-cyanopyridin-2-yl)amino]-6-(3,3-difluoropyrrolidin-1-yl)pyridin-4-yl]piperidine-1-carbonyl]cyclopropanecarbonyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)[C@@H]2C[C@H]2C(=O)N2CCC(c3cc(Nc4cc(C#N)ccn4)nc(N4CCC(F)(F)C4)c3)CC2)C(C)(C)C)cc1	C48H56F2N10O5S	LZK	O43283	VHL	WO-2022051326-A1
TPD-8ZNE7F	SCHEMBL24278205	(2S,4R)-1-[(2S)-2-[[(1S,2S)-2-[4-[2-[(4-cyanopyridin-2-yl)amino]-6-(3,3-difluoropyrrolidin-1-yl)pyridin-4-yl]piperidine-1-carbonyl]cyclopropanecarbonyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)[C@H]2C[C@@H]2C(=O)N2CCC(c3cc(Nc4cc(C#N)ccn4)nc(N4CCC(F)(F)C4)c3)CC2)C(C)(C)C)cc1	C48H56F2N10O5S	LZK	O43283	VHL	WO-2022051326-A1
TPD-LO8I15	SCHEMBL24278202	(2S,4S)-4-[[8-[4-[2-[(4-cyanopyridin-2-yl)amino]-6-(3,3-difluoropyrrolidin-1-yl)pyridin-4-yl]piperidin-1-yl]-8-oxooctanoyl]amino]-1-[(2S)-2-cyclohexyl-2-[[(2S)-2-(methylamino)propanoyl]amino]acetyl]-N-[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]pyrrolidine-2-carboxamide	CN[C@@H](C)C(=O)N[C@H](C(=O)N1C[C@@H](NC(=O)CCCCCCC(=O)N2CCC(c3cc(Nc4cc(C#N)ccn4)nc(N4CCC(F)(F)C4)c3)CC2)C[C@H]1C(=O)N[C@@H]1CCCc2ccccc21)C1CCCCC1	C55H73F2N11O5	LZK	O43283	VHL	WO-2022051326-A1
TPD-T5CD27	SCHEMBL24278201	(2S,4R)-1-[(2S)-2-[[(1S,2R)-2-[4-[2-[(4-cyanopyridin-2-yl)amino]-6-(3,3-difluoropyrrolidin-1-yl)pyridin-4-yl]piperidine-1-carbonyl]cyclopropanecarbonyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)[C@H]2C[C@H]2C(=O)N2CCC(c3cc(Nc4cc(C#N)ccn4)nc(N4CCC(F)(F)C4)c3)CC2)C(C)(C)C)cc1	C48H56F2N10O5S	LZK	O43283	VHL	WO-2022051326-A1
TPD-QCWXHJ	SCHEMBL24278199	(2S,4R)-1-[(2S)-2-[[(1R,2S)-2-[4-[2-[(4-cyanopyridin-2-yl)amino]-6-(3,3-difluoropyrrolidin-1-yl)pyridin-4-yl]piperidine-1-carbonyl]cyclopropanecarbonyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)[C@@H]2C[C@@H]2C(=O)N2CCC(c3cc(Nc4cc(C#N)ccn4)nc(N4CCC(F)(F)C4)c3)CC2)C(C)(C)C)cc1	C48H56F2N10O5S	LZK	O43283	VHL	WO-2022051326-A1
TPD-JY32EW	SCHEMBL24278204	(2S,4R)-1-[(2S)-2-[[(1S,2R)-2-[4-[2-[(4-cyanopyridin-2-yl)amino]-6-(3,3-difluoropyrrolidin-1-yl)pyridin-4-yl]piperidine-1-carbonyl]cyclobutanecarbonyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)[C@H]2CC[C@H]2C(=O)N2CCC(c3cc(Nc4cc(C#N)ccn4)nc(N4CCC(F)(F)C4)c3)CC2)C(C)(C)C)cc1	C49H58F2N10O5S	LZK	O43283	VHL	WO-2022051326-A1
TPD-SS6VOM	SCHEMBL24278153	(2S,4R)-1-[(2S)-2-[[(1R,2S)-2-[4-[2-[(4-cyanopyridin-2-yl)amino]-6-(3,3-difluoropyrrolidin-1-yl)pyridin-4-yl]piperidine-1-carbonyl]cyclobutanecarbonyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)[C@@H]2CC[C@@H]2C(=O)N2CCC(c3cc(Nc4cc(C#N)ccn4)nc(N4CCC(F)(F)C4)c3)CC2)C(C)(C)C)cc1	C49H58F2N10O5S	LZK	O43283	VHL	WO-2022051326-A1
TPD-JM489O	SCHEMBL24278152	(4R)-1-[(2R)-2-[[3-[4-[2-[(4-cyanopyridin-2-yl)amino]-6-(3,3-difluoropyrrolidin-1-yl)pyridin-4-yl]piperidine-1-carbonyl]cyclobutanecarbonyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)C2C[C@@H](O)CN2C(=O)[C@H](NC(=O)[C@H]2C[C@@H](C(=O)N3CCC(c4cc(Nc5cc(C#N)ccn5)nc(N5CCC(F)(F)C5)c4)CC3)C2)C(C)(C)C)cc1	C49H58F2N10O5S	LZK	O43283	VHL	WO-2022051326-A1
TPD-DX6WUZ	PROTAC BTK Degrader-3	PROTAC BTK Degrader-3; 2563861-90-3; CFM78G8GFB; orb2278211; CHEMBL5423706; SCHEMBL22720738; SCHEMBL29439205; BDBM588276; US11542266, Compound 17; HY-153536; CS-0783223; 1H-ISOINDOLE-1,3(2H)-DIONE, 5-(3-(4-(4-AMINO-3-(4-PHENOXYPHENYL)-1H-PYRAZOLO(3,4-D)PYRIMIDIN-1-YL)-1-PIPERIDINYL)(1,3'-BIAZETIDIN)-1'-YL)-2-(2,6-DIOXO-3-PIPERIDINYL)-; 5-[3-[3-[4-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]-1-piperidyl]azetidin-1-yl]azetidin-1-yl]-2-(2,6-dioxo-3-piperidyl)isoindoline-1,3-dione	NC1=C2C(C3=CC=C(OC4=CC=CC=C4)C=C3)=NN(C3CCN(C4CN(C5CN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)C4)CC3)C2=NC=N1	C41H40N10O5	BTK	Q06187	CRBN	WO-2022052950-A1
TPD-YWHWLT	SCHEMBL24351539	3-[4-[2-[4-[1-[2-fluoro-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazin-1-yl]ethyl]phenyl]piperidine-2,6-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC(F)=C(N5CCC(N6CCN(CCC7=CC=C(C8CCC(=O)NC8=O)C=C7)CC6)CC5)C=C4)=NC4=C3C=CN4)=C21	C43H49FN10O4S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-7V0U13	SCHEMBL24351528	3-[4-[2-[4-[1-[2-fluoro-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2-methoxyphenyl]piperidine-2,6-dione	COC1=CC(CCN2CCN(C3CCN(C4=C(F)C=C(NC5=NC6=C(C=CN6)C(NC6=C7C(=CC=C6)CCN7S(C)(=O)=O)=N5)C=C4)CC3)CC2)=CC=C1C1CCC(=O)NC1=O	C44H51FN10O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-NMZS0B	SCHEMBL27031722	3-[2-fluoro-4-[2-[4-[1-[2-fluoro-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazin-1-yl]ethyl]phenyl]piperidine-2,6-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC(F)=C(N5CCC(N6CCN(CCC7=CC=C(C8CCC(=O)NC8=O)C(F)=C7)CC6)CC5)C=C4)=NC4=C3C=CN4)=C21	C43H48F2N10O4S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-ECM92J	SCHEMBL24351176	3-[4-[3-[4-[1-[2-fluoro-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazin-1-yl]propoxy]phenoxy]piperidine-2,6-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC(F)=C(N5CCC(N6CCN(CCCOC7=CC=C(OC8CCC(=O)NC8=O)C=C7)CC6)CC5)C=C4)=NC4=C3C=CN4)=C21	C44H51FN10O6S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-9W67ME	SCHEMBL24352098	3-[3-[2-[4-[1-[2-fluoro-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazin-1-yl]ethoxy]phenyl]piperidine-2,6-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC(F)=C(N5CCC(N6CCN(CCOC7=CC=CC(C8CCC(=O)NC8=O)=C7)CC6)CC5)C=C4)=NC4=C3C=CN4)=C21	C43H49FN10O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-T0R81W	SCHEMBL24351541	3-[3-[2-[4-[1-[2-fluoro-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazin-1-yl]ethyl-methylamino]phenyl]piperidine-2,6-dione	CN(CCN1CCN(C2CCN(C3=C(F)C=C(NC4=NC5=C(C=CN5)C(NC5=C6C(=CC=C5)CCN6S(C)(=O)=O)=N4)C=C3)CC2)CC1)C1=CC=CC(C2CCC(=O)NC2=O)=C1	C44H52FN11O4S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-T1FVGS	SCHEMBL27048795	3-[3-[3-[4-[1-[2-fluoro-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazin-1-yl]propyl-methylamino]phenyl]piperidine-2,6-dione	CN(CCCN1CCN(C2CCN(C3=C(F)C=C(NC4=NC5=C(C=CN5)C(NC5=C6C(=CC=C5)CCN6S(C)(=O)=O)=N4)C=C3)CC2)CC1)C1=CC=CC(C2CCC(=O)NC2=O)=C1	C45H54FN11O4S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-ZSPC3L	SCHEMBL24351542	3-[4-[4-[2-[4-[1-[2-fluoro-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazin-1-yl]ethyl]piperidin-1-yl]phenyl]piperidine-2,6-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC(F)=C(N5CCC(N6CCN(CCC7CCN(C8=CC=C(C9CCC(=O)NC9=O)C=C8)CC7)CC6)CC5)C=C4)=NC4=C3C=CN4)=C21	C48H58FN11O4S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-PG53HZ	SCHEMBL27031703	3-[2-fluoro-4-[4-[2-[4-[1-[2-fluoro-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazin-1-yl]ethyl]piperidin-1-yl]phenyl]piperidine-2,6-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC(F)=C(N5CCC(N6CCN(CCC7CCN(C8=CC(F)=C(C9CCC(=O)NC9=O)C=C8)CC7)CC6)CC5)C=C4)=NC4=C3C=CN4)=C21	C48H57F2N11O4S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-O5XK21	SCHEMBL27031597	2-(2,6-dioxopiperidin-3-yl)-5-[4-[2-[4-[1-[2-fluoro-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazin-1-yl]ethyl]piperidin-1-yl]benzonitrile	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC(F)=C(N5CCC(N6CCN(CCC7CCN(C8=CC=C(C9CCC(=O)NC9=O)C(C#N)=C8)CC7)CC6)CC5)C=C4)=NC4=C3C=CN4)=C21	C49H57FN12O4S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-NM1N9K	SCHEMBL24351192	3-[4-[1-[3-[4-[1-[2-fluoro-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazin-1-yl]-3-oxopropyl]piperidin-4-yl]phenyl]piperidine-2,6-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC(F)=C(N5CCC(N6CCN(C(=O)CCN7CCC(C8=CC=C(C9CCC(=O)NC9=O)C=C8)CC7)CC6)CC5)C=C4)=NC4=C3C=CN4)=C21	C49H58FN11O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-14HU8V	SCHEMBL24351860	3-[4-[4-[2-[4-[1-[2-fluoro-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazin-1-yl]-2-oxoethyl]piperidin-1-yl]phenyl]piperidine-2,6-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC(F)=C(N5CCC(N6CCN(C(=O)CC7CCN(C8=CC=C(C9CCC(=O)NC9=O)C=C8)CC7)CC6)CC5)C=C4)=NC4=C3C=CN4)=C21	C48H56FN11O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-J1T1JB	SCHEMBL27031636	3-[4-[(3S)-3-[2-[4-[1-[2-fluoro-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazin-1-yl]ethyl]pyrrolidin-1-yl]phenyl]piperidine-2,6-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC(F)=C(N5CCC(N6CCN(CC[C@H]7CCN(C8=CC=C(C9CCC(=O)NC9=O)C=C8)C7)CC6)CC5)C=C4)=NC4=C3C=CN4)=C21	C47H56FN11O4S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-POE8TN	SCHEMBL24351908	2-(2,6-dioxopiperidin-3-yl)-5-[4-[[4-[4-[1-[2-fluoro-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazine-1-carbonyl]piperidin-1-yl]methyl]piperidin-1-yl]isoindole-1,3-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC(F)=C(N5CCC(N6CCN(C(=O)C7CCN(CC8CCN(C9=CC=C%10C(=O)N(C%11CCC(=O)NC%11=O)C(=O)C%10=C9)CC8)CC7)CC6)CC5)C=C4)=NC4=C3C=CN4)=C21	C55H64FN13O7S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-FGQAF5	SCHEMBL24352110	2-(2,6-dioxopiperidin-3-yl)-5-[4-[3-[4-[1-[2-fluoro-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazin-1-yl]-3-oxopropyl]piperazin-1-yl]isoindole-1,3-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC(F)=C(N5CCC(N6CCN(C(=O)CCN7CCN(C8=CC=C9C(=O)N(C%10CCC(=O)NC%10=O)C(=O)C9=C8)CC7)CC6)CC5)C=C4)=NC4=C3C=CN4)=C21	C50H56FN13O7S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-04Q35Q	SCHEMBL24351189	2-(2,6-dioxopiperidin-3-yl)-5-[4-[[4-[1-[2-fluoro-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazin-1-yl]methyl]piperidin-1-yl]isoindole-1,3-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC(F)=C(N5CCC(N6CCN(CC7CCN(C8=CC=C9C(=O)N(C%10CCC(=O)NC%10=O)C(=O)C9=C8)CC7)CC6)CC5)C=C4)=NC4=C3C=CN4)=C21	C49H55FN12O6S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-FPXO74	SCHEMBL27031710	2-(2,6-dioxopiperidin-3-yl)-5-[4-[2-[4-[1-[2-fluoro-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazin-1-yl]ethyl]piperidin-1-yl]isoindole-1,3-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC(F)=C(N5CCC(N6CCN(CCC7CCN(C8=CC9=C(C=C8)C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)C=C4)=NC4=C3C=CN4)=C21	C50H57FN12O6S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-YFLW7V	SCHEMBL24351913	3-[6-[4-[2-[4-[1-[2-fluoro-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazin-1-yl]ethyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC(F)=C(N5CCC(N6CCN(CCC7CCN(C8=CC9=C(C=C8)C(=O)N(C8CCC(=O)NC8=O)C9)CC7)CC6)CC5)C=C4)=NC4=C3C=CN4)=C21	C50H59FN12O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-955O4O	SCHEMBL27031613	2-(2,6-dioxopiperidin-3-yl)-5-[3-[3-[4-[1-[2-fluoro-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazin-1-yl]propyl]azetidin-1-yl]isoindole-1,3-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC(F)=C(N5CCC(N6CCN(CCCC7CN(C8=CC9=C(C=C8)C(=O)N(C8CCC(=O)NC8=O)C9=O)C7)CC6)CC5)C=C4)=NC4=C3C=CN4)=C21	C49H55FN12O6S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-G3ECJJ	SCHEMBL24351910	3-[7-[2-[4-[1-[2-fluoro-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazin-1-yl]ethoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC(F)=C(N5CCC(N6CCN(CCOC7=CC=CC8=C7CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)C=C4)=NC4=C3C=CN4)=C21	C45H50FN11O6S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-J3S4O5	SCHEMBL27031672	3-[4-[2-[4-[1-[3-methoxy-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazin-1-yl]ethyl]phenyl]piperidine-2,6-dione	COC1=CC(N2CCC(N3CCN(CCC4=CC=C(C5CCC(=O)NC5=O)C=C4)CC3)CC2)=CC=C1NC1=NC2=C(C=CN2)C(NC2=C3C(=CC=C2)CCN3S(C)(=O)=O)=N1	C44H52N10O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-W8DQAR	SCHEMBL24351917	3-[2-fluoro-4-[4-[2-[[1-[5-methoxy-2-methyl-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]-methylamino]ethyl]piperidin-1-yl]phenyl]piperidine-2,6-dione	COC1=C(NC2=NC3=C(C=CN3)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=C(C)C(N2CCC(N(C)CCC3CCN(C4=CC(F)=C(C5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C47H57FN10O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-TM12OT	SCHEMBL24351588	3-[4-[4-[2-[[1-[5-methoxy-2-methyl-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]-methylamino]ethyl]piperidin-1-yl]phenyl]piperidine-2,6-dione	COC1=C(NC2=NC3=C(C=CN3)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=C(C)C(N2CCC(N(C)CCC3CCN(C4=CC=C(C5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C47H58N10O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-DEIPWY	SCHEMBL24351577	2-(2,6-dioxopiperidin-3-yl)-5-[4-[2-[[1-[5-methoxy-2-methyl-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]-methylamino]ethyl]piperidin-1-yl]isoindole-1,3-dione	COC1=C(NC2=NC3=C(C=CN3)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=C(C)C(N2CCC(N(C)CCC3CCN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)=C1	C49H57N11O7S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-ENPNOT	SCHEMBL24351576	2-(2,6-dioxopiperidin-3-yl)-5-[3-[3-[[1-[5-methoxy-2-methyl-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]-methylamino]propyl]azetidin-1-yl]isoindole-1,3-dione	COC1=C(NC2=NC3=C(C=CN3)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=C(C)C(N2CCC(N(C)CCCC3CN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)CC2)=C1	C48H55N11O7S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-0OMMOL	SCHEMBL27048809	3-[2-fluoro-4-[2-[4-[2-fluoro-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperazin-1-yl]ethyl]phenyl]piperidine-2,6-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC(F)=C(N5CCN(CCC6=CC=C(C7CCC(=O)NC7=O)C(F)=C6)CC5)C=C4)=NC4=C3C=CN4)=C21	C38H39F2N9O4S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-DF0NP7	SCHEMBL24351591	3-[4-[4-[2-[4-[2-fluoro-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperazin-1-yl]ethyl]piperidin-1-yl]phenyl]piperidine-2,6-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC(F)=C(N5CCN(CCC6CCN(C7=CC=C(C8CCC(=O)NC8=O)C=C7)CC6)CC5)C=C4)=NC4=C3C=CN4)=C21	C43H49FN10O4S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-44M9NA	SCHEMBL27048810	3-[2-fluoro-4-[4-[2-[4-[2-fluoro-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperazin-1-yl]ethyl]piperidin-1-yl]phenyl]piperidine-2,6-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC(F)=C(N5CCN(CCC6CCN(C7=CC(F)=C(C8CCC(=O)NC8=O)C=C7)CC6)CC5)C=C4)=NC4=C3C=CN4)=C21	C43H48F2N10O4S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-5GMO84	SCHEMBL24351593	2-(2,6-dioxopiperidin-3-yl)-5-[4-[2-[4-[2-fluoro-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperazin-1-yl]ethyl]piperidin-1-yl]isoindole-1,3-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC(F)=C(N5CCN(CCC6CCN(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)C=C4)=NC4=C3C=CN4)=C21	C45H48FN11O6S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-O465BB	SCHEMBL27048812	2-(2,6-dioxopiperidin-3-yl)-5-[3-[3-[4-[2-fluoro-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperazin-1-yl]propyl]azetidin-1-yl]isoindole-1,3-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC(F)=C(N5CCN(CCCC6CN(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8=O)C6)CC5)C=C4)=NC4=C3C=CN4)=C21	C44H46FN11O6S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-GXCPO5	SCHEMBL24351580	3-[2-fluoro-4-[4-[2-[(2R)-4-[5-methoxy-2-methyl-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]-2-methylpiperazin-1-yl]ethyl]piperidin-1-yl]phenyl]piperidine-2,6-dione	COC1=C(NC2=NC3=C(C=CN3)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=C(C)C(N2CCN(CCC3CCN(C4=CC(F)=C(C5CCC(=O)NC5=O)C=C4)CC3)[C@H](C)C2)=C1	C46H55FN10O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-6BCVKV	SCHEMBL24351592	3-[4-[4-[2-[(2R)-4-[5-methoxy-2-methyl-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]-2-methylpiperazin-1-yl]ethyl]piperidin-1-yl]phenyl]piperidine-2,6-dione	COC1=C(NC2=NC3=C(C=CN3)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=C(C)C(N2CCN(CCC3CCN(C4=CC=C(C5CCC(=O)NC5=O)C=C4)CC3)[C@H](C)C2)=C1	C46H56N10O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-QLS0U8	SCHEMBL24351584	2-(2,6-dioxopiperidin-3-yl)-5-[4-[2-[(2R)-4-[5-methoxy-2-methyl-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]-2-methylpiperazin-1-yl]ethyl]piperidin-1-yl]isoindole-1,3-dione	COC1=C(NC2=NC3=C(C=CN3)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=C(C)C(N2CCN(CCC3CCN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)[C@H](C)C2)=C1	C48H55N11O7S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-P1HY8N	SCHEMBL24351707	3-[4-[2-[4-[1-[4-[[5-Chloro-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-3-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]phenyl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=CC(N2CCC(N3CCN(CCC4=CC=C(C5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C42H50ClN9O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-RTDJH1	SCHEMBL27031732	3-[4-[4-[2-[4-[1-[4-[[5-Chloro-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-3-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]piperidin-1-yl]phenyl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=CC(N2CCC(N3CCN(CCC4CCN(C5=CC=C(C6CCC(=O)NC6=O)C=C5)CC4)CC3)CC2)=C1	C47H59ClN10O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-QJ9AL4	SCHEMBL24351864	3-[4-[4-[2-[4-[1-[4-[[5-Chloro-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-3-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]piperidin-1-yl]-2-fluorophenyl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=CC(N2CCC(N3CCN(CCC4CCN(C5=CC=C(C6CCC(=O)NC6=O)C(F)=C5)CC4)CC3)CC2)=C1	C47H58ClFN10O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-4L7B0V	SCHEMBL24351866	5-[4-[2-[4-[1-[4-[[5-Chloro-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-3-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]piperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=CC(N2CCC(N3CCN(CCC4CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)CC2)=C1	C49H58ClN11O7S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-1DA9ML	SCHEMBL24352074	3-[4-[2-[4-[4-[4-[[5-Chloro-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-3-methoxyphenyl]piperazin-1-yl]piperidin-1-yl]ethyl]phenyl]piperidine-2,6-dione	COC1=CC(N2CCN(C3CCN(CCC4=CC=C(C5CCC(=O)NC5=O)C=C4)CC3)CC2)=CC=C1NC1=NC=C(Cl)C(NC2=C3C(=CC=C2)CCN3S(C)(=O)=O)=N1	C42H50ClN9O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-O8SU5F	SCHEMBL27031668	3-[4-[2-[4-[1-[4-[[5-Bromo-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]phenyl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Br)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=C(C)C(N2CCC(N3CCN(CCC4=CC=C(C5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C43H52BrN9O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-VWKEN4	SCHEMBL24351708	3-[4-[4-[[4-[1-[4-[[5-Bromo-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Br)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=C(C)C(N2CCC(N3CCN(CC4CCN(C5=CC=C(C6CCC(=O)NC6=O)C=C5)CC4)CC3)CC2)=C1	C47H59BrN10O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-I5IVLV	SCHEMBL24351875	3-[4-[4-[2-[4-[1-[4-[[5-Bromo-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]piperidin-1-yl]phenyl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Br)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=C(C)C(N2CCC(N3CCN(CCC4CCN(C5=CC=C(C6CCC(=O)NC6=O)C=C5)CC4)CC3)CC2)=C1	C48H61BrN10O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-HOUUTK	SCHEMBL24352067	5-[4-[3-[4-[1-[4-[[5-Bromo-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]-3-oxopropyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	COC1=C(NC2=NC=C(Br)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=C(C)C(N2CCC(N3CCN(C(=O)CCN4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)CC2)=C1	C50H59BrN12O8S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-VRICT3	SCHEMBL24352068	5-[4-[[4-[4-[1-[4-[[5-Bromo-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazine-1-carbonyl]piperidin-1-yl]methyl]piperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	COC1=C(NC2=NC=C(Br)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=C(C)C(N2CCC(N3CCN(C(=O)C4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)CC3)CC2)=C1	C55H67BrN12O8S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-T5RDVF	SCHEMBL24352069	5-[3-[3-[4-[1-[4-[[5-Bromo-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]propyl]azetidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	COC1=C(NC2=NC=C(Br)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=C(C)C(N2CCC(N3CCN(CCCC4CN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)CC2)=C1	C49H58BrN11O7S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-RM9LF2	SCHEMBL24352065	3-[4-[2-[4-[1-[4-[[5-Chloro-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-2-fluorophenyl]piperidin-4-yl]piperazin-1-yl]ethyl]phenyl]piperidine-2,6-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC=C(N5CCC(N6CCN(CCC7=CC=C(C8CCC(=O)NC8=O)C=C7)CC6)CC5)C(F)=C4)=NC=C3Cl)=C21	C41H47ClFN9O4S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-LZKFVO	SCHEMBL24352070	3-[4-[4-[2-[[1-[7-[[5-Chloro-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-2,3-dihydro-1-benzofuran-4-yl]piperidin-4-yl]-methylamino]ethyl]piperidin-1-yl]-2-fluorophenyl]piperidine-2,6-dione	CN(CCC1CCN(C2=CC=C(C3CCC(=O)NC3=O)C(F)=C2)CC1)C1CCN(C2=C3CCOC3=C(NC3=NC=C(Cl)C(NC4=C5C(=CC=C4)CCN5S(C)(=O)=O)=N3)C=C2)CC1	C45H53ClFN9O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-4YJM1V	SCHEMBL27031679	5-[4-[2-[[1-[7-[[5-Chloro-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-2,3-dihydro-1-benzofuran-4-yl]piperidin-4-yl]-methylamino]ethyl]piperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN(CCC1CCN(C2=CC=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=C2)CC1)C1CCN(C2=C3CCOC3=C(NC3=NC=C(Cl)C(NC4=C5C(=CC=C4)CCN5S(C)(=O)=O)=N3)C=C2)CC1	C47H53ClN10O7S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-51825Y	SCHEMBL24352071	3-[4-[2-[[1-[7-[[5-Chloro-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-2,3-dihydro-1-benzofuran-4-yl]piperidin-4-yl]-methylamino]ethyl]-2-fluorophenyl]piperidine-2,6-dione	CN(CCC1=CC=C(C2CCC(=O)NC2=O)C(F)=C1)C1CCN(C2=C3CCOC3=C(NC3=NC=C(Cl)C(NC4=C5C(=CC=C4)CCN5S(C)(=O)=O)=N3)C=C2)CC1	C40H44ClFN8O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-O1MC5Y	SCHEMBL24351683	3-[4-[4-[2-[[1-[7-[[5-Chloro-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-2,3-dihydro-1-benzofuran-4-yl]piperidin-4-yl]-methylamino]ethyl]piperidin-1-yl]phenyl]piperidine-2,6-dione	CN(CCC1CCN(C2=CC=C(C3CCC(=O)NC3=O)C=C2)CC1)C1CCN(C2=C3CCOC3=C(NC3=NC=C(Cl)C(NC4=C5C(=CC=C4)CCN5S(C)(=O)=O)=N3)C=C2)CC1	C45H54ClN9O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-M6Z05C	SCHEMBL24351685	5-[3-[3-[[1-[7-[[5-Chloro-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-2,3-dihydro-1-benzofuran-4-yl]piperidin-4-yl]-methylamino]propyl]azetidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN(CCCC1CN(C2=CC3=C(C=C2)C(=O)N(C2CCC(=O)NC2=O)C3=O)C1)C1CCN(C2=C3CCOC3=C(NC3=NC=C(Cl)C(NC4=C5C(=CC=C4)CCN5S(C)(=O)=O)=N3)C=C2)CC1	C46H51ClN10O7S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-OIZWXH	SCHEMBL24351658	3-[4-[4-[2-[4-[1-[7-[[5-Chloro-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-2,3-dihydro-1-benzofuran-4-yl]piperidin-4-yl]piperazin-1-yl]ethyl]piperidin-1-yl]-2-fluorophenyl]piperidine-2,6-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=C5OCCC5=C(N5CCC(N6CCN(CCC7CCN(C8=CC=C(C9CCC(=O)NC9=O)C(F)=C8)CC7)CC6)CC5)C=C4)=NC=C3Cl)=C21	C48H58ClFN10O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-CE2RBJ	SCHEMBL24352291	5-[4-[2-[4-[1-[7-[[5-Chloro-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-2,3-dihydro-1-benzofuran-4-yl]piperidin-4-yl]piperazin-1-yl]ethyl]piperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=C5OCCC5=C(N5CCC(N6CCN(CCC7CCN(C8=CC=C9C(=O)N(C%10CCC(=O)NC%10=O)C(=O)C9=C8)CC7)CC6)CC5)C=C4)=NC=C3Cl)=C21	C50H58ClN11O7S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-WCIZQD	SCHEMBL27031684	3-[4-[2-[4-[1-[7-[[5-Chloro-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-2,3-dihydro-1-benzofuran-4-yl]piperidin-4-yl]piperazin-1-yl]ethyl]-2-fluorophenyl]piperidine-2,6-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=C5OCCC5=C(N5CCC(N6CCN(CCC7=CC=C(C8CCC(=O)NC8=O)C(F)=C7)CC6)CC5)C=C4)=NC=C3Cl)=C21	C43H49ClFN9O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-H1FSZU	SCHEMBL24351842	3-[4-[4-[2-[4-[1-[7-[[5-Chloro-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-2,3-dihydro-1-benzofuran-4-yl]piperidin-4-yl]piperazin-1-yl]ethyl]piperidin-1-yl]phenyl]piperidine-2,6-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=C5OCCC5=C(N5CCC(N6CCN(CCC7CCN(C8=CC=C(C9CCC(=O)NC9=O)C=C8)CC7)CC6)CC5)C=C4)=NC=C3Cl)=C21	C48H59ClN10O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-92F805	SCHEMBL27031680	5-[3-[3-[4-[1-[7-[[5-Chloro-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-2,3-dihydro-1-benzofuran-4-yl]piperidin-4-yl]piperazin-1-yl]propyl]azetidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=C5OCCC5=C(N5CCC(N6CCN(CCCC7CN(C8=CC9=C(C=C8)C(=O)N(C8CCC(=O)NC8=O)C9=O)C7)CC6)CC5)C=C4)=NC=C3Cl)=C21	C49H56ClN11O7S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-AO0FPV	SCHEMBL24351681	3-[4-[4-[2-[4-[4-[[5-Chloro-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-3-methoxyphenyl]piperazin-1-yl]ethyl]piperidin-1-yl]phenyl]piperidine-2,6-dione	COC1=CC(N2CCN(CCC3CCN(C4=CC=C(C5CCC(=O)NC5=O)C=C4)CC3)CC2)=CC=C1NC1=NC=C(Cl)C(NC2=C3C(=CC=C2)CCN3S(C)(=O)=O)=N1	C42H50ClN9O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-RW8GVQ	SCHEMBL27048816	3-[4-[3-[2-[4-[1-[2-fluoro-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazin-1-yl]ethyl]azetidin-1-yl]phenyl]piperidine-2,6-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC(F)=C(N5CCC(N6CCN(CCC7CN(C8=CC=C(C9CCC(=O)NC9=O)C=C8)C7)CC6)CC5)C=C4)=NC4=C3C=CN4)=C21	C46H54FN11O4S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-9LVPZG	SCHEMBL24351232	3-[4-[3-[4-[1-[2-fluoro-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazine-1-carbonyl]azetidin-1-yl]phenyl]piperidine-2,6-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC(F)=C(N5CCC(N6CCN(C(=O)C7CN(C8=CC=C(C9CCC(=O)NC9=O)C=C8)C7)CC6)CC5)C=C4)=NC4=C3C=CN4)=C21	C45H50FN11O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-FM9C5Z	SCHEMBL24351687	3-[6-[3-[[4-[1-[2-fluoro-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazin-1-yl]methyl]azetidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC(F)=C(N5CCC(N6CCN(CC7CN(C8=CC9=C(C=C8)C(=O)N(C8CCC(=O)NC8=O)C9)C7)CC6)CC5)C=C4)=NC4=C3C=CN4)=C21	C47H53FN12O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-C83TUF	SCHEMBL24351863	2-(2,6-dioxopiperidin-3-yl)-5-[3-[[4-[1-[2-fluoro-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazin-1-yl]methyl]azetidin-1-yl]isoindole-1,3-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC(F)=C(N5CCC(N6CCN(CC7CN(C8=CC9=C(C=C8)C(=O)N(C8CCC(=O)NC8=O)C9=O)C7)CC6)CC5)C=C4)=NC4=C3C=CN4)=C21	C47H51FN12O6S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-1I70JU	SCHEMBL24351886	2-(2,6-dioxopiperidin-3-yl)-5-[3-[2-[4-[1-[2-fluoro-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazin-1-yl]-2-oxoethyl]azetidin-1-yl]isoindole-1,3-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC(F)=C(N5CCC(N6CCN(C(=O)CC7CN(C8=CC9=C(C=C8)C(=O)N(C8CCC(=O)NC8=O)C9=O)C7)CC6)CC5)C=C4)=NC4=C3C=CN4)=C21	C48H51FN12O7S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-HT726B	SCHEMBL24352293	2-(2,6-dioxopiperidin-3-yl)-5-[(3R)-3-[4-[1-[2-fluoro-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazine-1-carbonyl]pyrrolidin-1-yl]isoindole-1,3-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC(F)=C(N5CCC(N6CCN(C(=O)[C@@H]7CCN(C8=CC9=C(C=C8)C(=O)N(C8CCC(=O)NC8=O)C9=O)C7)CC6)CC5)C=C4)=NC4=C3C=CN4)=C21	C48H51FN12O7S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-S3XPC9	SCHEMBL27031615	2-(2,6-dioxopiperidin-3-yl)-5-[(3S)-3-[4-[1-[2-fluoro-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazine-1-carbonyl]pyrrolidin-1-yl]isoindole-1,3-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC(F)=C(N5CCC(N6CCN(C(=O)[C@H]7CCN(C8=CC9=C(C=C8)C(=O)N(C8CCC(=O)NC8=O)C9=O)C7)CC6)CC5)C=C4)=NC4=C3C=CN4)=C21	C48H51FN12O7S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-ADBILN	SCHEMBL24351858	3-[4-[(3R)-3-[2-[4-[1-[2-fluoro-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazin-1-yl]ethyl]pyrrolidin-1-yl]phenyl]piperidine-2,6-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC(F)=C(N5CCC(N6CCN(CC[C@@H]7CCN(C8=CC=C(C9CCC(=O)NC9=O)C=C8)C7)CC6)CC5)C=C4)=NC4=C3C=CN4)=C21	C47H56FN11O4S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-M82A8O	SCHEMBL24351848	3-[7-[3-[4-[1-[2-fluoro-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazin-1-yl]propoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC(F)=C(N5CCC(N6CCN(CCCOC7=CC=CC8=C7CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)C=C4)=NC4=C3C=CN4)=C21	C46H52FN11O6S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-3CR95Z	SCHEMBL27031681	3-[4-[2-[4-[1-[2-fluoro-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazin-1-yl]ethyl]anilino]piperidine-2,6-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC(F)=C(N5CCC(N6CCN(CCC7=CC=C(NC8CCC(=O)NC8=O)C=C7)CC6)CC5)C=C4)=NC4=C3C=CN4)=C21	C43H50FN11O4S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-GIMOSD	SCHEMBL27031611	3-[2,6-difluoro-4-[4-[2-[4-[1-[2-fluoro-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazin-1-yl]ethyl]piperidin-1-yl]phenyl]piperidine-2,6-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC(F)=C(N5CCC(N6CCN(CCC7CCN(C8=CC(F)=C(C9CCC(=O)NC9=O)C(F)=C8)CC7)CC6)CC5)C=C4)=NC4=C3C=CN4)=C21	C48H56F3N11O4S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-EHI55D	SCHEMBL27031653	3-[2,6-difluoro-4-[2-[4-[1-[2-fluoro-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazin-1-yl]ethyl]phenyl]piperidine-2,6-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC(F)=C(N5CCC(N6CCN(CCC7=CC(F)=C(C8CCC(=O)NC8=O)C(F)=C7)CC6)CC5)C=C4)=NC4=C3C=CN4)=C21	C43H47F3N10O4S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-R6E6C0	SCHEMBL24352113	3-[2,3-difluoro-4-[2-[4-[1-[2-fluoro-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazin-1-yl]ethyl]phenyl]piperidine-2,6-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC(F)=C(N5CCC(N6CCN(CCC7=C(F)C(F)=C(C8CCC(=O)NC8=O)C=C7)CC6)CC5)C=C4)=NC4=C3C=CN4)=C21	C43H47F3N10O4S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-YQ9CHR	SCHEMBL24351847	3-[4-[4-[[4-[2-fluoro-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]piperidine-2,6-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC(F)=C(N5CCN(CC6CCN(C7=CC=C(C8CCC(=O)NC8=O)C=C7)CC6)CC5)C=C4)=NC4=C3C=CN4)=C21	C42H47FN10O4S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-H2DU9I	SCHEMBL27048822	2-(2,6-dioxopiperidin-3-yl)-5-[3-[4-[2-fluoro-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperazine-1-carbonyl]azetidin-1-yl]isoindole-1,3-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC(F)=C(N5CCN(C(=O)C6CN(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8=O)C6)CC5)C=C4)=NC4=C3C=CN4)=C21	C42H40FN11O7S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-VK0GMI	SCHEMBL24351859	2-(2,6-dioxopiperidin-3-yl)-5-[3-[[4-[2-fluoro-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperazin-1-yl]methyl]azetidin-1-yl]isoindole-1,3-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC(F)=C(N5CCN(CC6CN(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8=O)C6)CC5)C=C4)=NC4=C3C=CN4)=C21	C42H42FN11O6S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-ELOOAN	SCHEMBL27031706	2-(2,6-dioxopiperidin-3-yl)-5-[3-[4-[1-[2-methoxy-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazine-1-carbonyl]azetidin-1-yl]isoindole-1,3-dione	COC1=CC(NC2=NC(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=C3C=CNC3=N2)=CC=C1N1CCC(N2CCN(C(=O)C3CN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)C3)CC2)CC1	C48H52N12O8S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-RA076S	SCHEMBL27031724	2-(2,6-dioxopiperidin-3-yl)-5-[(3S)-3-[4-[1-[2-methoxy-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazine-1-carbonyl]pyrrolidin-1-yl]isoindole-1,3-dione	COC1=CC(NC2=NC(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=C3C=CNC3=N2)=CC=C1N1CCC(N2CCN(C(=O)[C@H]3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)C3)CC2)CC1	C49H54N12O8S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-PYARMN	SCHEMBL24351849	2-(2,6-dioxopiperidin-3-yl)-5-[(3R)-3-[4-[1-[2-methoxy-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazine-1-carbonyl]pyrrolidin-1-yl]isoindole-1,3-dione	COC1=CC(NC2=NC(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=C3C=CNC3=N2)=CC=C1N1CCC(N2CCN(C(=O)[C@@H]3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)C3)CC2)CC1	C49H54N12O8S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-RUQ9F0	SCHEMBL24352306	5-[3-[[4-[1-[4-[[5-Chloro-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-2-fluorophenyl]piperidin-4-yl]piperazin-1-yl]methyl]azetidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC=C(N5CCC(N6CCN(CC7CN(C8=CC9=C(C=C8)C(=O)N(C8CCC(=O)NC8=O)C9=O)C7)CC6)CC5)C(F)=C4)=NC=C3Cl)=C21	C45H49ClFN11O6S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-JFAGOV	SCHEMBL24351636	5-[3-[4-[1-[4-[[5-Chloro-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-2-fluorophenyl]piperidin-4-yl]piperazine-1-carbonyl]azetidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC=C(N5CCC(N6CCN(C(=O)C7CN(C8=CC9=C(C=C8)C(=O)N(C8CCC(=O)NC8=O)C9=O)C7)CC6)CC5)C(F)=C4)=NC=C3Cl)=C21	C45H47ClFN11O7S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-JVMRK9	SCHEMBL24351867	5-[3-[3-[4-[1-[4-[[5-Chloro-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-2-fluorophenyl]piperidin-4-yl]piperazin-1-yl]propyl]azetidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC=C(N5CCC(N6CCN(CCCC7CN(C8=CC9=C(C=C8)C(=O)N(C8CCC(=O)NC8=O)C9=O)C7)CC6)CC5)C(F)=C4)=NC=C3Cl)=C21	C47H53ClFN11O6S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-FUOQQT	SCHEMBL27031685	3-[4-[4-[2-[4-[1-[4-[[5-Chloro-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-2-fluorophenyl]piperidin-4-yl]piperazin-1-yl]ethyl]piperidin-1-yl]phenyl]piperidine-2,6-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC=C(N5CCC(N6CCN(CCC7CCN(C8=CC=C(C9CCC(=O)NC9=O)C=C8)CC7)CC6)CC5)C(F)=C4)=NC=C3Cl)=C21	C46H56ClFN10O4S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-O1BFU9	SCHEMBL24351882	3-[4-[4-[2-[4-[1-[4-[[5-Chloro-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-2-fluorophenyl]piperidin-4-yl]piperazin-1-yl]ethyl]piperidin-1-yl]-2-fluorophenyl]piperidine-2,6-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC=C(N5CCC(N6CCN(CCC7CCN(C8=CC(F)=C(C9CCC(=O)NC9=O)C=C8)CC7)CC6)CC5)C(F)=C4)=NC=C3Cl)=C21	C46H55ClF2N10O4S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-Y1NV26	SCHEMBL24351643	5-[4-[2-[4-[1-[4-[[5-Chloro-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-2-fluorophenyl]piperidin-4-yl]piperazin-1-yl]ethyl]piperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC=C(N5CCC(N6CCN(CCC7CCN(C8=CC=C9C(=O)N(C%10CCC(=O)NC%10=O)C(=O)C9=C8)CC7)CC6)CC5)C(F)=C4)=NC=C3Cl)=C21	C48H55ClFN11O6S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-4ZXJU8	SCHEMBL24351644	5-[(3S)-3-[4-[1-[4-[[5-chloro-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-2-fluorophenyl]piperidin-4-yl]piperazine-1-carbonyl]pyrrolidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC=C(N5CCC(N6CCN(C(=O)[C@H]7CCN(C8=CC=C9C(=O)N(C%10CCC(=O)NC%10=O)C(=O)C9=C8)C7)CC6)CC5)C(F)=C4)=NC=C3Cl)=C21	C46H49ClFN11O7S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-VKQFJP	SCHEMBL24351639	5-[(3R)-3-[4-[1-[4-[[5-chloro-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-2-fluorophenyl]piperidin-4-yl]piperazine-1-carbonyl]pyrrolidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC=C(N5CCC(N6CCN(C(=O)[C@@H]7CCN(C8=CC=C9C(=O)N(C%10CCC(=O)NC%10=O)C(=O)C9=C8)C7)CC6)CC5)C(F)=C4)=NC=C3Cl)=C21	C46H49ClFN11O7S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-ZQ84H0	SCHEMBL24351645	3-[4-[3-[2-[4-[1-[4-[[5-Chloro-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-3-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]azetidin-1-yl]phenyl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=CC(N2CCC(N3CCN(CCC4CN(C5=CC=C(C6CCC(=O)NC6=O)C=C5)C4)CC3)CC2)=C1	C45H55ClN10O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-UN3Y75	SCHEMBL24351877	3-[6-[3-[[4-[1-[4-[[5-chloro-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-3-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]methyl]azetidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=CC(N2CCC(N3CCN(CC4CN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6)C4)CC3)CC2)=C1	C46H54ClN11O6S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-IL0QO4	WO2022068849A1_86	.	COC1=C(NC2=NC=C(Cl)C(NC3=C4C(CC=C3)CCN4S(C)(=O)=O)=N2)C=CC(N2CCC(N3CCN(CC4CN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)CC3)CC2)=C1	C46H54ClN11O7S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-H15E5M	SCHEMBL27031734	5-[(3S)-3-[4-[1-[4-[[5-chloro-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-3-methoxyphenyl]piperidin-4-yl]piperazine-1-carbonyl]pyrrolidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=CC(N2CCC(N3CCN(C(=O)[C@H]4CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)CC3)CC2)=C1	C47H52ClN11O8S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-06P9WK	SCHEMBL27031719	5-[(3R)-3-[4-[1-[4-[[5-chloro-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-3-methoxyphenyl]piperidin-4-yl]piperazine-1-carbonyl]pyrrolidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=CC(N2CCC(N3CCN(C(=O)[C@@H]4CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)CC3)CC2)=C1	C47H52ClN11O8S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-LQI0XE	SCHEMBL24351642	3-[4-[[1-[1-[4-[[5-Chloro-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-3-methoxyphenyl]piperidin-4-yl]piperidin-4-yl]methoxy]phenyl]piperidine-2,6-dione	COC1=CC(N2CCC(N3CCC(COC4=CC=C(C5CCC(=O)NC5=O)C=C4)CC3)CC2)=CC=C1NC1=NC=C(Cl)C(NC2=C3C(=CC=C2)CCN3S(C)(=O)=O)=N1	C42H49ClN8O6S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-W6BECN	SCHEMBL27031713	3-[4-[4-[2-[4-[1-[4-[[5-Bromo-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]piperidin-1-yl]-2-fluorophenyl]piperidine-2,6-dione	COC1=CC(N2CCC(N3CCN(CCC4CCN(C5=CC(F)=C(C6CCC(=O)NC6=O)C=C5)CC4)CC3)CC2)=C(C)C=C1NC1=NC=C(Br)C(NC2=C3C(=CC=C2)CCN3S(C)(=O)=O)=N1	C48H60BrFN10O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-1TKYDB	SCHEMBL27048826	5-[4-[2-[4-[1-[4-[[5-Bromo-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]piperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	COC1=CC(N2CCC(N3CCN(CCC4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)CC2)=C(C)C=C1NC1=NC=C(Br)C(NC2=C3C(=CC=C2)CCN3S(C)(=O)=O)=N1	C50H60BrN11O7S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-YEDVSU	SCHEMBL27048827	3-[4-[2-[4-[1-[4-[[5-Chloro-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-3-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2,6-difluorophenyl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=CC(N2CCC(N3CCN(CCC4=CC(F)=C(C5CCC(=O)NC5=O)C(F)=C4)CC3)CC2)=C1	C42H48ClF2N9O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-NQE3ZD	SCHEMBL27048828	3-[4-[2-[4-[1-[4-[[5-Chloro-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-3-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2,3-difluorophenyl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=CC(N2CCC(N3CCN(CCC4=C(F)C(F)=C(C5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C42H48ClF2N9O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-MSJ7GO	SCHEMBL24351142	3-[4-[3-[[4-[1-[4-[[5-Chloro-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-3-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]methyl]azetidin-1-yl]phenyl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=CC(N2CCC(N3CCN(CC4CN(C5=CC=C(C6CCC(=O)NC6=O)C=C5)C4)CC3)CC2)=C1	C44H53ClN10O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-LGJFKC	SCHEMBL27048829	3-[4-[(3S)-3-[4-[1-[2-fluoro-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazine-1-carbonyl]pyrrolidin-1-yl]phenyl]piperidine-2,6-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC(F)=C(N5CCC(N6CCN(C(=O)[C@H]7CCN(C8=CC=C(C9CCC(=O)NC9=O)C=C8)C7)CC6)CC5)C=C4)=NC4=C3C=CN4)=C21	C46H52FN11O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-V5U8IC	SCHEMBL27048830	3-[4-[(3S)-3-[4-[1-[4-[[5-chloro-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-3-methoxyphenyl]piperidin-4-yl]piperazine-1-carbonyl]pyrrolidin-1-yl]phenyl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=CC(N2CCC(N3CCN(C(=O)[C@H]4CCN(C5=CC=C(C6CCC(=O)NC6=O)C=C5)C4)CC3)CC2)=C1	C45H53ClN10O6S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-MGSZWR	WO2022068849A1_97	.	COC1=C(NC2=NC=C(Cl)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=CC(N2CCC(N3CCN(C(=O)C4CN(C5=CC=C(C6CCC(=O)NC6=O)C=C5)C4)CC3)CC2)=C1	C44H51ClN10O6S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-XO4TEM	SCHEMBL24351147	3-[4-[(3R)-3-[4-[1-[2-fluoro-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazine-1-carbonyl]pyrrolidin-1-yl]phenyl]piperidine-2,6-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC(F)=C(N5CCC(N6CCN(C(=O)[C@@H]7CCN(C8=CC=C(C9CCC(=O)NC9=O)C=C8)C7)CC6)CC5)C=C4)=NC4=C3C=CN4)=C21	C46H52FN11O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-LY5K5Z	SCHEMBL24351139	3-[4-[(3R)-3-[4-[1-[4-[[5-chloro-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-3-methoxyphenyl]piperidin-4-yl]piperazine-1-carbonyl]pyrrolidin-1-yl]phenyl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=CC(N2CCC(N3CCN(C(=O)[C@@H]4CCN(C5=CC=C(C6CCC(=O)NC6=O)C=C5)C4)CC3)CC2)=C1	C45H53ClN10O6S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-O8ZOSE	SCHEMBL27048832	3-[4-[3-[[4-[1-[2-fluoro-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazin-1-yl]methyl]azetidin-1-yl]phenyl]piperidine-2,6-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC(F)=C(N5CCC(N6CCN(CC7CN(C8=CC=C(C9CCC(=O)NC9=O)C=C8)C7)CC6)CC5)C=C4)=NC4=C3C=CN4)=C21	C45H52FN11O4S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-A58A0M	SCHEMBL24351140	3-[7-[2-[4-[1-[4-[[5-chloro-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-3-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]ethoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=CC(N2CCC(N3CCN(CCOC4=CC=CC5=C4CN(C4CCC(=O)NC4=O)C5=O)CC3)CC2)=C1	C44H51ClN10O7S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-BVY436	SCHEMBL24351145	3-[4-[(3R)-3-[[4-[1-[4-[[5-chloro-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-3-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]methyl]pyrrolidin-1-yl]phenyl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=CC(N2CCC(N3CCN(C[C@H]4CCN(C5=CC=C(C6CCC(=O)NC6=O)C=C5)C4)CC3)CC2)=C1	C45H55ClN10O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-GKPDVD	SCHEMBL27048833	3-[4-[2-[4-[1-[2-methoxy-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazin-1-yl]ethyl]phenyl]piperidine-2,6-dione	COC1=CC(NC2=NC(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=C3C=CNC3=N2)=CC=C1N1CCC(N2CCN(CCC3=CC=C(C4CCC(=O)NC4=O)C=C3)CC2)CC1	C44H52N10O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-K9AQIL	SCHEMBL27054910	3-[4-[4-[[4-[4-[[5-Chloro-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-3-methoxyphenyl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]piperidine-2,6-dione	COC1=CC(N2CCN(CC3CCN(C4=CC=C(C5CCC(=O)NC5=O)C=C4)CC3)CC2)=CC=C1NC1=NC(NC2=C3C(=CC=C2)CCN3S(C)(=O)=O)=C(Cl)C=N1	C41H48ClN9O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-8CN6P3	SCHEMBL24351146	2-(2,6-dioxopiperidin-3-yl)-5-[3-[2-[4-[1-[2-fluoro-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazin-1-yl]ethyl]azetidin-1-yl]isoindole-1,3-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC=C(N5CCC(N6CCN(CCC7CN(C8=CC9=C(C=C8)C(=O)N(C8CCC(=O)NC8=O)C9=O)C7)CC6)CC5)C(F)=C4)=NC4=C3C=CN4)=C21	C48H53FN12O6S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-RPDL2T	SCHEMBL24351141	5-[3-[2-[4-[1-[4-[[5-Chloro-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-3-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]azetidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=CC(N2CCC(N3CCN(CCC4CN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)CC3)CC2)=C1	C47H54ClN11O7S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-S7BDC6	SCHEMBL27048834	3-[4-[(3S)-3-[[4-[1-[2-fluoro-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazin-1-yl]methyl]pyrrolidin-1-yl]phenyl]piperidine-2,6-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC=C(N5CCC(N6CCN(C[C@@H]7CCN(C8=CC=C(C9CCC(=O)NC9=O)C=C8)C7)CC6)CC5)C(F)=C4)=NC4=C3C=CN4)=C21	C46H54FN11O4S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-0XCX1L	SCHEMBL24351161	3-[4-[(3R)-3-[[4-[1-[2-fluoro-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazin-1-yl]methyl]pyrrolidin-1-yl]phenyl]piperidine-2,6-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC=C(N5CCC(N6CCN(C[C@H]7CCN(C8=CC=C(C9CCC(=O)NC9=O)C=C8)C7)CC6)CC5)C(F)=C4)=NC4=C3C=CN4)=C21	C46H54FN11O4S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-HAGYE9	SCHEMBL27048835	3-[3-fluoro-4-[2-[4-[1-[2-fluoro-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazin-1-yl]ethyl]phenyl]piperidine-2,6-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC=C(N5CCC(N6CCN(CCC7=CC=C(C8CCC(=O)NC8=O)C=C7F)CC6)CC5)C(F)=C4)=NC4=C3C=CN4)=C21	C43H48F2N10O4S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-5LCNNM	SCHEMBL27048836	3-[4-[2-[4-[1-[4-[[5-Chloro-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-3-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-3-fluorophenyl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=CC(N2CCC(N3CCN(CCC4=CC=C(C5CCC(=O)NC5=O)C=C4F)CC3)CC2)=C1	C42H49ClFN9O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-9NTGM2	SCHEMBL24351152	3-[6-[2-[4-[1-[2-fluoro-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazin-1-yl]ethoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC=C(N5CCC(N6CCN(CCOC7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8)CC6)CC5)C(F)=C4)=NC4=C3C=CN4)=C21	C45H50FN11O6S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-OISCPM	SCHEMBL24351157	3-[6-[2-[4-[1-[4-[[5-chloro-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-3-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]ethoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=CC(N2CCC(N3CCN(CCOC4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5)CC3)CC2)=C1	C44H51ClN10O7S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-KFAYFN	SCHEMBL24351153	3-[5-[4-[2-[4-[1-[2-fluoro-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazin-1-yl]ethyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC(F)=C(N5CCC(N6CCN(CCC7CCN(C8=CC9=C(C=C8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)C=C4)=NC4=C3C=CN4)=C21	C50H59FN12O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-X6IP2J	SCHEMBL24351159	3-[7-[2-[4-[1-[5-methoxy-2-methyl-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazin-1-yl]ethoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	COC1=CC(N2CCC(N3CCN(CCOC4=CC=CC5=C4CN(C4CCC(=O)NC4=O)C5=O)CC3)CC2)=C(C)C=C1NC1=NC(NC2=C3C(=CC=C2)CCN3S(C)(=O)=O)=C2C=CNC2=N1	C47H55N11O7S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-D0AEWS	SCHEMBL24351160	2-(2,6-dioxopiperidin-3-yl)-5-[3-[[4-[1-[5-methoxy-2-methyl-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazin-1-yl]methyl]azetidin-1-yl]isoindole-1,3-dione	COC1=CC(N2CCC(N3CCN(CC4CN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)CC3)CC2)=C(C)C=C1NC1=NC(NC2=C3C(=CC=C2)CCN3S(C)(=O)=O)=C2C=CNC2=N1	C49H56N12O7S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-89D9V3	SCHEMBL27048838	3-[5-[4-[2-[4-[1-[4-[[5-chloro-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-3-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=CC(N2CCC(N3CCN(CCC4CCN(C5=CC6=C(C=C5)CN(C5CCC(=O)NC5=O)C6=O)CC4)CC3)CC2)=C1	C49H60ClN11O6S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-BG3L6Y	SCHEMBL24351156	3-[6-[2-[4-[1-[4-[[5-chloro-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-3-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]ethyl-methylamino]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=CC(N2CCC(N3CCN(CCN(C)C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5)CC3)CC2)=C1	C45H54ClN11O6S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-ELY8M8	SCHEMBL24351162	3-[3-[(3R)-3-[4-[1-[2-fluoro-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazine-1-carbonyl]pyrrolidin-1-yl]phenyl]piperidine-2,6-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC(F)=C(N5CCC(N6CCN(C(=O)[C@@H]7CCN(C8=CC=CC(C9CCC(=O)NC9=O)=C8)C7)CC6)CC5)C=C4)=NC4=C3C=CN4)=C21	C46H52FN11O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-S6MKT8	SCHEMBL24351154	3-[3-[(3R)-3-[4-[1-[4-[[5-chloro-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-3-methoxyphenyl]piperidin-4-yl]piperazine-1-carbonyl]pyrrolidin-1-yl]phenyl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=CC(N2CCC(N3CCN(C(=O)[C@@H]4CCN(C5=CC=CC(C6CCC(=O)NC6=O)=C5)C4)CC3)CC2)=C1	C45H53ClN10O6S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-9RE6TS	SCHEMBL24351164	3-[3-[(3S)-3-[[4-[1-[2-fluoro-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazin-1-yl]methyl]pyrrolidin-1-yl]phenyl]piperidine-2,6-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC(F)=C(N5CCC(N6CCN(C[C@@H]7CCN(C8=CC=CC(C9CCC(=O)NC9=O)=C8)C7)CC6)CC5)C=C4)=NC4=C3C=CN4)=C21	C46H54FN11O4S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-3CT57L	SCHEMBL24351552	3-[3-[(3S)-3-[[4-[1-[4-[[5-chloro-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-3-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]methyl]pyrrolidin-1-yl]phenyl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=CC(N2CCC(N3CCN(C[C@@H]4CCN(C5=CC=CC(C6CCC(=O)NC6=O)=C5)C4)CC3)CC2)=C1	C45H55ClN10O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-FT1IXP	SCHEMBL27048840	3-[5-chloro-2-fluoro-4-[2-[4-[1-[2-fluoro-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazin-1-yl]ethyl]phenyl]piperidine-2,6-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC(F)=C(N5CCC(N6CCN(CCC7=C(Cl)C=C(C8CCC(=O)NC8=O)C(F)=C7)CC6)CC5)C=C4)=NC4=C3C=CN4)=C21	C43H47ClF2N10O4S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-L5UG99	SCHEMBL24351562	3-[5-Chloro-4-[2-[4-[1-[4-[[5-chloro-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-3-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2-fluorophenyl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=CC(N2CCC(N3CCN(CCC4=CC(F)=C(C5CCC(=O)NC5=O)C=C4Cl)CC3)CC2)=C1	C42H48Cl2FN9O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-ZYN11N	SCHEMBL24351567	3-[4-[2-[4-[1-[4-[[5-Chloro-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-3-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]-2-oxoethyl]-2-fluorophenyl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=CC(N2CCC(N3CCN(C(=O)CC4=CC=C(C5CCC(=O)NC5=O)C(F)=C4)CC3)CC2)=C1	C42H47ClFN9O6S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-5QH8FR	SCHEMBL24351569	3-[5-[3-[4-[1-[4-[[5-chloro-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-3-methoxyphenyl]piperidin-4-yl]piperazine-1-carbonyl]azetidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=CC(N2CCC(N3CCN(C(=O)C4CN(C5=CC6=C(C=C5)CN(C5CCC(=O)NC5=O)C6=O)C4)CC3)CC2)=C1	C46H52ClN11O7S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-6F8LYU	SCHEMBL27048841	3-[3-[(3S)-3-[4-[1-[5-methoxy-2-methyl-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazine-1-carbonyl]pyrrolidin-1-yl]phenyl]piperidine-2,6-dione	COC1=CC(N2CCC(N3CCN(C(=O)[C@H]4CCN(C5=CC=CC(C6CCC(=O)NC6=O)=C5)C4)CC3)CC2)=C(C)C=C1NC1=NC(NC2=C3C(=CC=C2)CCN3S(C)(=O)=O)=C2C=CNC2=N1	C48H57N11O6S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-5M6K45	SCHEMBL27048842	3-[4-[2-[4-[1-[5-methoxy-2-methyl-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazin-1-yl]ethyl]phenyl]piperidine-2,6-dione	COC1=CC(N2CCC(N3CCN(CCC4=CC=C(C5CCC(=O)NC5=O)C=C4)CC3)CC2)=C(C)C=C1NC1=NC(NC2=C3C(=CC=C2)CCN3S(C)(=O)=O)=C2C=CNC2=N1	C45H54N10O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-VBIYPF	SCHEMBL24351568	3-[2-fluoro-4-[2-[4-[1-[2-fluoro-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazin-1-yl]-2-oxoethyl]phenyl]piperidine-2,6-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC(F)=C(N5CCC(N6CCN(C(=O)CC7=CC=C(C8CCC(=O)NC8=O)C(F)=C7)CC6)CC5)C=C4)=NC4=C3C=CN4)=C21	C43H46F2N10O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-3DAE1P	SCHEMBL24351564	3-[5-[3-[4-[1-[2-fluoro-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazine-1-carbonyl]azetidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC(F)=C(N5CCC(N6CCN(C(=O)C7CN(C8=CC9=C(C=C8)CN(C8CCC(=O)NC8=O)C9=O)C7)CC6)CC5)C=C4)=NC4=C3C=CN4)=C21	C47H51FN12O6S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-A05LP0	SCHEMBL24351563	3-[2-fluoro-4-[3-[4-[1-[2-fluoro-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazine-1-carbonyl]azetidin-1-yl]phenyl]piperidine-2,6-dione	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC(F)=C(N5CCC(N6CCN(C(=O)C7CN(C8=CC(F)=C(C9CCC(=O)NC9=O)C=C8)C7)CC6)CC5)C=C4)=NC4=C3C=CN4)=C21	C45H49F2N11O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-JJKA7Z	SCHEMBL27048844	3-[4-[3-[4-[1-[4-[[5-Chloro-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-3-methoxyphenyl]piperidin-4-yl]piperazine-1-carbonyl]azetidin-1-yl]-2-fluorophenyl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=CC(N2CCC(N3CCN(C(=O)C4CN(C5=CC(F)=C(C6CCC(=O)NC6=O)C=C5)C4)CC3)CC2)=C1	C44H50ClFN10O6S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-AOTS2Y	WO2022068849A1_132	.	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC(F)=C(N5CCC(N6CCN(C(=O)[C@H]7C[C@@H](OC8=CC=CC(C9CCC(=O)NC9=O)=C8)C7)CC6)CC5)C=C4)=NC4=C3C=CN4)=C21	C46H51FN10O6S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-O1HOQZ	WO2022068849A1_133	.	COC1=C(NC2=NC=C(Cl)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=CC(N2CCC(N3CCN(C(=O)[C@H]4C[C@@H](OC5=CC=CC(C6CCC(=O)NC6=O)=C5)C4)CC3)CC2)=C1	C45H52ClN9O7S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-RD261V	SCHEMBL24351288	3-[4-[2-[4-[1-[4-[[5-chloro-4-[(1-methylsulfonylspiro[2H-indole-3,1'-cyclopropane]-7-yl)amino]pyrimidin-2-yl]amino]-3-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2,6-difluorophenyl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C4C(=CC=C3)C3(CC3)CN4S(C)(=O)=O)=N2)C=CC(N2CCC(N3CCN(CCC4=CC(F)=C(C5CCC(=O)NC5=O)C(F)=C4)CC3)CC2)=C1	C44H50ClF2N9O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-R1PQTJ	SCHEMBL24351280	3-[4-[2-[4-[1-[4-[[5-chloro-4-[(1-methylsulfonylspiro[2H-indole-3,1'-cyclopropane]-7-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2,6-difluorophenyl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C4C(=CC=C3)C3(CC3)CN4S(C)(=O)=O)=N2)C=C(C)C(N2CCC(N3CCN(CCC4=CC(F)=C(C5CCC(=O)NC5=O)C(F)=C4)CC3)CC2)=C1	C45H52ClF2N9O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-1R9M1Y	WO2022068849A1_136	.	COC1=C(NC2=NC=C(Cl)C(NC3=C4C(=CC=C3)C3(CC3)CN4S(C)(=O)=O)=N2)C=C[C]([Ni]2[CH2]CC(N3CCN(CC4CN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)CC3)C[CH2]2)=C1	C48H54ClN10NiO7S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-M26UBN	SCHEMBL24351283	5-[3-[[4-[1-[4-[[5-chloro-4-[(1-methylsulfonylspiro[2H-indole-3,1'-cyclopropane]-7-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]methyl]azetidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C4C(=CC=C3)C3(CC3)CN4S(C)(=O)=O)=N2)C=C(C)C(N2CCC(N3CCN(CC4CN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)CC3)CC2)=C1	C49H56ClN11O7S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-VO5YXQ	SCHEMBL27055608	3-[4-[4-[2-[4-[1-[4-[[5-chloro-4-[(1-methylsulfonylspiro[2H-indole-3,1'-cyclopropane]-7-yl)amino]pyrimidin-2-yl]amino]-3-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]cyclohexyl]-2,6-difluorophenyl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C4C(=CC=C3)C3(CC3)CN4S(C)(=O)=O)=N2)C=CC(N2CCC(N3CCN(CCC4CCC(C5=CC(F)=C(C6CCC(=O)NC6=O)C(F)=C5)CC4)CC3)CC2)=C1	C50H60ClF2N9O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-7TY709	SCHEMBL27048848	5-[(3R)-3-[4-[1-[4-[[5-chloro-4-[(1-methylsulfonylspiro[2H-indole-3,1'-cyclopropane]-7-yl)amino]pyrimidin-2-yl]amino]-3-methoxyphenyl]piperidin-4-yl]piperazine-1-carbonyl]pyrrolidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C4C(=CC=C3)C3(CC3)CN4S(C)(=O)=O)=N2)C=CC(N2CCC(N3CCN(C(=O)[C@@H]4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)CC2)=C1	C49H54ClN11O8S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-4ZISIU	SCHEMBL27048850	3-[4-[4-[2-[4-[1-[4-[[5-chloro-4-[(1-methylsulfonylspiro[2H-indole-3,1'-cyclopropane]-7-yl)amino]pyrimidin-2-yl]amino]-3-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]cyclohexyl]-2-fluorophenyl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C4C(=CC=C3)C3(CC3)CN4S(C)(=O)=O)=N2)C=CC(N2CCC(N3CCN(CCC4CCC(C5=CC=C(C6CCC(=O)NC6=O)C(F)=C5)CC4)CC3)CC2)=C1	C50H61ClFN9O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-BL1WA6	SCHEMBL27048851	2-(2,6-dioxopiperidin-3-yl)-5-[(3R)-3-[4-[1-[5-methoxy-2-methyl-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazine-1-carbonyl]pyrrolidin-1-yl]isoindole-1,3-dione	COC1=CC(N2CCC(N3CCN(C(=O)[C@@H]4CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)CC3)CC2)=C(C)C=C1NC1=NC(NC2=C3C(=CC=C2)CCN3S(C)(=O)=O)=C2C=CNC2=N1	C50H56N12O8S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-MR7XJF	SCHEMBL24351285	3-[2-fluoro-4-[4-[2-[4-[1-[5-methoxy-2-methyl-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazin-1-yl]ethyl]piperidin-1-yl]phenyl]piperidine-2,6-dione	COC1=CC(N2CCC(N3CCN(CCC4CCN(C5=CC=C(C6CCC(=O)NC6=O)C(F)=C5)CC4)CC3)CC2)=C(C)C=C1NC1=NC(NC2=C3C(=CC=C2)CCN3S(C)(=O)=O)=C2C=CNC2=N1	C50H62FN11O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-0A2PKK	WO2022068849A1_143	.	CS(=O)(=O)N1CCC2=CC=CC(NC3=NC(NC4=CC(F)=C(N5CCC(N6CCN(C(=O)[C@H]7C[C@H](OC8=CC=CC(C9CCC(=O)NC9=O)=C8)C7)CC6)CC5)C=C4)=NC4=C3C=CN4)=C21	C46H51FN10O6S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-M47V28	WO2022068849A1_144	.	COC1=C(NC2=NC=C(Cl)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=CC(N2CCC(N3CCN(C(=O)[C@H]4C[C@H](OC5=CC=CC(C6CCC(=O)NC6=O)=C5)C4)CC3)CC2)=C1	C45H52ClN9O7S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-8F4F0K	SCHEMBL27048853	3-[4-[4-[2-[4-[1-[4-[[5-Chloro-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-3-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]piperidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=CC(N2CCC(N3CCN(CCC4CCN(C5=CC(F)=C(C6CCC(=O)NC6=O)C(F)=C5)CC4)CC3)CC2)=C1	C47H57ClF2N10O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-Q8K4CO	SCHEMBL27048854	3-[4-[(3S)-3-[4-[1-[4-[[5-bromo-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazine-1-carbonyl]pyrrolidin-1-yl]phenyl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Br)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=C(C)C(N2CCC(N3CCN(C(=O)[C@H]4CCN(C5=CC=C(C6CCC(=O)NC6=O)C=C5)C4)CC3)CC2)=C1	C46H55BrN10O6S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-AUC255	SCHEMBL27048855	5-[(3S)-3-[4-[1-[4-[[5-bromo-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazine-1-carbonyl]pyrrolidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	COC1=C(NC2=NC=C(Br)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=C(C)C(N2CCC(N3CCN(C(=O)[C@H]4CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)CC3)CC2)=C1	C48H54BrN11O8S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-BBBL2E	SCHEMBL24351916	3-[2,6-difluoro-4-[4-[2-[4-[1-[5-methoxy-2-methyl-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazin-1-yl]ethyl]piperidin-1-yl]phenyl]piperidine-2,6-dione	COC1=CC(N2CCC(N3CCN(CCC4CCN(C5=CC(F)=C(C6CCC(=O)NC6=O)C(F)=C5)CC4)CC3)CC2)=C(C)C=C1NC1=NC(NC2=C3C(=CC=C2)CCN3S(C)(=O)=O)=C2C=CNC2=N1	C50H61F2N11O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-N3VUZ4	SCHEMBL24351915	3-[4-[(3R)-3-[4-[1-[5-methoxy-2-methyl-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazine-1-carbonyl]pyrrolidin-1-yl]phenyl]piperidine-2,6-dione	COC1=CC(N2CCC(N3CCN(C(=O)[C@@H]4CCN(C5=CC=C(C6CCC(=O)NC6=O)C=C5)C4)CC3)CC2)=C(C)C=C1NC1=NC(NC2=C3C(=CC=C2)CCN3S(C)(=O)=O)=C2C=CNC2=N1	C48H57N11O6S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-YO7OMX	WO2022068849A1_150	.	COC1=C(NC2=NC=C(Cl)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=CC(N2CCC(N3CCN(C[C@@H]4CCN(C5=CC=C(C6CCC(=O)NC6=O)C=C5)C4)CC3)CC2)=C1	C45H55ClN10O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-W51BZP	SCHEMBL24351226	5-[3-[[4-[1-[4-[[5-Bromo-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]methyl]azetidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	COC1=C(NC2=NC=C(Br)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=C(C)C(N2CCC(N3CCN(CC4CN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)CC3)CC2)=C1	C47H54BrN11O7S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-FECU4G	SCHEMBL24351114	3-[4-[2-[4-[1-[4-[[5-Bromo-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]anilino]piperidine-2,6-dione	COC1=C(NC2=NC=C(Br)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=C(C)C(N2CCC(N3CCN(CCC4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C43H53BrN10O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-HMNHXY	SCHEMBL27031711	3-[4-[2-[4-[1-[4-[[5-Chloro-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-3-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]anilino]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=CC(N2CCC(N3CCN(CCC4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C42H51ClN10O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-2LTSQS	SCHEMBL27031607	3-[6-[(3S)-3-[[4-[1-[4-[[5-bromo-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]methyl]pyrrolidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Br)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=C(C)C(N2CCC(N3CCN(C[C@@H]4CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6)C4)CC3)CC2)=C1	C48H58BrN11O6S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-ZZ6QFZ	SCHEMBL24352078	3-[4-[2-[4-[1-[4-[[5-Bromo-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2,5-difluorophenyl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Br)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=C(C)C(N2CCC(N3CCN(CCC4=CC(F)=C(C5CCC(=O)NC5=O)C=C4F)CC3)CC2)=C1	C43H50BrF2N9O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-E4YFUE	SCHEMBL27031670	5-[(3R)-3-[[4-[1-[4-[[5-bromo-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]methyl]pyrrolidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	COC1=C(NC2=NC=C(Br)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=C(C)C(N2CCC(N3CCN(C[C@H]4CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)CC3)CC2)=C1	C48H56BrN11O7S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-IPY0KR	SCHEMBL24351619	3-[4-[1-[2-[4-[1-[4-[[5-Bromo-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]piperidin-4-yl]anilino]piperidine-2,6-dione	COC1=C(NC2=NC=C(Br)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=C(C)C(N2CCC(N3CCN(CCN4CCC(C5=CC=C(NC6CCC(=O)NC6=O)C=C5)CC4)CC3)CC2)=C1	C48H62BrN11O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-SAHHY2	SCHEMBL24351696	5-[[3-[4-[1-[4-[[5-Bromo-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazine-1-carbonyl]cyclobutyl]-methylamino]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione; SCHEMBL27141480	COC1=C(NC2=NC=C(Br)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=C(C)C(N2CCC(N3CCN(C(=O)[C@H]4C[C@H](N(C)C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)CC3)CC2)=C1	C49H56BrN11O8S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-WE1MG3	SCHEMBL24351248	3-[6-[3-[[4-[1-[4-[[5-bromo-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]methyl]cyclobutyl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL27131614	COC1=C(NC2=NC=C(Br)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=C(C)C(N2CCC(N3CCN(C[C@H]4C[C@H](C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6)C4)CC3)CC2)=C1	C48H57BrN10O6S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-DENK9G	SCHEMBL24352083	3-[4-[4-[2-[4-[1-[4-[[5-Bromo-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]piperidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=C(N2CCC(N3CCN(CCC4CCN(C5=CC(F)=C(C6CCC(=O)NC6=O)C(F)=C5)CC4)CC3)CC2)C=C(OC)C(NC2=NC(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=C(Br)C=N2)=C1	C49H61BrF2N10O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-B2ZF49	SCHEMBL24351709	5-[4-[4-[1-[4-[[5-Chloro-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-3-methoxyphenyl]piperidin-4-yl]piperazine-1-carbonyl]piperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	COC1=CC(N2CCC(N3CCN(C(=O)C4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)CC2)=CC=C1NC1=NC(NC2=C3C(=CC=C2)CCN3S(C)(=O)=O)=C(Cl)C=N1	C48H54ClN11O8S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-QLMCOB	SCHEMBL24352073	3-[2-fluoro-4-[2-[4-[1-[5-methoxy-2-methyl-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazin-1-yl]ethyl]phenyl]piperidine-2,6-dione	COC1=CC(N2CCC(N3CCN(CCC4=CC(F)=C(C5CCC(=O)NC5=O)C=C4)CC3)CC2)=C(C)C=C1NC1=NC(NC2=C3C(=CC=C2)CCN3S(C)(=O)=O)=C2C=CNC2=N1	C45H53FN10O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-7YYEXI	SCHEMBL24352066	3-[2,6-difluoro-4-[2-[4-[1-[5-methoxy-2-methyl-4-[[4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazin-1-yl]ethyl]phenyl]piperidine-2,6-dione	COC1=CC(N2CCC(N3CCN(CCC4=CC(F)=C(C5CCC(=O)NC5=O)C(F)=C4)CC3)CC2)=C(C)C=C1NC1=NC(NC2=C3C(=CC=C2)CCN3S(C)(=O)=O)=C2C=CNC2=N1	C45H52F2N10O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-38OJUE	SCHEMBL24352080	5-[(3S)-3-[[4-[1-[4-[[5-bromo-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]methyl]pyrrolidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	COC1=C(NC2=NC=C(Br)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=C(C)C(N2CCC(N3CCN(C[C@@H]4CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)CC3)CC2)=C1	C48H56BrN11O7S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-QXJ50R	SCHEMBL24351244	5-[[3-[[4-[1-[4-[[5-Bromo-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]methyl]cyclobutyl]-methylamino]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	COC1=C(NC2=NC=C(Br)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=C(C)C(N2CCC(N3CCN(C[C@H]4C[C@H](N(C)C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)CC3)CC2)=C1	C49H58BrN11O7S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-B41STF	WO2022068849A1_166	.	COC1=C(NC2=NC=C(Br)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)N2)C=C(C)C(N2CCC(N3CCN(CCOC4=CC=CC5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)=C1	C45H53BrN10O8S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-V7P49G	SCHEMBL24351586	5-[4-[4-[1-[4-[[5-Bromo-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]piperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	COC1=C(NC2=NC=C(Br)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=C(C)C(N2CCC(N3CCN(C4CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)CC2)=C1	C48H56BrN11O7S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-GUW7S4	SCHEMBL24351594	3-[6-[(3R)-3-[[4-[1-[4-[[5-bromo-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]methyl]pyrrolidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Br)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=C(C)C(N2CCC(N3CCN(C[C@H]4CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6)C4)CC3)CC2)=C1	C48H58BrN11O6S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-JV7M9F	SCHEMBL27031633	3-[4-[3-[[4-[1-[4-[[5-Bromo-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]methyl]azetidin-1-yl]-2-fluorophenyl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Br)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=C(C)C(N2CCC(N3CCN(CC4CN(C5=CC=C(C6CCC(=O)NC6=O)C(F)=C5)C4)CC3)CC2)=C1	C45H54BrFN10O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-2T8MZH	SCHEMBL24351572	3-[4-[[3-[4-[1-[4-[[5-Bromo-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazine-1-carbonyl]cyclobutyl]-methylamino]phenyl]piperidine-2,6-dione; SCHEMBL27130874	COC1=C(NC2=NC=C(Br)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=C(C)C(N2CCC(N3CCN(C(=O)[C@H]4C[C@H](N(C)C5=CC=C(C6CCC(=O)NC6=O)C=C5)C4)CC3)CC2)=C1	C47H57BrN10O6S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-40W2KS	SCHEMBL24351253	3-[5-[3-[4-[1-[4-[[5-bromo-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazine-1-carbonyl]azetidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Br)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=C(C)C(N2CCC(N3CCN(C(=O)C4CN(C5=CC6=C(C=C5)CN(C5CCC(=O)NC5=O)C6=O)C4)CC3)CC2)=C1	C47H54BrN11O7S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-4SZN7R	SCHEMBL27031618	3-[6-[3-[4-[1-[4-[[5-bromo-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazine-1-carbonyl]azetidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Br)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=C(C)C(N2CCC(N3CCN(C(=O)C4CN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6)C4)CC3)CC2)=C1	C47H54BrN11O7S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-0MFZVQ	SCHEMBL27031686	3-[7-[2-[4-[1-[4-[[5-bromo-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]ethylamino]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Br)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=C(C)C(N2CCC(N3CCN(CCNC4=CC=CC5=C4CN(C4CCC(=O)NC4=O)C5=O)CC3)CC2)=C1	C45H54BrN11O6S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-TQ6KSJ	SCHEMBL24351573	3-[4-[2-[4-[1-[4-[[5-Bromo-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2-chloro-5-fluorophenyl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Br)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=C(C)C(N2CCC(N3CCN(CCC4=C(F)C=C(C5CCC(=O)NC5=O)C(Cl)=C4)CC3)CC2)=C1	C43H50BrClFN9O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-QX00KW	SCHEMBL27031720	3-[6-[4-[[4-[1-[4-[[5-bromo-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Br)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=C(C)C(N2CCC(N3CCN(CC4CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6)CC4)CC3)CC2)=C1	C49H60BrN11O6S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-AUPOO9	SCHEMBL24352295	3-[4-[[3-[[4-[1-[4-[[5-Bromo-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]methyl]cyclobutyl]-methylamino]phenyl]piperidine-2,6-dione; SCHEMBL27129808	COC1=C(NC2=NC=C(Br)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=C(C)C(N2CCC(N3CCN(C[C@H]4C[C@H](N(C)C5=CC=C(C6CCC(=O)NC6=O)C=C5)C4)CC3)CC2)=C1	C47H59BrN10O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-4S1E29	SCHEMBL24351717	3-[3-[4-[4-[1-[4-[[5-Bromo-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]piperidin-1-yl]phenyl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Br)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=C(C)C(N2CCC(N3CCN(C4CCN(C5=CC=CC(C6CCC(=O)NC6=O)=C5)CC4)CC3)CC2)=C1	C46H57BrN10O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-7289UC	SCHEMBL24351671	5-[4-[4-[1-[4-[[5-Chloro-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazine-1-carbonyl]piperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	COC1=CC(N2CCC(N3CCN(C(=O)C4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)CC2)=C(C)C=C1NC1=NC(NC2=C3C(=CC=C2)CCN3S(C)(=O)=O)=C(Cl)C=N1	C49H56ClN11O8S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-966PLS	SCHEMBL24351890	3-[5-[3-[[4-[1-[4-[[5-bromo-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]methyl]azetidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Br)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=C(C)C(N2CCC(N3CCN(CC4CN(C5=CC6=C(C=C5)CN(C5CCC(=O)NC5=O)C6=O)C4)CC3)CC2)=C1	C47H56BrN11O6S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-JR4HCK	WO2022068849A1_181	.	COC1=C(NC2=NC=C(C)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=C(C)C(N2CCC(N3CCN(CC4CCN(C5=CC(F)=C(C6CCC(=O)NC6=O)C(F)=C5)CC4)CC3)CC2)=C1	C48H60F2N10O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-GFED5P	SCHEMBL27031658	3-[4-[3-[4-[1-[4-[[5-Bromo-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]cyclobutyl]anilino]piperidine-2,6-dione	COC1=C(NC2=NC=C(Br)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=C(C)C(N2CCC(N3CCN(C4CC(C5=CC=C(NC6CCC(=O)NC6=O)C=C5)C4)CC3)CC2)=C1	C45H55BrN10O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-WV2NFJ	SCHEMBL27031691	3-[4-[2-[4-[1-[4-[[5-Bromo-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]phenyl]-3-methylpiperidine-2,6-dione	COC1=C(NC2=NC=C(Br)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=C(C)C(N2CCC(N3CCN(CCC4=CC=C(C5(C)CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C44H54BrN9O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-5STO3T	SCHEMBL24351673	3-[4-[3-[[4-[1-[4-[[5-Bromo-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]methyl]azetidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Br)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=C(C)C(N2CCC(N3CCN(CC4CN(C5=CC(F)=C(C6CCC(=O)NC6=O)C(F)=C5)C4)CC3)CC2)=C1	C45H53BrF2N10O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-GE17UA	SCHEMBL27031675	3-[4-[2-[4-[1-[4-[[5-Bromo-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]-3-oxopiperazin-1-yl]ethyl]-2,6-difluorophenyl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Br)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=C(C)C(N2CCC(N3CCN(CCC4=CC(F)=C(C5CCC(=O)NC5=O)C(F)=C4)CC3=O)CC2)=C1	C43H48BrF2N9O6S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-2SSAJQ	SCHEMBL24351668	3-[4-[4-[2-[4-[1-[4-[[5-Bromo-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]-3-oxopiperazin-1-yl]ethyl]piperidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Br)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=C(C)C(N2CCC(N3CCN(CCC4CCN(C5=CC(F)=C(C6CCC(=O)NC6=O)C(F)=C5)CC4)CC3=O)CC2)=C1	C48H57BrF2N10O6S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-YWHUV6	SCHEMBL24351676	3-[4-[3-[4-[1-[4-[[5-Bromo-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazine-1-carbonyl]pyrrolidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Br)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=C(C)C(N2CCC(N3CCN(C(=O)C4CCN(C5=CC(F)=C(C6CCC(=O)NC6=O)C(F)=C5)C4)CC3)CC2)=C1	C46H53BrF2N10O6S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-OU35FY	SCHEMBL24351169	3-[4-[3-[4-[1-[4-[[5-Bromo-4-[(1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazine-1-carbonyl]azetidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Br)C(NC3=C4C(=CC=C3)CCN4S(C)(=O)=O)=N2)C=C(C)C(N2CCC(N3CCN(C(=O)C4CN(C5=CC(F)=C(C6CCC(=O)NC6=O)C(F)=C5)C4)CC3)CC2)=C1	C45H51BrF2N10O6S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-NOF049	SCHEMBL24351180	3-[4-[2-[4-[1-[4-[[5-Bromo-4-[(4-ethyl-1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C4C(=C(CC)C=C3)CCN4S(C)(=O)=O)=N2)=C(OC)C=C1N1CCC(N2CCN(CCC3=CC(F)=C(C4CCC(=O)NC4=O)C(F)=C3)CC2)CC1	C46H56BrF2N9O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-10S2N3	SCHEMBL27031721	3-[4-[2-[4-[1-[4-[[5-Bromo-4-[(4-cyclopropyl-1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C4C(=C(C5CC5)C=C3)CCN4S(C)(=O)=O)=N2)=C(OC)C=C1N1CCC(N2CCN(CCC3=CC(F)=C(C4CCC(=O)NC4=O)C(F)=C3)CC2)CC1	C47H56BrF2N9O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-FY6J7K	SCHEMBL27031718	(3R)-3-[4-[(3R)-3-[4-[1-[4-[[5-bromo-4-[(4-fluoro-1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazine-1-carbonyl]pyrrolidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C4C(=C(F)C=C3)CCN4S(C)(=O)=O)=N2)=C(OC)C=C1N1CCC(N2CCN(C(=O)[C@@H]3CCN(C4=CC(F)=C([C@H]5CCC(=O)NC5=O)C(F)=C4)C3)CC2)CC1	C47H54BrF3N10O6S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-MESH75	SCHEMBL27031716	(3R)-3-[4-[2-[4-[1-[4-[[5-bromo-4-[(4-fluoro-1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C4C(=C(F)C=C3)CCN4S(C)(=O)=O)=N2)=C(OC)C=C1N1CCC(N2CCN(CCC3=CC(F)=C([C@H]4CCC(=O)NC4=O)C(F)=C3)CC2)CC1	C44H51BrF3N9O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-BTW99U	SCHEMBL27031743	(3R)-3-[4-[3-[4-[1-[4-[[5-bromo-4-[[1-methylsulfonyl-4-(trifluoromethyl)-2,3-dihydroindol-7-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazine-1-carbonyl]azetidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=C(N2CCC(N3CCN(C(=O)C4CN(C5=CC(F)=C([C@H]6CCC(=O)NC6=O)C(F)=C5)C4)CC3)CC2)C=C(OC)C(NC2=NC=C(Br)C(NC3=C4C(=C(C(F)(F)F)C=C3)CCN4S(C)(=O)=O)=N2)=C1	C47H52BrF5N10O6S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-T3TSM9	SCHEMBL24351174	(3R)-3-[4-[(3R)-3-[4-[1-[4-[[5-bromo-4-[[1-methylsulfonyl-4-(trifluoromethyl)-2,3-dihydroindol-7-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazine-1-carbonyl]pyrrolidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=C(N2CCC(N3CCN(C(=O)[C@@H]4CCN(C5=CC(F)=C([C@H]6CCC(=O)NC6=O)C(F)=C5)C4)CC3)CC2)C=C(OC)C(NC2=NC=C(Br)C(NC3=C4C(=C(C(F)(F)F)C=C3)CCN4S(C)(=O)=O)=N2)=C1	C48H54BrF5N10O6S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-PKA4WX	SCHEMBL24351183	(3R)-3-[4-[(3R)-3-[4-[1-[4-[[5-bromo-4-[(4-ethyl-1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazine-1-carbonyl]pyrrolidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC=C(NC2=NC(NC3=CC(CC)=C(N4CCC(N5CCN(C(=O)[C@@H]6CCN(C7=CC(F)=C([C@H]8CCC(=O)NC8=O)C(F)=C7)C6)CC5)CC4)C=C3OC)=NC=C2Br)C2=C1CCN2S(C)(=O)=O	C49H59BrF2N10O6S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-O4LNRO	SCHEMBL27031609	(3R)-3-[4-[2-[4-[1-[4-[[5-bromo-4-[[4-(dimethylamino)-1-methylsulfonyl-2,3-dihydroindol-7-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=C(N2CCC(N3CCN(CCC4=CC(F)=C([C@H]5CCC(=O)NC5=O)C(F)=C4)CC3)CC2)C=C(OC)C(NC2=NC=C(Br)C(NC3=C4C(=C(N(C)C)C=C3)CCN4S(C)(=O)=O)=N2)=C1	C46H57BrF2N10O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-1OF3XJ	SCHEMBL24351173	(3R)-3-[4-[2-[4-[1-[4-[[5-bromo-4-[(4-ethyl-1-methylsulfonyl-2,3-dihydroindol-7-yl)amino]pyrimidin-2-yl]amino]-5-ethoxy-2-ethylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2,6-difluorophenyl]piperidine-2,6-dione	CCOC1=C(NC2=NC=C(Br)C(NC3=C4C(=C(CC)C=C3)CCN4S(C)(=O)=O)=N2)C=C(CC)C(N2CCC(N3CCN(CCC4=CC(F)=C([C@H]5CCC(=O)NC5=O)C(F)=C4)CC3)CC2)=C1	C47H58BrF2N9O5S	EGFR	P00533	CRBN	WO-2022068849-A1
TPD-1AGN0W	SCHEMBL24414421	3-Chloro-5-[5-[4-[5-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]pentyl]phenyl]-8-oxo-6-sulfanylidene-5,7-diazaspiro[3.4]octan-7-yl]pyridine-2-carbonitrile	N#CC1=NC=C(N2C(=O)C3(CCC3)N(C3=CC=C(CCCCCN4CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)C2=S)C=C1Cl	C40H39ClN8O5S	AR	P10275	CRBN	WO-2022098544-A1
TPD-9CBLBF	WO2022098544A1_2	.	N#CC1=NC=C(N2C(=O)N(C3=CC=C(N4CCC(CN5CCN(C6=CC7=C(C=C6)CN(C6CCC(=O)NC6=O)C7=O)CC5)CC4)C=C3)C3(CCC3)C2=O)C=C1Cl	C41H42ClN9O5	AR	P10275	CRBN	WO-2022098544-A1
TPD-UBC1Y9	SCHEMBL24414428	4-[3-[[6-[4-[[4-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]pyridin-3-yl]methyl]-4,4-dimethyl-5-oxo-2-sulfanylideneimidazolidin-1-yl]-2-(trifluoromethyl)benzonitrile	CC1(C)C(=O)N(C2=CC=C(C#N)C(C(F)(F)F)=C2)C(=S)N1CC1=CC=C(N2CCC(CN3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)N=C1	C42H42F3N9O5S	AR	P10275	CRBN	WO-2022098544-A1
TPD-WUTW8J	WO2022098544A1_4	.	CCN(CC1CCN(C2=NC=C(CN3C(=O)N(C4=CC=C(C#N)C(C(F)(F)F)=C4)C(=O)C3(C)C)C=C2)CC1)[C@H]1C[C@H](OC2=CC=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=C2)C1	C44H45F3N8O7	AR	P10275	CRBN	WO-2022098544-A1
TPD-S8HAF6	SCHEMBL24414437	2-Chloro-4-[5-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]-3-fluorophenyl]-8-oxo-6-sulfanylidene-5,7-diazaspiro[3.4]octan-7-yl]benzonitrile; SCHEMBL29632691	N#CC1=CC=C(N2C(=O)C3(CCC3)N(C3=CC(F)=C(N4CCC(CN5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C=C3)C2=S)C=C1Cl	C42H40ClFN8O5S	AR	P10275	CRBN	WO-2022098544-A1
TPD-FWIJ48	SCHEMBL24414395	4-[5-[4-[4-[[4-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]-3-fluorophenyl]-8-oxo-6-sulfanylidene-5,7-diazaspiro[3.4]octan-7-yl]-2-methoxybenzonitrile; SCHEMBL29632753	COC1=CC(N2C(=O)C3(CCC3)N(C3=CC(F)=C(N4CCC(CN5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C=C3)C2=S)=CC=C1C#N	C43H43FN8O6S	AR	P10275	CRBN	WO-2022098544-A1
TPD-DBUQU4	SCHEMBL24414405	4-[5-[4-[4-[[4-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]-8-oxo-6-sulfanylidene-5,7-diazaspiro[3.4]octan-7-yl]-2-methoxybenzonitrile	COC1=CC(N2C(=O)C3(CCC3)N(C3=CC=C(N4CCC(CN5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C=C3)C2=S)=CC=C1C#N	C43H44N8O6S	AR	P10275	CRBN	WO-2022098544-A1
TPD-BHMH1V	SCHEMBL24414436	5-[5-[6-[3-[[[3-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxycyclobutyl]-propan-2-ylamino]methyl]cyclobutyl]oxypyridin-3-yl]-8-oxo-6-sulfanylidene-5,7-diazaspiro[3.4]octan-7-yl]-3-(trifluoromethyl)pyridine-2-carbonitrile	CC(C)N(C[C@H]1C[C@H](OC2=NC=C(N3C(=S)N(C4=CN=C(C#N)C(C(F)(F)F)=C4)C(=O)C34CCC4)C=C2)C1)[C@H]1C[C@H](OC2=CC3=C(C=C2)C(=O)N(C2CCC(=O)NC2=O)C3=O)C1	C43H41F3N8O7S	AR	P10275	CRBN	WO-2022098544-A1
TPD-EUVVV4	SCHEMBL24414396	2-Chloro-4-[5-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]-8-oxo-6-sulfanylidene-5,7-diazaspiro[3.4]octan-7-yl]benzonitrile; SCHEMBL29632738	N#CC1=CC=C(N2C(=O)C3(CCC3)N(C3=CC=C(N4CCC(CN5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C=C3)C2=S)C=C1Cl	C42H41ClN8O5S	AR	P10275	CRBN	WO-2022098544-A1
TPD-HS7THX	SCHEMBL24414433	3-Chloro-5-[5-[4-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperidin-4-yl]oxy-3-fluorophenyl]-8-oxo-6-sulfanylidene-5,7-diazaspiro[3.4]octan-7-yl]pyridine-2-carbonitrile	N#CC1=NC=C(N2C(=O)C3(CCC3)N(C3=CC=C(OC4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C(F)=C3)C2=S)C=C1Cl	C42H40ClFN8O6S	AR	P10275	CRBN	WO-2022098544-A1
TPD-6E6CSI	WO2022098544A1_11	.	N#CC1=CC=C(N2C(=O)C3(CCC3)N(C3=CC=C(N4CCC(CC5CCN(C6=CC=C7CN(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C=C3)C2=S)C=C1Cl	C43H44ClN7O4S	AR	P10275	CRBN	WO-2022098544-A1
TPD-XCGXF2	SCHEMBL24414434	5-[5-[6-[1-[[1-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperidin-4-yl]oxypyridin-3-yl]-8-oxo-6-sulfanylidene-5,7-diazaspiro[3.4]octan-7-yl]-3-(trifluoromethyl)pyridine-2-carbonitrile	N#CC1=NC=C(N2C(=O)C3(CCC3)N(C3=CN=C(OC4CCN(CC5CCN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)C=C3)C2=S)C=C1C(F)(F)F	C42H40F3N9O6S	AR	P10275	CRBN	WO-2022098544-A1
TPD-ZHSC1S	SCHEMBL24411045	5-[5-[6-[4-[[[3-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxycyclobutyl]-propan-2-ylamino]methyl]piperidin-1-yl]pyridin-3-yl]-8-oxo-6-sulfanylidene-5,7-diazaspiro[3.4]octan-7-yl]-3-(trifluoromethyl)pyridine-2-carbonitrile	CC(C)N(CC1CCN(C2=NC=C(N3C(=S)N(C4=CN=C(C#N)C(C(F)(F)F)=C4)C(=O)C34CCC4)C=C2)CC1)[C@H]1C[C@H](OC2=CC3=C(C=C2)C(=O)N(C2CCC(=O)NC2=O)C3=O)C1	C44H44F3N9O6S	AR	P10275	CRBN	WO-2022098544-A1
TPD-Y86TKW	SCHEMBL24411056	4-[3-[[6-[2-[4-[[4-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]ethoxy]pyridin-3-yl]methyl]-4,4-dimethyl-5-oxo-2-sulfanylideneimidazolidin-1-yl]-2-(trifluoromethyl)benzonitrile	CC1(C)C(=O)N(C2=CC=C(C#N)C(C(F)(F)F)=C2)C(=S)N1CC1=CN=C(OCCN2CCC(CN3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)C=C1	C44H46F3N9O6S	AR	P10275	CRBN	WO-2022098544-A1
TPD-4SVI2F	SCHEMBL24411062	4-[3-[4-[[4-[[[3-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxycyclobutyl]-propan-2-ylamino]methyl]piperidin-1-yl]methyl]phenyl]-2-oxobenzimidazol-1-yl]-2-(trifluoromethyl)benzonitrile	CC(C)N(CC1CCN(CC2=CC=C(N3C(=O)N(C4=CC=C(C#N)C(C(F)(F)F)=C4)C4=C3C=CC=C4)C=C2)CC1)[C@H]1C[C@H](OC2=CC=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=C2)C1	C48H46F3N7O6	AR	P10275	CRBN	WO-2022098544-A1
TPD-94XNRL	SCHEMBL24411055	4-[3-[[6-[2-[4-[[[3-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxycyclobutyl]-ethylamino]methyl]piperidin-1-yl]ethoxy]pyridin-3-yl]methyl]-4,4-dimethyl-5-oxo-2-sulfanylideneimidazolidin-1-yl]-2-(trifluoromethyl)benzonitrile	CCN(CC1CCN(CCOC2=CC=C(CN3C(=S)N(C4=CC=C(C#N)C(C(F)(F)F)=C4)C(=O)C3(C)C)C=N2)CC1)[C@H]1C[C@H](OC2=CC=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=C2)C1	C46H49F3N8O7S	AR	P10275	CRBN	WO-2022098544-A1
TPD-4OCFSY	SCHEMBL24414484	4-[3-[2-[4-[4-[[[3-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxycyclobutyl]-propan-2-ylamino]methyl]piperidin-1-yl]phenyl]ethyl]-2-oxobenzimidazol-1-yl]-2-(trifluoromethyl)benzonitrile	CC(C)N(CC1CCN(C2=CC=C(CCN3C(=O)N(C4=CC=C(C#N)C(C(F)(F)F)=C4)C4=C3C=CC=C4)C=C2)CC1)[C@H]1C[C@H](OC2=CC=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=C2)C1	C49H48F3N7O6	AR	P10275	CRBN	WO-2022098544-A1
TPD-USZ6ZK	SCHEMBL24411070	4-(4-Cyanophenyl)-1-[[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]methyl]-2,5-dimethylpyrrole-3-carbonitrile	CC1=C(C#N)C(C2=CC=C(C#N)C=C2)=C(C)N1CC1=CC=C(N2CCC(CN3CCN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)C=C1	C44H44N8O4	AR	P10275	CRBN	WO-2022098544-A1
TPD-6166VC	SCHEMBL24414598	4-(4-Cyanophenyl)-1-[[4-[3-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]propoxy]phenyl]methyl]-2,5-dimethylpyrrole-3-carbonitrile	CC1=C(C#N)C(C2=CC=C(C#N)C=C2)=C(C)N1CC1=CC=C(OCCCN2CCC(CN3CCN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)C=C1	C47H50N8O5	AR	P10275	CRBN	WO-2022098544-A1
TPD-6EIXPG	WO2022098544A1_20	.	CC1=C(C#N)C(C2=CC=C(C#N)C=C2)=C(C)N1CC1=CC=C(OCCN2CCC(CN3CCN(C4=CC5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5C=C4)CC3)CC2)C=C1	C46H50N8O5	AR	P10275	CRBN	WO-2022098544-A1
TPD-OJ1LCY	SCHEMBL24414651	4-(4-Cyanophenyl)-1-[[4-[2-[2-[2-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]ethoxy]ethoxy]ethoxy]phenyl]methyl]-2,5-dimethylpyrrole-3-carbonitrile	CC1=C(C#N)C(C2=CC=C(C#N)C=C2)=C(C)N1CC1=CC=C(OCCOCCOCCN2CCC(CN3CCN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)C=C1	C50H56N8O7	AR	P10275	CRBN	WO-2022098544-A1
TPD-O69Y9F	SCHEMBL24414429	4-(4-Cyanophenyl)-1-[[4-[2-[2-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]ethoxy]ethoxy]phenyl]methyl]-2,5-dimethylpyrrole-3-carbonitrile	CC1=C(C#N)C(C2=CC=C(C#N)C=C2)=C(C)N1CC1=CC=C(OCCOCCN2CCC(CN3CCN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)C=C1	C48H52N8O6	AR	P10275	CRBN	WO-2022098544-A1
TPD-0BBMXD	SCHEMBL24411039	4-[3-[3-[4-[[[3-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxycyclobutyl]-propan-2-ylamino]methyl]piperidin-1-yl]propyl]-2-oxobenzimidazol-1-yl]-2-(trifluoromethyl)benzonitrile	CC(C)N(CC1CCN(CCCN2C(=O)N(C3=CC=C(C#N)C(C(F)(F)F)=C3)C3=C2C=CC=C3)CC1)[C@H]1C[C@H](OC2=CC=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=C2)C1	C44H46F3N7O6	AR	P10275	CRBN	WO-2022098544-A1
TPD-Z77XC9	SCHEMBL24414451	4-[3-[4-[4-[[[3-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxycyclobutyl]-propan-2-ylamino]methyl]piperidin-1-yl]butyl]-2-oxobenzimidazol-1-yl]-2-(trifluoromethyl)benzonitrile	CC(C)N(CC1CCN(CCCCN2C(=O)N(C3=CC=C(C#N)C(C(F)(F)F)=C3)C3=C2C=CC=C3)CC1)[C@H]1C[C@H](OC2=CC=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=C2)C1	C45H48F3N7O6	AR	P10275	CRBN	WO-2022098544-A1
TPD-TD7TWT	SCHEMBL24411104	4-[3-[[4-[4-[[[3-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxycyclobutyl]-propan-2-ylamino]methyl]piperidin-1-yl]phenyl]methyl]-2-oxobenzimidazol-1-yl]-2-(trifluoromethyl)benzonitrile	CC(C)N(CC1CCN(C2=CC=C(CN3C(=O)N(C4=CC=C(C#N)C(C(F)(F)F)=C4)C4=C3C=CC=C4)C=C2)CC1)[C@H]1C[C@H](OC2=CC=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=C2)C1	C48H46F3N7O6	AR	P10275	CRBN	WO-2022098544-A1
TPD-JDWZUM	WO2022101603A1_(R,S)-SIM1	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](CC(C)(C)C)NC(=O)COCC(C)(COCCOCCOCCNC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)COCCOCCOCCNC(=O)C[C@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)cc1	C80H100Cl2N14O13S3	BRD2	P25440	VHL	WO-2022101603-A1
TPD-WLEPWP	WO2022101603A1_cis-SIM1	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@H](O)CN2C(=O)[C@H](CC(C)(C)C)NC(=O)COCC(C)(COCCOCCOCCNC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)COCCOCCOCCNC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)cc1	C80H100Cl2N14O13S3	BRD2	P25440	VHL	WO-2022101603-A1
TPD-4BAM0Q	WO2022101603A1_SIM1	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](C)NC(=O)COCC(C)(COCCOCCOCCNC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)COCCOCCOCCNC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)cc1	C76H92Cl2N14O13S3	BRD2	P25440	VHL	WO-2022101603-A1
TPD-899NR9	WO2022101603A1_SIM3	.	CC1=C(C)C2=C(C1)n1c(C)nnc1[C@H](CC(=O)NCCOCCOCCOCCOCC(C)(COCCOCCOCCOCCNC(O)C[C@@H]1N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc31)COCC(=O)N[C@@H](C)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(-c3scnc3C)cc1)N=C2c1ccc(Cl)cc1	C81H104Cl2N14O15S2	BRD2	P25440	VHL	WO-2022101603-A1
TPD-ELJCZX	SIM4	2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]-N-[2-[2-[2-[2-[2-[2-[2-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]ethoxy]ethoxy]ethoxymethyl]-3-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethylamino]-2-oxoethoxy]-2-methylpropoxy]ethoxy]ethoxy]ethyl]acetamide; SCHEMBL29780162	Cc1sc2c(c1C)C(c1ccc(Cl)cc1)=N[C@@H](CC(=O)NCCOCCOCCOCC(C)(COCCOCCOCCNC(=O)C[C@@H]1N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc31)COCC(=O)NCCNc1cccc3c1C(=O)N(C1CCC(=O)NC1=O)C3=O)c1nnc(C)n1-2	C72H84Cl2N14O14S2	BRD2	P25440	VHL	WO-2022101603-A1
TPD-U04HJY	SCHEMBL29780164	2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]-N-[2-[2-[2-[2-[2-[2-[2-[2-[2-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]ethoxy]ethoxy]ethoxy]ethoxymethyl]-3-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethylamino]-2-oxoethoxy]-2-methylpropoxy]ethoxy]ethoxy]ethoxy]ethyl]acetamide	Cc1sc2c(c1C)C(c1ccc(Cl)cc1)=N[C@@H](CC(=O)NCCOCCOCCOCCOCC(C)(COCCOCCOCCOCCNC(=O)C[C@@H]1N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc31)COCC(=O)NCCNc1cccc3c1C(=O)N(C1CCC(=O)NC1=O)C3=O)c1nnc(C)n1-2	C76H92Cl2N14O16S2	BRD2	P25440	VHL	WO-2022101603-A1
TPD-TWXME3	SCHEMBL24480224	5-chloro-N-[2-chloro-4-(trifluoromethyl)phenyl]-2-[[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]sulfonylamino]benzamide; SCHEMBL29579009	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CC5CCN(S(=O)(=O)NC6=C(C(=O)NC7=C(Cl)C=C(C(F)(F)F)C=C7)C=C(Cl)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C37H36Cl2F3N7O7S	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-A3GG88	SCHEMBL24480225	N-[4-chloro-2-[4-chloro-6-(trifluoromethyl)-1H-benzimidazol-2-yl]phenyl]-4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperazine-1-sulfonamide; SCHEMBL29578874	O=C1CCC(N2C(=O)C3=CC=C(N4CC(N5CCN(S(=O)(=O)NC6=CC=C(Cl)C=C6C6=NC7=C(N6)C(Cl)=CC(C(F)(F)F)=C7)CC5)C4)C=C3C2=O)C(=O)N1	C34H29Cl2F3N8O6S	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-5O17JY	SCHEMBL24480286	5-chloro-N-[2-chloro-4-(trifluoromethyl)phenyl]-2-[[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]sulfonylamino]benzamide	O=C1CCC(N2C(=O)C3=CC=C(N4CCC(CN5CCN(S(=O)(=O)NC6=C(C(=O)NC7=C(Cl)C=C(C(F)(F)F)C=C7)C=C(Cl)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C37H36Cl2F3N7O7S	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-321RLT	SCHEMBL24480260	3-Chloro-2-(2-chloroethoxy)-5-[2-[4-[[2-[4-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]azetidin-3-yl]piperazin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL29578422	CC(C)(C1=CC=C(OCC2=NC(N3CCN(C4CN(C5CN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)C4)CC3)=NC=C2)C=C1)C1=CC(Cl)=C(OCCCl)C(C#N)=C1	C46H47Cl2N9O6	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-52GJIU	SCHEMBL24480488	3-Chloro-2-(2-chloroethoxy)-5-[2-[4-[[2-[4-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperidin-4-yl]piperazin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL31236705	CC(C)(C1=CC=C(OCC2=NC(N3CCN(C4CCN(C5CN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)=NC=C2)C=C1)C1=CC(C#N)=C(OCCCl)C(Cl)=C1	C48H51Cl2N9O6	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-0YSW66	SCHEMBL24480683	3-Chloro-2-(2-chloroethoxy)-5-[2-[4-[[2-[4-[1-[1-[[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-4-yl]methyl]azetidin-3-yl]piperidin-4-yl]piperazin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile	CN1C(=O)N(C2CCC(=O)NC2=O)C2=C1C(CN1CC(N3CCC(N4CCN(C5=NC=CC(COC6=CC=C(C(C)(C)C7=CC(C#N)=C(OCCCl)C(Cl)=C7)C=C6)=N5)CC4)CC3)C1)=CC=C2	C49H56Cl2N10O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-TCQX2S	SCHEMBL24480672	3-Chloro-2-(2-chloroethoxy)-5-[2-[4-[[2-[4-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperidin-4-yl]piperazin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL29578674	CC(C)(C1=CC=C(OCC2=NC(N3CCN(C4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)CC3)=NC=C2)C=C1)C1=CC(C#N)=C(OCCCl)C(Cl)=C1	C51H57Cl2N9O6	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-Z1N52N	SCHEMBL24480998	3-Chloro-2-(2-chloroethoxy)-5-[2-[4-[[2-[4-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperidin-4-yl]methyl]piperidin-4-yl]piperazin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile	CC(C)(C1=CC=C(OCC2=NC(N3CCN(C4CCN(CC5CCN(C6=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)CC5)CC4)CC3)=NC=C2)C=C1)C1=CC(C#N)=C(OCCCl)C(Cl)=C1	C51H57Cl2N9O6	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-G968OI	SCHEMBL24480460	3-Chloro-5-[2-[4-[[2-[4-[1-[1-[[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-4-yl]methyl]azetidin-3-yl]piperidin-4-yl]piperazin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL29579359	CN1C(=O)N(C2CCC(=O)NC2=O)C2=C1C(CN1CC(N3CCC(N4CCN(C5=NC=CC(COC6=CC=C(C(C)(C)C7=CC(C#N)=CC(Cl)=C7)C=C6)=N5)CC4)CC3)C1)=CC=C2	C47H53ClN10O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-AUSFL9	SCHEMBL24480449	3-Chloro-5-[2-[4-[[2-[4-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperidin-4-yl]piperazin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL29578859	CC(C)(C1=CC=C(OCC2=NC(N3CCN(C4CCN(C5CN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)=NC=C2)C=C1)C1=CC(C#N)=CC(Cl)=C1	C46H48ClN9O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-X8XJSX	SCHEMBL24481232	3-Chloro-2-(2-chloroethoxy)-5-[2-[4-[[2-[4-[[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperidin-4-yl]methyl]piperazin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL29579161	CC(C)(C1=CC=C(OCC2=CC=NC(N3CCN(CC4CCN(C5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)CC3)=N2)C=C1)C1=CC(Cl)=C(OCCCl)C(C#N)=C1	C51H57Cl2N9O6	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-VWLTLJ	SCHEMBL24481188	3-Chloro-2-(2-chloroethoxy)-5-[2-[4-[[2-[4-[[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperidin-4-yl]piperidin-4-yl]methyl]piperazin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL29579210	CC(C)(C1=CC=C(OCC2=CC=NC(N3CCN(CC4CCN(C5CCN(C6=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)CC5)CC4)CC3)=N2)C=C1)C1=CC(Cl)=C(OCCCl)C(C#N)=C1	C51H57Cl2N9O6	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-MLGKAE	SCHEMBL24480365	3-Chloro-2-(2-chloroethoxy)-5-[2-[4-[[2-[4-[[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL29579028	CC(C)(C1=CC=C(OCC2=CC=NC(N3CCN(CC4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)CC3)=N2)C=C1)C1=CC(Cl)=C(OCCCl)C(C#N)=C1	C52H59Cl2N9O6	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-THKVNC	SCHEMBL24480700	3-Chloro-2-(2-chloroethoxy)-5-[2-[4-[[2-[4-[[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperidin-4-yl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile	CC(C)(C1=CC=C(OCC2=CC=NC(N3CCN(CC4CCN(CC5CCN(C6=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)CC5)CC4)CC3)=N2)C=C1)C1=CC(Cl)=C(OCCCl)C(C#N)=C1	C52H59Cl2N9O6	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-UW68UD	SCHEMBL24481003	3-Chloro-2-(2-chloroethoxy)-5-[2-[4-[[2-[4-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperidin-4-yl]methyl]piperidin-4-yl]piperidin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL31236678	CC(C)(C1=CC=C(OCC2=NC(N3CCC(C4CCN(CC5CCN(C6=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)CC5)CC4)CC3)=NC=C2)C=C1)C1=CC(C#N)=C(OCCCl)C(Cl)=C1	C52H58Cl2N8O6	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-D78IZM	SCHEMBL29578914	5-[2-[4-[[2-[(3aS,6aR)-2-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperidin-4-yl]-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-5-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]-3-chloro-2-(2-chloroethoxy)benzonitrile	[H][C@@]12CN(C3=NC=CC(COC4=CC=C(C(C)(C)C5=CC(C#N)=C(OCCCl)C(Cl)=C5)C=C4)=N3)C[C@]1([H])CN(C1CCN(CC3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC1)C2	C53H59Cl2N9O6	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-LGQVQ4	SCHEMBL24481027	5-[2-[4-[[2-[(3aR,6aS)-2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperidin-4-yl]-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-5-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]-3-chloro-2-(2-chloroethoxy)benzonitrile; SCHEMBL29578658	[H][C@@]12CN(C3=NC=CC(COC4=CC=C(C(C)(C)C5=CC(C#N)=C(OCCCl)C(Cl)=C5)C=C4)=N3)C[C@]1([H])CN(C1CCN(C3CN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)C3)CC1)C2	C50H53Cl2N9O6	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-GBGB6X	SCHEMBL24481032	3-Chloro-5-[2-[4-[[2-[4-[1-[1-[[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-4-yl]methyl]azetidin-3-yl]piperidin-4-yl]piperazin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]-2-ethoxybenzonitrile; SCHEMBL29578956	CCOC1=C(C#N)C=C(C(C)(C)C2=CC=C(OCC3=NC(N4CCN(C5CCN(C6CN(CC7=CC=CC8=C7N(C)C(=O)N8C7CCC(=O)NC7=O)C6)CC5)CC4)=NC=C3)C=C2)C=C1Cl	C49H57ClN10O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-WWKROG	SCHEMBL24480487	3-Chloro-2-(2-chloroethoxy)-5-[2-[4-[[2-[4-[[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL31236674	CC(C)(C1=CC=C(OCC2=CC=NC(N3CCN(CC4CCN(CC5CN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)=N2)C=C1)C1=CC(Cl)=C(OCCCl)C(C#N)=C1	C50H55Cl2N9O6	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-SCFOVE	SCHEMBL24480692	3-Chloro-2-(2-chloroethoxy)-5-[2-[4-[[2-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperidin-4-yl]-2,7-diazaspiro[3.5]nonan-7-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL29579984	CC(C)(C1=CC=C(OCC2=CC=NC(N3CCC4(CC3)CN(C3CCN(C5CN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC3)C4)=N2)C=C1)C1=CC(Cl)=C(OCCCl)C(C#N)=C1	C51H55Cl2N9O6	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-OP19UJ	WO2022111526A1_21	.	CC(C)(C1=CC=C(OCCC2=CC=NC(N3CCC4(CC3)CN(C3CCN(CC5CCN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC3)C4)=N2)C=C1)C1=CC(Cl)=C(OCCCl)C(C#N)=C1	C55H63Cl2N9O6	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-899HV2	SCHEMBL31236666	3-Chloro-2-(2-chloroethoxy)-5-[2-[4-[[2-[2-[1-[1-[[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-4-yl]methyl]azetidin-3-yl]piperidin-4-yl]-2,7-diazaspiro[3.5]nonan-7-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile	CN1C(=O)N(C2CCC(=O)NC2=O)C2=C1C(CN1CC(N3CCC(N4CC5(CCN(C6=NC(COC7=CC=C(C(C)(C)C8=CC(Cl)=C(OCCCl)C(C#N)=C8)C=C7)=CC=N6)CC5)C4)CC3)C1)=CC=C2	C52H60Cl2N10O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-2Q8UMJ	SCHEMBL24480427	3-Chloro-2-(2-chloroethoxy)-5-[2-[4-[[2-[7-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperidin-4-yl]-2,7-diazaspiro[3.5]nonan-2-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL29579530	CC(C)(C1=CC=C(OCC2=CC=NC(N3CC4(CCN(C5CCN(C6CN(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8=O)C6)CC5)CC4)C3)=N2)C=C1)C1=CC(Cl)=C(OCCCl)C(C#N)=C1	C51H55Cl2N9O6	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-V5ZPAT	SCHEMBL24480296	3-Chloro-2-(2-chloroethoxy)-5-[2-[4-[[2-[7-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperidin-4-yl]-2,7-diazaspiro[3.5]nonan-2-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL29580257	CC(C)(C1=CC=C(OCC2=CC=NC(N3CC4(CCN(C5CCN(CC6CCN(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)CC4)C3)=N2)C=C1)C1=CC(Cl)=C(OCCCl)C(C#N)=C1	C54H61Cl2N9O6	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-6ZX6I7	SCHEMBL24480728	3-Chloro-2-(2-chloroethoxy)-5-[2-[4-[[2-[7-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperidin-4-yl]methyl]piperidin-4-yl]-2,7-diazaspiro[3.5]nonan-2-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL29578688	CC(C)(C1=CC=C(OCC2=CC=NC(N3CC4(CCN(C5CCN(CC6CCN(C7=CC=CC8=C7C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)CC4)C3)=N2)C=C1)C1=CC(Cl)=C(OCCCl)C(C#N)=C1	C54H61Cl2N9O6	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-B632KS	SCHEMBL24480426	3-Chloro-2-(2-chloroethoxy)-5-[2-[4-[[2-[7-[1-[1-[[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-4-yl]methyl]azetidin-3-yl]piperidin-4-yl]-2,7-diazaspiro[3.5]nonan-2-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL29579199	CN1C(=O)N(C2CCC(=O)NC2=O)C2=C1C(CN1CC(N3CCC(N4CCC5(CC4)CN(C4=NC(COC6=CC=C(C(C)(C)C7=CC(Cl)=C(OCCCl)C(C#N)=C7)C=C6)=CC=N4)C5)CC3)C1)=CC=C2	C52H60Cl2N10O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-N0W7TJ	SCHEMBL24481044	3-Chloro-2-(2-chloroethoxy)-5-[2-[4-[[2-[9-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperidin-4-yl]-3,9-diazaspiro[5.5]undecan-3-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL29579208	CC(C)(C1=CC=C(OCC2=CC=NC(N3CCC4(CC3)CCN(C3CCN(CC5CCN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC3)CC4)=N2)C=C1)C1=CC(Cl)=C(OCCCl)C(C#N)=C1	C56H65Cl2N9O6	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-NHPKRM	SCHEMBL24480431	3-Chloro-2-(2-chloroethoxy)-5-[2-[4-[[2-[9-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperidin-4-yl]methyl]piperidin-4-yl]-3,9-diazaspiro[5.5]undecan-3-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL29579124	CC(C)(C1=CC=C(OCC2=CC=NC(N3CCC4(CC3)CCN(C3CCN(CC5CCN(C6=CC=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC3)CC4)=N2)C=C1)C1=CC(Cl)=C(OCCCl)C(C#N)=C1	C56H65Cl2N9O6	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-ZYDGCY	SCHEMBL24480514	3-Chloro-2-(2-chloroethoxy)-5-[2-[4-[[2-[9-[1-[[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-4-yl]methyl]azetidin-3-yl]-3,9-diazaspiro[5.5]undecan-3-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL31236682	CN1C(=O)N(C2CCC(=O)NC2=O)C2=C1C(CN1CC(N3CCC4(CCN(C5=NC(COC6=CC=C(C(C)(C)C7=CC(Cl)=C(OCCCl)C(C#N)=C7)C=C6)=CC=N5)CC4)CC3)C1)=CC=C2	C49H55Cl2N9O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-GP0RHI	SCHEMBL24480432	3-Chloro-2-(2-chloroethoxy)-5-[2-[4-[[2-[9-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperidin-4-yl]-3,9-diazaspiro[5.5]undecan-3-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL31236712	CC(C)(C1=CC=C(OCC2=CC=NC(N3CCC4(CC3)CCN(C3CCN(C5CN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC3)CC4)=N2)C=C1)C1=CC(Cl)=C(OCCCl)C(C#N)=C1	C53H59Cl2N9O6	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-6G56BK	SCHEMBL24480273	3-Chloro-2-(2-chloroethoxy)-5-[2-[4-[[2-[9-[1-[1-[[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-4-yl]methyl]azetidin-3-yl]piperidin-4-yl]-3,9-diazaspiro[5.5]undecan-3-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL31236691	CN1C(=O)N(C2CCC(=O)NC2=O)C2=C1C(CN1CC(N3CCC(N4CCC5(CCN(C6=NC(COC7=CC=C(C(C)(C)C8=CC(Cl)=C(OCCCl)C(C#N)=C8)C=C7)=CC=N6)CC5)CC4)CC3)C1)=CC=C2	C54H64Cl2N10O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-VPF1XA	SCHEMBL24481260	3-Chloro-5-[2-[4-[[2-[4-[[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperidin-4-yl]methyl]piperazin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL29579143	CC(C)(C1=CC=C(OCC2=CC=NC(N3CCN(CC4CCN(C5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)CC3)=N2)C=C1)C1=CC(Cl)=CC(C#N)=C1	C49H54ClN9O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-3KCEVY	SCHEMBL24480708	3-Chloro-5-[2-[4-[[2-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL29578656	CC(C)(C1=CC=C(OCC2=CC=NC(N3CCN(CC4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)=N2)C=C1)C1=CC(Cl)=CC(C#N)=C1	C44H45ClN8O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-5TYJN2	SCHEMBL24480303	3-Chloro-5-[2-[4-[[2-[4-[1-[7-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-7-azaspiro[3.5]nonan-2-yl]piperidin-4-yl]piperazin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL29579155	CC(C)(C1=CC=C(OCC2=CC=NC(N3CCN(C4CCN(C5CC6(CCN(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)C5)CC4)CC3)=N2)C=C1)C1=CC(Cl)=CC(C#N)=C1	C51H56ClN9O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-XV1DKB	WO2022111526A1_35	.	CC(=O)C1=C(C(=O)NC2CCC(=O)NC2=O)C=CC(N2CCC(CN3CCC4(CC3)CCN(C3=NC(COC5=CC=C(C(C)(C)C6=CC(Cl)=C(OCCCl)C(C#N)=C6)C=C5)=CC=N3)CC4)CC2)=C1	C52H60Cl2N8O6	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-790W1E	SCHEMBL24480293	3-Chloro-2-(2-chloroethoxy)-5-[2-[4-[[2-[4-[1-[[1-[[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-4-yl]methyl]piperidin-4-yl]methyl]piperidin-4-yl]piperazin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL31236718	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=CC(CN3CCC(CN4CCC(N5CCN(C6=NC(COC7=CC=C(C(C)(C)C8=CC(Cl)=C(OCCCl)C(C#N)=C8)C=C7)=CC=N6)CC5)CC4)CC3)=C21	C52H62Cl2N10O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-MOLHW3	SCHEMBL24481233	3-Chloro-5-[2-[4-[[2-[4-[[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile	CC(C)(C1=CC=C(OCC2=NC(N3CCC(CN4CCC(C5CCN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)CC3)=NC=C2)C=C1)C1=CC(Cl)=CC(C#N)=C1	C50H55ClN8O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-60T553	SCHEMBL24480526	3-Chloro-5-[2-[4-[[2-[4-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperidin-4-yl]piperidin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile	CC(C)(C1=CC=C(OCC2=NC(N3CCC(C4CCN(CC5CCN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)CC3)=NC=C2)C=C1)C1=CC(Cl)=CC(C#N)=C1	C50H55ClN8O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-DNRCEO	SCHEMBL24480295	3-Chloro-5-[2-[4-[[2-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperazin-1-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL29578626	CC(C)(C1=CC=C(OCC2=NC(N3CCC(CN4CCN(C5=CC=CC6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)=NC=C2)C=C1)C1=CC(Cl)=CC(C#N)=C1	C44H45ClN8O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-MHPVST	SCHEMBL24480531	3-Chloro-5-[2-[4-[[2-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperazin-1-yl]methyl]piperidin-1-yl]piperidin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile	CC(C)(C1=CC=C(OCC2=NC(N3CCC(N4CCC(CN5CCN(C6=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)CC5)CC4)CC3)=NC=C2)C=C1)C1=CC(Cl)=CC(C#N)=C1	C49H54ClN9O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-P8VG1M	SCHEMBL24480685	3-Chloro-5-[2-[4-[[2-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile	CC(C)(C1=CC=C(OCC2=NC(N3CCC(CN4CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)=NC=C2)C=C1)C1=CC(Cl)=CC(C#N)=C1	C44H45ClN8O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-5AR2A9	SCHEMBL24481240	3-Chloro-5-[2-[4-[[2-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]piperidin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL31236668	CC(C)(C1=CC=C(OCC2=NC(N3CCC(N4CCC(CN5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)CC3)=NC=C2)C=C1)C1=CC(Cl)=CC(C#N)=C1	C49H54ClN9O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-82RXOQ	SCHEMBL31236700	(2S,4R)-1-[(2S)-2-[[2-[4-[4-[[4-[4-[[4-[2-(3-chloro-5-cyanophenyl)propan-2-yl]phenoxy]methyl]pyrimidin-2-yl]piperazin-1-yl]methyl]piperidin-1-yl]piperidin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCC(N4CCC(CN5CCN(C6=NC=CC(COC7=CC=C(C(C)(C)C8=CC(C#N)=CC(Cl)=C8)C=C7)=N6)CC5)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C61H78ClN11O5S	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-LVJ21R	SCHEMBL24480257	3-Chloro-5-[2-[4-[[2-[4-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-2,9-diazaspiro[5.5]undecan-9-yl]piperidin-1-yl]piperidin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL31236702	CC(C)(C1=CC=C(OCC2=CC=NC(N3CCC(N4CCC(N5CCC6(CCCN(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8=O)C6)CC5)CC4)CC3)=N2)C=C1)C1=CC(Cl)=CC(C#N)=C1	C53H60ClN9O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-09T7PC	SCHEMBL24480765	3-Chloro-5-[2-[4-[[2-[2-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]-2,7-diazaspiro[3.5]nonan-7-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile	CC(C)(C1=CC=C(OCC2=NC(N3CCC4(CC3)CN(CC3CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC3)C4)=NC=C2)C=C1)C1=CC(Cl)=CC(C#N)=C1	C47H49ClN8O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-QHS3GN	SCHEMBL24480323	3-Chloro-5-[2-[4-[[2-[4-[1-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-2-azaspiro[3.5]nonan-7-yl]piperidin-4-yl]piperazin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL29579905	CC(C)(C1=CC=C(OCC2=CC=NC(N3CCN(C4CCN(C5CCC6(CC5)CN(C5=CC7=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)CC3)=N2)C=C1)C1=CC(Cl)=CC(C#N)=C1	C51H56ClN9O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-IEPJCZ	SCHEMBL24480333	3-Chloro-5-[2-[4-[[2-[3-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]azetidin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL29580229	CC(C)(C1=CC=C(OCC2=NC(N3CC(N4CCC(CN5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C3)=NC=C2)C=C1)C1=CC(Cl)=CC(C#N)=C1	C47H50ClN9O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-ZSMFSX	SCHEMBL29579763	3-Chloro-5-[2-[4-[[2-[3-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperazin-1-yl]methyl]piperidin-1-yl]azetidin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile	CC(C)(C1=CC=C(OCC2=NC(N3CC(N4CCC(CN5CCN(C6=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)CC5)CC4)C3)=NC=C2)C=C1)C1=CC(Cl)=CC(C#N)=C1	C47H50ClN9O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-DN2TF2	SCHEMBL24480963	3-Chloro-5-[2-[4-[[2-[4-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperidin-4-yl]piperazin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile	CC(C)(C1=CC=C(OCC2=NC(N3CCN(C4CCN(CC5CCN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)CC3)=NC=C2)C=C1)C1=CC(Cl)=CC(C#N)=C1	C49H54ClN9O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-MZ7M29	SCHEMBL24480329	(2S,4R)-1-[(2S)-2-[[2-[4-[[4-[4-[4-[[4-[2-(3-chloro-5-cyanophenyl)propan-2-yl]phenoxy]methyl]pyrimidin-2-yl]piperazin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCC(CN4CCC(N5CCN(C6=NC=CC(COC7=CC=C(C(C)(C)C8=CC(C#N)=CC(Cl)=C8)C=C7)=N6)CC5)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C61H78ClN11O5S	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-S96EU6	SCHEMBL31236727	(2S,4R)-1-[(2S)-2-[[2-[4-[[4-[4-[[4-[2-(3-chloro-5-cyanophenyl)propan-2-yl]phenoxy]methyl]pyrimidin-2-yl]piperazin-1-yl]methyl]piperidin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCC(CN4CCN(C5=NC=CC(COC6=CC=C(C(C)(C)C7=CC(C#N)=CC(Cl)=C7)C=C6)=N5)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C56H69ClN10O5S	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-4WBQMQ	SCHEMBL24480549	3-Chloro-5-[2-[4-[[2-[4-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-3-yl]azetidin-3-yl]piperazin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL29578850	CC(C)(C1=CC=C(OCC2=NC(N3CCN(C4CN(C5CCCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)C4)CC3)=NC=C2)C=C1)C1=CC(C#N)=CC(Cl)=C1	C46H48ClN9O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-795WFS	SCHEMBL24480343	3-Chloro-5-[2-[4-[[2-[4-[1-[7-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-7-azaspiro[3.5]nonan-2-yl]azetidin-3-yl]piperazin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL29578720	CC(C)(C1=CC=C(OCC2=NC(N3CCN(C4CN(C5CC6(CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)C5)C4)CC3)=NC=C2)C=C1)C1=CC(C#N)=CC(Cl)=C1	C49H52ClN9O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-VJJXW9	SCHEMBL24480773	3-Chloro-5-[2-[4-[[2-[4-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]azetidin-3-yl]piperazin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL29579059	CC(C)(C1=CC=C(OCC2=NC(N3CCN(C4CN(C5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)C4)CC3)=NC=C2)C=C1)C1=CC(C#N)=CC(Cl)=C1	C46H48ClN9O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-RPT90G	SCHEMBL24481046	3-Chloro-5-[2-[4-[[2-[4-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]pyrrolidin-3-yl]azetidin-3-yl]piperazin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL31236716	CC(C)(C1=CC=C(OCC2=NC(N3CCN(C4CN(C5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)C4)CC3)=NC=C2)C=C1)C1=CC(C#N)=CC(Cl)=C1	C45H46ClN9O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-8CHOK8	SCHEMBL24480341	3-Chloro-5-[2-[4-[[2-[4-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]azetidin-3-yl]piperazin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL31236704	CC(C)(C1=CC=C(OCC2=NC(N3CCN(C4CN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)C4)CC3)=NC=C2)C=C1)C1=CC(C#N)=CC(Cl)=C1	C47H50ClN9O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-2HCNTG	SCHEMBL24480317	3-Chloro-5-[2-[4-[[2-[4-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]methyl]azetidin-3-yl]piperazin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL29578928	CC(C)(C1=CC=C(OCC2=NC(N3CCN(C4CN(CC5CN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)C4)CC3)=NC=C2)C=C1)C1=CC(C#N)=CC(Cl)=C1	C45H46ClN9O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-ZIF28F	SCHEMBL24480534	3-Chloro-5-[2-[4-[[2-[4-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]pyrrolidin-3-yl]methyl]azetidin-3-yl]piperazin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL29579078	CC(C)(C1=CC=C(OCC2=NC(N3CCN(C4CN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)C4)CC3)=NC=C2)C=C1)C1=CC(C#N)=CC(Cl)=C1	C46H48ClN9O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-Q0JO8A	SCHEMBL24480916	3-Chloro-5-[2-[4-[[2-[4-[7-[7-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-7-azaspiro[3.5]nonan-2-yl]-7-azaspiro[3.5]nonan-2-yl]piperazin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL31236706	CC(C)(C1=CC=C(OCC2=NC(N3CCN(C4CC5(CCN(C6CC7(CCN(C8=CC=C9C(=O)N(C%10CCC(=O)NC%10=O)C(=O)C9=C8)CC7)C6)CC5)C4)CC3)=NC=C2)C=C1)C1=CC(Cl)=CC(C#N)=C1	C54H60ClN9O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-VJ5EUS	SCHEMBL24481080	3-Chloro-5-[2-[4-[[2-[4-[7-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]-7-azaspiro[3.5]nonan-2-yl]piperazin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL29578966	CC(C)(C1=CC=C(OCC2=NC(N3CCN(C4CC5(CCN(CC6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)CC5)C4)CC3)=NC=C2)C=C1)C1=CC(Cl)=CC(C#N)=C1	C52H58ClN9O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-LOIX7X	SCHEMBL24481087	3-Chloro-5-[2-[4-[[2-[4-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]methyl]pyrrolidin-3-yl]piperazin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL29579007	CC(C)(C1=CC=C(OCC2=NC(N3CCN(C4CCN(CC5CN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)C4)CC3)=NC=C2)C=C1)C1=CC(Cl)=CC(C#N)=C1	C46H48ClN9O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-NZKG9C	SCHEMBL24480445	3-Chloro-5-[2-[4-[[2-[4-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]pyrrolidin-3-yl]methyl]pyrrolidin-3-yl]piperazin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL29579351	CC(C)(C1=CC=C(OCC2=NC(N3CCN(C4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)C4)CC3)=NC=C2)C=C1)C1=CC(Cl)=CC(C#N)=C1	C47H50ClN9O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-SCZYXS	SCHEMBL24480441	3-Chloro-5-[2-[4-[[2-[4-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]pyrrolidin-3-yl]piperazin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL29578572	CC(C)(C1=CC=C(OCC2=NC(N3CCN(C4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)C4)CC3)=NC=C2)C=C1)C1=CC(Cl)=CC(C#N)=C1	C48H52ClN9O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-4EDJZR	SCHEMBL24481025	3-Chloro-5-[2-[4-[[2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]azetidin-1-yl]piperidin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL29578472	CC(C)(C1=CC=C(OCC2=NC(N3CCC(N4CC(N5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)C4)CC3)=NC=C2)C=C1)C1=CC(Cl)=CC(C#N)=C1	C46H48ClN9O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-G1C92M	SCHEMBL24480536	3-Chloro-5-[2-[4-[[2-[4-[3-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperazin-1-yl]methyl]azetidin-1-yl]piperidin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile	CC(C)(C1=CC=C(OCC2=NC(N3CCC(N4CC(CN5CCN(C6=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)CC5)C4)CC3)=NC=C2)C=C1)C1=CC(Cl)=CC(C#N)=C1	C47H50ClN9O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-O00DKY	SCHEMBL24480788	3-Chloro-5-[2-[4-[[2-[4-[[1-[7-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-7-azaspiro[3.5]nonan-2-yl]pyrrolidin-3-yl]methyl]piperazin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL29579055	CC(C)(C1=CC=C(OCC2=NC(N3CCN(CC4CCN(C5CC6(CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)C5)C4)CC3)=NC=C2)C=C1)C1=CC(Cl)=CC(C#N)=C1	C51H56ClN9O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-S38LCC	SCHEMBL24481038	3-Chloro-5-[2-[4-[[2-[4-[[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-3-yl]pyrrolidin-3-yl]methyl]piperazin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL29579251	CC(C)(C1=CC=C(OCC2=NC(N3CCN(CC4CCN(C5CCCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)C4)CC3)=NC=C2)C=C1)C1=CC(Cl)=CC(C#N)=C1	C48H52ClN9O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-BIHZYS	SCHEMBL24480625	3-Chloro-5-[2-[4-[[2-[9-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]-3,9-diazaspiro[5.5]undecan-3-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile	CC(C)(C1=CC=C(OCC2=NC(N3CCC4(CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)CC3)=NC=C2)C=C1)C1=CC(Cl)=CC(C#N)=C1	C49H53ClN8O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-V0Z1C0	SCHEMBL24480372	3-Chloro-5-[2-[4-[[2-[7-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]-2,7-diazaspiro[3.5]nonan-2-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile	CC(C)(C1=CC=C(OCC2=NC(N3CC4(CCN(CC5CCN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)C3)=NC=C2)C=C1)C1=CC(Cl)=CC(C#N)=C1	C47H49ClN8O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-EZ9H3L	SCHEMBL24480371	3-Chloro-5-[2-[4-[[2-[7-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]methyl]-2,7-diazaspiro[3.5]nonan-2-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile	CC(C)(C1=CC=C(OCC2=NC(N3CC4(CCN(CC5CN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)C3)=NC=C2)C=C1)C1=CC(Cl)=CC(C#N)=C1	C45H45ClN8O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-5V4MSJ	SCHEMBL29579897	3-Chloro-5-[2-[4-[[2-[4-[1-[1-[[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]methyl]azetidin-3-yl]piperidin-4-yl]piperazin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile	CN1C(=O)N(C2CCC(=O)NC2=O)C2=C1C=C(CN1CC(N3CCC(N4CCN(C5=NC(COC6=CC=C(C(C)(C)C7=CC(Cl)=CC(C#N)=C7)C=C6)=CC=N5)CC4)CC3)C1)C=C2	C47H53ClN10O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-ADT84T	SCHEMBL24480535	3-Chloro-5-[2-[4-[[2-[2-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-5-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile	CC(C)(C1=CC=C(OCC2=NC(N3CC4CN(CC5CCN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4C3)=NC=C2)C=C1)C1=CC(Cl)=CC(C#N)=C1	C46H47ClN8O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-CAIB1M	SCHEMBL24481090	3-Chloro-5-[2-[4-[[2-[2-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]methyl]-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-5-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile	CC(C)(C1=CC=C(OCC2=NC(N3CC4CN(CC5CN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4C3)=NC=C2)C=C1)C1=CC(Cl)=CC(C#N)=C1	C44H43ClN8O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-LXQJ8H	SCHEMBL24480591	3-Chloro-5-[2-[4-[[2-[4-[1-[[1-[[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-4-yl]methyl]piperidin-4-yl]methyl]piperidin-4-yl]piperidin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL31236690	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=CC(CN3CCC(CN4CCC(C5CCN(C6=NC=CC(COC7=CC=C(C(C)(C)C8=CC(Cl)=CC(C#N)=C8)C=C7)=N6)CC5)CC4)CC3)=C21	C51H60ClN9O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-1C67WC	SCHEMBL24480425	3-Chloro-5-[2-[4-[[2-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperidin-4-yl]-2,7-diazaspiro[3.5]nonan-7-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL31236671	CC(C)(C1=CC=C(OCC2=CC=NC(N3CCC4(CC3)CN(C3CCN(C5CN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC3)C4)=N2)C=C1)C1=CC(Cl)=CC(C#N)=C1	C49H52ClN9O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-ZMTYIA	SCHEMBL24480781	3-Chloro-5-[2-[4-[[2-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]azetidin-3-yl]-2,7-diazaspiro[3.5]nonan-7-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL31236696; SCHEMBL31236697	CC(C)(C1=CC=C(OCC2=CC=NC(N3CCC4(CC3)CN(C3CN(C5CN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)C3)C4)=N2)C=C1)C1=CC(Cl)=CC(C#N)=C1	C47H48ClN9O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-D85T5F	SCHEMBL24481086	3-Chloro-5-[2-[4-[[2-[4-[[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-3,9-diazaspiro[5.5]undecan-9-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL29579554	CC(C)(C1=CC=C(OCC2=CC=NC(N3CCC(CN4CCC5(CC4)CCN(C4=CC6=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC5)CC3)=N2)C=C1)C1=CC(Cl)=CC(C#N)=C1	C49H53ClN8O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-KWCR4O	SCHEMBL24480520	3-Chloro-5-[2-[4-[[2-[4-[[4-[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile	CC(C)(C1=CC=C(OCC2=NC(N3CCC(CN4CCC(C5CCN(C6=CC7=C(C=C6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)CC3)=NC=C2)C=C1)C1=CC(Cl)=CC(C#N)=C1	C50H54ClFN8O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-R6NUFW	SCHEMBL24480824	3-Chloro-5-[2-[4-[[2-[4-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]methyl]piperidin-4-yl]piperidin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile	CC(C)(C1=CC=C(OCC2=NC(N3CCC(C4CCN(CC5CN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)CC3)=NC=C2)C=C1)C1=CC(Cl)=CC(C#N)=C1	C48H51ClN8O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-G0T348	SCHEMBL24481310	3-Chloro-5-[2-[4-[[2-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]ethynyl]piperidin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile	CC(C)(C1=CC=C(OCC2=NC(N3CCC(C#CC4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)=NC=C2)C=C1)C1=CC(Cl)=CC(C#N)=C1	C41H35ClN6O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-1B4XB6	SCHEMBL24480573	3-Chloro-5-[2-[4-[[2-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperidin-4-yl]-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-5-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL29579116	CC(C)(C1=CC=C(OCC2=NC(N3CC4CN(C5CCN(C6CN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)C6)CC5)CC4C3)=NC=C2)C=C1)C1=CC(Cl)=CC(C#N)=C1	C48H50ClN9O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-RV9HWJ	SCHEMBL24480412	3-Chloro-5-[2-[4-[[2-[2-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperidin-4-yl]-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-5-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL31236692	CC(C)(C1=CC=C(OCC2=NC(N3CC4CN(C5CCN(CC6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)CC5)CC4C3)=NC=C2)C=C1)C1=CC(Cl)=CC(C#N)=C1	C51H56ClN9O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-OL6XAB	SCHEMBL24480796	3-Chloro-5-[2-[4-[[2-[9-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]pyrrolidin-3-yl]methyl]-3,9-diazaspiro[5.5]undecan-3-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL29578740	CC(C)(C1=CC=C(OCC2=NC(N3CCC4(CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)=NC=C2)C=C1)C1=CC(Cl)=CC(C#N)=C1	C48H51ClN8O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-9DLZ71	SCHEMBL24480616	3-Chloro-5-[2-[4-[[2-[9-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperidin-4-yl]methyl]-3,9-diazaspiro[5.5]undecan-3-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile	CC(C)(C1=CC=C(OCC2=NC(N3CCC4(CCN(CC5CCN(C6=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)CC5)CC4)CC3)=NC=C2)C=C1)C1=CC(Cl)=CC(C#N)=C1	C49H53ClN8O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-XKI2J4	SCHEMBL24480660	3-Chloro-5-[2-[4-[[2-[4-[[4-[1-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-4-yl]piperidin-4-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL29579185	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=CC(N3CCC(C4CCN(CC5CCN(C6=NC=CC(COC7=CC=C(C(C)(C)C8=CC(Cl)=CC(C#N)=C8)C=C7)=N6)CC5)CC4)CC3)=C21	C50H58ClN9O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-BAUDOW	SCHEMBL24480405	3-Chloro-5-[2-[4-[[2-[3-[[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-3,9-diazaspiro[5.5]undecan-9-yl]methyl]pyrrolidin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL29578460	CC(C)(C1=CC=C(OCC2=CC=NC(N3CCC(CN4CCC5(CC4)CCN(C4=CC6=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC5)C3)=N2)C=C1)C1=CC(Cl)=CC(C#N)=C1	C48H51ClN8O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-ELRSPV	SCHEMBL24480593	3-Chloro-5-[2-[4-[[2-[3-[[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-3,9-diazaspiro[5.5]undecan-9-yl]methyl]azetidin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL29579585	CC(C)(C1=CC=C(OCC2=CC=NC(N3CC(CN4CCC5(CC4)CCN(C4=CC6=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC5)C3)=N2)C=C1)C1=CC(Cl)=CC(C#N)=C1	C47H49ClN8O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-H1G316	SCHEMBL24480563	3-Chloro-5-[2-[4-[[2-[4-[[4-[1-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidin-4-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL29579424	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(N3CCC(C4CCN(CC5CCN(C6=NC=CC(COC7=CC=C(C(C)(C)C8=CC(Cl)=CC(C#N)=C8)C=C7)=N6)CC5)CC4)CC3)C=C21	C50H58ClN9O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-1CRMN5	SCHEMBL24480668	3-Chloro-5-[2-[4-[[2-[4-[[4-[1-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidin-4-yl]piperidin-1-yl]methyl]-4-fluoropiperidin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL29578979	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(N3CCC(C4CCN(CC5(F)CCN(C6=NC=CC(COC7=CC=C(C(C)(C)C8=CC(Cl)=CC(C#N)=C8)C=C7)=N6)CC5)CC4)CC3)C=C21	C50H57ClFN9O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-7LUKTK	SCHEMBL24480670	3-Chloro-5-[2-[4-[[2-[4-[[4-[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidin-1-yl]piperidin-1-yl]methyl]-4-fluoropiperidin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL31236675	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(C3CCN(C4CCN(CC5(F)CCN(C6=NC=CC(COC7=CC=C(C(C)(C)C8=CC(Cl)=CC(C#N)=C8)C=C7)=N6)CC5)CC4)CC3)C=C21	C50H57ClFN9O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-FE4X5T	SCHEMBL24480680	3-Chloro-5-[2-[4-[[2-[4-[4-[[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]piperidin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL31236711	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(C3CCN(CC4CCN(C5CCN(C6=NC=CC(COC7=CC=C(C(C)(C)C8=CC(Cl)=CC(C#N)=C8)C=C7)=N6)CC5)CC4)CC3)C=C21	C50H58ClN9O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-0B9Z1T	SCHEMBL24481103	3-Chloro-5-[2-[4-[[2-[4-[[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]-2-methoxybenzonitrile; SCHEMBL31236722	COC1=C(Cl)C=C(C(C)(C)C2=CC=C(OCC3=NC(N4CCC(CN5CCC(C6=CC=C7C(=C6)N(C)C(=O)N7C6CCC(=O)NC6=O)CC5)CC4)=NC=C3)C=C2)C=C1C#N	C46H51ClN8O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-PMNY3E	SCHEMBL24480470	3-Chloro-5-[2-[4-[[2-[9-[[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidin-1-yl]methyl]-3-azaspiro[5.5]undecan-3-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]-2-methoxybenzonitrile; SCHEMBL31236715	COC1=C(Cl)C=C(C(C)(C)C2=CC=C(OCC3=NC(N4CCC5(CCC(CN6CCC(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC5)CC4)=NC=C3)C=C2)C=C1C#N	C51H59ClN8O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-LISN47	SCHEMBL24481292	3-Chloro-5-[2-[4-[[2-[4-[[4-[1-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidin-4-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]-2-ethoxybenzonitrile	CCOC1=C(Cl)C=C(C(C)(C)C2=CC=C(OCC3=NC(N4CCC(CN5CCC(C6CCN(C7=CC8=C(C=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)CC6)CC5)CC4)=NC=C3)C=C2)C=C1C#N	C52H62ClN9O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-AV6N46	SCHEMBL24480885	3-Chloro-5-[2-[4-[[2-[4-[1-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidin-4-yl]piperidin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]-2-methoxybenzonitrile	COC1=C(Cl)C=C(C(C)(C)C2=CC=C(OCC3=NC(N4CCC(C5CCN(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC5)CC4)=NC=C3)C=C2)C=C1C#N	C45H49ClN8O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-UX0H9Z	SCHEMBL24480869	3-Chloro-5-[2-[4-[[2-[9-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]-3,9-diazaspiro[5.5]undecan-3-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]-2-methoxybenzonitrile	COC1=C(Cl)C=C(C(C)(C)C2=CC=C(OCC3=NC(N4CCC5(CCN(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC5)CC4)=NC=C3)C=C2)C=C1C#N	C44H47ClN8O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-O49PGG	SCHEMBL24481322	3-Chloro-5-[2-[4-[[2-[4-[[4-[1-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidin-4-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]-2-methoxybenzonitrile	COC1=C(Cl)C=C(C(C)(C)C2=CC=C(OCC3=NC(N4CCC(CN5CCC(C6CCN(C7=CC8=C(C=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)CC6)CC5)CC4)=NC=C3)C=C2)C=C1C#N	C51H60ClN9O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-EVS1GM	SCHEMBL24480886	3-Chloro-2-(2-chloroethoxy)-5-[2-[4-[[2-[4-[[4-[1-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidin-4-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile	CN1C(=O)N(C2CCC(=O)NC2=O)C2=C1C=C(N1CCC(C3CCN(CC4CCN(C5=NC=CC(COC6=CC=C(C(C)(C)C7=CC(Cl)=C(OCCCl)C(C#N)=C7)C=C6)=N5)CC4)CC3)CC1)C=C2	C52H61Cl2N9O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-9578TR	SCHEMBL24480451	3-Chloro-5-[2-[4-[[2-[9-[1-[[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-4-yl]methyl]piperidin-4-yl]-3,9-diazaspiro[5.5]undecan-3-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile	CN1C(=O)N(C2CCC(=O)NC2=O)C2=C1C(CN1CCC(N3CCC4(CCN(C5=NC=CC(COC6=CC=C(C(C)(C)C7=CC(Cl)=CC(C#N)=C7)C=C6)=N5)CC4)CC3)CC1)=CC=C2	C49H56ClN9O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-SAVOZP	SCHEMBL24480622	3-Chloro-5-[2-[4-[[2-[9-[7-[[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-4-yl]methyl]-7-azaspiro[3.5]nonan-2-yl]-3,9-diazaspiro[5.5]undecan-3-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile	CN1C(=O)N(C2CCC(=O)NC2=O)C2=C1C(CN1CCC3(CC1)CC(N1CCC4(CCN(C5=NC=CC(COC6=CC=C(C(C)(C)C7=CC(Cl)=CC(C#N)=C7)C=C6)=N5)CC4)CC1)C3)=CC=C2	C52H60ClN9O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-VC42OV	SCHEMBL24480438	3-Chloro-5-[2-[4-[[2-[4-[[[1-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidin-4-yl]-methylamino]methyl]piperidin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]-2-ethoxybenzonitrile; SCHEMBL31236687	CCOC1=C(Cl)C=C(C(C)(C)C2=CC=C(OCC3=NC(N4CCC(CN(C)C5CCN(C6=CC=C7C(=C6)N(C)C(=O)N7C6CCC(=O)NC6=O)CC5)CC4)=NC=C3)C=C2)C=C1C#N	C48H56ClN9O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-7CYQ9U	SCHEMBL24480682	3-Chloro-5-[2-[4-[[2-[3-[[4-[1-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidin-4-yl]piperidin-1-yl]methyl]azetidin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL29578504	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(N3CCC(C4CCN(CC5CN(C6=NC=CC(COC7=CC=C(C(C)(C)C8=CC(Cl)=CC(C#N)=C8)C=C7)=N6)C5)CC4)CC3)C=C21	C48H54ClN9O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-NF05O8	SCHEMBL24481323	3-Chloro-5-[2-[4-[[2-[4-[4-[1-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidin-4-yl]piperidin-1-yl]piperidin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL31236684	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(N3CCC(C4CCN(C5CCN(C6=NC=CC(COC7=CC=C(C(C)(C)C8=CC(Cl)=CC(C#N)=C8)C=C7)=N6)CC5)CC4)CC3)C=C21	C49H56ClN9O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-J1R1J9	SCHEMBL24480730	3-Chloro-5-[2-[4-[[2-[4-[[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL31236703	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(C3CCN(CC4CCN(C5=NC=CC(COC6=CC=C(C(C)(C)C7=CC(Cl)=CC(C#N)=C7)C=C6)=N5)CC4)CC3)C=C21	C45H49ClN8O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-FQEVHO	SCHEMBL24480455	3-Chloro-5-[2-[4-[[2-[2-[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidin-1-yl]-7-azaspiro[3.5]nonan-7-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL29579774	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(C3CCN(C4CC5(CCN(C6=NC=CC(COC7=CC=C(C(C)(C)C8=CC(Cl)=CC(C#N)=C8)C=C7)=N6)CC5)C4)CC3)C=C21	C47H51ClN8O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-19B2OB	SCHEMBL24481082	3-Chloro-5-[2-[4-[[2-[2-[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidin-1-yl]-7-azaspiro[3.5]nonan-7-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]-2-ethoxybenzonitrile; SCHEMBL31236681	CCOC1=C(Cl)C=C(C(C)(C)C2=CC=C(OCC3=NC(N4CCC5(CC4)CC(N4CCC(C6=CC=C7C(=C6)N(C)C(=O)N7C6CCC(=O)NC6=O)CC4)C5)=NC=C3)C=C2)C=C1C#N	C49H55ClN8O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-R5XN2A	SCHEMBL24480865	3-Chloro-5-[2-[4-[[2-[2-[4-[[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]-7-azaspiro[3.5]nonan-7-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL29578788	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(C3CCN(CC4CCN(C5CC6(CCN(C7=NC=CC(COC8=CC=C(C(C)(C)C9=CC(Cl)=CC(C#N)=C9)C=C8)=N7)CC6)C5)CC4)CC3)C=C21	C53H62ClN9O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-KO1A25	SCHEMBL29578764	3-Chloro-5-[2-[4-[[2-[2-[4-[[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]-7-azaspiro[3.5]nonan-7-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]-2-ethoxybenzonitrile	CCOC1=C(Cl)C=C(C(C)(C)C2=CC=C(OCC3=NC(N4CCC5(CC4)CC(N4CCC(CN6CCC(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)C5)=NC=C3)C=C2)C=C1C#N	C55H66ClN9O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-7JJUGI	SCHEMBL24480727	5-[4-[1-[[1-[4-[[4-[2-(3-chloro-5-cyanophenyl)propan-2-yl]phenoxy]methyl]pyrimidin-2-yl]piperidin-4-yl]methyl]piperidin-4-yl]piperidin-1-yl]-N-(2,6-dioxopiperidin-3-yl)pyridine-2-carboxamide; SCHEMBL31236665	CC(C)(C1=CC=C(OCC2=NC(N3CCC(CN4CCC(C5CCN(C6=CC=C(C(=O)NC7CCC(=O)NC7=O)N=C6)CC5)CC4)CC3)=NC=C2)C=C1)C1=CC(Cl)=CC(C#N)=C1	C48H56ClN9O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-5UQ58W	SCHEMBL31236689	5-[4-[1-[[1-[4-[[4-[2-(3-chloro-5-cyano-4-ethoxyphenyl)propan-2-yl]phenoxy]methyl]pyrimidin-2-yl]piperidin-4-yl]methyl]piperidin-4-yl]piperidin-1-yl]-N-(2,6-dioxopiperidin-3-yl)pyridine-2-carboxamide	CCOC1=C(Cl)C=C(C(C)(C)C2=CC=C(OCC3=NC(N4CCC(CN5CCC(C6CCN(C7=CC=C(C(=O)NC8CCC(=O)NC8=O)N=C7)CC6)CC5)CC4)=NC=C3)C=C2)C=C1C#N	C50H60ClN9O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-SXEIE2	SCHEMBL24481312	5-[4-[1-[[1-[4-[[4-[2-(3-chloro-5-cyano-4-methoxyphenyl)propan-2-yl]phenoxy]methyl]pyrimidin-2-yl]piperidin-4-yl]methyl]piperidin-4-yl]piperidin-1-yl]-N-(2,6-dioxopiperidin-3-yl)pyridine-2-carboxamide; SCHEMBL31236677	COC1=C(Cl)C=C(C(C)(C)C2=CC=C(OCC3=NC(N4CCC(CN5CCC(C6CCN(C7=CC=C(C(=O)NC8CCC(=O)NC8=O)N=C7)CC6)CC5)CC4)=NC=C3)C=C2)C=C1C#N	C49H58ClN9O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-3MURLE	SCHEMBL24480707	3-Chloro-5-[2-[4-[[2-[2-[[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidin-1-yl]methyl]-7-azaspiro[3.5]nonan-7-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]-2-methoxybenzonitrile; SCHEMBL31236670	COC1=C(Cl)C=C(C(C)(C)C2=CC=C(OCC3=NC(N4CCC5(CC4)CC(CN4CCC(C6=CC=C7C(=C6)N(C)C(=O)N7C6CCC(=O)NC6=O)CC4)C5)=NC=C3)C=C2)C=C1C#N	C49H55ClN8O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-WYTV7V	SCHEMBL24480457	3-Chloro-5-[2-[4-[[2-[4-[[[1-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidin-4-yl]-methylamino]methyl]piperidin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL31236719	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(N3CCC(N(C)CC4CCN(C5=NC=CC(COC6=CC=C(C(C)(C)C7=CC(Cl)=CC(C#N)=C7)C=C6)=N5)CC4)CC3)C=C21	C46H52ClN9O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-86U90S	SCHEMBL24480458	3-Chloro-5-[2-[4-[[2-[2-[4-[[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-4-yl]piperidin-1-yl]methyl]-4-fluoropiperidin-1-yl]-7-azaspiro[3.5]nonan-7-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL29579873	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=CC(C3CCN(CC4(F)CCN(C5CC6(CCN(C7=NC=CC(COC8=CC=C(C(C)(C)C9=CC(Cl)=CC(C#N)=C9)C=C8)=N7)CC6)C5)CC4)CC3)=C21	C53H61ClFN9O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-937IEL	SCHEMBL24480903	3-Chloro-5-[2-[4-[[2-[4-[[4-[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]-2-methoxybenzonitrile	COC1=C(Cl)C=C(C(C)(C)C2=CC=C(OCC3=NC(N4CCC(CN5CCC(N6CCC(C7=CC8=C(C=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)CC6)CC5)CC4)=NC=C3)C=C2)C=C1C#N	C51H60ClN9O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-PR2HFJ	SCHEMBL24480360	3-Chloro-5-[2-[4-[[2-[4-[[2-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]-2,7-diazaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]-2-ethoxybenzonitrile	CCOC1=C(Cl)C=C(C(C)(C)C2=CC=C(OCC3=NC(N4CCC(CN5CCC6(CC5)CN(C5=CC7=C(C=C5)N(C5CCC(=O)NC5=O)C(=O)N7C)C6)CC4)=NC=C3)C=C2)C=C1C#N	C49H56ClN9O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-SJW4WP	SCHEMBL24480895	3-Chloro-5-[2-[4-[[2-[4-[[4-[1-[4-(2,6-dioxopiperidin-3-yl)phenyl]piperidin-4-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]-2-methoxybenzonitrile	COC1=C(Cl)C=C(C(C)(C)C2=CC=C(OCC3=NC(N4CCC(CN5CCC(C6CCN(C7=CC=C(C8CCC(=O)NC8=O)C=C7)CC6)CC5)CC4)=NC=C3)C=C2)C=C1C#N	C49H58ClN7O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-GIRC8A	SCHEMBL24481105	3-Chloro-5-[2-[4-[[2-[4-[[4-[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]-2-methoxybenzonitrile	COC1=C(Cl)C=C(C(C)(C)C2=CC=C(OCC3=NC(N4CCC(CN5CCC(C6CCN(C7=CC=C(N8CCC(=O)NC8=O)C=C7)CC6)CC5)CC4)=NC=C3)C=C2)C=C1C#N	C48H57ClN8O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-A669EM	SCHEMBL24480729	3-Chloro-5-[2-[4-[[2-[7-[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidin-1-yl]-2-azaspiro[3.5]nonan-2-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]-2-ethoxybenzonitrile; SCHEMBL29578965	CCOC1=C(Cl)C=C(C(C)(C)C2=CC=C(OCC3=NC(N4CC5(CCC(N6CCC(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC5)C4)=NC=C3)C=C2)C=C1C#N	C49H55ClN8O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-34Q16N	SCHEMBL24480476	3-Chloro-5-[2-[4-[[2-[7-[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidin-1-yl]-2-azaspiro[3.5]nonan-2-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL31236686	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(C3CCN(C4CCC5(CC4)CN(C4=NC=CC(COC6=CC=C(C(C)(C)C7=CC(Cl)=CC(C#N)=C7)C=C6)=N4)C5)CC3)C=C21	C47H51ClN8O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-9RIE0D	SCHEMBL24481320	3-Chloro-5-[2-[4-[[2-[4-[[4-[1-[1-(2,6-dioxopiperidin-3-yl)-6-fluoro-3-methyl-2-oxobenzimidazol-5-yl]piperidin-4-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]-2-methoxybenzonitrile; SCHEMBL31236669	COC1=C(Cl)C=C(C(C)(C)C2=CC=C(OCC3=NC(N4CCC(CN5CCC(C6CCN(C7=C(F)C=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC5)CC4)=NC=C3)C=C2)C=C1C#N	C51H59ClFN9O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-93JAGZ	SCHEMBL24480755	3-Chloro-5-[2-[4-[[2-[4-[4-[[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-4-yl]piperidin-1-yl]methyl]-4-fluoropiperidin-1-yl]piperidin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile; SCHEMBL31236679	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=CC(C3CCN(CC4(F)CCN(C5CCN(C6=NC=CC(COC7=CC=C(C(C)(C)C8=CC(Cl)=CC(C#N)=C8)C=C7)=N6)CC5)CC4)CC3)=C21	C50H57ClFN9O4	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-OM4TWH	SCHEMBL31236688	3-Chloro-2-(2-chloroethoxy)-5-[2-[4-[[2-[4-[1-[[1-[[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-4-yl]methyl]piperidin-4-yl]methyl]piperidin-4-yl]piperidin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile	CN1C(=O)N(C2CCC(=O)NC2=O)C2=C1C(CN1CCC(CN3CCC(C4CCN(C5=NC=CC(COC6=CC=C(C(C)(C)C7=CC(Cl)=C(OCCCl)C(C#N)=C7)C=C6)=N5)CC4)CC3)CC1)=CC=C2	C53H63Cl2N9O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-7US3HP	SCHEMBL24480494	3-Chloro-5-[2-[4-[1-[2-[4-[[4-[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]ethoxy]phenyl]propan-2-yl]benzonitrile	CC(OC1=CC=C(C(C)(C)C2=CC(Cl)=CC(C#N)=C2)C=C1)C1=NC(N2CCC(CN3CCC(C4CCN(C5=C(F)C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)CC2)=NC=C1	C51H56ClFN8O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-DLIXU6	SCHEMBL24480926	3-Chloro-5-[2-[4-[[2-[9-[7-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-7-azaspiro[3.5]nonan-2-yl]-3,9-diazaspiro[5.5]undecan-3-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile	CC(C)(C1=CC=C(OCC2=NC(N3CCC4(CC3)CCN(C3CC5(CCN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C3)CC4)=NC=C2)C=C1)C1=CC(Cl)=CC(C#N)=C1	C51H55ClN8O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-2DWI9W	SCHEMBL24480900	3-Chloro-5-[2-[4-[[2-[9-[[7-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-7-azaspiro[3.5]nonan-2-yl]methyl]-3,9-diazaspiro[5.5]undecan-3-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile	CC(C)(C1=CC=C(OCC2=NC(N3CCC4(CCN(CC5CC6(CCN(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)C5)CC4)CC3)=NC=C2)C=C1)C1=CC(Cl)=CC(C#N)=C1	C52H57ClN8O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-TIE5J3	SCHEMBL24481155	3-Chloro-5-[2-[4-[[2-[3-[[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperidin-1-yl]methyl]pyrrolidin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile	CC(C)(C1=CC=C(OCC2=NC(N3CCC(CN4CCC(C5CCN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)C3)=NC=C2)C=C1)C1=CC(Cl)=CC(C#N)=C1	C49H53ClN8O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-KBDLQM	SCHEMBL24480937	3-Chloro-5-[2-[4-[[2-[4-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperidin-1-yl]piperidin-1-yl]pyrimidin-4-yl]methoxy]phenyl]propan-2-yl]benzonitrile	CC(C)(C1=CC=C(OCC2=NC(N3CCC(N4CCC(C5CCN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)CC3)=NC=C2)C=C1)C1=CC(Cl)=CC(C#N)=C1	C49H53ClN8O5	AR;AR-V7	P10275/P10275-3	CRBN	WO-2022111526-A1
TPD-FPMBVE	SCHEMBL24620884	N-[1-benzofuran-2-yl(pyridin-3-yl)methyl]-2-[4-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethyl]piperazin-1-yl]acetamide	O=C1CCC(N2C(=O)c3cccc(NCCN4CCN(CC(=O)NC(c5cccnc5)c5cc6ccccc6o5)CC4)c3C2=O)C(=O)N1	C35H35N7O6	SMAD3	P84022	CRBN	WO-2022148459-A1
TPD-6IGO5W	SCHEMBL24621139	N-[1-benzofuran-2-yl(pyridin-3-yl)methyl]-2-[5-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]pent-4-ynoxy]acetamide	O=C1CCC(N2C(=O)c3cccc(C#CCCCOCC(=O)NC(c4cccnc4)c4cc5ccccc5o4)c3C2=O)C(=O)N1	C34H28N4O7	SMAD3	P84022	CRBN	WO-2022148459-A1
TPD-Y7YDZL	SCHEMBL24621153	N-[1-benzofuran-2-yl(pyridin-3-yl)methyl]-2-[5-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]pentoxy]acetamide	O=C1CCC(N2C(=O)c3cccc(CCCCCOCC(=O)NC(c4cccnc4)c4cc5ccccc5o4)c3C2=O)C(=O)N1	C34H32N4O7	SMAD3	P84022	CRBN	WO-2022148459-A1
TPD-PLVLJB	SCHEMBL24621185	N-[1-benzofuran-2-yl(pyridin-3-yl)methyl]-2-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxybutoxy]acetamide	O=C1CCC(N2C(=O)c3cccc(OCCCCOCC(=O)NC(c4cccnc4)c4cc5ccccc5o4)c3C2=O)C(=O)N1	C33H30N4O8	SMAD3	P84022	CRBN	WO-2022148459-A1
TPD-J9H2AR	SCHEMBL24621219	N-[1-benzofuran-2-yl(pyridin-3-yl)methyl]-3-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]butoxy]propanamide	O=C1CCC(N2C(=O)c3cccc(CCCCOCCC(=O)NC(c4cccnc4)c4cc5ccccc5o4)c3C2=O)C(=O)N1	C34H32N4O7	SMAD3	P84022	CRBN	WO-2022148459-A1
TPD-MB5N18	SCHEMBL24621190	N-[1-benzofuran-2-yl(pyridin-3-yl)methyl]-3-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]but-3-ynoxy]propanamide	O=C1CCC(N2C(=O)c3cccc(C#CCCOCCC(=O)NC(c4cccnc4)c4cc5ccccc5o4)c3C2=O)C(=O)N1	C34H28N4O7	SMAD3	P84022	CRBN	WO-2022148459-A1
TPD-LJWDUO	SCHEMBL24621221	N-[1-benzofuran-2-yl(pyridin-3-yl)methyl]-3-[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxypropoxy]propanamide	O=C1CCC(N2C(=O)c3cccc(OCCCOCCC(=O)NC(c4cccnc4)c4cc5ccccc5o4)c3C2=O)C(=O)N1	C33H30N4O8	SMAD3	P84022	CRBN	WO-2022148459-A1
TPD-0Y74H9	SCHEMBL24620978	N-[1-benzofuran-2-yl(pyridin-3-yl)methyl]-3-[3-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]propoxy]propanamide	O=C1CCC(N2C(=O)c3cccc(NCCCOCCC(=O)NC(c4cccnc4)c4cc5ccccc5o4)c3C2=O)C(=O)N1	C33H31N5O7	SMAD3	P84022	CRBN	WO-2022148459-A1
TPD-JX171I	SCHEMBL24621203	N-[1-benzofuran-2-yl(pyridin-3-yl)methyl]-7-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyheptanamide	O=C1CCC(N2C(=O)c3cccc(OCCCCCCC(=O)NC(c4cccnc4)c4cc5ccccc5o4)c3C2=O)C(=O)N1	C34H32N4O7	SMAD3	P84022	CRBN	WO-2022148459-A1
TPD-T7DZWZ	SCHEMBL24621222	N-[1-benzofuran-2-yl(pyridin-3-yl)methyl]-4-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyethoxy]butanamide	O=C1CCC(N2C(=O)c3cccc(OCCOCCCC(=O)NC(c4cccnc4)c4cc5ccccc5o4)c3C2=O)C(=O)N1	C33H30N4O8	SMAD3	P84022	CRBN	WO-2022148459-A1
TPD-WWK1O4	SCHEMBL24620953	2-[[1-benzofuran-2-yl(pyridin-3-yl)methyl]amino]-N-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]butyl]acetamide	O=C(CNC(c1cccnc1)c1cc2ccccc2o1)NCCCCNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O	C33H32N6O6	SMAD3	P84022	CRBN	WO-2022148459-A1
TPD-QHAE7Z	SCHEMBL24620954	2-[[1-benzofuran-2-yl(pyridin-3-yl)methyl]amino]-N-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxybutyl]acetamide	O=C(CNC(c1cccnc1)c1cc2ccccc2o1)NCCCCOc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O	C33H31N5O7	SMAD3	P84022	CRBN	WO-2022148459-A1
TPD-MKE75B	SCHEMBL24620975	2-[[1-benzofuran-2-yl(pyridin-3-yl)methyl]amino]-N-[5-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]pentyl]acetamide	O=C(CNC(c1cccnc1)c1cc2ccccc2o1)NCCCCCc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O	C34H33N5O6	SMAD3	P84022	CRBN	WO-2022148459-A1
TPD-5N78E6	SCHEMBL24620968	3-[[1-benzofuran-2-yl(pyridin-3-yl)methyl]amino]-N-[3-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]propyl]propanamide	O=C(CCNC(c1cccnc1)c1cc2ccccc2o1)NCCCNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O	C33H32N6O6	SMAD3	P84022	CRBN	WO-2022148459-A1
TPD-IANHZQ	SCHEMBL24620971	3-[[1-benzofuran-2-yl(pyridin-3-yl)methyl]amino]-N-[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxypropyl]propanamide	O=C(CCNC(c1cccnc1)c1cc2ccccc2o1)NCCCOc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O	C33H31N5O7	SMAD3	P84022	CRBN	WO-2022148459-A1
TPD-E7HI5O	SCHEMBL24620987	N-[2-[[1-benzofuran-2-yl(pyridin-3-yl)methyl]amino]ethyl]-4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]butanamide	O=C(CCCNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O)NCCNC(c1cccnc1)c1cc2ccccc2o1	C33H32N6O6	SMAD3	P84022	CRBN	WO-2022148459-A1
TPD-ZZTTA2	SCHEMBL24620995	N-[2-[[1-benzofuran-2-yl(pyridin-3-yl)methyl]amino]ethyl]-4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxybutanamide	O=C(CCCOc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O)NCCNC(c1cccnc1)c1cc2ccccc2o1	C33H31N5O7	SMAD3	P84022	CRBN	WO-2022148459-A1
TPD-2PECV5	SCHEMBL24620924	N-[3-[[1-benzofuran-2-yl(pyridin-3-yl)methyl]amino]propyl]-3-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]propanamide	O=C(CCNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O)NCCCNC(c1cccnc1)c1cc2ccccc2o1	C33H32N6O6	SMAD3	P84022	CRBN	WO-2022148459-A1
TPD-3O61HU	SCHEMBL24620989	N-[3-[[1-benzofuran-2-yl(pyridin-3-yl)methyl]amino]propyl]-3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxypropanamide	O=C(CCOc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O)NCCCNC(c1cccnc1)c1cc2ccccc2o1	C33H31N5O7	SMAD3	P84022	CRBN	WO-2022148459-A1
TPD-ZL4YN8	SCHEMBL24620846	N-[1-benzofuran-2-yl(pyridin-3-yl)methyl]-2-[4-[[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]methyl]piperidin-1-yl]acetamide	O=C1CCC(N2C(=O)c3cccc(NCC4CCN(CC(=O)NC(c5cccnc5)c5cc6ccccc6o5)CC4)c3C2=O)C(=O)N1	C35H34N6O6	SMAD3	P84022	CRBN	WO-2022148459-A1
TPD-RP4SK9	SCHEMBL24621142	N-[1-benzofuran-2-yl(pyridin-3-yl)methyl]-2-[4-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethyl]piperidin-1-yl]acetamide	O=C1CCC(N2C(=O)c3cccc(NCCC4CCN(CC(=O)NC(c5cccnc5)c5cc6ccccc6o5)CC4)c3C2=O)C(=O)N1	C36H36N6O6	SMAD3	P84022	CRBN	WO-2022148459-A1
TPD-WXU7I1	SCHEMBL24620826	N-[1-benzofuran-2-yl(pyridin-3-yl)methyl]-2-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]butoxy]acetamide	O=C1CCC(N2C(=O)c3cccc(NCCCCOCC(=O)NC(c4cccnc4)c4cc5ccccc5o4)c3C2=O)C(=O)N1	C33H31N5O7	SMAD3	P84022	CRBN	WO-2022148459-A1
TPD-DDANGV	SCHEMBL24620858	N-[1-benzofuran-2-yl(pyridin-4-yl)methyl]-7-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]heptanamide	O=C1CCC(N2C(=O)c3cccc(NCCCCCCC(=O)NC(c4ccncc4)c4cc5ccccc5o4)c3C2=O)C(=O)N1	C34H33N5O6	SMAD3	P84022	CRBN	WO-2022148459-A1
TPD-8NGV98	SCHEMBL24620854	N-[1-benzofuran-2-yl(pyridin-3-yl)methyl]-2-[1-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethyl]piperidin-4-yl]acetamide	O=C1CCC(N2C(=O)c3cccc(NCCN4CCC(CC(=O)NC(c5cccnc5)c5cc6ccccc6o5)CC4)c3C2=O)C(=O)N1	C36H36N6O6	SMAD3	P84022	CRBN	WO-2022148459-A1
TPD-86O2H6	SCHEMBL24621011	N-[1-benzofuran-2-yl(pyridin-3-yl)methyl]-2-[4-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethyl]phenyl]acetamide	O=C1CCC(N2C(=O)c3cccc(NCCc4ccc(CC(=O)NC(c5cccnc5)c5cc6ccccc6o5)cc4)c3C2=O)C(=O)N1	C37H31N5O6	SMAD3	P84022	CRBN	WO-2022148459-A1
TPD-V4UGNI	SCHEMBL24621031	N-[1-benzofuran-2-yl(pyridin-3-yl)methyl]-2-[4-[[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]methyl]phenyl]acetamide	O=C1CCC(N2C(=O)c3cccc(NCc4ccc(CC(=O)NC(c5cccnc5)c5cc6ccccc6o5)cc4)c3C2=O)C(=O)N1	C36H29N5O6	SMAD3	P84022	CRBN	WO-2022148459-A1
TPD-7TT55R	SCHEMBL24620880	7-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]-N-[(1-methylbenzimidazol-2-yl)-pyridin-3-ylmethyl]heptanamide	Cn1c(C(NC(=O)CCCCCCNc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)c2cccnc2)nc2ccccc21	C34H35N7O5	SMAD3	P84022	CRBN	WO-2022148459-A1
TPD-H8FGU0	SCHEMBL24621154	N-[1-benzofuran-2-yl(pyridin-3-yl)methyl]-4-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]butanamide	O=C1CCC(N2C(=O)c3cccc(NCCOCCCC(=O)NC(c4cccnc4)c4cc5ccccc5o4)c3C2=O)C(=O)N1	C33H31N5O7	SMAD3	P84022	CRBN	WO-2022148459-A1
TPD-PUFCIL	SCHEMBL24620918	N-[1-benzofuran-2-yl(pyridin-3-yl)methyl]-4-[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]prop-2-ynoxy]butanamide	O=C1CCC(N2C(=O)c3cccc(C#CCOCCCC(=O)NC(c4cccnc4)c4cc5ccccc5o4)c3C2=O)C(=O)N1	C34H28N4O7	SMAD3	P84022	CRBN	WO-2022148459-A1
TPD-56XNGO	SCHEMBL24621016	N-[1-benzofuran-2-yl(pyridin-3-yl)methyl]-2-[3-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethyl]phenyl]acetamide	O=C1CCC(N2C(=O)c3cccc(NCCc4cccc(CC(=O)NC(c5cccnc5)c5cc6ccccc6o5)c4)c3C2=O)C(=O)N1	C37H31N5O6	SMAD3	P84022	CRBN	WO-2022148459-A1
TPD-ML3YLV	SCHEMBL24620876	N-[1-benzofuran-2-yl(pyridin-2-yl)methyl]-7-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]heptanamide	O=C1CCC(N2C(=O)c3cccc(NCCCCCCC(=O)NC(c4ccccn4)c4cc5ccccc5o4)c3C2=O)C(=O)N1	C34H33N5O6	SMAD3	P84022	CRBN	WO-2022148459-A1
TPD-WYGSOU	SCHEMBL24620865	7-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]-N-[(1-methylindol-2-yl)-pyridin-3-ylmethyl]heptanamide	Cn1c(C(NC(=O)CCCCCCNc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)c2cccnc2)cc2ccccc21	C35H36N6O5	SMAD3	P84022	CRBN	WO-2022148459-A1
TPD-WQBNFQ	SCHEMBL24621209	N-[1-benzofuran-2-yl(pyridin-3-yl)methyl]-3-[3-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]propyl-methylamino]propanamide	CN(CCCNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O)CCC(=O)NC(c1cccnc1)c1cc2ccccc2o1	C34H34N6O6	SMAD3	P84022	CRBN	WO-2022148459-A1
TPD-3325F7	SCHEMBL24621013	N-[1-benzofuran-2-yl(pyridin-3-yl)methyl]-3-[3-[[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]methyl]phenyl]propanamide	O=C1CCC(N2C(=O)c3cccc(NCc4cccc(CCC(=O)NC(c5cccnc5)c5cc6ccccc6o5)c4)c3C2=O)C(=O)N1	C37H31N5O6	SMAD3	P84022	CRBN	WO-2022148459-A1
TPD-T1TPZU	SCHEMBL24620837	N-[1-benzofuran-2-yl(pyridin-3-yl)methyl]-3-[6-[[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]methyl]pyridin-2-yl]propanamide	O=C1CCC(N2C(=O)c3cccc(NCc4cccc(CCC(=O)NC(c5cccnc5)c5cc6ccccc6o5)n4)c3C2=O)C(=O)N1	C36H30N6O6	SMAD3	P84022	CRBN	WO-2022148459-A1
TPD-OCP3WV	SCHEMBL24620862	7-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]-N-[furo[2,3-c]pyridin-2-yl(pyridin-3-yl)methyl]heptanamide	O=C1CCC(N2C(=O)c3cccc(NCCCCCCC(=O)NC(c4cccnc4)c4cc5ccncc5o4)c3C2=O)C(=O)N1	C33H32N6O6	SMAD3	P84022	CRBN	WO-2022148459-A1
TPD-6OCW49	SCHEMBL24621474	N-[1-benzofuran-2-yl(pyridin-3-yl)methyl]-4-[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]propoxy]butanamide	O=C1CCC(N2C(=O)c3cccc(CCCOCCCC(=O)NC(c4cccnc4)c4cc5ccccc5o4)c3C2=O)C(=O)N1	C34H32N4O7	SMAD3	P84022	CRBN	WO-2022148459-A1
TPD-N94SRI	SCHEMBL24620860	7-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]-N-[furo[3,2-b]pyridin-2-yl(pyridin-3-yl)methyl]heptanamide	O=C1CCC(N2C(=O)c3cccc(NCCCCCCC(=O)NC(c4cccnc4)c4cc5ncccc5o4)c3C2=O)C(=O)N1	C33H32N6O6	SMAD3	P84022	CRBN	WO-2022148459-A1
TPD-UCSIOF	SCHEMBL24621238	N-[1-benzofuran-2-yl(pyridin-3-yl)methyl]-3-[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]sulfanylpropoxy]propanamide	O=C1CCC(N2C(=O)c3cccc(SCCCOCCC(=O)NC(c4cccnc4)c4cc5ccccc5o4)c3C2=O)C(=O)N1	C33H30N4O7S	SMAD3	P84022	CRBN	WO-2022148459-A1
TPD-K3FTN8	SCHEMBL24621034	N-[1-benzofuran-2-yl(pyridin-3-yl)methyl]-2-[3-[[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]methyl]phenyl]acetamide	O=C1CCC(N2C(=O)c3cccc(NCc4cccc(CC(=O)NC(c5cccnc5)c5cc6ccccc6o5)c4)c3C2=O)C(=O)N1	C36H29N5O6	SMAD3	P84022	CRBN	WO-2022148459-A1
TPD-395LNF	SCHEMBL24621015	N-[1-benzofuran-2-yl(pyridin-3-yl)methyl]-2-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxymethyl]phenyl]acetamide	O=C1CCC(N2C(=O)c3cccc(OCc4ccc(CC(=O)NC(c5cccnc5)c5cc6ccccc6o5)cc4)c3C2=O)C(=O)N1	C36H28N4O7	SMAD3	P84022	CRBN	WO-2022148459-A1
TPD-1MWE5Y	SCHEMBL24621207	N-[1-benzofuran-2-yl(pyridin-3-yl)methyl]-2-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]sulfanylbutoxy]acetamide	O=C1CCC(N2C(=O)c3cccc(SCCCCOCC(=O)NC(c4cccnc4)c4cc5ccccc5o4)c3C2=O)C(=O)N1	C33H30N4O7S	SMAD3	P84022	CRBN	WO-2022148459-A1
TPD-CVVS58	SCHEMBL24621206	N-[1-benzofuran-2-yl(pyridin-3-yl)methyl]-7-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]sulfanylheptanamide	O=C1CCC(N2C(=O)c3cccc(SCCCCCCC(=O)NC(c4cccnc4)c4cc5ccccc5o4)c3C2=O)C(=O)N1	C34H32N4O6S	SMAD3	P84022	CRBN	WO-2022148459-A1
TPD-BOBUWT	SCHEMBL24620834	N-[1-benzofuran-2-yl(pyridin-3-yl)methyl]-3-[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]sulfanylpropyl-methylamino]propanamide	CN(CCCSc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O)CCC(=O)NC(c1cccnc1)c1cc2ccccc2o1	C34H33N5O6S	SMAD3	P84022	CRBN	WO-2022148459-A1
TPD-18YTM1	SCHEMBL24621012	N-[1-benzofuran-2-yl(pyridin-3-yl)methyl]-3-[4-[[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]methyl]phenyl]propanamide	O=C1CCC(N2C(=O)c3cccc(NCc4ccc(CCC(=O)NC(c5cccnc5)c5cc6ccccc6o5)cc4)c3C2=O)C(=O)N1	C37H31N5O6	SMAD3	P84022	CRBN	WO-2022148459-A1
TPD-UJ6JUA	SCHEMBL24621025	N-[1-benzofuran-2-yl(pyridin-3-yl)methyl]-4-[[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]methyl]benzamide	O=C1CCC(N2C(=O)c3cccc(NCc4ccc(C(=O)NC(c5cccnc5)c5cc6ccccc6o5)cc4)c3C2=O)C(=O)N1	C35H27N5O6	SMAD3	P84022	CRBN	WO-2022148459-A1
TPD-ZJLGS5	SCHEMBL24620926	N-[1-benzofuran-2-yl(pyridin-3-yl)methyl]-2-[4-[[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]methyl]phenyl]acetamide	O=C1CCC(N2Cc3c(NCc4ccc(CC(=O)NC(c5cccnc5)c5cc6ccccc6o5)cc4)cccc3C2=O)C(=O)N1	C36H31N5O5	SMAD3	P84022	CRBN	WO-2022148459-A1
TPD-KG1CHY	SCHEMBL24620881	N-[1,3-benzothiazol-2-yl(pyridin-3-yl)methyl]-7-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]heptanamide	O=C1CCC(N2C(=O)c3cccc(NCCCCCCC(=O)NC(c4cccnc4)c4nc5ccccc5s4)c3C2=O)C(=O)N1	C33H32N6O5S	SMAD3	P84022	CRBN	WO-2022148459-A1
TPD-1MSR2N	SCHEMBL24620838	N-[1-benzofuran-2-yl(pyrimidin-5-yl)methyl]-7-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]heptanamide	O=C1CCC(N2C(=O)c3cccc(NCCCCCCC(=O)NC(c4cncnc4)c4cc5ccccc5o4)c3C2=O)C(=O)N1	C33H32N6O6	SMAD3	P84022	CRBN	WO-2022148459-A1
TPD-M9G98Z	SCHEMBL24620839	N-[1-benzothiophen-2-yl(pyridin-3-yl)methyl]-7-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]heptanamide	O=C1CCC(N2C(=O)c3cccc(NCCCCCCC(=O)NC(c4cccnc4)c4cc5ccccc5s4)c3C2=O)C(=O)N1	C34H33N5O5S	SMAD3	P84022	CRBN	WO-2022148459-A1
TPD-7PTAFL	SCHEMBL24620887	N-[1,3-benzoxazol-2-yl(pyridin-3-yl)methyl]-7-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]heptanamide	O=C1CCC(N2C(=O)c3cccc(NCCCCCCC(=O)NC(c4cccnc4)c4nc5ccccc5o4)c3C2=O)C(=O)N1	C33H32N6O6	SMAD3	P84022	CRBN	WO-2022148459-A1
TPD-49GOQ3	SCHEMBL24620864	7-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]-N-[furo[2,3-b]pyridin-2-yl(pyridin-3-yl)methyl]heptanamide	O=C1CCC(N2C(=O)c3cccc(NCCCCCCC(=O)NC(c4cccnc4)c4cc5cccnc5o4)c3C2=O)C(=O)N1	C33H32N6O6	SMAD3	P84022	CRBN	WO-2022148459-A1
TPD-5DNKFX	SCHEMBL24621029	N-[1-benzofuran-2-yl(pyridin-3-yl)methyl]-2-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]ethynyl]phenyl]acetamide	O=C1CCC(N2C(=O)c3cccc(C#Cc4ccc(CC(=O)NC(c5cccnc5)c5cc6ccccc6o5)cc4)c3C2=O)C(=O)N1	C37H26N4O6	SMAD3	P84022	CRBN	WO-2022148459-A1
TPD-U50R1Y	SCHEMBL24621032	N-[1-benzofuran-2-yl(pyridin-3-yl)methyl]-2-[4-[(Z)-2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]ethenyl]phenyl]acetamide	O=C1CCC(N2C(=O)c3cccc(/C=C\c4ccc(CC(=O)NC(c5cccnc5)c5cc6ccccc6o5)cc4)c3C2=O)C(=O)N1	C37H28N4O6	SMAD3	P84022	CRBN	WO-2022148459-A1
TPD-LQRZW9	SCHEMBL24621021	N-[1-benzofuran-2-yl(pyridin-3-yl)methyl]-2-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]ethyl]phenyl]acetamide	O=C1CCC(N2C(=O)c3cccc(CCc4ccc(CC(=O)NC(c5cccnc5)c5cc6ccccc6o5)cc4)c3C2=O)C(=O)N1	C37H30N4O6	SMAD3	P84022	CRBN	WO-2022148459-A1
TPD-73WT84	SCHEMBL24620913	N-[1-benzothiophen-2-yl(pyridin-3-yl)methyl]-2-[4-[[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]methyl]phenyl]acetamide	O=C1CCC(N2C(=O)c3cccc(NCc4ccc(CC(=O)NC(c5cccnc5)c5cc6ccccc6s5)cc4)c3C2=O)C(=O)N1	C36H29N5O5S	SMAD3	P84022	CRBN	WO-2022148459-A1
TPD-5G06IV	SCHEMBL24621017	N-[1-benzofuran-2-yl(pyridin-3-yl)methyl]-2-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]sulfanylmethyl]phenyl]acetamide	O=C1CCC(N2C(=O)c3cccc(SCc4ccc(CC(=O)NC(c5cccnc5)c5cc6ccccc6o5)cc4)c3C2=O)C(=O)N1	C36H28N4O6S	SMAD3	P84022	CRBN	WO-2022148459-A1
TPD-OKZS4O	SCHEMBL24620885	N-[1-benzofuran-2-yl(pyridin-3-yl)methyl]-2-[4-[[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]methyl]triazol-1-yl]acetamide	O=C1CCC(N2C(=O)c3cccc(NCc4cn(CC(=O)NC(c5cccnc5)c5cc6ccccc6o5)nn4)c3C2=O)C(=O)N1	C32H26N8O6	SMAD3	P84022	CRBN	WO-2022148459-A1
TPD-KA1VO2	SCHEMBL24621027	N-[1-benzofuran-2-yl(pyridin-3-yl)methyl]-2-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]phenyl]acetamide	O=C1CCC(N2C(=O)c3cccc(Nc4ccc(CC(=O)NC(c5cccnc5)c5cc6ccccc6o5)cc4)c3C2=O)C(=O)N1	C35H27N5O6	SMAD3	P84022	CRBN	WO-2022148459-A1
TPD-5JIQBP	CHEMBL5079358	2-[4-(3-chloro-4-fluoroanilino)-7-methoxyquinazolin-6-yl]oxy-N-[3-[4-[[1-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethyl]triazol-4-yl]methoxy]phenyl]-1-[4-[2-fluoro-5-[(4-oxo-3H-phthalazin-1-yl)methyl]benzoyl]piperazin-1-yl]-1-oxopropan-2-yl]acetamide; BDBM50582623	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1OCC(=O)NC(Cc1ccc(OCc2cn(CCOCCNc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)nn2)cc1)C(=O)N1CCN(C(=O)c2cc(Cc3n[nH]c(=O)c4ccccc34)ccc2F)CC1	C66H59ClF2N14O12	EGFR;PARP1	P00533/P09874	CRBN	WO-2022166570-A1
TPD-1DGUP1	CHEMBL5078576	4-[4-(3-chloro-4-fluoroanilino)-7-methoxyquinazolin-6-yl]oxy-N-[3-[[1-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethyl]triazol-4-yl]methoxy]-1-[4-[2-fluoro-5-[(4-oxo-3H-phthalazin-1-yl)methyl]benzoyl]piperazin-1-yl]-1-oxopropan-2-yl]butanamide	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1OCCCC(=O)NC(COCc1cn(CCOCCNc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)nn1)C(=O)N1CCN(C(=O)c2cc(Cc3n[nH]c(=O)c4ccccc34)ccc2F)CC1	C62H59ClF2N14O12	EGFR;PARP1	P00533/P09874	CRBN	WO-2022166570-A1
TPD-NHK41R	CHEMBL5084430	4-[4-(3-chloro-4-fluoroanilino)-7-methoxyquinazolin-6-yl]oxy-N-[3-[[1-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethyl]triazol-4-yl]methoxy]-1-[[4-[4-[2-fluoro-5-[(4-oxo-3H-phthalazin-1-yl)methyl]benzoyl]piperazin-1-yl]-4-oxobutyl]amino]-1-oxopropan-2-yl]butanamide	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1OCCCC(=O)NC(COCc1cn(CCOCCNc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)nn1)C(=O)NCCCC(=O)N1CCN(C(=O)c2cc(Cc3n[nH]c(=O)c4ccccc34)ccc2F)CC1	C66H66ClF2N15O13	EGFR;PARP1	P00533/P09874	CRBN	WO-2022166570-A1
TPD-NXV304	DP-C-4	CID 162641005; CHEMBL5077447; MS-32172; HY-141481; CS-0173214; G18225; 6-[4-(3-chloro-4-fluoroanilino)-7-methoxyquinazolin-6-yl]oxy-N-[3-[[1-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethyl]triazol-4-yl]methoxy]-1-[[6-[4-[2-fluoro-5-[(4-oxo-3H-phthalazin-1-yl)methyl]benzoyl]piperazin-1-yl]-6-oxohexyl]amino]-1-oxopropan-2-yl]hexanamide	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1OCCCCCC(=O)NC(COCc1cn(CCOCCOCCNc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)nn1)C(=O)NCCCCCC(=O)N1CCN(C(=O)c2cc(Cc3n[nH]c(=O)c4ccccc34)ccc2F)CC1	C72H78ClF2N15O14	EGFR;PARP1	P00533/P09874	CRBN	WO-2022166570-A1
TPD-Q5ISRB	CHEMBL5081703	(2S,4R)-1-[(2S)-2-[4-[4-[[4-[2-[[2-[4-(3-chloro-4-fluoroanilino)-7-methoxyquinazolin-6-yl]oxyacetyl]amino]-3-[4-[2-fluoro-5-[(4-oxo-3H-phthalazin-1-yl)methyl]benzoyl]piperazin-1-yl]-3-oxopropyl]phenoxy]methyl]triazol-1-yl]butanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1OCC(=O)NC(Cc1ccc(OCc2cn(CCCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCc3ccc(-c4scnc4C)cc3)C(C)(C)C)nn2)cc1)C(=O)N1CCN(C(=O)c2cc(Cc3n[nH]c(=O)c4ccccc34)ccc2F)CC1	C75H76ClF2N15O11S	EGFR;PARP1	P00533/P09874	VHL	WO-2022166570-A1
TPD-S26H10	CHEMBL5091185	(2S,4R)-1-[(2S)-2-[4-[4-[[2-[4-[4-(3-chloro-4-fluoroanilino)-7-methoxyquinazolin-6-yl]oxybutanoylamino]-3-[4-[2-fluoro-5-[(4-oxo-3H-phthalazin-1-yl)methyl]benzoyl]piperazin-1-yl]-3-oxopropoxy]methyl]triazol-1-yl]butanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1OCCCC(=O)NC(COCc1cn(CCCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCc2ccc(-c3scnc3C)cc2)C(C)(C)C)nn1)C(=O)N1CCN(C(=O)c2cc(Cc3n[nH]c(=O)c4ccccc34)ccc2F)CC1	C71H76ClF2N15O11S	EGFR;PARP1	P00533/P09874	VHL	WO-2022166570-A1
TPD-S59N05	CHEMBL5091616	(2S,4R)-1-[(2S)-2-[4-[4-[[2-[6-[4-(3-chloro-4-fluoroanilino)-7-methoxyquinazolin-6-yl]oxyhexanoylamino]-3-[[2-[4-[2-fluoro-5-[(4-oxo-3H-phthalazin-1-yl)methyl]benzoyl]piperazin-1-yl]-2-oxoethyl]amino]-3-oxopropoxy]methyl]triazol-1-yl]butanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1OCCCCCC(=O)NC(COCc1cn(CCCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCc2ccc(-c3scnc3C)cc2)C(C)(C)C)nn1)C(=O)NCC(=O)N1CCN(C(=O)c2cc(Cc3n[nH]c(=O)c4ccccc34)ccc2F)CC1	C75H83ClF2N16O12S	EGFR;PARP1	P00533/P09874	VHL	WO-2022166570-A1
TPD-5LJIK9	CHEMBL5091890	(2S,4R)-1-[(2S)-2-[4-[4-[[2-[6-[4-(3-chloro-4-fluoroanilino)-7-methoxyquinazolin-6-yl]oxyhexanoylamino]-3-[[6-[4-[2-fluoro-5-[(4-oxo-3H-phthalazin-1-yl)methyl]benzoyl]piperazin-1-yl]-6-oxohexyl]amino]-3-oxopropoxy]methyl]triazol-1-yl]butanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; BDBM50582622	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1OCCCCCC(=O)NC(COCc1cn(CCCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCc2ccc(-c3scnc3C)cc2)C(C)(C)C)nn1)C(=O)NCCCCCC(=O)N1CCN(C(=O)c2cc(Cc3n[nH]c(=O)c4ccccc34)ccc2F)CC1	C79H91ClF2N16O12S	EGFR;PARP1	P00533/P09874	VHL	WO-2022166570-A1
TPD-GB2WJW	CHEMBL5072342	4-[4-(3-chloro-4-fluoroanilino)-7-methoxyquinazolin-6-yl]oxy-N-[[1-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethyl]triazol-4-yl]methyl]butanamide	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1OCCCC(=O)NCc1cn(CCOCCNc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)nn1	C39H38ClFN10O8	EGFR;PARP1	P00533/P09874	CRBN	WO-2022166570-A1
TPD-RCSIEE	CHEMBL5076607	2-(2,6-dioxopiperidin-3-yl)-4-[2-[2-[4-[3-[4-[2-fluoro-5-[(4-oxo-3H-phthalazin-1-yl)methyl]benzoyl]piperazin-1-yl]-3-oxopropyl]triazol-1-yl]ethoxy]ethylamino]isoindole-1,3-dione	O=C1CCC(N2C(=O)c3cccc(NCCOCCn4cc(CCC(=O)N5CCN(C(=O)c6cc(Cc7n[nH]c(=O)c8ccccc78)ccc6F)CC5)nn4)c3C2=O)C(=O)N1	C42H41FN10O8	EGFR;PARP1	P00533/P09874	CRBN	WO-2022166570-A1
TPD-F8BONO	CHEMBL5086725	(2S,4R)-1-[(2S)-2-[4-[4-[[4-[4-(3-chloro-4-fluoroanilino)-7-methoxyquinazolin-6-yl]oxybutanoylamino]methyl]triazol-1-yl]butanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1OCCCC(=O)NCc1cn(CCCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCc2ccc(-c3scnc3C)cc2)C(C)(C)C)nn1	C48H55ClFN11O7S	EGFR;PARP1	P00533/P09874	VHL	WO-2022166570-A1
TPD-UWC8L1	CHEMBL5076946	(2S,4R)-1-[(2S)-2-[4-[4-[3-[4-[2-fluoro-5-[(4-oxo-3H-phthalazin-1-yl)methyl]benzoyl]piperazin-1-yl]-3-oxopropyl]triazol-1-yl]butanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCn2cc(CCC(=O)N3CCN(C(=O)c4cc(Cc5n[nH]c(=O)c6ccccc56)ccc4F)CC3)nn2)C(C)(C)C)cc1	C51H58FN11O7S	EGFR;PARP1	P00533/P09874	VHL	WO-2022166570-A1
TPD-ZUNETX	SCHEMBL26917667	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[[16-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-16-oxohexadecyl]-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL26917680	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCCCCCCCCCCN(C)CCOC23CC4(C)CC(C)(CC(Cn5ncc(-c6ccc(N7CCCc8c7nnc(Nc7nc9ccccc9s7)c8C)nc6C(=O)O)c5C)(C4)C2)C3)C(C)(C)C)cc1	C80H109N13O7S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-USLYHX	SCHEMBL26917995	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[[12-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-12-oxododecyl]-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL26918006	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCCCCCCN(C)CCOC23CC4(C)CC(C)(CC(Cn5ncc(-c6ccc(N7CCCc8c7nnc(Nc7nc9ccccc9s7)c8C)nc6C(=O)O)c5C)(C4)C2)C3)C(C)(C)C)cc1	C76H101N13O7S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-WL2JNS	WO2022169780A1_3	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@H]2C[C@H](O)CN2C(=O)[C@H](NC(=O)CCCCCCN(C)CCOC23CC4(C)CC(C)(CC(Cn5ncc(-c6ccc(N7CCCc8c7nnc(Nc7nc9ccccc9s7)c8C)nc6C(=O)O)c5C)(C4)C2)C3)C(C)(C)C)cc1	C71H91N13O7S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-SRW0D5	SCHEMBL26917893	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[[14-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-14-oxotetradecyl]-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL26917903	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCCCCCCCCN(C)CCOC23CC4(C)CC(C)(CC(Cn5ncc(-c6ccc(N7CCCc8c7nnc(Nc7nc9ccccc9s7)c8C)nc6C(=O)O)c5C)(C4)C2)C3)C(C)(C)C)cc1	C78H105N13O7S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-N9U153	WO2022169780A1_5	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@H]2C[C@H](O)CN2C(=O)[C@H](NC(=O)CCCCCCCCN(C)CCOC23CC4(C)CC(C)(CC(Cn5ncc(-c6ccc(N7CCCc8c7nnc(Nc7nc9ccccc9s7)c8C)nc6C(=O)O)c5C)(C4)C2)C3)C(C)(C)C)cc1	C73H95N13O7S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-XBMLTT	SCHEMBL26917983	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[[8-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-8-oxooctyl]-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL26917990	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCCN(C)CCOC23CC4(C)CC(C)(CC(Cn5ncc(-c6ccc(N7CCCc8c7nnc(Nc7nc9ccccc9s7)c8C)nc6C(=O)O)c5C)(C4)C2)C3)C(C)(C)C)cc1	C72H93N13O7S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-P9QHWQ	WO2022169780A1_7	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@H](O)CN2C(=O)[C@@H](CC(=O)CCCCCCCCCCCCCCN(C)CCOC23CC4(C)CC(C)(CC(Cn5ncc(-c6ccc(N7CCCc8c7nnc(Nc7nc9ccccc9s7)c8C)nc6C(=O)O)c5C)(C4)C2)C3)C(C)(C)C)cc1	C80H108N12O7S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-TA8HWR	WO2022169780A1_8	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@H]2C[C@@H](O)CN2C(=O)[C@H](NC(=O)CCCCCN(C)CCOC23CC4(C)CC(C)(CC(Cn5ncc(-c6ccc(N7CCCc8c7nnc(Nc7nc9ccccc9s7)c8C)nc6C(=O)O)c5C)(C4)C2)C3)C(C)(C)C)cc1	C70H89N13O7S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-6KLKKD	SCHEMBL26917790	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethyl-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL30670813	Cc1c(Nc2nc3ccccc3s2)nnc2c1CCCN2c1ccc(-c2cnn(CC34CC5(C)CC(C)(C3)CC(OCCN(C)CCOCCNc3cccc6c3C(=O)N(C3CCC(=O)NC3=O)C6=O)(C5)C4)c2C)c(C(=O)O)n1	C58H66N12O8S	BCL2L1	Q07817	CRBN	WO-2022169780-A1
TPD-JTHQJR	SCHEMBL26917702	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[8-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxyoctyl-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL30670803	Cc1c(Nc2nc3ccccc3s2)nnc2c1CCCN2c1ccc(-c2cnn(CC34CC5(C)CC(C)(C3)CC(OCCN(C)CCCCCCCCOc3ccc6c(c3)C(=O)N(C3CCC(=O)NC3=O)C6=O)(C5)C4)c2C)c(C(=O)O)n1	C62H73N11O8S	BCL2L1	Q07817	CRBN	WO-2022169780-A1
TPD-4MLHK6	SCHEMBL26917701	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethyl-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL30670800	Cc1c(Nc2nc3ccccc3s2)nnc2c1CCCN2c1ccc(-c2cnn(CC34CC5(C)CC(C)(C3)CC(OCCN(C)CCOCCOCCOCCNc3cccc6c3C(=O)N(C3CCC(=O)NC3=O)C6=O)(C5)C4)c2C)c(C(=O)O)n1	C62H74N12O10S	BCL2L1	Q07817	CRBN	WO-2022169780-A1
TPD-8487NG	SCHEMBL26917450	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethyl-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL30670780	Cc1c(Nc2nc3ccccc3s2)nnc2c1CCCN2c1ccc(-c2cnn(CC34CC5(C)CC(C)(C3)CC(OCCN(C)CCOCCOCCNc3cccc6c3C(=O)N(C3CCC(=O)NC3=O)C6=O)(C5)C4)c2C)c(C(=O)O)n1	C60H70N12O9S	BCL2L1	Q07817	CRBN	WO-2022169780-A1
TPD-CZDTO0	SCHEMBL26917715	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[2-[2-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethyl-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL30670926	Cc1c(Nc2nc3ccccc3s2)nnc2c1CCCN2c1ccc(-c2cnn(CC34CC5(C)CC(C)(C3)CC(OCCN(C)CCOCCOCCOCCOCCOCCNc3cccc6c3C(=O)N(C3CCC(=O)NC3=O)C6=O)(C5)C4)c2C)c(C(=O)O)n1	C66H82N12O12S	BCL2L1	Q07817	CRBN	WO-2022169780-A1
TPD-NJWY7O	SCHEMBL26918031	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[6-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxyhexyl-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL30670796	Cc1c(Nc2nc3ccccc3s2)nnc2c1CCCN2c1ccc(-c2cnn(CC34CC5(C)CC(C)(C3)CC(OCCN(C)CCCCCCOc3ccc6c(c3)C(=O)N(C3CCC(=O)NC3=O)C6=O)(C5)C4)c2C)c(C(=O)O)n1	C60H69N11O8S	BCL2L1	Q07817	CRBN	WO-2022169780-A1
TPD-S3JRYC	WO2022169780A1_15	2-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-5-[3-[2-fluoro-4-[3-[4-[7-[[(2R)-1-[(2R,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-7-oxoheptanoyl]piperazin-1-yl]prop-1-ynyl]phenoxy]propyl]-1,3-thiazole-4-carboxylic acid	Cc1ncsc1-c1ccc(CNC(=O)[C@H]2C[C@@H](O)CN2C(=O)[C@H](NC(=O)CCCCCC(=O)N2CCN(CC#Cc3ccc(OCCCc4sc(N5CCCc6c5nnc(Nc5nc7ccccc7s5)c6C)nc4C(=O)O)c(F)c3)CC2)C(C)(C)C)cc1	C64H73FN12O8S3	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-BJB54Y	WO2022169780A1_16	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@H]2C[C@@H](O)CN2C(=O)[C@H](NCCCCCCCC(=O)N2CCN(CC#Cc3ccc(OCCCc4sc(N5CCCc6c5nnc(Nc5nc7ccccc7s5)c6C)nc4C(=O)O)c(F)c3)CC2)C(C)(C)C)cc1	C66H79FN12O7S3	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-YS8ULN	WO2022169780A1_17	2-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-5-[3-[2-fluoro-4-[3-[4-[7-[[(2R)-1-[(2R,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-7-oxoheptanoyl]piperazin-1-yl]prop-1-ynyl]phenoxy]propyl]-1,3-thiazole-4-carboxylic acid	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@H]2C[C@@H](O)CN2C(=O)[C@H](NC(=O)CCCCCC(=O)N2CCN(CC#Cc3ccc(OCCCc4sc(N5CCCc6c5nnc(Nc5nc7ccccc7s5)c6C)nc4C(=O)O)c(F)c3)CC2)C(C)(C)C)cc1	C65H75FN12O8S3	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-B873XM	WO2022169780A1_18	2-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-5-[3-[2-fluoro-4-[3-[4-[5-[[(2R)-1-[(2R,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-5-oxopentanoyl]piperazin-1-yl]prop-1-ynyl]phenoxy]propyl]-1,3-thiazole-4-carboxylic acid	Cc1ncsc1-c1ccc(CNC(=O)[C@H]2C[C@@H](O)CN2C(=O)[C@H](NC(=O)CCCC(=O)N2CCN(CC#Cc3ccc(OCCCc4sc(N5CCCc6c5nnc(Nc5nc7ccccc7s5)c6C)nc4C(=O)O)c(F)c3)CC2)C(C)(C)C)cc1	C62H69FN12O8S3	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-3ZUES5	SCHEMBL26917570	2-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-5-[3-[2-fluoro-4-[3-[4-[6-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-6-oxohexanoyl]piperazin-1-yl]prop-1-ynyl]phenoxy]propyl]-1,3-thiazole-4-carboxylic acid; SCHEMBL30670854	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCC(=O)N2CCN(CC#Cc3ccc(OCCCc4sc(N5CCCc6c5nnc(Nc5nc7ccccc7s5)c6C)nc4C(=O)O)c(F)c3)CC2)C(C)(C)C)cc1	C63H71FN12O8S3	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-DID6LS	WO2022169780A1_20	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCC(=O)N2CCN(CC#Cc3ccc(OCCCc4sc(N5CCCc6c5nnc(Nc5nc7ccccc7s5)c6C)nc4C(=O)O)c(F)c3)CC2)C(C)(C)C)cc1	C65H75FN12O8S3	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-DH3OBB	WO2022169780A1_21	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@H](O)CN2C(=O)[C@@H](NC(=O)CCC(=O)N2CCN(CC#Cc3ccc(OCCCc4sc(N5CCCc6c5nnc(Nc5nc7ccccc7s5)c6C)nc4C(=O)O)c(F)c3)CC2)C(C)(C)C)cc1	C61H67FN12O8S3	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-8RF7MR	WO2022169780A1_22	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[4-[7-[[(2R)-1-[(2R,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-7-oxoheptanoyl]piperazin-1-yl]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid	Cc1ncsc1-c1ccc(CNC(=O)[C@H]2C[C@@H](O)CN2C(=O)[C@H](NC(=O)CCCCCC(=O)N2CCN(CCOC34CC5(C)CC(C)(CC(Cn6ncc(-c7ccc(N8CCCc9c8nnc(Nc8nc%10ccccc%10s8)c9C)nc7C(=O)O)c6C)(C5)C3)C4)CC2)C(C)(C)C)cc1	C73H92N14O8S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-PHTPKQ	WO2022169780A1_23	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[4-[6-[[(2R)-1-[(2S,4S)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-6-oxohexanoyl]piperazin-1-yl]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@H](O)CN2C(=O)[C@H](NC(=O)CCCCC(=O)N2CCN(CCOC34CC5(C)CC(C)(CC(Cn6ncc(-c7ccc(N8CCCc9c8nnc(Nc8nc%10ccccc%10s8)c9C)nc7C(=O)O)c6C)(C5)C3)C4)CC2)C(C)(C)C)cc1	C72H90N14O8S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-W64JLC	WO2022169780A1_24	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[4-[8-[[(2R)-1-[(2S,4S)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-8-oxooctanoyl]piperazin-1-yl]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@H](O)CN2C(=O)[C@H](NC(=O)CCCCCCC(=O)N2CCN(CCOC34CC5(C)CC(C)(CC(Cn6ncc(-c7ccc(N8CCCc9c8nnc(Nc8nc%10ccccc%10s8)c9C)nc7C(=O)O)c6C)(C5)C3)C4)CC2)C(C)(C)C)cc1	C74H94N14O8S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-LXXUPN	WO2022169780A1_25	.	Cc1c(Nc2nc3ccccc3s2)nnc2c1CCCN2c1nc(C(=O)O)c(CCCOc2ccc(C#CCN3CCN(C(=O)CCCCC(=O)NCCOCCNC(=O)COc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)cc2F)s1	C60H63FN12O12S2	BCL2L1	Q07817	CRBN	WO-2022169780-A1
TPD-LTVH73	SCHEMBL26917564	2-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-5-[3-[4-[3-[4-[5-[2-[2-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyacetyl]amino]ethoxy]ethylamino]-5-oxopentanoyl]piperazin-1-yl]prop-1-ynyl]-2-fluorophenoxy]propyl]-1,3-thiazole-4-carboxylic acid; SCHEMBL30670909	Cc1c(Nc2nc3ccccc3s2)nnc2c1CCCN2c1nc(C(=O)O)c(CCCOc2ccc(C#CCN3CCN(C(=O)CCCC(=O)NCCOCCNC(=O)COc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)cc2F)s1	C59H61FN12O12S2	BCL2L1	Q07817	CRBN	WO-2022169780-A1
TPD-D4YGJG	SCHEMBL26917547	2-[[6-(1,3-Benzothiazol-2-ylamino)-5-methylpyridazin-3-yl]-[3-[1-[2-[2-[2-[2-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyacetyl]amino]ethoxy]ethoxy]ethoxy]ethyl]triazol-4-yl]propyl]amino]-5-[3-[2-fluoro-4-[3-(methylamino)prop-1-ynyl]phenoxy]propyl]-1,3-thiazole-4-carboxylic acid; SCHEMBL30670911	CNCC#Cc1ccc(OCCCc2sc(N(CCCc3cn(CCOCCOCCOCCNC(=O)COc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)nn3)c3cc(C)c(Nc4nc5ccccc5s4)nn3)nc2C(=O)O)c(F)c1	C57H60FN13O12S2	BCL2L1	Q07817	CRBN	WO-2022169780-A1
TPD-SM79KQ	SCHEMBL26917949	6-[[6-(1,3-benzothiazol-2-ylamino)-5-methylpyridazin-3-yl]-[5-[4-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]-2-oxoethoxy]ethoxy]ethoxymethyl]triazol-1-yl]pentyl]amino]-3-[1-[[3-[2-(dimethylamino)ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid	Cc1cc(N(CCCCCn2cc(COCCOCCOCC(=O)Nc3cccc4c3CN(C3CCC(=O)NC3=O)C4=O)nn2)c2ccc(-c3cnn(CC45CC6(C)CC(C)(C4)CC(OCCN(C)C)(C6)C5)c3C)c(C(=O)O)n2)nnc1Nc1nc2ccccc2s1	C66H81N15O10S	BCL2L1	Q07817	CRBN	WO-2022169780-A1
TPD-6C1RFE	SCHEMBL26917800	2-[[6-(1,3-benzothiazol-2-ylamino)-5-methylpyridazin-3-yl]-[3-[1-[2-[2-[2-[2-[2-[3-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-3-oxopropoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethyl]triazol-4-yl]propyl]amino]-5-[3-[2-fluoro-4-[3-(methylamino)prop-1-ynyl]phenoxy]propyl]-1,3-thiazole-4-carboxylic acid; SCHEMBL26917810	CNCC#Cc1ccc(OCCCc2sc(N(CCCc3cn(CCOCCOCCOCCOCCOCCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)NCc4ccc(-c5scnc5C)cc4)C(C)(C)C)nn3)c3cc(C)c(Nc4nc5ccccc5s4)nn3)nc2C(=O)O)c(F)c1	C69H85FN14O12S3	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-EXI8LH	SCHEMBL26917851	2-[[6-(1,3-Benzothiazol-2-ylamino)-5-methylpyridazin-3-yl]-[3-[1-[8-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyacetyl]amino]octyl]triazol-4-yl]propyl]amino]-5-[3-[2-fluoro-4-[3-(methylamino)prop-1-ynyl]phenoxy]propyl]-1,3-thiazole-4-carboxylic acid; SCHEMBL26917890; SCHEMBL30670829; SCHEMBL30670863	CNCC#Cc1ccc(OCCCc2sc(N(CCCc3cn(CCCCCCCCNC(=O)COc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)nn3)c3cc(C)c(Nc4nc5ccccc5s4)nn3)nc2C(=O)O)c(F)c1	C57H60FN13O9S2	BCL2L1	Q07817	CRBN	WO-2022169780-A1
TPD-5FWC6S	WO2022169780A1_31	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@H]2C[C@H](O)CN2C(=O)[C@H](NC(=O)CCCCCCCCCCCN2CCN(CC#Cc3ccc(OCCCc4sc(N5CCCc6c5nnc(Nc5nc7ccccc7s5)c6C)nc4C(=O)O)c(F)c3)CC2)C(C)(C)C)cc1	C70H87FN12O7S3	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-PI5DLS	SCHEMBL26917379	2-[[6-(1,3-Benzothiazol-2-ylamino)-5-methylpyridazin-3-yl]-methylamino]-5-[3-[4-[3-[[2-[2-[2-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyacetyl]amino]ethoxy]ethylamino]-2-oxoethyl]-methylamino]prop-1-ynyl]-2-fluorophenoxy]propyl]-1,3-thiazole-4-carboxylic acid; SCHEMBL30670778	Cc1cc(N(C)c2nc(C(=O)O)c(CCCOc3ccc(C#CCN(C)CC(=O)NCCOCCNC(=O)COc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)cc3F)s2)nnc1Nc1nc2ccccc2s1	C51H50FN11O11S2	BCL2L1	Q07817	CRBN	WO-2022169780-A1
TPD-YA4C4T	SCHEMBL26917501	2-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-5-[3-[2-fluoro-4-[3-[4-[8-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-8-oxooctanoyl]piperazin-1-yl]prop-1-ynyl]phenoxy]propyl]-1,3-thiazole-4-carboxylic acid; SCHEMBL30670891	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCC(=O)N2CCN(CC#Cc3ccc(OCCCc4sc(N5CCCc6c5nnc(Nc5nc7ccccc7s5)c6C)nc4C(=O)O)c(F)c3)CC2)C(C)(C)C)cc1	C65H75FN12O8S3	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-NQ9E9L	SCHEMBL26917461	2-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-5-[3-[2-fluoro-4-[3-[4-[7-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-7-oxoheptanoyl]piperazin-1-yl]prop-1-ynyl]phenoxy]propyl]-1,3-thiazole-4-carboxylic acid; SCHEMBL30670823	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCC(=O)N2CCN(CC#Cc3ccc(OCCCc4sc(N5CCCc6c5nnc(Nc5nc7ccccc7s5)c6C)nc4C(=O)O)c(F)c3)CC2)C(C)(C)C)cc1	C65H75FN12O8S3	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-7638BK	SCHEMBL26917513	2-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-5-[3-[2-fluoro-4-[3-[4-[5-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-5-oxopentanoyl]piperazin-1-yl]prop-1-ynyl]phenoxy]propyl]-1,3-thiazole-4-carboxylic acid; SCHEMBL30671001; SCHEMBL30671003	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCC(=O)N2CCN(CC#Cc3ccc(OCCCc4sc(N5CCCc6c5nnc(Nc5nc7ccccc7s5)c6C)nc4C(=O)O)c(F)c3)CC2)C(C)(C)C)cc1	C63H71FN12O8S3	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-IVMBU6	SCHEMBL26917753	2-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-5-[3-[2-fluoro-4-[3-[4-[2-[[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethyl]-methylamino]acetyl]piperazin-1-yl]prop-1-ynyl]phenoxy]propyl]-1,3-thiazole-4-carboxylic acid; SCHEMBL30670790	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CN(C)CC(=O)N2CCN(CC#Cc3ccc(OCCCc4sc(N5CCCc6c5nnc(Nc5nc7ccccc7s5)c6C)nc4C(=O)O)c(F)c3)CC2)C(C)(C)C)cc1	C63H72FN13O8S3	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-PZS86I	SCHEMBL26917452	2-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-5-[3-[2-fluoro-4-[3-[4-[2-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethyl]sulfanylacetyl]piperazin-1-yl]prop-1-ynyl]phenoxy]propyl]-1,3-thiazole-4-carboxylic acid; SCHEMBL30670930	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CSCC(=O)N2CCN(CC#Cc3ccc(OCCCc4sc(N5CCCc6c5nnc(Nc5nc7ccccc7s5)c6C)nc4C(=O)O)c(F)c3)CC2)C(C)(C)C)cc1	C62H69FN12O8S4	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-SU39UL	SCHEMBL26917445	2-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-5-[3-[2-fluoro-4-[3-[4-[9-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-9-oxononanoyl]piperazin-1-yl]prop-1-ynyl]phenoxy]propyl]-1,3-thiazole-4-carboxylic acid; SCHEMBL30670905	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCCC(=O)N2CCN(CC#Cc3ccc(OCCCc4sc(N5CCCc6c5nnc(Nc5nc7ccccc7s5)c6C)nc4C(=O)O)c(F)c3)CC2)C(C)(C)C)cc1	C67H79FN12O8S3	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-ADYYWI	SCHEMBL26917688	2-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-5-[3-[2-fluoro-4-[3-[4-[2-[1-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethyl]cyclopentyl]acetyl]piperazin-1-yl]prop-1-ynyl]phenoxy]propyl]-1,3-thiazole-4-carboxylic acid; SCHEMBL30670841	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CC2(CC(=O)N3CCN(CC#Cc4ccc(OCCCc5sc(N6CCCc7c6nnc(Nc6nc8ccccc8s6)c7C)nc5C(=O)O)c(F)c4)CC3)CCCC2)C(C)(C)C)cc1	C67H77FN12O8S3	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-JRYKS0	SCHEMBL26917776	2-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-5-[3-[2-fluoro-4-[3-[4-[2-[2-[2-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]ethoxy]ethoxy]acetyl]piperazin-1-yl]prop-1-ynyl]phenoxy]propyl]-1,3-thiazole-4-carboxylic acid; SCHEMBL26917788	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCC(=O)N2CCN(CC#Cc3ccc(OCCCc4sc(N5CCCc6c5nnc(Nc5nc7ccccc7s5)c6C)nc4C(=O)O)c(F)c3)CC2)C(C)(C)C)cc1	C65H75FN12O11S3	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-5AFP0C	SCHEMBL26917510	2-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-5-[3-[2-fluoro-4-[3-[4-[6-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]carbamoyl]spiro[3.3]heptane-2-carbonyl]piperazin-1-yl]prop-1-ynyl]phenoxy]propyl]-1,3-thiazole-4-carboxylic acid; SCHEMBL30670904	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CC3(C2)CC(C(=O)N2CCN(CC#Cc4ccc(OCCCc5sc(N6CCCc7c6nnc(Nc6nc8ccccc8s6)c7C)nc5C(=O)O)c(F)c4)CC2)C3)C(C)(C)C)cc1	C67H75FN12O8S3	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-OIE71Q	WO2022169780A1_42	2-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-5-[3-[2-fluoro-4-[3-[4-[2-[3-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethyl]-1-adamantyl]acetyl]piperazin-1-yl]prop-1-ynyl]phenoxy]propyl]-1,3-thiazole-4-carboxylic acid	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CC23CC4CC(C2)CC(CC(=O)N2CCN(CC#Cc5ccc(OCCCc6sc(N7CCCc8c7nnc(Nc7nc9ccccc9s7)c8C)nc6C(=O)O)c(F)c5)CC2)(C4)C3)C(C)(C)C)cc1	C72H83FN12O8S3	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-MV0HGN	SCHEMBL26917730	2-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-5-[3-[2-fluoro-4-[3-[4-[3-fluoro-4-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]carbamoyl]benzoyl]piperazin-1-yl]prop-1-ynyl]phenoxy]propyl]-1,3-thiazole-4-carboxylic acid; SCHEMBL30670902	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)c2ccc(C(=O)N3CCN(CC#Cc4ccc(OCCCc5sc(N6CCCc7c6nnc(Nc6nc8ccccc8s6)c7C)nc5C(=O)O)c(F)c4)CC3)cc2F)C(C)(C)C)cc1	C66H68F2N12O8S3	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-8T3M6G	SCHEMBL26917411	2-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-5-[3-[2-fluoro-4-[3-[4-[5-[[2-[2-[[[(2S,4R)-1-[(2S)-2-[(1-fluorocyclopropanecarbonyl)amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carbonyl]amino]methyl]-5-(4-methyl-1,3-thiazol-5-yl)phenoxy]acetyl]amino]pentanoyl]piperazin-1-yl]prop-1-ynyl]phenoxy]propyl]-1,3-thiazole-4-carboxylic acid; SCHEMBL26917417; SCHEMBL30670784	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)C)c(OCC(=O)NCCCCC(=O)N2CCN(CC#Cc3ccc(OCCCc4sc(N5CCCc6c5nnc(Nc5nc7ccccc7s5)c6C)nc4C(=O)O)c(F)c3)CC2)c1	C68H77F2N13O10S3	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-NI2G1F	SCHEMBL26917563	2-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-5-[3-[2-fluoro-4-[3-[4-[12-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[2-hydroxy-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-12-oxododecanoyl]piperazin-1-yl]prop-1-ynyl]phenoxy]propyl]-1,3-thiazole-4-carboxylic acid; SCHEMBL26917574	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCCCCCC(=O)N2CCN(CC#Cc3ccc(OCCCc4sc(N5CCCc6c5nnc(Nc5nc7ccccc7s5)c6C)nc4C(=O)O)c(F)c3)CC2)C(C)(C)C)c(O)c1	C69H83FN12O9S3	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-BIREK2	SCHEMBL26918185	2-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-5-[3-[2-fluoro-4-[3-[4-[12-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-12-oxododecanoyl]piperazin-1-yl]prop-1-ynyl]phenoxy]propyl]-1,3-thiazole-4-carboxylic acid; SCHEMBL26918202	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCCCCCC(=O)N2CCN(CC#Cc3ccc(OCCCc4sc(N5CCCc6c5nnc(Nc5nc7ccccc7s5)c6C)nc4C(=O)O)c(F)c3)CC2)C(C)(C)C)cc1	C70H85FN12O8S3	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-98XV6X	WO2022169780A1_47	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[4-[12-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-12-oxododecanoyl]piperazin-1-yl]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCCCCCC(=O)N2CCN(CCOC34CC5(C)CC(C)(CC(Cn6ncc(-c7ccc(N8CCCc9c8nnc(Nc8nc%10ccccc%10s8)c9C)nc7C(=O)O)c6C)(C5)C3)C4)CC2)C(C)(C)C)cc1	C79H104N14O8S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-C6BOOY	SCHEMBL26918098	2-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-5-[3-[2-fluoro-4-[3-[4-[12-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-12-oxododecanoyl]piperazin-1-yl]prop-1-ynyl]phenoxy]propyl]-1,3-thiazole-4-carboxylic acid; SCHEMBL26918108	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCCCCCC(=O)N2CCN(CC#Cc3ccc(OCCCc4sc(N5CCCc6c5nnc(Nc5nc7ccccc7s5)c6C)nc4C(=O)O)c(F)c3)CC2)C(C)(C)C)cc1	C69H83FN12O8S3	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-XQB5GY	WO2022169780A1_49	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[4-[4-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-4-oxobutanoyl]piperazin-1-yl]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCC(=O)N2CCN(CCOC34CC5(C)CC(C)(CC(Cn6ncc(-c7ccc(N8CCCc9c8nnc(Nc8nc%10ccccc%10s8)c9C)nc7C(=O)O)c6C)(C5)C3)C4)CC2)C(C)(C)C)cc1	C71H88N14O8S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-VWJZQW	WO2022169780A1_50	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[4-[2-[2-[[[(2S,4R)-1-[(2S)-2-[(1-fluorocyclopropanecarbonyl)amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carbonyl]amino]methyl]-5-(4-methyl-1,3-thiazol-5-yl)phenoxy]acetyl]piperazin-1-yl]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)C)c(OCC(=O)N2CCN(CCOC34CC5(C)CC(C)(CC(Cn6ncc(-c7ccc(N8CCCc9c8nnc(Nc8nc%10ccccc%10s8)c9C)nc7C(=O)O)c6C)(C5)C3)C4)CC2)c1	C72H87FN14O9S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-QQ3ZHL	SCHEMBL26917391	2-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-5-[3-[2-fluoro-4-[3-[4-[12-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-12-oxododecyl]piperazin-1-yl]prop-1-ynyl]phenoxy]propyl]-1,3-thiazole-4-carboxylic acid; SCHEMBL26917407	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCCCCCCN2CCN(CC#Cc3ccc(OCCCc4sc(N5CCCc6c5nnc(Nc5nc7ccccc7s5)c6C)nc4C(=O)O)c(F)c3)CC2)C(C)(C)C)cc1	C70H87FN12O7S3	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-HMB3B7	SCHEMBL26918043	2-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-5-[3-[2-fluoro-4-[3-[4-[5-[[2-[2-[[[(2S,4R)-1-[(2S)-2-[(1-fluorocyclopropanecarbonyl)amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carbonyl]amino]methyl]-5-(4-methyl-1,3-thiazol-5-yl)phenoxy]acetyl]amino]pentyl]piperazin-1-yl]prop-1-ynyl]phenoxy]propyl]-1,3-thiazole-4-carboxylic acid; SCHEMBL26918059; SCHEMBL30670864	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)C)c(OCC(=O)NCCCCCN2CCN(CC#Cc3ccc(OCCCc4sc(N5CCCc6c5nnc(Nc5nc7ccccc7s5)c6C)nc4C(=O)O)c(F)c3)CC2)c1	C68H79F2N13O9S3	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-FRT1DY	SCHEMBL26917960	2-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-5-[3-[2-fluoro-4-[3-[4-[5-[[2-[2-[[[(2S,4R)-1-[(2S)-2-[(1-fluorocyclopropanecarbonyl)amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carbonyl]amino]methyl]-5-(4-methyl-1,3-thiazol-5-yl)phenoxy]acetyl]-methylamino]pentyl]piperazin-1-yl]prop-1-ynyl]phenoxy]propyl]-1,3-thiazole-4-carboxylic acid; SCHEMBL26917971; SCHEMBL30670878	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)C)c(OCC(=O)N(C)CCCCCN2CCN(CC#Cc3ccc(OCCCc4sc(N5CCCc6c5nnc(Nc5nc7ccccc7s5)c6C)nc4C(=O)O)c(F)c3)CC2)c1	C69H81F2N13O9S3	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-1OY5ZJ	WO2022169780A1_55	2-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-5-[3-[2-fluoro-4-[3-[4-[13-[2-[[[(2S,4R)-1-[(2S)-2-[(1-fluorocyclopropanecarbonyl)amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carbonyl]amino]methyl]-5-(4-methyl-1,3-thiazol-5-yl)phenoxy]tridecyl]piperazin-1-yl]prop-1-ynyl]phenoxy]propyl]-1,3-thiazole-4-carboxylic acid	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)C)c(OCCCCCCCCCCCCCN2CCN(CC#Cc3ccc(OCCCc4sc(N5CCCc6c5nnc(Nc5nc7ccccc7s5)c6C)nc4C(=O)O)c(F)c3)CC2)c1	C74H92F2N12O8S3	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-D19600	SCHEMBL26917592	2-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-5-[3-[2-fluoro-4-[3-[4-[8-[2-[[[(2S,4R)-1-[(2S)-2-[(1-fluorocyclopropanecarbonyl)amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carbonyl]amino]methyl]-5-(4-methyl-1,3-thiazol-5-yl)phenoxy]octyl]piperazin-1-yl]prop-1-ynyl]phenoxy]propyl]-1,3-thiazole-4-carboxylic acid; SCHEMBL26917607; SCHEMBL30670859	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)C)c(OCCCCCCCCN2CCN(CC#Cc3ccc(OCCCc4sc(N5CCCc6c5nnc(Nc5nc7ccccc7s5)c6C)nc4C(=O)O)c(F)c3)CC2)c1	C69H82F2N12O8S3	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-PZLASM	WO2022169780A1_57	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)C)c(OCCCCCCCCCCN2CCN(CC#Cc3ccc(OCCCc4sc(N5CCCc6c5nnc(Nc5nc7ccccc7s5)c6C)nc4C(=O)O)c(F)c3)CC2)c1	C71H86F2N12O8S3	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-RMGUJP	SCHEMBL26917566	2-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-5-[3-[2-fluoro-4-[3-[4-[[4-[[2-[[[(2S,4R)-1-[(2S)-2-[(1-fluorocyclopropanecarbonyl)amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carbonyl]amino]methyl]-5-(4-methyl-1,3-thiazol-5-yl)phenoxy]methyl]phenyl]methyl]piperazin-1-yl]prop-1-ynyl]phenoxy]propyl]-1,3-thiazole-4-carboxylic acid; SCHEMBL26917575; SCHEMBL30670922	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)C)c(OCc2ccc(CN3CCN(CC#Cc4ccc(OCCCc5sc(N6CCCc7c6nnc(Nc6nc8ccccc8s6)c7C)nc5C(=O)O)c(F)c4)CC3)cc2)c1	C69H74F2N12O8S3	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-MAVGA3	SCHEMBL26917545	2-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-5-[3-[2-fluoro-4-[3-[4-[2-[2-[2-[[[(2S,4R)-1-[(2S)-2-[(1-fluorocyclopropanecarbonyl)amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carbonyl]amino]methyl]-5-(4-methyl-1,3-thiazol-5-yl)phenoxy]ethyl-methylamino]acetyl]piperazin-1-yl]prop-1-ynyl]phenoxy]propyl]-1,3-thiazole-4-carboxylic acid; SCHEMBL26917551; SCHEMBL30670781	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)C)c(OCCN(C)CC(=O)N2CCN(CC#Cc3ccc(OCCCc4sc(N5CCCc6c5nnc(Nc5nc7ccccc7s5)c6C)nc4C(=O)O)c(F)c3)CC2)c1	C66H75F2N13O9S3	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-YVR69D	SCHEMBL26918028	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[10-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxydecyl-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL30670871	Cc1c(Nc2nc3ccccc3s2)nnc2c1CCCN2c1ccc(-c2cnn(CC34CC5(C)CC(C)(C3)CC(OCCN(C)CCCCCCCCCCOc3ccc6c(c3)C(=O)N(C3CCC(=O)NC3=O)C6=O)(C5)C4)c2C)c(C(=O)O)n1	C64H77N11O8S	BCL2L1	Q07817	CRBN	WO-2022169780-A1
TPD-194EVB	SCHEMBL26917997	6-[[6-(1,3-Benzothiazol-2-ylamino)-5-methylpyridazin-3-yl]-[5-[4-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxymethyl]triazol-1-yl]pentyl]amino]-3-[1-[[3-[2-(dimethylamino)ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL30670788	Cc1cc(N(CCCCCn2cc(COCCOCCNc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)nn2)c2ccc(-c3cnn(CC45CC6(C)CC(C)(C4)CC(OCCN(C)C)(C6)C5)c3C)c(C(=O)O)n2)nnc1Nc1nc2ccccc2s1	C64H77N15O9S	BCL2L1	Q07817	CRBN	WO-2022169780-A1
TPD-FRHUBF	WO2022169780A1_62	.	Cc1cc(N(CCCCCn2cc(COCCOCCNc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)nn2)c2ccc(-c3cnn(CC45C[C@@]6(C)C[C@@](C)(C4)C[C@](OCCN(C)C)(C5)C6)c3C)c(C(=O)O)n2)nnc1Nc1nc2ccccc2s1	C64H77N15O9S	BCL2L1	Q07817	CRBN	WO-2022169780-A1
TPD-48U3EG	SCHEMBL26918186	6-[[6-(1,3-Benzothiazol-2-ylamino)-5-methylpyridazin-3-yl]-[5-[4-[2-[2-[2-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyacetyl]amino]ethoxy]ethoxy]ethoxymethyl]triazol-1-yl]pentyl]amino]-3-[1-[[3-[2-(dimethylamino)ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL30670819	Cc1cc(N(CCCCCn2cc(COCCOCCOCCNC(=O)COc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)nn2)c2ccc(-c3cnn(CC45CC6(C)CC(C)(C4)CC(OCCN(C)C)(C6)C5)c3C)c(C(=O)O)n2)nnc1Nc1nc2ccccc2s1	C68H83N15O12S	BCL2L1	Q07817	CRBN	WO-2022169780-A1
TPD-0OSIS3	SCHEMBL26917754	6-[[6-(1,3-Benzothiazol-2-ylamino)-5-methylpyridazin-3-yl]-[5-[4-[7-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyacetyl]amino]heptyl]triazol-1-yl]pentyl]amino]-3-[1-[[3-[2-(dimethylamino)ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL30670792	Cc1cc(N(CCCCCn2cc(CCCCCCCNC(=O)COc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)nn2)c2ccc(-c3cnn(CC45CC6(C)CC(C)(C4)CC(OCCN(C)C)(C6)C5)c3C)c(C(=O)O)n2)nnc1Nc1nc2ccccc2s1	C68H83N15O9S	BCL2L1	Q07817	CRBN	WO-2022169780-A1
TPD-VCHYJX	SCHEMBL26917568	6-[[6-(1,3-Benzothiazol-2-ylamino)-5-methylpyridazin-3-yl]-[5-[4-[2-[2-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyacetyl]amino]ethoxy]ethoxymethyl]triazol-1-yl]pentyl]amino]-3-[1-[[3-[2-(dimethylamino)ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL30670929	Cc1cc(N(CCCCCn2cc(COCCOCCNC(=O)COc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)nn2)c2ccc(-c3cnn(CC45CC6(C)CC(C)(C4)CC(OCCN(C)C)(C6)C5)c3C)c(C(=O)O)n2)nnc1Nc1nc2ccccc2s1	C66H79N15O11S	BCL2L1	Q07817	CRBN	WO-2022169780-A1
TPD-F9YXGZ	WO2022169780A1_66	2-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-5-[3-[[5-[[(2S)-1-[(2S,4S)-4-hydroxy-2-[[(1R)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-5-oxopentyl]-methylamino]propyl]-1,3-thiazole-4-carboxylic acid	Cc1ncsc1-c1ccc([C@@H](C)NC(=O)[C@@H]2C[C@H](O)CN2C(=O)[C@@H](NC(=O)CCCCN(C)CCCc2sc(N3CCCc4c3nnc(Nc3nc5ccccc5s3)c4C)nc2C(=O)O)C(C)(C)C)cc1	C51H63N11O6S3	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-D5U24J	SCHEMBL26917745	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[[6-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]-6-oxohexyl]-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL30670885	Cc1c(Nc2nc3ccccc3s2)nnc2c1CCCN2c1ccc(-c2cnn(CC34CC5(C)CC(C)(C3)CC(OCCN(C)CCCCCC(=O)N3CCC(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC3)(C5)C4)c2C)c(C(=O)O)n1	C65H78N12O7S	BCL2L1	Q07817	CRBN	WO-2022169780-A1
TPD-0P2CNP	SCHEMBL26917713	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[[8-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]-8-oxooctyl]-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL30670838	Cc1c(Nc2nc3ccccc3s2)nnc2c1CCCN2c1ccc(-c2cnn(CC34CC5(C)CC(C)(C3)CC(OCCN(C)CCCCCCCC(=O)N3CCC(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC3)(C5)C4)c2C)c(C(=O)O)n1	C67H82N12O7S	BCL2L1	Q07817	CRBN	WO-2022169780-A1
TPD-9S05V0	SCHEMBL26917794	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[[12-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]-12-oxododecyl]-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL30670865	Cc1c(Nc2nc3ccccc3s2)nnc2c1CCCN2c1ccc(-c2cnn(CC34CC5(C)CC(C)(C3)CC(OCCN(C)CCCCCCCCCCCC(=O)N3CCC(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC3)(C5)C4)c2C)c(C(=O)O)n1	C71H90N12O7S	BCL2L1	Q07817	CRBN	WO-2022169780-A1
TPD-HACZHU	SCHEMBL26917383	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[[10-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]-10-oxodecyl]-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL30670810	Cc1c(Nc2nc3ccccc3s2)nnc2c1CCCN2c1ccc(-c2cnn(CC34CC5(C)CC(C)(C3)CC(OCCN(C)CCCCCCCCCC(=O)N3CCC(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC3)(C5)C4)c2C)c(C(=O)O)n1	C69H86N12O7S	BCL2L1	Q07817	CRBN	WO-2022169780-A1
TPD-HBCJT7	SCHEMBL26917994	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[[9-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]-9-oxononyl]-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL30670857	Cc1c(Nc2nc3ccccc3s2)nnc2c1CCCN2c1ccc(-c2cnn(CC34CC5(C)CC(C)(C3)CC(OCCN(C)CCCCCCCCC(=O)N3CCC(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC3)(C5)C4)c2C)c(C(=O)O)n1	C68H84N12O7S	BCL2L1	Q07817	CRBN	WO-2022169780-A1
TPD-PSP6UA	SCHEMBL26917673	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[9-[2-[[[(2S,4R)-1-[(2S)-2-[(1-fluorocyclopropanecarbonyl)amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carbonyl]amino]methyl]-5-(4-methyl-1,3-thiazol-5-yl)phenoxy]nonyl-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL26917686; SCHEMBL30670932	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)C)c(OCCCCCCCCCN(C)CCOC23CC4(C)CC(C)(CC(Cn5ncc(-c6ccc(N7CCCc8c7nnc(Nc7nc9ccccc9s7)c8C)nc6C(=O)O)c5C)(C4)C2)C3)c1	C76H98FN13O8S2	BCL2L1	Q07817	CRBN	WO-2022169780-A1
TPD-RL2H35	SCHEMBL26917468	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[10-[2-[[[(2S,4R)-1-[(2S)-2-[(1-fluorocyclopropanecarbonyl)amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carbonyl]amino]methyl]-5-(4-methyl-1,3-thiazol-5-yl)phenoxy]decyl-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL26917481; SCHEMBL30670959	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)C)c(OCCCCCCCCCCN(C)CCOC23CC4(C)CC(C)(CC(Cn5ncc(-c6ccc(N7CCCc8c7nnc(Nc7nc9ccccc9s7)c8C)nc6C(=O)O)c5C)(C4)C2)C3)c1	C77H100FN13O8S2	BCL2L1	Q07817	CRBN	WO-2022169780-A1
TPD-9MM3V3	SCHEMBL26917556	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[[16-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]-16-oxohexadecyl]-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL30670870	Cc1c(Nc2nc3ccccc3s2)nnc2c1CCCN2c1ccc(-c2cnn(CC34CC5(C)CC(C)(C3)CC(OCCN(C)CCCCCCCCCCCCCCCC(=O)N3CCC(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC3)(C5)C4)c2C)c(C(=O)O)n1	C75H98N12O7S	BCL2L1	Q07817	CRBN	WO-2022169780-A1
TPD-8MZGED	SCHEMBL26918094	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[[11-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]-11-oxoundecyl]-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL30670958	Cc1c(Nc2nc3ccccc3s2)nnc2c1CCCN2c1ccc(-c2cnn(CC34CC5(C)CC(C)(C3)CC(OCCN(C)CCCCCCCCCCC(=O)N3CCC(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC3)(C5)C4)c2C)c(C(=O)O)n1	C70H88N12O7S	BCL2L1	Q07817	CRBN	WO-2022169780-A1
TPD-0CGC8K	SCHEMBL26918236	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[11-[2-[[[(2S,4R)-1-[(2S)-2-[(1-fluorocyclopropanecarbonyl)amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carbonyl]amino]methyl]-5-(4-methyl-1,3-thiazol-5-yl)phenoxy]undecyl-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL26918256; SCHEMBL30670950	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)C)c(OCCCCCCCCCCCN(C)CCOC23CC4(C)CC(C)(CC(Cn5ncc(-c6ccc(N7CCCc8c7nnc(Nc7nc9ccccc9s7)c8C)nc6C(=O)O)c5C)(C4)C2)C3)c1	C78H102FN13O8S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-0EU6PY	SCHEMBL26917905	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[16-[2-[[[(2S,4R)-1-[(2S)-2-[(1-fluorocyclopropanecarbonyl)amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carbonyl]amino]methyl]-5-(4-methyl-1,3-thiazol-5-yl)phenoxy]hexadecyl-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL26917916; SCHEMBL30670836	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)C)c(OCCCCCCCCCCCCCCCCN(C)CCOC23CC4(C)CC(C)(CC(Cn5ncc(-c6ccc(N7CCCc8c7nnc(Nc7nc9ccccc9s7)c8C)nc6C(=O)O)c5C)(C4)C2)C3)c1	C83H112FN13O8S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-9TWBZJ	SCHEMBL26917832	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[[13-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]-13-oxotridecyl]-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL30670880	Cc1c(Nc2nc3ccccc3s2)nnc2c1CCCN2c1ccc(-c2cnn(CC34CC5(C)CC(C)(C3)CC(OCCN(C)CCCCCCCCCCCCC(=O)N3CCC(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC3)(C5)C4)c2C)c(C(=O)O)n1	C72H92N12O7S	BCL2L1	Q07817	CRBN	WO-2022169780-A1
TPD-PPJWGG	SCHEMBL26918855	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[12-[(3R)-3-[(1-fluorocyclopropanecarbonyl)amino]-4-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-2-methyl-4-oxobutan-2-yl]sulfanyldodecyl-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL26918878	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)SCCCCCCCCCCCCN(C)CCOC23CC4(C)CC(C)(CC(Cn5ncc(-c6ccc(N7CCCc8c7nnc(Nc7nc9ccccc9s7)c8C)nc6C(=O)O)c5C)(C4)C2)C3)cc1	C78H102FN13O7S3	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-0TN5HA	SCHEMBL26917930	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[14-[(3R)-3-[(1-fluorocyclopropanecarbonyl)amino]-4-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-2-methyl-4-oxobutan-2-yl]sulfanyltetradecyl-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL26917943	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)SCCCCCCCCCCCCCCN(C)CCOC23CC4(C)CC(C)(CC(Cn5ncc(-c6ccc(N7CCCc8c7nnc(Nc7nc9ccccc9s7)c8C)nc6C(=O)O)c5C)(C4)C2)C3)cc1	C80H106FN13O7S3	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-GU4QGB	SCHEMBL26917617	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[[8-[4-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]carbamoyl]piperidin-1-yl]-8-oxooctyl]-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL26917633	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCN(C(=O)CCCCCCCN(C)CCOC34CC5(C)CC(C)(CC(Cn6ncc(-c7ccc(N8CCCc9c8nnc(Nc8nc%10ccccc%10s8)c9C)nc7C(=O)O)c6C)(C5)C3)C4)CC2)C(C)(C)C)cc1	C78H102N14O8S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-B6PPX8	SCHEMBL26917389	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[[11-[4-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]carbamoyl]piperidin-1-yl]-11-oxoundecyl]-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL26917405	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCN(C(=O)CCCCCCCCCCN(C)CCOC34CC5(C)CC(C)(CC(Cn6ncc(-c7ccc(N8CCCc9c8nnc(Nc8nc%10ccccc%10s8)c9C)nc7C(=O)O)c6C)(C5)C3)C4)CC2)C(C)(C)C)cc1	C81H108N14O8S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-M76GNX	SCHEMBL26917596	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[15-[2-[[[(2S,4R)-1-[(2S)-2-[(1-fluorocyclopropanecarbonyl)amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carbonyl]amino]methyl]-5-(4-methyl-1,3-thiazol-5-yl)phenoxy]pentadecyl-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL26917610; SCHEMBL30670821	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)C)c(OCCCCCCCCCCCCCCCN(C)CCOC23CC4(C)CC(C)(CC(Cn5ncc(-c6ccc(N7CCCc8c7nnc(Nc7nc9ccccc9s7)c8C)nc6C(=O)O)c5C)(C4)C2)C3)c1	C82H110FN13O8S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-ABJ33Z	SCHEMBL26918076	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[[10-[4-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]carbamoyl]piperidin-1-yl]-10-oxodecyl]-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL26918096	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCN(C(=O)CCCCCCCCCN(C)CCOC34CC5(C)CC(C)(CC(Cn6ncc(-c7ccc(N8CCCc9c8nnc(Nc8nc%10ccccc%10s8)c9C)nc7C(=O)O)c6C)(C5)C3)C4)CC2)C(C)(C)C)cc1	C80H106N14O8S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-0W5T9H	SCHEMBL26917977	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[13-[2-[[[(2S,4R)-1-[(2S)-2-[(1-fluorocyclopropanecarbonyl)amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carbonyl]amino]methyl]-5-(4-methyl-1,3-thiazol-5-yl)phenoxy]tridecyl-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL26917986; SCHEMBL30670954	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)C)c(OCCCCCCCCCCCCCN(C)CCOC23CC4(C)CC(C)(CC(Cn5ncc(-c6ccc(N7CCCc8c7nnc(Nc7nc9ccccc9s7)c8C)nc6C(=O)O)c5C)(C4)C2)C3)c1	C80H106FN13O8S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-EVK1IA	SCHEMBL26917539	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[[12-[4-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]carbamoyl]piperidin-1-yl]-12-oxododecyl]-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL26917549	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCN(C(=O)CCCCCCCCCCCN(C)CCOC34CC5(C)CC(C)(CC(Cn6ncc(-c7ccc(N8CCCc9c8nnc(Nc8nc%10ccccc%10s8)c9C)nc7C(=O)O)c6C)(C5)C3)C4)CC2)C(C)(C)C)cc1	C82H110N14O8S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-RQST5R	WO2022169780A1_87	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@H]2C[C@@H](O)CN2C(=O)C(C)(NC(=O)COCCOCCOCCOCCN(C)CCOC23CC4(C)CC(C)(CC(Cn5ncc(-c6ccc(N7CCCc8c7nnc(Nc7nc9ccccc9s7)c8C)nc6C(=O)O)c5C)(C4)C2)C3)C(C)(C)C)cc1	C75H99N13O11S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-TLUMDB	WO2022169780A1_88	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@H]2C[C@@H](O)CN2C(=O)C(NC(=O)CCOCCOCCOCCN(C)CCOC23CC4(C)CC(C)(CC(Cn5ncc(-c6ccc(N7CCCc8c7nnc(Nc7nc9ccccc9s7)c8C)nc6C(=O)O)c5C)(C4)C2)C3)C(C)(C)C)cc1	C73H95N13O10S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-DSYX3J	SCHEMBL26918659	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[2-[2-[2-[2-[3-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-3-oxopropoxy]ethoxy]ethoxy]ethoxy]ethyl-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL26918681	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCOCCOCCOCCOCCN(C)CCOC23CC4(C)CC(C)(CC(Cn5ncc(-c6ccc(N7CCCc8c7nnc(Nc7nc9ccccc9s7)c8C)nc6C(=O)O)c5C)(C4)C2)C3)C(C)(C)C)cc1	C75H99N13O11S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-JZ61SX	SCHEMBL26918055	6-[[6-(1,3-Benzothiazol-2-ylamino)-5-methylpyridazin-3-yl]-[4-[11-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]undecanoyl-methylamino]butyl]amino]-3-[1-[[3-[2-(dimethylamino)ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL30670782	Cc1cc(N(CCCCN(C)C(=O)CCCCCCCCCCNc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)c2ccc(-c3cnn(CC45CC6(C)CC(C)(C4)CC(OCCN(C)C)(C6)C5)c3C)c(C(=O)O)n2)nnc1Nc1nc2ccccc2s1	C68H87N13O8S	BCL2L1	Q07817	CRBN	WO-2022169780-A1
TPD-XJAJX9	SCHEMBL26917518	6-[[6-(1,3-Benzothiazol-2-ylamino)-5-methylpyridazin-3-yl]-[4-[9-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]nonanoyl-methylamino]butyl]amino]-3-[1-[[3-[2-(dimethylamino)ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL30670896	Cc1cc(N(CCCCN(C)C(=O)CCCCCCCCNc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)c2ccc(-c3cnn(CC45CC6(C)CC(C)(C4)CC(OCCN(C)C)(C6)C5)c3C)c(C(=O)O)n2)nnc1Nc1nc2ccccc2s1	C66H83N13O8S	BCL2L1	Q07817	CRBN	WO-2022169780-A1
TPD-2GD2V1	WO2022169780A1_92	.	Cc1cc(N(CCCCN(C)C(=O)CCCCCCCCCNc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)c2ccc(-c3cnn(CC45CC6(C)CC(C)(C4)CC(OCCN(C)C)(C6)C5)c3)c(C(=O)O)n2)nnc1Nc1nc2ccccc2s1	C66H83N13O8S	BCL2L1	Q07817	CRBN	WO-2022169780-A1
TPD-1XB3XW	SCHEMBL26917630	6-[[6-(1,3-Benzothiazol-2-ylamino)-5-methylpyridazin-3-yl]-[4-[12-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]dodecanoyl-methylamino]butyl]amino]-3-[1-[[3-[2-(dimethylamino)ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL30670787	Cc1cc(N(CCCCN(C)C(=O)CCCCCCCCCCCNc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)c2ccc(-c3cnn(CC45CC6(C)CC(C)(C4)CC(OCCN(C)C)(C6)C5)c3C)c(C(=O)O)n2)nnc1Nc1nc2ccccc2s1	C69H89N13O8S	BCL2L1	Q07817	CRBN	WO-2022169780-A1
TPD-PZRY7E	SCHEMBL26917967	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[10-[(3R)-3-[(1-fluorocyclopropanecarbonyl)amino]-4-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-2-methyl-4-oxobutan-2-yl]sulfanyldecyl-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL26917980	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)SCCCCCCCCCCN(C)CCOC23CC4(C)CC(C)(CC(Cn5ncc(-c6ccc(N7CCCc8c7nnc(Nc7nc9ccccc9s7)c8C)nc6C(=O)O)c5C)(C4)C2)C3)cc1	C76H98FN13O7S3	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-L1ESQH	SCHEMBL26917714	6-[[6-(1,3-Benzothiazol-2-ylamino)-5-methylpyridazin-3-yl]-[4-[10-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxydecanoyl-methylamino]butyl]amino]-3-[1-[[3-[2-(dimethylamino)ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL30670817	Cc1cc(N(CCCCN(C)C(=O)CCCCCCCCCOc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)c2ccc(-c3cnn(CC45CC6(C)CC(C)(C4)CC(OCCN(C)C)(C6)C5)c3C)c(C(=O)O)n2)nnc1Nc1nc2ccccc2s1	C67H84N12O9S	BCL2L1	Q07817	CRBN	WO-2022169780-A1
TPD-B0ROAG	SCHEMBL26917822	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[12-[3-[2-[(2S)-1-[(2S)-2-cyclohexyl-2-[[(2S)-2-(methylamino)propanoyl]amino]acetyl]pyrrolidin-2-yl]-1,3-thiazole-4-carbonyl]phenoxy]dodecyl-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL26917838	CN[C@@H](C)C(=O)N[C@H](C(=O)N1CCC[C@H]1c1nc(C(=O)c2cccc(OCCCCCCCCCCCCN(C)CCOC34CC5(C)CC(C)(CC(Cn6ncc(-c7ccc(N8CCCc9c8nnc(Nc8nc%10ccccc%10s8)c9C)nc7C(=O)O)c6C)(C5)C3)C4)c2)cs1)C1CCCCC1	C79H105N13O7S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-56HPIM	SCHEMBL26917793	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[8-[3-[2-[(2S)-1-[(2S)-2-cyclohexyl-2-[[(2S)-2-(methylamino)propanoyl]amino]acetyl]pyrrolidin-2-yl]-1,3-thiazole-4-carbonyl]phenoxy]octyl-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL26917803	CN[C@@H](C)C(=O)N[C@H](C(=O)N1CCC[C@H]1c1nc(C(=O)c2cccc(OCCCCCCCCN(C)CCOC34CC5(C)CC(C)(CC(Cn6ncc(-c7ccc(N8CCCc9c8nnc(Nc8nc%10ccccc%10s8)c9C)nc7C(=O)O)c6C)(C5)C3)C4)c2)cs1)C1CCCCC1	C75H97N13O7S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-GSJ3SV	SCHEMBL26917625	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[10-[3-[2-[(2S)-1-[(2S)-2-cyclohexyl-2-[[(2S)-2-(methylamino)propanoyl]amino]acetyl]pyrrolidin-2-yl]-1,3-thiazole-4-carbonyl]phenoxy]decyl-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL26917634	CN[C@@H](C)C(=O)N[C@H](C(=O)N1CCC[C@H]1c1nc(C(=O)c2cccc(OCCCCCCCCCCN(C)CCOC34CC5(C)CC(C)(CC(Cn6ncc(-c7ccc(N8CCCc9c8nnc(Nc8nc%10ccccc%10s8)c9C)nc7C(=O)O)c6C)(C5)C3)C4)c2)cs1)C1CCCCC1	C77H101N13O7S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-GSNSQ2	SCHEMBL26917533	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[4-[3-[2-[(2S)-1-[(2S)-2-cyclohexyl-2-[[(2S)-2-(methylamino)propanoyl]amino]acetyl]pyrrolidin-2-yl]-1,3-thiazole-4-carbonyl]phenoxy]butyl-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL30670840	CN[C@@H](C)C(=O)N[C@H](C(=O)N1CCC[C@H]1c1nc(C(=O)c2cccc(OCCCCN(C)CCOC34CC5(C)CC(C)(CC(Cn6ncc(-c7ccc(N8CCCc9c8nnc(Nc8nc%10ccccc%10s8)c9C)nc7C(=O)O)c6C)(C5)C3)C4)c2)cs1)C1CCCCC1	C71H89N13O7S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-S1L5SG	SCHEMBL26917947	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[14-[3-[2-[(2S)-1-[(2S)-2-cyclohexyl-2-[[(2S)-2-(methylamino)propanoyl]amino]acetyl]pyrrolidin-2-yl]-1,3-thiazole-4-carbonyl]phenoxy]tetradecyl-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL26917957	CN[C@@H](C)C(=O)N[C@H](C(=O)N1CCC[C@H]1c1nc(C(=O)c2cccc(OCCCCCCCCCCCCCCN(C)CCOC34CC5(C)CC(C)(CC(Cn6ncc(-c7ccc(N8CCCc9c8nnc(Nc8nc%10ccccc%10s8)c9C)nc7C(=O)O)c6C)(C5)C3)C4)c2)cs1)C1CCCCC1	C81H109N13O7S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-CTGEQ2	SCHEMBL26917854	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[2-[3-[2-[(2S)-1-[(2S)-2-cyclohexyl-2-[[(2S)-2-(methylamino)propanoyl]amino]acetyl]pyrrolidin-2-yl]-1,3-thiazole-4-carbonyl]phenoxy]ethyl-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL30670917	CN[C@@H](C)C(=O)N[C@H](C(=O)N1CCC[C@H]1c1nc(C(=O)c2cccc(OCCN(C)CCOC34CC5(C)CC(C)(CC(Cn6ncc(-c7ccc(N8CCCc9c8nnc(Nc8nc%10ccccc%10s8)c9C)nc7C(=O)O)c6C)(C5)C3)C4)c2)cs1)C1CCCCC1	C69H85N13O7S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-L3DB83	SCHEMBL26917591	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[6-[3-[2-[(2S)-1-[(2S)-2-cyclohexyl-2-[[(2S)-2-(methylamino)propanoyl]amino]acetyl]pyrrolidin-2-yl]-1,3-thiazole-4-carbonyl]phenoxy]hexyl-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL26917601	CN[C@@H](C)C(=O)N[C@H](C(=O)N1CCC[C@H]1c1nc(C(=O)c2cccc(OCCCCCCN(C)CCOC34CC5(C)CC(C)(CC(Cn6ncc(-c7ccc(N8CCCc9c8nnc(Nc8nc%10ccccc%10s8)c9C)nc7C(=O)O)c6C)(C5)C3)C4)c2)cs1)C1CCCCC1	C73H93N13O7S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-NJLZE2	SCHEMBL26918144	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[2-[3-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-3-oxopropoxy]ethyl-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL30670951	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCOCCN(C)CCOC23CC4(C)CC(C)(CC(Cn5ncc(-c6ccc(N7CCCc8c7nnc(Nc7nc9ccccc9s7)c8C)nc6C(=O)O)c5C)(C4)C2)C3)C(C)(C)C)cc1	C69H87N13O8S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-LUYXO4	SCHEMBL26917453	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[9-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxynonyl-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL30670916	Cc1c(Nc2nc3ccccc3s2)nnc2c1CCCN2c1ccc(-c2cnn(CC34CC5(C)CC(C)(C3)CC(OCCN(C)CCCCCCCCCOc3ccc6c(c3)C(=O)N(C3CCC(=O)NC3=O)C6=O)(C5)C4)c2C)c(C(=O)O)n1	C63H75N11O8S	BCL2L1	Q07817	CRBN	WO-2022169780-A1
TPD-IBREF0	SCHEMBL26917659	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[11-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxyundecyl-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL30670900	Cc1c(Nc2nc3ccccc3s2)nnc2c1CCCN2c1ccc(-c2cnn(CC34CC5(C)CC(C)(C3)CC(OCCN(C)CCCCCCCCCCCOc3ccc6c(c3)C(=O)N(C3CCC(=O)NC3=O)C6=O)(C5)C4)c2C)c(C(=O)O)n1	C65H79N11O8S	BCL2L1	Q07817	CRBN	WO-2022169780-A1
TPD-KODQEU	SCHEMBL26917636	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[7-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxyheptyl-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL30670849	Cc1c(Nc2nc3ccccc3s2)nnc2c1CCCN2c1ccc(-c2cnn(CC34CC5(C)CC(C)(C3)CC(OCCN(C)CCCCCCCOc3ccc6c(c3)C(=O)N(C3CCC(=O)NC3=O)C6=O)(C5)C4)c2C)c(C(=O)O)n1	C61H71N11O8S	BCL2L1	Q07817	CRBN	WO-2022169780-A1
TPD-WVARXV	SCHEMBL26917755	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[5-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxypentyl-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL30670779	Cc1c(Nc2nc3ccccc3s2)nnc2c1CCCN2c1ccc(-c2cnn(CC34CC5(C)CC(C)(C3)CC(OCCN(C)CCCCCOc3ccc6c(c3)C(=O)N(C3CCC(=O)NC3=O)C6=O)(C5)C4)c2C)c(C(=O)O)n1	C59H67N11O8S	BCL2L1	Q07817	CRBN	WO-2022169780-A1
TPD-V5R6I9	SCHEMBL26918210	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[6-[3-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-3-oxopropoxy]hexyl-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL26918231	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCOCCCCCCN(C)CCOC23CC4(C)CC(C)(CC(Cn5ncc(-c6ccc(N7CCCc8c7nnc(Nc7nc9ccccc9s7)c8C)nc6C(=O)O)c5C)(C4)C2)C3)C(C)(C)C)cc1	C73H95N13O8S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-1R9SII	SCHEMBL26917695	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[9-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]nonyl-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL26917704	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCCCCCCCCN(C)CCOC23CC4(C)CC(C)(CC(Cn5ncc(-c6ccc(N7CCCc8c7nnc(Nc7nc9ccccc9s7)c8C)nc6C(=O)O)c5C)(C4)C2)C3)C(C)(C)C)cc1	C75H99N13O8S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-BCOMRT	SCHEMBL26917969	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[11-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]undecyl-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL26917982	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCCCCCCCCCCN(C)CCOC23CC4(C)CC(C)(CC(Cn5ncc(-c6ccc(N7CCCc8c7nnc(Nc7nc9ccccc9s7)c8C)nc6C(=O)O)c5C)(C4)C2)C3)C(C)(C)C)cc1	C77H103N13O8S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-0PMGM2	SCHEMBL26917437	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[13-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]tridecyl-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL26917447	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCCCCCCCCCCCCN(C)CCOC23CC4(C)CC(C)(CC(Cn5ncc(-c6ccc(N7CCCc8c7nnc(Nc7nc9ccccc9s7)c8C)nc6C(=O)O)c5C)(C4)C2)C3)C(C)(C)C)cc1	C79H107N13O8S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-41C1NC	SCHEMBL26917900	6-[[6-(1,3-benzothiazol-2-ylamino)-5-methylpyridazin-3-yl]-[4-[[12-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-12-oxododecanoyl]-methylamino]butyl]amino]-3-[1-[[3-[2-(dimethylamino)ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL26917914	Cc1cc(N(CCCCN(C)C(=O)CCCCCCCCCCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)c2ccc(-c3scnc3C)cc2)C(C)(C)C)c2ccc(-c3cnn(CC45CC6(C)CC(C)(C4)CC(OCCN(C)C)(C6)C5)c3C)c(C(=O)O)n2)nnc1Nc1nc2ccccc2s1	C79H108N14O8S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-FNC886	SCHEMBL26918000	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[2-[2-[2-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]ethoxy]ethoxy]ethyl-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL26918017	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCOCCOCCN(C)CCOC23CC4(C)CC(C)(CC(Cn5ncc(-c6ccc(N7CCCc8c7nnc(Nc7nc9ccccc9s7)c8C)nc6C(=O)O)c5C)(C4)C2)C3)C(C)(C)C)cc1	C72H93N13O10S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-7U5ANE	SCHEMBL26917961	6-[[6-(1,3-benzothiazol-2-ylamino)-5-methylpyridazin-3-yl]-[4-[[11-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-11-oxoundecanoyl]-methylamino]butyl]amino]-3-[1-[[3-[2-(dimethylamino)ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL26917973	Cc1cc(N(CCCCN(C)C(=O)CCCCCCCCCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)c2ccc(-c3scnc3C)cc2)C(C)(C)C)c2ccc(-c3cnn(CC45CC6(C)CC(C)(C4)CC(OCCN(C)C)(C6)C5)c3C)c(C(=O)O)n2)nnc1Nc1nc2ccccc2s1	C78H106N14O8S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-UJ2ARF	SCHEMBL26917771	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[13-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxytridecyl-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL30670943	Cc1c(Nc2nc3ccccc3s2)nnc2c1CCCN2c1ccc(-c2cnn(CC34CC5(C)CC(C)(C3)CC(OCCN(C)CCCCCCCCCCCCCOc3ccc6c(c3)C(=O)N(C3CCC(=O)NC3=O)C6=O)(C5)C4)c2C)c(C(=O)O)n1	C67H83N11O8S	BCL2L1	Q07817	CRBN	WO-2022169780-A1
TPD-WT9J3N	SCHEMBL26917537	6-[[6-(1,3-benzothiazol-2-ylamino)-5-methylpyridazin-3-yl]-[4-[[14-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-14-oxotetradecanoyl]-methylamino]butyl]amino]-3-[1-[[3-[2-(dimethylamino)ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL26917548	Cc1cc(N(CCCCN(C)C(=O)CCCCCCCCCCCCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)c2ccc(-c3scnc3C)cc2)C(C)(C)C)c2ccc(-c3cnn(CC45CC6(C)CC(C)(C4)CC(OCCN(C)C)(C6)C5)c3C)c(C(=O)O)n2)nnc1Nc1nc2ccccc2s1	C81H112N14O8S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-4WIWN8	SCHEMBL26917500	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[11-[(3R)-3-[(1-fluorocyclopropanecarbonyl)amino]-4-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-2-methyl-4-oxobutan-2-yl]sulfanylundecyl-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL26917514	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)SCCCCCCCCCCCN(C)CCOC23CC4(C)CC(C)(CC(Cn5ncc(-c6ccc(N7CCCc8c7nnc(Nc7nc9ccccc9s7)c8C)nc6C(=O)O)c5C)(C4)C2)C3)cc1	C77H100FN13O7S3	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-0IDNWT	SCHEMBL26918104	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[13-[(3R)-3-[(1-fluorocyclopropanecarbonyl)amino]-4-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-2-methyl-4-oxobutan-2-yl]sulfanyltridecyl-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL26918120	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)SCCCCCCCCCCCCCN(C)CCOC23CC4(C)CC(C)(CC(Cn5ncc(-c6ccc(N7CCCc8c7nnc(Nc7nc9ccccc9s7)c8C)nc6C(=O)O)c5C)(C4)C2)C3)cc1	C79H104FN13O7S3	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-EPGWED	SCHEMBL26917540	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[15-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxypentadecyl-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL30670893	Cc1c(Nc2nc3ccccc3s2)nnc2c1CCCN2c1ccc(-c2cnn(CC34CC5(C)CC(C)(C3)CC(OCCN(C)CCCCCCCCCCCCCCCOc3ccc6c(c3)C(=O)N(C3CCC(=O)NC3=O)C6=O)(C5)C4)c2C)c(C(=O)O)n1	C69H87N11O8S	BCL2L1	Q07817	CRBN	WO-2022169780-A1
TPD-C7BL6K	SCHEMBL26917669	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3,5-dimethyl-7-(2-pyrrolidin-1-ylethoxy)-1-adamantyl]methyl]-5-methylpyrazol-4-yl]-N-[7-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-7-oxoheptyl]pyridine-2-carboxamide; SCHEMBL26917684	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCNC(=O)c2nc(N3CCCc4c3nnc(Nc3nc5ccccc5s3)c4C)ccc2-c2cnn(CC34CC5(C)CC(C)(C3)CC(OCCN3CCCC3)(C5)C4)c2C)C(C)(C)C)cc1	C74H96N14O6S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-XTNTND	WO2022169780A1_121	.	Cc1cc(N(CCCCN(C)C(=O)CCCCCCCCCCCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)c2ccc(-c3scnc3C)cc2)C(C)(C)C)c2ccc(-c3cnn(C[C@@]45C[C@@]6(C)C[C@@](O)(C4)C[C@](OCCN(C)C)(C6)C5)c3C)c(C(=O)O)n2)nnc1Nc1nc2ccccc2s1	C79H108N14O9S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-0Z037N	SCHEMBL26918002	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3,5-dimethyl-7-(2-pyrrolidin-1-ylethoxy)-1-adamantyl]methyl]-5-methylpyrazol-4-yl]-N-[5-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-5-oxopentyl]pyridine-2-carboxamide; SCHEMBL26918020	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCNC(=O)c2nc(N3CCCc4c3nnc(Nc3nc5ccccc5s3)c4C)ccc2-c2cnn(CC34CC5(C)CC(C)(C3)CC(OCCN3CCCC3)(C5)C4)c2C)C(C)(C)C)cc1	C72H92N14O6S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-8B3P3Y	WO2022169780A1_123	.	Cc1ncsc1-c1ccc([C@@H](C)NC(=O)C2C[C@H](O)CN2C(=O)[C@@H](NC(=O)CCNC(=O)c2nc(N3CCCc4c3nnc(Nc3nc5ccccc5s3)c4C)ccc2-c2cnn(CC34CC5(C)CC(C)(C3)CC(OCCN3CCCC3)(C5)C4)c2C)C(C)(C)C)cc1	C70H88N14O6S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-MERMPE	WO2022169780A1_124	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[(3R,5S)-3,5-dimethyl-7-(2-pyrrolidin-1-ylethoxy)-1-adamantyl]methyl]-5-methylpyrazol-4-yl]-N-[9-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-9-oxononyl]pyridine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCCCNC(=O)c2nc(N3CCCc4c3nnc(Nc3nc5ccccc5s3)c4C)ccc2-c2cnn(C[C@]34C[C@]5(C)C[C@](C)(C3)C[C@@](OCCN3CCCC3)(C5)C4)c2C)C(C)(C)C)cc1	C76H100N14O6S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-4A3RX9	SCHEMBL26917409	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3,5-dimethyl-7-(2-pyrrolidin-1-ylethoxy)-1-adamantyl]methyl]-5-methylpyrazol-4-yl]-N-[11-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-11-oxoundecyl]pyridine-2-carboxamide; SCHEMBL26917424	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCCCCCNC(=O)c2nc(N3CCCc4c3nnc(Nc3nc5ccccc5s3)c4C)ccc2-c2cnn(CC34CC5(C)CC(C)(C3)CC(OCCN3CCCC3)(C5)C4)c2C)C(C)(C)C)cc1	C78H104N14O6S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-WSNTVT	SCHEMBL26918331	6-[[6-(1,3-benzothiazol-2-ylamino)-5-methylpyridazin-3-yl]-[4-[10-[(3R)-3-[(1-fluorocyclopropanecarbonyl)amino]-4-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-2-methyl-4-oxobutan-2-yl]sulfanyldecanoyl-methylamino]butyl]amino]-3-[1-[[3-[2-(dimethylamino)ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL26918347	Cc1cc(N(CCCCN(C)C(=O)CCCCCCCCCSC(C)(C)[C@H](NC(=O)C2(F)CC2)C(=O)N2C[C@H](O)C[C@H]2C(=O)NCc2ccc(-c3scnc3C)cc2)c2ccc(-c3cnn(CC45CC6(C)CC(C)(C4)CC(OCCN(C)C)(C6)C5)c3C)c(C(=O)O)n2)nnc1Nc1nc2ccccc2s1	C79H105FN14O8S3	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-S1HFV9	SCHEMBL26917559	6-[[6-(1,3-benzothiazol-2-ylamino)-5-methylpyridazin-3-yl]-[4-[13-[(3R)-3-[(1-fluorocyclopropanecarbonyl)amino]-4-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-2-methyl-4-oxobutan-2-yl]sulfanyltridecanoyl-methylamino]butyl]amino]-3-[1-[[3-[2-(dimethylamino)ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL26917571	Cc1cc(N(CCCCN(C)C(=O)CCCCCCCCCCCCSC(C)(C)[C@H](NC(=O)C2(F)CC2)C(=O)N2C[C@H](O)C[C@H]2C(=O)NCc2ccc(-c3scnc3C)cc2)c2ccc(-c3cnn(CC45CC6(C)CC(C)(C4)CC(OCCN(C)C)(C6)C5)c3C)c(C(=O)O)n2)nnc1Nc1nc2ccccc2s1	C82H111FN14O8S3	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-YF0PMV	SCHEMBL26917716	N'-[4-[[6-(1,3-benzothiazol-2-ylamino)-5-methylpyridazin-3-yl]-[5-[1-[[3-[2-(dimethylamino)ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]-6-(dimethylcarbamoyl)pyridin-2-yl]amino]butyl]-N-[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]-N'-methyldodecanediamide; SCHEMBL26917724	Cc1cc(N(CCCCN(C)C(=O)CCCCCCCCCCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)c2ccc(-c3scnc3C)cc2)C(C)(C)C)c2ccc(-c3cnn(CC45CC6(C)CC(C)(C4)CC(OCCN(C)C)(C6)C5)c3C)c(C(=O)N(C)C)n2)nnc1Nc1nc2ccccc2s1	C81H113N15O7S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-LLR5FR	SCHEMBL26917451	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3,5-dimethyl-7-(2-pyrrolidin-1-ylethoxy)-1-adamantyl]methyl]-5-methylpyrazol-4-yl]-N-[8-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-8-oxooctyl]pyridine-2-carboxamide; SCHEMBL26917460	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCCNC(=O)c2nc(N3CCCc4c3nnc(Nc3nc5ccccc5s3)c4C)ccc2-c2cnn(CC34CC5(C)CC(C)(C3)CC(OCCN3CCCC3)(C5)C4)c2C)C(C)(C)C)cc1	C75H98N14O6S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-ZDMI29	SCHEMBL26917734	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3,5-dimethyl-7-(2-pyrrolidin-1-ylethoxy)-1-adamantyl]methyl]-5-methylpyrazol-4-yl]-N-[10-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-10-oxodecyl]pyridine-2-carboxamide; SCHEMBL26917746	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCCCCNC(=O)c2nc(N3CCCc4c3nnc(Nc3nc5ccccc5s3)c4C)ccc2-c2cnn(CC34CC5(C)CC(C)(C3)CC(OCCN3CCCC3)(C5)C4)c2C)C(C)(C)C)cc1	C77H102N14O6S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-1TY9B7	SCHEMBL26917710	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3,5-dimethyl-7-(2-pyrrolidin-1-ylethoxy)-1-adamantyl]methyl]-5-methylpyrazol-4-yl]-N-[12-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-12-oxododecyl]pyridine-2-carboxamide; SCHEMBL26917718	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCCCCCCNC(=O)c2nc(N3CCCc4c3nnc(Nc3nc5ccccc5s3)c4C)ccc2-c2cnn(CC34CC5(C)CC(C)(C3)CC(OCCN3CCCC3)(C5)C4)c2C)C(C)(C)C)cc1	C79H106N14O6S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-I92MI5	SCHEMBL26917581	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[2-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethyl-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL30670895	Cc1c(Nc2nc3ccccc3s2)nnc2c1CCCN2c1ccc(-c2cnn(CC34CC5(C)CC(C)(C3)CC(OCCN(C)CCOCCOCCOCCOCCNc3cccc6c3C(=O)N(C3CCC(=O)NC3=O)C6=O)(C5)C4)c2C)c(C(=O)O)n1	C64H78N12O11S	BCL2L1	Q07817	CRBN	WO-2022169780-A1
TPD-TFR030	SCHEMBL26918944	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[[10-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-10-oxodecyl]-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL26918967	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCCCCN(C)CCOC23CC4(C)CC(C)(CC(Cn5ncc(-c6ccc(N7CCCc8c7nnc(Nc7nc9ccccc9s7)c8C)nc6C(=O)O)c5C)(C4)C2)C3)C(C)(C)C)cc1	C74H97N13O7S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-1DTE58	SCHEMBL26917974	2-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-5-[3-[2-fluoro-4-[3-[4-[10-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-10-oxodecyl]piperazin-1-yl]prop-1-ynyl]phenoxy]propyl]-1,3-thiazole-4-carboxylic acid; SCHEMBL30670925	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCCCCN2CCN(CC#Cc3ccc(OCCCc4sc(N5CCCc6c5nnc(Nc5nc7ccccc7s5)c6C)nc4C(=O)O)c(F)c3)CC2)C(C)(C)C)cc1	C68H83FN12O7S3	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-K2HKNI	SCHEMBL26917853	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[[11-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-11-oxoundecyl]-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL26917863	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCCCCCN(C)CCOC23CC4(C)CC(C)(CC(Cn5ncc(-c6ccc(N7CCCc8c7nnc(Nc7nc9ccccc9s7)c8C)nc6C(=O)O)c5C)(C4)C2)C3)C(C)(C)C)cc1	C75H99N13O7S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-9GIBXM	SCHEMBL26917897	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[[13-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-13-oxotridecyl]-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL26917908	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCCCCCCCN(C)CCOC23CC4(C)CC(C)(CC(Cn5ncc(-c6ccc(N7CCCc8c7nnc(Nc7nc9ccccc9s7)c8C)nc6C(=O)O)c5C)(C4)C2)C3)C(C)(C)C)cc1	C77H103N13O7S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-1V4B2D	SCHEMBL26917664	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[6-[2-[[[(2S,4R)-1-[(2S)-2-[(1-fluorocyclopropanecarbonyl)amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carbonyl]amino]methyl]-5-(4-methyl-1,3-thiazol-5-yl)phenoxy]hexyl-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL26917675; SCHEMBL30670825	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)C)c(OCCCCCCN(C)CCOC23CC4(C)CC(C)(CC(Cn5ncc(-c6ccc(N7CCCc8c7nnc(Nc7nc9ccccc9s7)c8C)nc6C(=O)O)c5C)(C4)C2)C3)c1	C73H92FN13O8S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-LYCIOI	SCHEMBL26917786	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[8-[2-[[[(2S,4R)-1-[(2S)-2-[(1-fluorocyclopropanecarbonyl)amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carbonyl]amino]methyl]-5-(4-methyl-1,3-thiazol-5-yl)phenoxy]octyl-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL26917799; SCHEMBL30670820	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)C)c(OCCCCCCCCN(C)CCOC23CC4(C)CC(C)(CC(Cn5ncc(-c6ccc(N7CCCc8c7nnc(Nc7nc9ccccc9s7)c8C)nc6C(=O)O)c5C)(C4)C2)C3)c1	C75H96FN13O8S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-79BPQ6	SCHEMBL26917826	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[12-[2-[[[(2S,4R)-1-[(2S)-2-[(1-fluorocyclopropanecarbonyl)amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carbonyl]amino]methyl]-5-(4-methyl-1,3-thiazol-5-yl)phenoxy]dodecyl-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL26917846; SCHEMBL30670953	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)C)c(OCCCCCCCCCCCCN(C)CCOC23CC4(C)CC(C)(CC(Cn5ncc(-c6ccc(N7CCCc8c7nnc(Nc7nc9ccccc9s7)c8C)nc6C(=O)O)c5C)(C4)C2)C3)c1	C79H104FN13O8S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-GI60ZT	SCHEMBL26917597	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[12-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxydodecyl-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL30670812	Cc1c(Nc2nc3ccccc3s2)nnc2c1CCCN2c1ccc(-c2cnn(CC34CC5(C)CC(C)(C3)CC(OCCN(C)CCCCCCCCCCCCOc3ccc6c(c3)C(=O)N(C3CCC(=O)NC3=O)C6=O)(C5)C4)c2C)c(C(=O)O)n1	C66H81N11O8S	BCL2L1	Q07817	CRBN	WO-2022169780-A1
TPD-YUSHSO	SCHEMBL26917922	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[6-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyhexyl-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL30670883	Cc1c(Nc2nc3ccccc3s2)nnc2c1CCCN2c1ccc(-c2cnn(CC34CC5(C)CC(C)(C3)CC(OCCN(C)CCCCCCOc3cccc6c3C(=O)N(C3CCC(=O)NC3=O)C6=O)(C5)C4)c2C)c(C(=O)O)n1	C60H69N11O8S	BCL2L1	Q07817	CRBN	WO-2022169780-A1
TPD-CFMZ7X	SCHEMBL26917720	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[14-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxytetradecyl-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL30670982	Cc1c(Nc2nc3ccccc3s2)nnc2c1CCCN2c1ccc(-c2cnn(CC34CC5(C)CC(C)(C3)CC(OCCN(C)CCCCCCCCCCCCCCOc3ccc6c(c3)C(=O)N(C3CCC(=O)NC3=O)C6=O)(C5)C4)c2C)c(C(=O)O)n1	C68H85N11O8S	BCL2L1	Q07817	CRBN	WO-2022169780-A1
TPD-DFZFTT	SCHEMBL26917894	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[8-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyoctyl-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL30670931	Cc1c(Nc2nc3ccccc3s2)nnc2c1CCCN2c1ccc(-c2cnn(CC34CC5(C)CC(C)(C3)CC(OCCN(C)CCCCCCCCOc3cccc6c3C(=O)N(C3CCC(=O)NC3=O)C6=O)(C5)C4)c2C)c(C(=O)O)n1	C62H73N11O8S	BCL2L1	Q07817	CRBN	WO-2022169780-A1
TPD-A67W0G	SCHEMBL26918182	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[10-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxydecyl-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL30670824	Cc1c(Nc2nc3ccccc3s2)nnc2c1CCCN2c1ccc(-c2cnn(CC34CC5(C)CC(C)(C3)CC(OCCN(C)CCCCCCCCCCOc3cccc6c3C(=O)N(C3CCC(=O)NC3=O)C6=O)(C5)C4)c2C)c(C(=O)O)n1	C64H77N11O8S	BCL2L1	Q07817	CRBN	WO-2022169780-A1
TPD-1TO1TW	SCHEMBL26918176	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[[17-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-17-oxoheptadecyl]-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL26918192	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCCCCCCCCCCCN(C)CCOC23CC4(C)CC(C)(CC(Cn5ncc(-c6ccc(N7CCCc8c7nnc(Nc7nc9ccccc9s7)c8C)nc6C(=O)O)c5C)(C4)C2)C3)C(C)(C)C)cc1	C81H111N13O7S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-DQ51VL	SCHEMBL26917384	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[14-[2-[[[(2S,4R)-1-[(2S)-2-[(1-fluorocyclopropanecarbonyl)amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carbonyl]amino]methyl]-5-(4-methyl-1,3-thiazol-5-yl)phenoxy]tetradecyl-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL26917395; SCHEMBL30670879	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)C)c(OCCCCCCCCCCCCCCN(C)CCOC23CC4(C)CC(C)(CC(Cn5ncc(-c6ccc(N7CCCc8c7nnc(Nc7nc9ccccc9s7)c8C)nc6C(=O)O)c5C)(C4)C2)C3)c1	C81H108FN13O8S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-A077ZM	SCHEMBL26917758	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[16-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxyhexadecyl-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL30670816	Cc1c(Nc2nc3ccccc3s2)nnc2c1CCCN2c1ccc(-c2cnn(CC34CC5(C)CC(C)(C3)CC(OCCN(C)CCCCCCCCCCCCCCCCOc3ccc6c(c3)C(=O)N(C3CCC(=O)NC3=O)C6=O)(C5)C4)c2C)c(C(=O)O)n1	C70H89N11O8S	BCL2L1	Q07817	CRBN	WO-2022169780-A1
TPD-25A18S	SCHEMBL26917731	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[[14-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-14-oxotetradecyl]-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]-N,N-dimethylpyridine-2-carboxamide; SCHEMBL26917743	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCCCCCCCCN(C)CCOC23CC4(C)CC(C)(CC(Cn5ncc(-c6ccc(N7CCCc8c7nnc(Nc7nc9ccccc9s7)c8C)nc6C(=O)N(C)C)c5C)(C4)C2)C3)C(C)(C)C)cc1	C80H110N14O6S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-B61EJ1	SCHEMBL26917386	2-[[6-(1,3-Benzothiazol-2-ylamino)-5-methylpyridazin-3-yl]-[4-[3-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethoxy]propanoylamino]butyl]amino]-5-[3-[4-[3-(dimethylamino)prop-1-ynyl]-2-fluorophenoxy]propyl]-1,3-thiazole-4-carboxylic acid; SCHEMBL30670783	Cc1cc(N(CCCCNC(=O)CCOCCOCCOCCOCCNc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)c2nc(C(=O)O)c(CCCOc3ccc(C#CCN(C)C)cc3F)s2)nnc1Nc1nc2ccccc2s1	C58H66FN11O12S2	BCL2L1	Q07817	CRBN	WO-2022169780-A1
TPD-MSNIOK	SCHEMBL26917935	6-[[6-(1,3-Benzothiazol-2-ylamino)-5-methylpyridazin-3-yl]-[5-[4-[7-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]heptyl]triazol-1-yl]pentyl]amino]-3-[1-[[3-[2-(dimethylamino)ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL30670961	Cc1cc(N(CCCCCn2cc(CCCCCCCNc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)nn2)c2ccc(-c3cnn(CC45CC6(C)CC(C)(C4)CC(OCCN(C)C)(C6)C5)c3C)c(C(=O)O)n2)nnc1Nc1nc2ccccc2s1	C66H81N15O7S	BCL2L1	Q07817	CRBN	WO-2022169780-A1
TPD-5AAN1B	WO2022169780A1_151	.	Cc1cc(N(CCCCCn2cc(COCCOCCOCCOCCOCCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCc3ccc(-c4scnc4C)cc3)C(C)(C)C)nn2)c2ccc(-c3cnn(CC45CC6(C)CC(C)(C4)CC(OCCN(C)C)(C6)C5)c3C)c(C(=O)O)n2)nnc1Nc1nc2ccccc2s1	C80H108N16O12S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-X9UD0F	SCHEMBL26918073	6-[[6-(1,3-benzothiazol-2-ylamino)-5-methylpyridazin-3-yl]-[5-[4-[9-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-9-oxononyl]triazol-1-yl]pentyl]amino]-3-[1-[[3-[2-(dimethylamino)ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL26918092	Cc1cc(N(CCCCCn2cc(CCCCCCCCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCc3ccc(-c4scnc4C)cc3)C(C)(C)C)nn2)c2ccc(-c3cnn(CC45CC6(C)CC(C)(C4)CC(OCCN(C)C)(C6)C5)c3C)c(C(=O)O)n2)nnc1Nc1nc2ccccc2s1	C77H102N16O7S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-SQG3SX	SCHEMBL26917728	6-[[6-(1,3-Benzothiazol-2-ylamino)-5-methylpyridazin-3-yl]-[5-[4-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethoxymethyl]triazol-1-yl]pentyl]amino]-3-[1-[[3-[2-(dimethylamino)ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL30670774	Cc1cc(N(CCCCCn2cc(COCCOCCOCCOCCNc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)nn2)c2ccc(-c3cnn(CC45CC6(C)CC(C)(C4)CC(OCCN(C)C)(C6)C5)c3C)c(C(=O)O)n2)nnc1Nc1nc2ccccc2s1	C68H85N15O11S	BCL2L1	Q07817	CRBN	WO-2022169780-A1
TPD-NSIURM	SCHEMBL26917682	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[[14-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-14-oxotetradecyl]-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxamide; SCHEMBL26917689	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCCCCCCCCN(C)CCOC23CC4(C)CC(C)(CC(Cn5ncc(-c6ccc(N7CCCc8c7nnc(Nc7nc9ccccc9s7)c8C)nc6C(N)=O)c5C)(C4)C2)C3)C(C)(C)C)cc1	C78H106N14O6S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-YWFUJC	WO2022169780A1_155	.	C/C(NCC12CC3(C)CC(C)(C1)CC(OCCN(C)CCCCCCCCCCCCCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)c1ccc(-c4scnc4C)cc1)C(C)(C)C)(C3)C2)=C(/C=N)c1ccc(N2CCCc3c2nnc(Nc2nc4ccccc4s2)c3C)nc1CO	C78H109N13O6S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-9DQWCO	WO2022169780A1_156	.	CNC(=O)c1nc(N2CCCc3c2nnc(Nc2nc4ccccc4s2)c3C)ccc1/C(C=N)=C(\C)NCC12CC3(C)CC(C)(C1)CC(OCCN(C)CCCCCCCCCCCCCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)c1ccc(-c4scnc4C)cc1)C(C)(C)C)(C3)C2	C79H110N14O6S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-H4F1SG	SCHEMBL26917783	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[[14-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-14-oxotetradecyl]-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]-N-propan-2-ylpyridine-2-carboxamide; SCHEMBL26917798	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCCCCCCCCN(C)CCOC23CC4(C)CC(C)(CC(Cn5ncc(-c6ccc(N7CCCc8c7nnc(Nc7nc9ccccc9s7)c8C)nc6C(=O)NC(C)C)c5C)(C4)C2)C3)C(C)(C)C)cc1	C81H112N14O6S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-27S09T	WO2022169780A1_158	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3,5-dimethyl-7-(2-pyrrolidin-1-ylethoxy)-1-adamantyl]methyl]-5-methylpyrazol-4-yl]-N-[2-[2-[3-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-3-oxopropoxy]ethoxy]ethyl]pyridine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCOCCOCCNC(=O)c2nc(N3CCCc4c3nnc(Nc3nc5ccccc5s3)c4C)ccc2-c2cnn(CC34CC5(C)CC(C)(C3)CC(OCCN3CCCC3)(C5)C4)c2C)C(C)(C)C)cc1	C74H96N14O8S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-SQ4BT1	WO2022169780A1_159	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3,5-dimethyl-7-(2-pyrrolidin-1-ylethoxy)-1-adamantyl]methyl]-5-methylpyrazol-4-yl]-N-[2-[2-[2-[3-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-3-oxopropoxy]ethoxy]ethoxy]ethyl]pyridine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCOCCOCCOCCNC(=O)c2nc(N3CCCc4c3nnc(Nc3nc5ccccc5s3)c4C)ccc2-c2cnn(CC34CC5(C)CC(C)(C3)CC(OCCN3CCCC3)(C5)C4)c2C)C(C)(C)C)cc1	C76H100N14O9S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-UZ56K7	WO2022169780A1_160	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3,5-dimethyl-7-(2-pyrrolidin-1-ylethoxy)-1-adamantyl]methyl]-5-methylpyrazol-4-yl]-N-[2-[2-[2-[3-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-3-oxopropoxy]ethoxy]ethoxy]ethyl]-N-methylpyridine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCOCCOCCOCCN(C)C(=O)c2nc(N3CCCc4c3nnc(Nc3nc5ccccc5s3)c4C)ccc2-c2cnn(CC34CC5(C)CC(C)(C3)CC(OCCN3CCCC3)(C5)C4)c2C)C(C)(C)C)cc1	C77H102N14O9S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-EESM2G	WO2022169780A1_161	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3,5-dimethyl-7-(2-pyrrolidin-1-ylethoxy)-1-adamantyl]methyl]-5-methylpyrazol-4-yl]-N-[9-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-9-oxononyl]-N-methylpyridine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCCCN(C)C(=O)c2nc(N3CCCc4c3nnc(Nc3nc5ccccc5s3)c4C)ccc2-c2cnn(CC34CC5(C)CC(C)(C3)CC(OCCN3CCCC3)(C5)C4)c2C)C(C)(C)C)cc1	C77H102N14O6S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-MBHHFZ	WO2022169780A1_162	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3,5-dimethyl-7-(2-pyrrolidin-1-ylethoxy)-1-adamantyl]methyl]-5-methylpyrazol-4-yl]-N-[4-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]carbamoyl]cyclohexyl]pyridine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)[C@H]2CC[C@H](NC(=O)c3nc(N4CCCc5c4nnc(Nc4nc6ccccc6s4)c5C)ccc3-c3cnn(CC45CC6(C)CC(C)(C4)CC(OCCN4CCCC4)(C6)C5)c3C)CC2)C(C)(C)C)cc1	C74H94N14O6S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-S2HZEC	WO2022169780A1_163	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C[C@H]2CC[C@@H](NC(=O)c3nc(N4CCCc5c4nnc(Nc4nc6ccccc6s4)c5C)ccc3-c3cnn(CC45CC6(C)CC(C)(C4)CC(OCCN4CCCC4)(C6)C5)c3C)CC2)C(C)(C)C)cc1	C75H96N14O6S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-5LDU64	WO2022169780A1_164	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C[C@H]2CC[C@H](NC(=O)c3nc(N4CCCc5c4nnc(Nc4nc6ccccc6s4)c5C)ccc3-c3cnn(CC45CC6(C)CC(C)(C4)CC(OCCN4CCCC4)(C6)C5)c3C)CC2)C(C)(C)C)cc1	C75H96N14O6S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-T2O1RN	WO2022169780A1_165	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3,5-dimethyl-7-(2-pyrrolidin-1-ylethoxy)-1-adamantyl]methyl]-5-methylpyrazol-4-yl]-N-[3-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]carbamoyl]cyclobutyl]pyridine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)[C@H]2C[C@H](NC(=O)c3nc(N4CCCc5c4nnc(Nc4nc6ccccc6s4)c5C)ccc3-c3cnn(CC45CC6(C)CC(C)(C4)CC(OCCN4CCCC4)(C6)C5)c3C)C2)C(C)(C)C)cc1	C72H90N14O6S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-YL1DY3	WO2022169780A1_166	(2S,4R)-1-[(2S)-2-[[2-[1-[6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3,5-dimethyl-7-(2-pyrrolidin-1-ylethoxy)-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carbonyl]piperidin-4-yl]oxyacetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COC2CCN(C(=O)c3nc(N4CCCc5c4nnc(Nc4nc6ccccc6s4)c5C)ccc3-c3cnn(CC45CC6(C)CC(C)(C4)CC(OCCN4CCCC4)(C6)C5)c3C)CC2)C(C)(C)C)cc1	C74H94N14O7S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-N31QMR	WO2022169780A1_167	(2S,4R)-1-[(2S)-2-[3-[1-[6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3,5-dimethyl-7-(2-pyrrolidin-1-ylethoxy)-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carbonyl]piperidin-4-yl]oxypropanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCOC2CCN(C(=O)c3nc(N4CCCc5c4nnc(Nc4nc6ccccc6s4)c5C)ccc3-c3cnn(CC45CC6(C)CC(C)(C4)CC(OCCN4CCCC4)(C6)C5)c3C)CC2)C(C)(C)C)cc1	C75H96N14O7S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-XAS5OF	WO2022169780A1_168	(3S)-1-[6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3,5-dimethyl-7-(2-pyrrolidin-1-ylethoxy)-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carbonyl]-N-[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]piperidine-3-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)[C@H]2CCCN(C(=O)c3nc(N4CCCc5c4nnc(Nc4nc6ccccc6s4)c5C)ccc3-c3cnn(CC45CC6(C)CC(C)(C4)CC(OCCN4CCCC4)(C6)C5)c3C)C2)C(C)(C)C)cc1	C73H92N14O6S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-NDWSWK	WO2022169780A1_169	(3R)-1-[6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3,5-dimethyl-7-(2-pyrrolidin-1-ylethoxy)-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carbonyl]-N-[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]piperidine-3-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)[C@@H]2CCCN(C(=O)c3nc(N4CCCc5c4nnc(Nc4nc6ccccc6s4)c5C)ccc3-c3cnn(CC45CC6(C)CC(C)(C4)CC(OCCN4CCCC4)(C6)C5)c3C)C2)C(C)(C)C)cc1	C73H92N14O6S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-R7536K	WO2022169780A1_170	(2S,4R)-1-[(2S)-2-[[2-[2-[6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3,5-dimethyl-7-(2-pyrrolidin-1-ylethoxy)-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carbonyl]-2-azaspiro[3.3]heptan-6-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CC2CC3(C2)CN(C(=O)c2nc(N4CCCc5c4nnc(Nc4nc6ccccc6s4)c5C)ccc2-c2cnn(CC45CC6(C)CC(C)(C4)CC(OCCN4CCCC4)(C6)C5)c2C)C3)C(C)(C)C)cc1	C75H94N14O6S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-4S6P7W	WO2022169780A1_171	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3,5-dimethyl-7-(2-pyrrolidin-1-ylethoxy)-1-adamantyl]methyl]-5-methylpyrazol-4-yl]-N-[(3R)-1-[4-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-4-oxobutanoyl]piperidin-3-yl]pyridine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCC(=O)N2CCC[C@@H](NC(=O)c3nc(N4CCCc5c4nnc(Nc4nc6ccccc6s4)c5C)ccc3-c3cnn(CC45CC6(C)CC(C)(C4)CC(OCCN4CCCC4)(C6)C5)c3C)C2)C(C)(C)C)cc1	C76H97N15O7S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-1T9MYT	WO2022169780A1_172	.	Cc1ncsc1-c1ccc([C@@H](C)NC(=O)[C@@H]2C[C@H](O)CN2C(=O)[C@H](NC(=O)CCCCCCS(=O)(=O)NC(=O)c2nc(N3CCCc4c3nnc(Nc3nc5ccccc5s3)c4C)ccc2-c2cnn(CC34CC5(C)CC(C)(C3)CC(OCCN3CCCC3)(C5)C4)c2C)C(C)(C)C)cc1	C74H96N14O8S3	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-CUCJJF	SCHEMBL26917541	6-[3-(1,3-benzothiazol-2-ylamino)-4-methyl-6,7-dihydro-5H-pyrido[2,3-c]pyridazin-8-yl]-3-[1-[[3-[2-[2-[2-[3-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-3-oxopropoxy]ethoxy]ethyl-methylamino]ethoxy]-5,7-dimethyl-1-adamantyl]methyl]-5-methylpyrazol-4-yl]pyridine-2-carboxylic acid; SCHEMBL26917552	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCOCCOCCN(C)CCOC23CC4(C)CC(C)(CC(Cn5ncc(-c6ccc(N7CCCc8c7nnc(Nc7nc9ccccc9s7)c8C)nc6C(=O)O)c5C)(C4)C2)C3)C(C)(C)C)cc1	C71H91N13O9S2	BCL2L1	Q07817	VHL	WO-2022169780-A1
TPD-9F2GIG	WO2022187417A1_CP-001	6-[2-[4-[5-acetyl-3-[7-(difluoromethyl)-6-(1-methylpyrazol-4-yl)-3,4-dihydro-2H-quinolin-1-yl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]piperidin-1-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-7,8-dihydro-5H-pyrrolo[3,4-g]isoquinoline-1,3-dione	CC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C(C(F)F)C(C1=CN(C)N=C1)=C3)=NN2C1CCN(C(=O)CN2CCC3=CC4=C(C=C3C2)C(=O)N(C2CCC(=O)NC2=O)C4=O)CC1	C45H48F2N10O6	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-VLOJU3	WO2022187417A1_CP-002	6-[2-[4-[5-acetyl-3-[7-(difluoromethyl)-6-(1-methylpyrazol-4-yl)-3,4-dihydro-2H-quinolin-1-yl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]piperidin-1-yl]acetyl]-2-(2,6-dioxopiperidin-3-yl)-7,8-dihydro-5H-pyrrolo[3,4-g]isoquinoline-1,3-dione	CC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C(C(F)F)C(C1=CN(C)N=C1)=C3)=NN2C1CCN(CC(=O)N2CCC3=CC4=C(C=C3C2)C(=O)N(C2CCC(=O)NC2=O)C4=O)CC1	C45H48F2N10O6	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-CRK0JM	WO2022187417A1_CP-003	6-[3-[4-[5-acetyl-3-[7-(difluoromethyl)-6-(1-methylpyrazol-4-yl)-3,4-dihydro-2H-quinolin-1-yl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]piperidin-1-yl]-3-oxopropyl]-2-(2,6-dioxopiperidin-3-yl)-7,8-dihydro-5H-pyrrolo[3,4-g]isoquinoline-1,3-dione	CC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C(C(F)F)C(C1=CN(C)N=C1)=C3)=NN2C1CCN(C(=O)CCN2CCC3=CC4=C(C=C3C2)C(=O)N(C2CCC(=O)NC2=O)C4=O)CC1	C46H50F2N10O6	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-0VPTLW	WO2022187417A1_CP-004	6-[4-[4-[5-acetyl-3-[7-(difluoromethyl)-6-(1-methylpyrazol-4-yl)-3,4-dihydro-2H-quinolin-1-yl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]piperidin-1-yl]-4-oxobutyl]-2-(2,6-dioxopiperidin-3-yl)-7,8-dihydro-5H-pyrrolo[3,4-g]isoquinoline-1,3-dione	CC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C(C(F)F)C(C1=CN(C)N=C1)=C3)=NN2C1CCN(C(=O)CCCN2CCC3=CC4=C(C=C3C2)C(=O)N(C2CCC(=O)NC2=O)C4=O)CC1	C47H52F2N10O6	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-VXD994	WO2022187417A1_CP-005	6-[2-[4-[5-acetyl-3-[7-(difluoromethyl)-6-(1-methylpyrazol-4-yl)-3,4-dihydro-2H-quinolin-1-yl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]piperidin-1-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	CC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C(C(F)F)C(C1=CN(C)N=C1)=C3)=NN2C1CCN(C(=O)CN2CC3=CC4=C(C=C3C2)C(=O)N(C2CCC(=O)NC2=O)C4=O)CC1	C44H46F2N10O6	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-CJX699	WO2022187417A1_CP-006	6-[2-[4-[5-acetyl-3-[7-(difluoromethyl)-6-(1-methylpyrazol-4-yl)-3,4-dihydro-2H-quinolin-1-yl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]piperidin-1-yl]acetyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	CC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C(C(F)F)C(C1=CN(C)N=C1)=C3)=NN2C1CCN(CC(=O)N2CC3=CC4=C(C=C3C2)C(=O)N(C2CCC(=O)NC2=O)C4=O)CC1	C44H46F2N10O6	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-HVAL7S	WO2022187417A1_CP-007	6-[3-[4-[5-acetyl-3-[7-(difluoromethyl)-6-(1-methylpyrazol-4-yl)-3,4-dihydro-2H-quinolin-1-yl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]piperidin-1-yl]-3-oxopropyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	CC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C(C(F)F)C(C1=CN(C)N=C1)=C3)=NN2C1CCN(C(=O)CCN2CC3=CC4=C(C=C3C2)C(=O)N(C2CCC(=O)NC2=O)C4=O)CC1	C45H48F2N10O6	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-SR4MPA	WO2022187417A1_CP-008	.	CC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C(C(F)F)C(C1=CN(C)N=C1)=C3)=NN2C1CCN(C(=O)CCCN2CC3=CC4=C(C=C3C2)C(=O)N(C2CCC(=O)NC2=O)C4=O)CC1	C46H50F2N10O6	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-CG2LIQ	WO2022187417A1_CP-009	6-[2-[4-[5-acetyl-3-[7-(difluoromethyl)-3,4-dihydro-2H-quinolin-1-yl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]piperidin-1-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-7,8-dihydro-5H-pyrrolo[3,4-g]isoquinoline-1,3-dione	[H]C1=CC2=C(C=C1C(F)F)N(C1=NN(C3CCN(C(=O)CN4CCC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C3=C1CN(C(C)=O)CC3)CCC2	C41H44F2N8O6	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-AHR4B0	WO2022187417A1_CP-010	6-[2-[4-[5-acetyl-3-[7-(difluoromethyl)-3,4-dihydro-2H-quinolin-1-yl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]piperidin-1-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	[H]C1=CC2=C(C=C1C(F)F)N(C1=NN(C3CCN(C(=O)CN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C3=C1CN(C(C)=O)CC3)CCC2	C40H42F2N8O6	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-3DZ0VS	WO2022187417A1_CP-011	6-[2-[4-[5-acetyl-3-[7-(difluoromethyl)-6-methyl-3,4-dihydro-2H-quinolin-1-yl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]piperidin-1-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	CC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C(C(F)F)C(C)=C3)=NN2C1CCN(C(=O)CN2CC3=CC4=C(C=C3C2)C(=O)N(C2CCC(=O)NC2=O)C4=O)CC1	C41H44F2N8O6	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-TE1YQB	WO2022187417A1_CP-012	6-[2-[4-[5-acetyl-3-[7-(difluoromethyl)-6-ethyl-3,4-dihydro-2H-quinolin-1-yl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]piperidin-1-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	CCC1=CC2=C(C=C1C(F)F)N(C1=NN(C3CCN(C(=O)CN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C3=C1CN(C(C)=O)CC3)CCC2	C42H46F2N8O6	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-WENW2D	WO2022187417A1_CP-013	6-[2-[4-[5-acetyl-3-[6-cyclopropyl-7-(difluoromethyl)-3,4-dihydro-2H-quinolin-1-yl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]piperidin-1-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	CC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C(C(F)F)C(C1CC1)=C3)=NN2C1CCN(C(=O)CN2CC3=CC4=C(C=C3C2)C(=O)N(C2CCC(=O)NC2=O)C4=O)CC1	C43H46F2N8O6	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-LSY1Z0	WO2022187417A1_CP-014	6-[2-[4-[5-acetyl-3-[6-cyclopropyl-7-(difluoromethyl)-3,4-dihydro-2H-quinolin-1-yl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]piperidin-1-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-7,8-dihydro-5H-pyrrolo[3,4-g]isoquinoline-1,3-dione	CC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C(C(F)F)C(C1CC1)=C3)=NN2C1CCN(C(=O)CN2CCC3=CC4=C(C=C3C2)C(=O)N(C2CCC(=O)NC2=O)C4=O)CC1	C44H48F2N8O6	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-WHTUZB	WO2022187417A1_CP-015	6-[2-[4-[5-acetyl-3-[7-(difluoromethyl)-6-propan-2-yl-3,4-dihydro-2H-quinolin-1-yl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]piperidin-1-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	CC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C(C(F)F)C(C(C)C)=C3)=NN2C1CCN(C(=O)CN2CC3=CC4=C(C=C3C2)C(=O)N(C2CCC(=O)NC2=O)C4=O)CC1	C43H48F2N8O6	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-4S55PV	WO2022187417A1_CP-016	6-[2-[4-[5-acetyl-3-[6-bromo-7-(difluoromethyl)-3,4-dihydro-2H-quinolin-1-yl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]piperidin-1-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	CC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C(C(F)F)C(Br)=C3)=NN2C1CCN(C(=O)CN2CC3=CC4=C(C=C3C2)C(=O)N(C2CCC(=O)NC2=O)C4=O)CC1	C40H41BrF2N8O6	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-7ITD39	WO2022187417A1_CP-017	6-[2-[4-[5-acetyl-3-[6-chloro-7-(difluoromethyl)-3,4-dihydro-2H-quinolin-1-yl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]piperidin-1-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	CC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C(C(F)F)C(Cl)=C3)=NN2C1CCN(C(=O)CN2CC3=CC4=C(C=C3C2)C(=O)N(C2CCC(=O)NC2=O)C4=O)CC1	C40H41ClF2N8O6	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-HVNJQJ	WO2022187417A1_CP-018	6-[2-[4-[5-acetyl-3-[6-chloro-7-(difluoromethyl)-3,4-dihydro-2H-quinolin-1-yl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]piperidin-1-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-7,8-dihydro-5H-pyrrolo[3,4-g]isoquinoline-1,3-dione	CC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C(C(F)F)C(Cl)=C3)=NN2C1CCN(C(=O)CN2CCC3=CC4=C(C=C3C2)C(=O)N(C2CCC(=O)NC2=O)C4=O)CC1	C41H43ClF2N8O6	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-XCSTE8	WO2022187417A1_CP-019	6-[2-[4-[5-acetyl-3-[6-acetyl-7-(difluoromethyl)-3,4-dihydro-2H-quinolin-1-yl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]piperidin-1-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	CC(=O)C1=CC2=C(C=C1C(F)F)N(C1=NN(C3CCN(C(=O)CN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C3=C1CN(C(C)=O)CC3)CCC2	C42H44F2N8O7	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-7BIMXE	WO2022187417A1_CP-020	6-[2-[4-[5-acetyl-3-[6-acetyl-7-(difluoromethyl)-3,4-dihydro-2H-quinolin-1-yl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]piperidin-1-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-7,8-dihydro-5H-pyrrolo[3,4-g]isoquinoline-1,3-dione	CC(=O)C1=CC2=C(C=C1C(F)F)N(C1=NN(C3CCN(C(=O)CN4CCC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C3=C1CN(C(C)=O)CC3)CCC2	C43H46F2N8O7	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-S9GCG5	WO2022187417A1_CP-021	6-[2-[4-[5-acetyl-3-[6-cyclohexyl-7-(difluoromethyl)-3,4-dihydro-2H-quinolin-1-yl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]piperidin-1-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	CC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C(C(F)F)C(C1CCCCC1)=C3)=NN2C1CCN(C(=O)CN2CC3=C(C=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)C2)CC1	C46H52F2N8O6	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-94PYUC	SCHEMBL27214134	6-[2-[4-[5-acetyl-3-[7-(difluoromethyl)-6-phenyl-3,4-dihydro-2H-quinolin-1-yl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]piperidin-1-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	CC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C(C(F)F)C(C1=CC=CC=C1)=C3)=NN2C1CCN(C(=O)CN2CC3=C(C=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)C2)CC1	C46H46F2N8O6	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-IFLONN	SCHEMBL27214140	6-[2-[4-[5-acetyl-3-[7-(difluoromethyl)-6-(4-fluorophenyl)-3,4-dihydro-2H-quinolin-1-yl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]piperidin-1-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	CC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C(C(F)F)C(C1=CC=C(F)C=C1)=C3)=NN2C1CCN(C(=O)CN2CC3=C(C=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)C2)CC1	C46H45F3N8O6	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-GKT4ZG	WO2022187417A1_CP-024	6-[2-[4-[5-acetyl-3-[7-(difluoromethyl)-6-thiophen-2-yl-3,4-dihydro-2H-quinolin-1-yl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]piperidin-1-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	CC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C(C(F)F)C(C1=CC=CS1)=C3)=NN2C1CCN(C(=O)CN2CC3=C(C=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)C2)CC1	C44H44F2N8O6S	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-J5Y8UL	WO2022187417A1_CP-025	6-[2-[4-[5-acetyl-3-[6-(2-cyclopropylethyl)-7-(difluoromethyl)-3,4-dihydro-2H-quinolin-1-yl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]piperidin-1-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	CC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C(C(F)F)C(CCC1CC1)=C3)=NN2C1CCN(C(=O)CN2CC3=C(C=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)C2)CC1	C45H50F2N8O6	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-7G43VM	WO2022187417A1_CP-026	6-[2-[4-[5-acetyl-3-[7-(difluoromethyl)-6-(3-methylbutyl)-3,4-dihydro-2H-quinolin-1-yl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]piperidin-1-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	CC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C(C(F)F)C(CCC(C)C)=C3)=NN2C1CCN(C(=O)CN2CC3=C(C=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)C2)CC1	C45H52F2N8O6	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-D9QEL8	WO2022187417A1_CP-027	6-[2-[4-[5-acetyl-3-[7-(difluoromethyl)-6-(1-methylpyrazol-4-yl)-3,4-dihydro-2H-quinolin-1-yl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]cyclohexyl]acetyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	CC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C(C(F)F)C(C1=CN(C)N=C1)=C3)=NN2C1CCC(CC(=O)N2CC3=C(C=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)C2)CC1	C45H47F2N9O6	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-L7P7UD	WO2022187417A1_CP-028	6-[2-[4-[5-acetyl-3-[7-(difluoromethyl)-6-(1-methylpyrazol-4-yl)-3,4-dihydro-2H-quinolin-1-yl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]cyclohexyl]acetyl]-2-(2,6-dioxopiperidin-3-yl)-7,8-dihydro-5H-pyrrolo[3,4-g]isoquinoline-1,3-dione	CC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C(C(F)F)C(C1=CN(C)N=C1)=C3)=NN2C1CCC(CC(=O)N2CCC3=C(C=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)C2)CC1	C46H49F2N9O6	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-3GWR6Y	WO2022187417A1_CP-029	.	CC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C(C(F)F)C(C1=CN(C)N=C1)=C3)=NN2C[C@H]1CC[C@H](C(=O)N2CC3=C(C=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)C2)CC1	C45H47F2N9O6	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-3MOAUN	WO2022187417A1_CP-030	.	CC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C(C(F)F)C(C1=CN(C)N=C1)=C3)=NN2C[C@H]1CC[C@H](C(=O)N2CCC3=C(C=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)C2)CC1	C46H49F2N9O6	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-5U7W9F	WO2022187417A1_CP-031	.	CC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C(C(F)F)C(C1=CN(C)N=C1)=C3)=NN2C[C@H]1CC[C@@H](C(=O)N2CC3=C(C=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)C2)CC1	C45H47F2N9O6	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-FJT3TY	WO2022187417A1_CP-032	.	CC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C(C(F)F)C(C1=CN(C)N=C1)=C3)=NN2C[C@H]1CC[C@@H](C(=O)N2CCC3=C(C=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)C2)CC1	C46H49F2N9O6	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-03XC9G	WO2022187417A1_CP-033	6-[4-[5-acetyl-3-[7-(difluoromethyl)-6-(1-methylpyrazol-4-yl)-3,4-dihydro-2H-quinolin-1-yl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]cyclohexanecarbonyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	CC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C(C(F)F)C(C1=CN(C)N=C1)=C3)=NN2C1CCC(C(=O)N2CC3=C(C=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)C2)CC1	C44H45F2N9O6	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-XDDREI	WO2022187417A1_CP-035	6-[4-[5-acetyl-3-[7-(difluoromethyl)-6-(1-methylpyrazol-4-yl)-3,4-dihydro-2H-quinolin-1-yl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]cyclohexanecarbonyl]-2-(2,6-dioxopiperidin-3-yl)-7,8-dihydro-5H-pyrrolo[3,4-g]isoquinoline-1,3-dione	CC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C(C(F)F)C(C1=CN(C)N=C1)=C3)=NN2C1CCC(C(=O)N2CCC3=C(C=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)C2)CC1	C45H47F2N9O6	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-3P3WN7	WO2022187417A1_CP-037	6-[4-[5-acetyl-3-[7-(difluoromethyl)-6-(1-methylpyrazol-4-yl)-3,4-dihydro-2H-quinolin-1-yl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]cyclohexyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	CC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C(C(F)F)C(C1=CN(C)N=C1)=C3)=NN2C1CCC(N2CC3=CC4=C(C=C3C2)C(=O)N(C2CCC(=O)NC2=O)C4=O)CC1	C43H45F2N9O5	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-RL36MN	WO2022187417A1_CP-038	6-[4-[5-acetyl-3-[7-(difluoromethyl)-6-(1-methylpyrazol-4-yl)-3,4-dihydro-2H-quinolin-1-yl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]cyclohexyl]-2-(2,6-dioxopiperidin-3-yl)-7,8-dihydro-5H-pyrrolo[3,4-g]isoquinoline-1,3-dione	CC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C(C(F)F)C(C1=CN(C)N=C1)=C3)=NN2C1CCC(N2CCC3=CC4=C(C=C3C2)C(=O)N(C2CCC(=O)NC2=O)C4=O)CC1	C44H47F2N9O5	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-L0E3UB	WO2022187417A1_CP-039	.	CC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C(C(F)F)C(C1=CN(C)N=C1)=C3)=NN2C[C@H]1CC[C@H](N2CC3=CC4=C(C=C3C2)C(=O)N(C2CCC(=O)NC2=O)C4=O)CC1	C44H47F2N9O5	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-TSVUKA	WO2022187417A1_CP-040	.	CC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C(C(F)F)C(C1=CN(C)N=C1)=C3)=NN2C[C@H]1CC[C@@H](N2CC3=CC4=C(C=C3C2)C(=O)N(C2CCC(=O)NC2=O)C4=O)CC1	C44H47F2N9O5	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-M3BICE	WO2022187417A1_CP-041	.	CC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C(C(F)F)C(C1=CN(C)N=C1)=C3)=NN2C[C@H]1CC[C@H](N2CCC3=CC4=C(C=C3C2)C(=O)N(C2CCC(=O)NC2=O)C4=O)CC1	C45H49F2N9O5	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-S84AAY	WO2022187417A1_CP-042	.	CC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C(C(F)F)C(C1=CN(C)N=C1)=C3)=NN2C[C@H]1CC[C@@H](N2CCC3=CC4=C(C=C3C2)C(=O)N(C2CCC(=O)NC2=O)C4=O)CC1	C45H49F2N9O5	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-HKZXBN	WO2022187417A1_CP-043	6-[[4-[[5-acetyl-3-[7-(difluoromethyl)-6-(1-methylpyrazol-4-yl)-3,4-dihydro-2H-quinolin-1-yl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]methyl]cyclohexyl]methyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	CC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C(C(F)F)C(C1=CN(C)N=C1)=C3)=NN2C[C@H]1CC[C@H](CN2CC3=CC4=C(C=C3C2)C(=O)N(C2CCC(=O)NC2=O)C4=O)CC1	C45H49F2N9O5	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-G9IS6Q	WO2022187417A1_CP-044	6-[2-[4-[5-acetyl-3-[7-(difluoromethyl)-6-(1-methylpyrazol-4-yl)-3,4-dihydro-2H-quinolin-1-yl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]cyclohexyl]ethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	CC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C(C(F)F)C(C1=CN(C)N=C1)=C3)=NN2C1CCC(CCN2CC3=C(C=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)C2)CC1	C45H49F2N9O5	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-RZSP3F	WO2022187417A1_CP-045	6-[2-[4-[5-acetyl-3-[7-(difluoromethyl)-6-(1-methylpyrazol-4-yl)-3,4-dihydro-2H-quinolin-1-yl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]cyclohexyl]ethyl]-2-(2,6-dioxopiperidin-3-yl)-7,8-dihydro-5H-pyrrolo[3,4-g]isoquinoline-1,3-dione	CC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C(C(F)F)C(C1=CN(C)N=C1)=C3)=NN2C1CCC(CCN2CCC3=C(C=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)C2)CC1	C46H51F2N9O5	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-XK5G5Q	WO2022187417A1_CP-046	.	CC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C(C(F)F)C(C1=CN(C)N=C1)=C3)=NN2[C@H]1CC[C@@H](CN2CC3=C(C=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)C2)CC1	C44H47F2N9O5	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-77WZXA	WO2022187417A1_CP-047	.	CC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C(C(F)F)C(C1=CN(C)N=C1)=C3)=NN2[C@H]1CC[C@H](CN2CC3=C(C=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)C2)CC1	C44H47F2N9O5	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-JAJRID	WO2022187417A1_CP-048	3-[6-[[4-[5-acetyl-3-[7-(difluoromethyl)-6-(1-methylpyrazol-4-yl)-3,4-dihydro-2H-quinolin-1-yl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]cyclohexyl]methyl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione	CC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C(C(F)F)C(C1=CN(C)N=C1)=C3)=NN2[C@H]1CC[C@H](CN2CC3=C(C=C4C(=O)N(C5CCC(=O)NC5=O)CC4=C3)C2)CC1	C44H49F2N9O4	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-AVAH6N	WO2022187417A1_CP-049	.	CC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C(C(F)F)C(C1=CN(C)N=C1)=C3)=NN2[C@H]1CC[C@H](CN2CCC3=C(C=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)C2)CC1	C45H49F2N9O5	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-ZNED2A	WO2022187417A1_CP-050	.	CC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C(C(F)F)C(C1=CN(C)N=C1)=C3)=NN2[C@H]1CC[C@@H](CN2CCC3=C(C=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)C2)CC1	C45H49F2N9O5	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-VY86TL	WO2022187417A1_CP-051	6-[2-[4-[5-acetyl-3-[7-(difluoromethyl)-6-(1-methylpyrazol-4-yl)-3,4-dihydro-2H-quinolin-1-yl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]cyclohexyl]propyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	CC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C(C(F)F)C(C1=CN(C)N=C1)=C3)=NN2C1CCC(C(C)CN2CC3=C(C=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)C2)CC1	C46H51F2N9O5	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-TRRILI	WO2022187417A1_CP-052	6-[[4-[5-acetyl-3-[7-(difluoromethyl)-6-(1-methylpyrazol-4-yl)-3,4-dihydro-2H-quinolin-1-yl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]piperidin-1-yl]methyl]-2-(2,6-dioxopiperidin-3-yl)-6,7-dihydro-5H-cyclopenta[f]isoindole-1,3-dione	CC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C(C(F)F)C(C1=CN(C)N=C1)=C3)=NN2C1CCN(CC2CC3=C(C=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)C2)CC1	C44H47F2N9O5	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-EBBIEL	WO2022187417A1_CP-053	6-[2-[4-[3-[7-(difluoromethyl)-6-(1-methylpyrazol-4-yl)-3,4-dihydro-2H-quinolin-1-yl]-5-(2-fluoroacetyl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]piperidin-1-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	CN1C=C(C2=CC3=C(C=C2C(F)F)N(C2=NN(C4CCN(C(=O)CN5CC6=CC7=C(C=C6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)C4=C2CN(C(=O)CF)CC4)CCC3)C=N1	C44H45F3N10O6	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-7DIZLQ	WO2022187417A1_CP-054	6-[2-[4-[5-(cyclopropanecarbonyl)-3-[7-(difluoromethyl)-6-(1-methylpyrazol-4-yl)-3,4-dihydro-2H-quinolin-1-yl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]piperidin-1-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	CN1C=C(C2=CC3=C(C=C2C(F)F)N(C2=NN(C4CCN(C(=O)CN5CC6=CC7=C(C=C6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)C4=C2CN(C(=O)C2CC2)CC4)CCC3)C=N1	C46H48F2N10O6	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-VUZSKL	WO2022187417A1_CP-055	6-[2-[4-[3-[7-(difluoromethyl)-6-(1-methylpyrazol-4-yl)-3,4-dihydro-2H-quinolin-1-yl]-5-propanoyl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]piperidin-1-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	CCC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C(C(F)F)C(C1=CN(C)N=C1)=C3)=NN2C1CCN(C(=O)CN2CC3=CC4=C(C=C3C2)C(=O)N(C2CCC(=O)NC2=O)C4=O)CC1	C45H48F2N10O6	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-20KKFA	WO2022187417A1_CP-056	6-[2-[4-[5-(2,2-difluoroacetyl)-3-[7-(difluoromethyl)-6-(1-methylpyrazol-4-yl)-3,4-dihydro-2H-quinolin-1-yl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]piperidin-1-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	CN1C=C(C2=CC3=C(C=C2C(F)F)N(C2=NN(C4CCN(C(=O)CN5CC6=CC7=C(C=C6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)C4=C2CN(C(=O)C(F)F)CC4)CCC3)C=N1	C44H44F4N10O6	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-HEUZ57	SCHEMBL27214138	6-[2-[4-[3-[7-(difluoromethyl)-6-(1-methylpyrazol-4-yl)-3,4-dihydro-2H-quinolin-1-yl]-4,5,6,7-tetrahydropyrazolo[4,3-c]pyridin-1-yl]piperidin-1-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	CN1C=C(C2=CC3=C(C=C2C(F)F)N(C2=NN(C4CCN(C(=O)CN5CC6=CC7=C(C=C6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)C4=C2CNCC4)CCC3)C=N1	C42H44F2N10O5	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-DVEAU9	WO2022187417A1_CP-058	6-[2-[4-[5-(2,2-difluoroethyl)-3-[7-(difluoromethyl)-6-(1-methylpyrazol-4-yl)-3,4-dihydro-2H-quinolin-1-yl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]piperidin-1-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	CN1C=C(C2=CC3=C(C=C2C(F)F)N(C2=NN(C4CCN(C(=O)CN5CC6=CC7=C(C=C6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)C4=C2CN(CC(F)F)CC4)CCC3)C=N1	C44H46F4N10O5	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-NPIEXE	WO2022187417A1_CP-059	6-[2-[4-[3-[7-(difluoromethyl)-6-(1-methylpyrazol-4-yl)-3,4-dihydro-2H-quinolin-1-yl]-5-(2,2-difluoropropyl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]piperidin-1-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	CN1C=C(C2=CC3=C(C=C2C(F)F)N(C2=NN(C4CCN(C(=O)CN5CC6=CC7=C(C=C6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)C4=C2CN(CC(C)(F)F)CC4)CCC3)C=N1	C45H48F4N10O5	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-9JP6XQ	WO2022187417A1_CP-060	6-[2-[4-[3-[7-(difluoromethyl)-6-(1-methylpyrazol-4-yl)-3,4-dihydro-2H-quinolin-1-yl]-5-(2,2,2-trifluoroethyl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]piperidin-1-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	CN1C=C(C2=CC3=C(C=C2C(F)F)N(C2=NN(C4CCN(C(=O)CN5CC6=CC7=C(C=C6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)C4=C2CN(CC(F)(F)F)CC4)CCC3)C=N1	C44H45F5N10O5	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-ALZJ46	WO2022187417A1_CP-061	6-[2-[4-[2-[(2S)-1-(3,4-difluorophenyl)-6-oxopiperidin-2-yl]-5-(3,5-dimethyl-1,2-oxazol-4-yl)benzimidazol-1-yl]piperidin-1-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	CC1=NOC(C)=C1C1=CC=C2C(=C1)N=C([C@@H]1CCCC(=O)N1C1=CC(F)=C(F)C=C1)N2C1CCN(C(=O)CN2CC3=C(C=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)C2)CC1	C45H42F2N8O7	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-JYLOI3	SCHEMBL27214137	3-[6-[2-[4-[2-[(2S)-1-(3,4-difluorophenyl)-6-oxopiperidin-2-yl]-5-(3,5-dimethyl-1,2-oxazol-4-yl)benzimidazol-1-yl]piperidin-1-yl]-2-oxoethyl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione	CC1=NOC(C)=C1C1=CC=C2C(=C1)N=C([C@@H]1CCCC(=O)N1C1=CC(F)=C(F)C=C1)N2C1CCN(C(=O)CN2CC3=C(C=C4C(=O)N(C5CCC(=O)NC5=O)CC4=C3)C2)CC1	C45H44F2N8O6	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-RVPKL5	WO2022187417A1_CP-063	6-[2-[4-[2-[(2S)-1-(3,4-difluorophenyl)-6-oxopiperidin-2-yl]-5-(3,5-dimethyl-1,2-oxazol-4-yl)benzimidazol-1-yl]piperidin-1-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-7,8-dihydro-5H-pyrrolo[3,4-g]isoquinoline-1,3-dione	CC1=NOC(C)=C1C1=CC=C2C(=C1)N=C([C@@H]1CCCC(=O)N1C1=CC(F)=C(F)C=C1)N2C1CCN(C(=O)CN2CCC3=C(C=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)C2)CC1	C46H44F2N8O7	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-8UBM8U	WO2022187417A1_CP-064	7-[2-[4-[2-[(2S)-1-(3,4-difluorophenyl)-6-oxopiperidin-2-yl]-5-(3,5-dimethyl-1,2-oxazol-4-yl)benzimidazol-1-yl]piperidin-1-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,6,8,9-tetrahydropyrrolo[3,4-h][3]benzazepine-1,3-dione	CC1=NOC(C)=C1C1=CC=C2C(=C1)N=C([C@@H]1CCCC(=O)N1C1=CC(F)=C(F)C=C1)N2C1CCN(C(=O)CN2CCC3=C(C=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)CC2)CC1	C47H46F2N8O7	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-I6C8H9	SCHEMBL27214136	6-[3-[4-[2-[(2S)-1-(3,4-difluorophenyl)-6-oxopiperidin-2-yl]-5-(3,5-dimethyl-1,2-oxazol-4-yl)benzimidazol-1-yl]piperidin-1-yl]-3-oxopropyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	CC1=NOC(C)=C1C1=CC=C2C(=C1)N=C([C@@H]1CCCC(=O)N1C1=CC(F)=C(F)C=C1)N2C1CCN(C(=O)CCN2CC3=C(C=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)C2)CC1	C46H44F2N8O7	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-BFXQ2G	WO2022187417A1_CP-066	6-[4-[4-[2-[(2S)-1-(3,4-difluorophenyl)-6-oxopiperidin-2-yl]-5-(3,5-dimethyl-1,2-oxazol-4-yl)benzimidazol-1-yl]piperidin-1-yl]-4-oxobutyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	CC1=NOC(C)=C1C1=CC=C2C(=C1)N=C([C@@H]1CCCC(=O)N1C1=CC(F)=C(F)C=C1)N2C1CCN(C(=O)CCCN2CC3=C(C=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)C2)CC1	C47H46F2N8O7	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-808VR7	WO2022187417A1_CP-067	6-[5-[4-[1-[5-acetyl-1-(oxan-4-yl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-3-yl]-7-(difluoromethyl)-3,4-dihydro-2H-quinolin-6-yl]pyrazol-1-yl]pentyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	CC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C(C(F)F)C(C1=CN(CCCCCN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)N=C1)=C3)=NN2C1CCOCC1	C46H51F2N9O6	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-MVVFI1	WO2022187417A1_CP-068	6-[4-[4-[1-[5-acetyl-1-(oxan-4-yl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-3-yl]-7-(difluoromethyl)-3,4-dihydro-2H-quinolin-6-yl]pyrazol-1-yl]butyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	CC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C(C(F)F)C(C1=CN(CCCCN4CC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)N=C1)=C3)=NN2C1CCOCC1	C45H49F2N9O6	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-SQEJS6	WO2022187417A1_CP-069	6-[5-[4-[1-[5-acetyl-1-(oxan-4-yl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-3-yl]-7-(difluoromethyl)-3,4-dihydro-2H-quinolin-6-yl]pyrazol-1-yl]pentyl]-2-(2,6-dioxopiperidin-3-yl)-7,8-dihydro-5H-pyrrolo[3,4-g]isoquinoline-1,3-dione	CC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C(C(F)F)C(C1=CN(CCCCCN4CCC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)N=C1)=C3)=NN2C1CCOCC1	C47H53F2N9O6	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-1RE1K6	WO2022187417A1_CP-070	6-[4-[4-[1-[5-acetyl-1-(oxan-4-yl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-3-yl]-7-(difluoromethyl)-3,4-dihydro-2H-quinolin-6-yl]pyrazol-1-yl]butyl]-2-(2,6-dioxopiperidin-3-yl)-7,8-dihydro-5H-pyrrolo[3,4-g]isoquinoline-1,3-dione	CC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C(C(F)F)C(C1=CN(CCCCN4CCC5=CC6=C(C=C5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)N=C1)=C3)=NN2C1CCOCC1	C46H51F2N9O6	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-J2HNMZ	WO2022187417A1_CP-071	6-[2-[4-[4-[1-[5-acetyl-1-(oxan-4-yl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-3-yl]-7-(difluoromethyl)-3,4-dihydro-2H-quinolin-6-yl]pyrazol-1-yl]piperidin-1-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-7,8-dihydro-5H-pyrrolo[3,4-g]isoquinoline-1,3-dione	CC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C(C(F)F)C(C1=CN(C4CCN(C(=O)CN5CCC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)N=C1)=C3)=NN2C1CCOCC1	C49H54F2N10O7	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-L78EXD	WO2022187417A1_CP-072	.	CC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C(C(F)F)C(C1=CN(C4CCN(C(=O)CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)N=C1)=C3)=NN2C1CCOCC1	C48H52F2N10O7	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-0DI0T5	WO2022187417A1_CP-073	6-[3-[4-[1-[5-acetyl-1-(oxan-4-yl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-3-yl]-7-(difluoromethyl)-3,4-dihydro-2H-quinolin-6-yl]pyrazol-1-yl]propyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	CC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C(C(F)F)C(C1=CN(CCCN4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)N=C1)=C3)=NN2C1CCOCC1	C44H47F2N9O6	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-68MM0P	WO2022187417A1_CP-074	.	CC(=O)C1CCC2=C(C1)C(N1CCCC3=C1C=C(C(F)F)C(C1=CN(CCCN4CCC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)N=C1)=C3)=NN2C1CCOCC1	C46H50F2N8O6	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-NFCXEX	WO2022187417A1_CP-075	6-[2-[4-(5-acetyl-3-naphthalen-1-yl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl)piperidin-1-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	CC(=O)N1CCC2=C(C1)C(C1=CC=CC3=C1C=CC=C3)=NN2C1CCN(C(=O)CN2CC3=C(C=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)C2)CC1	C40H39N7O6	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-5KTEXU	WO2022187417A1_CP-076	6-[2-[4-(5-acetyl-3-naphthalen-1-yl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl)piperidin-1-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-7,8-dihydro-5H-pyrrolo[3,4-g]isoquinoline-1,3-dione	CC(=O)N1CCC2=C(C1)C(C1=CC=CC3=C1C=CC=C3)=NN2C1CCN(C(=O)CN2CCC3=C(C=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)C2)CC1	C41H41N7O6	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-2GWLR1	WO2022187417A1_CP-077	6-[2-[4-[5-acetyl-3-(3,4,6,7,8,9-hexahydro-2H-benzo[g]quinolin-1-yl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]piperidin-1-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	CC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C1CCCCC1=C3)=NN2C1CCN(C(=O)CN2CC3=C(C=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)C2)CC1	C43H48N8O6	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-PIKVPT	WO2022187417A1_CP-078	6-[2-[4-[5-acetyl-3-(3,4,6,7,8,9-hexahydro-2H-benzo[g]quinolin-1-yl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]piperidin-1-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-7,8-dihydro-5H-pyrrolo[3,4-g]isoquinoline-1,3-dione	CC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C1CCCCC1=C3)=NN2C1CCN(C(=O)CN2CCC3=C(C=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)C2)CC1	C44H50N8O6	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-XEFKZB	WO2022187417A1_CP-079	6-[2-[4-[5-acetyl-3-(9-methyl-3,4,6,7,8,9-hexahydro-2H-benzo[g]quinolin-1-yl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]piperidin-1-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	CC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C1C(=C3)CCCC1C)=NN2C1CCN(C(=O)CN2CC3=C(C=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)C2)CC1	C44H50N8O6	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-UII9IC	WO2022187417A1_CP-080	6-[2-[4-[5-acetyl-3-(7-acetyl-2,3,4,6,8,9-hexahydropyrido[3,4-g]quinolin-1-yl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]piperidin-1-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	CC(=O)N1CCC2=CC3=C(C=C2C1)CCCN3C1=NN(C2CCN(C(=O)CN3CC4=C(C=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)C3)CC2)C2=C1CN(C(C)=O)CC2	C44H49N9O7	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-S0EH0C	WO2022187417A1_CP-081	6-[2-[4-[5-acetyl-3-(3-acetyl-1,2,4,8,9,10-hexahydro-3,7-phenanthrolin-7-yl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]piperidin-1-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	CC(=O)N1CCC2=C(C=CC3=C2CCCN3C2=NN(C3CCN(C(=O)CN4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C3=C2CN(C(C)=O)CC3)C1	C44H49N9O7	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-A74BY9	WO2022187417A1_CP-082	6-[2-[4-(5-acetyl-3-isoquinolin-8-yl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl)piperidin-1-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	CC(=O)N1CCC2=C(C1)C(C1=CC=CC3=C1C=NC=C3)=NN2C1CCN(C(=O)CN2CC3=C(C=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)C2)CC1	C39H38N8O6	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-T2J6MJ	WO2022187417A1_CP-083	6-[2-[4-[5-acetyl-3-(9,9-dimethyl-2,3,4,6,7,8-hexahydrobenzo[g]quinolin-1-yl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]piperidin-1-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	CC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C1C(=C3)CCCC1(C)C)=NN2C1CCN(C(=O)CN2CC3=C(C=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)C2)CC1	C45H52N8O6	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-PJC3ZX	WO2022187417A1_CP-084	6-[2-[4-[5-acetyl-3-[7-(difluoromethyl)-6-(1-methylpyrazol-4-yl)-3,4-dihydro-2H-quinolin-1-yl]-7,7-dimethyl-4,6-dihydropyrazolo[4,3-c]pyridin-1-yl]piperidin-1-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	CC(=O)N1CC2=C(N(C3CCN(C(=O)CN4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)N=C2N2CCCC3=C2C=C(C(F)F)C(C2=CN(C)N=C2)=C3)C(C)(C)C1	C46H50F2N10O6	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-WRX3RW	WO2022187417A1_CP-085	6-[2-[4-[5-acetyl-3-[7-(difluoromethyl)-6-(2-methylpyrazol-3-yl)-3,4-dihydro-2H-quinolin-1-yl]-7,7-dimethyl-4,6-dihydropyrazolo[4,3-c]pyridin-1-yl]piperidin-1-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	CC(=O)N1CC2=C(N(C3CCN(C(=O)CN4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)N=C2N2CCCC3=C2C=C(C(F)F)C(C2=CC=NN2C)=C3)C(C)(C)C1	C46H50F2N10O6	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-BKRI9U	WO2022187417A1_CP-086	1'-[4-[5-acetyl-3-[7-(difluoromethyl)-6-(1-methylpyrazol-4-yl)-3,4-dihydro-2H-quinolin-1-yl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]cyclohexyl]-2-(2,6-dioxopiperidin-3-yl)spiro[5,7-dihydrocyclopenta[f]isoindole-6,3'-azetidine]-1,3-dione	CC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C(C(F)F)C(C1=CN(C)N=C1)=C3)=NN2C1CCC(N2CC3(CC4=C(C=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)C3)C2)CC1	C46H49F2N9O5	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-G6DW03	WO2022187417A1_CP-087	8-[4-[5-acetyl-3-[7-(difluoromethyl)-6-(1-methylpyrazol-4-yl)-3,4-dihydro-2H-quinolin-1-yl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]cyclohexyl]-2-(2,6-dioxopiperidin-3-yl)-7,9-dihydro-6H-pyrrolo[3,4-h]isoquinoline-1,3-dione	CC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C(C(F)F)C(C1=CN(C)N=C1)=C3)=NN2C1CCC(N2CCC3=CC=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3C2)CC1	C44H47F2N9O5	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-ZF2FLE	WO2022187417A1_CP-088	1'-[[4-[5-acetyl-3-[7-(difluoromethyl)-6-(1-methylpyrazol-4-yl)-3,4-dihydro-2H-quinolin-1-yl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]cyclohexyl]methyl]-2-(2,6-dioxopiperidin-3-yl)spiro[5,7-dihydrocyclopenta[f]isoindole-6,3'-azetidine]-1,3-dione	CC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C(C(F)F)C(C1=CN(C)N=C1)=C3)=NN2[C@H]1CC[C@H](CN2CC3(CC4=C(C=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)C3)C2)CC1	C47H51F2N9O5	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-5WM7JC	WO2022187417A1_CP-089	8-[[4-[5-acetyl-3-[7-(difluoromethyl)-6-(1-methylpyrazol-4-yl)-3,4-dihydro-2H-quinolin-1-yl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]cyclohexyl]methyl]-2-(2,6-dioxopiperidin-3-yl)-7,9-dihydro-6H-pyrrolo[3,4-h]isoquinoline-1,3-dione	CC(=O)N1CCC2=C(C1)C(N1CCCC3=C1C=C(C(F)F)C(C1=CN(C)N=C1)=C3)=NN2[C@H]1CC[C@H](CN2CCC3=CC=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3C2)CC1	C45H49F2N9O5	CBP;P300	Q92793/Q09472	CRBN	WO-2022187417-A1
TPD-BHX2T2	WO2022187419A1_1	2-chloro-4-[(3S)-8-[4-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperazin-1-yl]sulfonylphenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(S(=O)(=O)N4CCN(C5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H49ClN8O6S	AR	P10275	CRBN	WO-2022187419-A1
TPD-25VH4L	WO2022187419A1_10	.	C[C@H]1CC2(CCN(c3ccc(CN4CCN(C5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)c(F)c3)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H50ClFN8O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-N05KYH	WO2022187419A1_100	.	C[C@H]1CC2(CCN(c3ccc(N4CCC(N5CC(Oc6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)nn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C41H44ClN9O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-LCXAFT	WO2022187419A1_101	2-chloro-4-[(3S)-8-[2-[4-[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxyazetidin-1-yl]piperidin-1-yl]pyrimidin-5-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3cnc(N4CCC(N5CC(Oc6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C41H44ClN9O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-HGJDVC	WO2022187419A1_102	.	C[C@H]1CC2(CCN(c3cnc(N4CCC(N5CC(Oc6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C41H44ClN9O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-UE0O2G	WO2022187419A1_103	.	C[C@H]1CC2(CCN(c3ncc(N4CCC(N5CC(Oc6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C41H44ClN9O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-SWT9PN	WO2022187419A1_104	2-chloro-4-[(3S)-8-[4-[4-[3-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]amino]azetidin-1-yl]piperidin-1-yl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(N4CCC(N5CC(Nc6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H47ClN8O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-0E9VGV	WO2022187419A1_105	2-chloro-4-[(3S)-8-[6-[4-[3-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]amino]azetidin-1-yl]piperidin-1-yl]pyridin-3-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(N4CCC(N5CC(Nc6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H46ClN9O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-M5IVPA	WO2022187419A1_106	.	C[C@H]1CC2(CCN(c3ccc(N4CCC(N5CC(Nc6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H46ClN9O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-QJ9NK1	WO2022187419A1_107	.	C[C@H]1CC2(CCN(c3ccc(N4CCC(N5CC(Nc6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)nn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C41H45ClN10O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-PXRKF4	WO2022187419A1_108	2-chloro-4-[(3S)-8-[2-[4-[3-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]amino]azetidin-1-yl]piperidin-1-yl]pyrimidin-5-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3cnc(N4CCC(N5CC(Nc6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C41H45ClN10O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-1PCXM0	WO2022187419A1_109	.	C[C@H]1CC2(CCN(c3cnc(N4CCC(N5CC(Nc6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C41H45ClN10O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-XR3VMJ	WO2022187419A1_11	.	C[C@H]1CC2(CCN(c3ccc(CC(=O)N4CCC(N5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H46ClN7O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-2VLM05	WO2022187419A1_110	.	C[C@H]1CC2(CCN(c3ncc(N4CCC(N5CC(Nc6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C41H45ClN10O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-OKI96Q	WO2022187419A1_111	2-chloro-4-[(3S)-8-[4-[4-[3-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-methylamino]azetidin-1-yl]piperidin-1-yl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(N4CCC(N5CC(N(C)c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H49ClN8O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-9JGBUK	WO2022187419A1_112	.	C[C@H]1CC2(CCN(c3ccc(N4CCC(N5CC(N(C)c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H48ClN9O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-O9385F	WO2022187419A1_113	.	C[C@H]1CC2(CCN(c3ccc(N4CCC(N5CC(N(C)c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H48ClN9O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-R34BPI	WO2022187419A1_114	.	C[C@H]1CC2(CCN(c3ccc(N4CCC(N5CC(N(C)c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)nn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H47ClN10O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-I32MTO	WO2022187419A1_115	.	C[C@H]1CC2(CCN(c3cnc(N4CCC(N5CC(N(C)c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H47ClN10O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-V3B09A	WO2022187419A1_116	.	C[C@H]1CC2(CCN(c3cnc(N4CCC(N5CC(N(C)c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H47ClN10O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-SOMZDF	WO2022187419A1_117	.	C[C@H]1CC2(CCN(c3ncc(N4CCC(N5CC(N(C)c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H47ClN10O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-OTKQQJ	WO2022187419A1_118	.	C[C@H]1CC2(CCN(c3nnc(N4CCC(N5CC(N(C)c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)nn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C40H45ClN12O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-LJUBB9	SCHEMBL27241113	2-chloro-4-[(3S)-8-[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]-methylamino]piperidin-1-yl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(N4CCC(N(C)C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H49ClN8O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-UUV9UB	WO2022187419A1_12	.	C[C@H]1CC2(CCN(c3ccc(CC(=O)N4CCC(CN5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H48ClN7O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-8QGRAK	WO2022187419A1_120	2-chloro-4-[(3S)-8-[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]amino]piperidin-1-yl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(N4CCC(NC5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H47ClN8O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-ZZHLLD	WO2022187419A1_121	2-chloro-4-[(3S)-8-[4-[3-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]-methylamino]azetidin-1-yl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(N4CC(N(C)C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)C4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H45ClN8O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-QKDTIA	WO2022187419A1_123	2-chloro-4-[(3S)-8-[5-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]-methylamino]piperidin-1-yl]pyridin-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(N4CCC(N(C)C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H48ClN9O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-Y3HBOY	WO2022187419A1_124	2-chloro-4-[(3S)-8-[6-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]-methylamino]piperidin-1-yl]pyridin-3-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(N4CCC(N(C)C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H48ClN9O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-UHCEBD	WO2022187419A1_125	2-chloro-4-[(3S)-8-[6-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]-methylamino]piperidin-1-yl]pyridazin-3-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(N4CCC(N(C)C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)nn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H47ClN10O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-549KVW	WO2022187419A1_128	2-chloro-4-[(3S)-8-[6-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]amino]piperidin-1-yl]pyridazin-3-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(N4CCC(NC5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)nn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C41H45ClN10O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-09QQRR	WO2022187419A1_129	.	C[C@H]1CC2(CCN(c3ccc(N4CC(N(C)C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)C4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C41H44ClN9O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-GLO7Y3	WO2022187419A1_13	.	COC1(CN2Cc3cc4c(cc3C2)C(=O)N(C2CCC(=O)NC2=O)C4=O)CCN(C(=O)c2ccc(N3CCC4(CC3)C[C@H](C)N(c3ccc(C#N)c(F)c3)C4)cc2)CC1	C45H48FN7O6	AR	P10275	CRBN	WO-2022187419-A1
TPD-55XH4Z	WO2022187419A1_130	2-chloro-4-[(3S)-8-[6-[3-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]-methylamino]azetidin-1-yl]pyridazin-3-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(N4CC(N(C)C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)C4)nn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C40H43ClN10O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-SC34OG	WO2022187419A1_131	2-chloro-4-[(3S)-8-[4-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperidin-4-yl]oxyphenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(OC4CCN(C5CN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H45ClFN7O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-C5QLY5	WO2022187419A1_132	2-chloro-4-[(3S)-8-[5-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperidin-4-yl]oxypyridin-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(OC4CCN(C5CN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H44ClFN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-6LNSGJ	WO2022187419A1_133	.	C[C@H]1CC2(CCN(c3ccc(OC4CCN(C5CN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H44ClFN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-ZPA711	WO2022187419A1_134	.	C[C@H]1CC2(CCN(c3ccc(OC4CCN(C5CN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)nn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C41H43ClFN9O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-4XCF5K	WO2022187419A1_135	2-chloro-4-[(3S)-8-[5-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperazine-1-carbonyl]thiophen-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)s3)CC2)CN1c1ccc(C#N)c(Cl)c1	C41H43ClN8O5S	AR	P10275	CRBN	WO-2022187419-A1
TPD-362CDP	WO2022187419A1_136	.	C[C@H]1CC2(CCN(c3ncc(C(=O)N4CCN(C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)s3)CC2)CN1c1ccc(C#N)c(Cl)c1	C40H42ClN9O5S	AR	P10275	CRBN	WO-2022187419-A1
TPD-SFYJSX	WO2022187419A1_137	2-chloro-4-[(3S)-8-[2-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperazine-1-carbonyl]-1,3-thiazol-5-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3cnc(C(=O)N4CCN(C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)s3)CC2)CN1c1ccc(C#N)c(Cl)c1	C40H42ClN9O5S	AR	P10275	CRBN	WO-2022187419-A1
TPD-OOO22Y	WO2022187419A1_138	2-chloro-4-[(3S)-8-[5-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]piperidine-1-carbonyl]thiophen-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(N5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)s3)CC2)CN1c1ccc(C#N)c(Cl)c1	C41H42ClN7O5S	AR	P10275	CRBN	WO-2022187419-A1
TPD-CTIRTE	WO2022187419A1_139	.	C[C@H]1CC2(CCN(c3ncc(C(=O)N4CCC(N5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)s3)CC2)CN1c1ccc(C#N)c(Cl)c1	C40H41ClN8O5S	AR	P10275	CRBN	WO-2022187419-A1
TPD-8N4QE2	WO2022187419A1_14	.	C[C@H]1CC2(CCN(c3ccc(C4CCN(CC(=O)N5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H46ClN7O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-H5MUHB	WO2022187419A1_140	2-chloro-4-[(3S)-8-[4-[4-[1-[3-(2,6-dioxopiperidin-3-yl)-1-methyl-2-oxobenzimidazol-5-yl]azetidin-3-yl]piperazine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(C5CN(c6ccc7c(c6)n(C6CCC(=O)NC6=O)c(=O)n7C)C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H48ClN9O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-ZE04LJ	WO2022187419A1_141	2-chloro-4-[(3S)-8-[4-[4-[1-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]azetidin-3-yl]piperazine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(C5CN(c6ccc7c(c6)n(C)c(=O)n7C6CCC(=O)NC6=O)C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H48ClN9O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-X4E9UE	WO2022187419A1_142	2-chloro-4-[(3S)-8-[4-[4-[1-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-4-yl]azetidin-3-yl]piperazine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(C5CN(c6cccc7c6n(C)c(=O)n7C6CCC(=O)NC6=O)C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H48ClN9O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-Y0DSY7	SCHEMBL27241108	2-chloro-4-[(3S)-8-[4-[4-[1-[6-(2,6-dioxopiperidin-3-yl)-5,7-dioxopyrrolo[3,4-b]pyridin-3-yl]piperidin-4-yl]piperazine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL30069550; SCHEMBL30069551	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(C5CCN(c6cnc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H48ClN9O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-1N2R6J	WO2022187419A1_144	2-chloro-4-[(3S)-8-[4-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxopyrrolo[3,4-c]pyridin-6-yl]piperidin-4-yl]piperazine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(C5CCN(c6cc7c(cn6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H48ClN9O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-88F1KR	WO2022187419A1_145	2-chloro-4-[(3S)-8-[4-[4-[1-[6-(2,6-dioxopiperidin-3-yl)-5,7-dioxopyrrolo[3,4-b]pyridin-2-yl]piperidin-4-yl]piperazine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(C5CCN(c6ccc7c(n6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H48ClN9O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-XW0Y1U	WO2022187419A1_146	2-chloro-4-[(3S)-8-[4-[4-[1-[6-(2,6-dioxopiperidin-3-yl)-5,7-dioxopyrrolo[3,4-d]pyrimidin-2-yl]piperidin-4-yl]piperazine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(C5CCN(c6ncc7c(n6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H47ClN10O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-CC5W5G	SCHEMBL27241123	2-chloro-4-[(3S)-8-[4-[1-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]-2-oxoethyl]piperidine-4-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)C4CCN(CC(=O)N5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H46ClN7O6	AR	P10275	CRBN	WO-2022187419-A1
TPD-3Q1UAM	SCHEMBL27241119	2-chloro-4-[(3S)-8-[4-[1-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]acetyl]piperidine-4-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)C4CCN(C(=O)CN5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H46ClN7O6	AR	P10275	CRBN	WO-2022187419-A1
TPD-64GYE0	WO2022187419A1_149	2-chloro-4-[(3S)-8-[4-[1-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]acetyl]azetidin-3-yl]sulfonylphenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(S(=O)(=O)C4CN(C(=O)CN5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H42ClN7O7S	AR	P10275	CRBN	WO-2022187419-A1
TPD-C2FCE8	WO2022187419A1_15	.	C[C@H]1CC2(CCN(c3ccc(C4CCN(C(=O)CN5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H46ClN7O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-HPBCT6	WO2022187419A1_150	2-chloro-4-[(3S)-8-[4-[1-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]acetyl]azetidine-3-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)C4CN(C(=O)CN5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H42ClN7O6	AR	P10275	CRBN	WO-2022187419-A1
TPD-ABT8MM	WO2022187419A1_151	2-chloro-4-[(3S)-8-[4-[1-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]-2-oxoethyl]piperidin-4-yl]sulfonylphenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(S(=O)(=O)C4CCN(CC(=O)N5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H46ClN7O7S	AR	P10275	CRBN	WO-2022187419-A1
TPD-ZXFVBU	WO2022187419A1_152	.	C[C@H]1CC2(CCN(c3ccc(S(=O)(=O)C4CCN(C(=O)CN5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H46ClN7O7S	AR	P10275	CRBN	WO-2022187419-A1
TPD-P4I55T	SCHEMBL27241130	2-chloro-4-[(3S)-8-[5-[[4-[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperazin-1-yl]methyl]pyridin-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(CN4CCN(C5CN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H45ClFN9O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-P4W63E	WO2022187419A1_154	.	C[C@H]1CC2(CCN(c3ccc(CN4CCN(C5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H50ClN9O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-TF3MAK	SCHEMBL23125284	2-chloro-4-[(3S)-8-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindole-6-carbonyl]piperidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(C(=O)N5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H44ClN7O6	AR	P10275	CRBN	WO-2022187419-A1
TPD-MF6R8A	WO2022187419A1_156	2-chloro-4-[(3S)-8-[5-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindole-6-carbonyl]piperidine-1-carbonyl]pyridin-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(C(=O)N5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H43ClN8O6	AR	P10275	CRBN	WO-2022187419-A1
TPD-JJLUXP	WO2022187419A1_157	2-chloro-4-[(3S)-8-[6-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindole-6-carbonyl]piperidine-1-carbonyl]pyridin-3-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(C(=O)N5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H43ClN8O6	AR	P10275	CRBN	WO-2022187419-A1
TPD-LCMT6B	WO2022187419A1_158	2-chloro-4-[(3S)-8-[4-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]acetyl]piperidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(C(=O)CN5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H46ClN7O6	AR	P10275	CRBN	WO-2022187419-A1
TPD-OO6BAM	WO2022187419A1_159	2-chloro-4-[(3S)-8-[5-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]acetyl]piperidine-1-carbonyl]pyridin-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(C(=O)CN5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H45ClN8O6	AR	P10275	CRBN	WO-2022187419-A1
TPD-O48N7K	WO2022187419A1_16	.	C[C@H]1CC2(CCN(c3ccc(CN4CCC(C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H48ClN7O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-JVZDK3	WO2022187419A1_160	2-chloro-4-[(3S)-8-[6-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]acetyl]piperidine-1-carbonyl]pyridin-3-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(C(=O)CN5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H45ClN8O6	AR	P10275	CRBN	WO-2022187419-A1
TPD-7TPJJR	WO2022187419A1_161	2-chloro-4-[(3S)-8-[4-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperidin-4-yl]sulfonylphenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(S(=O)(=O)C4CCN(C5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H50ClN7O6S	AR	P10275	CRBN	WO-2022187419-A1
TPD-H7ATR6	WO2022187419A1_162	2-chloro-4-[(3S)-8-[4-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperidin-4-yl]sulfonylphenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(S(=O)(=O)C4CCN(CC5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C46H52ClN7O6S	AR	P10275	CRBN	WO-2022187419-A1
TPD-20GQEL	WO2022187419A1_163	2-chloro-4-[(3S)-8-[4-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperidin-4-yl]sulfonylphenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(S(=O)(=O)C4CCN(C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H46ClN7O6S	AR	P10275	CRBN	WO-2022187419-A1
TPD-WZZLL7	WO2022187419A1_164	2-chloro-4-[(3S)-8-[4-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]methyl]piperidin-4-yl]sulfonylphenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(S(=O)(=O)C4CCN(CC5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H48ClN7O6S	AR	P10275	CRBN	WO-2022187419-A1
TPD-GYYGY1	WO2022187419A1_165	2-chloro-4-[(3S)-8-[5-[[4-[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperazin-1-yl]methyl]pyridin-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(CN4CCN(C5CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H49ClFN9O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-OA553Q	WO2022187419A1_166	2-chloro-4-[(3S)-8-[5-[[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]piperidin-1-yl]methyl]pyridin-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(CN4CCC(N5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H50ClN9O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-7ZNX9J	WO2022187419A1_167	2-chloro-4-[(3S)-8-[5-[[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperazin-1-yl]methyl]pyridin-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(CN4CCN(C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H46ClN9O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-AL7ARM	WO2022187419A1_168	2-chloro-4-[(3S)-8-[5-[[4-[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]piperidin-1-yl]methyl]pyridin-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(CN4CCC(N5CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H49ClFN9O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-1AFY66	SCHEMBL27241097	2-chloro-4-[(3S)-8-[6-[[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperazin-1-yl]methyl]pyridin-3-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL30069547	C[C@H]1CC2(CCN(c3ccc(CN4CCN(C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H46ClN9O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-T92TZJ	WO2022187419A1_17	.	C[C@H]1CC2(CCN(c3ccc(CN4CCC(C5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C46H52ClN7O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-MQ9WX8	SCHEMBL27241110	2-chloro-4-[(3S)-8-[2-[[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperazin-1-yl]methyl]pyrimidin-5-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3cnc(CN4CCN(C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C41H45ClN10O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-LVMLQV	WO2022187419A1_171	2-chloro-4-[(3S)-8-[2-[[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperazin-1-yl]methyl]pyrimidin-5-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3cnc(CN4CCN(C5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H49ClN10O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-CX4LXK	WO2022187419A1_172	2-chloro-4-[(3S)-8-[6-[[4-[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperazin-1-yl]methyl]pyridin-3-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(CN4CCN(C5CN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H45ClFN9O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-STDA20	WO2022187419A1_173	2-chloro-4-[(3S)-8-[6-[[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperazin-1-yl]methyl]pyridazin-3-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(CN4CCN(C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)nn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C41H45ClN10O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-RX2E0O	WO2022187419A1_174	2-chloro-4-[(3S)-8-[6-[[4-[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperazin-1-yl]methyl]pyridazin-3-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(CN4CCN(C5CN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)nn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C41H44ClFN10O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-SLFAOR	WO2022187419A1_175	2-chloro-4-[(3S)-8-[2-[[4-[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperazin-1-yl]methyl]pyrimidin-5-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3cnc(CN4CCN(C5CN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C41H44ClFN10O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-771MNU	WO2022187419A1_176	2-chloro-4-[(3S)-8-[5-[[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperidin-1-yl]methyl]pyridin-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(CN4CCC(C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H47ClN8O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-65W42F	WO2022187419A1_177	2-chloro-4-[(3S)-8-[6-[[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperidin-1-yl]methyl]pyridin-3-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(CN4CCC(C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H47ClN8O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-LAL0GY	WO2022187419A1_178	2-chloro-4-[(3S)-8-[5-[[3-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]azetidin-1-yl]methyl]pyridin-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(CN4CC(C5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H47ClN8O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-6JF9S1	WO2022187419A1_179	2-chloro-4-[(3S)-8-[6-[[3-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]azetidin-1-yl]methyl]pyridin-3-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(CN4CC(C5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H47ClN8O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-R704FJ	WO2022187419A1_18	.	C[C@H]1CC2(CCN(c3ccc(CN4CCN(C5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H51ClN8O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-6WGEDO	SCHEMBL27241096	2-chloro-4-[(3S)-8-[5-[[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperidin-1-yl]methyl]pyridin-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(CN4CCC(C5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H51ClN8O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-CQTD5Q	WO2022187419A1_181	2-chloro-4-[(3S)-8-[6-[[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperidin-1-yl]methyl]pyridin-3-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(CN4CCC(C5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H51ClN8O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-C5BE3R	WO2022187419A1_182	2-chloro-4-[(3S)-8-[6-[[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperazin-1-yl]methyl]pyridin-3-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(CN4CCN(C5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H50ClN9O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-YD7A6T	WO2022187419A1_183	2-chloro-4-[(3S)-8-[5-[[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperazin-1-yl]methyl]pyrimidin-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ncc(CN4CCN(C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C41H45ClN10O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-V729PY	WO2022187419A1_184	2-chloro-4-[(3S)-8-[5-[[4-[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperazin-1-yl]methyl]pyrimidin-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ncc(CN4CCN(C5CN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C41H44ClFN10O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-JYBCBW	WO2022187419A1_185	2-chloro-4-[(3S)-8-[5-[[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperazin-1-yl]methyl]pyrazin-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3cnc(CN4CCN(C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C41H45ClN10O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-IY7UWE	WO2022187419A1_186	.	C[C@H]1CC2(CCN(c3cnc(CN4CCN(C5CN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C41H44ClFN10O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-3WUB5T	WO2022187419A1_187	.	C[C@H]1CC2(CCN(c3ccc(CN4CCC(C(=O)N5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H45ClN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-2LYFHB	WO2022187419A1_188	.	C[C@H]1CC2(CCN(c3ccc(CN4CCC(C(=O)N5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H45ClN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-KC1F5Q	WO2022187419A1_189	.	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(C5CCN(c6cnc7c(n6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H47ClN10O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-SWX50O	WO2022187419A1_19	.	C[C@H]1CC2(CCN(c3ccc(CN4CCC(N5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H46ClN7O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-5VKD83	WO2022187419A1_190	.	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(CC5CCN(c6cnc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H50ClN9O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-Z26UZ0	WO2022187419A1_191	.	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(CC5CCN(c6cc7c(cn6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H50ClN9O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-CCA5KZ	WO2022187419A1_192	.	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(CC5CCN(c6ccc7c(n6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H50ClN9O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-IYN17M	WO2022187419A1_193	.	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(CC5CCN(c6ncc7c(n6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H49ClN10O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-AAR4FR	WO2022187419A1_194	.	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(N5CCOc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H46ClN7O6	AR	P10275	CRBN	WO-2022187419-A1
TPD-SAFKG9	WO2022187419A1_195	.	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(CN5CCOc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H48ClN7O6	AR	P10275	CRBN	WO-2022187419-A1
TPD-2E4AIS	WO2022187419A1_196	.	C[C@H]1CC2(CCN(c3ccc(CC4CCN(C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H47ClN8O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-BX4TMA	WO2022187419A1_197	.	C[C@H]1CC2(CCN(c3ccc(CC4CCN(C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H47ClN8O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-V1P3AH	WO2022187419A1_198	.	C[C@H]1CC2(CCN(c3ccc(CC4CCN(C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)nn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H46ClN9O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-Z373EI	WO2022187419A1_199	.	C[C@H]1CC2(CCN(c3ncc(CC4CCN(C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H46ClN9O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-O4OGEM	WO2022187419A1_2	.	C[C@H]1CC2(CCN(c3ccc(S(=O)(=O)N4CCN(C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H45ClN8O6S	AR	P10275	CRBN	WO-2022187419-A1
TPD-1G1UYQ	WO2022187419A1_20	.	C[C@H]1CC2(CCN(c3ccc(CN4CCC(CN5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H48ClN7O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-14D2NC	WO2022187419A1_200	.	C[C@H]1CC2(CCN(c3cnc(CC4CCN(C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H46ClN9O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-3A71MB	WO2022187419A1_201	.	C[C@H]1CC2(CCN(c3cnc(CC4CCN(C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H46ClN9O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-PZHFZD	WO2022187419A1_202	.	C[C@H]1CC2(CCN(c3ccc(CN4CCC(N5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)nn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H49ClN10O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-M5E79H	WO2022187419A1_203	.	C[C@H]1CC2(CCN(c3ccc(CN4CCC(N5CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)nn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H48ClFN10O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-CWVEMP	WO2022187419A1_204	.	C[C@H]1CC2(CCN(c3ccc(CN4CC(N5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H46ClN9O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-YOEOBQ	WO2022187419A1_205	.	C[C@H]1CC2(CCN(c3ccc(CN4CC(N5CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H45ClFN9O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-L6Z7EZ	SCHEMBL27241114	2-chloro-4-[(3S)-8-[4-[4-[3-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]amino]azetidin-1-yl]piperidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(N5CC(Nc6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H47ClN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-25RZD9	SCHEMBL27241106	2-chloro-4-[(3S)-8-[4-[4-[3-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-methylamino]azetidin-1-yl]piperidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(N5CC(N(C)c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H49ClN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-DH8W1K	WO2022187419A1_208	2-chloro-4-[(3S)-8-[4-[4-[3-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]amino]-3-methylazetidin-1-yl]piperidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(N5CC(C)(Nc6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H49ClN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-NB9TS2	WO2022187419A1_209	2-chloro-4-[(3S)-8-[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]-methylamino]piperidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(N(C)C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H49ClN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-E6GRXJ	WO2022187419A1_21	.	C[C@H]1CC2(CCN(c3ccc(C4CCN(CC5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H48ClN7O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-2HBW67	WO2022187419A1_210	.	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(CC5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H48ClN7O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-4YNL4A	WO2022187419A1_211	2-chloro-4-[(3S)-8-[4-[4-[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxyazetidin-1-yl]piperidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(N5CC(Oc6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H46ClN7O6	AR	P10275	CRBN	WO-2022187419-A1
TPD-NOSSDU	WO2022187419A1_212	2-chloro-4-[(3S)-8-[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]amino]piperidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(NC5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H47ClN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-H0YGBJ	WO2022187419A1_213	2-chloro-4-[(3S)-8-[4-[3-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]amino]azetidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CC(NC5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)C4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H43ClN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-C16REG	WO2022187419A1_214	2-chloro-4-[(3S)-8-[4-[3-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]-methylamino]azetidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CC(N(C)C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)C4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H45ClN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-XJVDHR	WO2022187419A1_215	2-chloro-4-[(3S)-8-[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-3-methylazetidin-3-yl]amino]piperidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(NC5(C)CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H49ClN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-FD9LPS	WO2022187419A1_216	2-chloro-4-[(3S)-8-[4-[3-[3-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-methylamino]azetidin-1-yl]azetidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CC(N5CC(N(C)c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)C4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H45ClN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-EZSGCO	WO2022187419A1_217	2-chloro-4-[(3S)-8-[4-[3-[3-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]amino]azetidin-1-yl]azetidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CC(N5CC(Nc6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)C4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H43ClN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-YAMOFK	WO2022187419A1_218	.	C[C@H]1CC2(CCN(c3ccc(CN4CCC(N5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H51ClN8O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-DJJE4J	WO2022187419A1_219	.	C[C@H]1CC2(CCN(c3ncc(CN4CCC(N5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H49ClN10O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-AALPXG	WO2022187419A1_22	.	C[C@H]1CC2(CCN(c3ccc(C4CCN(C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H46ClN7O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-48MFKO	WO2022187419A1_220	.	C[C@H]1CC2(CCN(c3ccc(CN4CCC(N5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H50ClN9O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-748SGG	WO2022187419A1_221	.	C[C@H]1CC2(CCN(c3cnc(CN4CCC(N5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H49ClN10O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-7F8IJ6	WO2022187419A1_222	.	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CC(N(C)C5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H49ClN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-W62YQZ	WO2022187419A1_223	.	C[C@H]1CC2(CCN(c3ccc(CN4CC(N5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H46ClN9O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-3HQIGE	WO2022187419A1_224	.	C[C@H]1CC2(CCN(c3ccc(CN4CC(N5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)nn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C41H45ClN10O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-CBIHRB	WO2022187419A1_225	.	C[C@H]1CC2(CCN(c3cnc(CN4CC(N5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C41H45ClN10O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-M3DVJO	WO2022187419A1_226	2-chloro-4-[(3S)-8-[5-[[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]azetidin-1-yl]methyl]pyrimidin-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ncc(CN4CC(N5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C41H45ClN10O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-FY6ZOY	WO2022187419A1_227	2-chloro-4-[(3S)-8-[5-[[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]azetidin-1-yl]methyl]pyrazin-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3cnc(CN4CC(N5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C41H45ClN10O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-HUINB2	WO2022187419A1_228	2-chloro-4-[(3S)-8-[6-[[3-[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]azetidin-1-yl]methyl]pyridin-3-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(CN4CC(N5CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H45ClFN9O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-3DJYL5	WO2022187419A1_229	.	C[C@H]1CC2(CCN(c3ccc(CN4CC(N5CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)nn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C41H44ClFN10O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-2TG1MX	WO2022187419A1_23	.	C[C@H]1CC2(CCN(c3ccc(CC4CCN(C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H48ClN7O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-NC3C0T	WO2022187419A1_230	.	C[C@H]1CC2(CCN(c3cnc(CN4CC(N5CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C41H44ClFN10O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-Y9LQOC	WO2022187419A1_231	2-chloro-4-[(3S)-8-[5-[[3-[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]azetidin-1-yl]methyl]pyrimidin-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ncc(CN4CC(N5CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C41H44ClFN10O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-THYXHR	WO2022187419A1_232	.	C[C@H]1CC2(CCN(c3cnc(CN4CC(N5CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C41H44ClFN10O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-1V3Q9Z	WO2022187419A1_233	2-chloro-4-[(3S)-8-[4-[[4-[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]piperidin-1-yl]methyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(CN4CCC(N5CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H50ClFN8O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-XQ0J2D	WO2022187419A1_234	2-chloro-4-[(3S)-8-[5-[[4-[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]piperidin-1-yl]methyl]pyrimidin-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ncc(CN4CCC(N5CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H48ClFN10O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-EGWHTB	WO2022187419A1_235	2-chloro-4-[(3S)-8-[6-[[4-[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]piperidin-1-yl]methyl]pyridin-3-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(CN4CCC(N5CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H49ClFN9O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-AL8W2F	WO2022187419A1_236	2-chloro-4-[(3S)-8-[2-[[4-[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]piperidin-1-yl]methyl]pyrimidin-5-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3cnc(CN4CCC(N5CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H48ClFN10O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-A18QEL	WO2022187419A1_237	2-chloro-4-[(3S)-8-[5-[[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]piperidin-1-yl]methyl]pyrazin-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3cnc(CN4CCC(N5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H49ClN10O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-D4YST6	WO2022187419A1_238	2-chloro-4-[(3S)-8-[5-[[4-[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]piperidin-1-yl]methyl]pyrazin-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3cnc(CN4CCC(N5CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H48ClFN10O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-NH208A	WO2022187419A1_239	2-chloro-4-[(3S)-8-[6-[[4-[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperazin-1-yl]methyl]pyridin-3-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(CN4CCN(C5CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H49ClFN9O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-71Z4BD	WO2022187419A1_24	.	C[C@H]1CC2(CCN(c3ccc(CC4CCN(C5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C46H52ClN7O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-ZQGNAF	WO2022187419A1_240	2-chloro-4-[(3S)-8-[2-[[4-[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperazin-1-yl]methyl]pyrimidin-5-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3cnc(CN4CCN(C5CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H48ClFN10O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-5GWEG4	WO2022187419A1_241	2-chloro-4-[(3S)-8-[5-[[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperazin-1-yl]methyl]pyrazin-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3cnc(CN4CCN(C5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H49ClN10O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-7BCWPF	WO2022187419A1_242	2-chloro-4-[(3S)-8-[5-[[4-[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperazin-1-yl]methyl]pyrazin-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3cnc(CN4CCN(C5CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H48ClFN10O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-D9HRAD	WO2022187419A1_243	2-chloro-4-[(3S)-8-[6-[[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperazin-1-yl]methyl]pyridazin-3-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(CN4CCN(C5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)nn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H49ClN10O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-ZRWA1X	WO2022187419A1_244	2-chloro-4-[(3S)-8-[6-[[4-[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperazin-1-yl]methyl]pyridazin-3-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(CN4CCN(C5CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)nn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H48ClFN10O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-FEH949	WO2022187419A1_245	2-chloro-4-[(3S)-8-[5-[[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperazin-1-yl]methyl]pyrimidin-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ncc(CN4CCN(C5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H49ClN10O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-19U9KU	WO2022187419A1_246	.	C[C@H]1CC2(CCN(c3ncc(CN4CCN(C5CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H48ClFN10O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-UIP66Q	WO2022187419A1_247	2-chloro-4-[(3S)-8-[5-[[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperazin-1-yl]methyl]-1,3-thiazol-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ncc(CN4CCN(C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)s3)CC2)CN1c1ccc(C#N)c(Cl)c1	C40H44ClN9O4S	AR	P10275	CRBN	WO-2022187419-A1
TPD-FHXRD4	WO2022187419A1_248	2-chloro-4-[(3S)-8-[5-[[4-[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperazin-1-yl]methyl]-1,3-thiazol-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ncc(CN4CCN(C5CN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)s3)CC2)CN1c1ccc(C#N)c(Cl)c1	C40H43ClFN9O4S	AR	P10275	CRBN	WO-2022187419-A1
TPD-QNL7O9	WO2022187419A1_249	2-chloro-4-[(3S)-8-[5-[[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]azetidin-1-yl]methyl]-1,3-thiazol-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ncc(CN4CC(N5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)s3)CC2)CN1c1ccc(C#N)c(Cl)c1	C40H44ClN9O4S	AR	P10275	CRBN	WO-2022187419-A1
TPD-N8IF01	WO2022187419A1_25	.	C[C@H]1CC2(CCN(c3ccc(CC4CCN(CC5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H50ClN7O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-H1KGNK	WO2022187419A1_250	2-chloro-4-[(3S)-8-[5-[[3-[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]azetidin-1-yl]methyl]-1,3-thiazol-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ncc(CN4CC(N5CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)s3)CC2)CN1c1ccc(C#N)c(Cl)c1	C40H43ClFN9O4S	AR	P10275	CRBN	WO-2022187419-A1
TPD-UXW2D3	WO2022187419A1_251	2-chloro-4-[(3S)-8-[5-[[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperazin-1-yl]methyl]-1,3-thiazol-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ncc(CN4CCN(C5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)s3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H48ClN9O4S	AR	P10275	CRBN	WO-2022187419-A1
TPD-0VYUR0	WO2022187419A1_252	2-chloro-4-[(3S)-8-[5-[[4-[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperazin-1-yl]methyl]-1,3-thiazol-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ncc(CN4CCN(C5CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)s3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H47ClFN9O4S	AR	P10275	CRBN	WO-2022187419-A1
TPD-MT8PQ3	WO2022187419A1_253	.	C[C@H]1CC2(CCN(c3ncc(CN4CCC(N5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)s3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H48ClN9O4S	AR	P10275	CRBN	WO-2022187419-A1
TPD-CFJBGX	WO2022187419A1_254	2-chloro-4-[(3S)-8-[5-[[4-[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]piperidin-1-yl]methyl]-1,3-thiazol-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ncc(CN4CCC(N5CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)s3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H47ClFN9O4S	AR	P10275	CRBN	WO-2022187419-A1
TPD-GQS9LW	WO2022187419A1_26	.	C[C@H]1CC2(CCN(c3ccc(CC4CCN(CC5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C47H54ClN7O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-MUQW2K	WO2022187419A1_27	.	C[C@H]1CC2(CCN(c3ccc(N4CCN(C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H45ClN8O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-BQEHUK	SCHEMBL27241120	2-chloro-4-[(3S)-8-[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]methyl]piperazin-1-yl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(N4CCN(CC5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H47ClN8O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-0FIELA	WO2022187419A1_29	.	C[C@H]1CC2(CCN(c3ccc(N4CCN(C5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H49ClN8O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-B8KIFN	WO2022187419A1_3	.	C[C@H]1CC2(CCN(c3ccc(S(=O)(=O)N4CCC(CN5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H46ClN7O6S	AR	P10275	CRBN	WO-2022187419-A1
TPD-JBP525	WO2022187419A1_30	.	C[C@H]1CC2(CCN(c3ccc(N4CCN(CC5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H51ClN8O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-NC43Z1	WO2022187419A1_31	.	C[C@H]1CC2(CCN(c3ccc(N4CCN(CC5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H46ClN9O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-3SW0CR	WO2022187419A1_32	.	C[C@H]1CC2(CCN(c3ccc(N4CCN(CC5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H50ClN9O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-DAZ5P9	WO2022187419A1_33	.	C[C@H]1CC2(CCN(c3ccc(N4CCN(C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C41H44ClN9O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-WCF77H	WO2022187419A1_34	.	C[C@H]1CC2(CCN(c3ccc(N4CCN(CC5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H46ClN9O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-OE7QC8	WO2022187419A1_35	.	C[C@H]1CC2(CCN(c3ccc(N4CCN(CC5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H50ClN9O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-KHV9WQ	WO2022187419A1_36 	.	C[C@H]1CC2(CCN(c3ccc(N4CCN(C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C41H44ClN9O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-51UHT2	WO2022187419A1_37 	2-chloro-4-[(3S)-8-[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]methyl]piperazin-1-yl]-2-fluorophenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(N4CCN(CC5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cc3F)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H46ClFN8O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-CYU6D9	WO2022187419A1_38	.	C[C@H]1CC2(CCN(c3ccc(N4CCN(CC5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3F)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H50ClFN8O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-KUVUOC	WO2022187419A1_39	.	C[C@H]1CC2(CCN(c3ccc(N4CCN(C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cc3F)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H44ClFN8O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-XHV8ED	WO2022187419A1_4	.	C[C@H]1CC2(CCN(c3ccc(S(=O)(=O)N4CCC(N5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H44ClN7O6S	AR	P10275	CRBN	WO-2022187419-A1
TPD-23PZTC	WO2022187419A1_40	2-chloro-4-[(3S)-8-[4-[[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperazin-1-yl]methyl]-3-fluorophenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(CN4CCN(C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)c(F)c3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H46ClFN8O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-U7Z593	WO2022187419A1_41	2-chloro-4-[(3S)-8-[4-[[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperidin-1-yl]methyl]-3-fluorophenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(CN4CCC(C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)c(F)c3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H47ClFN7O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-BIERVJ	WO2022187419A1_43	.	C[C@H]1CC2(CCN(c3ccc(C4CCN(CC5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H47ClN8O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-PO2I44	WO2022187419A1_44	.	C[C@H]1CC2(CCN(c3ccc(C4CCN(CC5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H51ClN8O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-W6HF2L	WO2022187419A1_45	.	C[C@H]1CC2(CCN(c3ccc(C4CCN(CC5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H47ClN8O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-MYUAEP	WO2022187419A1_46	.	C[C@H]1CC2(CCN(c3ccc(C4CCN(CC5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H51ClN8O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-M750NL	WO2022187419A1_47	.	C[C@H]1CC2(CCN(c3ccc(N4CCN(CC5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)nn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C41H45ClN10O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-1PKTVZ	WO2022187419A1_48	.	C[C@H]1CC2(CCN(c3ccc(N4CCN(CC5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)nn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H49ClN10O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-EC5FVP	WO2022187419A1_49	.	C[C@H]1CC2(CCN(c3cnc(N4CCN(CC5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C41H45ClN10O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-B51V4Y	WO2022187419A1_5	2-chloro-4-[(3S)-8-[4-[[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperazin-1-yl]methyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(CN4CCN(C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H47ClN8O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-ABKAUZ	WO2022187419A1_50	.	C[C@H]1CC2(CCN(c3cnc(N4CCN(CC5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H49ClN10O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-GZ67CA	WO2022187419A1_51	2-chloro-4-[(3S)-8-[5-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]pyridin-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(N4CCC(CN5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H50ClN9O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-ELFCGU	WO2022187419A1_52	.	C[C@H]1CC2(CCN(c3ccc(N4CCC(CN5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H45ClN8O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-1QM7ET	WO2022187419A1_53	2-chloro-4-[(3S)-8-[6-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]pyridin-3-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(N4CCC(CN5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H50ClN9O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-YSYI4D	WO2022187419A1_54	.	C[C@H]1CC2(CCN(c3ccc(N4CCC(CN5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H45ClN8O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-YOZXFH	WO2022187419A1_55	2-chloro-4-[(3S)-8-[6-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]pyridazin-3-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(N4CCC(CN5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)nn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H49ClN10O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-1BWN2S	WO2022187419A1_56	.	C[C@H]1CC2(CCN(c3ccc(N4CCC(CN5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)nn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C41H44ClN9O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-6LC7QH	WO2022187419A1_57	.	C[C@H]1CC2(CCN(c3ccc(OC4CCN(C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H46ClN7O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-P56T45	WO2022187419A1_58	.	C[C@H]1CC2(CCN(c3ccc(OC4CCN(C5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H50ClN7O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-RLP0EJ	WO2022187419A1_59	.	C[C@H]1CC2(CCN(c3ccc(OC4CN(C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)C4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C41H42ClN7O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-4TKS2R	WO2022187419A1_60	.	C[C@H]1CC2(CCN(c3ccc(OC4CN(C5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H46ClN7O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-I9TNQF	SCHEMBL27241104	2-chloro-4-[(3S)-8-[5-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperidin-4-yl]oxypyridin-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL30069552	C[C@H]1CC2(CCN(c3ccc(OC4CCN(C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H45ClN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-WDEAXX	WO2022187419A1_62	.	C[C@H]1CC2(CCN(c3ccc(OC4CCN(C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)nn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C41H44ClN9O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-LAYRP0	WO2022187419A1_63	.	C[C@H]1CC2(CCN(c3ccc(OC4CCN(C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H45ClN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-BJTR74	WO2022187419A1_64	.	C[C@H]1CC2(CCN(c3cnc(OC4CCN(C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C41H44ClN9O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-RT93IW	WO2022187419A1_65	.	C[C@H]1CC2(CCN(c3ccc(OC4CCN(C5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H49ClN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-OW4TDM	WO2022187419A1_66	2-chloro-4-[(3S)-8-[6-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperidin-4-yl]oxypyridazin-3-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(OC4CCN(C5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)nn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H48ClN9O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-I4NOH2	WO2022187419A1_67	.	C[C@H]1CC2(CCN(c3ccc(OC4CCN(C5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H49ClN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-T3AYTB	WO2022187419A1_68	.	C[C@H]1CC2(CCN(c3cnc(OC4CCN(C5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H48ClN9O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-L25PB0	WO2022187419A1_69	.	C[C@H]1CC2(CCN(c3ccc(OC4CN(C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)C4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C40H41ClN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-WN9CYT	WO2022187419A1_7 	2-chloro-4-[(3S)-8-[2-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]-1,3-dihydroisoindol-5-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc4c(c3)CN(CC3CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC3)C4)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H46ClN7O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-NS3RBR	WO2022187419A1_70	2-chloro-4-[(3S)-8-[5-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]azetidin-3-yl]oxypyridin-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(OC4CN(C5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H45ClN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-AV4JV9	WO2022187419A1_71	2-chloro-4-[(3S)-8-[6-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]azetidin-3-yl]oxypyridin-3-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(OC4CN(C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)C4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C40H41ClN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-MW25E9	WO2022187419A1_72 	.	C[C@H]1CC2(CCN(c3ccc(OC4CN(C5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H45ClN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-UW56VZ	WO2022187419A1_73	2-chloro-4-[(3S)-8-[6-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]azetidin-3-yl]oxypyridazin-3-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(OC4CN(C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)C4)nn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C39H40ClN9O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-PZ6HI9	WO2022187419A1_74	2-chloro-4-[(3S)-8-[6-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]azetidin-3-yl]oxypyridazin-3-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(OC4CN(C5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)nn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C41H44ClN9O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-Y7KZUT	WO2022187419A1_75	.	C[C@H]1CC2(CCN(c3ncc(C4CCN(CC5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H46ClN9O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-8IPB4S	WO2022187419A1_76	2-chloro-4-[(3S)-8-[2-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]methyl]piperazin-1-yl]pyrimidin-5-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3cnc(N4CCN(CC5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C41H45ClN10O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-OZ38KX	WO2022187419A1_77	.	C[C@H]1CC2(CCN(c3ncc(N4CCN(CC5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C41H45ClN10O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-ZFW7B2	ARD-1671	2-chloro-4-[(3S)-8-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]piperidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; CHEMBL5399633; SCHEMBL23125339	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(N5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H44ClN7O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-OW7KNE	WO2022187419A1_83	2-chloro-4-[(3S)-8-[2-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]pyrimidin-5-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3cnc(N4CCN(CC5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H49ClN10O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-GII9Z5	WO2022187419A1_84	2-chloro-4-[(3S)-8-[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-3-fluoroazetidin-3-yl]methyl]piperazin-1-yl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(N4CCN(CC5(F)CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H46ClFN8O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-P9MLKN	WO2022187419A1_85	.	COC1(CN2CCN(c3ccc(N4CCC5(CC4)C[C@H](C)N(c4ccc(C#N)c(Cl)c4)C5)cc3)CC2)CN(c2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)C1	C44H49ClN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-A9MF5L	WO2022187419A1_86	2-chloro-4-[(3S)-8-[6-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-3-fluoroazetidin-3-yl]methyl]piperazin-1-yl]pyridin-3-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(N4CCN(CC5(F)CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H45ClFN9O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-2W62GL	WO2022187419A1_87	2-chloro-4-[(3S)-8-[6-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-3-methoxyazetidin-3-yl]methyl]piperazin-1-yl]pyridin-3-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	COC1(CN2CCN(c3ccc(N4CCC5(CC4)C[C@H](C)N(c4ccc(C#N)c(Cl)c4)C5)cn3)CC2)CN(c2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)C1	C43H48ClN9O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-5JHYJT	WO2022187419A1_88	2-chloro-4-[(3S)-8-[5-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-3-fluoroazetidin-3-yl]methyl]piperazin-1-yl]pyridin-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(N4CCN(CC5(F)CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H45ClFN9O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-5FQPRZ	WO2022187419A1_89	2-chloro-4-[(3S)-8-[5-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-3-methoxyazetidin-3-yl]methyl]piperazin-1-yl]pyridin-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	COC1(CN2CCN(c3ccc(N4CCC5(CC4)C[C@H](C)N(c4ccc(C#N)c(Cl)c4)C5)nc3)CC2)CN(c2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)C1	C43H48ClN9O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-G8RYET	WO2022187419A1_90	2-chloro-4-[(3S)-8-[4-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]oxypiperidin-1-yl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(N4CCC(OC5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H46ClN7O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-JENNOW	WO2022187419A1_91	2-chloro-4-[(3S)-8-[6-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]oxypiperidin-1-yl]pyridin-3-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(N4CCC(OC5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H45ClN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-W0SVOI	WO2022187419A1_92	2-chloro-4-[(3S)-8-[5-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]oxypiperidin-1-yl]pyridin-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(N4CCC(OC5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H45ClN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-RFKK3Z	WO2022187419A1_93	2-chloro-4-[(3S)-8-[6-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]oxypiperidin-1-yl]pyridazin-3-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(N4CCC(OC5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)nn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C41H44ClN9O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-908T82	WO2022187419A1_94	2-chloro-4-[(3S)-8-[2-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]oxypiperidin-1-yl]pyrimidin-5-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3cnc(N4CCC(OC5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C41H44ClN9O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-WBSUCF	WO2022187419A1_95	2-chloro-4-[(3S)-8-[5-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]oxypiperidin-1-yl]pyrazin-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3cnc(N4CCC(OC5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C41H44ClN9O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-JWYYPI	WO2022187419A1_96	2-chloro-4-[(3S)-8-[5-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]oxypiperidin-1-yl]pyrimidin-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ncc(N4CCC(OC5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C41H44ClN9O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-ZKN3Q1	WO2022187419A1_97	.	C[C@H]1CC2(CCN(c3ccc(N4CCC(N5CC(Oc6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H46ClN7O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-2XVU79	WO2022187419A1_98	.	C[C@H]1CC2(CCN(c3ccc(N4CCC(N5CC(Oc6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H45ClN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-G9GA6P	WO2022187419A1_99	.	C[C@H]1CC2(CCN(c3ccc(N4CCC(N5CC(Oc6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H45ClN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-GCVGSE	ARD-2051	2-chloro-4-[(3S)-8-[4-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperazine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; 2632305-17-8; CHEMBL5404267; orb2278305; SCHEMBL23125320; SCHEMBL29795965; GLXC-27543; BDBM50620470; EX-A12444; AT40049; BP-42200; DA-71028; HY-149862; CS-0866810; 2-Chloro-4-((3S)-8-(4-(4-(1-(2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindolin-5-yl)azetidin-3-yl)piperazine-1-carbonyl)phenyl)-3-methyl-2,8-diazaspiro[4.5]decan-2-yl)benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H45ClN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-92CR53	SCHEMBL23125225	2-chloro-4-[(3S)-8-[4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-6-yl]methyl]piperidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(CN5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H48ClN7O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-NEPZY4	SCHEMBL23125385	2-chloro-4-[(3S)-8-[5-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazine-1-carbonyl]pyrazin-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL29796029	C[C@H]1CC2(CCN(c3cnc(C(=O)N4CCN(CC5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H49ClN10O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-TCJIRS	ARD-7064	2-chloro-4-[(3S)-8-[5-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidine-1-carbonyl]pyrazin-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; CHEMBL5436760; SCHEMBL23125249	C[C@H]1CC2(CCN(c3cnc(C(=O)N4CCC(CN5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H44ClN9O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-2PAKBN	ARD-7063	2-chloro-4-[(3S)-8-[6-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidine-1-carbonyl]pyridazin-3-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; CHEMBL5437356; SCHEMBL23125164; SCHEMBL29796052	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(CN5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)nn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H44ClN9O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-JN03KV	SCHEMBL23125271	2-chloro-4-[(3S)-8-[5-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]piperidine-1-carbonyl]pyrazin-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL29795940	C[C@H]1CC2(CCN(c3cnc(C(=O)N4CCC(N5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H47ClN10O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-WWWAVC	SCHEMBL23125247	2-chloro-4-[(3S)-8-[5-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]piperidine-1-carbonyl]pyrazin-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL29795907	C[C@H]1CC2(CCN(c3cnc(C(=O)N4CCC(N5CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H46ClFN10O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-UQ7FD4	SCHEMBL23125286	2-chloro-4-[(3S)-8-[6-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]piperidine-1-carbonyl]pyridazin-3-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL29795809	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(N5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)nn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H47ClN10O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-4GA2F0	SCHEMBL23125382	2-chloro-4-[(3S)-8-[6-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]piperidine-1-carbonyl]pyridazin-3-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL29795979	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(N5CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)nn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H46ClFN10O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-100YOG	SCHEMBL23125334	2-chloro-4-[(3S)-8-[6-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperazine-1-carbonyl]pyridazin-3-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL29796051	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(C5CN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)nn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C41H42ClFN10O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-APSWPN	SCHEMBL23125279	2-chloro-4-[(3S)-8-[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]azetidin-3-yl]methyl]piperazine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL29795840	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(CC5CN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H46ClFN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-EQDYMB	SCHEMBL23125131	2-chloro-4-[(3S)-8-[6-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]azetidin-3-yl]methyl]piperazine-1-carbonyl]pyridazin-3-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL29795932	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(CC5CN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)nn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H44ClFN10O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-JO5F20	ARD-1683	2-chloro-4-[(3S)-8-[4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]-4-fluoropiperidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; CHEMBL5440609; SCHEMBL23125296	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(F)(CN5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H45ClFN7O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-X712EU	SCHEMBL23125076	2-chloro-4-[(3S)-8-[5-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperazine-1-carbonyl]pyridin-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL29795814	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(C5CN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H43ClFN9O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-WQCQPD	SCHEMBL23125153	2-chloro-4-[(3S)-8-[5-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperazine-1-carbonyl]pyridin-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL29795952	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(C5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H48ClN9O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-QZKNM4	SCHEMBL23125128	2-chloro-4-[(3S)-8-[4-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperazine-1-carbonyl]-2-fluorophenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL29788756	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cc3F)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H44ClFN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-DQWMK8	SCHEMBL23125142	2-chloro-4-[(3S)-8-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]piperidine-1-carbonyl]-2-fluorophenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL29795974	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(N5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3F)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H48ClFN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-KBFFJQ	SCHEMBL23125208	2-chloro-4-[(3S)-8-[5-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperazine-1-carbonyl]pyrimidin-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL29796037	C[C@H]1CC2(CCN(c3ncc(C(=O)N4CCN(C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C41H43ClN10O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-EJ8M1R	SCHEMBL23125282	2-chloro-4-[(3S)-8-[5-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperazine-1-carbonyl]pyrimidin-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL29795904	C[C@H]1CC2(CCN(c3ncc(C(=O)N4CCN(C5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H47ClN10O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-ETLWNP	ARD-1684	2-chloro-4-[(3S)-8-[4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]-4-methoxypiperidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; CHEMBL4851345; SCHEMBL23125380	COC1(CN2Cc3cc4c(cc3C2)C(=O)N(C2CCC(=O)NC2=O)C4=O)CCN(C(=O)c2ccc(N3CCC4(CC3)C[C@H](C)N(c3ccc(C#N)c(Cl)c3)C4)cc2)CC1	C45H48ClN7O6	AR	P10275	CRBN	WO-2022187419-A1
TPD-2YRKDM	SCHEMBL23125398	2-chloro-4-[(3S)-8-[5-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]piperidine-1-carbonyl]pyrimidin-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL29795934	C[C@H]1CC2(CCN(c3ncc(C(=O)N4CCC(N5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H47ClN10O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-WT4YZT	SCHEMBL23125336	2-chloro-4-[(3S)-8-[4-[(3R)-3-[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]pyrrolidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL29795939	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CC[C@@H](N5CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H46ClFN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-UJDHMA	SCHEMBL23124910	2-chloro-4-[(3S)-8-[4-[(3S)-3-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]pyrrolidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL29795829	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CC[C@H](N5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H47ClN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-32T3YB	SCHEMBL23125263	2-chloro-4-[(3S)-8-[4-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperazine-1-carbonyl]-2-fluorophenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL29795875	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(C5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3F)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H48ClFN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-V2IQFZ	SCHEMBL23125302	2-chloro-4-[(3S)-8-[5-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperazine-1-carbonyl]pyrimidin-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL29796012	C[C@H]1CC2(CCN(c3ncc(C(=O)N4CCN(C5CN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C41H42ClFN10O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-KQ8DOE	WO2022187419A1_A13	.	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CC(N5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7)C4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C41H42ClN7O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-3A4Z9D	SCHEMBL23125361	2-chloro-4-[(3S)-8-[5-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperazine-1-carbonyl]pyrimidin-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL29795966	C[C@H]1CC2(CCN(c3ncc(C(=O)N4CCN(C5CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H46ClFN10O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-RVWUTR	SCHEMBL23125280	2-chloro-4-[(3S)-8-[5-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]piperidine-1-carbonyl]pyrimidin-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL29795851	C[C@H]1CC2(CCN(c3ncc(C(=O)N4CCC(N5CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H46ClFN10O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-T391XT	SCHEMBL23125107	2-chloro-4-[(3S)-8-[5-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidine-1-carbonyl]pyrimidin-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ncc(C(=O)N4CCC(CN5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H44ClN9O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-L0IV98	SCHEMBL23125364	2-chloro-4-[(3S)-8-[4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidine-1-carbonyl]-2-fluorophenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL29795824	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(CN5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)cc3F)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H45ClFN7O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-5MR78N	SCHEMBL23125307	2-chloro-4-[(3S)-8-[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]methyl]piperazine-1-carbonyl]-2-fluorophenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL29795917	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(CC5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cc3F)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H46ClFN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-8PUNEQ	SCHEMBL23124914	2-chloro-4-[(3S)-8-[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]methyl]piperazine-1-carbonyl]-3-fluorophenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL29795982	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(CC5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)c(F)c3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H46ClFN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-7RTZ7Q	SCHEMBL23124940	2-chloro-4-[(3S)-8-[4-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperazine-1-carbonyl]-3-fluorophenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL29795950	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(C5CN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)c(F)c3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H43ClF2N8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-NJ3UE8	SCHEMBL23125193	2-chloro-4-[(3S)-8-[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]azetidin-3-yl]methyl]piperazine-1-carbonyl]-3-fluorophenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL29795871	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(CC5CN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)c(F)c3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H45ClF2N8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-Q1SCVR	SCHEMBL23125399	2-chloro-4-[(3S)-8-[4-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperazine-1-carbonyl]-2-fluorophenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL29788764	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(C5CN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cc3F)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H43ClF2N8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-XOIPHR	SCHEMBL23125212	2-chloro-4-[(3S)-8-[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]azetidin-3-yl]methyl]piperazine-1-carbonyl]-2-fluorophenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL29795994	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(CC5CN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cc3F)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H45ClF2N8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-NG7HOK	ARD-1690	2-chloro-4-[(3S)-8-[4-[3-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]azetidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; CHEMBL4862208; SCHEMBL23125344	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CC(CN5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H42ClN7O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-67AS20	SCHEMBL23125071	2-chloro-4-[(3S)-8-[4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidine-1-carbonyl]-3-fluorophenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL29796106	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(CN5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)c(F)c3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H45ClFN7O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-7KAVBN	CHEMBL5437794	2-chloro-4-[(3S)-8-[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]methyl]piperazine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL23125392; SCHEMBL29795914	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(CC5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H47ClN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-E7F25L	SCHEMBL23125372	2-chloro-4-[(3S)-8-[6-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]azetidine-1-carbonyl]pyridazin-3-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL29795795	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CC(N5CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)nn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C41H42ClFN10O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-PUOMU8	SCHEMBL23125091	2-chloro-4-[(3S)-8-[6-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]azetidine-1-carbonyl]pyridin-3-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL29795852	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CC(N5CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H43ClFN9O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-I57MK1	SCHEMBL23125180	2-chloro-4-[(3S)-8-[5-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]azetidine-1-carbonyl]pyridin-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL29795925	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CC(N5CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H43ClFN9O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-WF75UK	SCHEMBL23138872	2-chloro-4-[(3S)-8-[4-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperazine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(C5CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H48ClFN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-HZO79I	SCHEMBL23138020	2-chloro-4-[(3S)-8-[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(CC5CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C46H50ClFN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-X9DYUV	SCHEMBL23138021	2-chloro-4-[(3S)-8-[6-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperazine-1-carbonyl]pyridin-3-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(C5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H48ClN9O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-QLDN6G	SCHEMBL23138028	2-chloro-4-[(3S)-8-[6-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazine-1-carbonyl]pyridin-3-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(CC5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H50ClN9O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-QKNBEK	CHEMBL4867200	2-chloro-4-[(3S)-8-[4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-6-yl]methyl]-4-fluoropiperidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; PD173206	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(F)(CN5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H47ClFN7O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-R6IVOZ	SCHEMBL23138029	2-chloro-4-[(3S)-8-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-7,8-dihydro-5H-pyrrolo[3,4-g]isoquinolin-6-yl]piperidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(N5CCc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H46ClN7O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-NIE2OL	SCHEMBL23138867	2-chloro-4-[(3S)-8-[4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-7,8-dihydro-5H-pyrrolo[3,4-g]isoquinolin-6-yl]methyl]piperidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(CN5CCc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H48ClN7O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-YPP0L1	SCHEMBL23138868	2-chloro-4-[(3S)-8-[4-[4-[(3S)-1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]pyrrolidin-3-yl]piperazine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN([C@H]5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H47ClN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-6YLPKW	SCHEMBL23138863	2-chloro-4-[(3S)-8-[4-[4-[(3R)-1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]pyrrolidin-3-yl]piperazine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN([C@@H]5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H47ClN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-RK7LYK	SCHEMBL23138865	2-chloro-4-[(3S)-8-[4-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]pyrrolidin-3-yl]piperazine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(C5CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H46ClFN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-GAQ7AY	SCHEMBL23138866	2-chloro-4-[(3S)-8-[4-[4-[(3R)-1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]pyrrolidin-3-yl]piperazine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN([C@@H]5CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H46ClFN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-P9TYXP	SCHEMBL23138878	2-chloro-4-[(3S)-8-[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazine-1-carbonyl]-2-fluorophenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(CC5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3F)CC2)CN1c1ccc(C#N)c(Cl)c1	C46H50ClFN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-841KLO	SCHEMBL23138877	2-chloro-4-[(3S)-8-[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazine-1-carbonyl]-3-fluorophenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(CC5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)c(F)c3)CC2)CN1c1ccc(C#N)c(Cl)c1	C46H50ClFN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-AXH1MD	SCHEMBL23138880	2-chloro-4-[(3S)-8-[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazine-1-carbonyl]-2-fluorophenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(CC5CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3F)CC2)CN1c1ccc(C#N)c(Cl)c1	C46H49ClF2N8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-5NBYP3	SCHEMBL23138876	2-chloro-4-[(3S)-8-[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazine-1-carbonyl]-3-fluorophenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(CC5CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)c(F)c3)CC2)CN1c1ccc(C#N)c(Cl)c1	C46H49ClF2N8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-U7Y9L2	SCHEMBL23138714	2-chloro-4-[(3S)-8-[4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-6-yl]methyl]-4-methoxypiperidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	COC1(CN2Cc3cc4c(cc3C2)C(=O)N(C2CCC(=O)NC2=O)C4)CCN(C(=O)c2ccc(N3CCC4(CC3)C[C@H](C)N(c3ccc(C#N)c(Cl)c3)C4)cc2)CC1	C45H50ClN7O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-B1N43U	WO2022187419A1_A161	.	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(C5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)c(F)c3)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H48ClFN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-2JKGPV	SCHEMBL23125357	2-chloro-4-[(3S)-8-[4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,6,8,9-tetrahydropyrrolo[3,4-h][3]benzazepin-7-yl]methyl]piperidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(CN5CCc6cc7c(cc6CC5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C46H50ClN7O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-JB45KP	WO2022187419A1_A163	.	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(N5CCc6cc7c(cc6CC5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H48ClN7O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-0MKQF5	WO2022187419A1_A164	.	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(CN5CCCc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C46H50ClN7O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-I8OGKD	WO2022187419A1_A165	.	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CC(CN5CCc6cc7c(cc6CC5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H46ClN7O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-68PX05	SCHEMBL23138776	2-chloro-4-[(3S)-8-[4-[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,6,8,9-tetrahydropyrrolo[3,4-h][3]benzazepin-7-yl]azetidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CC(N5CCc6cc7c(cc6CC5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H44ClN7O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-PP14EG	WO2022187419A1_A167	.	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(N5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H48ClN9O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-3UFPMW	ARD-4055	2-chloro-4-[(3S)-8-[6-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidine-1-carbonyl]pyridin-3-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; CHEMBL5398110	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(CN5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H45ClN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-KPD7HF	WO2022187419A1_A169	.	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(N5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H43ClN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-5AJE3C	ARD-1694	2-chloro-4-[(3S)-8-[4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]-4-methylpiperidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; CHEMBL5437017; SCHEMBL23138948	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(C)(CN5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H48ClN7O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-LDIUK0	SCHEMBL23139069	2-chloro-4-[(3S)-8-[6-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperazine-1-carbonyl]pyridazin-3-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(C5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)nn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H47ClN10O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-S3K1WZ	SCHEMBL23139070	2-chloro-4-[(3S)-8-[5-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperazine-1-carbonyl]pyrazin-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3cnc(C(=O)N4CCN(C5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H47ClN10O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-8DOIVX	SCHEMBL23125322	2-chloro-4-[(3S)-8-[6-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperidine-1-carbonyl]pyridazin-3-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL29795967	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(C5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)nn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H48ClN9O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-3397US	WO2022187419A1_A173	.	C[C@H]1CC2(CCN(c3cnc(C(=O)N4CCC(C5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H48ClN9O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-LYZRH0	WO2022187419A1_A174	.	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(C5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H49ClN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-CMNKIK	WO2022187419A1_A175	.	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(C5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H49ClN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-V74DMY	WO2022187419A1_A176	.	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CC(C5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)nn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H44ClN9O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-TMX8RP	WO2022187419A1_A177	.	C[C@H]1CC2(CCN(c3cnc(C(=O)N4CC(C5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H44ClN9O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-ZHGTXA	WO2022187419A1_A178	.	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CC(C5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H45ClN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-SQ78LO	WO2022187419A1_A179	.	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CC(C5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H45ClN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-C36TO8	CHEMBL4852425	2-chloro-4-[(3S)-8-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]-7-azaspiro[3.5]nonane-7-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL23138946; PD173208	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC5(CC4)CC(N4Cc6cc7c(cc6C4)C(=O)N(C4CCC(=O)NC4=O)C7=O)C5)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C46H48ClN7O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-5KWWK5	WO2022187419A1_A180	.	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)nn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H44ClN9O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-MLV1C2	WO2022187419A1_A181	.	C[C@H]1CC2(CCN(c3cnc(C(=O)N4CCC(C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H44ClN9O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-TGLQAH	WO2022187419A1_A182	.	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H45ClN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-8SVBHE	WO2022187419A1_A183	.	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H45ClN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-7HDOL3	WO2022187419A1_A184	.	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CC(N5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)nn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C41H43ClN10O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-XBHJCI	WO2022187419A1_A185	.	C[C@H]1CC2(CCN(c3cnc(C(=O)N4CC(N5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C41H43ClN10O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-FHPSFG	WO2022187419A1_A186	.	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CC(N5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H44ClN9O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-OI98WK	WO2022187419A1_A187	.	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CC(N5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H44ClN9O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-4HWAFZ	WO2022187419A1_A188	.	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CC(C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)C4)nn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C40H40ClN9O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-FV64SG	WO2022187419A1_A189	.	C[C@H]1CC2(CCN(c3cnc(C(=O)N4CC(C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)C4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C40H40ClN9O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-69UTHS	WO2022187419A1_A19	2-chloro-4-[(3S)-8-[4-[6-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]-2-azaspiro[3.3]heptane-2-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CC5(CC(N6Cc7cc8c(cc7C6)C(=O)N(C6CCC(=O)NC6=O)C8=O)C5)C4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H44ClN7O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-XRO20V	WO2022187419A1_A190	.	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CC(C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)C4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C41H41ClN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-5U9IXJ	WO2022187419A1_A191	.	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CC(C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)C4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C41H41ClN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-HTIR4V	SCHEMBL23138833	2-chloro-4-[(3S)-8-[6-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazine-1-carbonyl]pyridazin-3-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(CC5CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)nn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H48ClFN10O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-T27TBE	CHEMBL5431770	2-chloro-4-[(3S)-8-[4-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperazine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL23138706	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(C5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H49ClN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-56VZ7G	WO2022187419A1_A20	.	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CC[C@@H](CN5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H44ClN7O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-1IWVZ6	WO2022187419A1_A21	.	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CC[C@H](CN5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H44ClN7O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-3ZDGVB	SCHEMBL23138952	2-chloro-4-[(3S)-8-[4-[3-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]-3-fluoroazetidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CC(F)(CN5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H41ClFN7O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-34IRDR	SCHEMBL23138953	2-chloro-4-[(3S)-8-[4-[3-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]-3-methoxyazetidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	COC1(CN2Cc3cc4c(cc3C2)C(=O)N(C2CCC(=O)NC2=O)C4=O)CN(C(=O)c2ccc(N3CCC4(CC3)C[C@H](C)N(c3ccc(C#N)c(Cl)c3)C4)cc2)C1	C43H44ClN7O6	AR	P10275	CRBN	WO-2022187419-A1
TPD-LGBWC6	SCHEMBL23138949	2-chloro-4-[(3S)-8-[4-[3-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]-3-methylazetidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CC(C)(CN5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H44ClN7O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-BC8KGK	SCHEMBL23138954	2-chloro-4-[(3S)-8-[4-[3-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-6-yl]methyl]-3-fluoroazetidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CC(F)(CN5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7)C4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H43ClFN7O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-K2SMFE	SCHEMBL23138852	2-chloro-4-[(3S)-8-[4-[3-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-6-yl]methyl]-3-methoxyazetidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	COC1(CN2Cc3cc4c(cc3C2)C(=O)N(C2CCC(=O)NC2=O)C4)CN(C(=O)c2ccc(N3CCC4(CC3)C[C@H](C)N(c3ccc(C#N)c(Cl)c3)C4)cc2)C1	C43H46ClN7O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-37HS0R	SCHEMBL23138847	2-chloro-4-[(3S)-8-[4-[3-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-6-yl]methyl]-3-methylazetidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CC(C)(CN5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7)C4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H46ClN7O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-51NYUQ	ARD-1705	2-chloro-4-[(3S)-8-[4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]-4-hydroxypiperidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; CHEMBL5403307; SCHEMBL23138850	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(O)(CN5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H46ClN7O6	AR	P10275	CRBN	WO-2022187419-A1
TPD-OU33OU	SCHEMBL23138853	2-chloro-4-[(3S)-8-[4-[3-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]-3-hydroxyazetidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CC(O)(CN5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H42ClN7O6	AR	P10275	CRBN	WO-2022187419-A1
TPD-A59OTW	SCHEMBL23138855	2-chloro-4-[(3S)-8-[4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-6-yl]methyl]-4-methylpiperidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(C)(CN5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H50ClN7O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-BVM6XX	SCHEMBL23138849	2-chloro-4-[(3S)-8-[4-[3-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-6-yl]methyl]azetidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CC(CN5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7)C4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H44ClN7O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-EL5GM3	SCHEMBL23138857	2-chloro-4-[(3S)-3-methyl-8-[4-[4-[[2-(1-methyl-2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidine-1-carbonyl]phenyl]-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(CN5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)N(C)C5=O)C7=O)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H48ClN7O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-OHUMQ6	SCHEMBL23138888	2-chloro-4-[(3S)-3-methyl-8-[4-[4-[2-(1-methyl-2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]piperidine-1-carbonyl]phenyl]-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(N5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)N(C)C5=O)C7=O)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H46ClN7O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-P31ZXM	WO2022187419A1_A34	.	C[C@H]1CC2(CCN(C(=O)c3ccc(N4CCN(CC(=O)N5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H45ClN8O6	AR	P10275	CRBN	WO-2022187419-A1
TPD-7X978W	CHEMBL4846160	2-chloro-4-[(3S)-8-[4-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]-2-oxoethyl]piperazine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL23125408; PD173210	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(CC(=O)N5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H45ClN8O6	AR	P10275	CRBN	WO-2022187419-A1
TPD-OMP7OB	CHEMBL4851046	2-chloro-4-[(3S)-8-[4-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]acetyl]piperazine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL23125205	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(C(=O)CN5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H45ClN8O6	AR	P10275	CRBN	WO-2022187419-A1
TPD-SMLUOI	CHEMBL4871674	2-chloro-4-[(3S)-8-[4-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-6-yl]acetyl]piperazine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL23138784; PD173214	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(C(=O)CN5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H47ClN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-LWFR2C	CHEMBL5427973	2-chloro-4-[(3S)-8-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]azetidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL23125229; SCHEMBL29795826	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CC(N5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H45ClN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-V1WL4P	SCHEMBL23125222	2-chloro-4-[(3S)-8-[4-[7-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]-2-azaspiro[3.5]nonane-2-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CC5(CCC(N6Cc7cc8c(cc7C6)C(=O)N(C6CCC(=O)NC6=O)C8=O)CC5)C4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C46H48ClN7O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-X4M41D	SCHEMBL23124907	2-chloro-4-[(3S)-8-[4-[6-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]-2-azaspiro[3.3]heptane-2-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CC5(CC(CN6Cc7cc8c(cc7C6)C(=O)N(C6CCC(=O)NC6=O)C8=O)C5)C4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H46ClN7O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-84CFBI	CHEMBL5427499	2-chloro-4-[(3S)-8-[4-[(1S,4S)-5-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]-2,5-diazabicyclo[2.2.1]heptane-2-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL23125176	C[C@H]1CC2(CCN(c3ccc(C(=O)N4C[C@@H]5C[C@H]4CN5C4CN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H45ClN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-OS7JHH	CHEMBL5409000	2-chloro-4-[(3S)-8-[4-[(1R,4R)-5-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]-2,5-diazabicyclo[2.2.1]heptane-2-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL23125395	C[C@H]1CC2(CCN(c3ccc(C(=O)N4C[C@H]5C[C@@H]4CN5C4CN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H45ClN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-N5R0N3	SCHEMBL23125403	2-chloro-4-[(3S)-8-[4-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxopyrrolo[3,4-c]pyridin-6-yl]azetidin-3-yl]piperazine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL29795817	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(C5CN(c6cc7c(cn6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H44ClN9O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-7FQITW	SCHEMBL23125086	2-chloro-4-[(3S)-8-[4-[4-[1-[6-(2,6-dioxopiperidin-3-yl)-5,7-dioxopyrrolo[3,4-b]pyridin-3-yl]azetidin-3-yl]piperazine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(C5CN(c6cnc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H44ClN9O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-316CYO	SCHEMBL23125093	2-chloro-4-[(3S)-8-[6-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperazine-1-carbonyl]pyridin-3-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL29795896	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H44ClN9O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-AP0GVV	SCHEMBL23125384	2-chloro-4-[(3S)-8-[4-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]azetidin-3-yl]piperazine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(C5CN(c6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H45ClN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-QD2NEW	SCHEMBL23125353	2-chloro-4-[(3S)-8-[6-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperazine-1-carbonyl]pyridazin-3-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL29795988	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)nn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C41H43ClN10O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-RYOFYQ	SCHEMBL23125297	2-chloro-4-[(3S)-8-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindole-6-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4Cc5cc6c(cc5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C38H35ClN6O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-I5RVS4	SCHEMBL23125363	2-chloro-4-[(3S)-8-[4-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperazine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL29795927	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(C5CN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H44ClFN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-BWAMMR	SCHEMBL23125234	2-chloro-4-[(3S)-8-[5-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperazine-1-carbonyl]pyridin-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL29795984	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H44ClN9O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-F6YBMX	SCHEMBL23125359	2-chloro-4-[(3S)-8-[5-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]piperidine-1-carbonyl]pyridin-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL29795951	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(N5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H43ClN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-848S7J	ARD-4056	2-chloro-4-[(3S)-8-[5-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidine-1-carbonyl]pyridin-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; CHEMBL5396008; SCHEMBL23125374; SCHEMBL29795938	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(CN5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H45ClN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-SMSDC5	SCHEMBL23125273	2-chloro-4-[(3S)-8-[4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-6,7-dihydro-5H-cyclopenta[f]isoindol-6-yl]methyl]piperazine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL29795843	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(CC5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H46ClN7O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-6OV81K	SCHEMBL23125360	2-chloro-4-[(3S)-8-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-6,7-dihydro-5H-cyclopenta[f]isoindol-6-yl]piperazine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL29788760	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(C5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H44ClN7O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-PZ685I	CHEMBL5419206	2-chloro-4-[(3S)-8-[4-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL23125228; SCHEMBL29795919	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H46ClN7O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-80DMOV	CHEMBL5400020	3-[4-[4-[(3S)-2-(3-chloro-4-cyanophenyl)-3-methyl-2,8-diazaspiro[4.5]decan-8-yl]benzoyl]piperazin-1-yl]-1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidine-3-carbonitrile; SCHEMBL23125199; SCHEMBL29788754	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(C5(C#N)CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H44ClN9O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-9R58OE	SCHEMBL23125326	2-chloro-4-[(3S)-8-[6-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]piperidine-1-carbonyl]pyridazin-3-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL29795980	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(N5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)nn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C41H42ClN9O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-GFH8U7	SCHEMBL23138937	2-chloro-4-[(3S)-3-methyl-8-[4-[4-[1-[2-(1-methyl-2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperazine-1-carbonyl]phenyl]-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)N(C)C6=O)C7=O)C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H47ClN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-QRSMEM	SCHEMBL23125375	2-chloro-4-[(3S)-8-[4-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]azetidin-3-yl]piperazine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL29796010	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(C5CN(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H47ClN8O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-IS6LGX	SCHEMBL23125211	2-chloro-4-[(3S)-8-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-6,7-dihydro-5H-cyclopenta[f]isoindole-6-carbonyl]piperazine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL29788763	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(C(=O)C5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H44ClN7O6	AR	P10275	CRBN	WO-2022187419-A1
TPD-KDCM38	SCHEMBL23125295	2-chloro-4-[(3S)-8-[4-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-6,7-dihydro-5H-cyclopenta[f]isoindol-6-yl]acetyl]piperazine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL29795799	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(C(=O)CC5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H46ClN7O6	AR	P10275	CRBN	WO-2022187419-A1
TPD-GLZP8Y	SCHEMBL23125088	2-chloro-4-[(3S)-8-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxospiro[5,7-dihydrocyclopenta[f]isoindole-6,3'-azetidine]-1'-yl]piperidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL29788784	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(N5CC6(Cc7cc8c(cc7C6)C(=O)N(C6CCC(=O)NC6=O)C8=O)C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C46H48ClN7O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-47NNOF	SCHEMBL23125102	2-chloro-4-[(3S)-8-[4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxospiro[5,7-dihydrocyclopenta[f]isoindole-6,3'-azetidine]-1'-yl]methyl]piperidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL29796048	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(CN5CC6(Cc7cc8c(cc7C6)C(=O)N(C6CCC(=O)NC6=O)C8=O)C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C47H50ClN7O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-JV8VFB	SCHEMBL23125406	2-chloro-4-[(3S)-8-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxospiro[5,7-dihydrocyclopenta[f]isoindole-6,4'-piperidine]-1'-yl]piperidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL29788768	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(N5CCC6(CC5)Cc5cc7c(cc5C6)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C48H52ClN7O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-CP7BXM	SCHEMBL23125266	2-chloro-4-[(3S)-8-[4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxospiro[5,7-dihydrocyclopenta[f]isoindole-6,4'-piperidine]-1'-yl]methyl]piperidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL29795853	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(CN5CCC6(CC5)Cc5cc7c(cc5C6)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C49H54ClN7O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-3VHW65	CHEMBL5415103	2-chloro-4-[(3S)-8-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL23125355; SCHEMBL29795822	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(CN5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C46H51ClN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-JOKG7B	CHEMBL5410066	2-chloro-4-[(3S)-8-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]piperidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL23125368; SCHEMBL29795956	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(N5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H49ClN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-O3M5IS	SCHEMBL23125112	2-chloro-4-[(3S)-8-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL29795995	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(CN5CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C46H50ClFN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-OJQWSC	SCHEMBL23125092	2-chloro-4-[(3S)-8-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]piperidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL29795781	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(N5CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H48ClFN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-AZXKNR	SCHEMBL23125333	2-chloro-4-[(3S)-8-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]piperidin-1-yl]benzoyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(C(=O)c3ccc(N4CCC(N5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H44ClN7O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-CA9P80	SCHEMBL23125209	2-chloro-4-[(3S)-8-[2-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidine-1-carbonyl]pyrimidin-5-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL29795999	C[C@H]1CC2(CCN(c3cnc(C(=O)N4CCC(CN5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H49ClN10O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-47P1ID	SCHEMBL23125097	2-chloro-4-[(3S)-8-[6-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidine-1-carbonyl]pyridazin-3-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL29795908	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(CN5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)nn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H49ClN10O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-U1JXBV	SCHEMBL23138726	2-chloro-4-[(3S)-8-[4-[(3S)-3-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]pyrrolidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CC[C@@H](CN5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H49ClN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-DSLZDA	SCHEMBL23138727	2-chloro-4-[(3S)-8-[4-[(3R)-3-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]pyrrolidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CC[C@@H](N5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H47ClN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-97UOYL	WO2022187419A1_A74	.	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(CN5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H50ClN9O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-I09P7K	WO2022187419A1_A76	.	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(CN5CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H49ClFN9O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-F5XOPW	WO2022187419A1_A77	.	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(N5CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H47ClFN9O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-PX7TYJ	WO2022187419A1_A78	.	C[C@H]1CC2(CCN(c3cnc(C(=O)N4CCC(CN5CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H48ClFN10O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-I9BHQ5	WO2022187419A1_A79	.	C[C@H]1CC2(CCN(c3cnc(C(=O)N4CCC(N5CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H46ClFN10O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-KBKIDN	SCHEMBL23125256	2-chloro-4-[(3S)-8-[4-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-3-oxo-1H-isoindol-5-yl]azetidin-3-yl]piperazine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL29796009	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7)C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H47ClN8O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-6A01Q8	SCHEMBL23125146	2-chloro-4-[(3S)-8-[6-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidine-1-carbonyl]pyridazin-3-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL29795978	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(CN5CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)nn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H48ClFN10O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-80H0UQ	WO2022187419A1_A82	.	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CC[C@@H](CN5CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H48ClFN8O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-HN7V2X	SCHEMBL23138975	2-chloro-4-[(3S)-8-[2-[(3S)-3-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]pyrrolidine-1-carbonyl]pyrimidin-5-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3cnc(C(=O)N4CC[C@@H](CN5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H47ClN10O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-CRBOGH	SCHEMBL23138976	2-chloro-4-[(3S)-8-[2-[(3R)-3-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]pyrrolidine-1-carbonyl]pyrimidin-5-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3cnc(C(=O)N4CC[C@@H](N5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H45ClN10O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-CT0EQU	SCHEMBL23138973	2-chloro-4-[(3S)-8-[6-[(3S)-3-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]pyrrolidine-1-carbonyl]pyridazin-3-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CC[C@@H](CN5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)nn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H47ClN10O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-JT6U0Q	SCHEMBL23138974	2-chloro-4-[(3S)-8-[6-[(3R)-3-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]pyrrolidine-1-carbonyl]pyridazin-3-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CC[C@@H](N5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)nn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H45ClN10O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-5EY7T9	SCHEMBL23138055	2-chloro-4-[(3S)-8-[4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxopyrrolo[3,4-f]isoindol-6-yl]methyl]piperidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(Cn5cc6cc7c(cc6c5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H44ClN7O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-MN7LOL	SCHEMBL23138027	2-chloro-4-[(3S)-8-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxopyrrolo[3,4-f]isoindol-6-yl]piperidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(n5cc6cc7c(cc6c5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H42ClN7O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-IB4TG7	SCHEMBL23138891	2-chloro-4-[(3S)-8-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-6-yl]piperidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(N5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H46ClN7O4	AR	P10275	CRBN	WO-2022187419-A1
TPD-KOHUOK	SCHEMBL23125350	2-chloro-4-[(3S)-8-[6-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]methyl]piperazine-1-carbonyl]pyridazin-3-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL29796071	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(CC5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)nn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H45ClN10O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-FAK1HS	SCHEMBL23138978	2-chloro-4-[(3S)-8-[5-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]methyl]piperazine-1-carbonyl]pyrazin-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3cnc(C(=O)N4CCN(CC5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H45ClN10O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-OX10J3	SCHEMBL23124934	2-chloro-4-[(3S)-8-[5-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]azetidin-3-yl]methyl]piperazine-1-carbonyl]pyrazin-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL29796006	C[C@H]1CC2(CCN(c3cnc(C(=O)N4CCN(CC5CN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H44ClFN10O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-1Q3CDS	SCHEMBL23125170	2-chloro-4-[(3S)-8-[6-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazine-1-carbonyl]pyridazin-3-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL29796025	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(CC5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)nn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H49ClN10O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-4MNQAZ	SCHEMBL23125109	2-chloro-4-[(3S)-8-[5-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidine-1-carbonyl]pyrazin-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL29795848	C[C@H]1CC2(CCN(c3cnc(C(=O)N4CCC(CN5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H49ClN10O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-1F7OPB	SCHEMBL23125254	2-chloro-4-[(3S)-8-[5-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidine-1-carbonyl]pyrazin-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL29796023	C[C@H]1CC2(CCN(c3cnc(C(=O)N4CCC(CN5CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H48ClFN10O5	AR	P10275	CRBN	WO-2022187419-A1
TPD-BFU8XQ	SCHEMBL27239381	3-[6-[[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC4=C(C=C3C2=O)CN(CC2CCN(C3=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=CC=C5)C=C3)CC2)C4)C(=O)N1	C43H44N4O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-GEXC5E	ERD-821	2-(2,6-dioxopiperidin-3-yl)-6-[[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; CHEMBL5415025; SCHEMBL27239531	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC2CCN(C3=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=CC=C5)C=C3)CC2)C4)C(=O)N1	C43H42N4O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-O17H7F	SCHEMBL27239517	3-[6-[1-[[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperidin-4-yl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC4=C(C=C3C2=O)CN(C2CCN(CC3CCN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC3)CC2)C4)C(=O)N1	C48H53N5O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-I772S8	SCHEMBL27239387	3-[6-[2-[8-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-2,8-diazaspiro[4.5]decan-2-yl]-2-oxoethyl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC4=C(C=C3C2=O)CN(CC(=O)N2CCC3(CCN(C5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC3)C2)C4)C(=O)N1	C47H49N5O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-ODODF6	SCHEMBL27239165	3-[6-[2-[2-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-2,7-diazaspiro[3.5]nonan-7-yl]-2-oxoethyl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC4=C(C=C3C2=O)CN(CC(=O)N2CCC3(CC2)CN(C2=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=CC=C5)C=C2)C3)C4)C(=O)N1	C46H47N5O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-XF67I3	SCHEMBL27239198	3-[6-[2-[2-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-2,7-diazaspiro[3.4]octan-7-yl]-2-oxoethyl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC4=C(C=C3C2=O)CN(CC(=O)N2CCC3(C2)CN(C2=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=CC=C5)C=C2)C3)C4)C(=O)N1	C45H45N5O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-0WXEWF	ERD-851	2-(2,6-dioxopiperidin-3-yl)-6-[2-[8-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-2,8-diazaspiro[4.5]decan-2-yl]-2-oxoethyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; CHEMBL5400354; SCHEMBL27239251	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC(=O)N2CCC3(CCN(C5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC3)C2)C4)C(=O)N1	C47H47N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-IV4FJK	ERD-853	2-(2,6-dioxopiperidin-3-yl)-6-[2-[6-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-2,6-diazaspiro[3.3]heptan-2-yl]-2-oxoethyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; CHEMBL5434699; SCHEMBL27239269; SCHEMBL29911887	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC(=O)N2CC3(C2)CN(C2=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=CC=C5)C=C2)C3)C4)C(=O)N1	C44H41N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-CF2HP4	ERD-1152	2-(2,6-dioxopiperidin-3-yl)-6-[2-[7-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-2,7-diazaspiro[3.5]nonan-2-yl]-2-oxoethyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; CHEMBL5427139; SCHEMBL27239295; SCHEMBL30934183	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC(=O)N2CC3(CCN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC3)C2)C4)C(=O)N1	C46H45N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-621ZMV	ERD-856	2-(2,6-dioxopiperidin-3-yl)-6-[2-[2-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-2,7-diazaspiro[3.5]nonan-7-yl]-2-oxoethyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; CHEMBL5396338; SCHEMBL27239238	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC(=O)N2CCC3(CC2)CN(C2=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=CC=C5)C=C2)C3)C4)C(=O)N1	C46H45N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-C56CDX	SCHEMBL27239440	6-[2-[2-[4-[(1R,2S)-2-(2-chloro-4-fluorophenyl)-6-hydroxy-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-2,7-diazaspiro[3.5]nonan-7-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC(=O)N2CCC3(CC2)CN(C2=CC=C([C@@H]5C6=C(C=C(O)C=C6)CC[C@@H]5C5=CC=C(F)C=C5Cl)C=C2)C3)C4)C(=O)N1	C46H43ClFN5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-FUNFXB	SCHEMBL27239494	2-(2,6-dioxopiperidin-3-yl)-6-[1-[1-[4-[(1R,2S)-2-(4-fluorophenyl)-6-hydroxy-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]piperidine-4-carbonyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=C(C=C4CN(C(=O)C5CCN(C6CCN(C7=CC=C([C@@H]8C9=C(C=C(O)C=C9)CC[C@@H]8C8=CC=C(F)C=C8)C=C7)CC6)CC5)CC4=C3)C2=O)C(=O)N1	C48H48FN5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-HV1JYP	WO2022187588A1_E013	.	C=C/C=C\C(=C)[C@@H](C)[C@H](C1=CC=C(N2CCC(C(=O)N3CCC(N4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)CC2)C=C1)C1=CC=C(O)C=C1C	C48H53N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-J41XFQ	ERD-10108	2-(2,6-dioxopiperidin-3-yl)-6-[[1-[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidine-4-carbonyl]piperidin-4-yl]methyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; CHEMBL5397189; SCHEMBL27239275; SCHEMBL30934523	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC2CCN(C(=O)C3CCN(C5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC3)CC2)C4)C(=O)N1	C49H51N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-VKT01B	SCHEMBL27239152	2-(2,6-dioxopiperidin-3-yl)-6-[1-[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidine-4-carbonyl]azetidin-3-yl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(C2CN(C(=O)C3CCN(C5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC3)C2)C4)C(=O)N1	C46H45N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-TPQB2G	WO2022187588A1_E016	.	O=C1CCC(N2C(=O)C3=CC4CN(CC5CN(C(=O)C6CCN(C7=CC=C([C@@H]8C9=C(C=C(O)C=C9)CC[C@@H]8C8=CC=CC=C8)C=C7)CC6)C5)CC4C=C3C2=O)C(=O)N1	C47H49N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-04Q0EN	ERD-854	2-(2,6-dioxopiperidin-3-yl)-6-[2-[2-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-2,7-diazaspiro[3.4]octan-7-yl]-2-oxoethyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; CHEMBL5437374; SCHEMBL27239467	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC(=O)N2CCC3(C2)CN(C2=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=CC=C5)C=C2)C3)C4)C(=O)N1	C45H43N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-9IICDJ	SCHEMBL27239210	2-(2,6-dioxopiperidin-3-yl)-6-[2-[6-[4-[(1R,2S)-2-(4-fluorophenyl)-6-hydroxy-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-2,6-diazaspiro[3.3]heptan-2-yl]-2-oxoethyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC(=O)N2CC3(C2)CN(C2=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=C(F)C=C5)C=C2)C3)C4)C(=O)N1	C44H40FN5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-W0J3E5	SCHEMBL27239630	2-(2,6-dioxopiperidin-3-yl)-6-[2-[7-[4-[(1R,2S)-2-(4-fluorophenyl)-6-hydroxy-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-2,7-diazaspiro[3.5]nonan-2-yl]-2-oxoethyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC(=O)N2CC3(CCN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=C(F)C=C6)C=C5)CC3)C2)C4)C(=O)N1	C46H44FN5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-229EOM	ERD-1173	2-(2,6-dioxopiperidin-3-yl)-6-[2-[9-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-oxoethyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; CHEMBL5439513; SCHEMBL27239235; SCHEMBL29911559	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC(=O)N2CCC3(CC2)CCN(C2=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=CC=C5)C=C2)CC3)C4)C(=O)N1	C48H49N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-VUAA2D	SCHEMBL27239221	2-(2,6-dioxopiperidin-3-yl)-6-[2-[3-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]piperidin-1-yl]-2-oxoethyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934170	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC(=O)N2CCCC(OC3=CC=C([C@@H]5C6=C(C=C(O)C=C6)CC[C@@H]5C5=CC=CC=C5)C=C3)C2)C4)C(=O)N1	C44H42N4O7	ERα	P03372	CRBN	WO-2022187588-A1
TPD-GDQRAW	SCHEMBL27239435	2-(2,6-dioxopiperidin-3-yl)-6-[3-[3-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]piperidine-1-carbonyl]cyclobutyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934264	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(C2CC(C(=O)N3CCCC(OC5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)C3)C2)C4)C(=O)N1	C47H46N4O7	ERα	P03372	CRBN	WO-2022187588-A1
TPD-LYLY37	SCHEMBL27239239	2-(2,6-dioxopiperidin-3-yl)-6-[4-[3-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]piperidine-1-carbonyl]cyclohexyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934376	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(C2CCC(C(=O)N3CCCC(OC5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)C3)CC2)C4)C(=O)N1	C49H50N4O7	ERα	P03372	CRBN	WO-2022187588-A1
TPD-568UNP	SCHEMBL27239516	2-(2,6-dioxopiperidin-3-yl)-6-[4-[2-[3-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]piperidin-1-yl]-2-oxoethyl]benzoyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934451	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(C(=O)C2=CC=C(CC(=O)N3CCCC(OC5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)C3)C=C2)C4)C(=O)N1	C51H46N4O8	ERα	P03372	CRBN	WO-2022187588-A1
TPD-QCI18W	SCHEMBL27239474	6-[2-[2-[4-[(1S,3R)-2-(2,2-difluoropropyl)-6-hydroxy-3-methyl-3,4-dihydro-1H-isoquinolin-1-yl]-3,5-difluorophenyl]-2,7-diazaspiro[3.5]nonan-7-yl]acetyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934219	C[C@@H]1CC2=CC(O)=CC=C2[C@@H](C2=C(F)C=C(N3CC4(CCN(CC(=O)N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C3)C=C2F)N1CC(C)(F)F	C43H44F4N6O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-RA5CVV	SCHEMBL27239268	3-[6-[2-[2-[4-[(1S,3R)-2-(2,2-difluoropropyl)-6-hydroxy-3-methyl-3,4-dihydro-1H-isoquinolin-1-yl]-3,5-difluorophenyl]-2,7-diazaspiro[3.5]nonan-7-yl]acetyl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30934123	C[C@@H]1CC2=CC(O)=CC=C2[C@@H](C2=C(F)C=C(N3CC4(CCN(CC(=O)N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)C5)CC4)C3)C=C2F)N1CC(C)(F)F	C43H46F4N6O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-DYA594	SCHEMBL27239285	3-[6-[2-[2-[4-[(1S,3R)-2-(2,2-difluoropropyl)-6-hydroxy-3-methyl-3,4-dihydro-1H-isoquinolin-1-yl]-3,5-difluorophenyl]-2,7-diazaspiro[3.5]nonan-7-yl]-2-oxoethyl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30934190	C[C@@H]1CC2=CC(O)=CC=C2[C@@H](C2=C(F)C=C(N3CC4(CCN(C(=O)CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)C5)CC4)C3)C=C2F)N1CC(C)(F)F	C43H46F4N6O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-B63XJU	SCHEMBL27239582	3-[6-[2-[7-[4-[(1S,3R)-2-(2,2-difluoropropyl)-6-hydroxy-3-methyl-3,4-dihydro-1H-isoquinolin-1-yl]-3,5-difluorophenyl]-2,7-diazaspiro[4.4]nonan-2-yl]-2-oxoethyl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30934401	C[C@@H]1CC2=CC(O)=CC=C2[C@@H](C2=C(F)C=C(N3CCC4(CCN(C(=O)CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)C5)C4)C3)C=C2F)N1CC(C)(F)F	C43H46F4N6O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-TTN51N	SCHEMBL27239469	6-[1-[1-[4-[(1S,3R)-2-(2,2-difluoropropyl)-6-hydroxy-3-methyl-3,4-dihydro-1H-isoquinolin-1-yl]-3,5-difluorophenyl]piperidin-4-yl]piperidine-4-carbonyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934326	C[C@@H]1CC2=CC(O)=CC=C2[C@@H](C2=C(F)C=C(N3CCC(N4CCC(C(=O)N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2F)N1CC(C)(F)F	C45H48F4N6O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-E2Y14C	SCHEMBL27239496	3-[6-[1-[1-[4-[(1S,3R)-2-(2,2-difluoropropyl)-6-hydroxy-3-methyl-3,4-dihydro-1H-isoquinolin-1-yl]-3,5-difluorophenyl]piperidin-4-yl]piperidine-4-carbonyl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30934444	C[C@@H]1CC2=CC(O)=CC=C2[C@@H](C2=C(F)C=C(N3CCC(N4CCC(C(=O)N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)C5)CC4)CC3)C=C2F)N1CC(C)(F)F	C45H50F4N6O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-IEBFDH	SCHEMBL27239160	6-[2-[2-[4-[(1S,3R)-2-(2,2-difluoropropyl)-6-hydroxy-3-methyl-3,4-dihydro-1H-isoquinolin-1-yl]-3,5-difluorophenyl]-2,7-diazaspiro[4.4]nonan-7-yl]acetyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934239	C[C@@H]1CC2=CC(O)=CC=C2[C@@H](C2=C(F)C=C(N3CCC4(CCN(CC(=O)N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)C4)C3)C=C2F)N1CC(C)(F)F	C43H44F4N6O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-74XKFD	SCHEMBL27239158	3-[6-[2-[2-[4-[(1S,3R)-2-(2,2-difluoropropyl)-6-hydroxy-3-methyl-3,4-dihydro-1H-isoquinolin-1-yl]-3,5-difluorophenyl]-2,7-diazaspiro[4.4]nonan-7-yl]acetyl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30934492	C[C@@H]1CC2=CC(O)=CC=C2[C@@H](C2=C(F)C=C(N3CCC4(CCN(CC(=O)N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)C5)C4)C3)C=C2F)N1CC(C)(F)F	C43H46F4N6O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-O4YAHW	SCHEMBL27239380	6-[2-[8-[4-[(1S,3R)-2-(2,2-difluoropropyl)-6-hydroxy-3-methyl-3,4-dihydro-1H-isoquinolin-1-yl]-3,5-difluorophenyl]-2,8-diazaspiro[4.5]decan-2-yl]acetyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934224	C[C@@H]1CC2=CC(O)=CC=C2[C@@H](C2=C(F)C=C(N3CCC4(CCN(CC(=O)N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)C4)CC3)C=C2F)N1CC(C)(F)F	C44H46F4N6O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-NNYLVT	SCHEMBL27239460	3-[6-[2-[8-[4-[(1S,3R)-2-(2,2-difluoropropyl)-6-hydroxy-3-methyl-3,4-dihydro-1H-isoquinolin-1-yl]-3,5-difluorophenyl]-2,8-diazaspiro[4.5]decan-2-yl]acetyl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30934061	C[C@@H]1CC2=CC(O)=CC=C2[C@@H](C2=C(F)C=C(N3CCC4(CCN(CC(=O)N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)C5)C4)CC3)C=C2F)N1CC(C)(F)F	C44H48F4N6O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-2EJ1YV	SCHEMBL30934445	3-[6-[2-[7-[4-[(1S,3R)-2-(2,2-difluoroethyl)-6-hydroxy-3-methyl-3,4-dihydro-1H-isoquinolin-1-yl]-3,5-difluorophenyl]-2,7-diazaspiro[3.5]nonan-2-yl]-2-oxoethyl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione	C[C@@H]1CC2=CC(O)=CC=C2[C@@H](C2=C(F)C=C(N3CCC4(CC3)CN(C(=O)CN3CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)CC6=C5)C3)C4)C=C2F)N1CC(F)F	C42H44F4N6O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-CGVEO8	WO2022187588A1_E036	.	C[C@@H]1CC2=CC(O)=CC=C2[C@@H](C2=C(F)C=C(N3CC4(CCN(C(=O)CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)C5)C4)C3)C=C2F)N1CC(F)F	C41H42F4N6O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-9X7OSF	SCHEMBL27239330	3-[6-[2-[7-[4-[(1S,3R)-2-(2,2-difluoroethyl)-6-hydroxy-3-methyl-3,4-dihydro-1H-isoquinolin-1-yl]-3,5-difluorophenyl]-2,7-diazaspiro[3.4]octan-2-yl]-2-oxoethyl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30934234	C[C@@H]1CC2=CC(O)=CC=C2[C@@H](C2=C(F)C=C(N3CCC4(CN(C(=O)CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)C5)C4)C3)C=C2F)N1CC(F)F	C41H42F4N6O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-3ZPZ2Y	SCHEMBL27239305	3-[6-[2-[7-[4-[(1S,3R)-2-(2,2-difluoroethyl)-6-hydroxy-3-methyl-3,4-dihydro-1H-isoquinolin-1-yl]-3,5-difluorophenyl]-2,7-diazaspiro[3.4]octan-2-yl]acetyl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30934317	C[C@@H]1CC2=CC(O)=CC=C2[C@@H](C2=C(F)C=C(N3CCC4(CN(CC(=O)N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)C5)C4)C3)C=C2F)N1CC(F)F	C41H42F4N6O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-RJDRNM	SCHEMBL30934231	3-[6-[2-[7-[4-[(1S,3R)-2-(2,2-difluoroethyl)-6-hydroxy-3-methyl-3,4-dihydro-1H-isoquinolin-1-yl]-3,5-difluorophenyl]-2,7-diazaspiro[3.5]nonan-2-yl]acetyl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione	C[C@@H]1CC2=CC(O)=CC=C2[C@@H](C2=C(F)C=C(N3CCC4(CC3)CN(CC(=O)N3CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)CC6=C5)C3)C4)C=C2F)N1CC(F)F	C42H44F4N6O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-0TDIHX	SCHEMBL27239462	3-[6-[2-[2-[4-[(1S,3R)-2-(2,2-difluoroethyl)-6-hydroxy-3-methyl-3,4-dihydro-1H-isoquinolin-1-yl]-3,5-difluorophenyl]-2,7-diazaspiro[3.4]octan-7-yl]acetyl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30934210	C[C@@H]1CC2=CC(O)=CC=C2[C@@H](C2=C(F)C=C(N3CC4(CCN(CC(=O)N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)C5)C4)C3)C=C2F)N1CC(F)F	C41H42F4N6O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-RCC7AS	SCHEMBL27239477	6-[2-[7-[4-[(1S,3R)-2-(2,2-difluoroethyl)-6-hydroxy-3-methyl-3,4-dihydro-1H-isoquinolin-1-yl]-3,5-difluorophenyl]-2,7-diazaspiro[3.5]nonan-2-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934269	C[C@@H]1CC2=CC(O)=CC=C2[C@@H](C2=C(F)C=C(N3CCC4(CC3)CN(C(=O)CN3CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C3)C4)C=C2F)N1CC(F)F	C42H42F4N6O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-V6RYOO	SCHEMBL27239536	6-[2-[6-[4-[(1S,3R)-2-(2,2-difluoroethyl)-6-hydroxy-3-methyl-3,4-dihydro-1H-isoquinolin-1-yl]-3,5-difluorophenyl]-2,6-diazaspiro[3.3]heptan-2-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934421	C[C@@H]1CC2=CC(O)=CC=C2[C@@H](C2=C(F)C=C(N3CC4(CN(C(=O)CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)C4)C3)C=C2F)N1CC(F)F	C40H38F4N6O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-MMW5OF	SCHEMBL27239597	6-[2-[2-[4-[(1S,3R)-2-(2,2-difluoroethyl)-6-hydroxy-3-methyl-3,4-dihydro-1H-isoquinolin-1-yl]-3,5-difluorophenyl]-2,7-diazaspiro[3.4]octan-7-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934381	C[C@@H]1CC2=CC(O)=CC=C2[C@@H](C2=C(F)C=C(N3CC4(CCN(C(=O)CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)C4)C3)C=C2F)N1CC(F)F	C41H40F4N6O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-I4BCEN	SCHEMBL27239446	6-[2-[7-[4-[(1S,3R)-2-(2,2-difluoroethyl)-6-hydroxy-3-methyl-3,4-dihydro-1H-isoquinolin-1-yl]-3,5-difluorophenyl]-2,7-diazaspiro[3.4]octan-2-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934255	C[C@@H]1CC2=CC(O)=CC=C2[C@@H](C2=C(F)C=C(N3CCC4(CN(C(=O)CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)C4)C3)C=C2F)N1CC(F)F	C41H40F4N6O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-9CGZCY	SCHEMBL27239281	6-[2-[2-[4-[(1S,3R)-2-(2,2-difluoroethyl)-6-hydroxy-3-methyl-3,4-dihydro-1H-isoquinolin-1-yl]-3,5-difluorophenyl]-2,7-diazaspiro[3.5]nonan-7-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934375	C[C@@H]1CC2=CC(O)=CC=C2[C@@H](C2=C(F)C=C(N3CC4(CCN(C(=O)CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C3)C=C2F)N1CC(F)F	C42H42F4N6O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-7EUDMV	SCHEMBL27239297	6-[[1-[1-[4-[(1S,3R)-2-(2,2-difluoroethyl)-6-hydroxy-3-methyl-3,4-dihydro-1H-isoquinolin-1-yl]-3,5-difluorophenyl]piperidin-4-yl]azetidin-3-yl]methyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934434	C[C@@H]1CC2=CC(O)=CC=C2[C@@H](C2=C(F)C=C(N3CCC(N4CC(CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)C4)CC3)C=C2F)N1CC(F)F	C42H44F4N6O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-79RWN2	SCHEMBL27239577	6-[1-[[1-[4-[(1S,3R)-2-(2,2-difluoroethyl)-6-hydroxy-3-methyl-3,4-dihydro-1H-isoquinolin-1-yl]-3,5-difluorophenyl]piperidin-4-yl]methyl]azetidin-3-yl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934182	C[C@@H]1CC2=CC(O)=CC=C2[C@@H](C2=C(F)C=C(N3CCC(CN4CC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)C4)CC3)C=C2F)N1CC(F)F	C42H44F4N6O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-KD5K8X	SCHEMBL30934253	3-[6-[2-[2-[4-[6-(4-fluorophenyl)-2-hydroxy-8,9-dihydro-7H-benzo[7]annulen-5-yl]phenyl]-2,6-diazaspiro[3.3]heptan-6-yl]acetyl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC4=C(C=C3C2=O)CN(C(=O)CN2CC3(C2)CN(C2=CC=C(C5=C(C6=CC=C(F)C=C6)CCCC6=CC(O)=CC=C65)C=C2)C3)C4)C(=O)N1	C45H42FN5O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-OLA3WF	SCHEMBL27239419	2-(2,6-dioxopiperidin-3-yl)-6-[2-[2-[4-[6-(4-fluorophenyl)-2-hydroxy-8,9-dihydro-7H-benzo[7]annulen-5-yl]phenyl]-2,6-diazaspiro[3.3]heptan-6-yl]acetyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL29911854	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(C(=O)CN2CC3(C2)CN(C2=CC=C(C5=C(C6=CC=C(F)C=C6)CCCC6=CC(O)=CC=C65)C=C2)C3)C4)C(=O)N1	C45H40FN5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-WTUHAH	SCHEMBL27239265	6-[1-[[1-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]piperidin-4-yl]methyl]azetidin-3-yl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934055	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCC(CN4CC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)C4)CC3)C=C2F)N1CC(F)F	C44H45F4N7O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-NYWKKZ	SCHEMBL27239396	6-[1-[[1-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]piperidin-4-yl]methyl]piperidin-4-yl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934462	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCC(CN4CCC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2F)N1CC(F)F	C46H49F4N7O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-EALEME	SCHEMBL27239227	3-[6-[1-[[1-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]piperidin-4-yl]methyl]azetidin-3-yl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30934322	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCC(CN4CC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)C5)C4)CC3)C=C2F)N1CC(F)F	C44H47F4N7O3	ERα	P03372	CRBN	WO-2022187588-A1
TPD-3MA94O	SCHEMBL27239302	3-[6-[2-[4-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]piperazin-1-yl]ethyl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30934241	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCN(CCN4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)CC6=C5)C4)CC3)C=C2F)N1CC(F)F	C41H43F4N7O3	ERα	P03372	CRBN	WO-2022187588-A1
TPD-T0WFZ2	SCHEMBL27239427	6-[2-[1-[1-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]piperidin-4-yl]azetidin-3-yl]acetyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934141	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCC(N4CC(CC(=O)N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)C4)CC3)C=C2F)N1CC(F)F	C45H45F4N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-T1Z292	SCHEMBL27239220	3-[6-[2-[1-[1-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]piperidin-4-yl]azetidin-3-yl]acetyl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30934069	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCC(N4CC(CC(=O)N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)C5)C4)CC3)C=C2F)N1CC(F)F	C45H47F4N7O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-HQYBE5	SCHEMBL27239171	6-[1-[[1-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]pyrrolidin-3-yl]methyl]piperidine-4-carbonyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934129	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCC(CN4CCC(C(=O)N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C3)C=C2F)N1CC(F)F	C46H47F4N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-A42EA4	SCHEMBL27239258	6-[1-[[1-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]piperidin-3-yl]methyl]piperidine-4-carbonyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934328	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCCC(CN4CCC(C(=O)N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C3)C=C2F)N1CC(F)F	C47H49F4N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-6Q1RXE	SCHEMBL27239219	6-[1-[[1-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]piperidin-3-yl]methyl]piperidin-4-yl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934399	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCCC(CN4CCC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C3)C=C2F)N1CC(F)F	C46H49F4N7O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-0U0Z0H	SCHEMBL27239561	6-[2-[6-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]-1,6-diazaspiro[3.3]heptan-1-yl]acetyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934198	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CC4(CCN4CC(=O)N4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)C3)C=C2F)N1CC(F)F	C42H39F4N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-L8V8GK	SCHEMBL27239321	3-[6-[2-[6-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]-1,6-diazaspiro[3.3]heptan-1-yl]acetyl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30934300	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CC4(CCN4CC(=O)N4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)CC6=C5)C4)C3)C=C2F)N1CC(F)F	C42H41F4N7O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-4OWT58	SCHEMBL27239340	6-[2-[8-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]-2,8-diazaspiro[4.5]decan-2-yl]acetyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934212	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCC4(CCN(CC(=O)N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)C4)CC3)C=C2F)N1CC(F)F	C45H45F4N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-2VSQQC	SCHEMBL27239214	3-[6-[2-[8-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]-2,8-diazaspiro[4.5]decan-2-yl]acetyl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30934456	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCC4(CCN(CC(=O)N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)C5)C4)CC3)C=C2F)N1CC(F)F	C45H47F4N7O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-MYBWMK	SCHEMBL27239447	3-[6-[2-[8-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]-2,8-diazaspiro[4.5]decan-2-yl]-2-oxoethyl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30934094	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCC4(CCN(C(=O)CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)C5)C4)CC3)C=C2F)N1CC(F)F	C45H47F4N7O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-0DSKH5	SCHEMBL27239358	3-[6-[2-[2-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]-2,6-diazaspiro[3.3]heptan-6-yl]acetyl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30934289	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CC4(CN(CC(=O)N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)C5)C4)C3)C=C2F)N1CC(F)F	C42H41F4N7O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-YK3D01	SCHEMBL27239432	3-[6-[2-[2-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]-2,7-diazaspiro[3.4]octan-7-yl]-2-oxoethyl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30934373	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CC4(CCN(C(=O)CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)C5)C4)C3)C=C2F)N1CC(F)F	C43H43F4N7O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-F7OZXS	SCHEMBL27239490	3-[6-[2-[9-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]-2,9-diazaspiro[4.5]decan-2-yl]-2-oxoethyl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30934310	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCCC4(CCN(C(=O)CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)C5)C4)C3)C=C2F)N1CC(F)F	C45H47F4N7O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-DXUA5E	SCHEMBL27239538	3-[6-[2-[7-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]-2,7-diazaspiro[4.4]nonan-2-yl]-2-oxoethyl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30934347	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCC4(CCN(C(=O)CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)C5)C4)C3)C=C2F)N1CC(F)F	C44H45F4N7O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-RQK7SR	WO2022187588A1_E069	6-[2-[2-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]-2,8-diazaspiro[3.5]nonan-8-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CC4(CCCN(C(=O)CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)C4)C3)C=C2F)N1CC(F)F	C44H43F4N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-8THSYQ	SCHEMBL27239337	3-[6-[2-[8-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]-2,8-diazaspiro[3.5]nonan-2-yl]-2-oxoethyl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30934114	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCCC4(CN(C(=O)CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)C5)C4)C3)C=C2F)N1CC(F)F	C44H45F4N7O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-F120W4	SCHEMBL27239262	3-[6-[2-[6-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]-2,6-diazaspiro[3.3]heptan-2-yl]-2-oxoethyl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30934387	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CC4(CN(C(=O)CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)C5)C4)C3)C=C2F)N1CC(F)F	C42H41F4N7O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-KHK46J	SCHEMBL27239261	3-[6-[2-[7-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]-2,7-diazaspiro[3.4]octan-2-yl]-2-oxoethyl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30934437	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCC4(CN(C(=O)CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)C5)C4)C3)C=C2F)N1CC(F)F	C43H43F4N7O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-HCA597	SCHEMBL27239359	3-[6-[2-[2-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]-2,7-diazaspiro[3.4]octan-7-yl]acetyl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30934350	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CC4(CCN(CC(=O)N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)C5)C4)C3)C=C2F)N1CC(F)F	C43H43F4N7O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-62NOJS	SCHEMBL27239509	6-[2-[2-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]-2,7-diazaspiro[3.4]octan-7-yl]acetyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934151	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CC4(CCN(CC(=O)N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)C4)C3)C=C2F)N1CC(F)F	C43H41F4N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-TUA9KG	SCHEMBL27239544	3-[6-[2-[2-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]-2,7-diazaspiro[4.4]nonan-7-yl]acetyl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30934214	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCC4(CCN(CC(=O)N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)C5)C4)C3)C=C2F)N1CC(F)F	C44H45F4N7O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-JBZZHA	SCHEMBL27239290	6-[2-[2-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]-2,7-diazaspiro[4.4]nonan-7-yl]acetyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934517	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCC4(CCN(CC(=O)N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)C4)C3)C=C2F)N1CC(F)F	C44H43F4N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-RCVACX	SCHEMBL27239209	6-[2-[2-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]-2,7-diazaspiro[3.4]octan-7-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934446	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CC4(CCN(C(=O)CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)C4)C3)C=C2F)N1CC(F)F	C43H41F4N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-HK1ZT0	SCHEMBL27239343	6-[2-[9-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]-2,9-diazaspiro[4.5]decan-2-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934261	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCCC4(CCN(C(=O)CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)C4)C3)C=C2F)N1CC(F)F	C45H45F4N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-K5ORG7	SCHEMBL27239218	6-[2-[7-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]-2,7-diazaspiro[4.4]nonan-2-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934384	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCC4(CCN(C(=O)CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)C4)C3)C=C2F)N1CC(F)F	C44H43F4N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-2NCJB6	WO2022187588A1_E081	.	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCCC4(CN(C(=O)CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)C4)C3)C=C2F)N1CC(F)F	C44H43F4N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-A8ONI9	SCHEMBL27239309	6-[2-[6-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]-2,6-diazaspiro[3.3]heptan-2-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934324	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CC4(CN(C(=O)CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)C4)C3)C=C2F)N1CC(F)F	C42H39F4N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-C1ZDXQ	SCHEMBL27239623	6-[2-[7-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]-2,7-diazaspiro[3.4]octan-2-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934426	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCC4(CN(C(=O)CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)C4)C3)C=C2F)N1CC(F)F	C43H41F4N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-83B8MM	WO2022187588A1_E084	6-[2-[2-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]-2,7-diazaspiro[3.5]nonan-7-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CC4(CCN(C(=O)CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C3)C=C2F)N1CC(F)F	C44H43F4N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-H19NZR	WO2022187588A1_E085	3-[6-[2-[2-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]-2,7-diazaspiro[3.5]nonan-7-yl]-2-oxoethyl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CC4(CCN(C(=O)CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)C5)CC4)C3)C=C2F)N1CC(F)F	C44H45F4N7O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-V1AD0P	SCHEMBL27239339	3-[6-[[1-[1-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]piperidin-4-yl]piperidin-4-yl]methyl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30934369	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCC(N4CCC(CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)C5)CC4)CC3)C=C2F)N1CC(F)F	C46H51F4N7O3	ERα	P03372	CRBN	WO-2022187588-A1
TPD-HV0M8P	SCHEMBL30934131	6-[1-[1-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]piperidin-4-yl]piperidin-4-yl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCC(N4CCC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2F)N1CC(F)F	C45H47F4N7O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-FLZ93D	SCHEMBL27239605	6-[1-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]piperidin-4-yl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934275	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCC(N4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=C2F)N1CC(F)F	C40H38F4N6O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-TTEZCR	SCHEMBL27239433	6-[[1-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]piperidin-4-yl]methyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934073	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCC(CN4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C=C2F)N1CC(F)F	C41H40F4N6O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-FOKUYO	SCHEMBL27239273	3-[6-[1-[[(3S)-1-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]pyrrolidin-3-yl]methyl]piperidine-4-carbonyl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30934320	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CC[C@@H](CN4CCC(C(=O)N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)C5)CC4)C3)C=C2F)N1CC(F)F	C46H49F4N7O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-IINWNR	SCHEMBL27239168	6-[1-[[(3S)-1-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]pyrrolidin-3-yl]methyl]piperidine-4-carbonyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934108	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CC[C@@H](CN4CCC(C(=O)N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C3)C=C2F)N1CC(F)F	C46H47F4N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-AL8W3O	SCHEMBL27239326	3-[6-[1-[[1-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]piperidin-3-yl]methyl]piperidine-4-carbonyl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30934112	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCCC(CN4CCC(C(=O)N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)C5)CC4)C3)C=C2F)N1CC(F)F	C47H51F4N7O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-WP1OHT	SCHEMBL27239641	6-[2-[1-[1-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]piperidin-4-yl]piperidin-4-yl]acetyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934436	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCC(N4CCC(CC(=O)N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2F)N1CC(F)F	C47H49F4N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-974TV0	SCHEMBL27239539	3-[6-[2-[1-[1-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]piperidin-4-yl]piperidin-4-yl]acetyl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30934502	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCC(N4CCC(CC(=O)N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)C5)CC4)CC3)C=C2F)N1CC(F)F	C47H51F4N7O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-WTK3OJ	SCHEMBL27239454	6-[2-[4-[1-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]piperidin-4-yl]piperazin-1-yl]acetyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934547	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCC(N4CCN(CC(=O)N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2F)N1CC(F)F	C46H48F4N8O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-ATWVMX	SCHEMBL27239184	3-[6-[2-[4-[1-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]piperidin-4-yl]piperazin-1-yl]acetyl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30934064	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCC(N4CCN(CC(=O)N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)C5)CC4)CC3)C=C2F)N1CC(F)F	C46H50F4N8O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-E9QA8V	SCHEMBL27239470	6-[2-[2-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]-2,7-diazaspiro[3.5]nonan-7-yl]acetyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934046	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CC4(CCN(CC(=O)N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C3)C=C2F)N1CC(F)F	C44H43F4N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-LVXERQ	SCHEMBL27239411	3-[6-[2-[2-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]-2,7-diazaspiro[3.5]nonan-7-yl]acetyl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30934271	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CC4(CCN(CC(=O)N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)C5)CC4)C3)C=C2F)N1CC(F)F	C44H45F4N7O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-CJE6D1	SCHEMBL27239231	6-[[1-[7-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]-7-azaspiro[3.5]nonane-2-carbonyl]piperidin-4-yl]methyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934107	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCC4(CC3)CC(C(=O)N3CCC(CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC3)C4)C=C2F)N1CC(F)F	C50H53F4N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-RI444E	SCHEMBL27239514	6-[1-[7-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]-7-azaspiro[3.5]nonane-2-carbonyl]piperidin-4-yl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934058	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCC4(CC3)CC(C(=O)N3CCC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC3)C4)C=C2F)N1CC(F)F	C49H51F4N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-8NINNM	SCHEMBL27239170	3-[6-[1-[7-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]-7-azaspiro[3.5]nonane-2-carbonyl]piperidin-4-yl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30934125	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCC4(CC3)CC(C(=O)N3CCC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)C5)CC3)C4)C=C2F)N1CC(F)F	C49H53F4N7O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-FQWEX1	SCHEMBL27239237	3-[6-[2-[1-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]azetidin-3-yl]acetyl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30934145	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CC(CC(=O)N4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)CC6=C5)C4)C3)C=C2F)N1CC(F)F	C40H38F4N6O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-69JZ37	WO2022187588A1_E103	.	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CC(CC(=O)N4CC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)C4)C3)C=C2F)N1CC(F)F	C43H41F4N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-DA69NT	SCHEMBL27239398	3-[6-[2-[1-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]piperidin-4-yl]acetyl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30934079	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCC(CC(=O)N4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)CC6=C5)C4)CC3)C=C2F)N1CC(F)F	C42H42F4N6O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-SMZF86	SCHEMBL27239459	6-[2-[2-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]-2,8-diazaspiro[3.5]nonan-8-yl]acetyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934104	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CC4(CCCN(CC(=O)N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)C4)C3)C=C2F)N1CC(F)F	C44H43F4N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-0WOBVO	SCHEMBL27239139	3-[6-[2-[2-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]-2,8-diazaspiro[3.5]nonan-8-yl]acetyl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30934242	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CC4(CCCN(CC(=O)N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)C5)C4)C3)C=C2F)N1CC(F)F	C44H45F4N7O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-MJM6BS	SCHEMBL27239354	6-[2-[2-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]-2,8-diazaspiro[4.5]decan-8-yl]acetyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934371	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCC4(CCN(CC(=O)N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C3)C=C2F)N1CC(F)F	C45H45F4N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-IFWGM7	SCHEMBL27239548	3-[6-[2-[2-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]-2,8-diazaspiro[4.5]decan-8-yl]acetyl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30934296	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCC4(CCN(CC(=O)N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)C5)CC4)C3)C=C2F)N1CC(F)F	C45H47F4N7O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-7D4XYL	WO2022187588A1_E109	6-[2-[4-[1-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]piperidin-4-yl]piperazin-1-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCC(N4CCN(C(=O)CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2F)N1CC(F)F	C46H48F4N8O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-ALEYTK	SCHEMBL27239196	6-[1-[1-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]pyrrolidin-3-yl]piperidine-4-carbonyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934450	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCC(N4CCC(C(=O)N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C3)C=C2F)N1CC(F)F	C45H45F4N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-KUKU7S	SCHEMBL27239216	6-[2-[7-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]-2,7-diazaspiro[3.5]nonan-2-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934424	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCC4(CC3)CN(C(=O)CN3CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C3)C4)C=C2F)N1CC(F)F	C44H43F4N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-27STP8	ERD-1099	6-[2-[9-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; CHEMBL5434591; SCHEMBL27239256; SCHEMBL30934428	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCC4(CCN(C(=O)CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2F)N1CC(F)F	C46H47F4N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-M5WJL5	SCHEMBL27239422	6-[[1-[1-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]piperidine-4-carbonyl]piperidin-4-yl]methyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934410	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCC(C(=O)N4CCC(CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2F)N1CC(F)F	C47H49F4N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-PLJMG5	SCHEMBL27239233	6-[1-[1-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]piperidine-4-carbonyl]piperidin-4-yl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934537	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCC(C(=O)N4CCC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2F)N1CC(F)F	C46H47F4N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-7HVXML	SCHEMBL27239551	6-[[1-[2-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]-2-azaspiro[3.3]heptane-6-carbonyl]piperidin-4-yl]methyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934357	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CC4(CC(C(=O)N5CCC(CN6CC7=C(C=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)C6)CC5)C4)C3)C=C2F)N1CC(F)F	C48H49F4N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-SRX7RV	SCHEMBL27239282	6-[1-[2-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]-2-azaspiro[3.3]heptane-6-carbonyl]piperidin-4-yl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934595	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CC4(CC(C(=O)N5CCC(N6CC7=C(C=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)C6)CC5)C4)C3)C=C2F)N1CC(F)F	C47H47F4N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-OXO4Y1	SCHEMBL27239352	6-[[1-[1-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]piperidin-4-yl]azetidin-3-yl]methyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934385	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCC(N4CC(CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)C4)CC3)C=C2F)N1CC(F)F	C44H45F4N7O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-9G3ASD	SCHEMBL27239569	6-[[1-[1-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]piperidin-4-yl]piperidin-4-yl]methyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934205	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCC(N4CCC(CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2F)N1CC(F)F	C46H49F4N7O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-56XABI	SCHEMBL27239202	6-[1-[1-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]piperidin-4-yl]azetidine-3-carbonyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934512	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCC(N4CC(C(=O)N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)C4)CC3)C=C2F)N1CC(F)F	C44H43F4N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-DJ2C51	SCHEMBL27239560	3-[6-[1-[1-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]piperidin-4-yl]azetidine-3-carbonyl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30934337	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCC(N4CC(C(=O)N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)C5)C4)CC3)C=C2F)N1CC(F)F	C44H45F4N7O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-YFSVAP	SCHEMBL27239287	6-[[1-[1-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]azetidine-3-carbonyl]piperidin-4-yl]methyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934314	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CC(C(=O)N4CCC(CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C3)C=C2F)N1CC(F)F	C45H45F4N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-9PPEQC	SCHEMBL27239389	6-[1-[1-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]azetidine-3-carbonyl]piperidin-4-yl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934243	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CC(C(=O)N4CCC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C3)C=C2F)N1CC(F)F	C44H43F4N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-WX2QNI	SCHEMBL27239263	6-[[1-[1-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]pyrrolidin-3-yl]piperidin-4-yl]methyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934457	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCC(N4CCC(CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C3)C=C2F)N1CC(F)F	C45H47F4N7O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-07VA8M	WO2022187588A1_E125	.	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(C(=O)CN2CC3(CCN(C5=CC=C6C[C@@H]7C8=C(C=C(O)C=C8)CC[C@@]7(C7=CC=CC=C7)C6=C5)CC3)C2)C4)C(=O)N1	C47H45N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-3I85QH	ERD-858	2-(2,6-dioxopiperidin-3-yl)-6-[2-[3-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-3,9-diazaspiro[5.5]undecan-9-yl]acetyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; CHEMBL5434908; SCHEMBL27239205	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(C(=O)CN2CCC3(CC2)CCN(C2=CC=C([C@@H]5C6=C(C=C(O)C=C6)CC[C@@H]5C5=CC=CC=C5)C=C2)CC3)C4)C(=O)N1	C48H49N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-JA9QOD	SCHEMBL27239250	2-(2,6-dioxopiperidin-3-yl)-6-[2-[7-[4-[(1R,2S)-2-(4-fluorophenyl)-6-hydroxy-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-2,7-diazaspiro[3.5]nonan-2-yl]acetyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL29911589	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(C(=O)CN2CC3(CCN(C5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=C(F)C=C6)C=C5)CC3)C2)C4)C(=O)N1	C46H44FN5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-TU3I4J	SCHEMBL27239338	6-[[1-[[1-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]piperidin-4-yl]methyl]piperidin-4-yl]methyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934356	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCC(CN4CCC(CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2F)N1CC(F)F	C47H51F4N7O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-W4F3AM	SCHEMBL27239270	6-[1-[[1-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]piperidin-4-yl]methyl]pyrrolidin-3-yl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934093	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCC(CN4CCC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)C4)CC3)C=C2F)N1CC(F)F	C45H47F4N7O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-AHQ3CR	SCHEMBL27239259	6-[1-[[1-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]piperidin-4-yl]methyl]azepan-4-yl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934087	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCC(CN4CCCC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2F)N1CC(F)F	C47H51F4N7O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-IVN2VA	SCHEMBL27239406	6-[2-[[1-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]piperidin-4-yl]methyl]-2-azaspiro[3.3]heptan-6-yl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934056	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCC(CN4CC5(CC(N6CC7=C(C=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)C6)C5)C4)CC3)C=C2F)N1CC(F)F	C47H49F4N7O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-1FP2DJ	SCHEMBL27239232	6-[7-[[1-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]piperidin-4-yl]methyl]-7-azaspiro[3.5]nonan-2-yl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934455	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCC(CN4CCC5(CC4)CC(N4CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C4)C5)CC3)C=C2F)N1CC(F)F	C49H53F4N7O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-LRPYC7	SCHEMBL27239442	6-[8-[[1-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]piperidin-4-yl]methyl]-8-azaspiro[4.5]decan-3-yl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934475	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCC(CN4CCC5(CCC(N6CC7=C(C=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)C6)C5)CC4)CC3)C=C2F)N1CC(F)F	C50H55F4N7O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-ND1HSE	SCHEMBL27239308	3-[6-[1-[2-[1-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]azetidin-3-yl]acetyl]azetidin-3-yl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30934147	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CC(CC(=O)N4CC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)C5)C4)C3)C=C2F)N1CC(F)F	C43H43F4N7O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-ID0OES	SCHEMBL27239318	6-[2-[2-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]-2,8-diazaspiro[4.5]decan-8-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934458	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCC4(CCN(C(=O)CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C3)C=C2F)N1CC(F)F	C45H45F4N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-UQXY6S	SCHEMBL27239173	6-[1-[[1-[4-[(6S,8R)-7-(2,2-difluoroethyl)-8-methyl-3,6,8,9-tetrahydropyrazolo[4,3-f]isoquinolin-6-yl]-3,5-difluorophenyl]piperidin-4-yl]methyl]piperidin-4-yl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934133	C[C@@H]1CC2=C(C=CC3=C2C=NN3)[C@@H](C2=C(F)C=C(N3CCC(CN4CCC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2F)N1CC(F)F	C45H48F4N8O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-2AWUPM	WO2022187588A1_E137	.	C[C@@H]1CC2=C(C=CC3=C2C=NN3)[C@@H](C2=C(F)C=C(N3CCC(CN4CCC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)C5)CC4)CC3)C=C2F)N1CC(F)F	C45H50F4N8O3	ERα	P03372	CRBN	WO-2022187588-A1
TPD-93C97G	WO2022187588A1_E138	3-[6-[2-[8-[4-[(1S,3R)-2-(2,2-difluoropropyl)-6-hydroxy-3-methyl-3,4-dihydro-1H-isoquinolin-1-yl]-3,5-difluorophenyl]-2,8-diazaspiro[4.5]decan-2-yl]-2-oxoethyl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione	C[C@@H]1CC2=CC(O)=CC=C2[C@@H](C2=C(F)C=C(N3CCC4(CCN(C(=O)CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)C5)C4)CC3)C=C2F)N1CC(C)(F)F	C44H48F4N6O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-ETQ1X3	ERD-857	2-(2,6-dioxopiperidin-3-yl)-6-[2-[2-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-2,8-diazaspiro[4.5]decan-8-yl]-2-oxoethyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL27239187	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC(=O)N2CCC3(CC2)CCN(C2=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=CC=C5)C=C2)C3)C4)C(=O)N1	C47H47N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-ZOOR07	SCHEMBL27239401	2-(2,6-dioxopiperidin-3-yl)-6-[2-[8-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-2,8-diazaspiro[4.5]decan-2-yl]acetyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(C(=O)CN2CCC3(CCN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC3)C2)C4)C(=O)N1	C47H47N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-2TD8FA	SCHEMBL27239479	2-(2,6-dioxopiperidin-3-yl)-6-[2-[2-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-2,8-diazaspiro[4.5]decan-8-yl]acetyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(C(=O)CN2CCC3(CC2)CCN(C2=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=CC=C5)C=C2)C3)C4)C(=O)N1	C47H47N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-9659O7	SCHEMBL27239522	2-(2,6-dioxopiperidin-3-yl)-6-[2-[(3S)-8-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]-2-oxoethyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	C[C@H]1CC2(CCN(C3=CC=C([C@@H]4C5=CC=C(O)C=C5CC[C@@H]4C4=CC=CC=C4)C=C3)CC2)CN1C(=O)CN1CC2=C(C=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=C2)C1	C48H49N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-N6DNMS	SCHEMBL27239188	2-(2,6-dioxopiperidin-3-yl)-6-[2-[(3S)-2-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-8-yl]-2-oxoethyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	C[C@H]1CC2(CCN(C(=O)CN3CC4=C(C=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)C3)CC2)CN1C1=CC=C([C@@H]2C3=CC=C(O)C=C3CC[C@@H]2C2=CC=CC=C2)C=C1	C48H49N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-MRSHGR	SCHEMBL27239346	2-(2,6-dioxopiperidin-3-yl)-6-[2-[(3S)-2-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-8-yl]acetyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	C[C@H]1CC2(CCN(CC(=O)N3CC4=C(C=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)C3)CC2)CN1C1=CC=C([C@@H]2C3=CC=C(O)C=C3CC[C@@H]2C2=CC=CC=C2)C=C1	C48H49N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-SIZXBT	SCHEMBL27239189	2-(2,6-dioxopiperidin-3-yl)-6-[2-[(3R)-8-[4-[(1R,2S)-2-(4-fluorophenyl)-6-hydroxy-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]-2-oxoethyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	C[C@@H]1CC2(CCN(C3=CC=C([C@@H]4C5=C(C=C(O)C=C5)CC[C@@H]4C4=CC=C(F)C=C4)C=C3)CC2)CN1C(=O)CN1CC2=C(C=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=C2)C1	C48H48FN5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-DIC546	SCHEMBL27239425	2-(2,6-dioxopiperidin-3-yl)-6-[2-[(3R)-8-[4-[(1R,2S)-2-(4-fluorophenyl)-6-hydroxy-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]acetyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	C[C@@H]1CC2(CCN(C3=CC=C([C@@H]4C5=C(C=C(O)C=C5)CC[C@@H]4C4=CC=C(F)C=C4)C=C3)CC2)CN1CC(=O)N1CC2=C(C=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=C2)C1	C48H48FN5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-EATDKZ	SCHEMBL27239598	3-[6-[[1-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]piperidin-4-yl]methyl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30934173	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCC(CN4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)CC6=C5)C4)CC3)C=C2F)N1CC(F)F	C41H42F4N6O3	ERα	P03372	CRBN	WO-2022187588-A1
TPD-WY4ELP	SCHEMBL27239225	2-(2,6-dioxopiperidin-3-yl)-6-[2-[2-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-2,7-diazaspiro[3.5]nonan-7-yl]acetyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(C(=O)CN2CCC3(CC2)CN(C2=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=CC=C5)C=C2)C3)C4)C(=O)N1	C46H45N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-6X9QXP	SCHEMBL27239342	2-(2,6-dioxopiperidin-3-yl)-6-[2-[(3S)-8-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]acetyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	C[C@H]1CC2(CCN(C3=CC=C([C@@H]4C5=CC=C(O)C=C5CC[C@@H]4C4=CC=CC=C4)C=C3)CC2)CN1CC(=O)N1CC2=C(C=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=C2)C1	C48H49N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-Y6RI4R	WO2022187588A1_E152	.	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(C(=O)CN2CCC3(CC2)CCN(C2=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=C(F)C=C5)C=C2)C3)C4)C(=O)N1	C47H46FN5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-17J5GA	SCHEMBL27239370	2-(2,6-dioxopiperidin-3-yl)-6-[2-[2-[3-fluoro-4-[(1S,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-2,8-diazaspiro[4.5]decan-8-yl]acetyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(C(=O)CN2CCC3(CC2)CCN(C2=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=CC=C5)C(F)=C2)C3)C4)C(=O)N1	C47H46FN5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-7SNPVV	SCHEMBL27239164	2-(2,6-dioxopiperidin-3-yl)-6-[2-[2-[2-fluoro-4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-2,8-diazaspiro[4.5]decan-8-yl]acetyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(C(=O)CN2CCC3(CC2)CCN(C2=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=CC=C5)C=C2F)C3)C4)C(=O)N1	C47H46FN5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-WZ6JLE	SCHEMBL27239366	6-[2-[2-[2,6-difluoro-4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-2,8-diazaspiro[4.5]decan-8-yl]acetyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(C(=O)CN2CCC3(CC2)CCN(C2=C(F)C=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=CC=C5)C=C2F)C3)C4)C(=O)N1	C47H45F2N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-VQP6EI	ERD-9096	2-(2,6-dioxopiperidin-3-yl)-6-[[1-[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]azetidine-3-carbonyl]piperidin-4-yl]methyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; CHEMBL5430447; SCHEMBL27239236; SCHEMBL30934270	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC2CCN(C(=O)C3CN(C5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)C3)CC2)C4)C(=O)N1	C47H47N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-ESF97E	SCHEMBL27239502	2-(2,6-dioxopiperidin-3-yl)-6-[2-[(3S)-3-[4-[(1R,2S)-2-(4-fluorophenyl)-6-hydroxy-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]piperidin-1-yl]-2-oxoethyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC(=O)N2CCC[C@H](OC3=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=C(F)C=C5)C=C3)C2)C4)C(=O)N1	C44H41FN4O7	ERα	P03372	CRBN	WO-2022187588-A1
TPD-1QYK39	SCHEMBL27239513	2-(2,6-dioxopiperidin-3-yl)-6-[[1-[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]azetidine-3-carbonyl]azetidin-3-yl]methyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934592	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC2CN(C(=O)C3CN(C5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)C3)C2)C4)C(=O)N1	C45H43N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-L459X8	SCHEMBL27239428	2-(2,6-dioxopiperidin-3-yl)-6-[2-[(3S)-3-[4-[(1R,2S)-2-(4-fluorophenyl)-6-hydroxy-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]piperidin-1-yl]acetyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(C(=O)CN2CCC[C@H](OC3=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=C(F)C=C5)C=C3)C2)C4)C(=O)N1	C44H41FN4O7	ERα	P03372	CRBN	WO-2022187588-A1
TPD-7LNS29	SCHEMBL27239241	2-(2,6-dioxopiperidin-3-yl)-6-[3-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-3-azaspiro[5.5]undecan-9-yl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934252	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(C2CCC3(CC2)CCN(C2=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=CC=C5)C=C2)CC3)C4)C(=O)N1	C47H48N4O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-5S1BLF	WO2022187588A1_E161	2-(2,6-dioxopiperidin-3-yl)-6-[2-[3-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-3,9-diazaspiro[5.5]undecan-9-yl]acetyl]-7,8-dihydro-5H-pyrrolo[3,4-g]isoquinoline-1,3-dione	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(C(=O)CN2CCC3(CC2)CCN(C2=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=CC=C5)C=C2)CC3)CC4)C(=O)N1	C49H51N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-5VAX2P	WO2022187588A1_E162	2-(2,6-dioxopiperidin-3-yl)-6-[2-[9-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-oxoethyl]-7,8-dihydro-5H-pyrrolo[3,4-g]isoquinoline-1,3-dione	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC(=O)N2CCC3(CC2)CCN(C2=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=CC=C5)C=C2)CC3)CC4)C(=O)N1	C49H51N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-LHUEXF	WO2022187588A1_E163	2-(2,6-dioxopiperidin-3-yl)-6-[2-[7-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-2,7-diazaspiro[3.5]nonan-2-yl]-2-oxoethyl]-7,8-dihydro-5H-pyrrolo[3,4-g]isoquinoline-1,3-dione	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC(=O)N2CC3(CCN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC3)C2)CC4)C(=O)N1	C47H47N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-WBKFSR	WO2022187588A1_E164	2-(2,6-dioxopiperidin-3-yl)-6-[2-[7-[4-[(1R,2S)-2-(4-fluorophenyl)-6-hydroxy-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-2,7-diazaspiro[3.5]nonan-2-yl]-2-oxoethyl]-7,8-dihydro-5H-pyrrolo[3,4-g]isoquinoline-1,3-dione	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC(=O)N2CC3(CCN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=C(F)C=C6)C=C5)CC3)C2)CC4)C(=O)N1	C47H46FN5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-QU2J07	WO2022187588A1_E165	2-(2,6-dioxopiperidin-3-yl)-6-[2-[9-[4-[(1R,2S)-2-(4-fluorophenyl)-6-hydroxy-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-oxoethyl]-7,8-dihydro-5H-pyrrolo[3,4-g]isoquinoline-1,3-dione	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC(=O)N2CCC3(CC2)CCN(C2=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=C(F)C=C5)C=C2)CC3)CC4)C(=O)N1	C49H50FN5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-0J7VAG	SCHEMBL27239391	2-(2,6-dioxopiperidin-3-yl)-7-[2-[9-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-oxoethyl]-5,6,8,9-tetrahydropyrrolo[3,4-h][3]benzazepine-1,3-dione; SCHEMBL30934051	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CCN(CC(=O)N2CCC3(CC2)CCN(C2=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=CC=C5)C=C2)CC3)CC4)C(=O)N1	C50H53N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-CRM3DN	SCHEMBL27239190	2-(2,6-dioxopiperidin-3-yl)-7-[2-[3-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-3,9-diazaspiro[5.5]undecan-9-yl]acetyl]-5,6,8,9-tetrahydropyrrolo[3,4-h][3]benzazepine-1,3-dione; SCHEMBL30934237	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CCN(C(=O)CN2CCC3(CC2)CCN(C2=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=CC=C5)C=C2)CC3)CC4)C(=O)N1	C50H53N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-ZRKZMC	SCHEMBL27239412	2-(2,6-dioxopiperidin-3-yl)-6-[2-[7-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-2,7-diazaspiro[3.5]nonan-2-yl]acetyl]-5,7,8,9-tetrahydropyrrolo[3,4-h][2]benzazepine-1,3-dione	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(C(=O)CN2CC3(CCN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC3)C2)CCC4)C(=O)N1	C48H49N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-CDG3Y8	SCHEMBL27239511	2-(2,6-dioxopiperidin-3-yl)-7-[2-[7-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-2,7-diazaspiro[3.5]nonan-2-yl]-2-oxoethyl]-5,6,8,9-tetrahydropyrrolo[3,4-h][3]benzazepine-1,3-dione; SCHEMBL30934345	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CCN(CC(=O)N2CC3(CCN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC3)C2)CC4)C(=O)N1	C48H49N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-DZ4HIW	SCHEMBL27239461	2-(2,6-dioxopiperidin-3-yl)-7-[2-[7-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-2,7-diazaspiro[3.5]nonan-2-yl]acetyl]-5,6,8,9-tetrahydropyrrolo[3,4-h][3]benzazepine-1,3-dione; SCHEMBL30934152	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CCN(C(=O)CN2CC3(CCN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC3)C2)CC4)C(=O)N1	C48H49N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-Z49J39	SCHEMBL27239393	2-(2,6-dioxopiperidin-3-yl)-6-[2-[7-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-2,7-diazaspiro[3.5]nonan-2-yl]-2-oxoethyl]-5,7,8,9-tetrahydropyrrolo[3,4-h][2]benzazepine-1,3-dione; SCHEMBL30934404	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC(=O)N2CC3(CCN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC3)C2)CCC4)C(=O)N1	C48H49N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-BWBBZA	SCHEMBL27239615	2-(2,6-dioxopiperidin-3-yl)-6-[2-[7-[2-fluoro-4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-2,7-diazaspiro[3.5]nonan-2-yl]-2-oxoethyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC(=O)N2CC3(CCN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5F)CC3)C2)C4)C(=O)N1	C46H44FN5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-I1LOAT	SCHEMBL27239254	2-(2,6-dioxopiperidin-3-yl)-6-[2-[7-[3-fluoro-4-[(1S,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-2,7-diazaspiro[3.5]nonan-2-yl]-2-oxoethyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC(=O)N2CC3(CCN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C(F)=C5)CC3)C2)C4)C(=O)N1	C46H44FN5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-5NEQGE	SCHEMBL27239363	6-[2-[9-[2,6-difluoro-4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC(=O)N2CCC3(CC2)CCN(C2=C(F)C=C([C@@H]5C6=C(C=C(O)C=C6)CC[C@@H]5C5=CC=CC=C5)C=C2F)CC3)C4)C(=O)N1	C48H47F2N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-WAEH3E	SCHEMBL27239335	6-[2-[9-[3,5-difluoro-4-[(1S,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC(=O)N2CCC3(CC2)CCN(C2=CC(F)=C([C@@H]5C6=C(C=C(O)C=C6)CC[C@@H]5C5=CC=CC=C5)C(F)=C2)CC3)C4)C(=O)N1	C48H47F2N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-N7LBQE	SCHEMBL27239475	6-[2-[9-[4-[(1R,2R)-2-cyclohexyl-6-hydroxy-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC(=O)N2CCC3(CC2)CCN(C2=CC=C([C@@H]5C6=C(C=C(O)C=C6)CC[C@@H]5C5CCCCC5)C=C2)CC3)C4)C(=O)N1	C48H55N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-AG8EQH	WO2022187588A1_E178	.	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC(=O)N2CCC3(CC2)CCN(C2=CC=C([C@H]5C6CCC(C7=CC=C(O)C=C76)[C@@H]5C5CCC(F)(F)CC5)C=C2)CC3)C4)C(=O)N1	C50H55F2N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-KGKZO8	SCHEMBL27239452	2-(2,6-dioxopiperidin-3-yl)-6-[2-[9-[4-[(1R)-6-hydroxyspiro[3,4-dihydro-1H-naphthalene-2,1'-cyclopentane]-1-yl]phenyl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-oxoethyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC(=O)N2CCC3(CC2)CCN(C2=CC=C([C@@H]5C6=C(C=C(O)C=C6)CCC56CCCC6)C=C2)CC3)C4)C(=O)N1	C46H51N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-DJ5JN1	WO2022187588A1_E180	.	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC(=O)N2CCC3(CC2)CCN(C2=CC=C([C@@H]5C6=CC=C(S(=O)(=O)O)C=C6CC[C@@H]5C5=CC=CC=C5)C=C2)CC3)C4)C(=O)N1	C48H49N5O8S	ERα	P03372	CRBN	WO-2022187588-A1
TPD-4647VG	WO2022187588A1_E181	.	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(C(=O)CCN2CCC3(CC2)CCN(C2=CC=C([C@@H]5C6=CC=C(S(=O)(=O)O)C=C6CC[C@@H]5C5=CC=CC=C5)C=C2)CC3)C4)C(=O)N1	C49H51N5O8S	ERα	P03372	CRBN	WO-2022187588-A1
TPD-RVUCQF	WO2022187588A1_E182	6-[2-[9-[4-[(E)-4-chloro-1-(4-hydroxyphenyl)-2-phenylbut-1-enyl]phenyl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC(=O)N2CCC3(CC2)CCN(C2=CC=C(/C(C5=CC=C(O)C=C5)=C(/CCCl)C5=CC=CC=C5)C=C2)CC3)C4)C(=O)N1	C48H48ClN5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-PMJEUL	SCHEMBL27239421	2-(2,6-dioxopiperidin-3-yl)-7-[2-[9-[4-[(1R,2S)-2-(4-fluorophenyl)-6-hydroxy-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-oxoethyl]-5,6,8,9-tetrahydropyrrolo[3,4-h][3]benzazepine-1,3-dione; SCHEMBL30934580	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CCN(CC(=O)N2CCC3(CC2)CCN(C2=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=C(F)C=C5)C=C2)CC3)CC4)C(=O)N1	C50H52FN5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-AS35U1	SCHEMBL27239361	2-(2,6-dioxopiperidin-3-yl)-7-[2-[7-[4-[(1R,2S)-2-(4-fluorophenyl)-6-hydroxy-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-2,7-diazaspiro[3.5]nonan-2-yl]-2-oxoethyl]-5,6,8,9-tetrahydropyrrolo[3,4-h][3]benzazepine-1,3-dione; SCHEMBL30934433	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CCN(CC(=O)N2CC3(CCN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=C(F)C=C6)C=C5)CC3)C2)CC4)C(=O)N1	C48H48FN5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-68RN3R	SCHEMBL27239148	2-(2,6-dioxopiperidin-3-yl)-6-[2-[9-[5-[(1S,2S)-2-(4-fluorophenyl)-6-hydroxy-1,2,3,4-tetrahydronaphthalen-1-yl]pyridin-2-yl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-oxoethyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC(=O)N2CCC3(CC2)CCN(C2=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=C(F)C=C5)C=N2)CC3)C4)C(=O)N1	C47H47FN6O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-W7EBL3	SCHEMBL27239567	2-(2,6-dioxopiperidin-3-yl)-6-[2-[2-[4-[(1R,2S)-2-(4-fluorophenyl)-6-hydroxy-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-2,8-diazaspiro[4.5]decan-8-yl]-2-oxoethyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934166	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC(=O)N2CCC3(CC2)CCN(C2=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=C(F)C=C5)C=C2)C3)C4)C(=O)N1	C47H46FN5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-FI8LH1	WO2022187588A1_E187	6-[2-[7-[4-[(E)-4-chloro-1-(4-hydroxyphenyl)-2-phenylbut-1-enyl]phenyl]-2,7-diazaspiro[3.5]nonan-2-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC(=O)N2CC3(CCN(C5=CC=C(/C(C6=CC=C(O)C=C6)=C(/CCCl)C6=CC=CC=C6)C=C5)CC3)C2)C4)C(=O)N1	C46H44ClN5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-1469V0	WO2022187588A1_E188	2-(2,6-dioxopiperidin-3-yl)-6-[2-[9-[4-[(E)-1-(4-hydroxyphenyl)-2-phenylbut-1-enyl]phenyl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-oxoethyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	CC/C(C1=CC=CC=C1)=C(\C1=CC=C(O)C=C1)C1=CC=C(N2CCC3(CCN(C(=O)CN4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)CC2)C=C1	C48H49N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-47GN5D	WO2022187588A1_E189	.	CC/C(C1=CC=CC=C1)=C(/C1=CC=C(O)C=C1)C1=CC=C(N2CCC3(CCN(C(=O)CN4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C2)C=C1	C47H47N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-W0LYAE	WO2022187588A1_E190	6-[2-[2-[4-[(E)-4-chloro-1-(4-hydroxyphenyl)-2-phenylbut-1-enyl]phenyl]-2,8-diazaspiro[4.5]decan-8-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC(=O)N2CCC3(CC2)CCN(C2=CC=C(/C(C5=CC=C(O)C=C5)=C(/CCCl)C5=CC=CC=C5)C=C2)C3)C4)C(=O)N1	C47H46ClN5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-SM5QPK	WO2022187588A1_E191	6-[2-[2-[4-[(E)-4-chloro-1-(4-hydroxyphenyl)-2-phenylbut-1-enyl]phenyl]-2,8-diazaspiro[4.5]decan-8-yl]acetyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(C(=O)CN2CCC3(CC2)CCN(C2=CC=C(/C(C5=CC=C(O)C=C5)=C(/CCCl)C5=CC=CC=C5)C=C2)C3)C4)C(=O)N1	C47H46ClN5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-0C96HH	WO2022187588A1_E192	.	CC/C(C1=CC=CC=C1)=C(/C1=CC=C(O)C=C1)C1=CC=C(N2CCC3(CCN(CC(=O)N4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)C2)C=C1	C47H47N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-Z6M7XN	WO2022187588A1_E193	6-[2-[9-[4-[(E)-4-chloro-2-(4-fluorophenyl)-1-(4-hydroxyphenyl)but-1-enyl]phenyl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-7,8-dihydro-5H-pyrrolo[3,4-g]isoquinoline-1,3-dione	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC(=O)N2CCC3(CC2)CCN(C2=CC=C(/C(C5=CC=C(O)C=C5)=C(/CCCl)C5=CC=C(F)C=C5)C=C2)CC3)CC4)C(=O)N1	C49H49ClFN5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-0IHSWM	WO2022187588A1_E194	2-(2,6-dioxopiperidin-3-yl)-6-[2-[7-[4-[(E)-1-(4-hydroxyphenyl)-2-phenylbut-1-enyl]phenyl]-2,7-diazaspiro[3.5]nonan-2-yl]-2-oxoethyl]-7,8-dihydro-5H-pyrrolo[3,4-g]isoquinoline-1,3-dione	CC/C(C1=CC=CC=C1)=C(\C1=CC=C(O)C=C1)C1=CC=C(N2CCC3(CC2)CN(C(=O)CN2CCC4=C(C=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)C2)C3)C=C1	C47H47N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-GZFYIW	WO2022187588A1_E195	6-[2-[3-[4-[(E)-4-chloro-1-(4-hydroxyphenyl)-2-phenylbut-1-enyl]phenyl]-3,9-diazaspiro[5.5]undecan-9-yl]acetyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(C(=O)CN2CCC3(CC2)CCN(C2=CC=C(/C(C5=CC=C(O)C=C5)=C(/CCCl)C5=CC=CC=C5)C=C2)CC3)C4)C(=O)N1	C48H48ClN5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-EUVFT5	WO2022187588A1_E196	6-[2-[9-[4-[(E)-4-chloro-2-(4-fluorophenyl)-1-(4-hydroxyphenyl)but-1-enyl]phenyl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC(=O)N2CCC3(CC2)CCN(C2=CC=C(/C(C5=CC=C(O)C=C5)=C(/CCCl)C5=CC=C(F)C=C5)C=C2)CC3)C4)C(=O)N1	C48H47ClFN5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-79HICP	WO2022187588A1_E197	.	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC(=O)N2CCC3(CC2)CCN(C2=CC=C(/C(C5=CC=C(S(O)(O)O)C=C5)=C(/CCCl)C5=CC=CC=C5)C=C2)CC3)C4)C(=O)N1	C48H50ClN5O8S	ERα	P03372	CRBN	WO-2022187588-A1
TPD-UHH58Q	WO2022187588A1_E198	.	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(C(=O)CN2CCC3(CC2)CCN(C2=CC=C(/C(C5=CC=C(B(O)O)C=C5)=C(\CCCl)C5=CC=CC=C5)C=C2)CC3)C4)C(=O)N1	C48H49BClN5O7	ERα	P03372	CRBN	WO-2022187588-A1
TPD-9TY9ZE	SCHEMBL27239444	2-(2,6-dioxopiperidin-3-yl)-6-[[4-fluoro-1-[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]azetidine-3-carbonyl]piperidin-4-yl]methyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934351	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC2(F)CCN(C(=O)C3CN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)C3)CC2)C4)C(=O)N1	C47H46FN5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-933Q8D	SCHEMBL27239512	2-(2,6-dioxopiperidin-3-yl)-6-[[4-fluoro-1-[3-fluoro-1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]azetidine-3-carbonyl]piperidin-4-yl]methyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934215	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC2(F)CCN(C(=O)C3(F)CN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)C3)CC2)C4)C(=O)N1	C47H45F2N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-JU9KGQ	SCHEMBL27239528	2-(2,6-dioxopiperidin-3-yl)-6-[[1-[3-fluoro-1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]azetidine-3-carbonyl]piperidin-4-yl]methyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934117	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC2CCN(C(=O)C3(F)CN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)C3)CC2)C4)C(=O)N1	C47H46FN5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-K5PS83	WO2022187588A1_E205	.	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(C(=O)C2CCN(CC3CCN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC3)CC2)C4)C(=O)N1	C49H51N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-PIMTVZ	SCHEMBL27239553	2-(2,6-dioxopiperidin-3-yl)-6-[[4-fluoro-1-[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidine-4-carbonyl]piperidin-4-yl]methyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934229	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC2(F)CCN(C(=O)C3CCN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC3)CC2)C4)C(=O)N1	C49H50FN5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-3T9JNZ	SCHEMBL27239260	2-(2,6-dioxopiperidin-3-yl)-6-[[3-fluoro-1-[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidine-4-carbonyl]azetidin-3-yl]methyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934406	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC2(F)CN(C(=O)C3CCN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC3)C2)C4)C(=O)N1	C47H46FN5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-BK5DKF	SCHEMBL27239472	2-(2,6-dioxopiperidin-3-yl)-6-[[1-[4-fluoro-1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidine-4-carbonyl]piperidin-4-yl]methyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934440	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC2CCN(C(=O)C3(F)CCN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC3)CC2)C4)C(=O)N1	C49H50FN5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-YTA7QZ	SCHEMBL27239289	6-[[1-[1-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]-3-fluoroazetidine-3-carbonyl]piperidin-4-yl]methyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934420	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CC(F)(C(=O)N4CCC(CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C3)C=C2F)N1CC(F)F	C45H44F5N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-QHDMP2	SCHEMBL27239537	6-[[1-[1-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]-3-fluoroazetidine-3-carbonyl]-4-fluoropiperidin-4-yl]methyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934480	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CC(F)(C(=O)N4CCC(F)(CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C3)C=C2F)N1CC(F)F	C45H43F6N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-QTPN01	SCHEMBL27239376	2-(2,6-dioxopiperidin-3-yl)-6-[[4-fluoro-1-[[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperidin-4-yl]methyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934081	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC2(F)CCN(CC3CCN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC3)CC2)C4)C(=O)N1	C49H52FN5O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-GR2GZ4	SCHEMBL27239521	2-(2,6-dioxopiperidin-3-yl)-6-[[3-fluoro-1-[[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]azetidin-3-yl]methyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934542	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC2(F)CN(CC3CCN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC3)C2)C4)C(=O)N1	C47H48FN5O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-DX4W8O	SCHEMBL27239355	2-(2,6-dioxopiperidin-3-yl)-6-[2-[9-[4-[(1S,2R)-2-(4-fluorophenyl)-6-hydroxy-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-oxoethyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934208	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC(=O)N2CCC3(CC2)CCN(C2=CC=C([C@H]5C6=C(C=C(O)C=C6)CC[C@H]5C5=CC=C(F)C=C5)C=C2)CC3)C4)C(=O)N1	C48H48FN5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-VUGZE2	SCHEMBL27239507	2-(2,6-dioxopiperidin-3-yl)-6-[2-[4-[4-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]pyrazol-1-yl]piperidin-1-yl]-2-oxoethyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934312	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC(=O)N2CCC(N3C=C(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)C=N3)CC2)C4)C(=O)N1	C47H44N6O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-2UTXJE	SCHEMBL27239185	2-(2,6-dioxopiperidin-3-yl)-6-[2-[3-[4-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]pyrazol-1-yl]azetidin-1-yl]-2-oxoethyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934301	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC(=O)N2CC(N3C=C(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)C=N3)C2)C4)C(=O)N1	C45H40N6O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-3A1GTX	ERD-9033	2-(2,6-dioxopiperidin-3-yl)-6-[[1-[[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperidin-4-yl]methyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; CHEMBL5428271; SCHEMBL27239307; SCHEMBL30934429	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC2CCN(CC3CCN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC3)CC2)C4)C(=O)N1	C49H53N5O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-49XD5O	ERD-9038	2-(2,6-dioxopiperidin-3-yl)-6-[[1-[[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]azetidin-3-yl]methyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; CHEMBL5401181; SCHEMBL27239242; SCHEMBL30934192	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC2CN(CC3CCN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC3)C2)C4)C(=O)N1	C47H49N5O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-8L5VJ3	SCHEMBL27239143	2-(2,6-dioxopiperidin-3-yl)-6-[2-[4-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]piperidin-1-yl]-2-oxoethyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934247	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC(=O)N2CCC(OC3=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=CC=C5)C=C3)CC2)C4)C(=O)N1	C44H42N4O7	ERα	P03372	CRBN	WO-2022187588-A1
TPD-3SO8EU	SCHEMBL27239481	2-(2,6-dioxopiperidin-3-yl)-6-[2-[2-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]-7-azaspiro[3.5]nonan-7-yl]-2-oxoethyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934068	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC(=O)N2CCC3(CC2)CC(OC2=CC=C([C@@H]5C6=C(C=C(O)C=C6)CC[C@@H]5C5=CC=CC=C5)C=C2)C3)C4)C(=O)N1	C47H46N4O7	ERα	P03372	CRBN	WO-2022187588-A1
TPD-08LETR	WO2022187588A1_E221	2-(2,6-dioxopiperidin-3-yl)-6-[2-[6-[4-[(1R)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]-2-azaspiro[3.3]heptan-2-yl]-2-oxoethyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC(=O)N2CC3(CC(OC5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CCC6C6=CC=CC=C6)C=C5)C3)C2)C4)C(=O)N1	C45H42N4O7	ERα	P03372	CRBN	WO-2022187588-A1
TPD-2PB2PD	SCHEMBL27239458	2-(2,6-dioxopiperidin-3-yl)-6-[2-[2-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]-7-azaspiro[3.5]nonan-7-yl]acetyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934467	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(C(=O)CN2CCC3(CC2)CC(OC2=CC=C([C@@H]5C6=C(C=C(O)C=C6)CC[C@@H]5C5=CC=CC=C5)C=C2)C3)C4)C(=O)N1	C47H46N4O7	ERα	P03372	CRBN	WO-2022187588-A1
TPD-CSDGK7	SCHEMBL27239471	2-(2,6-dioxopiperidin-3-yl)-6-[2-[7-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]-2-azaspiro[3.5]nonan-2-yl]-2-oxoethyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934308	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC(=O)N2CC3(CCC(OC5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC3)C2)C4)C(=O)N1	C47H46N4O7	ERα	P03372	CRBN	WO-2022187588-A1
TPD-U6813J	SCHEMBL27239498	2-(2,6-dioxopiperidin-3-yl)-6-[2-[9-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]-3-azaspiro[5.5]undecan-3-yl]-2-oxoethyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934372	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC(=O)N2CCC3(CCC(OC5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC3)CC2)C4)C(=O)N1	C49H50N4O7	ERα	P03372	CRBN	WO-2022187588-A1
TPD-47HWAU	SCHEMBL27239215	6-[2-[9-[3,5-difluoro-4-[(1S,3R)-6-hydroxy-3-methyl-2-(2,2,2-trifluoroethyl)-3,4-dihydro-1H-isoquinolin-1-yl]phenyl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934148	C[C@@H]1CC2=C(C=CC(O)=C2)[C@@H](C2=C(F)C=C(N3CCC4(CCN(C(=O)CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2F)N1CC(F)(F)F	C44H45F5N6O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-KNQGCT	SCHEMBL27239365	6-[2-[9-[3,5-difluoro-4-[(1R,3R)-3-methyl-2-(2,2,2-trifluoroethyl)-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]phenyl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934292	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCC4(CCN(C(=O)CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2F)N1CC(F)(F)F	C46H46F5N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-0RZF1F	SCHEMBL27239434	6-[2-[7-[3,5-difluoro-4-[(1R,3R)-3-methyl-2-(2,2,2-trifluoroethyl)-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]phenyl]-2,7-diazaspiro[3.5]nonan-2-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934280	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCC4(CC3)CN(C(=O)CN3CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C3)C4)C=C2F)N1CC(F)(F)F	C44H42F5N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-UA318H	SCHEMBL27239530	6-[1-[1-[3,5-difluoro-4-[(1R,3R)-3-methyl-2-(2,2,2-trifluoroethyl)-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]phenyl]piperidine-4-carbonyl]piperidin-4-yl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934050	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCC(C(=O)N4CCC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2F)N1CC(F)(F)F	C46H46F5N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-3649V5	SCHEMBL27239534	6-[1-[1-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]azetidine-3-carbonyl]azetidin-3-yl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934323	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CC(C(=O)N4CC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)C4)C3)C=C2F)N1CC(F)F	C42H39F4N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-4PZHXV	SCHEMBL27239532	6-[[1-[1-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]azetidine-3-carbonyl]azetidin-3-yl]methyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934200	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CC(C(=O)N4CC(CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)C4)C3)C=C2F)N1CC(F)F	C43H41F4N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-J43LVS	SCHEMBL27239413	6-[[3-[3,5-difluoro-4-[(1R,3R)-3-methyl-2-(2,2,2-trifluoroethyl)-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]phenyl]-3,9-diazaspiro[5.5]undecan-9-yl]methyl]-2-(2,6-dioxopiperidin-3-yl)-6,7-dihydro-5H-cyclopenta[f]isoindole-1,3-dione; SCHEMBL30934168	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCC4(CCN(CC5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2F)N1CC(F)(F)F	C46H47F5N6O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-LS5KMO	SCHEMBL27239488	6-[[7-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]-2,7-diazaspiro[3.5]nonan-2-yl]methyl]-2-(2,6-dioxopiperidin-3-yl)-6,7-dihydro-5H-cyclopenta[f]isoindole-1,3-dione; SCHEMBL30934262	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCC4(CC3)CN(CC3CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C3)C4)C=C2F)N1CC(F)F	C44H44F4N6O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-897PCM	SCHEMBL27239212	6-[[1-[1-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]piperidine-4-carbonyl]azetidin-3-yl]methyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934122	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCC(C(=O)N4CC(CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)C4)CC3)C=C2F)N1CC(F)F	C45H45F4N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-BVULWL	SCHEMBL27239430	6-[1-[1-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]piperidine-4-carbonyl]azetidin-3-yl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934497	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCC(C(=O)N4CC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)C4)CC3)C=C2F)N1CC(F)F	C44H43F4N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-76BUYV	SCHEMBL27239449	6-[1-[[1-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]piperidin-4-yl]methyl]piperidine-4-carbonyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934082	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCC(CN4CCC(C(=O)N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2F)N1CC(F)F	C47H49F4N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-Z6TK5R	SCHEMBL27239177	6-[1-[[1-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]piperidin-4-yl]methyl]azetidine-3-carbonyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934394	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCC(CN4CC(C(=O)N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)C4)CC3)C=C2F)N1CC(F)F	C45H45F4N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-W9BQVS	ERD-9115	2-(2,6-dioxopiperidin-3-yl)-6-[1-[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidine-4-carbonyl]piperidin-4-yl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; CHEMBL5407068; SCHEMBL27239191; SCHEMBL30934303	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(C2CCN(C(=O)C3CCN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC3)CC2)C4)C(=O)N1	C48H49N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-MMUGH7	SCHEMBL27239200	2-(2,6-dioxopiperidin-3-yl)-6-[1-[4-fluoro-1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidine-4-carbonyl]piperidin-4-yl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934286	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(C2CCN(C(=O)C3(F)CCN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC3)CC2)C4)C(=O)N1	C48H48FN5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-BO7TTD	WO2022187588A1_E242	2-(2,6-dioxopiperidin-3-yl)-6-[2-[7-[4-[(E)-1-(4-hydroxyphenyl)-2-phenylbut-1-enyl]phenyl]-2,7-diazaspiro[3.5]nonan-2-yl]-2-oxoethyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	CC/C(C1=CC=CC=C1)=C(\C1=CC=C(O)C=C1)C1=CC=C(N2CCC3(CC2)CN(C(=O)CN2CC4=C(C=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)C2)C3)C=C1	C46H45N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-SEB7LB	ERD-2141	2-(2,6-dioxopiperidin-3-yl)-6-[1-[[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]azetidin-3-yl]methyl]piperidin-4-yl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; CHEMBL5432713; SCHEMBL27239504; SCHEMBL30934495	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(C2CCN(CC3CN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)C3)CC2)C4)C(=O)N1	C46H47N5O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-HDX1UJ	ERD-2142	2-(2,6-dioxopiperidin-3-yl)-6-[[1-[[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]azetidin-3-yl]methyl]piperidin-4-yl]methyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; CHEMBL5406248; SCHEMBL27239443; SCHEMBL30934583	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC2CCN(CC3CN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)C3)CC2)C4)C(=O)N1	C47H49N5O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-O58XJP	SCHEMBL27239578	2-(2,6-dioxopiperidin-3-yl)-6-[[4-fluoro-1-[[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]azetidin-3-yl]methyl]piperidin-4-yl]methyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934413	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC2(F)CCN(CC3CN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)C3)CC2)C4)C(=O)N1	C47H48FN5O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-8A81W8	SCHEMBL27239144	6-[1-[4-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]cyclohexanecarbonyl]piperidin-4-yl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934435	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(C3CCC(C(=O)N4CCC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2F)N1CC(F)F	C47H48F4N6O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-VD8OO5	SCHEMBL27239369	6-[[1-[4-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]cyclohexanecarbonyl]-4-fluoropiperidin-4-yl]methyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934427	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(C3CCC(C(=O)N4CCC(F)(CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2F)N1CC(F)F	C48H49F5N6O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-6W5ICK	SCHEMBL27239267	6-[[1-[4-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]cyclohexanecarbonyl]piperidin-4-yl]methyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934352	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(C3CCC(C(=O)N4CCC(CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2F)N1CC(F)F	C48H50F4N6O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-PBN63Q	SCHEMBL27239604	6-[1-[4-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]cyclohexanecarbonyl]azetidin-3-yl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934283	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(C3CCC(C(=O)N4CC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)C4)CC3)C=C2F)N1CC(F)F	C45H44F4N6O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-OKYSZ4	SCHEMBL27239344	6-[[1-[4-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]cyclohexanecarbonyl]azetidin-3-yl]methyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934378	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(C3CCC(C(=O)N4CC(CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)C4)CC3)C=C2F)N1CC(F)F	C46H46F4N6O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-KNJ3CZ	SCHEMBL27239559	6-[1-[1-[4-[(1R,3R)-2-(2,2-difluoropropyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]piperidine-4-carbonyl]piperidin-4-yl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934075	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCC(C(=O)N4CCC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2F)N1CC(C)(F)F	C47H49F4N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-BWWHD4	SCHEMBL27239384	2-(2,6-dioxopiperidin-3-yl)-6-[2-[9-[5-[(1R,3R)-3-methyl-2-(2,2,2-trifluoroethyl)-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyrimidin-2-yl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-oxoethyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=CN=C(N3CCC4(CCN(C(=O)CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)N=C2)N1CC(F)(F)F	C44H46F3N9O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-C6WJ0P	SCHEMBL27239499	2-(2,6-dioxopiperidin-3-yl)-6-[2-[7-[5-[(1R,3R)-3-methyl-2-(2,2,2-trifluoroethyl)-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyrimidin-2-yl]-2,7-diazaspiro[3.5]nonan-2-yl]-2-oxoethyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=CN=C(N3CCC4(CC3)CN(C(=O)CN3CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C3)C4)N=C2)N1CC(F)(F)F	C42H42F3N9O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-8FBKV5	SCHEMBL27239224	2-(2,6-dioxopiperidin-3-yl)-6-[1-[[1-[5-[(1R,3R)-3-methyl-2-(2,2,2-trifluoroethyl)-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyrimidin-2-yl]piperidin-4-yl]methyl]piperidin-4-yl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=CN=C(N3CCC(CN4CCC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)N=C2)N1CC(F)(F)F	C44H48F3N9O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-S0XE43	SCHEMBL27239314	2-(2,6-dioxopiperidin-3-yl)-6-[1-[1-[5-[(1R,3R)-3-methyl-2-(2,2,2-trifluoroethyl)-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyrimidin-2-yl]piperidine-4-carbonyl]piperidin-4-yl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=CN=C(N3CCC(C(=O)N4CCC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)N=C2)N1CC(F)(F)F	C44H46F3N9O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-DS1BKI	WO2022187588A1_E258	.	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=CN=C(N3CCC4(CCN(C(=O)CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)N=C2)N1CC(=O)O	C44H47N9O7	ERα	P03372	CRBN	WO-2022187588-A1
TPD-68XZD0	WO2022187588A1_E259	.	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=CN=C(N3CCC4(CC3)CN(C(=O)CN3CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C3)C4)N=C2)N1CC(=O)O	C42H43N9O7	ERα	P03372	CRBN	WO-2022187588-A1
TPD-BKSZ6G	WO2022187588A1_E262	.	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=CC=C(N3CCC4(CC3)CN(C(=O)CN3CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C3)C4)C=C2)N1CC(=O)O	C44H45N7O7	ERα	P03372	CRBN	WO-2022187588-A1
TPD-HCH4JN	WO2022187588A1_E263	.	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=CC=C(N3CCC(C(=O)N4CCC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2)N1CC(=O)O	C46H49N7O7	ERα	P03372	CRBN	WO-2022187588-A1
TPD-Y1E4S5	WO2022187588A1_E264	.	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=CC=C(N3CCC(CN4CCC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2)N1CC(F)(F)F	C46H50F3N7O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-YQHGI1	WO2022187588A1_E265	.	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=CC=C(N3CCC4(CCN(C(=O)CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2)N1CC(=O)O	C46H49N7O7	ERα	P03372	CRBN	WO-2022187588-A1
TPD-OK3HOY	SCHEMBL27239495	2-(2,6-dioxopiperidin-3-yl)-6-[2-[2-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-2,7-diazaspiro[3.5]nonan-7-yl]ethyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CCN2CCC3(CC2)CN(C2=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=CC=C5)C=C2)C3)C4)C(=O)N1	C46H47N5O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-KNFYKA	SCHEMBL27239349	2-(2,6-dioxopiperidin-3-yl)-6-[2-[7-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-2,7-diazaspiro[3.5]nonan-2-yl]ethyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CCN2CC3(CCN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC3)C2)C4)C(=O)N1	C46H47N5O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-AH227H	SCHEMBL27239466	2-(2,6-dioxopiperidin-3-yl)-6-[2-[3-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-3,9-diazaspiro[5.5]undecan-9-yl]ethyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CCN2CCC3(CC2)CCN(C2=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=CC=C5)C=C2)CC3)C4)C(=O)N1	C48H51N5O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-24DQAO	SCHEMBL27239535	6-[1-[1-[4-[(1S,3R)-2-(2,2-difluoroethyl)-6-hydroxy-3-methyl-3,4-dihydro-1H-isoquinolin-1-yl]-3,5-difluorophenyl]piperidine-4-carbonyl]piperidin-4-yl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934090	C[C@@H]1CC2=CC(O)=CC=C2[C@@H](C2=C(F)C=C(N3CCC(C(=O)N4CCC(N5CC6=CC7=C(C=C6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)CC3)C=C2F)N1CC(F)F	C44H46F4N6O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-1R3EJC	SCHEMBL27239364	6-[1-[[1-[4-[(1S,3R)-2-(2,2-difluoroethyl)-6-hydroxy-3-methyl-3,4-dihydro-1H-isoquinolin-1-yl]-3,5-difluorophenyl]piperidin-4-yl]methyl]piperidin-4-yl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934306	C[C@@H]1CC2=CC(O)=CC=C2[C@@H](C2=C(F)C=C(N3CCC(CN4CCC(N5CC6=CC7=C(C=C6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)CC3)C=C2F)N1CC(F)F	C44H48F4N6O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-BD8L8V	ERD-2217	2-(2,6-dioxopiperidin-3-yl)-6-[1-[[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperidin-4-yl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; CHEMBL5434207; SCHEMBL27239292; SCHEMBL30934274	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(C2CCN(CC3CCN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC3)CC2)C4)C(=O)N1	C48H51N5O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-VCW9NA	ERD-2218	2-(2,6-dioxopiperidin-3-yl)-6-[1-[[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]azetidin-3-yl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; CHEMBL5396634; SCHEMBL27239142; SCHEMBL30934405	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(C2CN(CC3CCN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC3)C2)C4)C(=O)N1	C46H47N5O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-9FVYQI	SCHEMBL27239439	2-(2,6-dioxopiperidin-3-yl)-6-[1-[[1-[4-[(1R,2S)-2-(4-fluorophenyl)-6-hydroxy-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperidin-4-yl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934083	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(C2CCN(CC3CCN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=C(F)C=C6)C=C5)CC3)CC2)C4)C(=O)N1	C48H50FN5O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-U02QNJ	SCHEMBL27239574	2-(2,6-dioxopiperidin-3-yl)-6-[[1-[[1-[4-[(1R,2S)-2-(4-fluorophenyl)-6-hydroxy-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]azetidin-3-yl]methyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934201	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC2CN(CC3CCN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=C(F)C=C6)C=C5)CC3)C2)C4)C(=O)N1	C47H48FN5O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-VDNLM9	SCHEMBL27239243	3-[6-[1-[[1-[4-[(1R,2S)-2-(4-fluorophenyl)-6-hydroxy-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperidin-4-yl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30934414	O=C1CCC(N2CC3=CC4=C(C=C3C2=O)CN(C2CCN(CC3CCN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=C(F)C=C6)C=C5)CC3)CC2)C4)C(=O)N1	C48H52FN5O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-FSJWOA	SCHEMBL27239334	2-(2,6-dioxopiperidin-3-yl)-6-[1-[[1-[4-[(1S,2R)-2-(4-fluorophenyl)-6-hydroxy-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]azetidin-3-yl]methyl]piperidin-4-yl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934315	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(C2CCN(CC3CN(C5=CC=C([C@H]6C7=C(C=C(O)C=C7)CC[C@H]6C6=CC=C(F)C=C6)C=C5)C3)CC2)C4)C(=O)N1	C46H46FN5O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-H6RUU4	SCHEMBL27239397	2-(2,6-dioxopiperidin-3-yl)-6-[[1-[[1-[4-[(1R,2S)-2-(4-fluorophenyl)-6-hydroxy-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]azetidin-3-yl]methyl]piperidin-4-yl]methyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934311	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC2CCN(CC3CN(C5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=C(F)C=C6)C=C5)C3)CC2)C4)C(=O)N1	C47H48FN5O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-6KUIM8	SCHEMBL27239333	2-(2,6-dioxopiperidin-3-yl)-6-[[1-[[1-[4-[(1R,2S)-2-(4-fluorophenyl)-6-hydroxy-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]azetidin-3-yl]methyl]azetidin-3-yl]methyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934268	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC2CN(CC3CN(C5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=C(F)C=C6)C=C5)C3)C2)C4)C(=O)N1	C45H44FN5O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-K9QICT	SCHEMBL27239217	3-[6-[1-[[1-[4-[(1S,2R)-2-(4-fluorophenyl)-6-hydroxy-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]azetidin-3-yl]methyl]piperidin-4-yl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30934402	O=C1CCC(N2CC3=CC4=C(C=C3C2=O)CN(C2CCN(CC3CN(C5=CC=C([C@H]6C7=C(C=C(O)C=C7)CC[C@H]6C6=CC=C(F)C=C6)C=C5)C3)CC2)C4)C(=O)N1	C46H48FN5O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-OP1B37	WO2022187588A1_E280	.	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=NC=C(N3CCC4(CCN(C(=O)CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2)N1CC(=O)O	C45H48N8O7	ERα	P03372	CRBN	WO-2022187588-A1
TPD-P9ZA6N	WO2022187588A1_E281	.	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=CN=C(N3CCC4(CCN(C(=O)CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2)N1CC(=O)O	C45H48N8O7	ERα	P03372	CRBN	WO-2022187588-A1
TPD-VC2XZG	SCHEMBL27239149	6-[1-[[4-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]cyclohexyl]methyl]piperidin-4-yl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934206	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(C3CCC(CN4CCC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2F)N1CC(F)F	C47H50F4N6O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-WFR99C	SCHEMBL27239312	6-[[1-[[4-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]cyclohexyl]methyl]azetidin-3-yl]methyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934216	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(C3CCC(CN4CC(CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)C4)CC3)C=C2F)N1CC(F)F	C46H48F4N6O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-QIZTRK	SCHEMBL27239244	3-[6-[1-[[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperidine-4-carbonyl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30934172	O=C1CCC(N2CC3=CC4=C(C=C3C2=O)CN(C(=O)C2CCN(CC3CCN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC3)CC2)C4)C(=O)N1	C49H53N5O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-0K91VU	SCHEMBL27239586	2-(2,6-dioxopiperidin-3-yl)-6-[1-[[3-fluoro-1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]azetidin-3-yl]methyl]piperidin-4-yl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934360	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(C2CCN(CC3(F)CN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)C3)CC2)C4)C(=O)N1	C46H46FN5O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-UD6SQJ	SCHEMBL27239450	2-(2,6-dioxopiperidin-3-yl)-6-[[1-[[3-fluoro-1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]azetidin-3-yl]methyl]piperidin-4-yl]methyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934576	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC2CCN(CC3(F)CN(C5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)C3)CC2)C4)C(=O)N1	C47H48FN5O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-BRSP09	WO2022187588A1_E288	.	CN(C1CCN(C2=CC=C([C@@H]3C4=CC=C(O)C=C4CC[C@@H]3C3=CC=CC=C3)C=C2)CC1)[N+]12CCC(C(=O)N3CC4=C(C=C5C(=O)N(C6CCC(=O)NC6=O)CC5=C4)C3)(CC1)CC2	C51H57N6O5+	ERα	P03372	CRBN	WO-2022187588-A1
TPD-V52N6M	SCHEMBL27239266	2-(2,6-dioxopiperidin-3-yl)-6-[[4-[[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]-methylamino]cyclohexyl]methyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934257	CN(C1CCC(CN2CC3=C(C=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)C2)CC1)C1CCN(C2=CC=C([C@@H]3C4=CC=C(O)C=C4CC[C@@H]3C3=CC=CC=C3)C=C2)CC1	C50H55N5O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-53OQMW	SCHEMBL27239409	2-(2,6-dioxopiperidin-3-yl)-6-[4-[[4-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperazin-1-yl]methyl]cyclohexyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934469	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(C2CCC(CN3CCN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC3)CC2)C4)C(=O)N1	C48H51N5O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-I46JYR	SCHEMBL27239546	2-(2,6-dioxopiperidin-3-yl)-6-[4-[4-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperazine-1-carbonyl]cyclohexyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934162	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(C2CCC(C(=O)N3CCN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC3)CC2)C4)C(=O)N1	C48H49N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-P6OL2T	WO2022187588A1_E292	.	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=NC=C(N3CCC4(CCN(CC(=O)N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2)N1CC(F)(F)F	C45H47F3N8O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-GTH0A1	WO2022187588A1_E293	.	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=CC=C(N3CCC4(CCN(C(=O)CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2F)N1CC(=O)O	C46H48FN7O7	ERα	P03372	CRBN	WO-2022187588-A1
TPD-6EDJUT	SCHEMBL27239395	3-[6-[1-[[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]azetidin-3-yl]methyl]piperidin-4-yl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30934097	O=C1CCC(N2CC3=CC4=C(C=C3C2=O)CN(C2CCN(CC3CN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)C3)CC2)C4)C(=O)N1	C46H49N5O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-10MOD9	ERD-2270	2-(2,6-dioxopiperidin-3-yl)-6-[1-[[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]azetidin-3-yl]methyl]piperidine-4-carbonyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; CHEMBL5409697; SCHEMBL27239166; SCHEMBL30934067	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(C(=O)C2CCN(CC3CN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)C3)CC2)C4)C(=O)N1	C47H47N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-AREUJG	SCHEMBL27239400	3-[6-[1-[[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]azetidin-3-yl]methyl]piperidine-4-carbonyl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30934110	O=C1CCC(N2CC3=CC4=C(C=C3C2=O)CN(C(=O)C2CCN(CC3CN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)C3)CC2)C4)C(=O)N1	C47H49N5O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-R75DGE	SCHEMBL27239557	2-(2,6-dioxopiperidin-3-yl)-6-[2-[9-[5-[(1S,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]pyridin-2-yl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-oxoethyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC(=O)N2CCC3(CC2)CCN(C2=NC=C([C@@H]5C6=C(C=C(O)C=C6)CC[C@@H]5C5=CC=CC=C5)C=C2)CC3)C4)C(=O)N1	C47H48N6O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-W0MZP5	SCHEMBL27239506	2-(2,6-dioxopiperidin-3-yl)-6-[2-[9-[5-[(1S,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]pyrimidin-2-yl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-oxoethyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC(=O)N2CCC3(CC2)CCN(C2=NC=C([C@@H]5C6=C(C=C(O)C=C6)CC[C@@H]5C5=CC=CC=C5)C=N2)CC3)C4)C(=O)N1	C46H47N7O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-LXX6YL	SCHEMBL27239323	2-(2,6-dioxopiperidin-3-yl)-6-[[4-[4-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperazin-1-yl]cyclohexyl]methyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934575	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC2CCC(N3CCN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC3)CC2)C4)C(=O)N1	C48H51N5O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-98AXB2	WO2022187588A1_E300	.	CN(C1CCN(C2=CC=C([C@@H]3C4=CC=C(O)C=C4CC[C@@H]3C3=CC=CC=C3)C=C2)CC1)[N+]12CCC(CN3CC4=C(C=C5C(=O)N(C6CCC(=O)NC6=O)CC5=C4)C3)(CC1)CC2	C51H59N6O4+	ERα	P03372	CRBN	WO-2022187588-A1
TPD-2R8PV8	SCHEMBL27239543	6-[2-[9-[4-[(1R,3R)-2-(2,2-difluoroethyl)-6-hydroxy-3-methyl-3,4-dihydro-1H-isoquinolin-1-yl]phenyl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934265	C[C@@H]1CC2=CC(O)=CC=C2[C@@H](C2=CC=C(N3CCC4(CCN(C(=O)CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2)N1CC(F)F	C44H48F2N6O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-MBG2D1	WO2022187588A1_E302	.	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCC(C(=O)N4CCC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2)N1CC(F)(F)F	C46H47F4N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-4OIEMO	WO2022187588A1_E303	.	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(C2CCC(NC3CCN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC3)CC2)C4)C(=O)N1	C48H51N5O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-7TYBO3	SCHEMBL27239455	2-(2,6-dioxopiperidin-3-yl)-6-[2-[9-[5-[(1S,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]pyrazin-2-yl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-oxoethyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC(=O)N2CCC3(CC2)CCN(C2=CN=C([C@@H]5C6=C(C=C(O)C=C6)CC[C@@H]5C5=CC=CC=C5)C=N2)CC3)C4)C(=O)N1	C46H47N7O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-54X7OS	SCHEMBL27239301	2-(2,6-dioxopiperidin-3-yl)-6-[2-[9-[6-[(1S,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]pyridin-3-yl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-oxoethyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC(=O)N2CCC3(CC2)CCN(C2=CN=C([C@@H]5C6=C(C=C(O)C=C6)CC[C@@H]5C5=CC=CC=C5)C=C2)CC3)C4)C(=O)N1	C47H48N6O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-UXDZJ4	WO2022187588A1_E306	.	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC(=O)N2CCC3(CC2)CCN(C2=NN=C([C@@H]5C6=C(C=C(O)C=C6)CC[C@@H]5C5=CC=CC=C5)C=C2)CC3)C4)C(=O)N1	C46H47N7O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-8PFXKF	SCHEMBL27239286	3-[6-[1-[4-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]cyclohexanecarbonyl]piperidin-4-yl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30934174	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(C3CCC(C(=O)N4CCC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)C5)CC4)CC3)C=C2F)N1CC(F)F	C47H50F4N6O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-MRTCER	SCHEMBL27239347	3-[6-[1-[[4-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]cyclohexyl]methyl]piperidin-4-yl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30934491	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(C3CCC(CN4CCC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)C5)CC4)CC3)C=C2F)N1CC(F)F	C47H52F4N6O3	ERα	P03372	CRBN	WO-2022187588-A1
TPD-YT8HXC	SCHEMBL27239288	6-[1-[5-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]pyrimidine-2-carbonyl]piperidin-4-yl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934095	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(C3=CN=C(C(=O)N4CCC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)N=C3)C=C2F)N1CC(F)F	C45H40F4N8O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-0R0R72	SCHEMBL27239169	2-(2,6-dioxopiperidin-3-yl)-6-[4-[[3-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]azetidin-1-yl]methyl]cyclohexanecarbonyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934382	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(C(=O)[C@H]2CC[C@H](CN3CC(OC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)C3)CC2)C4)C(=O)N1	C48H48N4O7	ERα	P03372	CRBN	WO-2022187588-A1
TPD-KFSG64	SCHEMBL27239588	2-(2,6-dioxopiperidin-3-yl)-6-[[6-[4-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperazin-1-yl]pyridin-3-yl]methyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934358	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC2=CN=C(N3CCN(C5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC3)C=C2)C4)C(=O)N1	C47H44N6O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-64HV8Y	SCHEMBL27239408	6-[1-[4-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3-fluorophenyl]cyclohexanecarbonyl]piperidin-4-yl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934130	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(C3CCC(C(=O)N4CCC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2)N1CC(F)F	C47H49F3N6O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-O52QEB	SCHEMBL27239255	6-[1-[4-[6-[(1S,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyridin-3-yl]cyclohexanecarbonyl]piperidin-4-yl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934321	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=NC=C(C3CCC(C(=O)N4CCC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2)N1CC(F)F	C46H49F2N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-TUEHVB	SCHEMBL27239563	6-[1-[4-[5-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyridin-2-yl]cyclohex-3-ene-1-carbonyl]piperidin-4-yl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934085	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=CN=C(C3=CCC(C(=O)N4CCC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2)N1CC(F)F	C46H47F2N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-BYKAGH	SCHEMBL27239405	6-[1-[4-[5-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyrimidin-2-yl]cyclohex-3-ene-1-carbonyl]piperidin-4-yl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934230	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=CN=C(C3=CCC(C(=O)N4CCC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)N=C2)N1CC(F)F	C45H46F2N8O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-AQOE7N	SCHEMBL27239199	6-[1-[4-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]phenyl]cyclohex-3-ene-1-carbonyl]piperidin-4-yl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934238	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=CC=C(C3=CCC(C(=O)N4CCC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2)N1CC(F)F	C47H48F2N6O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-4DYOKX	SCHEMBL27239503	6-[1-[4-[4-[(1S,3R)-2-(2,2-difluoroethyl)-6-hydroxy-3-methyl-3,4-dihydro-1H-isoquinolin-1-yl]-3-fluorophenyl]cyclohexanecarbonyl]piperidin-4-yl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934044	C[C@@H]1CC2=CC(O)=CC=C2[C@@H](C2=CC=C(C3CCC(C(=O)N4CCC(N5CC6=CC7=C(C=C6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)CC3)C=C2F)N1CC(F)F	C45H48F3N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-2UHP1Y	SCHEMBL27239524	6-[1-[1-[4-[(1R,3R)-2-(2,2-difluoroethyl)-6-hydroxy-3-methyl-3,4-dihydro-1H-isoquinolin-1-yl]phenyl]piperidine-4-carbonyl]piperidin-4-yl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	C[C@@H]1CC2=CC(O)=CC=C2[C@@H](C2=CC=C(N3CCC(C(=O)N4CCC(N5CC6=CC7=C(C=C6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)CC3)C=C2)N1CC(F)F	C44H48F2N6O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-J0T9QL	SCHEMBL27239325	6-[1-[4-[5-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyridin-2-yl]cyclohexanecarbonyl]piperidin-4-yl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934142	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=CN=C(C3CCC(C(=O)N4CCC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2)N1CC(F)F	C46H49F2N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-GXT89C	SCHEMBL27239549	6-[2-[9-[4-[(1S,3R)-2-(2,2-difluoroethyl)-6-hydroxy-3-methyl-3,4-dihydro-1H-isoquinolin-1-yl]-3,5-difluorophenyl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934244	C[C@@H]1CC2=CC(O)=CC=C2[C@@H](C2=C(F)C=C(N3CCC4(CCN(C(=O)CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2F)N1CC(F)F	C44H46F4N6O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-2WW4VR	SCHEMBL27239375	6-[1-[1-[4-[(3R)-2-(2,2-difluoroethyl)-6-hydroxy-3-methyl-3,4-dihydro-1H-isoquinolin-1-yl]phenyl]piperidine-4-carbonyl]piperidin-4-yl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934070	C[C@@H]1CC2=CC(O)=CC=C2C(C2=CC=C(N3CCC(C(=O)N4CCC(N5CC6=CC7=C(C=C6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)CC3)C=C2)N1CC(F)F	C44H48F2N6O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-C4R3PC	WO2022187588A1_E322	.	C[C@@H]1CC2=CC(O)=CC=C2[C@@H](C2=CC=C(N3CCC(C(=O)N4CCC(N5CC6=CC7=C(C=C6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)CC3)C=N2)N1CC(F)F	C43H47F2N7O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-I1917C	SCHEMBL27239473	6-[1-[1-[4-[(1S,3R)-2-(2,2-difluoroethyl)-6-hydroxy-3-methyl-3,4-dihydro-1H-isoquinolin-1-yl]-3-fluorophenyl]piperidine-4-carbonyl]piperidin-4-yl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934412	C[C@@H]1CC2=CC(O)=CC=C2[C@@H](C2=CC=C(N3CCC(C(=O)N4CCC(N5CC6=CC7=C(C=C6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)CC3)C=C2F)N1CC(F)F	C44H47F3N6O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-XA8DE9	SCHEMBL27239500	2-(2,6-dioxopiperidin-3-yl)-6-[4-[[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]-methylamino]cyclohexyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934100	CN(C1CCC(N2CC3=C(C=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)C2)CC1)C1CCN(C2=CC=C([C@@H]3C4=CC=C(O)C=C4CC[C@@H]3C3=CC=CC=C3)C=C2)CC1	C49H53N5O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-SI83GQ	SCHEMBL27239278	6-[1-[5-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]pyridine-2-carbonyl]piperidin-4-yl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934207	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(C3=CN=C(C(=O)N4CCC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C3)C=C2F)N1CC(F)F	C46H41F4N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-USMVP6	SCHEMBL27239194	6-[1-[[5-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]pyridin-2-yl]methyl]piperidin-4-yl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934102	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(C3=CN=C(CN4CCC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C3)C=C2F)N1CC(F)F	C46H43F4N7O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-BP6PZM	SCHEMBL27239379	2-(2,6-dioxopiperidin-3-yl)-6-[5-[[3-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]azetidin-1-yl]methyl]pyrimidin-2-yl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934293	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(C2=NC=C(CN3CC(OC5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)C3)C=N2)C4)C(=O)N1	C45H40N6O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-DP7VJ0	SCHEMBL27239547	2-(2,6-dioxopiperidin-3-yl)-6-[5-[[3-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]azetidin-1-yl]methyl]pyridin-2-yl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934540	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(C2=CC=C(CN3CC(OC5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)C3)C=N2)C4)C(=O)N1	C46H41N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-CPRI7H	SCHEMBL27239399	2-(2,6-dioxopiperidin-3-yl)-6-[[6-[3-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]azetidin-1-yl]pyridin-3-yl]methyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934447	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC2=CN=C(N3CC(OC5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)C3)C=C2)C4)C(=O)N1	C46H41N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-D2BBUG	SCHEMBL27239247	2-(2,6-dioxopiperidin-3-yl)-6-[[2-[3-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]azetidin-1-yl]pyrimidin-5-yl]methyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934159	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC2=CN=C(N3CC(OC5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)C3)N=C2)C4)C(=O)N1	C45H40N6O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-XATKGV	SCHEMBL27239423	2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]-N-[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]acetamide; SCHEMBL30934353	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC(=O)NC2CCN(C3=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=CC=C5)C=C3)CC2)C4)C(=O)N1	C44H43N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-X4XXI6	SCHEMBL27239145	3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]-N-[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]propanamide; SCHEMBL30934124	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CCC(=O)NC2CCN(C3=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=CC=C5)C=C3)CC2)C4)C(=O)N1	C45H45N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-E9F7PU	SCHEMBL27239201	2-(2,6-dioxopiperidin-3-yl)-6-[4-[[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]azetidin-3-yl]methyl-methylamino]cyclohexyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934276	CN(CC1CN(C2=CC=C([C@@H]3C4=CC=C(O)C=C4CC[C@@H]3C3=CC=CC=C3)C=C2)C1)C1CCC(N2CC3=C(C=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)C2)CC1	C48H51N5O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-HTCTRG	WO2022187588A1_E334	.	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN([C@H]2CC[C@H](NC3CCN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC3)CC2)C4)C(=O)N1	C48H51N5O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-GA9FX5	WO2022187588A1_E335	.	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN([C@H]2CC[C@@H](NC3CCN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC3)CC2)C4)C(=O)N1	C48H51N5O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-7TOBRE	WO2022187588A1_E336	.	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(C2CCC(C(=O)NC3CN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)C3)CC2)C4)C(=O)N1	C47H47N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-JFVKRF	SCHEMBL27239505	2-(2,6-dioxopiperidin-3-yl)-6-[[4-[[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]azetidin-3-yl]amino]cyclohexyl]methyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934279	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC2CCC(NC3CN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)C3)CC2)C4)C(=O)N1	C47H49N5O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-BGHHO6	SCHEMBL27239371	2-(2,6-dioxopiperidin-3-yl)-6-[4-[[[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]azetidin-3-yl]amino]methyl]cyclohexyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934438	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(C2CCC(CNC3CN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)C3)CC2)C4)C(=O)N1	C47H49N5O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-G3QNBI	SCHEMBL27239193	2-(2,6-dioxopiperidin-3-yl)-6-[4-[[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]azetidin-3-yl]methylamino]cyclohexyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934143	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(C2CCC(NCC3CN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)C3)CC2)C4)C(=O)N1	C47H49N5O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-AM5H3L	SCHEMBL27239163	2-(2,6-dioxopiperidin-3-yl)-6-[4-[[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]azetidin-3-yl]amino]cyclohexyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934160	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN([C@H]2CC[C@H](NC3CN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)C3)CC2)C4)C(=O)N1	C46H47N5O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-Y76XZZ	SCHEMBL27239306	2-(2,6-dioxopiperidin-3-yl)-6-[[5-[3-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]azetidin-1-yl]pyrazin-2-yl]methyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934099	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC2=NC=C(N3CC(OC5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)C3)N=C2)C4)C(=O)N1	C45H40N6O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-SM01DD	SCHEMBL27239453	6-[1-[6-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]pyridine-3-carbonyl]piperidin-4-yl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934272	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(C3=CC=C(C(=O)N4CCC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=N3)C=C2F)N1CC(F)F	C46H41F4N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-8O38Z2	SCHEMBL27239162	6-[1-[5-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]pyrazine-2-carbonyl]piperidin-4-yl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934267	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(C3=CN=C(C(=O)N4CCC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=N3)C=C2F)N1CC(F)F	C45H40F4N8O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-AR6980	SCHEMBL27239204	6-[1-[6-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]pyridazine-3-carbonyl]piperidin-4-yl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934157	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(C3=CC=C(C(=O)N4CCC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)N=N3)C=C2F)N1CC(F)F	C45H40F4N8O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-1XHYB7	SCHEMBL27239596	6-[1-[2-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]pyrimidine-5-carbonyl]piperidin-4-yl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934415	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(C3=NC=C(C(=O)N4CCC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=N3)C=C2F)N1CC(F)F	C45H40F4N8O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-G8HOYY	SCHEMBL27239319	6-[1-[4-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]benzoyl]piperidin-4-yl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934120	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(C3=CC=C(C(=O)N4CCC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C3)C=C2F)N1CC(F)F	C47H42F4N6O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-8KWBKB	WO2022187588A1_E348	.	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(C3CCN(C(=O)C4CCC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2F)N1CC(F)F	C47H48F4N6O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-QPN4RO	SCHEMBL27239558	6-[[1-[1-[4-[(1S,3R)-2-(2,2-difluoroethyl)-6-hydroxy-3-methyl-3,4-dihydro-1H-isoquinolin-1-yl]-3-fluorophenyl]piperidine-4-carbonyl]azetidin-3-yl]methyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934163	C[C@@H]1CC2=CC(O)=CC=C2[C@@H](C2=C(F)C=C(N3CCC(C(=O)N4CC(CN5CC6=CC7=C(C=C6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C4)CC3)C=C2)N1CC(F)F	C43H45F3N6O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-IPOYSE	SCHEMBL27239180	6-[[1-[1-[4-[(1R,3R)-2-(2,2-difluoroethyl)-6-hydroxy-3-methyl-3,4-dihydro-1H-isoquinolin-1-yl]phenyl]piperidine-4-carbonyl]azetidin-3-yl]methyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934305	C[C@@H]1CC2=CC(O)=CC=C2[C@@H](C2=CC=C(N3CCC(C(=O)N4CC(CN5CC6=CC7=C(C=C6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C4)CC3)C=C2)N1CC(F)F	C43H46F2N6O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-66YCEW	SCHEMBL27239464	6-[[1-[1-[6-[(1S,3R)-2-(2,2-difluoroethyl)-6-hydroxy-3-methyl-3,4-dihydro-1H-isoquinolin-1-yl]pyridin-3-yl]piperidine-4-carbonyl]azetidin-3-yl]methyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934341	C[C@@H]1CC2=CC(O)=CC=C2[C@@H](C2=NC=C(N3CCC(C(=O)N4CC(CN5CC6=CC7=C(C=C6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C4)CC3)C=C2)N1CC(F)F	C42H45F2N7O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-7EQDMQ	SCHEMBL27239310	6-[4-[4-[4-[(1S,3R)-2-(2,2-difluoroethyl)-6-hydroxy-3-methyl-3,4-dihydro-1H-isoquinolin-1-yl]-3,5-difluorophenyl]piperazine-1-carbonyl]cyclohexyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	C[C@@H]1CC2=CC(O)=CC=C2[C@@H](C2=C(F)C=C(N3CCN(C(=O)C4CCC(N5CC6=CC7=C(C=C6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)CC3)C=C2F)N1CC(F)F	C44H46F4N6O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-L4O28P	WO2022187588A1_E353	.	C[C@@H]1CC2=CC(O)=CC=C2[C@@H](C2=C(F)C=C(N3CCN(C(=O)C45CCC(N6CC7=CC8=C(C=C7C6)C(=O)N(C6CCC(=O)NC6=O)C8=O)(CC4)CC5)CC3)C=C2F)N1CC(F)F	C46H48F4N6O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-4R1BFA	SCHEMBL27239519	3-[6-[2-[3-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-3,9-diazaspiro[5.5]undecan-9-yl]acetyl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30934354	O=C1CCC(N2CC3=CC4=C(C=C3C2=O)CN(C(=O)CN2CCC3(CC2)CCN(C2=CC=C([C@@H]5C6=C(C=C(O)C=C6)CC[C@@H]5C5=CC=CC=C5)C=C2)CC3)C4)C(=O)N1	C48H51N5O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-SUJY1F	WO2022187588A1_E355	.	CN(C1CN(C2=CC=C([C@@H]3C4=C(C=C(O)C=C4)CC[C@@H]3C3=CC=CC=C3)C=C2)C1)[C@H]1CC[C@H](C(=O)N2CC3=C(C=C4C(=O)N(C5CCC(=O)NC5=O)CC4=C3)C2)CC1	C48H51N5O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-F2TK3A	WO2022187588A1_E356	.	CN(C1CN(C2=CC=C([C@@H]3C4=C(C=C(O)C=C4)CC[C@@H]3C3=CC=CC=C3)C=C2)C1)[C@H]1CC[C@@H](C(=O)N2CC3=C(C=C4C(=O)N(C5CCC(=O)NC5=O)CC4=C3)C2)CC1	C48H51N5O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-SKIE0R	WO2022187588A1_E357	.	O=C1CCC(N2CC3=CC4=C(C=C3C2=O)CN(C(=O)[C@H]2CC[C@H](N3CC(OC5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)C3)CC2)C4)C(=O)N1	C47H48N4O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-DHWH3C	WO2022187588A1_E358	.	O=C1CCC(N2CC3=CC4=C(C=C3C2=O)CN(C(=O)[C@H]2CC[C@@H](N3CC(OC5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)C3)CC2)C4)C(=O)N1	C47H48N4O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-5Y8HJ8	SCHEMBL27239556	3-[6-[4-[[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]azetidin-3-yl]amino]cyclohexanecarbonyl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30934188	O=C1CCC(N2CC3=CC4=C(C=C3C2=O)CN(C(=O)C2CCC(NC3CN(C5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)C3)CC2)C4)C(=O)N1	C47H49N5O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-RP726D	WO2022187588A1_E360	.	O=C1CCC(N2CC3=CC4=C(C=C3C2=O)CN(C(=O)[C@H]2CC[C@H](N3CC(NC5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)C3)CC2)C4)C(=O)N1	C47H49N5O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-FWCAIX	WO2022187588A1_E361	.	O=C1CCC(N2CC3=CC4=C(C=C3C2=O)CN(C(=O)[C@H]2CC[C@@H](N3CC(NC5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)C3)CC2)C4)C(=O)N1	C47H49N5O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-T9KP9Y	SCHEMBL27239257	2-(2,6-dioxopiperidin-3-yl)-6-[3-[[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]-methylamino]cyclobutanecarbonyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934149	CN(C1CCN(C2=CC=C([C@@H]3C4=C(C=C(O)C=C4)CC[C@@H]3C3=CC=CC=C3)C=C2)CC1)C1CC(C(=O)N2CC3=C(C=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)C2)C1	C48H49N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-JB2ZA1	WO2022187588A1_E363	.	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(C(=O)[C@H]2CC[C@@H](CN3CC(NC5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)C3)CC2)C4)C(=O)N1	C48H49N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-T2O5G0	WO2022187588A1_E364	.	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(C(=O)[C@H]2CC[C@H](CN3CC(NC5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)C3)CC2)C4)C(=O)N1	C48H49N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-PCORJ9	SCHEMBL27239181	2-(2,6-dioxopiperidin-3-yl)-6-[4-[[4-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperazin-1-yl]methyl]cyclohexanecarbonyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934464	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(C(=O)C2CCC(CN3CCN(C5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC3)CC2)C4)C(=O)N1	C49H51N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-CATR4F	WO2022187588A1_E366	.	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(C3CCN(C[C@H]4CC[C@@H](N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2F)N1CC(F)F	C47H50F4N6O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-53J7Q8	WO2022187588A1_E367	.	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(C3CCN(CC4CCC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2F)N1CC(F)F	C47H50F4N6O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-7BR5RJ	ERD-3111	CID 164924072; 2832865-25-3; CHEMBL5438736; orb2278378; SCHEMBL27239485; SCHEMBL29911585; GTPL13249; ERD3111; GLXC-27637; EX-A9186; BDBM50618119; compound 44 [PMID: 37647546]; DA-63255; HY-149480; CS-0890777; 6-(2-(9-(4-((6S,8R)-7-(2,2-Difluoroethyl)-8-methyl-6,7,8,9-tetrahydro-3H-pyrazolo[4,3-f]isoquinolin-6-yl)-3,5-difluorophenyl)-3,9-diazaspiro[5.5]undecan-3-yl)-2-oxoethyl)-2-(2,6-dioxopiperidin-3-yl)-6,7-dihydropyrrolo[3,4-f]isoindole-1,3(2H,5H)-dione; 6-[2-[9-[4-[(6S,8R)-7-(2,2-difluoroethyl)-8-methyl-3,6,8,9-tetrahydropyrazolo[4,3-f]isoquinolin-6-yl]-3,5-difluorophenyl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	C[C@@H]1CC2=C(C=CC3=C2C=NN3)[C@@H](C2=C(F)C=C(N3CCC4(CCN(C(=O)CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2F)N1CC(F)F	C45H46F4N8O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-9STXLD	WO2022187588A1_E369	.	C[C@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(C(=O)N3CCC4(CC3)CC(CN3CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C3)C4)C=C2F)N1CC(F)F	C45H44F4N6O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-RBJ6F5	SCHEMBL27239482	6-[[7-[[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]methyl]-7-azaspiro[3.5]nonan-2-yl]methyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934246	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(CN3CCC4(CC3)CC(CN3CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C3)C4)C=C2F)N1CC(F)F	C45H46F4N6O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-RHB1YD	WO2022187588A1_E371	.	C[C@@H]1CC2=C(C=CC3=C2C=NN3)[C@@H](C2=C(F)C=C([C@H]3CC[C@@H](C(=O)N4CCC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2F)N1CC(F)F	C46H47F4N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-T91ICM	WO2022187588A1_E372	.	C[C@@H]1CC2=C(C=CC3=C2C=NN3)[C@@H](C2=C(F)C=C([C@H]3CC[C@H](C(=O)N4CCC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2F)N1CC(F)F	C46H47F4N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-5WT8QP	SCHEMBL27239331	2-(2,6-dioxopiperidin-3-yl)-6-[[6-[3-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]anilino]azetidin-1-yl]pyridin-3-yl]methyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934146	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC2=CC=C(N3CC(NC5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)C3)N=C2)C4)C(=O)N1	C46H42N6O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-KER110	WO2022187588A1_E374	.	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(C[C@H]2CC[C@@H](N3CC(NC5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)C3)CC2)C4)C(=O)N1	C47H49N5O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-PFFLXK	WO2022187588A1_E375	.	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC2CCC(N3CC(NC5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)C3)CC2)C4)C(=O)N1	C47H49N5O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-FBIGBX	SCHEMBL27239416	2-(2,6-dioxopiperidin-3-yl)-6-[2-[4-[3-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]azetidine-1-carbonyl]piperidin-1-yl]-2-oxoethyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934228	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC(=O)N2CCC(C(=O)N3CC(OC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)C3)CC2)C4)C(=O)N1	C48H47N5O8	ERα	P03372	CRBN	WO-2022187588-A1
TPD-295J6N	SCHEMBL27239415	2-(2,6-dioxopiperidin-3-yl)-6-[2-[4-[3-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]azetidin-1-yl]piperidin-1-yl]-2-oxoethyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934203	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC(=O)N2CCC(N3CC(OC5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)C3)CC2)C4)C(=O)N1	C47H47N5O7	ERα	P03372	CRBN	WO-2022187588-A1
TPD-HWHFDH	SCHEMBL27239213	6-[[3-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorobenzoyl]-3-azaspiro[5.5]undecan-9-yl]methyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934291	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(C(=O)N3CCC4(CCC(CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2F)N1CC(F)F	C47H48F4N6O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-3SEZQA	SCHEMBL27239580	6-[[3-[4-[(1S,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorobenzoyl]-3-azaspiro[5.5]undecan-9-yl]methyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934509	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@H](C2=C(F)C=C(C(=O)N3CCC4(CCC(CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2F)N1CC(F)F	C47H48F4N6O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-YALVB9	SCHEMBL27239600	6-[[3-[[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]methyl]-3-azaspiro[5.5]undecan-9-yl]methyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934127	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(CN3CCC4(CCC(CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2F)N1CC(F)F	C47H50F4N6O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-7XDBWE	SCHEMBL27239317	6-[[3-[[4-[(1S,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]methyl]-3-azaspiro[5.5]undecan-9-yl]methyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934197	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@H](C2=C(F)C=C(CN3CCC4(CCC(CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2F)N1CC(F)F	C47H50F4N6O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-W2QBTO	SCHEMBL27239176	6-[3-[[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]methyl]-3-azaspiro[5.5]undecane-9-carbonyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934570	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(CN3CCC4(CCC(C(=O)N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2F)N1CC(F)F	C47H48F4N6O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-WJIM6M	SCHEMBL27239385	6-[3-[[4-[(1S,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]methyl]-3-azaspiro[5.5]undecane-9-carbonyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934423	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@H](C2=C(F)C=C(CN3CCC4(CCC(C(=O)N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2F)N1CC(F)F	C47H48F4N6O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-J6AV0R	SCHEMBL27239186	2-(2,6-dioxopiperidin-3-yl)-6-[4-[3-[4-[(1S,2R)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]azetidine-1-carbonyl]cyclohexyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934391	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(C2CCC(C(=O)N3CC(OC5=CC=C([C@H]6C7=C(C=C(O)C=C7)CC[C@H]6C6=CC=CC=C6)C=C5)C3)CC2)C4)C(=O)N1	C47H46N4O7	ERα	P03372	CRBN	WO-2022187588-A1
TPD-MU44Y5	SCHEMBL27239230	2-(2,6-dioxopiperidin-3-yl)-6-[4-[3-[4-[(1S,2R)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]anilino]azetidine-1-carbonyl]cyclohexyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934144	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(C2CCC(C(=O)N3CC(NC5=CC=C([C@H]6C7=C(C=C(O)C=C7)CC[C@H]6C6=CC=CC=C6)C=C5)C3)CC2)C4)C(=O)N1	C47H47N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-3YFDA6	WO2022187588A1_E388	.	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(C(=O)[C@H]2CC[C@H](N3CC(OC5=CC=C([C@H]6C7=C(C=C(O)C=C7)CC[C@H]6C6=CC=CC=C6)C=C5)C3)CC2)C4)C(=O)N1	C47H46N4O7	ERα	P03372	CRBN	WO-2022187588-A1
TPD-7AZZ06	WO2022187588A1_E389	.	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(C(=O)C2CCC(N3CC(OC5=CC=C([C@H]6C7=C(C=C(O)C=C7)CC[C@H]6C6=CC=CC=C6)C=C5)C3)CC2)C4)C(=O)N1	C47H46N4O7	ERα	P03372	CRBN	WO-2022187588-A1
TPD-XUX8I0	SCHEMBL27239362	2-(2,6-dioxopiperidin-3-yl)-6-[4-[3-[4-[(1S,2R)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]anilino]azetidin-1-yl]cyclohexanecarbonyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934134	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(C(=O)[C@H]2CC[C@H](N3CC(NC5=CC=C([C@H]6C7=C(C=C(O)C=C7)CC[C@H]6C6=CC=CC=C6)C=C5)C3)CC2)C4)C(=O)N1	C47H47N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-5YUT8P	WO2022187588A1_E392	.	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(C3CCN(C(=O)[C@H]4CC[C@H](N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2F)N1CC(F)F	C47H48F4N6O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-E530IR	WO2022187588A1_E393	.	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(C3CCN(C(=O)[C@H]4CC[C@@H](N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2F)N1CC(F)F	C47H48F4N6O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-MYY1LJ	WO2022187588A1_E394	.	CN(C1=CC=C([C@H]2C3=C(C=C(O)C=C3)CC[C@H]2C2=CC=CC=C2)C=C1)C1CN([C@H]2CC[C@H](C(=O)N3CC4=C(C=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)C3)CC2)C1	C48H49N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-HA3HD7	WO2022187588A1_E395	.	CN(C1=CC=C([C@H]2C3=C(C=C(O)C=C3)CC[C@H]2C2=CC=CC=C2)C=C1)C1CN([C@H]2CC[C@@H](C(=O)N3CC4=C(C=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)C3)CC2)C1	C48H49N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-0P6PB9	WO2022187588A1_E396	.	COC1=C([C@@H]2C3=C(C[C@@H](C)N2CC(F)F)C2=C(C=CC=C2)N3)C=NC([C@H]2CC[C@@H](C(=O)N3CCC(N4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)CC2)=C1	C47H51F2N7O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-D4S8OF	WO2022187588A1_E397	.	COC1=C([C@@H]2C3=C(C[C@@H](C)N2CC(F)F)C2=C(C=CC=C2)N3)C=NC([C@H]2CC[C@H](C(=O)N3CCC(N4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)CC2)=C1	C47H51F2N7O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-OE62FM	SCHEMBL27239274	2-(2,6-dioxopiperidin-3-yl)-6-[4-[[3-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]-N-methylanilino]azetidin-1-yl]methyl]cyclohexanecarbonyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934179	CN(C1=CC=C([C@@H]2C3=C(C=C(O)C=C3)CC[C@@H]2C2=CC=CC=C2)C=C1)C1CN(C[C@H]2CC[C@H](C(=O)N3CC4=C(C=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)C3)CC2)C1	C49H51N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-4PF81J	SCHEMBL27239192	6-[1-[4-[6-[(1S,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-5-fluoropyridin-3-yl]cyclohex-3-ene-1-carbonyl]piperidin-4-yl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934209	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(C3=CCC(C(=O)N4CCC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=N2)N1CC(F)F	C46H46F3N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-YW2W5X	SCHEMBL27239394	6-[1-[4-[4-[(1R,3R)-2-(2,2-difluoro-3-hydroxypropyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]cyclohexanecarbonyl]piperidin-4-yl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934418	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(C3CCC(C(=O)N4CCC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2F)N1CC(F)(F)CO	C48H50F4N6O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-1NR07Y	SCHEMBL27239353	6-[1-[4-[5-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-6-methoxypyridin-2-yl]cyclohexanecarbonyl]piperidin-4-yl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934346	COC1=C([C@@H]2C3=C(C[C@@H](C)N2CC(F)F)C2=C(C=CC=C2)N3)C=CC(C2CCC(C(=O)N3CCC(N4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)CC2)=N1	C47H51F2N7O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-MRJESV	WO2022187588A1_E403	.	COC1=C([C@@H]2C3=C(C[C@@H](C)N2CC(F)F)C2=C(C=CC=C2)N3)C=CC([C@H]2CC[C@H](C(=O)N3CCC(N4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)CC2)=C1	C48H52F2N6O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-38TUF9	WO2022187588A1_E404	.	COC1=C([C@@H]2C3=C(C[C@@H](C)N2CC(F)F)C2=C(C=CC=C2)N3)C=CC([C@H]2CC[C@@H](C(=O)N3CCC(N4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)CC2)=C1	C48H52F2N6O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-PBS359	SCHEMBL27239211	6-[1-[4-[6-[(1S,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-5-methoxypyridin-3-yl]cyclohexanecarbonyl]piperidin-4-yl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934442	COC1=C([C@@H]2C3=C(C[C@@H](C)N2CC(F)F)C2=C(C=CC=C2)N3)N=CC(C2CCC(C(=O)N3CCC(N4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)CC2)=C1	C47H51F2N7O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-Q2HITS	SCHEMBL27239614	6-[1-[4-[6-[(1S,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-5-fluoropyridin-3-yl]cyclohexanecarbonyl]piperidin-4-yl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934318	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(C3CCC(C(=O)N4CCC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=N2)N1CC(F)F	C46H48F3N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-5YW9VV	SCHEMBL30934155	6-[[1-[4-[4-[(6S,8R)-7-(2,2-difluoroethyl)-8-methyl-3,6,8,9-tetrahydropyrazolo[4,3-f]isoquinolin-6-yl]-3,5-difluorophenyl]cyclohexanecarbonyl]azetidin-3-yl]methyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	C[C@@H]1CC2=C(C=CC3=C2C=NN3)[C@@H](C2=C(F)C=C([C@H]3CC[C@@H](C(=O)N4CC(CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)C4)CC3)C=C2F)N1CC(F)F	C45H45F4N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-M75T8G	SCHEMBL30934368	6-[2-[7-[4-[(6S,8R)-7-(2,2-difluoroethyl)-8-methyl-3,6,8,9-tetrahydropyrazolo[4,3-f]isoquinolin-6-yl]-3,5-difluorophenyl]-2,7-diazaspiro[3.5]nonan-2-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	C[C@@H]1CC2=C(C=CC3=C2C=NN3)[C@@H](C2=C(F)C=C(N3CCC4(CC3)CN(C(=O)CN3CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C3)C4)C=C2F)N1CC(F)F	C43H42F4N8O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-B3QTZB	SCHEMBL30934403	6-[2-[3-[4-[(6S,8R)-7-(2,2-difluoroethyl)-8-methyl-3,6,8,9-tetrahydropyrazolo[4,3-f]isoquinolin-6-yl]-3,5-difluorophenyl]-3,9-diazaspiro[5.5]undecan-9-yl]acetyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	C[C@@H]1CC2=C(C=CC3=C2C=NN3)[C@@H](C2=C(F)C=C(N3CCC4(CCN(CC(=O)N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2F)N1CC(F)F	C45H46F4N8O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-8IZ0Q8	WO2022187588A1_E410	.	C[C@@H]1CC2=C(C=CC3=C2C=NN3)[C@@H](C2=C(F)C=C(N3CCC(C(=O)N4CCC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2F)N1CC(F)F	C45H46F4N8O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-AP0FXT	WO2022187588A1_E411	.	C[C@@H]1CC2=C(C=CC3=C2C=NN3)[C@@H](C2=C(F)C=C(C3CCN(C(=O)[C@H]4CC[C@H](N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2F)N1CC(F)F	C46H47F4N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-5NF1IL	WO2022187588A1_E412	.	C[C@@H]1CC2=C(C=CC3=C2C=NN3)[C@@H](C2=C(F)C=C(C3CCN(C(=O)[C@H]4CC[C@@H](N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2F)N1CC(F)F	C46H47F4N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-M62PS6	ERD-3327	2-(2,6-dioxopiperidin-3-yl)-6-[2-[9-[6-[(6S,8R)-8-methyl-7-(2,2,2-trifluoroethyl)-3,6,8,9-tetrahydropyrazolo[4,3-f]isoquinolin-6-yl]pyridin-3-yl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-oxoethyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; CHEMBL5407461; SCHEMBL27239510; SCHEMBL30934218	C[C@@H]1CC2=C(C=CC3=C2C=NN3)[C@@H](C2=CC=C(N3CCC4(CCN(C(=O)CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=N2)N1CC(F)(F)F	C44H46F3N9O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-SKT58H	SCHEMBL27239463	2-(2,6-dioxopiperidin-3-yl)-6-[1-[4-[6-[(6S,8R)-8-methyl-7-(2,2,2-trifluoroethyl)-3,6,8,9-tetrahydropyrazolo[4,3-f]isoquinolin-6-yl]pyridin-3-yl]cyclohexanecarbonyl]piperidin-4-yl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934515	C[C@@H]1CC2=C(C=CC3=C2C=NN3)[C@@H](C2=CC=C(C3CCC(C(=O)N4CCC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=N2)N1CC(F)(F)F	C45H47F3N8O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-M1HCCT	SCHEMBL27239456	2-(2,6-dioxopiperidin-3-yl)-6-[1-[4-[6-[(6S,8R)-8-methyl-7-(2,2,2-trifluoroethyl)-3,6,8,9-tetrahydropyrazolo[4,3-f]isoquinolin-6-yl]pyridin-3-yl]cyclohex-3-ene-1-carbonyl]piperidin-4-yl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934076	C[C@@H]1CC2=C(C=CC3=C2C=NN3)[C@@H](C2=CC=C(C3=CCC(C(=O)N4CCC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=N2)N1CC(F)(F)F	C45H45F3N8O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-FM4P9I	WO2022187588A1_E416	.	C[C@@H]1CC2=C(C=CC3=C2C=NN3)[C@@H](C2=C(F)C=C(N3CCC4(CCN(C(=O)CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C3)C=C2F)N1CC(F)F	C44H44F4N8O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-63BXGU	WO2022187588A1_E417	.	C[C@@H]1CC2=C(C=CC3=C2C=NN3)[C@@H](C2=C(F)C=C(N3CC4(CCN(C(=O)CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C3)C=C2F)N1CC(F)F	C43H42F4N8O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-DXX0VK	SCHEMBL27239327	1'-[[1-[4-[(6S,8R)-7-(2,2-difluoroethyl)-8-methyl-3,6,8,9-tetrahydropyrazolo[4,3-f]isoquinolin-6-yl]-3,5-difluorophenyl]piperidin-4-yl]methyl]-2-(2,6-dioxopiperidin-3-yl)spiro[5,7-dihydrocyclopenta[f]isoindole-6,3'-azetidine]-1,3-dione; SCHEMBL30934196	C[C@@H]1CC2=C(C=CC3=C2C=NN3)[C@@H](C2=C(F)C=C(N3CCC(CN4CC5(CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)C4)CC3)C=C2F)N1CC(F)F	C43H43F4N7O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-BD7EK2	WO2022187588A1_E419	.	COC1=C2C(=O)N(C3CCC(=O)NC3=O)C(=O)C2=CC2=C1CN(CC(=O)N1CCC3(CC1)CCN(C1=CC(F)=C([C@@H]4C5=C(C[C@@H](C)N4CC(F)F)C4=C(C=C5)NN=C4)C(F)=C1)CC3)C2	C46H48F4N8O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-38KNH2	SCHEMBL27239431	2-(2,6-dioxopiperidin-3-yl)-6-[2-[9-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-oxoethyl]-8-methoxy-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934543	COC1=C2C(=O)N(C3CCC(=O)NC3=O)C(=O)C2=CC2=C1CN(CC(=O)N1CCC3(CC1)CCN(C1=CC=C([C@@H]4C5=C(C=C(O)C=C5)CC[C@@H]4C4=CC=CC=C4)C=C1)CC3)C2	C49H51N5O7	ERα	P03372	CRBN	WO-2022187588-A1
TPD-V1QZT5	SCHEMBL27239402	6-[1-[[1-[4-[(6S,8R)-7-(2,2-difluoroethyl)-8-methyl-3,6,8,9-tetrahydropyrazolo[4,3-f]isoquinolin-6-yl]-3,5-difluorophenyl]piperidin-4-yl]methyl]piperidin-4-yl]-2-(2,6-dioxopiperidin-3-yl)-1,5-dihydropyrrolo[3,4-f]isoindole-3,7-dione; SCHEMBL30934273	C[C@@H]1CC2=C(C=CC3=C2C=NN3)[C@@H](C2=C(F)C=C(N3CCC(CN4CCC(N5CC6=C(C=C7CN(C8CCC(=O)NC8=O)C(=O)C7=C6)C5=O)CC4)CC3)C=C2F)N1CC(F)F	C45H48F4N8O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-PW59M0	SCHEMBL27239367	2-(2,6-dioxopiperidin-3-yl)-6-[2-oxo-2-[9-[4-[(6S,7R)-7-phenyl-6,7,8,9-tetrahydro-3H-benzo[e]indazol-6-yl]phenyl]-3,9-diazaspiro[5.5]undecan-3-yl]ethyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934178	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC(=O)N2CCC3(CC2)CCN(C2=CC=C([C@H]5C6=C(CC[C@H]5C5=CC=CC=C5)C5=C(C=C6)NN=C5)C=C2)CC3)C4)C(=O)N1	C49H49N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-JT49NN	SCHEMBL27239234	2-(2,6-dioxopiperidin-3-yl)-6-[2-oxo-2-[9-[4-[(6R,7S)-7-phenyl-6,7,8,9-tetrahydro-3H-benzo[e]indazol-6-yl]phenyl]-3,9-diazaspiro[5.5]undecan-3-yl]ethyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934333	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC(=O)N2CCC3(CC2)CCN(C2=CC=C([C@@H]5C6=C(CC[C@@H]5C5=CC=CC=C5)C5=C(C=C6)NN=C5)C=C2)CC3)C4)C(=O)N1	C49H49N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-PXED6S	WO2022187588A1_E424	.	C[C@@H]1CC2=C(C=CC3=C2C=NN3)[C@@H](C2=C(F)C=C(NC3CN(C(=O)[C@H]4CC[C@@H](N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C3)C=C2F)N1CC(F)F	C44H44F4N8O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-3JCTR7	WO2022187588A1_E425	.	C[C@@H]1CC2=C(C=CC3=C2C=NN3)[C@@H](C2=C(F)C=C(NC3CN(C(=O)[C@H]4CC[C@H](N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C3)C=C2F)N1CC(F)F	C44H44F4N8O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-VNEHUV	SCHEMBL27239322	2-(2,6-dioxopiperidin-3-yl)-6-[2-[6-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]anilino]-2-azaspiro[3.3]heptan-2-yl]-2-oxoethyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934432	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC(=O)N2CC3(CC(NC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)C3)C2)C4)C(=O)N1	C45H43N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-87JLYN	SCHEMBL27239424	6-[2-[6-[4-[(6S,8R)-7-(2,2-difluoroethyl)-8-methyl-3,6,8,9-tetrahydropyrazolo[4,3-f]isoquinolin-6-yl]-3,5-difluoroanilino]-2-azaspiro[3.3]heptan-2-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934362	C[C@@H]1CC2=C(C=CC3=C2C=NN3)[C@@H](C2=C(F)C=C(NC3CC4(C3)CN(C(=O)CN3CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C3)C4)C=C2F)N1CC(F)F	C42H40F4N8O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-NQNV7U	WO2022187588A1_E428	.	C[C@@H]1CC2=C(C=CC3=C2C=NN3)[C@@H](C2=C(F)C=C(NC3CC4(C3)CN(CC(=O)N3CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C3)C4)C=C2F)N1CC(F)F	C42H40F4N8O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-RJD0LZ	SCHEMBL27239291	3-[6-[2-[9-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-oxoethyl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30934431	O=C1CCC(N2CC3=CC4=C(C=C3C2=O)CN(CC(=O)N2CCC3(CC2)CCN(C2=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=CC=C5)C=C2)CC3)C4)C(=O)N1	C48H51N5O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-G98HK5	SCHEMBL27239150	6-[2-[9-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3-methoxyphenyl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934185	COC1=CC(N2CCC3(CCN(C(=O)CN4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)CC2)=CC=C1[C@@H]1C2=C(C[C@@H](C)N1CC(F)F)C1=C(C=CC=C1)N2	C47H51F2N7O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-H0S19N	ERD-570	6-[2-[9-[4-[(6S,8R)-7-(2,2-difluoroethyl)-8-methyl-3,6,8,9-tetrahydropyrazolo[4,3-f]isoquinolin-6-yl]-3-methoxyphenyl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; CHEMBL5423055; SCHEMBL30934473	COC1=CC(N2CCC3(CCN(C(=O)CN4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)CC2)=CC=C1[C@@H]1C2=C(C[C@@H](C)N1CC(F)F)C1=C(C=C2)NN=C1	C46H50F2N8O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-N7CI0W	WO2022187588A1_E432	.	COC1=CC(N2CCC3(CCN(C(=O)CN4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)CC6=C5)C4)CC3)CC2)=CC=C1[C@@H]1C2=C(C[C@@H](C)N1CC(F)F)C1=C(C=C2)NN=C1	C46H52F2N8O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-62DYWI	SCHEMBL27239249	2-(2,6-dioxopiperidin-3-yl)-6-[2-[3-[6-[(6S,8R)-8-methyl-7-(2,2,2-trifluoroethyl)-3,6,8,9-tetrahydropyrazolo[4,3-f]isoquinolin-6-yl]pyridin-3-yl]-3,9-diazaspiro[5.5]undecan-9-yl]acetyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934161	C[C@@H]1CC2=C(C=CC3=C2C=NN3)[C@@H](C2=CC=C(N3CCC4(CCN(CC(=O)N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=N2)N1CC(F)(F)F	C44H46F3N9O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-E3QWYT	ERD-576	6-[2-[9-[6-[(6S,8R)-7-(2,2-difluoroethyl)-8-methyl-3,6,8,9-tetrahydropyrazolo[4,3-f]isoquinolin-6-yl]pyridin-3-yl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; CHEMBL5403887; SCHEMBL30934126	C[C@@H]1CC2=C(C=CC3=C2C=NN3)[C@@H](C2=CC=C(N3CCC4(CCN(C(=O)CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=N2)N1CC(F)F	C44H47F2N9O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-A32PRB	WO2022187588A1_E435	.	C[C@@H]1CC2=C(C=CC3=C2C=NN3)[C@@H](C2=CC=C(N3CCC4(CCN(CC(=O)N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2)N1CC(F)F	C45H48F2N8O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-D18KX7	SCHEMBL30934479	6-[2-[3-[4-[(6S,8R)-7-(2,2-difluoroethyl)-8-methyl-3,6,8,9-tetrahydropyrazolo[4,3-f]isoquinolin-6-yl]-3-methoxyphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]acetyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	COC1=CC(N2CCC3(CCN(CC(=O)N4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)CC2)=CC=C1[C@@H]1C2=C(C[C@@H](C)N1CC(F)F)C1=C(C=C2)NN=C1	C46H50F2N8O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-GH0EJ1	SCHEMBL27239576	2-(2,6-dioxopiperidin-3-yl)-6-[2-[9-[4-[(1S,2R)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-oxoethyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934195	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC(=O)N2CCC3(CC2)CCN(C2=CC=C([C@H]5C6=C(C=C(O)C=C6)CC[C@H]5C5=CC=CC=C5)C=C2)CC3)C4)C(=O)N1	C48H49N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-G8586A	SCHEMBL27239313	2-(2,6-dioxopiperidin-3-yl)-6-[2-[7-[4-[(1S,2R)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-2,7-diazaspiro[3.5]nonan-2-yl]-2-oxoethyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934364	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC(=O)N2CC3(CCN(C5=CC=C([C@H]6C7=C(C=C(O)C=C7)CC[C@H]6C6=CC=CC=C6)C=C5)CC3)C2)C4)C(=O)N1	C46H45N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-BQ7ZOX	SCHEMBL27239140	3-[6-[2-[9-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-oxoethyl]-8-methoxy-3-oxo-5,7-dihydro-1H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30934348	COC1=C2CN(C3CCC(=O)NC3=O)C(=O)C2=CC2=C1CN(CC(=O)N1CCC3(CC1)CCN(C1=CC=C([C@@H]4C5=CC=C(O)C=C5CC[C@@H]4C4=CC=CC=C4)C=C1)CC3)C2	C49H53N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-IBSA98	WO2022187588A1_E440	.	COC1=C2CN(C3CCC(=O)NC3=O)C(=O)C2=CC2=C1CN(CC(=O)N1CCC3(CC1)CCN(C1=CC(F)=C([C@@H]4C5=CC=C6NN=CC6=C5C[C@@H](C)N4CC(F)F)C(F)=C1)CC3)C2	C46H50F4N8O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-AFMSMH	SCHEMBL30934287	3-[6-[2-[7-[4-[(6S,8R)-7-(2,2-difluoroethyl)-8-methyl-3,6,8,9-tetrahydropyrazolo[4,3-f]isoquinolin-6-yl]-3,5-difluorophenyl]-2,7-diazaspiro[3.5]nonan-2-yl]-2-oxoethyl]-8-methoxy-3-oxo-5,7-dihydro-1H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione	COC1=C2CN(C3CCC(=O)NC3=O)C(=O)C2=CC2=C1CN(CC(=O)N1CC3(CCN(C4=CC(F)=C([C@@H]5C6=CC=C7NN=CC7=C6C[C@@H](C)N5CC(F)F)C(F)=C4)CC3)C1)C2	C44H46F4N8O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-A5F2EK	WO2022187588A1_E442	.	COC1=C2CN(C3CCC(=O)NC3=O)C(=O)C2=CC2=C1CN(CC(=O)N1CCC3(CC1)CCN(C1=CN=C([C@@H]4C5=C(C[C@@H](C)N4CC(F)(F)F)C4=C(C=C5)NN=C4)C=C1)CC3)C2	C45H50F3N9O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-C4HS02	SCHEMBL27239386	3-[6-[2-[9-[6-[(6S,8R)-8-methyl-7-(2,2,2-trifluoroethyl)-3,6,8,9-tetrahydropyrazolo[4,3-f]isoquinolin-6-yl]pyridin-3-yl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-oxoethyl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30934343	C[C@@H]1CC2=C(C=CC3=C2C=NN3)[C@@H](C2=NC=C(N3CCC4(CCN(C(=O)CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)C5)CC4)CC3)C=C2)N1CC(F)(F)F	C44H48F3N9O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-0KQBOQ	SCHEMBL27239271	3-[6-[2-[9-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-oxoethyl]-8-methoxy-3-oxo-5,7-dihydro-1H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30934344	COC1=C2CN(C3CCC(=O)NC3=O)C(=O)C2=CC2=C1CN(CC(=O)N1CCC3(CC1)CCN(C1=CC(F)=C([C@@H]4C5=C(C[C@@H](C)N4CC(F)F)C4=C(C=CC=C4)N5)C(F)=C1)CC3)C2	C47H51F4N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-4J66QV	SCHEMBL27239228	3-[6-[2-[9-[5-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyrimidin-2-yl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-oxoethyl]-8-methoxy-3-oxo-5,7-dihydro-1H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30934586	COC1=C2CN(C3CCC(=O)NC3=O)C(=O)C2=CC2=C1CN(CC(=O)N1CCC3(CC1)CCN(C1=NC=C([C@@H]4C5=C(C[C@@H](C)N4CC(F)F)C4=C(C=CC=C4)N5)C=N1)CC3)C2	C45H51F2N9O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-25G3RN	SCHEMBL30934167	6-[2-[9-[4-[(1S,3R)-2-(2,2-difluoroethyl)-6-hydroxy-3-methyl-3,4-dihydro-1H-isoquinolin-1-yl]-3,5-difluorophenyl]-3-azaspiro[5.5]undec-9-en-3-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	C[C@@H]1CC2=CC(O)=CC=C2[C@@H](C2=C(F)C=C(C3=CCC4(CC3)CCN(C(=O)CN3CC5=CC6=C(C=C5C3)C(=O)N(C3CCC(=O)NC3=O)C6=O)CC4)C=C2F)N1CC(F)F	C45H45F4N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-DL107W	SCHEMBL27239329	6-[2-[9-[4-[(1S,3R)-2-(2,2-difluoroethyl)-6-hydroxy-3-methyl-3,4-dihydro-1H-isoquinolin-1-yl]-3,5-difluorophenyl]-3-azaspiro[5.5]undecan-3-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934582	C[C@@H]1CC2=CC(O)=CC=C2[C@@H](C2=C(F)C=C(C3CCC4(CC3)CCN(C(=O)CN3CC5=CC6=C(C=C5C3)C(=O)N(C3CCC(=O)NC3=O)C6=O)CC4)C=C2F)N1CC(F)F	C45H47F4N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-LRC5YO	SCHEMBL27239527	6-[2-[9-[4-[(1R,3R)-2-(2,2-difluoroethyl)-6-hydroxy-3-methyl-3,4-dihydro-1H-isoquinolin-1-yl]phenyl]-3-azaspiro[5.5]undec-9-en-3-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934092	C[C@@H]1CC2=CC(O)=CC=C2[C@@H](C2=CC=C(C3=CCC4(CC3)CCN(C(=O)CN3CC5=CC6=C(C=C5C3)C(=O)N(C3CCC(=O)NC3=O)C6=O)CC4)C=C2)N1CC(F)F	C45H47F2N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-IQS5CQ	SCHEMBL27239438	6-[2-[9-[4-[(1S,3R)-2-(2,2-difluoroethyl)-6-hydroxy-3-methyl-3,4-dihydro-1H-isoquinolin-1-yl]phenyl]-3-azaspiro[5.5]undec-9-en-3-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934393	C[C@@H]1CC2=CC(O)=CC=C2[C@H](C2=CC=C(C3=CCC4(CC3)CCN(C(=O)CN3CC5=CC6=C(C=C5C3)C(=O)N(C3CCC(=O)NC3=O)C6=O)CC4)C=C2)N1CC(F)F	C45H47F2N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-R6RM0P	SCHEMBL27239279	6-[2-[9-[4-[(3R)-2-(2,2-difluoroethyl)-6-hydroxy-3-methyl-3,4-dihydro-1H-isoquinolin-1-yl]phenyl]-3-azaspiro[5.5]undecan-3-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934138	C[C@@H]1CC2=CC(O)=CC=C2C(C2=CC=C(C3CCC4(CC3)CCN(C(=O)CN3CC5=CC6=C(C=C5C3)C(=O)N(C3CCC(=O)NC3=O)C6=O)CC4)C=C2)N1CC(F)F	C45H49F2N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-0EUBU4	WO2022187588A1_E451	.	C[C@H]1CC2=CC(O)=CC=C2[C@@H](C2=C(F)C=C(NC3CC4(CCN(C(=O)CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C3)C=C2F)N1CC(F)F	C43H44F4N6O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-IJZSFU	SCHEMBL27239304	6-[2-[2-[4-[(1S,3R)-2-(2,2-difluoroethyl)-6-hydroxy-3-methyl-3,4-dihydro-1H-isoquinolin-1-yl]-3,5-difluoro-N-methylanilino]-7-azaspiro[3.5]nonan-7-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934411	C[C@@H]1CC2=CC(O)=CC=C2[C@@H](C2=C(F)C=C(N(C)C3CC4(CCN(C(=O)CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C3)C=C2F)N1CC(F)F	C44H46F4N6O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-0VGZPN	SCHEMBL27239332	6-[2-[7-[[4-[(1S,3R)-2-(2,2-difluoroethyl)-6-hydroxy-3-methyl-3,4-dihydro-1H-isoquinolin-1-yl]-3,5-difluorophenoxy]methyl]-2-azaspiro[3.5]nonan-2-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934199	C[C@@H]1CC2=CC(O)=CC=C2[C@@H](C2=C(F)C=C(OCC3CCC4(CC3)CN(C(=O)CN3CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C3)C4)C=C2F)N1CC(F)F	C44H45F4N5O7	ERα	P03372	CRBN	WO-2022187588-A1
TPD-MSASQE	SCHEMBL27239465	6-[[3-[4-[(1R,3R)-2-(2,2-difluoroethyl)-6-hydroxy-3-methyl-3,4-dihydro-1H-isoquinolin-1-yl]benzoyl]-3-azaspiro[5.5]undecan-9-yl]methyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934419	C[C@@H]1CC2=CC(O)=CC=C2[C@@H](C2=CC=C(C(=O)N3CCC4(CCC(CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2)N1CC(F)F	C45H49F2N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-TDEKKD	SCHEMBL27239555	6-[2-[2-[4-[(1S,3R)-2-(2,2-difluoroethyl)-6-hydroxy-3-methyl-3,4-dihydro-1H-isoquinolin-1-yl]-3,5-difluorophenoxy]-7-azaspiro[3.5]nonan-7-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934177	C[C@@H]1CC2=CC(O)=CC=C2[C@@H](C2=C(F)C=C(OC3CC4(CCN(C(=O)CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C3)C=C2F)N1CC(F)F	C43H43F4N5O7	ERα	P03372	CRBN	WO-2022187588-A1
TPD-UPLSVI	SCHEMBL27239378	6-[2-[2-[4-[(1R,3R)-2-(2,2-difluoroethyl)-6-hydroxy-3-methyl-3,4-dihydro-1H-isoquinolin-1-yl]-3,5-difluorophenoxy]-7-azaspiro[3.5]nonan-7-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934259	C[C@@H]1CC2=CC(O)=CC=C2[C@H](C2=C(F)C=C(OC3CC4(CCN(C(=O)CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C3)C=C2F)N1CC(F)F	C43H43F4N5O7	ERα	P03372	CRBN	WO-2022187588-A1
TPD-ZUBUWV	SCHEMBL27239476	6-[2-[2-[4-[(1S,3R)-2-(2,2-difluoroethyl)-6-hydroxy-3-methyl-3,4-dihydro-1H-isoquinolin-1-yl]-3,5-difluorobenzoyl]-2,7-diazaspiro[3.5]nonan-7-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934263	C[C@@H]1CC2=CC(O)=CC=C2[C@@H](C2=C(F)C=C(C(=O)N3CC4(CCN(C(=O)CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C3)C=C2F)N1CC(F)F	C43H42F4N6O7	ERα	P03372	CRBN	WO-2022187588-A1
TPD-1T0QEO	SCHEMBL27239374	6-[2-[2-[4-[(1R,3R)-2-(2,2-difluoroethyl)-6-hydroxy-3-methyl-3,4-dihydro-1H-isoquinolin-1-yl]-3,5-difluorobenzoyl]-2,7-diazaspiro[3.5]nonan-7-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934290	C[C@@H]1CC2=CC(O)=CC=C2[C@H](C2=C(F)C=C(C(=O)N3CC4(CCN(C(=O)CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C3)C=C2F)N1CC(F)F	C43H42F4N6O7	ERα	P03372	CRBN	WO-2022187588-A1
TPD-36RIF2	SCHEMBL27239480	6-[2-[2-[4-[(1R,3R)-2-(2,2-difluoroethyl)-6-hydroxy-3-methyl-3,4-dihydro-1H-isoquinolin-1-yl]benzoyl]-2,7-diazaspiro[3.5]nonan-7-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934417	C[C@@H]1CC2=CC(O)=CC=C2[C@@H](C2=CC=C(C(=O)N3CC4(CCN(C(=O)CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C3)C=C2)N1CC(F)F	C43H44F2N6O7	ERα	P03372	CRBN	WO-2022187588-A1
TPD-7338LU	SCHEMBL27239253	6-[2-[2-[4-[(1S,3R)-2-(2,2-difluoroethyl)-6-hydroxy-3-methyl-3,4-dihydro-1H-isoquinolin-1-yl]benzoyl]-2,7-diazaspiro[3.5]nonan-7-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934471	C[C@@H]1CC2=CC(O)=CC=C2[C@H](C2=CC=C(C(=O)N3CC4(CCN(C(=O)CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C3)C=C2)N1CC(F)F	C43H44F2N6O7	ERα	P03372	CRBN	WO-2022187588-A1
TPD-9E4OQN	WO2022187588A1_E461	.	COC1=C2CN(C3CCC(=O)NC3=O)C(=O)C2=CC2=C1CN(C(=O)CN1CCC3(CC1)CCN(C1=CC(F)=C([C@@H]4C5=CC=C(O)C=C5C[C@H](SC)N4CC(F)F)C(F)=C1)CC3)C2	C45H50F4N6O6S	ERα	P03372	CRBN	WO-2022187588-A1
TPD-WM9IN6	SCHEMBL27239410	2-(2,6-dioxopiperidin-3-yl)-6-[2-[9-[4-[(1R,3R)-2-(4-fluorophenyl)-6-hydroxy-3-methyl-3,4-dihydro-1H-isoquinolin-1-yl]phenyl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-oxoethyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934176	C[C@@H]1CC2=CC(O)=CC=C2[C@@H](C2=CC=C(N3CCC4(CCN(C(=O)CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2)N1C1=CC=C(F)C=C1	C48H49FN6O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-VVU5C2	SCHEMBL27239390	6-[[2-[4-[(1S,3R)-2-(2,2-difluoroethyl)-6-hydroxy-3-methyl-3,4-dihydro-1H-isoquinolin-1-yl]-3,5-difluorobenzoyl]-2-azaspiro[3.5]nonan-7-yl]methyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934171	C[C@@H]1CC2=CC(O)=CC=C2[C@@H](C2=C(F)C=C(C(=O)N3CC4(CCC(CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C3)C=C2F)N1CC(F)F	C43H43F4N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-50D6UL	SCHEMBL27239179	6-[[7-[4-[(1S,3R)-2-(2,2-difluoroethyl)-6-hydroxy-3-methyl-3,4-dihydro-1H-isoquinolin-1-yl]-3,5-difluorobenzoyl]-7-azaspiro[3.5]nonan-2-yl]methyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934193	C[C@@H]1CC2=CC(O)=CC=C2[C@@H](C2=C(F)C=C(C(=O)N3CCC4(CC3)CC(CN3CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C3)C4)C=C2F)N1CC(F)F	C43H43F4N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-32LR5Q	SCHEMBL30720119	2-(2,6-dioxopiperidin-3-yl)-6-[2-[9-[4-[(3S,4R)-7-hydroxy-3-phenyl-3,4-dihydro-2H-chromen-4-yl]phenyl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-oxoethyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC(=O)N2CCC3(CC2)CCN(C2=CC=C([C@@H]5C6=CC=C(O)C=C6OC[C@@H]5C5=CC=CC=C5)C=C2)CC3)C4)C(=O)N1	C47H47N5O7	ERα	P03372	CRBN	WO-2022187588-A1
TPD-WKW6RY	SCHEMBL27239161	6-[1-[4-[4-[(6S,8R)-7-(2,2-difluoroethyl)-8-methyl-3,6,8,9-tetrahydropyrazolo[4,3-f]isoquinolin-6-yl]-3,5-difluorophenyl]cyclohex-3-ene-1-carbonyl]piperidin-4-yl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934335	C[C@@H]1CC2=C(C=CC3=C2C=NN3)[C@@H](C2=C(F)C=C(C3=CCC(C(=O)N4CCC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2F)N1CC(F)F	C46H45F4N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-5YHG7T	SCHEMBL30934164	6-[8-[1-[4-[(6S,8R)-7-(2,2-difluoroethyl)-8-methyl-3,6,8,9-tetrahydropyrazolo[4,3-f]isoquinolin-6-yl]-3,5-difluorophenyl]piperidine-4-carbonyl]-8-azabicyclo[3.2.1]octan-3-yl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	C[C@@H]1CC2=C(C=CC3=C2C=NN3)[C@@H](C2=C(F)C=C(N3CCC(C(=O)N4C5CCC4CC(N4CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C4)C5)CC3)C=C2F)N1CC(F)F	C47H48F4N8O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-TQE3UN	SCHEMBL27239245	2-(2,6-dioxopiperidin-3-yl)-6-[2-[9-[6-[(6S,8R)-8-methyl-7-(2,2,2-trifluoroethyl)-3,6,8,9-tetrahydropyrazolo[4,3-f]isoquinolin-6-yl]pyridin-3-yl]-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl]-2-oxoethyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934249	C[C@@H]1CC2=C(C=CC3=C2C=NN3)[C@@H](C2=NC=C(N3CCC4(CC3)CN(C(=O)CN3CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C3)CCO4)C=C2)N1CC(F)(F)F	C43H44F3N9O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-31TU8Q	SCHEMBL27239486	2-(2,6-dioxopiperidin-3-yl)-6-[[2-[5-[(1R,3R)-2-(2-fluoro-2-methylpropyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyrimidin-2-yl]-2-azaspiro[3.5]nonan-7-yl]methyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=CN=C(N3CC4(CCC(CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C3)N=C2)N1CC(C)(C)F	C44H49FN8O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-TM6QLN	SCHEMBL27239590	6-[[2-[5-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyrimidin-2-yl]-2-azaspiro[3.5]nonan-7-yl]methyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934062	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=CN=C(N3CC4(CCC(CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C3)N=C2)N1CC(F)F	C42H44F2N8O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-MLLZ5C	SCHEMBL27239264	2-(2,6-dioxopiperidin-3-yl)-6-[[7-[5-[(1R,3R)-2-(2-fluoro-2-methylpropyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyrimidin-2-yl]-7-azaspiro[3.5]nonan-2-yl]methyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=CN=C(N3CCC4(CC3)CC(CN3CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C3)C4)N=C2)N1CC(C)(C)F	C44H49FN8O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-GLH23K	SCHEMBL27239328	6-[[7-[5-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyrimidin-2-yl]-7-azaspiro[3.5]nonan-2-yl]methyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934524	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=CN=C(N3CCC4(CC3)CC(CN3CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C3)C4)N=C2)N1CC(F)F	C42H44F2N8O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-MAT2X5	SCHEMBL27239277	6-[1-[4-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-2-fluorophenyl]cyclohexanecarbonyl]piperidin-4-yl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934282	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=CC(F)=C(C3CCC(C(=O)N4CCC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2)N1CC(F)F	C47H49F3N6O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-0R6WFA	SCHEMBL27239417	6-[2-[9-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]-3-azaspiro[5.5]undec-9-en-3-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934260	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(C3=CCC4(CC3)CCN(C(=O)CN3CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C3)CC4)C=C2F)N1CC(F)F	C47H46F4N6O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-VUMGTJ	WO2022187588A1_E477	.	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(C3=CCC4(CC3)CCN(C(=O)CN3CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C3)CC4)C=C2)N1CC(F)F	C47H47F3N6O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-K44NNT	SCHEMBL27239388	6-[2-[9-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]phenyl]-3-azaspiro[5.5]undec-9-en-3-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934220	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=CC=C(C3=CCC4(CC3)CCN(C(=O)CN3CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C3)CC4)C=C2)N1CC(F)F	C47H48F2N6O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-MQ0KFQ	SCHEMBL27239523	6-[2-[9-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3-fluorophenyl]-3-azaspiro[5.5]undecan-3-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934063	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(C3CCC4(CC3)CCN(C(=O)CN3CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C3)CC4)C=C2)N1CC(F)F	C47H49F3N6O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-MU9R9F	SCHEMBL27239383	6-[2-[9-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3,5-difluorophenyl]-3-azaspiro[5.5]undecan-3-yl]-2-oxoethyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934211	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(C3CCC4(CC3)CCN(C(=O)CN3CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C3)CC4)C=C2F)N1CC(F)F	C47H48F4N6O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-0YVQP7	SCHEMBL27239174	2-(2,6-dioxopiperidin-3-yl)-6-[1-[4-[3-fluoro-4-[(1R,3R)-2-(2-fluoro-2-methylpropyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]phenyl]cyclohex-3-ene-1-carbonyl]piperidin-4-yl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(C3=CCC(C(=O)N4CCC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2)N1CC(C)(C)F	C49H52F2N6O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-TZZ65H	SCHEMBL27239226	6-[1-[4-[4-[(1R,3R)-2-(2,2-difluoropropyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3-fluorophenyl]cyclohex-3-ene-1-carbonyl]piperidin-4-yl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934460	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(C3=CCC(C(=O)N4CCC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2)N1CC(C)(F)F	C48H49F3N6O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-87I8QM	SCHEMBL27239293	6-[1-[4-[6-[(1S,3R)-2-(2,2-difluoropropyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-5-fluoropyridin-3-yl]cyclohex-3-ene-1-carbonyl]piperidin-4-yl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934150	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(C3=CCC(C(=O)N4CCC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=N2)N1CC(C)(F)F	C47H48F3N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-GXOGG5	SCHEMBL27239240	2-(2,6-dioxopiperidin-3-yl)-6-[1-[4-[5-fluoro-6-[(1S,3R)-2-(2-fluoro-2-methylpropyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyridin-3-yl]cyclohex-3-ene-1-carbonyl]piperidin-4-yl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934217	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(C3=CCC(C(=O)N4CCC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=N2)N1CC(C)(C)F	C48H51F2N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-QMH392	SCHEMBL27239515	6-[1-[4-[3,5-difluoro-4-[(1R,3R)-2-[(1-fluorocyclopropyl)methyl]-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]phenyl]cyclohex-3-ene-1-carbonyl]piperidin-4-yl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934227	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(C3=CCC(C(=O)N4CCC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2F)N1CC1(F)CC1	C49H49F3N6O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-72J82N	WO2022187588A1_E486	.	C[C@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(C3=CCC(C(=O)N4CCC(N5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C=C2)N1CC1(F)CC1	C49H50F2N6O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-3CG5MS	SCHEMBL27239315	6-[1-[4-[4-[(1S,3R)-2-(2,2-difluoroethyl)-6-hydroxy-3-methyl-3,4-dihydro-1H-isoquinolin-1-yl]-3,5-difluorophenyl]cyclohexanecarbonyl]piperidin-4-yl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934441	C[C@@H]1CC2=CC(O)=CC=C2[C@@H](C2=C(F)C=C(C3CCC(C(=O)N4CCC(N5CC6=CC7=C(C=C6C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)CC3)C=C2F)N1CC(F)F	C45H47F4N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-JPI08E	SCHEMBL27239487	2-(2,6-dioxopiperidin-3-yl)-6-[1-[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-4-methylpiperidine-4-carbonyl]piperidin-4-yl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	CC1(C(=O)N2CCC(N3CC4=C(C=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)C3)CC2)CCN(C2=CC=C([C@@H]3C4=C(C=C(O)C=C4)CC[C@@H]3C3=CC=CC=C3)C=C2)CC1	C49H51N5O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-KIRA2B	SCHEMBL27239613	2-(2,6-dioxopiperidin-3-yl)-6-[1-[3-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]cyclobutanecarbonyl]piperidin-4-yl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(C2CCN(C(=O)[C@H]3C[C@@H](OC5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)C3)CC2)C4)C(=O)N1	C47H46N4O7	ERα	P03372	CRBN	WO-2022187588-A1
TPD-2X3C8I	WO2022187588A1_E491	.	O=C1CCC(N2CC3=CC4=C(C=C3C2=O)CN(C(=O)[C@H]2CC[C@H](CN3CC(OC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)C3)CC2)C4)C(=O)N1	C48H50N4O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-ICDVR7	SCHEMBL27239628	2-(2,6-dioxopiperidin-3-yl)-6-[[3-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]benzoyl]-3-azaspiro[5.5]undecan-9-yl]methyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934235	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC2CCC3(CC2)CCN(C(=O)C2=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=CC=C5)C=C2)CC3)C4)C(=O)N1	C49H50N4O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-5OI53I	SCHEMBL27239303	2-(2,6-dioxopiperidin-3-yl)-6-[[2-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]benzoyl]-2-azaspiro[3.5]nonan-7-yl]methyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934135	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC2CCC3(CC2)CN(C(=O)C2=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=CC=C5)C=C2)C3)C4)C(=O)N1	C47H46N4O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-H2JI0N	WO2022187588A1_E494	.	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC2CC3(CCN(C(=O)C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC3)C2)C4)C(=O)N1	C47H46N4O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-AC0JVL	SCHEMBL27239550	2-(2,6-dioxopiperidin-3-yl)-6-[2-[3-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]benzoyl]-3,9-diazaspiro[5.5]undecan-9-yl]-2-oxoethyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934254	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC(=O)N2CCC3(CC2)CCN(C(=O)C2=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=CC=C5)C=C2)CC3)C4)C(=O)N1	C49H49N5O7	ERα	P03372	CRBN	WO-2022187588-A1
TPD-Z8M6B6	SCHEMBL27239351	2-(2,6-dioxopiperidin-3-yl)-6-[2-[2-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]benzoyl]-2,7-diazaspiro[3.5]nonan-7-yl]-2-oxoethyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC(=O)N2CCC3(CC2)CN(C(=O)C2=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=CC=C5)C=C2)C3)C4)C(=O)N1	C47H45N5O7	ERα	P03372	CRBN	WO-2022187588-A1
TPD-Q9QKYN	SCHEMBL27239403	2-(2,6-dioxopiperidin-3-yl)-6-[8-[[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]-8-azabicyclo[3.2.1]octan-3-yl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934530	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(C2CC3CCC(C2)N3CC2CCN(C3=CC=C([C@@H]5C6=C(C=C(O)C=C6)CC[C@@H]5C5=CC=CC=C5)C=C3)CC2)C4)C(=O)N1	C50H53N5O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-R3A9BX	SCHEMBL27239541	2-(2,6-dioxopiperidin-3-yl)-6-[[4-[3-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]azetidine-1-carbonyl]cyclohexyl]methyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(C[C@H]2CC[C@@H](C(=O)N3CC(OC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)C3)CC2)C4)C(=O)N1	C48H48N4O7	ERα	P03372	CRBN	WO-2022187588-A1
TPD-5Z1D8J	SCHEMBL27239478	3-[6-[[4-[3-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]azetidine-1-carbonyl]cyclohexyl]methyl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30934504	O=C1CCC(N2CC3=CC4=C(C=C3C2=O)CN(C[C@H]2CC[C@H](C(=O)N3CC(OC5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)C3)CC2)C4)C(=O)N1	C48H50N4O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-UCN9QS	SCHEMBL27239437	2-(2,6-dioxopiperidin-3-yl)-1'-[[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]spiro[5,7-dihydrocyclopenta[f]isoindole-6,3'-azetidine]-1,3-dione; SCHEMBL30934527	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CC2(C4)CN(CC3CCN(C4=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=CC=C5)C=C4)CC3)C2)C(=O)N1	C46H46N4O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-IHPQNE	SCHEMBL27239141	2-(2,6-dioxopiperidin-3-yl)-1'-[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidine-4-carbonyl]spiro[5,7-dihydrocyclopenta[f]isoindole-6,3'-azetidine]-1,3-dione; SCHEMBL30934156	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CC2(C4)CN(C(=O)C3CCN(C4=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=CC=C5)C=C4)CC3)C2)C(=O)N1	C46H44N4O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-Q284CE	SCHEMBL27239448	2-(2,6-dioxopiperidin-3-yl)-1'-[2-[3-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]azetidin-1-yl]acetyl]spiro[5,7-dihydrocyclopenta[f]isoindole-6,3'-azetidine]-1,3-dione; SCHEMBL30934077	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CC2(C4)CN(C(=O)CN3CC(OC4=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=CC=C5)C=C4)C3)C2)C(=O)N1	C45H42N4O7	ERα	P03372	CRBN	WO-2022187588-A1
TPD-WUE78M	SCHEMBL27239175	2-(2,6-dioxopiperidin-3-yl)-1'-[2-[3-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]azetidin-1-yl]-2-oxoethyl]spiro[5,7-dihydrocyclopenta[f]isoindole-6,3'-azetidine]-1,3-dione; SCHEMBL30934507	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CC2(C4)CN(CC(=O)N3CC(OC4=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=CC=C5)C=C4)C3)C2)C(=O)N1	C45H42N4O7	ERα	P03372	CRBN	WO-2022187588-A1
TPD-ZUKZZ1	SCHEMBL27239208	2-(2,6-dioxopiperidin-3-yl)-6-[[1-[[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]azetidin-3-yl]methyl]-1,5-dihydropyrrolo[3,4-f]isoindole-3,7-dione; SCHEMBL30934448	O=C1CCC(N2CC3=CC4=C(C=C3C2=O)CN(CC2CN(CC3CCN(C5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC3)C2)C4=O)C(=O)N1	C47H49N5O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-LWCRR6	SCHEMBL27239542	6-(2,6-dioxopiperidin-3-yl)-2-[1-[[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]azetidin-3-yl]-1,5-dihydropyrrolo[3,4-f]isoindole-3,7-dione; SCHEMBL30934103	O=C1CCC(N2CC3=CC4=C(C=C3C2=O)CN(C2CN(CC3CCN(C5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC3)C2)C4=O)C(=O)N1	C46H47N5O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-68IFFP	SCHEMBL27239203	2-(2,6-dioxopiperidin-3-yl)-6-[1-[[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperidin-4-yl]-1,5-dihydropyrrolo[3,4-f]isoindole-3,7-dione; SCHEMBL30934363	O=C1CCC(N2CC3=CC4=C(C=C3C2=O)CN(C2CCN(CC3CCN(C5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC3)CC2)C4=O)C(=O)N1	C48H51N5O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-6RZBSZ	SCHEMBL27239182	2-(2,6-dioxopiperidin-3-yl)-6-[1-[[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperidin-4-yl]-3,5-dihydropyrrolo[3,4-f]isoindole-1,7-dione; SCHEMBL30934060	O=C1CCC(N2CC3=CC4=C(C=C3C2=O)C(=O)N(C2CCN(CC3CCN(C5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC3)CC2)C4)C(=O)N1	C48H51N5O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-PK2ZQJ	SCHEMBL27239283	2-(2,6-dioxopiperidin-3-yl)-6-[[1-[[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]azetidin-3-yl]methyl]-3,5-dihydropyrrolo[3,4-f]isoindole-1,7-dione; SCHEMBL30934359	O=C1CCC(N2CC3=CC4=C(C=C3C2=O)C(=O)N(CC2CN(CC3CCN(C5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC3)C2)C4)C(=O)N1	C47H49N5O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-J25QHR	SCHEMBL27239252	2-(2,6-dioxopiperidin-3-yl)-6-[2-[9-[4-[(1R,2S)-6-(1-methylpyrazol-4-yl)-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-oxoethyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934118	CN1C=C(C2=CC3=C(C=C2)[C@@H](C2=CC=C(N4CCC5(CCN(C(=O)CN6CC7=C(C=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)C6)CC5)CC4)C=C2)[C@@H](C2=CC=CC=C2)CC3)C=N1	C52H53N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-LNIE9O	SCHEMBL27239451	2-(2,6-dioxopiperidin-3-yl)-6-[2-oxo-2-[9-[4-[(1R,2S)-2-phenyl-6-(1H-pyrazol-4-yl)-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-3,9-diazaspiro[5.5]undecan-3-yl]ethyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934181	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC(=O)N2CCC3(CC2)CCN(C2=CC=C([C@@H]5C6=C(C=C(C7=CNN=C7)C=C6)CC[C@@H]5C5=CC=CC=C5)C=C2)CC3)C4)C(=O)N1	C51H51N7O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-EF6P6I	SCHEMBL27239404	2-(2,6-dioxopiperidin-3-yl)-6-[2-[9-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl]-2-oxoethyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934355	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC(=O)N2CCOC3(CCN(C5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC3)C2)C4)C(=O)N1	C47H47N5O7	ERα	P03372	CRBN	WO-2022187588-A1
TPD-E7Y3TI	SCHEMBL27239568	6-[[7-[5-[(1R,3R)-2-(2,2-difluoro-3-hydroxypropyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyrimidin-2-yl]-7-azaspiro[3.5]nonan-2-yl]methyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=CN=C(N3CCC4(CC3)CC(CN3CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C3)C4)N=C2)N1CC(F)(F)CO	C43H46F2N8O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-RG8D34	SCHEMBL27239151	6-[[2-[5-[(1R,3R)-2-(2,2-difluoro-3-hydroxypropyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyrimidin-2-yl]-2-azaspiro[3.5]nonan-7-yl]methyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934295	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=CN=C(N3CC4(CCC(CN5CC6=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C3)N=C2)N1CC(F)(F)CO	C43H46F2N8O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-D0RCHW	SCHEMBL27239414	2-(2,6-dioxopiperidin-3-yl)-6-[2-[9-[4-[(1R,3R)-2-(2-fluoro-2-methylpropyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3-methoxyphenyl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-oxoethyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	COC1=C([C@@H]2C3=C(C[C@@H](C)N2CC(C)(C)F)C2=C(C=CC=C2)N3)C=CC(N2CCC3(CCN(C(=O)CN4CC5=C(C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)CC2)=C1	C49H56FN7O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-OYNAOO	SCHEMBL27239552	2-(2,6-dioxopiperidin-3-yl)-6-[[8-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-1-oxa-8-azaspiro[4.5]decan-3-yl]methyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934408	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC2COC3(CCN(C5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC3)C2)C4)C(=O)N1	C46H46N4O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-SY8CCT	SCHEMBL27239518	3-[6-[[8-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-1-oxa-8-azaspiro[4.5]decan-3-yl]methyl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30934045	O=C1CCC(N2CC3=CC4=C(C=C3C2=O)CN(CC2COC3(CCN(C5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC3)C2)C4)C(=O)N1	C46H48N4O5	ERα	P03372	CRBN	WO-2022187588-A1
TPD-US816W	SCHEMBL27239357	2-(2,6-dioxopiperidin-3-yl)-6-[[9-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-1,5-dioxa-9-azaspiro[5.5]undecan-3-yl]methyl]-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione; SCHEMBL30934327	O=C1CCC(N2C(=O)C3=CC4=C(C=C3C2=O)CN(CC2COC3(CCN(C5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC3)OC2)C4)C(=O)N1	C46H46N4O7	ERα	P03372	CRBN	WO-2022187588-A1
TPD-OZ629H	SCHEMBL30934047	3-[6-[[9-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-1,5-dioxa-9-azaspiro[5.5]undecan-3-yl]methyl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC4=C(C=C3C2=O)CN(CC2COC3(CCN(C5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC3)OC2)C4)C(=O)N1	C46H48N4O6	ERα	P03372	CRBN	WO-2022187588-A1
TPD-K49KSN	SCHEMBL27239407	3-[1'-[[(3S)-1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]pyrrolidin-3-yl]methyl]-1-oxospiro[5,7-dihydro-3H-cyclopenta[f]isoindole-6,3'-azetidine]-2-yl]piperidine-2,6-dione; SCHEMBL30934374	O=C1CCC(N2CC3=CC4=C(C=C3C2=O)CC2(C4)CN(C[C@@H]3CCN(C4=CC=C([C@@H]5C6=C(C=C(O)C=C6)CC[C@@H]5C5=CC=CC=C5)C=C4)C3)C2)C(=O)N1	C45H46N4O4	ERα	P03372	CRBN	WO-2022187588-A1
TPD-3754PX	SCHEMBL24677977	N-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]-2-[[1-[[4-[[(1R)-1-[2-fluoro-3-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxymethyl]cyclopropyl]methyl-methylamino]acetamide	COC1=CC2=C(C=C1OCC1(CN(C)CC(=O)NC3=CC=CC4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC1)C(N[C@H](C)C1=CC=CC(C(F)(F)F)=C1F)=NC(C)=N2	C40H39F4N7O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-3A7LAV	SCHEMBL24677710	7-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]-N-[[1-[[4-[[(1R)-1-[2-fluoro-3-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxymethyl]cyclopropyl]methyl]-N-methylheptanamide	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CCCCCCNC3=CC=CC4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC1)C(N[C@H](C)C1=CC=CC(C(F)(F)F)=C1F)=NC(C)=N2	C45H49F4N7O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-86KXG7	SCHEMBL29922325	4-[[6-[(3S)-3-[4-[[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxypyrrolidin-1-yl]-6-oxohexyl]amino]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	COC1=CC2=C(C=C1O[C@H]1CCN(C(=O)CCCCCNC3=CC=CC4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)C1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C42H45F3N8O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-ERQ0XV	WO2022188819A1_101	.	COC1=CC2=C(C=C1O[C@H]1CCN(C(=O)CCOCCOCCNC3=CC=CC4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)C1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C43H47F3N8O9	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-RZFSVG	WO2022188819A1_102	.	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)C(C)(C)OCCCCNC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C46H53F3N8O8	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-A0U8QT	SCHEMBL28863575	N-[[1-[[4-[[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxymethyl]cyclopropyl]methyl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]cyclohexyl]oxy-N-methylbutanamide; PD216675	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CCCOC3CCC(NC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C48H55F3N8O8	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-TET2HB	WO2022188819A1_104	.	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CCC(=O)N(C)C3CCC(NC4=CC=CC5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C49H56F3N9O8	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-A3JECI	SCHEMBL28863606	N-[[1-[[4-[[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxymethyl]cyclopropyl]methyl]-4-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]-N-methylbutanamide	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CCCOCCNC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C44H49F3N8O8	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-54K3SR	WO2022188819A1_106	.	COC1=CC2=C(C=C1OCC(C)(C)CN(C)C(=O)CCCN1CCN(C3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C46H54F3N9O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-T5YZHZ	SCHEMBL28863585	N-[[1-[[4-[[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxymethyl]cyclopropyl]methyl]-5-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]-N-methylpentanamide	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CCCCN3CCN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C47H54F3N9O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-ROANM5	SCHEMBL28863614	N-[[1-[[4-[[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxymethyl]cyclopropyl]methyl]-3-[4-[4-[(2,6-dioxopiperidin-3-yl)amino]phenyl]piperidin-1-yl]-N-methylpropanamide	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CCN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C44H53F3N8O5	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-H7DJ9E	WO2022188819A1_109	.	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CN3CCN(C4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)N2	C49H59F3N10O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-FIWUUY	SCHEMBL24678228	3-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]-N-[[1-[[4-[[(1R)-1-[2-fluoro-3-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxymethyl]cyclopropyl]methyl]-N-methylpropanamide	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CCOCCOCCNC3=CC=CC4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC1)C(N[C@H](C)C1=CC=CC(C(F)(F)F)=C1F)=NC(C)=N2	C45H49F4N7O9	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-AY8VO6	WO2022188819A1_110	.	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)C3CCN(C(=O)C4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C50H56F3N9O8	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-Y70HLN	WO2022188819A1_111	.	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CN3CCC4(CC3)CCN(C3=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C3)CC4)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C49H56F3N9O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-NSGNTU	WO2022188819A1_112	.	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CN3CCC(CNC4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C46H52F3N9O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-3QQNHO	WO2022188819A1_113	.	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CCCCCCNC3=C4C(=CC=C3)N(C3CCC(=O)NC3=O)C(=O)N4C)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C45H54F3N9O6	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-9IOWC6	SCHEMBL29922135	N-[[1-[[4-[[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxymethyl]cyclopropyl]methyl]-2-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]-N-methylacetamide	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CN3CCC(CN4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C50H59F3N10O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-Z81ZAN	SCHEMBL28863647	N-[[1-[[4-[[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxymethyl]cyclopropyl]methyl]-4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]-N-methylcyclohexane-1-carboxamide	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)C3CCC(N4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C49H56F3N9O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-BHI6E1	SCHEMBL29922551	N-[[1-[[4-[[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxymethyl]cyclopropyl]methyl]-2-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]-N-methylacetamide	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CN3CCC(CN4CCN(C5=C(F)C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C50H58F4N10O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-LDA7B8	SCHEMBL29922573	N-[[1-[[4-[[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxymethyl]cyclopropyl]methyl]-4-[[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]cyclohexyl]-methylamino]-N-methylbutanamide	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CCCN(C)C3CCC(NC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C49H58F3N9O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-IE6643	SCHEMBL24678242	N-[[1-[[4-[[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxymethyl]cyclopropyl]methyl]-1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]-N-methylpiperidine-4-carboxamide	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)C3CCN(C4CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C49H56F3N9O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-P5XQPV	SCHEMBL29922187	N-[[1-[[4-[[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxymethyl]cyclopropyl]methyl]-2-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]oxypiperidin-1-yl]-N-methylacetamide	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CN3CCC(OC4CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C50H58F3N9O8	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-X3PG6U	SCHEMBL28863642	1-[[4-[[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxymethyl]-N-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethyl]cyclopropane-1-carboxamide; SCHEMBL29922351	COC1=CC2=C(C=C1OCC1(C(=O)NCCNC3=CC=CC4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C39H39F3N8O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-I7MUGN	WO2022188819A1_120	.	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CN3CCN(C4CN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C47H53F3N10O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-426LNM	SCHEMBL24677866	N-[[1-[[4-[[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxymethyl]cyclopropyl]methyl]-4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]amino]-N-methylcyclohexane-1-carboxamide	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)C3CCC(NC4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C50H58F3N9O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-8KDUWC	WO2022188819A1_122	.	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)C3CCN(CCN4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C50H59F3N10O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-YDOPHF	SCHEMBL28863640	N-[[1-[[4-[[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxymethyl]cyclopropyl]methyl]-4-[4-[4-[(2,6-dioxopiperidin-3-yl)amino]phenyl]piperidin-1-yl]-N-methylbutanamide	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CCCN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C45H55F3N8O5	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-MNHZPS	SCHEMBL29922583	N-[[1-[[4-[[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxymethyl]cyclopropyl]methyl]-2-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]-N-methylacetamide	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CN3CCC(CN4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)CC6=C5)CC4)CC3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C50H61F3N10O6	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-JJKBBN	SCHEMBL28956619	N-[[1-[[4-[[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxymethyl]cyclopropyl]methyl]-3-[4-[[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]methyl]piperidin-1-yl]-N-methylpropanamide	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CCN3CCC(CNC4=CC=CC5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C47H54F3N9O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-I1L0P3	WO2022188819A1_126	.	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)C3CCC(OC4CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C50H57F3N8O8	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-IINOFJ	WO2022188819A1_127	.	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)COCCN3CCN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C46H52F3N9O8	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-6QCHEZ	SCHEMBL28863561	N-[[1-[[4-[[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxymethyl]cyclopropyl]methyl]-1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]-N-methylpiperidine-4-carboxamide; SCHEMBL29922255	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)C3CCN(C4=CC=C(N5CCC(=O)NC5=O)C=C4)CC3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C41H47F3N8O5	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-RXIA83	WO2022188819A1_129	.	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CN3CCN(C4=CC=C(N5CCC(=O)NC5=O)C=C4)CC3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C41H48F3N9O5	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-JFE127	SCHEMBL24677956	1-[[4-[[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxymethyl]-N-[3-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]propyl]cyclopropane-1-carboxamide; SCHEMBL29922412	COC1=CC2=C(C=C1OCC1(C(=O)NCCCNC3=CC=CC4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C40H41F3N8O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-HWFYRL	WO2022188819A1_130	.	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CCN3CCN(C4=CC=C(N5CCC(=O)NC5=O)C=C4)CC3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C42H50F3N9O5	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-GU7CQS	SCHEMBL24678207	N-[[1-[[4-[[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxymethyl]cyclopropyl]methyl]-4-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperazin-1-yl]-N-methylbutanamide	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CCCN3CCN(C4=CC=C(N5CCC(=O)NC5=O)C=C4)CC3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C43H52F3N9O5	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-YHXLMI	WO2022188819A1_132	.	COC1=CC2=C(C=C1OCC(C)(C)CN(C)C(=O)CCCCN1CCN(C3=CC=C(N4CCC(=O)NC4=O)C=C3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C44H56F3N9O5	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-YEHJPE	WO2022188819A1_133	.	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CCOCCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCC3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C53H66F3N9O8S	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-L4K776	WO2022188819A1_134	.	COC1=CC2=C(C=C1OCC1(CN(C)CC3CCN(C4=CC=C(N5CCC(=O)NC5=O)C=C4)CC3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C41H49F3N8O4	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-LTMX42	WO2022188819A1_135-1	.	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)C3CCN([C@H]4C[C@@H](NC5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)C4)CC3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C48H54F3N9O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-UFGVCZ	WO2022188819A1_135-2	.	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)C3CCN([C@H]4C[C@H](NC5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)C4)CC3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C48H54F3N9O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-31JX2D	SCHEMBL24677963	5-[[7-[[1-[[4-[[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxymethyl]cyclopropyl]methyl-methylamino]-7-oxoheptyl]amino]-N-(2,6-dioxopiperidin-3-yl)-2-fluorobenzamide	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CCCCCCNC3=CC(C(=O)NC4CCC(=O)NC4=O)=C(F)C=C3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C44H52F4N8O6	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-RFSI4D	SCHEMBL24677721	N-[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]-6-(2-methoxyethoxy)-2-methyl-7-piperidin-4-yloxyquinazolin-4-amine; SCHEMBL29922333	COCCOC1=CC2=C(C=C1OC1CCNCC1)N=C(C)N=C2N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1	C26H32F3N5O3	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-4U359S	SCHEMBL29922558	N-[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]-7-(azetidin-3-yloxy)-6-(2-methoxyethoxy)-2-methylquinazolin-4-amine	COCCOC1=CC2=C(C=C1OC1CNC1)N=C(C)N=C2N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1	C24H28F3N5O3	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-F4KRH8	WO2022188819A1_139	.	COCCOC1=CC2=C(C=C1OC1CCN(CC3CCN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC1)N=C(C)N=C2N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1	C45H51F3N8O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-HQ6277	WO2022188819A1_14	.	COC1=CC2=C(C=C1OCC1(C(=O)NCCCCNC3=CC=CC4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C41H43F3N8O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-9WRNKR	WO2022188819A1_140	.	COCCOC1=CC2=C(C=C1OC1CCN(CC3CCN(C4=CC=C(N5CCC(=O)NC5=O)C=C4)CC3)CC1)N=C(C)N=C2N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1	C42H51F3N8O5	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-THXQNW	WO2022188819A1_141	.	COCCOC1=CC2=C(C=C1OC1CCN(C3CCN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC1)N=C(C)N=C2N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1	C44H49F3N8O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-8UMXUV	SCHEMBL29922335	5-[4-[4-[[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]amino]-2-methyl-6-[(3S)-oxolan-3-yl]oxyquinazolin-7-yl]oxypiperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CC1=NC2=C(C=C(O[C@H]3CCOC3)C(OC3CCN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)=C2)C(N[C@H](C)C2=CC(N)=CC(C(F)(F)F)=C2)=N1	C40H40F3N7O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-P657YJ	SCHEMBL29922676	1-[[4-[[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxymethyl]-N-[5-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]pentyl]cyclopropane-1-carboxamide	COC1=CC2=C(C=C1OCC1(C(=O)NCCCCCNC3=CC=CC4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C42H45F3N8O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-CS3NLQ	WO2022188819A1_16	.	COC1=CC2=C(C=C1OCC1(C(=O)NCCCCCCNC3=CC=CC4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C43H47F3N8O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-EXVQ04	SCHEMBL24677854	1-[[4-[[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxymethyl]-N-[7-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]heptyl]cyclopropane-1-carboxamide	COC1=CC2=C(C=C1OCC1(C(=O)NCCCCCCCNC3=CC=CC4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C44H49F3N8O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-KZTR50	WO2022188819A1_18	.	COC1=CC2=C(C=C1OCC1(C(=O)NCCCCCCCCNC3=CC=CC4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C45H51F3N8O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-541M8X	WO2022188819A1_19	.	COC1=CC2=C(C=C1OCC1(C(=O)NCCOCC(=O)NC3=CC=CC4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C41H41F3N8O9	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-V7C8XQ	WO2022188819A1_2	.	COC1=CC2=C(C=C1OCC1(CN(C)CC(=O)NC3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC1)C(N[C@H](C)C1=CC=CC(C(F)(F)F)=C1F)=NC(C)=N2	C40H39F4N7O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-DHS47C	SCHEMBL24677855	1-[[4-[[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxymethyl]-N-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]-2-oxoethoxy]ethoxy]ethyl]cyclopropane-1-carboxamide	COC1=CC2=C(C=C1OCC1(C(=O)NCCOCCOCC(=O)NC3=CC=CC4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C43H45F3N8O10	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-LNLGUM	WO2022188819A1_21	.	COC1=CC2=C(C=C1OCC1(C(=O)NCCCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCC3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C50H60F3N9O7S	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-TNA1R1	WO2022188819A1_22	N-[[1-[[4-[[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxymethyl]cyclopropyl]methyl]-3-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]-N-methylpropanamide	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CCNC3=CC=CC4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C41H43F3N8O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-F9QT19	SCHEMBL24677951	N-[[1-[[4-[[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxymethyl]cyclopropyl]methyl]-4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]-N-methylbutanamide	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CCCNC3=CC=CC4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C42H45F3N8O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-K41QEH	PD216659	N-[[1-[[4-[[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxymethyl]cyclopropyl]methyl]-5-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]-N-methylpentanamide	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CCCCNC3=CC=CC4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C43H47F3N8O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-BFMJZY	SCHEMBL24677853	N-[[1-[[4-[[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxymethyl]cyclopropyl]methyl]-6-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]-N-methylhexanamide	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CCCCCNC3=CC=CC4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C44H49F3N8O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-E4585B	PROTAC SOS1 degrader-5	PROTAC SOS1 degrader-5; 2836273-61-9; orb2565416; EX-A9151; PD216661; HY-161173; CS-0979282	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CCCCCCNC3=CC=CC4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C45H51F3N8O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-F8KYFI	SCHEMBL24678219	N-[[1-[[4-[[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxymethyl]cyclopropyl]methyl]-10-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]-N-methyldecanamide	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CCCCCCCCCNC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C48H57F3N8O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-9FTAWY	WO2022188819A1_28	.	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)COCCNC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C42H45F3N8O8	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-1TFOH6	WO2022188819A1_29	.	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CCOCCNC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C43H47F3N8O8	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-2V1W4I	WO2022188819A1_3	.	COC1=CC2=C(C=C1OCC1(CN(C)CC(=O)NC3=CC=CC4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C40H41F3N8O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-EHMCS8	SCHEMBL29922427	N-[[1-[[4-[[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxymethyl]cyclopropyl]methyl]-3-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]-N-methylpropanamide	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CCOCCOCCNC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C45H51F3N8O9	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-Q9YH11	WO2022188819A1_31	.	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CNC(=O)CNC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C42H44F3N9O8	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-FZB650	WO2022188819A1_32	.	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CCNC(=O)CNC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C43H46F3N9O8	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-84PA8L	WO2022188819A1_33	.	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CCCNC(=O)CNC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C44H48F3N9O8	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-6LRR3G	SCHEMBL24677980	N-[[1-[[4-[[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxymethyl]cyclopropyl]methyl]-2-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyacetyl]amino]-N-methylacetamide	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CNC(=O)COC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C42H43F3N8O9	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-ALUM4Q	SCHEMBL24677708	N-[[1-[[4-[[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxymethyl]cyclopropyl]methyl]-3-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyacetyl]amino]-N-methylpropanamide	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CCNC(=O)COC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C43H45F3N8O9	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-D6ZFHV	WO2022188819A1_36	.	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CCCNC(=O)COC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C44H47F3N8O9	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-NGQW2P	WO2022188819A1_37	.	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CNC(=O)CNC3=CC=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)N2	C42H46F3N9O8	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-UJ1QBR	SCHEMBL24677978	N-[[1-[[4-[[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxymethyl]cyclopropyl]methyl]-3-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]amino]acetyl]amino]-N-methylpropanamide	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CCNC(=O)CNC3=CC=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C43H46F3N9O8	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-4L12AF	SCHEMBL24678225	N-[[1-[[4-[[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxymethyl]cyclopropyl]methyl]-4-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]amino]acetyl]amino]-N-methylbutanamide	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CCCNC(=O)CNC3=CC=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C44H48F3N9O8	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-E2UAIP	SCHEMBL24678186	2-[[1-[[4-[[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxymethyl]cyclopropyl]methyl-methylamino]-N-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]acetamide	COC1=CC2=C(C=C1OCC1(CN(C)CC(=O)NC3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C40H41F3N8O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-G0ZIBM	WO2022188819A1_40	.	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CNC(=O)COC3=CC=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C42H43F3N8O9	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-C3G1OT	WO2022188819A1_41	N-[[1-[[4-[[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxymethyl]cyclopropyl]methyl]-3-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxyacetyl]amino]-N-methylpropanamide	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CCNC(=O)COC3=CC=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C43H45F3N8O9	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-KC2FN6	WO2022188819A1_42	.	COC1=CC2=C(C=C1OCC(C)(C)CN(C)C(=O)CCCNC(=O)COC1=CC=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=C1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C44H49F3N8O9	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-F5OF4N	SCHEMBL24677860	5-[4-[(3S)-3-[4-[[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxypyrrolidin-1-yl]piperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione; SCHEMBL29922554	COC1=CC2=C(C=C1O[C@H]1CCN(C3CCN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)C1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C41H43F3N8O6	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-L1C7EJ	WO2022188819A1_44	.	COC1=CC2=C(C=C1O[C@H]1CCN(C3CCN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5)CC3)C1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C41H45F3N8O5	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-O0ZORG	SCHEMBL29922540	5-[4-[(3S)-3-[4-[[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxypyrrolidin-1-yl]piperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)-6-fluoroisoindole-1,3-dione	COC1=CC2=C(C=C1O[C@H]1CCN(C3CCN(C4=CC5=C(C=C4F)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)C1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C41H42F4N8O6	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-RRONRY	SCHEMBL29922519	3-[6-[4-[[(3S)-3-[4-[[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxypyrrolidin-1-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	COC1=CC2=C(C=C1O[C@H]1CCN(CC3CCN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5)CC3)C1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C42H47F3N8O5	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-7HQCRM	WO2022188819A1_47	.	COC1=CC2=C(C=C1O[C@H]1CCN(C(=O)C3CCN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5)CC3)C1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C42H45F3N8O6	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-494HAV	WO2022188819A1_48	.	COC1=CC2=NC(C)=NC(N[C@H](C)C3=CC(N)=CC(C(F)(F)F)=C3)=C2C=C1OCCCCC(=O)NC1=CC2=C(C=C1)C(=O)N(C1CCC(=O)NC1=O)C2=O	C37H36F3N7O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-7HUXTU	WO2022188819A1_49	.	COC1=CC2=NC(C)=NC(N[C@H](C)C3=CC(N)=CC(C(F)(F)F)=C3)=C2C=C1OCCOCCC(=O)NC1=CC2=C(C=C1)C(=O)N(C1CCC(=O)NC1=O)C2=O	C37H36F3N7O8	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-O5K238	WO2022188819A1_5	.	COC1=CC2=C(C=C1OCC1(CN(C)CCC(=O)NC3=CC=CC4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC1)C(N[C@H](C)C1=CC=CC(C(F)(F)F)=C1F)=NC(C)=N2	C41H41F4N7O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-ECPAXV	WO2022188819A1_50	.	COC1=CC2=NC(C)=NC(N[C@H](C)C3=CC(N)=CC(C(F)(F)F)=C3)=C2C=C1OCCOCCOCCC(=O)NC1=CC2=C(C=C1)C(=O)N(C1CCC(=O)NC1=O)C2=O	C39H40F3N7O9	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-B8D7WF	SCHEMBL24678237	4-[4-[(3S)-3-[4-[[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxypyrrolidin-1-yl]piperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione; SCHEMBL29922249	COC1=CC2=C(C=C1O[C@H]1CCN(C3CCN(C4=CC=CC5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)C1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C41H43F3N8O6	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-F5Q76I	SCHEMBL29922556	4-[4-[[(3S)-3-[4-[[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxypyrrolidin-1-yl]methyl]piperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	COC1=CC2=C(C=C1O[C@H]1CCN(CC3CCN(C4=CC=CC5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)C1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C42H45F3N8O6	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-MOZHHJ	WO2022188819A1_53	.	COC1=CC2=C(C=C1OCC1(C(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCC3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C46H53F3N8O6S	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-VCVLDT	WO2022188819A1_54	.	COC1=CC2=C(C=C1OCC1(C(=O)NC3=CC=CC4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C37H34F3N7O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-XCIZ68	WO2022188819A1_55	.	COC1=CC2=C(C=C1OCC1(C(=O)NC3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C37H34F3N7O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-R5MFOB	WO2022188819A1_56	.	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CC3CCN(C4=CC=CC5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C45H49F3N8O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-WDKCJ6	SCHEMBL24677969	N-[[1-[[4-[[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxymethyl]cyclopropyl]methyl]-1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]-N-methylpiperidine-4-carboxamide	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)C3CCN(C4=CC=CC5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C44H47F3N8O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-WES51M	SCHEMBL29922586	4-[4-[(3S)-3-[4-[[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxypyrrolidine-1-carbonyl]piperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	COC1=CC2=C(C=C1O[C@H]1CCN(C(=O)C3CCN(C4=CC=CC5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)C1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C42H43F3N8O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-J8LYEV	WO2022188819A1_59	.	COC1=CC2=C(C=C1O[C@H]1CCN(C(=O)CC3CCN(C4=CC=CC5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)C1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C43H45F3N8O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-91INE8	SCHEMBL24677724	N-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-3-[[1-[[4-[[(1R)-1-[2-fluoro-3-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxymethyl]cyclopropyl]methyl-methylamino]propanamide	COC1=CC2=C(C=C1OCC1(CN(C)CCC(=O)NC3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC1)C(N[C@H](C)C1=CC=CC(C(F)(F)F)=C1F)=NC(C)=N2	C41H41F4N7O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-NTVD5V	WO2022188819A1_60	.	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)C3CCN(C4CN(C5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)C4)CC3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C47H52F3N9O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-B9Q0U7	WO2022188819A1_61	.	COC1=CC2=C(C=C1OCC1(C(=O)N3CC4CN(C(=O)CNC5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)CC4C3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C45H46F3N9O8	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-JC0MI5	WO2022188819A1_62	.	COC1=CC2=C(C=C1OCC1(C(=O)N3CC4(CCN(C(=O)CNC5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)CC4)C3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C46H48F3N9O8	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-8DGBT6	WO2022188819A1_63	.	COC1=CC2=C(C=C1OCC1(C(=O)N3CCC4(CCN(C(=O)CNC5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)CC4)C3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C47H50F3N9O8	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-FLEBBM	SCHEMBL24677718	4-[5-[4-[[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxypent-1-ynyl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione; SCHEMBL29922245	COC1=CC2=C(C=C1OCCCC#CC1=CC=CC3=C1C(=O)N(C1CCC(=O)NC1=O)C3=O)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C37H33F3N6O6	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-A2F4EZ	SCHEMBL28863584	N-[[1-[[4-[[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxymethyl]cyclopropyl]methyl]-N-methyl-7-[[2-(1-methyl-2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]heptanamide	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CCCCCCNC3=C4C(=O)N(C5CCC(=O)N(C)C5=O)C(=O)C4=CC=C3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C46H53F3N8O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-LTG47F	PD216665	N-[[1-[[4-[[(1R)-1-[3-(difluoromethyl)-2-fluorophenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxymethyl]cyclopropyl]methyl]-7-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]-N-methylheptanamide	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CCCCCCNC3=CC=CC4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC1)C(N[C@H](C)C1=CC=CC(C(F)F)=C1F)=NC(C)=N2	C45H50F3N7O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-XI2NKZ	PD216663	N-[[1-[[4-[[(1R)-1-[3-amino-5-(difluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxymethyl]cyclopropyl]methyl]-7-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]-N-methylheptanamide	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CCCCCCNC3=CC=CC4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)F)=C1)=NC(C)=N2	C45H52F2N8O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-29UTYT	WO2022188819A1_68	.	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CCCCCCNC3=CC=CC4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)C(C)(C)O)=C1F)=NC(C)=N2	C48H57F3N8O8	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-VZZ65M	WO2022188819A1_69	.	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CCCCCCNC3=CC=CC4=C3C(=O)N(C3CCC(=O)N(COC(=O)C(C)(C)C)C3=O)C4=O)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C51H61F3N8O9	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-U2ZBIO	SCHEMBL24677722	2-(2,6-dioxopiperidin-3-yl)-4-[[1-[[4-[[(1R)-1-[2-fluoro-3-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxymethyl]cyclopropyl]methylamino]isoindole-1,3-dione	COC1=CC2=C(C=C1OCC1(CNC3=CC=CC4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC1)C(N[C@H](C)C1=CC=CC(C(F)(F)F)=C1F)=NC(C)=N2	C37H34F4N6O6	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-MXH3IB	WO2022188819A1_70	.	COC1=CC2=C(C=C1OCC1(COC(=O)CCCCCCNC3=CC=CC4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C44H48F3N7O8	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-KGBUWA	WO2022188819A1_71	.	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CCCCCCNC3=CC=CC4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC1)C(N[C@H](C)C1=CC=CC(C#N)=C1C)=NC(C)=N2	C46H52N8O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-XA38CH	WO2022188819A1_72	.	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)C3CCN(C4CCN(C5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)CC4)CC3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C49H56F3N9O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-RK06CO	SCHEMBL28956701	N-[[1-[[4-[[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxymethyl]cyclopropyl]methyl]-3-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperazin-1-yl]-N-methylpropanamide	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CCN3CCN(C4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C45H50F3N9O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-GCSLT7	WO2022188819A1_74	.	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CCCCCCNC3=CC=CC4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)C(C)(C)O)=C1)=NC(C)=N2	C48H58F2N8O8	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-B6KXZO	SCHEMBL24678190	N-[[1-[[4-[[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxymethyl]cyclopropyl]methyl]-7-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]-N-methylheptanamide; PD216667	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CCCCCCNC3=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C45H53F3N8O6	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-TADS6Y	SCHEMBL28863659	N-[[1-[[4-[[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxymethyl]cyclopropyl]methyl]-4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperazin-1-yl]-N-methylcyclohexane-1-carboxamide	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)C3CCC(N4CCN(C5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)CC4)CC3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C49H56F3N9O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-N5IX86	SCHEMBL28863625	N-[[1-[[4-[[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxymethyl]cyclopropyl]methyl]-5-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperazin-1-yl]-N-methylpentanamide	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CCCCN3CCN(C4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C47H54F3N9O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-133SKS	SCHEMBL28863628	N-[[1-[[4-[[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxymethyl]cyclopropyl]methyl]-4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperazin-1-yl]-N-methylbutanamide	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CCCN3CCN(C4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C46H52F3N9O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-FIXKGY	SCHEMBL28863586	N-[[1-[[4-[[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxymethyl]cyclopropyl]methyl]-3-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperidin-4-yl]oxy-N-methylpropanamide	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CCOC3CCN(C4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C46H51F3N8O8	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-1TYQGD	SCHEMBL24677725	2-(2,6-dioxopiperidin-3-yl)-5-[[1-[[4-[[(1R)-1-[2-fluoro-3-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxymethyl]cyclopropyl]methylamino]isoindole-1,3-dione	COC1=CC2=C(C=C1OCC1(CNC3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC1)C(N[C@H](C)C1=CC=CC(C(F)(F)F)=C1F)=NC(C)=N2	C37H34F4N6O6	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-6JADWH	SCHEMBL24677954	N-[[1-[[4-[[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxymethyl]cyclopropyl]methyl]-2-[5-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-2-yl]-N-methylacetamide	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CN3CC4CN(C5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)CC4C3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C46H50F3N9O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-6DSQG2	WO2022188819A1_81	.	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CN3CCC4(CC3)CCN(C3=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C3)CC4)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C49H56F3N9O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-T2X9XZ	WO2022188819A1_82	.	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)COCCCCNC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C44H49F3N8O8	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-T2KR5Y	WO2022188819A1_83	.	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CCCCCCOC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C45H50F3N7O8	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-NSBNEZ	WO2022188819A1_84	.	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CCCCCCNC3=CC=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C45H51F3N8O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-JMVRAI	WO2022188819A1_85	.	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CCCCCCOC3=CC=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C45H50F3N7O8	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-ASGOIH	WO2022188819A1_86	.	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CCCCCCNC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3F)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C45H50F4N8O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-OMZ9E3	WO2022188819A1_87	.	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CCCCCCNC3=CC=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3F)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C45H50F4N8O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-CY4PAB	PD216669	N-[[1-[[4-[[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxymethyl]cyclopropyl]methyl]-7-[[2-(2,6-dioxopiperidin-3-yl)-7-fluoro-1,3-dioxoisoindol-4-yl]amino]-N-methylheptanamide	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CCCCCCNC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C(F)C=C3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C45H50F4N8O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-EF6BWP	WO2022188819A1_89	.	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CN3CCC4(CCN(C5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)CC4)C3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C48H54F3N9O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-RT1FFS	SCHEMBL24678179	4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]-N-[[1-[[4-[[(1R)-1-[2-fluoro-3-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxymethyl]cyclopropyl]methyl]-N-methylbutanamide	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CCCNC3=CC=CC4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC1)C(N[C@H](C)C1=CC=CC(C(F)(F)F)=C1F)=NC(C)=N2	C42H43F4N7O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-ZDHWSQ	WO2022188819A1_90	.	COC1=CC2=C(C=C1OCC(C)(C)CN(C)C(=O)CCOCCCNC1=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=CC=C1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C44H51F3N8O8	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-JZB0NZ	SCHEMBL28863618	N-[[1-[[4-[[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxymethyl]cyclopropyl]methyl]-8-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]-N-methyloct-7-ynamide	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CCCCCC#CC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C46H48F3N7O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-CDFL0D	SCHEMBL28863607	N-[[1-[[4-[[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxymethyl]cyclopropyl]methyl]-3-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]but-3-ynoxy]-N-methylpropanamide	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CCOCCC#CC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C45H46F3N7O8	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-BTZE31	WO2022188819A1_93	.	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)CCCCCCNC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=N3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C44H50F3N9O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-ZK9XSF	PD216671	N-[[1-[[4-[[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxymethyl]cyclopropyl]methyl]-1-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethyl]-N-methylpiperidine-4-carboxamide	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)C3CCN(CCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C46H52F3N9O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-K1KFGM	WO2022188819A1_95	.	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)C3CCN(C(=O)CNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C46H50F3N9O8	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-T8CMMF	SCHEMBL28863656	N-[[1-[[4-[[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxymethyl]cyclopropyl]methyl]-1-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]cyclohexyl]-N-methylpiperidine-4-carboxamide; SCHEMBL29922616; PD216673	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)C3CCN(C4CCC(NC5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)CC4)CC3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C50H58F3N9O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-2972LM	SCHEMBL24677858	N-[[1-[[4-[[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxymethyl]cyclopropyl]methyl]-1-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]azetidin-3-yl]-N-methylpiperidine-4-carboxamide	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)C3CCN(C4CN(C5CN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)C4)CC3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C50H57F3N10O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-54Y8D8	WO2022188819A1_98	.	COC1=CC2=C(C=C1OCC1(CN(C)C(=O)C3CCN(C4CN(C5CN(C6=CC=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)C4)CC3)CC1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C50H57F3N10O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-6XBKQ0	SCHEMBL29922131	4-[[7-[(3S)-3-[4-[[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]amino]-7-methoxy-2-methylquinazolin-6-yl]oxypyrrolidin-1-yl]-7-oxoheptyl]amino]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	COC1=CC2=C(C=C1O[C@H]1CCN(C(=O)CCCCCCNC3=CC=CC4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)C1)C(N[C@H](C)C1=CC(N)=CC(C(F)(F)F)=C1)=NC(C)=N2	C43H47F3N8O7	SOS1	Q07889	CRBN	WO-2022188819-A1
TPD-FLJQ8K	WO2022201162A1_R4VP	.	Cc1ncsc1-c1ccc(CNC(=O)C2CC(=O)CN2C(=O)C(NC(=O)CCC(=O)NCCCCOc2ccc(Oc3ccc(N(Cc4ccccc4)C(=O)CCl)cc3)cc2)C(C)(C)C)cc1	C51H57ClN6O8S	RNF4	P78317	VHL	WO-2022201162-A1
TPD-8KS6G0	SCHEMBL27081396	3-[6-[4-[[1-[4-(6-hydroxyspiro[3,4-dihydro-1H-naphthalene-2,1'-cyclopentane]-1-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2Cc3cc(N4CCN(CC5CCN(c6ccc(C7c8ccc(O)cc8CCC78CCCC8)cc6)CC5)CC4)ccc3C2=O)C(=O)N1	C43H51N5O4	ERα	P03372	CRBN	WO-2022206737-A1
TPD-7J8VOF	SCHEMBL27081314	3-[6-[4-[[1-[4-[(1R,2R)-2-(4,4-difluorocyclohexyl)-6-hydroxy-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30773576	O=C1CCC(N2Cc3cc(N4CCN(CC5CCN(c6ccc([C@@H]7c8ccc(O)cc8CC[C@@H]7C7CCC(F)(F)CC7)cc6)CC5)CC4)ccc3C2=O)C(=O)N1	C45H53F2N5O4	ERα	P03372	CRBN	WO-2022206737-A1
TPD-8IAD98	WO2022206737A1_11	.	CN1CCC(C2CCc3cc(O)ccc3C2c2ccc(N3CCC(CN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)CC3)cc2)CC1	C45H56N6O4	ERα	P03372	CRBN	WO-2022206737-A1
TPD-ZN68V5	SCHEMBL30773592	3-[6-[4-[[1-[3-fluoro-4-[(1S,2R)-6-hydroxy-2-(oxan-4-yl)-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2Cc3cc(N4CCN(CC5CCN(c6ccc([C@@H]7c8ccc(O)cc8CC[C@@H]7C7CCOCC7)c(F)c6)CC5)CC4)ccc3C2=O)C(=O)N1	C44H52FN5O5	ERα	P03372	CRBN	WO-2022206737-A1
TPD-1JDCQE	SCHEMBL30773562	3-[6-[4-[[1-[3-fluoro-4-[(1R,2S)-6-hydroxy-2-(oxan-4-yl)-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2Cc3cc(N4CCN(CC5CCN(c6ccc([C@H]7c8ccc(O)cc8CC[C@H]7C7CCOCC7)c(F)c6)CC5)CC4)ccc3C2=O)C(=O)N1	C44H52FN5O5	ERα	P03372	CRBN	WO-2022206737-A1
TPD-020FXK	SCHEMBL29965912	(3S)-3-[6-[4-[[1-[4-[(1R,2R)-2-cyclobutyl-6-hydroxy-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CC[C@H](N2Cc3cc(N4CCN(CC5CCN(c6ccc([C@@H]7c8ccc(O)cc8CC[C@@H]7C7CCC7)cc6)CC5)CC4)ccc3C2=O)C(=O)N1	C43H51N5O4	ERα	P03372	CRBN	WO-2022206737-A1
TPD-QN60PZ	SCHEMBL27081240	3-[6-[4-[[1-[4-[(1S,2S)-2-cyclobutyl-6-hydroxy-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL29965896	O=C1CCC(N2Cc3cc(N4CCN(CC5CCN(c6ccc([C@H]7c8ccc(O)cc8CC[C@H]7C7CCC7)cc6)CC5)CC4)ccc3C2=O)C(=O)N1	C43H51N5O4	ERα	P03372	CRBN	WO-2022206737-A1
TPD-T6H1ID	SCHEMBL29966789	3-[6-[4-[[1-[4-[(1R,2R)-2-cyclopentyl-6-hydroxy-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2Cc3cc(N4CCN(CC5CCN(c6ccc([C@@H]7c8ccc(O)cc8CC[C@@H]7C7CCCC7)cc6)CC5)CC4)ccc3C2=O)C(=O)N1	C44H53N5O4	ERα	P03372	CRBN	WO-2022206737-A1
TPD-UP2BTM	SCHEMBL29965880	3-[6-[4-[[1-[4-[(1S,2S)-2-cyclopentyl-6-hydroxy-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2Cc3cc(N4CCN(CC5CCN(c6ccc([C@H]7c8ccc(O)cc8CC[C@H]7C7CCCC7)cc6)CC5)CC4)ccc3C2=O)C(=O)N1	C44H53N5O4	ERα	P03372	CRBN	WO-2022206737-A1
TPD-PW7RFK	SCHEMBL29966323	3-[6-[4-[[1-[4-[(1R,2R)-2-cyclohexyl-6-hydroxy-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2Cc3cc(N4CCN(CC5CCN(c6ccc([C@@H]7c8ccc(O)cc8CC[C@@H]7C7CCCCC7)cc6)CC5)CC4)ccc3C2=O)C(=O)N1	C45H55N5O4	ERα	P03372	CRBN	WO-2022206737-A1
TPD-YAE3HA	WO2022206737A1_15-2	.	O=C1CCC(N2Cc3cc(N4C=CN(CC5CCN(c6ccc([C@H]7c8ccc(O)cc8CC[C@H]7C7CCCCC7)cc6)CC5)CC4)ccc3C2=O)C(=O)N1	C45H53N5O4	ERα	P03372	CRBN	WO-2022206737-A1
TPD-W324HF	WO2022206737A1_16	.	O=C1CCC(N2Cc3cc(N4CCN(CC5CCN(c6ccc(C7c8ccc(O)cc8CCC7C7CC7)cc6)CC5)CC4)ccc3C2=O)C(=O)N1	C42H49N5O4	ERα	P03372	CRBN	WO-2022206737-A1
TPD-P3W13M	WO2022206737A1_17-1	(3S)-3-[6-[4-[[1-[4-[(1R,2R)-2-cyclopropyl-6-hydroxy-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CC[C@H](N2Cc3cc(N4CCN(CC5CCN(c6ccc([C@@H]7c8ccc(O)cc8CC[C@@H]7C7CC7)cc6)CC5)CC4)ccc3C2=O)C(=O)N1	C42H49N5O4	ERα	P03372	CRBN	WO-2022206737-A1
TPD-5RH978	WO2022206737A1_17-2	(3S)-3-[6-[4-[[1-[4-[(1S,2S)-2-cyclopropyl-6-hydroxy-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CC[C@H](N2Cc3cc(N4CCN(CC5CCN(c6ccc([C@H]7c8ccc(O)cc8CC[C@H]7C7CC7)cc6)CC5)CC4)ccc3C2=O)C(=O)N1	C42H49N5O4	ERα	P03372	CRBN	WO-2022206737-A1
TPD-Q6NF0F	SCHEMBL29966492	(3S)-3-[6-[4-[[1-[4-[(1R,2R)-2-cyclobutyl-6-hydroxy-1,2,3,4-tetrahydronaphthalen-1-yl]-2-fluorophenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CC[C@H](N2Cc3cc(N4CCN(CC5CCN(c6ccc([C@@H]7c8ccc(O)cc8CC[C@@H]7C7CCC7)cc6F)CC5)CC4)ccc3C2=O)C(=O)N1	C43H50FN5O4	ERα	P03372	CRBN	WO-2022206737-A1
TPD-U0NHOI	WO2022206737A1_18-2	.	O=C1CC[C@H](N2Cc3cc(N4C=CN(CC5CCN(c6ccc([C@H]7c8ccc(O)cc8CC[C@H]7C7CCC7)cc6F)CC5)CC4)ccc3C2=O)C(=O)N1	C43H48FN5O4	ERα	P03372	CRBN	WO-2022206737-A1
TPD-YZV3P5	WO2022206737A1_19	.	O=C1CC[C@@H](N2Cc3cc(N4CCN(CC5CCN(c6ccc([C@@H]7c8ccc(O)cc8CC[C@@H]7C7CCCC7)cc6F)CC5)CC4)ccc3C2=O)C(=O)N1	C44H52FN5O4	ERα	P03372	CRBN	WO-2022206737-A1
TPD-MZDQ5G	SCHEMBL29093046	3-[6-[4-[[1-[4-[(1R)-6-hydroxyspiro[3,4-dihydro-1H-naphthalene-2,1'-cyclopentane]-1-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL29966958	O=C1CCC(N2Cc3cc(N4CCN(CC5CCN(c6ccc([C@@H]7c8ccc(O)cc8CCC78CCCC8)cc6)CC5)CC4)ccc3C2=O)C(=O)N1	C43H51N5O4	ERα	P03372	CRBN	WO-2022206737-A1
TPD-C7BKTD	WO2022206737A1_2-2	.	O=C1CCC(N2Cc3cc(N4C=CN(CC5CCN(c6ccc([C@H]7c8ccc(O)cc8CCC78CCCC8)cc6)CC5)CC4)ccc3C2=O)C(=O)N1	C43H49N5O4	ERα	P03372	CRBN	WO-2022206737-A1
TPD-0HOM0O	SCHEMBL27080986	(3S)-3-[6-[4-[[1-[4-[(1R,2R)-2-cyclohexyl-6-hydroxy-1,2,3,4-tetrahydronaphthalen-1-yl]-2-fluorophenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL29966984	O=C1CC[C@H](N2Cc3cc(N4CCN(CC5CCN(c6ccc([C@@H]7c8ccc(O)cc8CC[C@@H]7C7CCCCC7)cc6F)CC5)CC4)ccc3C2=O)C(=O)N1	C45H54FN5O4	ERα	P03372	CRBN	WO-2022206737-A1
TPD-SYRLZH	SCHEMBL27081116	(3S)-3-[6-[4-[[1-[4-[(1R,2R)-2-cyclopropyl-6-hydroxy-1,2,3,4-tetrahydronaphthalen-1-yl]-2-fluorophenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL29966745	O=C1CC[C@H](N2Cc3cc(N4CCN(CC5CCN(c6ccc([C@@H]7c8ccc(O)cc8CC[C@@H]7C7CC7)cc6F)CC5)CC4)ccc3C2=O)C(=O)N1	C42H48FN5O4	ERα	P03372	CRBN	WO-2022206737-A1
TPD-XO7A1S	SCHEMBL27081085	(3S)-3-[6-[4-[[1-[4-[(1R)-6-hydroxyspiro[3,4-dihydro-1H-naphthalene-2,4'-oxane]-1-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CC[C@H](N2Cc3cc(N4CCN(CC5CCN(c6ccc([C@@H]7c8ccc(O)cc8CCC78CCOCC8)cc6)CC5)CC4)ccc3C2=O)C(=O)N1	C43H51N5O5	ERα	P03372	CRBN	WO-2022206737-A1
TPD-F6HIEG	SCHEMBL29092612	3-[6-[4-[[1-[4-[(1R)-6-hydroxyspiro[3,4-dihydro-1H-naphthalene-2,1'-cyclobutane]-1-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL29965926	O=C1CCC(N2Cc3cc(N4CCN(CC5CCN(c6ccc([C@@H]7c8ccc(O)cc8CCC78CCC8)cc6)CC5)CC4)ccc3C2=O)C(=O)N1	C42H49N5O4	ERα	P03372	CRBN	WO-2022206737-A1
TPD-X4R25N	SCHEMBL29093050	3-[6-[4-[[1-[4-[(1S)-6-hydroxyspiro[3,4-dihydro-1H-naphthalene-2,1'-cyclobutane]-1-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL29966027	O=C1CCC(N2Cc3cc(N4CCN(CC5CCN(c6ccc([C@H]7c8ccc(O)cc8CCC78CCC8)cc6)CC5)CC4)ccc3C2=O)C(=O)N1	C42H49N5O4	ERα	P03372	CRBN	WO-2022206737-A1
TPD-HXK3RG	SCHEMBL27081154	(3S)-3-[6-[4-[[1-[4-[(1R,2R)-6-hydroxy-2-propan-2-yl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CC(C)[C@H]1CCc2cc(O)ccc2[C@H]1c1ccc(N2CCC(CN3CCN(c4ccc5c(c4)CN([C@H]4CCC(=O)NC4=O)C5=O)CC3)CC2)cc1	C42H51N5O4	ERα	P03372	CRBN	WO-2022206737-A1
TPD-48WYIP	SCHEMBL29966326	3-[6-[4-[[1-[4-[(1R)-6-hydroxy-2,2-dimethyl-3,4-dihydro-1H-naphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CC1(C)CCc2cc(O)ccc2[C@H]1c1ccc(N2CCC(CN3CCN(c4ccc5c(c4)CN(C4CCC(=O)NC4=O)C5=O)CC3)CC2)cc1	C41H49N5O4	ERα	P03372	CRBN	WO-2022206737-A1
TPD-6RRJ36	SCHEMBL30773591	3-[6-[4-[[1-[4-[(1S)-6-hydroxy-2,2-dimethyl-3,4-dihydro-1H-naphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CC1(C)CCc2cc(O)ccc2[C@@H]1c1ccc(N2CCC(CN3CCN(c4ccc5c(c4)CN(C4CCC(=O)NC4=O)C5=O)CC3)CC2)cc1	C41H49N5O4	ERα	P03372	CRBN	WO-2022206737-A1
TPD-FMKB82	orb2802200	(3S)-3-[6-[4-[[1-[4-[(1R,2R)-6-hydroxy-2-(2-methylpropyl)-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL27188723; 2846112-04-5	CC(C)C[C@H]1CCc2cc(O)ccc2[C@H]1c1ccc(N2CCC(CN3CCN(c4ccc5c(c4)CN([C@H]4CCC(=O)NC4=O)C5=O)CC3)CC2)cc1	C43H53N5O4	ERα	P03372	CRBN	WO-2022206737-A1
TPD-67BX9S	SCHEMBL29966524	(3S)-3-[6-[4-[[1-[4-[(1S,2S)-6-hydroxy-2-(2-methylpropyl)-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CC(C)C[C@@H]1CCc2cc(O)ccc2[C@@H]1c1ccc(N2CCC(CN3CCN(c4ccc5c(c4)CN([C@H]4CCC(=O)NC4=O)C5=O)CC3)CC2)cc1	C43H53N5O4	ERα	P03372	CRBN	WO-2022206737-A1
TPD-NY2G2V	WO2022206737A1_27	.	C[C@H]1CCc2cc(O)ccc2[C@H]1c1ccc(N2CCC(CN3C=CN(c4ccc5c(c4)CN([C@H]4CCC(=O)NC4=O)C5=O)CC3)CC2)cc1	C40H45N5O4	ERα	P03372	CRBN	WO-2022206737-A1
TPD-SCZT01	SCHEMBL27081321	(3S)-3-[6-[4-[[1-[4-[(1R,2S)-2-ethyl-6-hydroxy-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30768603	CC[C@H]1CCc2cc(O)ccc2[C@H]1c1ccc(N2CCC(CN3CCN(c4ccc5c(c4)CN([C@H]4CCC(=O)NC4=O)C5=O)CC3)CC2)cc1	C41H49N5O4	ERα	P03372	CRBN	WO-2022206737-A1
TPD-CWIC0Z	WO2022206737A1_29	.	CCC[C@H]1CCc2cc(O)ccc2C1c1ccc(N2CCC(CN3CCN(c4ccc5c(c4)CN([C@H]4CCC(=O)NC4=O)C5=O)CC3)CC2)cc1	C42H51N5O4	ERα	P03372	CRBN	WO-2022206737-A1
TPD-1W1LVR	WO2022206737A1_3	.	O=C1CCC(N2Cc3cc(N4CCN(CC5CCN(c6ccc(C7c8ccc(O)cc8CCC7C7CCOCC7)cc6F)CC5)CC4)ccc3C2=O)C(=O)N1	C44H52FN5O5	ERα	P03372	CRBN	WO-2022206737-A1
TPD-BBARKK	SCHEMBL27081236	(3S)-3-[6-[4-[[1-[4-[(1R,2R)-2-benzyl-6-hydroxy-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL29966544	O=C1CC[C@H](N2Cc3cc(N4CCN(CC5CCN(c6ccc([C@@H]7c8ccc(O)cc8CC[C@@H]7Cc7ccccc7)cc6)CC5)CC4)ccc3C2=O)C(=O)N1	C46H51N5O4	ERα	P03372	CRBN	WO-2022206737-A1
TPD-SHH80H	WO2022206737A1_31	.	Cc1cc([C@@H]2c3ccc(O)cc3OC[C@@H]2C2CCOCC2)ccc1N1CCC(CN2CCN(c3ccc4c(c3)CN([C@@H]3CCC(=O)NC3=O)C4=O)CC2)CC1	C44H53N5O6	ERα	P03372	CRBN	WO-2022206737-A1
TPD-DMO7SH	SCHEMBL27081552	(3S)-3-[6-[4-[[1-[4-[(3R,4R)-3-cyclobutyl-7-hydroxy-3,4-dihydro-2H-chromen-4-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CC[C@H](N2Cc3cc(N4CCN(CC5CCN(c6ccc([C@@H]7c8ccc(O)cc8OC[C@@H]7C7CCC7)cc6)CC5)CC4)ccc3C2=O)C(=O)N1	C42H49N5O5	ERα	P03372	CRBN	WO-2022206737-A1
TPD-XKLZJJ	SCHEMBL27081457	2-(2,6-dioxopiperidin-3-yl)-5-[4-[[1-[2-fluoro-4-[(1R,2R)-6-hydroxy-2-(oxan-4-yl)-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]isoindole-1,3-dione; SCHEMBL30773561	O=C1CCC(N2C(=O)c3ccc(N4CCN(CC5CCN(c6ccc([C@@H]7c8ccc(O)cc8CC[C@@H]7C7CCOCC7)cc6F)CC5)CC4)cc3C2=O)C(=O)N1	C44H50FN5O6	ERα	P03372	CRBN	WO-2022206737-A1
TPD-XC62LK	WO2022206737A1_34	.	O=C1CC[C@@H](N2Cc3cc(N4CCN(CC5CCN(c6ccc([C@@H]7c8ccc(O)cc8CC[C@@H]7CC7CC7)cc6)CC5)CC4)ccc3C2=O)C(=O)N1	C43H51N5O4	ERα	P03372	CRBN	WO-2022206737-A1
TPD-BFAZ5U	WO2022206737A1_35	.	O=C1CC[C@@H](N2Cc3cc(N4CCN(CC5CCN(c6ccc([C@@H]7c8ccc(O)cc8CC[C@@H]7CC7CCC7)cc6)CC5)CC4)ccc3C2=O)C(=O)N1	C44H53N5O4	ERα	P03372	CRBN	WO-2022206737-A1
TPD-B6NDDH	WO2022206737A1_36	.	O=C1CC[C@@H](N2Cc3cc(N4CCN(CC5CCN(c6ccc([C@@H]7c8ccc(O)cc8CCC78CCCC8)cc6F)CC5)CC4)ccc3C2=O)C(=O)N1	C43H50FN5O4	ERα	P03372	CRBN	WO-2022206737-A1
TPD-KR1WQ0	WO2022206737A1_37	.	CC(C)C[C@H]1CCc2cc(O)ccc2[C@H]1c1ccc(N2CCC(CN3CCN(c4ccc5c(c4)CN([C@@H]4CCC(=O)NC4=O)C5=O)CC3)CC2)c(F)c1	C43H52FN5O4	ERα	P03372	CRBN	WO-2022206737-A1
TPD-7E3VUJ	WO2022206737A1_38	.	CCC(CC)C[C@H]1CCc2cc(O)ccc2[C@H]1c1ccc(N2CCC(CN3CCN(c4ccc5c(c4)CN([C@@H]4CCC(=O)NC4=O)C5=O)CC3)CC2)cc1	C45H57N5O4	ERα	P03372	CRBN	WO-2022206737-A1
TPD-TJ7L1B	SCHEMBL27081378	(3S)-3-[6-[4-[[1-[4-[(1R,2R)-2-(2,2-dimethylpropyl)-6-hydroxy-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CC(C)(C)C[C@H]1CCc2cc(O)ccc2[C@H]1c1ccc(N2CCC(CN3CCN(c4ccc5c(c4)CN([C@H]4CCC(=O)NC4=O)C5=O)CC3)CC2)cc1	C44H55N5O4	ERα	P03372	CRBN	WO-2022206737-A1
TPD-3IBKF2	SCHEMBL29966615	3-[6-[4-[[1-[2-fluoro-4-[(1R,2R)-6-hydroxy-2-(oxan-4-yl)-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2Cc3cc(N4CCN(CC5CCN(c6ccc([C@@H]7c8ccc(O)cc8CC[C@@H]7C7CCOCC7)cc6F)CC5)CC4)ccc3C2=O)C(=O)N1	C44H52FN5O5	ERα	P03372	CRBN	WO-2022206737-A1
TPD-S8FHQV	SCHEMBL30773563	3-[6-[4-[[1-[2-fluoro-4-[(1S,2S)-6-hydroxy-2-(oxan-4-yl)-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2Cc3cc(N4CCN(CC5CCN(c6ccc([C@H]7c8ccc(O)cc8CC[C@H]7C7CCOCC7)cc6F)CC5)CC4)ccc3C2=O)C(=O)N1	C44H52FN5O5	ERα	P03372	CRBN	WO-2022206737-A1
TPD-FDRYH1	WO2022206737A1_40	.	CC(C)CC[C@H]1CCc2cc(O)ccc2[C@H]1c1ccc(N2CCC(CN3CCN(c4ccc5c(c4)CN([C@@H]4CCC(=O)NC4=O)C5=O)CC3)CC2)cc1	C44H55N5O4	ERα	P03372	CRBN	WO-2022206737-A1
TPD-905Y6C	SCHEMBL27081158	3-[6-[4-[[1-[4-[(1R,2R)-6-hydroxy-2-(2-methylpropyl)-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CC(C)C[C@H]1CCc2cc(O)ccc2[C@H]1c1ccc(N2CCC(CN3CCN(c4ccc5c(c4)CN(C4CCC(=O)NC4=O)C5=O)CC3)CC2)cc1	C43H53N5O4	ERα	P03372	CRBN	WO-2022206737-A1
TPD-1RC6G6	SCHEMBL27081194	(3R)-3-[6-[4-[[1-[4-[(1R,2R)-6-hydroxy-2-(2-methylpropyl)-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CC(C)C[C@H]1CCc2cc(O)ccc2[C@H]1c1ccc(N2CCC(CN3CCN(c4ccc5c(c4)CN([C@@H]4CCC(=O)NC4=O)C5=O)CC3)CC2)cc1	C43H53N5O4	ERα	P03372	CRBN	WO-2022206737-A1
TPD-AZ8V24	SCHEMBL27081290	(3R)-3-[6-[4-[[1-[2-fluoro-4-[(1R,2R)-6-hydroxy-2-(oxan-4-yl)-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL29966485	O=C1CC[C@@H](N2Cc3cc(N4CCN(CC5CCN(c6ccc([C@@H]7c8ccc(O)cc8CC[C@@H]7C7CCOCC7)cc6F)CC5)CC4)ccc3C2=O)C(=O)N1	C44H52FN5O5	ERα	P03372	CRBN	WO-2022206737-A1
TPD-PDDXMB	SCHEMBL27080998	(3S)-3-[6-[4-[[1-[2-fluoro-4-[(1R,2R)-6-hydroxy-2-(oxan-4-yl)-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL29966604	O=C1CC[C@H](N2Cc3cc(N4CCN(CC5CCN(c6ccc([C@@H]7c8ccc(O)cc8CC[C@@H]7C7CCOCC7)cc6F)CC5)CC4)ccc3C2=O)C(=O)N1	C44H52FN5O5	ERα	P03372	CRBN	WO-2022206737-A1
TPD-GRSFRM	SCHEMBL27081054	3-[2-[4-[[1-[4-[(1R)-6-hydroxyspiro[3,4-dihydro-1H-naphthalene-2,1'-cyclopentane]-1-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-5-oxo-7H-pyrrolo[3,4-b]pyridin-6-yl]piperidine-2,6-dione	O=C1CCC(N2Cc3nc(N4CCN(CC5CCN(c6ccc([C@@H]7c8ccc(O)cc8CCC78CCCC8)cc6)CC5)CC4)ccc3C2=O)C(=O)N1	C42H50N6O4	ERα	P03372	CRBN	WO-2022206737-A1
TPD-RUN2N4	WO2022206737A1_7	.	O=C1CCC(N2Cc3cc(N4CCN(CC5CCN(c6ccc(C7c8ccc(O)cc8CCC7C7CCOCC7)cc6)CC5)CC4)ccc3C2=O)C(=O)N1	C44H53N5O5	ERα	P03372	CRBN	WO-2022206737-A1
TPD-CTN5JX	SCHEMBL30773572	3-[6-[4-[[1-[4-[(1R,2R)-6-hydroxy-2-(oxan-4-yl)-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2Cc3cc(N4CCN(CC5CCN(c6ccc([C@@H]7c8ccc(O)cc8CC[C@@H]7C7CCOCC7)cc6)CC5)CC4)ccc3C2=O)C(=O)N1	C44H53N5O5	ERα	P03372	CRBN	WO-2022206737-A1
TPD-GASAZM	SCHEMBL30773579	3-[6-[4-[[1-[4-[(1S,2S)-6-hydroxy-2-(oxan-4-yl)-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30773580	O=C1CCC(N2Cc3cc(N4CCN(CC5CCN(c6ccc([C@H]7c8ccc(O)cc8CC[C@H]7C7CCOCC7)cc6)CC5)CC4)ccc3C2=O)C(=O)N1	C44H53N5O5	ERα	P03372	CRBN	WO-2022206737-A1
TPD-Y01UK5	WO2022206737A1_9	.	O=C1CCC(N2Cc3cc(N4CCN(CC5CCN(c6ccc(C7c8ccc(O)cc8CCC7C7CCC(F)(F)CC7)cc6)CC5)CC4)ccc3C2=O)C(=O)N1	C45H53F2N5O4	ERα	P03372	CRBN	WO-2022206737-A1
TPD-EJ6CYL	SCHEMBL25342345	5-[4-[[(3S)-4-[6-[[5-[2-(4,4-dimethyl-9-oxo-1,10-diazatricyclo[6.4.0.02,6]dodeca-2(6),7-dien-10-yl)-3-(hydroxymethyl)pyridin-4-yl]-1-methyl-2-oxopyridin-3-yl]amino]pyridin-3-yl]-3-methylpiperazin-1-yl]methyl]piperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	C[C@H]1CN(CC2CCN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)CCN1c1ccc(Nc2cc(-c3ccnc(N4CCn5c(cc6c5CC(C)(C)C6)C4=O)c3CO)cn(C)c2=O)nc1	C53H59N11O7	BTK	Q06187	CRBN	WO-2022206924-A1
TPD-3SO2BR	WO2022206924A1_2	.	Cn1cc(-c2ccnc(N3CCn4c(cc5c4CC(C)(C)C5)C3=O)c2CO)cc(Nc2ccc(C3CCN(CC4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)cn2)c1=O	C53H58N10O7	BTK	Q06187	CRBN	WO-2022206924-A1
TPD-8U99RT	WO2022206924A1_3	.	C[C@H]1CN(CC2CCN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)CCN1c1ccc(Nc2cc(-c3ccnc(N4CCn5c(cc6c5CC(C)(C)C6)C4=O)c3CO)cn(C)c2=O)nc1	C52H57N11O7	BTK	Q06187	CRBN	WO-2022206924-A1
TPD-2K8JE6	WO2022206924A1_4	.	C[C@H]1CN(CCC2CCN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)CCN1c1ccc(Nc2cc(-c3ccnc(N4CCn5c(cc6c5CC(C)(C)C6)C4=O)c3CO)cn(C)c2=O)nc1	C54H61N11O7	BTK	Q06187	CRBN	WO-2022206924-A1
TPD-5HGR7P	WO2022206924A1_5	.	C[C@H]1CN(CC2CCN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4)CC2)CCN1c1ccc(Nc2cc(-c3ccnc(N4CCn5c(cc6c5CC(C)(C)C6)C4=O)c3CO)cn(C)c2=O)nc1	C53H61N11O6	BTK	Q06187	CRBN	WO-2022206924-A1
TPD-NS5P5F	SCHEMBL27095755	5-[3-[(3S)-4-[6-[[5-[2-(4,4-dimethyl-9-oxo-1,10-diazatricyclo[6.4.0.02,6]dodeca-2(6),7-dien-10-yl)-3-(hydroxymethyl)pyridin-4-yl]-1-methyl-2-oxopyridin-3-yl]amino]pyridin-3-yl]-3-methylpiperazin-1-yl]azetidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	C[C@H]1CN(C2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)CCN1c1ccc(Nc2cc(-c3ccnc(N4CCn5c(cc6c5CC(C)(C)C6)C4=O)c3CO)cn(C)c2=O)nc1	C50H53N11O7	BTK	Q06187	CRBN	WO-2022206924-A1
TPD-P32ZJE	WO2022206924A1_7	.	C[C@H]1CN(C2CN(CC3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)C2)CCN1c1ccc(Nc2cc(-c3ccnc(N4CCn5c(cc6c5CC(C)(C)C6)C4=O)c3CO)cn(C)c2=O)nc1	C56H64N12O7	BTK	Q06187	CRBN	WO-2022206924-A1
TPD-BN4TJS	WO2022206924A1_8	.	C=C1c2cc3c(n2CCN1c1nccc(-c2cc(Nc4ccc(N5CCC6(CC5)CCN(c5ccc7c(c5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC6)cn4)c(=O)n(C)c2)c1CO)CC(C)(C)C3	C52H56N10O6	BTK	Q06187	CRBN	WO-2022206924-A1
TPD-WD3OQQ	WO2022206924A1_9	.	C[C@H]1CN(C2CN(C3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)C2)CCN1c1ccc(Nc2cc(-c3ccnc(N4CCn5c(cc6c5CC(C)(C)C6)C4=O)c3CO)cn(C)c2=O)nc1	C55H62N12O7	BTK	Q06187	CRBN	WO-2022206924-A1
TPD-JWI5PV	WO2022206924A1_12	.	Cn1cc(-c2ccnc(N3CCn4c(cc5c4CC(C)(C)C5)C3=O)c2CO)cc(Nc2ccc(N3CC4(CN(CC5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)C3)cn2)c1=O	C53H57N11O7	BTK	Q06187	CRBN	WO-2022206924-A1
TPD-J4W73J	WO2022206924A1_13	.	COc1ccc(C(=O)N2CCC(CN3CCC(CN4CCN(c5ccc(Nc6cc(-c7ccnc(N8CCn9c(cc%10c9CC(C)(C)C%10)C8=O)c7CO)cn(C)c6=O)nc5)[C@@H](C)C4)CC3)CC2)cc1N1CCC(=O)NC1=O	C58H72N12O7	BTK	Q06187	CRBN	WO-2022206924-A1
TPD-976DCK	WO2022206924A1_14	.	COc1ccc(C(=O)N2CCC3(CCN(CCN4CCN(c5ccc(Nc6cc(-c7ccnc(N8CCn9c(cc%10c9CC(C)(C)C%10)C8=O)c7CO)cn(C)c6=O)nc5)[C@@H](C)C4)CC3)CC2)cc1N1CCC(=O)NC1=O	C57H70N12O7	BTK	Q06187	CRBN	WO-2022206924-A1
TPD-8CC6VV	WO2022206924A1_15	.	Cc1ccc(C(=O)N2CCC3(CCN(CCN4CCN(c5ccc(Nc6cc(-c7ccnc(N8CCn9c(cc%10c9CC(C)(C)C%10)C8=O)c7CO)cn(C)c6=O)nc5)[C@@H](C)C4)CC3)CC2)cc1N1CCC(=O)NC1=O	C57H70N12O6	BTK	Q06187	CRBN	WO-2022206924-A1
TPD-IBOYQ2	WO2022206924A1_16	.	Cn1cc(-c2ccnc(N3CCn4c(cc5c4CC(C)(C)C5)C3=O)c2CO)cc(Nc2ccc(N3CCN(CC4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C4(CC4)C3)cn2)c1=O	C54H59N11O7	BTK	Q06187	CRBN	WO-2022206924-A1
TPD-5PVOAK	WO2022206924A1_17	.	Cn1cc(-c2ccnc(N3CCn4c(cc5c4CC(C)(C)C5)C3=O)c2CO)cc(Nc2ccc(N3CCN(CC4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC34CC4)cn2)c1=O	C54H59N11O7	BTK	Q06187	CRBN	WO-2022206924-A1
TPD-8A9I79	WO2022206924A1_18	.	CC1Cc2cc3n(c2C1)CCN(c1nccc(-c2cc(Nc4ccc(N5CCC6(CCCN(c7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)C6)CC5)cn4)c(=O)n(C)c2)c1CO)C3=O	C50H52N10O7	BTK	Q06187	CRBN	WO-2022206924-A1
TPD-57CR3R	WO2022206924A1_19	.	C[C@H]1CN(C2CCCN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)CCN1c1ccc(Nc2cc(-c3ccnc(N4CCn5c(cc6c5CC(C)(C)C6)C4=O)c3CO)cn(C)c2=O)nc1	C52H57N11O7	BTK	Q06187	CRBN	WO-2022206924-A1
TPD-JP4TOF	SCHEMBL27095666	5-[4-[(3S)-4-[6-[[5-[2-(4,4-dimethyl-9-oxo-1,10-diazatricyclo[6.4.0.02,6]dodeca-2(6),7-dien-10-yl)-3-(hydroxymethyl)pyridin-4-yl]-1-methyl-2-oxopyridin-3-yl]amino]pyridin-3-yl]-3-methylpiperazin-1-yl]piperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	C[C@H]1CN(C2CCN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)CCN1c1ccc(Nc2cc(-c3ccnc(N4CCn5c(cc6c5CC(C)(C)C6)C4=O)c3CO)cn(C)c2=O)nc1	C52H57N11O7	BTK	Q06187	CRBN	WO-2022206924-A1
TPD-ZAG8AO	WO2022228421A1_1	.	Cn1cc(-c2sc(C(C)(C)O)cc2N2CCc3ccccc32)c2c(c1=O)NC(C(=O)NCCCCC(=O)Nc1cccc3c1CN(C1CCC(=O)NC1=O)C3=O)O2	C41H43N7O8S	BRD4	O60885	CRBN	WO-2022228421-A1
TPD-WE6DPI	WO2022228421A1_2	.	Cn1cc(-c2sc(C(C)(C)O)cc2N2CCc3ccccc32)c2cc(C(=O)NCCCC(=O)Nc3cccc4c3CN(C3CCC(=O)NC3=O)C4=O)[nH]c2c1=O	C41H41N7O7S	BRD4	O60885	CRBN	WO-2022228421-A1
TPD-ODU4P4	WO2022228421A1_3	.	Cn1cc(-c2sc(C(C)(C)O)cc2N2CCc3ccccc32)c2cc(C(=O)NCCC(=O)Nc3cccc4c3CN(C3CCC(=O)NC3=O)C4=O)[nH]c2c1=O	C40H39N7O7S	BRD4	O60885	CRBN	WO-2022228421-A1
TPD-ZF2K0A	WO2022228421A1_4	.	Cn1cc(-c2sc(C(C)(C)O)cc2N2CCc3ccccc32)c2cc(C(=O)NCCOCCC(=O)Nc3cccc4c3CN(C3CCC(=O)NC3=O)C4=O)[nH]c2c1=O	C42H43N7O8S	BRD4	O60885	CRBN	WO-2022228421-A1
TPD-T60O6M	WO2022228421A1_5	.	Cn1cc(-c2sc(C(C)(C)O)cc2N2CCc3ccccc32)c2cc(C(=O)NCCOCCOCC(=O)Nc3cccc4c3CN(C3CCC(=O)NC3=O)C4=O)[nH]c2c1=O	C43H45N7O9S	BRD4	O60885	CRBN	WO-2022228421-A1
TPD-699PRT	WO2022228421A1_6	.	Cn1cc(-c2sc(C(C)(C)O)cc2N2CCc3ccccc32)c2cc(C(=O)NCCCC(=O)Nc3ccc4c(c3)CN(C3CCC(=O)NC3=O)C4=O)[nH]c2c1=O	C41H41N7O7S	BRD4	O60885	CRBN	WO-2022228421-A1
TPD-0G4YN9	WO2022228421A1_7	.	Cn1cc(-c2sc(C(C)(C)O)cc2N2CCC3C=CC=CC32)c2cc(C(=O)NCCC(=O)Nc3ccc4c(c3)CN(C3CCC(=O)NC3=O)C4=O)[nH]c2c1=O	C40H41N7O7S	BRD4	O60885	CRBN	WO-2022228421-A1
TPD-I6TBY3	WO2022228421A1_8	.	Cn1cc(-c2sc(C(C)(C)O)cc2N2CCc3ccccc32)c2cc(C(=O)NCCOCCC(=O)Nc3ccc4c(c3)CN(C3CCC(=O)NC3=O)C4=O)[nH]c2c1=O	C42H43N7O8S	BRD4	O60885	CRBN	WO-2022228421-A1
TPD-DK16EI	WO2022228421A1_9	.	Cn1cc(-c2sc(C(C)(C)O)cc2N2CCc3ccccc32)c2cc(C(=O)NCCOCCOCC(=O)Nc3ccc4c(c3)CN(C3CCC(=O)NC3=O)C4=O)[nH]c2c1=O	C43H45N7O9S	BRD4	O60885	CRBN	WO-2022228421-A1
TPD-7QI4BY	WO2022228421A1_10	.	Cn1cc(-c2sc(C(C)(C)O)cc2N2CCc3ccccc32)c2cc(C(=O)NCCCCNc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)[nH]c2c1=O	C41H41N7O7S	BRD4	O60885	CRBN	WO-2022228421-A1
TPD-H4H7GS	WO2022228421A1_11	.	Cn1cc(-c2sc(C(C)(C)O)cc2N2CCc3ccccc32)c2cc(C(=O)NCCCCCNC(=O)COc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)[nH]c2c1=O	C44H45N7O9S	BRD4	O60885	CRBN	WO-2022228421-A1
TPD-FU40EK	WO2022228421A1_12	.	Cn1cc(-c2sc(C(C)(C)O)cc2N2CCc3ccccc32)c2cc(C(=O)NCCOCCNC(=O)COc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)[nH]c2c1=O	C43H43N7O10S	BRD4	O60885	CRBN	WO-2022228421-A1
TPD-TAMI0U	WO2022228421A1_13	.	Cn1cc(-c2sc(C(C)(C)O)cc2N2CCc3ccccc32)c2cc(C(=O)NCCCCCCNC(=O)COc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)[nH]c2c1=O	C45H47N7O9S	BRD4	O60885	CRBN	WO-2022228421-A1
TPD-WTEDJY	WO2022228421A1_14	.	Cn1cc(-c2sc(C(C)(C)O)cc2N2CCc3ccccc32)c2cc(C(=O)Nc3ccc(OCCOCCOCCOCCNc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)cc3)[nH]c2c1=O	C51H53N7O11S	BRD4	O60885	CRBN	WO-2022228421-A1
TPD-GEGJKF	WO2022228421A1_15	.	Cn1cc(-c2sc(C(C)(C)O)cc2N2CCc3ccccc32)c2cc(C(=O)NCCOCCNc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)[nH]c2c1=O	C41H41N7O8S	BRD4	O60885	CRBN	WO-2022228421-A1
TPD-38ZHLN	WO2022228421A1_16	.	Cn1cc(-c2sc(C(C)(C)O)cc2N2CCc3ccccc32)c2cc(C(=O)NCCCCCCOc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)[nH]c2c1=O	C43H44N6O8S	BRD4	O60885	CRBN	WO-2022228421-A1
TPD-OJHL8S	WO2022228421A1_17	.	Cn1cc(-c2sc(C(C)(C)O)cc2N2CCc3ccccc32)c2cc(C(=O)NCCCCCNc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)[nH]c2c1=O	C42H43N7O7S	BRD4	O60885	CRBN	WO-2022228421-A1
TPD-8R8VU7	WO2022235220A1_A	.	Cc1sc2c(c1C)C(c1ccc(Cl)cc1)=N[C@@H](CC(=O)Oc1ccc3sc(C4=NC(C(=O)Nc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6=O)CS4)nc3c1)c1nnc(C)n1-2	C43H32ClN9O7S3	BRD4	O60885	CRBN	WO-2022235220-A1
TPD-RPW7BI	WO2022235220A1_B	.	Cc1sc2c(c1C)C(c1ccc(Cl)cc1)=N[C@@H](CC(=O)NCCCNc1ccc3nc(C4=NC(C(=O)NCCCNc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6=O)CS4)sc3c1)c1nnc(C)n1-2	C49H47ClN12O6S3	BRD4	O60885	CRBN	WO-2022235220-A1
TPD-84MU5I	SCHEMBL29315716	[2-[4-[3-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]propylcarbamoyl]-2,5-dihydro-1,3-thiazol-2-yl]-1,3-benzothiazol-6-yl] 2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetate	Cc1sc2c(c1C)C(c1ccc(Cl)cc1)=N[C@@H](CC(=O)Oc1ccc3nc(C4N=C(C(=O)NCCCNc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6=O)CS4)sc3c1)c1nnc(C)n1-2	C46H39ClN10O7S3	BRD4	O60885	CRBN	WO-2022235220-A1
TPD-JGRYBF	SCHEMBL29317293	[2-[4-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]-2-oxoethoxy]ethoxy]ethylcarbamoyl]-2,5-dihydro-1,3-thiazol-2-yl]-1,3-benzothiazol-6-yl] 2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetate	Cc1sc2c(c1C)C(c1ccc(Cl)cc1)=N[C@@H](CC(=O)Oc1ccc3nc(C4N=C(C(=O)NCCOCCOCC(=O)Nc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6=O)CS4)sc3c1)c1nnc(C)n1-2	C49H43ClN10O10S3	BRD4	O60885	CRBN	WO-2022235220-A1
TPD-DSJ6G5	WO2022235220A1_T208	.	Cc1sc2c(c1C)C(c1ccc(Cl)cc1)=N[C@@H](CC(=O)NCCCOc1ccc3nc(C4=NC(C(=O)NCCOCCOCC(=O)Nc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6=O)CS4)sc3c1)c1nnc(C)n1-2	C52H50ClN11O10S3	BRD4	O60885	CRBN	WO-2022235220-A1
TPD-4BIYFI	WO2022235220A1_T44	.	COc1cc(/C=N/n2c(SC)nnc2-c2ccc(OCCOCCOCCOCc3cn(CCOCC(=O)Nc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)nn3)cc2)c(Br)cc1O	C43H45BrN10O12S	BRD4	O60885	CRBN	WO-2022235220-A1
TPD-1GTFT6	WO2022242725A1_1	.	COc1cc(N2CCC(N3CCN(CC#Cc4cccc5c4CN(C4CCC(=O)NC4=O)C5=O)CC3)CC2)ccc1Nc1ncc(Cl)c(Nc2ccccc2P(C)(C)=O)n1	C44H49ClN9O5P	ALK;ROS1;EGFR	Q9UM73/P08922/P00533	CRBN	WO-2022242725-A1
TPD-DWSPD9	HJM-561	3-[7-[4-[4-[1-[4-[[5-chloro-4-(2-dimethylphosphorylanilino)pyrimidin-2-yl]amino]-3-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]but-1-ynyl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; 2570251-68-0; orb1942573; CHEMBL5284115; SCHEMBL23066080; AT42456; DA-54027; HY-156698; CS-0889810	COc1cc(N2CCC(N3CCN(CCC#Cc4cccc5c4CN(C4CCC(=O)NC4=O)C5=O)CC3)CC2)ccc1Nc1ncc(Cl)c(Nc2ccccc2P(C)(C)=O)n1	C45H51ClN9O5P	ALK;ROS1;EGFR	Q9UM73/P08922/P00533	CRBN	WO-2022242725-A1
TPD-Y8IEO4	WO2022242725A1_3	3-[7-[3-[4-[1-[4-[[5-chloro-4-(2-dimethylphosphorylanilino)pyrimidin-2-yl]amino]-3-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]propyl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	COc1cc(N2CCC(N3CCN(CCCc4cccc5c4CN(C4CCC(=O)NC4=O)C5=O)CC3)CC2)ccc1Nc1ncc(Cl)c(Nc2ccccc2P(C)(C)=O)n1	C44H53ClN9O5P	ALK;ROS1;EGFR	Q9UM73/P08922/P00533	CRBN	WO-2022242725-A1
TPD-X4E0WD	SCHEMBL23044789	3-[7-[6-[4-[1-[4-[[5-chloro-4-(2-dimethylphosphorylanilino)pyrimidin-2-yl]amino]-3-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]hexyl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	COc1cc(N2CCC(N3CCN(CCCCCCc4cccc5c4CN(C4CCC(=O)NC4=O)C5=O)CC3)CC2)ccc1Nc1ncc(Cl)c(Nc2ccccc2P(C)(C)=O)n1	C47H59ClN9O5P	ALK;ROS1;EGFR	Q9UM73/P08922/P00533	CRBN	WO-2022242725-A1
TPD-D4JSFC	SCHEMBL23066105	3-[7-[7-[4-[1-[4-[[5-chloro-4-(2-dimethylphosphorylanilino)pyrimidin-2-yl]amino]-3-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]heptyl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	COc1cc(N2CCC(N3CCN(CCCCCCCc4cccc5c4CN(C4CCC(=O)NC4=O)C5=O)CC3)CC2)ccc1Nc1ncc(Cl)c(Nc2ccccc2P(C)(C)=O)n1	C48H61ClN9O5P	ALK;ROS1;EGFR	Q9UM73/P08922/P00533	CRBN	WO-2022242725-A1
TPD-ERKCDC	WO2022242725A1_6	.	COc1cc(N2CCC(N3CCN(Cc4ccc(C#Cc5cccc6c5CN(C5CCC(=O)NC5=O)C6=O)cc4)CC3)CC2)ccc1Nc1ncc(Cl)c(Nc2ccccc2P(C)(C)=O)n1	C50H53ClN9O5P	ALK;ROS1;EGFR	Q9UM73/P08922/P00533	CRBN	WO-2022242725-A1
TPD-FB7GRJ	WO2022242725A1_7	.	COc1cc(N2CCC(N3CCN(CCC/C=C\c4cccc5c4CN(C4CCC(=O)NC4=O)C5=O)CC3)CC2)ccc1Nc1ncc(Cl)c(Nc2ccccc2P(C)(C)=O)n1	C46H55ClN9O5P	ALK;ROS1;EGFR	Q9UM73/P08922/P00533	CRBN	WO-2022242725-A1
TPD-QQM5I1	WO2022242725A1_8	.	COc1cc(N2CCC(N3CCN(CCN(C)c4cccc5c4CN(C4CCC(=O)NC4=O)C5=O)CC3)CC2)ccc1Nc1ncc(Cl)c(Nc2ccccc2P(C)(C)=O)n1	C44H54ClN10O5P	ALK;ROS1;EGFR	Q9UM73/P08922/P00533	CRBN	WO-2022242725-A1
TPD-RBAKLQ	WO2022242725A1_9	.	COc1cc(N2CCC(N3CCN(CCCC#Cc4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5)CC3)CC2)ccc1Nc1ncc(Cl)c(Nc2ccccc2P(C)(C)=O)n1	C46H53ClN9O5P	ALK;ROS1;EGFR	Q9UM73/P08922/P00533	CRBN	WO-2022242725-A1
TPD-WSW8DY	WO2022242725A1_10	.	COc1cc(N2CCC(N3CCN(CCCCNc4cccc5c4CN(C4CCC(=O)NC4=O)C5=O)CC3)CC2)ccc1Nc1ncc(Cl)c(Nc2ccccc2P(C)(C)=O)n1	C45H56ClN10O5P	ALK;ROS1;EGFR	Q9UM73/P08922/P00533	CRBN	WO-2022242725-A1
TPD-PDA243	WO2022242725A1_11	.	COc1cc(N2CCC(N3CCN(CCCCCCCCCC(=O)N[C@H](C(=O)N4C[C@@H](O)C[C@H]4C(=O)NCc4ccc(-c5scnc5C)cc4)C(C)(C)C)CC3)CC2)ccc1Nc1ncc(Cl)c(Nc2ccccc2P(C)(C)=O)n1	C60H83ClN11O6PS	ALK;ROS1;EGFR	Q9UM73/P08922/P00533	VHL	WO-2022242725-A1
TPD-Z04F6B	WO2022242725A1_12	.	COc1cc(N2CCC(N3CCN(CCC/C=C/c4cccc5c4CN(C4CCC(=O)NC4=O)C5=O)CC3)CC2)ccc1Nc1ncc(Cl)c(Nc2ccccc2P(C)(C)=O)n1	C46H55ClN9O5P	ALK;ROS1;EGFR	Q9UM73/P08922/P00533	CRBN	WO-2022242725-A1
TPD-CUKMC5	WO2022242725A1_13	.	COc1cc(N2CCC(N3CCN(CCOc4cccc5c4CN(C4CCC(=O)NC4=O)C5=O)CC3)CC2)ccc1Nc1ncc(Cl)c(Nc2ccccc2P(C)(C)=O)n1	C43H51ClN9O6P	ALK;ROS1;EGFR	Q9UM73/P08922/P00533	CRBN	WO-2022242725-A1
TPD-B3KVOP	SCHEMBL22974006	3-[7-[4-[4-[1-[4-[[5-chloro-4-(2-dimethylphosphorylanilino)pyrimidin-2-yl]amino]-3-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]butylsulfanyl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	COc1cc(N2CCC(N3CCN(CCCCSc4cccc5c4CN(C4CCC(=O)NC4=O)C5=O)CC3)CC2)ccc1Nc1ncc(Cl)c(Nc2ccccc2P(C)(C)=O)n1	C45H55ClN9O5PS	ALK;ROS1;EGFR	Q9UM73/P08922/P00533	CRBN	WO-2022242725-A1
TPD-0UZEDS	WO2022242725A1_15	.	COc1cc(N2CCC(N3CCN(CCCCCSc4cccc5c4CN(C4CCC(=O)NC4=O)C5=O)CC3)CC2)ccc1Nc1ncc(Cl)c(Nc2ccccc2P(C)(C)=O)n1	C46H57ClN9O5PS	ALK;ROS1;EGFR	Q9UM73/P08922/P00533	CRBN	WO-2022242725-A1
TPD-8GCQ3Z	WO2022242725A1_16	.	COc1cc(N2CCC(N3CCN(C/C=C\c4cccc5c4CN(C4CCC(=O)NC4=O)C5=O)CC3)CC2)ccc1Nc1ncc(Cl)c(Nc2ccccc2P(C)(C)=O)n1	C44H51ClN9O5P	ALK;ROS1;EGFR	Q9UM73/P08922/P00533	CRBN	WO-2022242725-A1
TPD-71ZQHK	WO2022242725A1_17	.	COc1cc(N2CCC(N3CCN(CCCCS(=O)(=O)c4cccc5c4CN(C4CCC(=O)NC4=O)C5=O)CC3)CC2)ccc1Nc1ncc(Cl)c(Nc2ccccc2P(C)(C)=O)n1	C45H55ClN9O7PS	ALK;ROS1;EGFR	Q9UM73/P08922/P00533	CRBN	WO-2022242725-A1
TPD-M1PIS0	WO2022242725A1_18	.	COc1cc(N2CCC(N3CCN(CC/C=C\c4cccc5c4CN(C4CCC(=O)NC4=O)C5=O)CC3)CC2)ccc1Nc1ncc(Cl)c(Nc2ccccc2P(C)(C)=O)n1	C45H53ClN9O5P	ALK;ROS1;EGFR	Q9UM73/P08922/P00533	CRBN	WO-2022242725-A1
TPD-DCW6A4	WO2022242725A1_19	.	CCc1cc2c(cc1N1CCC(N3CCN(CCCCOc4cccc5c4CN(C4CCC(=O)NC4=O)C5=O)CC3)CC1)C(C)(C)c1[nH]c3cc(C#N)ccc3c1C2=O	C47H53N7O5	ALK;ROS1;EGFR	Q9UM73/P08922/P00533	CRBN	WO-2022242725-A1
TPD-64OPTL	WO2022242725A1_20	.	COc1cc(N2CCC(N3CCN(S(=O)(=O)CC/C=C/c4cccc5c4CN(C4CCC(=O)NC4=O)C5=O)CC3)CC2)ccc1Nc1ncc(Cl)c(Nc2ccccc2P(C)(C)=O)n1	C45H53ClN9O7PS	ALK;ROS1;EGFR	Q9UM73/P08922/P00533	CRBN	WO-2022242725-A1
TPD-VWA3ZA	WO2022242725A1_21	.	COc1cc(N2CCC(N(C)CCCCCOc3cccc4c3CN(C3CCC(=O)NC3=O)C4=O)CC2)ccc1Nc1ncc(Cl)c(Nc2ccccc2P(C)(C)=O)n1	C43H52ClN8O6P	ALK;ROS1;EGFR	Q9UM73/P08922/P00533	CRBN	WO-2022242725-A1
TPD-HHERC5	WO2022242725A1_22	.	COc1cc(N2CCC(N(C)CCCCOc3cccc4c3CN(C3CCC(=O)NC3=O)C4=O)CC2)ccc1Nc1ncc(Cl)c(Nc2ccccc2P(C)(C)=O)n1	C42H50ClN8O6P	ALK;ROS1;EGFR	Q9UM73/P08922/P00533	CRBN	WO-2022242725-A1
TPD-FPSUR3	WO2022242725A1_23	.	COc1cc(N2CCC(N(C)CCCCCCc3cccc4c3CN(C3CCC(=O)NC3=O)C4=O)CC2)ccc1Nc1ncc(Cl)c(Nc2ccccc2P(C)(C)=O)n1	C44H54ClN8O5P	ALK;ROS1;EGFR	Q9UM73/P08922/P00533	CRBN	WO-2022242725-A1
TPD-FRPFGM	WO2022242725A1_24	.	COc1cc(N2CCC(N3CCN(C/C=C/c4cccc5c4CN(C4CCC(=O)NC4=O)C5=O)CC3)CC2)ccc1Nc1ncc(Cl)c(Nc2ccccc2P(C)(C)=O)n1	C44H51ClN9O5P	ALK;ROS1;EGFR	Q9UM73/P08922/P00533	CRBN	WO-2022242725-A1
TPD-08H0UX	WO2022242725A1_25	.	COc1cc(N2CCC(N3CCN(C/C=C/CN(C)c4cccc5c4CN(C4CCC(=O)NC4=O)C5=O)CC3)CC2)ccc1Nc1ncc(Cl)c(Nc2ccccc2P(C)(C)=O)n1	C46H56ClN10O5P	ALK;ROS1;EGFR	Q9UM73/P08922/P00533	CRBN	WO-2022242725-A1
TPD-ZTU38Q	WO2022242725A1_26	.	COc1cc(N2CCC(N3CCN(CCCCN(C)c4cccc5c4CN(C4CCC(=O)NC4=O)C5=O)CC3)CC2)ccc1Nc1ncc(Cl)c(Nc2ccccc2P(C)(C)=O)n1	C46H58ClN10O5P	ALK;ROS1;EGFR	Q9UM73/P08922/P00533	CRBN	WO-2022242725-A1
TPD-98430N	WO2022242725A1_27	.	COc1cc(N2CCC(N(C)CCCCCCCc3cccc4c3CN(C3CCC(=O)NC3=O)C4=O)CC2)ccc1Nc1ncc(Cl)c(Nc2ccccc2P(C)(C)=O)n1	C45H56ClN8O5P	ALK;ROS1;EGFR	Q9UM73/P08922/P00533	CRBN	WO-2022242725-A1
TPD-B1NVJ9	WO2022242725A1_28	.	COc1cc(N2CCC(N(C)CCCCCCOc3cccc4c3CN(C3CCC(=O)NC3=O)C4=O)CC2)ccc1Nc1ncc(Cl)c(Nc2ccccc2P(C)(C)=O)n1	C44H54ClN8O6P	ALK;ROS1;EGFR	Q9UM73/P08922/P00533	CRBN	WO-2022242725-A1
TPD-64KCKI	WO2022242725A1_29	.	COc1cc(N2CCC(N3CCN(CCCCCCCCCCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)NCc4ccc(-c5scnc5C)cc4)C(C)(C)C)CC3)CC2)ccc1Nc1ncc(Cl)c(Nc2ccccc2P(C)(C)=O)n1	C61H85ClN11O6PS	ALK;ROS1;EGFR	Q9UM73/P08922/P00533	VHL	WO-2022242725-A1
TPD-263U1M	SCHEMBL24697205	4-[8-amino-3-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]oxy]ethoxy]ethoxy]ethyl]-2,7-diazaspiro[3.5]nonan-7-yl]imidazo[1,5-a]pyrazin-1-yl]-N-(4-chloropyridin-2-yl)-3-fluorobenzamide	NC1=NC=CN2C(N3CCC4(CC3)CN(CCOCCOCCOC3=CC=C5C(=O)N(C6CCC(=O)NC6=O)CC5=C3)C4)=NC(C3=C(F)C=C(C(=O)NC4=CC(Cl)=CC=N4)C=C3)=C12	C44H46ClFN10O7	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-M5O58Y	SCHEMBL24697397	4-[8-amino-3-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]oxy]ethyl]-2,7-diazaspiro[3.5]nonan-7-yl]imidazo[1,5-a]pyrazin-1-yl]-N-(4-chloropyridin-2-yl)-3-fluorobenzamide	NC1=NC=CN2C(N3CCC4(CC3)CN(CCOC3=CC=C5C(=O)N(C6CCC(=O)NC6=O)CC5=C3)C4)=NC(C3=C(F)C=C(C(=O)NC4=CC(Cl)=CC=N4)C=C3)=C12	C40H38ClFN10O5	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-JFEH3I	SCHEMBL24697227	4-[8-amino-3-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]ethyl]-2,7-diazaspiro[3.5]nonan-7-yl]imidazo[1,5-a]pyrazin-1-yl]-N-(4-chloropyridin-2-yl)-3-fluorobenzamide	NC1=NC=CN2C(N3CCC4(CC3)CN(CCC3=CC=C5C(=O)N(C6CCC(=O)NC6=O)CC5=C3)C4)=NC(C3=C(F)C=C(C(=O)NC4=CC(Cl)=CC=N4)C=C3)=C12	C40H38ClFN10O4	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-YTYEXZ	SCHEMBL24696567	4-[8-amino-3-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]methyl]-2,7-diazaspiro[3.5]nonan-7-yl]imidazo[1,5-a]pyrazin-1-yl]-N-(4-chloropyridin-2-yl)-3-fluorobenzamide	NC1=NC=CN2C(N3CCC4(CC3)CN(CC3=CC=C5C(=O)N(C6CCC(=O)NC6=O)CC5=C3)C4)=NC(C3=C(F)C=C(C(=O)NC4=CC(Cl)=CC=N4)C=C3)=C12	C39H36ClFN10O4	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-NKP4I2	SCHEMBL24696550	4-[8-amino-3-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-2,7-diazaspiro[3.5]nonan-7-yl]imidazo[1,5-a]pyrazin-1-yl]-N-(4-chloropyridin-2-yl)-3-fluorobenzamide	NC1=NC=CN2C(N3CCC4(CC3)CN(C3=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C3)C4)=NC(C3=C(F)C=C(C(=O)NC4=CC(Cl)=CC=N4)C=C3)=C12	C38H32ClFN10O5	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-IJK0L4	SCHEMBL24696603	4-[8-amino-3-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]oxy]ethoxy]ethoxy]ethyl]-2,7-diazaspiro[3.5]nonan-7-yl]imidazo[1,5-a]pyrazin-1-yl]-N-pyridin-2-ylbenzamide	NC1=NC=CN2C(N3CCC4(CC3)CN(CCOCCOCCOC3=CC=C5C(=O)N(C6CCC(=O)NC6=O)CC5=C3)C4)=NC(C3=CC=C(C(=O)NC4=CC=CC=N4)C=C3)=C12	C44H48N10O7	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-8P50ED	SCHEMBL24696607	4-[8-amino-3-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]amino]ethoxy]ethoxy]ethyl]-2,7-diazaspiro[3.5]nonan-7-yl]imidazo[1,5-a]pyrazin-1-yl]-N-(4-chloropyridin-2-yl)-3-fluorobenzamide	NC1=NC=CN2C(N3CCC4(CC3)CN(CCOCCOCCNC3=CC=C5C(=O)N(C6CCC(=O)NC6=O)CC5=C3)C4)=NC(C3=C(F)C=C(C(=O)NC4=CC(Cl)=CC=N4)C=C3)=C12	C44H47ClFN11O6	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-A2U29V	SCHEMBL24696609	4-[3-[(2S,3aR,6aS)-1-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]oxy]ethoxy]ethoxy]ethyl]-2,3,3a,4,6,6a-hexahydrofuro[3,4-b]pyrrol-2-yl]-8-aminoimidazo[1,5-a]pyrazin-1-yl]-N-pyridin-2-ylbenzamide	[H][C@]12COC[C@@]1([H])N(CCOCCOCCOC1=CC=C3C(=O)N(C4CCC(=O)NC4=O)CC3=C1)[C@H](C1=NC(C3=CC=C(C(=O)NC4=CC=CC=N4)C=C3)=C3C(N)=NC=CN13)C2	C43H45N9O8	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-UO9R40	SCHEMBL24696604	4-[8-amino-3-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]oxy]ethoxy]ethoxy]ethyl]-1-oxo-2,8-diazaspiro[4.5]decan-8-yl]imidazo[1,5-a]pyrazin-1-yl]-N-(4-chloropyridin-2-yl)-3-fluorobenzamide	NC1=NC=CN2C(N3CCC4(CCN(CCOCCOCCOC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6)C4=O)CC3)=NC(C3=C(F)C=C(C(=O)NC4=CC(Cl)=CC=N4)C=C3)=C12	C45H46ClFN10O8	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-6VXFA4	WO2022253250A1_18	.	NC1=NC=CN2C(N3CC4(CN(CCOCCOCCOC5=CC=C6C(=O)N(C7CCC(=O)NC7=O)CC6=C5)C4)C3)=NC(C3=C(F)C=C(C(=O)NC4=CC(Cl)=CC=N4)C=C3)=C12	C42H42ClFN10O7	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-RBOCQN	SCHEMBL24696605	4-[8-amino-3-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-3-oxo-1H-isoindol-5-yl]oxy]ethoxy]ethoxy]ethyl]-2,7-diazaspiro[3.5]nonan-7-yl]imidazo[1,5-a]pyrazin-1-yl]-N-(4-chloropyridin-2-yl)-3-fluorobenzamide	NC1=NC=CN2C(N3CCC4(CC3)CN(CCOCCOCCOC3=CC=C5CN(C6CCC(=O)NC6=O)C(=O)C5=C3)C4)=NC(C3=C(F)C=C(C(=O)NC4=CC(Cl)=CC=N4)C=C3)=C12	C44H46ClFN10O7	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-57QO9Z	SCHEMBL24696598	4-[8-amino-3-[2-[4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]oxy]butoxy]butyl]-2,7-diazaspiro[3.5]nonan-7-yl]imidazo[1,5-a]pyrazin-1-yl]-N-(4-chloropyridin-2-yl)-3-fluorobenzamide	NC1=NC=CN2C(N3CCC4(CC3)CN(CCCCOCCCCOC3=CC=C5C(=O)N(C6CCC(=O)NC6=O)CC5=C3)C4)=NC(C3=C(F)C=C(C(=O)NC4=CC(Cl)=CC=N4)C=C3)=C12	C46H50ClFN10O6	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-Y05ZO3	SCHEMBL24696714	4-[8-amino-3-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-3-oxo-1H-isoindol-4-yl]oxy]ethoxy]ethoxy]ethyl]-2,7-diazaspiro[3.5]nonan-7-yl]imidazo[1,5-a]pyrazin-1-yl]-N-(4-chloropyridin-2-yl)-3-fluorobenzamide	NC1=NC=CN2C(N3CCC4(CC3)CN(CCOCCOCCOC3=C5C(=O)N(C6CCC(=O)NC6=O)CC5=CC=C3)C4)=NC(C3=C(F)C=C(C(=O)NC4=CC(Cl)=CC=N4)C=C3)=C12	C44H46ClFN10O7	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-Q7D0PG	SCHEMBL24696739	4-[8-amino-3-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]oxy]ethoxy]ethoxy]ethyl]-2,7-diazaspiro[3.5]nonan-7-yl]imidazo[1,5-a]pyrazin-1-yl]-N-(4-chloropyridin-2-yl)-3-fluorobenzamide	NC1=NC=CN2C(N3CCC4(CC3)CN(CCOCCOCCOC3=C5CN(C6CCC(=O)NC6=O)C(=O)C5=CC=C3)C4)=NC(C3=C(F)C=C(C(=O)NC4=CC(Cl)=CC=N4)C=C3)=C12	C44H46ClFN10O7	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-RWNK89	SCHEMBL24696961	4-[8-amino-3-[2-[8-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]amino]octyl]-2,7-diazaspiro[3.5]nonan-7-yl]imidazo[1,5-a]pyrazin-1-yl]-N-(4-chloropyridin-2-yl)-3-fluorobenzamide	NC1=NC=CN2C(N3CCC4(CC3)CN(CCCCCCCCNC3=CC=C5C(=O)N(C6CCC(=O)NC6=O)CC5=C3)C4)=NC(C3=C(F)C=C(C(=O)NC4=CC(Cl)=CC=N4)C=C3)=C12	C46H51ClFN11O4	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-KK7H0G	SCHEMBL24697234	4-[8-amino-3-[2-[9-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]nonyl]-2,7-diazaspiro[3.5]nonan-7-yl]imidazo[1,5-a]pyrazin-1-yl]-N-(4-chloropyridin-2-yl)-3-fluorobenzamide	NC1=NC=CN2C(N3CCC4(CC3)CN(CCCCCCCCCC3=CC=C5C(=O)N(C6CCC(=O)NC6=O)CC5=C3)C4)=NC(C3=C(F)C=C(C(=O)NC4=CC(Cl)=CC=N4)C=C3)=C12	C47H52ClFN10O4	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-UU0MT1	SCHEMBL24696579	4-[8-amino-3-[2-[2-[5-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]oxy]pentoxy]ethyl]-2,7-diazaspiro[3.5]nonan-7-yl]imidazo[1,5-a]pyrazin-1-yl]-N-(4-chloropyridin-2-yl)-3-fluorobenzamide	NC1=NC=CN2C(N3CCC4(CC3)CN(CCOCCCCCOC3=CC=C5C(=O)N(C6CCC(=O)NC6=O)CC5=C3)C4)=NC(C3=C(F)C=C(C(=O)NC4=CC(Cl)=CC=N4)C=C3)=C12	C45H48ClFN10O6	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-HDN9LL	SCHEMBL24697431	4-[8-amino-3-[2-[4-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]amino]butyl]-2,7-diazaspiro[3.5]nonan-7-yl]imidazo[1,5-a]pyrazin-1-yl]-N-(4-chloropyridin-2-yl)-3-fluorobenzamide	NC1=NC=CN2C(N3CCC4(CC3)CN(CCCCNC3=CC=C5C(=O)N(C6CCC(=O)NC6=O)CC5=C3)C4)=NC(C3=C(F)C=C(C(=O)NC4=CC(Cl)=CC=N4)C=C3)=C12	C42H43ClFN11O4	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-VMVNQ8	SCHEMBL24697011	4-[8-amino-3-[2-[[(3R)-1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]pyrrolidin-3-yl]methyl]-2,7-diazaspiro[3.5]nonan-7-yl]imidazo[1,5-a]pyrazin-1-yl]-N-(4-chloropyridin-2-yl)-3-fluorobenzamide	NC1=NC=CN2C(N3CCC4(CC3)CN(C[C@H]3CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C3)C4)=NC(C3=C(F)C=C(C(=O)NC4=CC(Cl)=CC=N4)C=C3)=C12	C43H41ClFN11O5	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-H0W06Y	WO2022253250A1_27	.	NC1=NC=CN2C(N3CCC4(CC3)CN(C[C@@H]3CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C3)C4)=NC(C3=C(F)C=C(C(=O)NC4=CC(Cl)=CC=N4)C=C3)=C12	C43H41ClFN11O5	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-9I7HKG	SCHEMBL24697032	4-[8-amino-3-[2-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]-2,7-diazaspiro[3.5]nonan-7-yl]imidazo[1,5-a]pyrazin-1-yl]-N-(4-chloropyridin-2-yl)-3-fluorobenzamide	NC1=NC=CN2C(N3CCC4(CC3)CN(CC3CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC3)C4)=NC(C3=C(F)C=C(C(=O)NC4=CC(Cl)=CC=N4)C=C3)=C12	C44H43ClFN11O5	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-7KGCUF	SCHEMBL24696761	4-[8-amino-3-[2-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]ethyl]-2,7-diazaspiro[3.5]nonan-7-yl]imidazo[1,5-a]pyrazin-1-yl]-N-(4-chloropyridin-2-yl)-3-fluorobenzamide	NC1=NC=CN2C(N3CCC4(CC3)CN(CCN3CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC3)C4)=NC(C3=C(F)C=C(C(=O)NC4=CC(Cl)=CC=N4)C=C3)=C12	C44H44ClFN12O5	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-C4L460	SCHEMBL24696597	4-[8-amino-3-[2-[8-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]oxy]octyl]-2,7-diazaspiro[3.5]nonan-7-yl]imidazo[1,5-a]pyrazin-1-yl]-N-(4-chloropyridin-2-yl)-3-fluorobenzamide	NC1=NC=CN2C(N3CCC4(CC3)CN(CCCCCCCCOC3=CC=C5C(=O)N(C6CCC(=O)NC6=O)CC5=C3)C4)=NC(C3=C(F)C=C(C(=O)NC4=CC(Cl)=CC=N4)C=C3)=C12	C46H50ClFN10O5	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-OVV52X	SCHEMBL24697029	4-[8-amino-3-[2-[[(1R,5S)-3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-3-azabicyclo[3.1.0]hexan-6-yl]methyl]-2,7-diazaspiro[3.5]nonan-7-yl]imidazo[1,5-a]pyrazin-1-yl]-N-(4-chloropyridin-2-yl)-3-fluorobenzamide	[H][C@@]12CN(C3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C[C@]1([H])C2CN1CC2(CCN(C3=NC(C4=C(F)C=C(C(=O)NC5=CC(Cl)=CC=N5)C=C4)=C4C(N)=NC=CN34)CC2)C1	C44H41ClFN11O5	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-0SM67W	SCHEMBL24697033	4-[8-amino-3-[2-[[(1R,5S)-3-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]-3-azabicyclo[3.1.0]hexan-6-yl]methyl]-2,7-diazaspiro[3.5]nonan-7-yl]imidazo[1,5-a]pyrazin-1-yl]-N-(4-chloropyridin-2-yl)-3-fluorobenzamide	[H][C@@]12CN(C3=CC4=C(C=C3F)C(=O)N(C3CCC(=O)NC3=O)C4=O)C[C@]1([H])[C@H]2CN1CC2(CCN(C3=NC(C4=C(F)C=C(C(=O)NC5=CC(Cl)=CC=N5)C=C4)=C4C(N)=NC=CN34)CC2)C1	C44H40ClF2N11O5	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-HFI5FO	SCHEMBL24697759	4-[8-amino-3-[2-[[(3R)-1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]pyrrolidin-3-yl]methyl]-2,7-diazaspiro[3.5]nonan-7-yl]imidazo[1,5-a]pyrazin-1-yl]-N-(4-chloropyridin-2-yl)-3-fluorobenzamide	NC1=NC=CN2C(N3CCC4(CC3)CN(C[C@H]3CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)CC6=C5)C3)C4)=NC(C3=C(F)C=C(C(=O)NC4=CC(Cl)=CC=N4)C=C3)=C12	C43H43ClFN11O4	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-LKLWP1	SCHEMBL24696742	4-[8-amino-3-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]-2,7-diazaspiro[3.5]nonan-7-yl]imidazo[1,5-a]pyrazin-1-yl]-N-(4-chloropyridin-2-yl)-3-fluorobenzamide	NC1=NC=CN2C(N3CCC4(CC3)CN(C3CN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C3)C4)=NC(C3=C(F)C=C(C(=O)NC4=CC(Cl)=CC=N4)C=C3)=C12	C41H37ClFN11O5	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-ONFG3E	SCHEMBL24697226	4-[8-amino-3-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]azetidin-3-yl]-2,7-diazaspiro[3.5]nonan-7-yl]imidazo[1,5-a]pyrazin-1-yl]-N-(4-chloropyridin-2-yl)-3-fluorobenzamide	NC1=NC=CN2C(N3CCC4(CC3)CN(C3CN(C5=C(F)C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C3)C4)=NC(C3=C(F)C=C(C(=O)NC4=CC(Cl)=CC=N4)C=C3)=C12	C41H36ClF2N11O5	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-1U96FT	SCHEMBL24697001	4-[8-amino-3-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]azetidin-3-yl]-2,7-diazaspiro[3.5]nonan-7-yl]imidazo[1,5-a]pyrazin-1-yl]-N-(4-chloropyridin-2-yl)-3-fluorobenzamide	NC1=NC=CN2C(N3CCC4(CC3)CN(C3CN(C5CN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)C3)C4)=NC(C3=C(F)C=C(C(=O)NC4=CC(Cl)=CC=N4)C=C3)=C12	C44H42ClFN12O5	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-JWXHL5	SCHEMBL24696737	4-[8-amino-3-[2-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]methyl]-2,7-diazaspiro[3.5]nonan-7-yl]imidazo[1,5-a]pyrazin-1-yl]-N-(4-chloropyridin-2-yl)-3-fluorobenzamide	NC1=NC=CN2C(N3CCC4(CC3)CN(CC3CN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C3)C4)=NC(C3=C(F)C=C(C(=O)NC4=CC(Cl)=CC=N4)C=C3)=C12	C42H39ClFN11O5	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-3JNG6D	SCHEMBL24697052	4-[8-amino-3-[2-[(3S)-1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]pyrrolidin-3-yl]-2,7-diazaspiro[3.5]nonan-7-yl]imidazo[1,5-a]pyrazin-1-yl]-N-(4-chloropyridin-2-yl)-3-fluorobenzamide	NC1=NC=CN2C(N3CCC4(CC3)CN([C@H]3CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C3)C4)=NC(C3=C(F)C=C(C(=O)NC4=CC(Cl)=CC=N4)C=C3)=C12	C42H39ClFN11O5	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-RED0B0	SCHEMBL24696729	4-[8-amino-3-[2-[(3S)-1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]pyrrolidin-3-yl]-2,7-diazaspiro[3.5]nonan-7-yl]imidazo[1,5-a]pyrazin-1-yl]-N-(4-chloropyridin-2-yl)-3-fluorobenzamide	NC1=NC=CN2C(N3CCC4(CC3)CN([C@H]3CCN(C5CN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)C3)C4)=NC(C3=C(F)C=C(C(=O)NC4=CC(Cl)=CC=N4)C=C3)=C12	C45H44ClFN12O5	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-TPH0A1	SCHEMBL24697012	4-[8-amino-3-[2-[(3R)-1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]pyrrolidin-3-yl]-2,7-diazaspiro[3.5]nonan-7-yl]imidazo[1,5-a]pyrazin-1-yl]-N-(4-chloropyridin-2-yl)-3-fluorobenzamide	NC1=NC=CN2C(N3CCC4(CC3)CN([C@@H]3CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C3)C4)=NC(C3=C(F)C=C(C(=O)NC4=CC(Cl)=CC=N4)C=C3)=C12	C42H39ClFN11O5	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-DLWSET	SCHEMBL24696599	4-[8-amino-3-[2-[8-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]oxy]octyl]-2,7-diazaspiro[3.5]nonan-7-yl]imidazo[1,5-a]pyrazin-1-yl]-3-fluoro-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide	NC1=NC=CN2C(N3CCC4(CC3)CN(CCCCCCCCOC3=CC=C5C(=O)N(C6CCC(=O)NC6=O)CC5=C3)C4)=NC(C3=C(F)C=C(C(=O)NC4=CC(C(F)(F)F)=CC=N4)C=C3)=C12	C47H50F4N10O5	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-MWJZ6N	SCHEMBL24696555	4-[8-amino-3-[2-[(3R)-1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]pyrrolidin-3-yl]-2,7-diazaspiro[3.5]nonan-7-yl]imidazo[1,5-a]pyrazin-1-yl]-N-(4-chloropyridin-2-yl)-3-fluorobenzamide	NC1=NC=CN2C(N3CCC4(CC3)CN([C@@H]3CCN(C5CN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)C3)C4)=NC(C3=C(F)C=C(C(=O)NC4=CC(Cl)=CC=N4)C=C3)=C12	C45H44ClFN12O5	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-2JTRNM	SCHEMBL24696733	4-[8-amino-3-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]-2,7-diazaspiro[3.5]nonan-7-yl]imidazo[1,5-a]pyrazin-1-yl]-N-(4-chloropyridin-2-yl)-3-fluorobenzamide	NC1=NC=CN2C(N3CCC4(CC3)CN(C3CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC3)C4)=NC(C3=C(F)C=C(C(=O)NC4=CC(Cl)=CC=N4)C=C3)=C12	C43H41ClFN11O5	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-EKLET3	SCHEMBL24697048	4-[8-amino-3-[2-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperidin-4-yl]-2,7-diazaspiro[3.5]nonan-7-yl]imidazo[1,5-a]pyrazin-1-yl]-N-(4-chloropyridin-2-yl)-3-fluorobenzamide	NC1=NC=CN2C(N3CCC4(CC3)CN(C3CCN(C5CN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC3)C4)=NC(C3=C(F)C=C(C(=O)NC4=CC(Cl)=CC=N4)C=C3)=C12	C46H46ClFN12O5	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-3W86RA	SCHEMBL24696721	3-[6-[8-[7-[8-amino-1-(4-phenoxyphenyl)imidazo[1,5-a]pyrazin-3-yl]-2,7-diazaspiro[3.5]nonan-2-yl]octoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	NC1=NC=CN2C(N3CCC4(CC3)CN(CCCCCCCCOC3=CC=C5C(=O)N(C6CCC(=O)NC6=O)CC5=C3)C4)=NC(C3=CC=C(OC4=CC=CC=C4)C=C3)=C12	C46H52N8O5	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-RCTVT4	SCHEMBL24696725	5-[3-[7-[8-Amino-1-(4-phenoxyphenyl)imidazo[1,5-a]pyrazin-3-yl]-2,7-diazaspiro[3.5]nonan-2-yl]azetidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	NC1=NC=CN2C(N3CCC4(CC3)CN(C3CN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C3)C4)=NC(C3=CC=C(OC4=CC=CC=C4)C=C3)=C12	C41H39N9O5	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-MFQHIW	SCHEMBL24696730	5-[3-[3-[7-[8-Amino-1-(4-phenoxyphenyl)imidazo[1,5-a]pyrazin-3-yl]-2,7-diazaspiro[3.5]nonan-2-yl]azetidin-1-yl]azetidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	NC1=NC=CN2C(N3CCC4(CC3)CN(C3CN(C5CN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)C3)C4)=NC(C3=CC=C(OC4=CC=CC=C4)C=C3)=C12	C44H44N10O5	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-8BYUWM	SCHEMBL24197195	5-[3-[7-[4-Amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]-2-azaspiro[3.5]nonan-2-yl]azetidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione; SCHEMBL30331164	NC1=C2C(C3=CC=C(OC4=CC=CC=C4)C=C3)=NN(C3CCC4(CC3)CN(C3CN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C3)C4)C2=NC=N1	C41H39N9O5	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-F4HJL6	SCHEMBL24196966	5-[3-[3-[7-[4-Amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]-2-azaspiro[3.5]nonan-2-yl]azetidin-1-yl]azetidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	NC1=C2C(C3=CC=C(OC4=CC=CC=C4)C=C3)=NN(C3CCC4(CC3)CN(C3CN(C5CN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)C3)C4)C2=NC=N1	C44H44N10O5	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-3XY38G	SCHEMBL24696554	5-[3-[7-[4-Amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]-2-azaspiro[3.5]nonan-2-yl]azetidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)-6-fluoroisoindole-1,3-dione	NC1=C2C(C3=CC=C(OC4=CC=CC=C4)C=C3)=NN(C3CCC4(CC3)CN(C3CN(C5=C(F)C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C3)C4)C2=NC=N1	C41H38FN9O5	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-T00T6I	SCHEMBL24696585	3-[6-[3-[7-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]-2-azaspiro[3.5]nonan-2-yl]azetidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	NC1=C2C(C3=CC=C(OC4=CC=CC=C4)C=C3)=NN(C3CCC4(CC3)CN(C3CN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)CC6=C5)C3)C4)C2=NC=N1	C41H41N9O4	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-UQ2NFS	SCHEMBL24696989	4-[8-amino-3-[2-[3-[3-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]oxy]propoxy]propyl]-2,7-diazaspiro[3.5]nonan-7-yl]imidazo[1,5-a]pyrazin-1-yl]-N-(4-chloropyridin-2-yl)-3-fluorobenzamide	NC1=NC=CN2C(N3CCC4(CC3)CN(CCCOCCCOC3=CC=C5C(=O)N(C6CCC(=O)NC6=O)CC5=C3)C4)=NC(C3=C(F)C=C(C(=O)NC4=CC(Cl)=CC=N4)C=C3)=C12	C44H46ClFN10O6	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-50KLMB	SCHEMBL24696727	5-[3-[[7-[4-Amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]-2-azaspiro[3.5]nonan-2-yl]methyl]azetidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	NC1=C2C(C3=CC=C(OC4=CC=CC=C4)C=C3)=NN(C3CCC4(CC3)CN(CC3CN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C3)C4)C2=NC=N1	C42H41N9O5	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-P9ZCJR	SCHEMBL24697024	5-[(3R)-3-[7-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]-2-azaspiro[3.5]nonan-2-yl]pyrrolidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	NC1=C2C(C3=CC=C(OC4=CC=CC=C4)C=C3)=NN(C3CCC4(CC3)CN([C@@H]3CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C3)C4)C2=NC=N1	C42H41N9O5	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-KHK3M8	SCHEMBL24697004	5-[(3S)-3-[7-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]-2-azaspiro[3.5]nonan-2-yl]pyrrolidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	NC1=C2C(C3=CC=C(OC4=CC=CC=C4)C=C3)=NN(C3CCC4(CC3)CN([C@H]3CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C3)C4)C2=NC=N1	C42H41N9O5	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-XQC7HA	SCHEMBL24697022	5-[4-[7-[4-Amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]-2-azaspiro[3.5]nonan-2-yl]piperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	NC1=C2C(C3=CC=C(OC4=CC=CC=C4)C=C3)=NN(C3CCC4(CC3)CN(C3CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC3)C4)C2=NC=N1	C43H43N9O5	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-C3FLDY	SCHEMBL24696589	5-[3-[9-[4-Amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]-3-azaspiro[5.5]undecan-3-yl]azetidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	NC1=C2C(C3=CC=C(OC4=CC=CC=C4)C=C3)=NN(C3CCC4(CC3)CCN(C3CN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C3)CC4)C2=NC=N1	C43H43N9O5	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-GDAFDR	SCHEMBL24696978	5-[4-[9-[4-Amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]-3-azaspiro[5.5]undecan-3-yl]piperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	NC1=C2C(C3=CC=C(OC4=CC=CC=C4)C=C3)=NN(C3CCC4(CC3)CCN(C3CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC3)CC4)C2=NC=N1	C45H47N9O5	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-3EYZK9	SCHEMBL24697404	5-[4-[[9-[4-Amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]-3-azaspiro[5.5]undecan-3-yl]methyl]piperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	NC1=C2C(C3=CC=C(OC4=CC=CC=C4)C=C3)=NN(C3CCC4(CC3)CCN(CC3CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC3)CC4)C2=NC=N1	C46H49N9O5	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-YPU1NC	SCHEMBL24196797	5-[3-[2-[4-Amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]-7-azaspiro[3.5]nonan-7-yl]azetidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione; SCHEMBL30332194	NC1=C2C(C3=CC=C(OC4=CC=CC=C4)C=C3)=NN(C3CC4(CCN(C5CN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C3)C2=NC=N1	C41H39N9O5	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-08SXEY	SCHEMBL24697199	5-[3-[8-[4-Amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]-2-azaspiro[4.5]decan-2-yl]azetidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	NC1=C2C(C3=CC=C(OC4=CC=CC=C4)C=C3)=NN(C3CCC4(CC3)CCN(C3CN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C3)C4)C2=NC=N1	C42H41N9O5	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-ZSYWH8	SCHEMBL24697241	5-[3-[(3aR,6aS)-5-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]-3,3a,4,5,6,6a-hexahydro-1H-cyclopenta[c]pyrrol-2-yl]azetidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	[H][C@@]12C[C@@H](N3N=C(C4=CC=C(OC5=CC=CC=C5)C=C4)C4=C(N)N=CN=C43)C[C@]1([H])CN(C1CN(C3=CC=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)C1)C2	C40H37N9O5	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-94KQNH	SCHEMBL24696600	4-[8-amino-3-[2-[2-[3-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]oxy]propoxy]ethyl]-2,7-diazaspiro[3.5]nonan-7-yl]imidazo[1,5-a]pyrazin-1-yl]-N-(4-chloropyridin-2-yl)-3-fluorobenzamide	NC1=NC=CN2C(N3CCC4(CC3)CN(CCOCCCOC3=CC=C5C(=O)N(C6CCC(=O)NC6=O)CC5=C3)C4)=NC(C3=C(F)C=C(C(=O)NC4=CC(Cl)=CC=N4)C=C3)=C12	C43H44ClFN10O6	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-S1C4TO	SCHEMBL24697746	5-[3-[3-[(3aR,6aS)-5-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]-3,3a,4,5,6,6a-hexahydro-1H-cyclopenta[c]pyrrol-2-yl]azetidin-1-yl]azetidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione; SCHEMBL26477430	[H][C@@]12C[C@@H](N3N=C(C4=CC=C(OC5=CC=CC=C5)C=C4)C4=C(N)N=CN=C43)C[C@]1([H])CN(C1CN(C3CN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)C3)C1)C2	C43H42N10O5	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-JUEEAE	SCHEMBL24697230	5-[3-[3-[4-Amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]-8-azaspiro[4.5]decan-8-yl]azetidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	NC1=C2C(C3=CC=C(OC4=CC=CC=C4)C=C3)=NN(C3CCC4(CCN(C5CN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C3)C2=NC=N1	C42H41N9O5	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-W5TYJ1	SCHEMBL24697020	5-[3-[9-[4-Amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]-2-azaspiro[5.5]undecan-2-yl]azetidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	NC1=C2C(C3=CC=C(OC4=CC=CC=C4)C=C3)=NN(C3CCC4(CCCN(C5CN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)C4)CC3)C2=NC=N1	C43H43N9O5	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-CI77K4	SCHEMBL24697813	5-[3-[6-[4-Amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]-2-azaspiro[3.3]heptan-2-yl]azetidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione; SCHEMBL30954853	NC1=C2C(C3=CC=C(OC4=CC=CC=C4)C=C3)=NN(C3CC4(C3)CN(C3CN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C3)C4)C2=NC=N1	C39H35N9O5	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-I50ELY	WO2022253250A1_64	.	NC1=C2C(C3=CC=C(OC4=CC=CC=C4)C=C3)=NN(C3CCC4(C3)CN(C3CN(C5=CC=C6C(=O)C(C7CCC(=O)NC7=O)C(=O)C6=C5)C3)C4)C2=NC=C1	C42H39N7O5	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-VOSIDD	SCHEMBL24697044	5-[3-[7-[4-Amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]-6-fluoro-2-azaspiro[3.5]nonan-2-yl]azetidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	NC1=C2C(C3=CC=C(OC4=CC=CC=C4)C=C3)=NN(C3CCC4(CC3F)CN(C3CN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C3)C4)C2=NC=N1	C41H38FN9O5	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-SYA72B	SCHEMBL24696561	5-[3-[7-[4-Amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]-3-fluoro-2-azaspiro[3.5]nonan-2-yl]azetidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	NC1=C2C(C3=CC=C(OC4=CC=CC=C4)C=C3)=NN(C3CCC4(CC3)CN(C3CN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C3)C4F)C2=NC=N1	C41H38FN9O5	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-B2FVJV	SCHEMBL24697045	3-[6-[3-[7-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]-2-azaspiro[3.5]nonan-2-yl]azetidin-1-yl]-5-fluoro-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	NC1=C2C(C3=CC=C(OC4=CC=CC=C4)C=C3)=NN(C3CCC4(CC3)CN(C3CN(C5=C(F)C=C6C(=O)N(C7CCC(=O)NC7=O)CC6=C5)C3)C4)C2=NC=N1	C41H40FN9O4	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-4PPEVK	SCHEMBL24697038	5-[4-[2-[4-Amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]-7-azaspiro[3.5]nonan-7-yl]piperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	NC1=C2C(C3=CC=C(OC4=CC=CC=C4)C=C3)=NN(C3CC4(CCN(C5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C3)C2=NC=N1	C43H43N9O5	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-4VFI4M	SCHEMBL24696569	5-[3-[6-[4-Amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]-3-azabicyclo[3.1.0]hexan-3-yl]azetidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	NC1=C2C(C3=CC=C(OC4=CC=CC=C4)C=C3)=NN(C3C4CN(C5CN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC43)C2=NC=N1	C38H33N9O5	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-BZPG9Q	SCHEMBL24697756	4-[8-amino-3-[2-[5-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]oxy]pentyl]-2,7-diazaspiro[3.5]nonan-7-yl]imidazo[1,5-a]pyrazin-1-yl]-N-(4-chloropyridin-2-yl)-3-fluorobenzamide	NC1=NC=CN2C(N3CCC4(CC3)CN(CCCCCOC3=CC=C5C(=O)N(C6CCC(=O)NC6=O)CC5=C3)C4)=NC(C3=C(F)C=C(C(=O)NC4=CC(Cl)=CC=N4)C=C3)=C12	C43H44ClFN10O5	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-8ZGG3G	SCHEMBL24697000	5-[3-[7-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]-3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinolin-2-yl]azetidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	NC1=C2C(C3=CC=C(OC4=CC=CC=C4)C=C3)=NN(C3CCC4CCN(C5CN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4C3)C2=NC=N1	C42H41N9O5	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-ULSNFO	SCHEMBL24697460	5-[3-[6-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]-3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinolin-2-yl]azetidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	NC1=C2C(C3=CC=C(OC4=CC=CC=C4)C=C3)=NN(C3CCC4CN(C5CN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CCC4C3)C2=NC=N1	C42H41N9O5	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-A5RKXP	SCHEMBL24697039	5-[3-[5-[4-Amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]-1,3,3a,4,5,6,7,7a-octahydroisoindol-2-yl]azetidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	NC1=C2C(C3=CC=C(OC4=CC=CC=C4)C=C3)=NN(C3CCC4CN(C5CN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4C3)C2=NC=N1	C41H39N9O5	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-YW1FBX	SCHEMBL24696996	5-[3-[6-[4-Amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]-3-azabicyclo[3.2.0]heptan-3-yl]azetidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	NC1=C2C(C3=CC=C(OC4=CC=CC=C4)C=C3)=NN(C3CC4CN(C5CN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC43)C2=NC=N1	C39H35N9O5	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-32VECR	SCHEMBL24697040	5-[3-[6-[4-Amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]-1,3,4,4a,5,6,7,7a-octahydrocyclopenta[c]pyridin-2-yl]azetidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	NC1=C2C(C3=CC=C(OC4=CC=CC=C4)C=C3)=NN(C3CC4CCN(C5CN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4C3)C2=NC=N1	C41H39N9O5	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-ZAVXVI	SCHEMBL24696731	5-[3-[7-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]-2-azaspiro[3.5]nonan-2-yl]azetidin-1-yl]-2-[(3R)-2,6-dioxopiperidin-3-yl]isoindole-1,3-dione	NC1=C2C(C3=CC=C(OC4=CC=CC=C4)C=C3)=NN(C3CCC4(CC3)CN(C3CN(C5=CC=C6C(=O)N([C@@H]7CCC(=O)NC7=O)C(=O)C6=C5)C3)C4)C2=NC=N1	C41H39N9O5	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-3BMOUW	SCHEMBL24696726	5-[3-[7-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]-2-azaspiro[3.5]nonan-2-yl]azetidin-1-yl]-2-[(3S)-2,6-dioxopiperidin-3-yl]isoindole-1,3-dione	NC1=C2C(C3=CC=C(OC4=CC=CC=C4)C=C3)=NN(C3CCC4(CC3)CN(C3CN(C5=CC=C6C(=O)N([C@H]7CCC(=O)NC7=O)C(=O)C6=C5)C3)C4)C2=NC=N1	C41H39N9O5	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-AP5QRJ	SCHEMBL24697021	(3R)-3-[6-[3-[7-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]-2-azaspiro[3.5]nonan-2-yl]azetidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	NC1=C2C(C3=CC=C(OC4=CC=CC=C4)C=C3)=NN(C3CCC4(CC3)CN(C3CN(C5=CC=C6C(=O)N([C@@H]7CCC(=O)NC7=O)CC6=C5)C3)C4)C2=NC=N1	C41H41N9O4	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-EVRGDN	SCHEMBL24696728	5-[3-[[7-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]-2-azaspiro[3.5]nonan-2-yl]methyl]azetidin-1-yl]-2-[(3R)-2,6-dioxopiperidin-3-yl]isoindole-1,3-dione	NC1=C2C(C3=CC=C(OC4=CC=CC=C4)C=C3)=NN(C3CCC4(CC3)CN(CC3CN(C5=CC=C6C(=O)N([C@@H]7CCC(=O)NC7=O)C(=O)C6=C5)C3)C4)C2=NC=N1	C42H41N9O5	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-CB2UT6	SCHEMBL24696601	4-[8-amino-3-[2-[4-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]oxy]butyl]-2,7-diazaspiro[3.5]nonan-7-yl]imidazo[1,5-a]pyrazin-1-yl]-N-(4-chloropyridin-2-yl)-3-fluorobenzamide	NC1=NC=CN2C(N3CCC4(CC3)CN(CCCCOC3=CC=C5C(=O)N(C6CCC(=O)NC6=O)CC5=C3)C4)=NC(C3=C(F)C=C(C(=O)NC4=CC(Cl)=CC=N4)C=C3)=C12	C42H42ClFN10O5	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-X6SI15	SCHEMBL24696724	5-[3-[[7-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]-2-azaspiro[3.5]nonan-2-yl]methyl]azetidin-1-yl]-2-[(3S)-2,6-dioxopiperidin-3-yl]isoindole-1,3-dione	NC1=C2C(C3=CC=C(OC4=CC=CC=C4)C=C3)=NN(C3CCC4(CC3)CN(CC3CN(C5=CC=C6C(=O)N([C@H]7CCC(=O)NC7=O)C(=O)C6=C5)C3)C4)C2=NC=N1	C42H41N9O5	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-340DM1	SCHEMBL24696740	4-[8-amino-3-[2-[3-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]oxy]propyl]-2,7-diazaspiro[3.5]nonan-7-yl]imidazo[1,5-a]pyrazin-1-yl]-N-(4-chloropyridin-2-yl)-3-fluorobenzamide	NC1=NC=CN2C(N3CCC4(CC3)CN(CCCOC3=CC=C5C(=O)N(C6CCC(=O)NC6=O)CC5=C3)C4)=NC(C3=C(F)C=C(C(=O)NC4=CC(Cl)=CC=N4)C=C3)=C12	C41H40ClFN10O5	BTK	Q06187	CRBN	WO-2022253250-A1
TPD-4M7M70	CHEMBL5428135	N-[4-[7-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]-2-oxoethoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-6-ethyl-1,2-dimethyl-4-oxoquinoline-3-carboxamide; SCHEMBL24737279; PD216107	CCC1=CC2=C(C=C1)N(C)C(C)=C(C(=O)NC1=CC=C(OC3=NC=NC4=CC(OCC(=O)NC5=CC=CC6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)=C(OC)C=C43)C(F)=C1)C2=O	C44H36FN7O10	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-EHCM3B	CHEMBL5415358	N-[4-[7-[6-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]-6-oxohexoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-6-ethyl-1,2-dimethyl-4-oxoquinoline-3-carboxamide; SCHEMBL24737928; SCHEMBL30002295; PD216119	CCC1=CC2=C(C=C1)N(C)C(C)=C(C(=O)NC1=CC=C(OC3=NC=NC4=CC(OCCCCCC(=O)NC5=CC=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)=C(OC)C=C43)C(F)=C1)C2=O	C48H46FN7O9	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-KVVPTZ	CHEMBL5422023	N-[4-[7-[6-[[2-(2,6-dioxopiperidin-3-yl)-3-oxo-1H-isoindol-4-yl]amino]-6-oxohexoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-6-ethyl-1,2-dimethyl-4-oxoquinoline-3-carboxamide; SCHEMBL24737299; SCHEMBL30002201; PD216122	CCC1=CC2=C(C=C1)N(C)C(C)=C(C(=O)NC1=CC=C(OC3=NC=NC4=CC(OCCCCCC(=O)NC5=CC=CC6=C5C(=O)N(C5CCC(=O)NC5=O)C6)=C(OC)C=C43)C(F)=C1)C2=O	C48H46FN7O9	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-MQZZEJ	CHEMBL5403126	N-[4-[7-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]amino]-2-oxoethoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-6-ethyl-1,2-dimethyl-4-oxoquinoline-3-carboxamide; SCHEMBL24737305; PD216113	CCC1=CC2=C(C=C1)N(C)C(C)=C(C(=O)NC1=CC=C(OC3=NC=NC4=CC(OCC(=O)NC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)=C(OC)C=C43)C(F)=C1)C2=O	C44H36FN7O10	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-Y3OHUP	SCHEMBL24737263	N-[4-[7-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]amino]-2-oxoethoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-6-ethyl-1,2-dimethyl-4-oxoquinoline-3-carboxamide	CCC1=CC2=C(C=C1)N(C)C(C)=C(C(=O)NC1=CC=C(OC3=NC=NC4=CC(OCC(=O)NC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6)=C(OC)C=C43)C(F)=C1)C2=O	C44H38FN7O9	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-VTD25G	CHEMBL5429906	N-[4-[7-[8-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]-8-oxooctoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-6-ethyl-1,2-dimethyl-4-oxoquinoline-3-carboxamide; SCHEMBL24737306; PD216110	CCC1=CC2=C(C=C1)N(C)C(C)=C(C(=O)NC1=CC=C(OC3=NC=NC4=CC(OCCCCCCCC(=O)NC5=CC=CC6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)=C(OC)C=C43)C(F)=C1)C2=O	C50H48FN7O10	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-3WGRAG	SCHEMBL24737313	N-[4-[7-[8-[[2-(2,6-dioxopiperidin-3-yl)-3-oxo-1H-isoindol-4-yl]amino]-8-oxooctoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-6-ethyl-1,2-dimethyl-4-oxoquinoline-3-carboxamide	CCC1=CC2=C(C=C1)N(C)C(C)=C(C(=O)NC1=CC=C(OC3=NC=NC4=CC(OCCCCCCCC(=O)NC5=CC=CC6=C5C(=O)N(C5CCC(=O)NC5=O)C6)=C(OC)C=C43)C(F)=C1)C2=O	C50H50FN7O9	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-U9H2V3	SCHEMBL24737287	N-[4-[7-[8-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]amino]-8-oxooctoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-6-ethyl-1,2-dimethyl-4-oxoquinoline-3-carboxamide	CCC1=CC2=C(C=C1)N(C)C(C)=C(C(=O)NC1=CC=C(OC3=NC=NC4=CC(OCCCCCCCC(=O)NC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6)=C(OC)C=C43)C(F)=C1)C2=O	C50H50FN7O9	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-A4S89R	SCHEMBL24737301	N-[4-[7-[10-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]-10-oxodecoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-6-ethyl-1,2-dimethyl-4-oxoquinoline-3-carboxamide	CCC1=CC2=C(C=C1)N(C)C(C)=C(C(=O)NC1=CC=C(OC3=NC=NC4=CC(OCCCCCCCCCC(=O)NC5=CC=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)=C(OC)C=C43)C(F)=C1)C2=O	C52H54FN7O9	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-SE5V82	SCHEMBL24737308	N-[4-[7-[8-[[2-(2,6-dioxopiperidin-3-yl)-3-oxo-1H-isoindol-5-yl]amino]-8-oxooctoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-6-ethyl-1,2-dimethyl-4-oxoquinoline-3-carboxamide	CCC1=CC2=C(C=C1)N(C)C(C)=C(C(=O)NC1=CC=C(OC3=NC=NC4=CC(OCCCCCCCC(=O)NC5=CC6=C(C=C5)CN(C5CCC(=O)NC5=O)C6=O)=C(OC)C=C43)C(F)=C1)C2=O	C50H50FN7O9	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-6TICK0	SCHEMBL24737262	N-[4-[7-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]-2-oxoethoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-6-ethyl-1,2-dimethyl-4-oxoquinoline-3-carboxamide; SCHEMBL30002116	CCC1=CC2=C(C=C1)N(C)C(C)=C(C(=O)NC1=CC=C(OC3=NC=NC4=CC(OCC(=O)NC5=CC=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)=C(OC)C=C43)C(F)=C1)C2=O	C44H38FN7O9	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-PUYITD	SCHEMBL24737285	N-[4-[7-[2-[[2-(2,6-dioxopiperidin-3-yl)-3-oxo-1H-isoindol-5-yl]amino]-2-oxoethoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-6-ethyl-1,2-dimethyl-4-oxoquinoline-3-carboxamide	CCC1=CC2=C(C=C1)N(C)C(C)=C(C(=O)NC1=CC=C(OC3=NC=NC4=CC(OCC(=O)NC5=CC6=C(C=C5)CN(C5CCC(=O)NC5=O)C6=O)=C(OC)C=C43)C(F)=C1)C2=O	C44H38FN7O9	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-7Q9V8O	CHEMBL5434192	N-[4-[7-[5-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]-5-oxopentoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-6-ethyl-1,2-dimethyl-4-oxoquinoline-3-carboxamide; SCHEMBL24737309; PD216108	CCC1=CC2=C(C=C1)N(C)C(C)=C(C(=O)NC1=CC=C(OC3=NC=NC4=CC(OCCCCC(=O)NC5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)=C(OC)C=C43)C(F)=C1)C2=O	C47H42FN7O10	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-VUU5ZJ	SCHEMBL24737310	N-[4-[7-[5-[[2-(2,6-dioxopiperidin-3-yl)-3-oxo-1H-isoindol-5-yl]amino]-5-oxopentoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-6-ethyl-1,2-dimethyl-4-oxoquinoline-3-carboxamide; SCHEMBL30002795	CCC1=CC2=C(C=C1)N(C)C(C)=C(C(=O)NC1=CC=C(OC3=NC=NC4=CC(OCCCCC(=O)NC5=CC=C6CN(C7CCC(=O)NC7=O)C(=O)C6=C5)=C(OC)C=C43)C(F)=C1)C2=O	C47H44FN7O9	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-UHMGTQ	CHEMBL5408071	N-[4-[7-[10-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]amino]-10-oxodecoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-6-ethyl-1,2-dimethyl-4-oxoquinoline-3-carboxamide; SCHEMBL24737291; PD216117	CCC1=CC2=C(C=C1)N(C)C(C)=C(C(=O)NC1=CC=C(OC3=NC=NC4=CC(OCCCCCCCCCC(=O)NC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)=C(OC)C=C43)C(F)=C1)C2=O	C52H52FN7O10	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-YUPO2H	SCHEMBL24737314	N-[4-[7-[10-[[2-(2,6-dioxopiperidin-3-yl)-3-oxo-1H-isoindol-5-yl]amino]-10-oxodecoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-6-ethyl-1,2-dimethyl-4-oxoquinoline-3-carboxamide; SCHEMBL30002015	CCC1=CC2=C(C=C1)N(C)C(C)=C(C(=O)NC1=CC=C(OC3=NC=NC4=CC(OCCCCCCCCCC(=O)NC5=CC6=C(C=C5)CN(C5CCC(=O)NC5=O)C6=O)=C(OC)C=C43)C(F)=C1)C2=O	C52H54FN7O9	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-YHZN6I	SCHEMBL24737294	N-[4-[7-[5-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]-5-oxopentoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-6-ethyl-1,2-dimethyl-4-oxoquinoline-3-carboxamide; SCHEMBL30002252	CCC1=CC2=C(C=C1)N(C)C(C)=C(C(=O)NC1=CC=C(OC3=NC=NC4=CC(OCCCCC(=O)NC5=C6CN(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)=C(OC)C=C43)C(F)=C1)C2=O	C47H44FN7O9	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-6FNH75	SCHEMBL24737303	N-[4-[7-[8-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]-8-oxooctoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-6-ethyl-1,2-dimethyl-4-oxoquinoline-3-carboxamide	CCC1=CC2=C(C=C1)N(C)C(C)=C(C(=O)NC1=CC=C(OC3=NC=NC4=CC(OCCCCCCCC(=O)NC5=CC=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)=C(OC)C=C43)C(F)=C1)C2=O	C50H50FN7O9	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-XW9T2U	CHEMBL5433966	N-[4-[7-[6-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]amino]-6-oxohexoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-6-ethyl-1,2-dimethyl-4-oxoquinoline-3-carboxamide; SCHEMBL24737290; PD216115	CCC1=CC2=C(C=C1)N(C)C(C)=C(C(=O)NC1=CC=C(OC3=NC=NC4=CC(OCCCCCC(=O)NC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)=C(OC)C=C43)C(F)=C1)C2=O	C48H44FN7O10	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-R8WDXS	CHEMBL5412649	N-[4-[7-[12-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]amino]-12-oxododecoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-6-ethyl-1,2-dimethyl-4-oxoquinoline-3-carboxamide; SCHEMBL24737304; SCHEMBL30002328; PD216118	CCC1=CC2=C(C=C1)N(C)C(C)=C(C(=O)NC1=CC=C(OC3=NC=NC4=CC(OCCCCCCCCCCCC(=O)NC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)=C(OC)C=C43)C(F)=C1)C2=O	C54H56FN7O10	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-Y2E838	SCHEMBL24737292	N-[4-[7-[10-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]amino]-10-oxodecoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-6-ethyl-1,2-dimethyl-4-oxoquinoline-3-carboxamide	CCC1=CC2=C(C=C1)N(C)C(C)=C(C(=O)NC1=CC=C(OC3=NC=NC4=CC(OCCCCCCCCCC(=O)NC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6)=C(OC)C=C43)C(F)=C1)C2=O	C52H54FN7O9	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-E7V888	CHEMBL5394454	N-[4-[7-[6-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]amino]-6-oxohexoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-6-ethyl-1,2-dimethyl-4-oxoquinoline-3-carboxamide; SCHEMBL24737256; SCHEMBL30002244; BDBM50616896; PD216120	CCC1=CC2=C(C=C1)N(C)C(C)=C(C(=O)NC1=CC=C(OC3=NC=NC4=CC(OCCCCCC(=O)NC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6)=C(OC)C=C43)C(F)=C1)C2=O	C48H46FN7O9	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-PQOEZN	SCHEMBL24737251	N-[4-[7-[5-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]amino]-5-oxopentoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-6-ethyl-1,2-dimethyl-4-oxoquinoline-3-carboxamide; SCHEMBL30002708	CCC1=CC2=C(C=C1)N(C)C(C)=C(C(=O)NC1=CC=C(OC3=NC=NC4=CC(OCCCCC(=O)NC5=CC=C6C(=O)N(C7CCC(=O)NC7=O)CC6=C5)=C(OC)C=C43)C(F)=C1)C2=O	C47H44FN7O9	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-LK894A	CHEMBL5424653	N-[4-[7-[6-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]-6-oxohexoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-6-ethyl-1,2-dimethyl-4-oxoquinoline-3-carboxamide; SCHEMBL24737234; PD216109	CCC1=CC2=C(C=C1)N(C)C(C)=C(C(=O)NC1=CC=C(OC3=NC=NC4=CC(OCCCCCC(=O)NC5=CC=CC6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)=C(OC)C=C43)C(F)=C1)C2=O	C48H44FN7O10	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-51AS8A	CHEMBL5425980	N-[4-[7-[5-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]amino]-5-oxopentoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-6-ethyl-1,2-dimethyl-4-oxoquinoline-3-carboxamide; SCHEMBL24737841; PD216114	CCC1=CC2=C(C=C1)N(C)C(C)=C(C(=O)NC1=CC=C(OC3=NC=NC4=CC(OCCCCC(=O)NC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)=C(OC)C=C43)C(F)=C1)C2=O	C47H42FN7O10	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-B4I5VB	CHEMBL5394497	N-[4-[7-[10-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]-10-oxodecoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-6-ethyl-1,2-dimethyl-4-oxoquinoline-3-carboxamide; SCHEMBL24737768; PD216111	CCC1=CC2=C(C=C1)N(C)C(C)=C(C(=O)NC1=CC=C(OC3=NC=NC4=CC(OCCCCCCCCCC(=O)NC5=CC=CC6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)=C(OC)C=C43)C(F)=C1)C2=O	C52H52FN7O10	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-8YJPQG	SCHEMBL30002066	N-[4-[7-[6-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]amino]-6-oxohexoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-6-methoxy-1,2-dimethyl-4-oxoquinoline-3-carboxamide	COC1=CC2=C(C=C1)N(C)C(C)=C(C(=O)NC1=CC(F)=C(OC3=NC=NC4=CC(OCCCCCC(=O)NC5=CC=C6C(=O)N(C7CCC(=O)NC7=O)CC6=C5)=C(OC)C=C43)C=C1)C2=O	C47H44FN7O10	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-VT54LB	SCHEMBL30001934	N-[4-[7-[6-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]amino]-6-oxohexoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide	COC1=C(OCCCCCC(=O)NC2=CC=C3C(=O)N(C4CCC(=O)NC4=O)CC3=C2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C47H41F4N7O10	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-NPUVBU	WO2022253283A1_37	.	COC1=C(OCC(=O)N2CC3CN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5)CC3C2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C49H42F4N8O10	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-B483R0	WO2022253283A1_38	.	COC1=C(OCC(=O)N2CC3(C2)CN(C2=CC4=C(C=C2)C(=O)N(C2CCC(=O)NC2=O)C4)C3)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C48H40F4N8O10	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-DULHCD	SCHEMBL30002255	N-[4-[7-[2-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]azetidin-3-yl]amino]-2-oxoethoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide	COC1=C(OCC(=O)NC2CN(C3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4)C2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C46H38F4N8O10	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-0BM9RN	SCHEMBL30002057	N-[4-[7-[2-[7-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-2,7-diazaspiro[3.5]nonan-2-yl]-2-oxoethoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide	COC1=C(OCC(=O)N2CC3(CCN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5)CC3)C2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C50H44F4N8O10	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-4U7KMJ	SCHEMBL24737775	N-[4-[7-[2-[4-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]oxy]ethyl]piperidin-1-yl]-2-oxoethoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide	COC1=C(OCC(=O)N2CCC(CCOC3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4)CC2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C50H45F4N7O11	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-UUDU3V	WO2022253283A1_42	.	COC1=C(OCC(=O)NC2CCC(CC(=O)NC3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4)CC2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C51H46F4N8O11	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-A2J34C	SCHEMBL30002198	N-[4-[7-[2-[4-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]amino]-2-oxoethyl]piperidin-1-yl]-2-oxoethoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide	COC1=C(OCC(=O)N2CCC(CC(=O)NC3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4)CC2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C50H44F4N8O11	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-KDQZPN	SCHEMBL30002250	N-[4-[7-[2-[4-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]carbamoyl]piperidin-1-yl]-2-oxoethoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide	COC1=C(OCC(=O)N2CCC(C(=O)NC3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4)CC2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C49H42F4N8O11	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-YMUYD4	SCHEMBL30001602	N-[4-[7-[2-[[4-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]carbamoyl]cyclohexyl]methylamino]-2-oxoethoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide	COC1=C(OCC(=O)NCC2CCC(C(=O)NC3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4)CC2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C51H46F4N8O11	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-JTCE60	SCHEMBL30002022	N-[4-[7-[2-[3-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]carbamoyl]azetidin-1-yl]-2-oxoethoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide	COC1=C(OCC(=O)N2CC(C(=O)NC3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4)C2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C47H38F4N8O11	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-8NY1PY	WO2022253283A1_47	N-[4-[7-[2-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]ethynyl]piperidin-1-yl]-2-oxoethoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide	COC1=C(OCC(=O)N2CCC(C#CC3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4)CC2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C50H41F4N7O10	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-G870HU	SCHEMBL30002327	N-[4-[7-[2-[(3S)-3-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]carbamoyl]piperidin-1-yl]-2-oxoethoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide	COC1=C(OCC(=O)N2CCC[C@H](C(=O)NC3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4)C2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C49H42F4N8O11	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-DOAG8G	SCHEMBL24737777	N-[4-[7-[2-[3-[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]ethynyl]anilino]-2-oxoethoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide; SCHEMBL30002284	COC1=C(OCC(=O)NC2=CC(C#CC3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4)=CC=C2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C51H37F4N7O10	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-KLI3AO	SCHEMBL30001539	N-[4-[7-[2-[3-[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]ethynyl]azetidin-1-yl]-2-oxoethoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide	COC1=C(OCC(=O)N2CC(C#CC3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4)C2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C48H37F4N7O10	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-6IWRNI	SCHEMBL30001547	N-[4-[7-[2-[[4-[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]ethynyl]cyclohexyl]amino]-2-oxoethoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide	COC1=C(OCC(=O)NC2CCC(C#CC3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4)CC2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C51H43F4N7O10	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-ECN4KZ	SCHEMBL30002859	N-[4-[7-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]carbamoyl]-6-azaspiro[2.5]octan-6-yl]-2-oxoethoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide	COC1=C(OCC(=O)N2CCC3(CC2)CC3C(=O)NC2=CC3=C(C=C2)C(=O)N(C2CCC(=O)NC2=O)C3)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C51H44F4N8O11	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-0PS2X5	WO2022253283A1_53	.	COC1=C(OCC(=O)N2CCN(CC(=O)NC3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4)CC2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C49H43F4N9O11	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-UGF1L2	SCHEMBL30002241	N-[4-[7-[2-[4-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]amino]ethyl]piperidin-1-yl]-2-oxoethoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide	COC1=C(OCC(=O)N2CCC(CCNC3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4)CC2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C50H46F4N8O10	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-C9P7CQ	WO2022253283A1_55	.	COC1=C(OCC(=O)N2CCC3(CC2)CCN(C(=O)C2=CC4=C(C=C2)C(=O)N(C2CCC(=O)NC2=O)C4)C3)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C52H46F4N8O11	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-R1FIIJ	WO2022253283A1_56	.	COC1=C(OCC(=O)N2CCC(CNC(=O)C3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4)CC2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C50H44F4N8O11	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-KK4EAC	WO2022253283A1_57	.	COC1=C(OCC(=O)N2CC3CN(CC(=O)NC4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5)CC3C2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C51H45F4N9O11	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-0FCPYO	WO2022253283A1_58	N-[4-[7-[2-[3-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]amino]-2-oxoethyl]-3,8-diazabicyclo[3.2.1]octan-8-yl]-2-oxoethoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide	COC1=C(OCC(=O)N2C3CCC2CN(CC(=O)NC2=CC4=C(C=C2)C(=O)N(C2CCC(=O)NC2=O)C4)C3)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C51H45F4N9O11	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-15U9MC	SCHEMBL30001560	N-[4-[7-[2-[3-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]amino]-2-oxoethyl]-3,6-diazabicyclo[3.1.1]heptan-6-yl]-2-oxoethoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide	COC1=C(OCC(=O)N2C3CC2CN(CC(=O)NC2=CC4=C(C=C2)C(=O)N(C2CCC(=O)NC2=O)C4)C3)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C50H43F4N9O11	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-AEI0XC	WO2022253283A1_60	N-[4-[7-[2-[[4-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]amino]-2-oxoethyl]piperazin-1-yl]amino]-2-oxoethoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide	COC1=C(OCC(=O)NN2CCN(CC(=O)NC3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4)CC2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C49H44F4N10O11	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-LW96MO	SCHEMBL30001619	N-[4-[7-[2-[4-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]carbamoylamino]piperazin-1-yl]-2-oxoethoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide	COC1=C(OCC(=O)N2CCN(NC(=O)NC3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4)CC2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C48H42F4N10O11	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-144JMZ	WO2022253283A1_62	.	COC1=C(OCC(=O)N2CCC3(CCN(CC(=O)NC4=CC=C5C(=O)N(C6CCC(=O)NC6=O)CC5=C4)CC3)CC2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C54H51F4N9O11	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-9L5A3Q	SCHEMBL30002097	N-[4-[7-[2-[8-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]amino]-2-oxoethyl]-3,8-diazabicyclo[3.2.1]octan-3-yl]-2-oxoethoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide	COC1=C(OCC(=O)N2CC3CCC(C2)N3CC(=O)NC2=CC3=C(C=C2)C(=O)N(C2CCC(=O)NC2=O)C3)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C51H45F4N9O11	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-0IB82D	SCHEMBL30001600	N-[4-[7-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindole-5-carbonyl]-2,7-diazaspiro[3.5]nonan-7-yl]-2-oxoethoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide	COC1=C(OCC(=O)N2CCC3(CC2)CN(C(=O)C2=CC4=C(C=C2)C(=O)N(C2CCC(=O)NC2=O)C4)C3)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C51H44F4N8O11	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-NOUC62	WO2022253283A1_65	.	COC1=C(OCC(=O)N2CC3(CCN(C(=O)C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5)CC3)C2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C51H44F4N8O11	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-32MBS8	SCHEMBL30002069	N-[4-[7-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindole-5-carbonyl]-2,6-diazaspiro[3.3]heptan-6-yl]-2-oxoethoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide	COC1=C(OCC(=O)N2CC3(C2)CN(C(=O)C2=CC4=C(C=C2)C(=O)N(C2CCC(=O)NC2=O)C4)C3)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C49H40F4N8O11	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-23DWAY	SCHEMBL30002234	N-[4-[7-[2-[3-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindole-5-carbonyl]-3,9-diazaspiro[5.5]undecan-9-yl]-2-oxoethoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide	COC1=C(OCC(=O)N2CCC3(CC2)CCN(C(=O)C2=CC4=C(C=C2)C(=O)N(C2CCC(=O)NC2=O)C4)CC3)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C53H48F4N8O11	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-KX7FWL	SCHEMBL30002065	N-[4-[7-[2-[4-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]-2-oxoethyl]piperidin-1-yl]-2-oxoethoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide	COC1=C(OCC(=O)N2CCC(CC(=O)NC3=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)CC2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C50H44F4N8O11	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-S1G2OE	SCHEMBL30002064	N-[4-[7-[2-[4-[2-[[2-(2,6-dioxopiperidin-3-yl)-3-oxo-1H-isoindol-5-yl]amino]-2-oxoethyl]piperidin-1-yl]-2-oxoethoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide	COC1=C(OCC(=O)N2CCC(CC(=O)NC3=CC4=C(C=C3)CN(C3CCC(=O)NC3=O)C4=O)CC2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C50H44F4N8O11	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-AI7236	SCHEMBL30002004	N-[4-[7-[2-[[4-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]carbamoyl]cyclohexyl]methylamino]-2-oxoethoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide	COC1=C(OCC(=O)NCC2CCC(C(=O)NC3=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)CC2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C51H46F4N8O11	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-MK3TY5	WO2022253283A1_71	.	COC1=C(OCC(=O)N2CCC(CC(=O)NC3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C50H42F4N8O12	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-321XEF	WO2022253283A1_72	.	COC1=C(OCCCC(=O)N2CC3CN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5)CC3C2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C51H46F4N8O10	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-M4YOX2	SCHEMBL30002242	N-[4-[7-[4-[6-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-2,6-diazaspiro[3.3]heptan-2-yl]-4-oxobutoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide	COC1=C(OCCCC(=O)N2CC3(C2)CN(C2=CC4=C(C=C2)C(=O)N(C2CCC(=O)NC2=O)C4)C3)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C50H44F4N8O10	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-C323MO	WO2022253283A1_74	N-[4-[7-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]azetidin-3-yl]amino]-4-oxobutoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide	COC1=C(OCCCC(=O)NC2CN(C3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4)C2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C48H42F4N8O10	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-38LKWK	WO2022253283A1_75	N-[4-[7-[4-[7-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-2,7-diazaspiro[3.5]nonan-2-yl]-4-oxobutoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide	COC1=C(OCCCC(=O)N2CC3(CCN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5)CC3)C2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C52H48F4N8O10	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-93BUB0	SCHEMBL30002761	N-[4-[7-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]-4-oxobutoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide	COC1=C(OCCCC(=O)N2CCN(C3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4)CC2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C49H44F4N8O10	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-LJFFE3	WO2022253283A1_77	N-[4-[7-[4-[[4-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]amino]-2-oxoethyl]cyclohexyl]amino]-4-oxobutoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide	COC1=C(OCCCC(=O)NC2CCC(CC(=O)NC3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4)CC2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C53H50F4N8O11	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-NZOIVO	WO2022253283A1_78	.	COC1=C(OCCCC(=O)NC2CCC(C(=O)NC3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4)CC2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C52H48F4N8O11	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-8PON7R	WO2022253283A1_79	N-[4-[7-[4-[[4-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]oxy]ethyl]cyclohexyl]amino]-4-oxobutoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide	COC1=C(OCCCC(=O)NC2CCC(CCOC3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4)CC2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C53H51F4N7O11	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-5NQ1PR	WO2022253283A1_80	N-[4-[7-[4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]carbamoyl]piperidin-1-yl]-4-oxobutoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide	COC1=C(OCCCC(=O)N2CCC(C(=O)NC3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4)CC2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C51H46F4N8O11	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-49MQGB	SCHEMBL30002030	N-[4-[7-[4-[4-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]amino]-2-oxoethyl]piperidin-1-yl]-4-oxobutoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide	COC1=C(OCCCC(=O)N2CCC(CC(=O)NC3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4)CC2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C52H48F4N8O11	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-HFIVW3	WO2022253283A1_82	N-[4-[7-[4-[3-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]carbamoyl]azetidin-1-yl]-4-oxobutoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide	COC1=C(OCCCC(=O)N2CC(C(=O)NC3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4)C2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C49H42F4N8O11	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-5M1V3N	WO2022253283A1_83	N-[4-[7-[4-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]ethynyl]piperidin-1-yl]-4-oxobutoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide	COC1=C(OCCCC(=O)N2CCC(C#CC3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4)CC2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C52H45F4N7O10	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-VTDE3C	WO2022253283A1_84	N-[4-[7-[4-[(3S)-3-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]carbamoyl]piperidin-1-yl]-4-oxobutoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide	COC1=C(OCCCC(=O)N2CCC[C@H](C(=O)NC3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4)C2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C51H46F4N8O11	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-7BV7A8	SCHEMBL24737261	N-[4-[7-[4-[3-[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]ethynyl]anilino]-4-oxobutoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide; SCHEMBL30002748	COC1=C(OCCCC(=O)NC2=CC(C#CC3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4)=CC=C2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C53H41F4N7O10	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-6QL265	WO2022253283A1_86	N-[4-[7-[4-[3-[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]ethynyl]azetidin-1-yl]-4-oxobutoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide	COC1=C(OCCCC(=O)N2CC(C#CC3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4)C2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C50H41F4N7O10	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-Q8C6B2	WO2022253283A1_87	.	COC1=C(OCCCC(=O)NC2CCC(C#CC3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4)CC2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C53H47F4N7O10	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-QDRLHQ	WO2022253283A1_88	N-[4-[7-[4-[3-[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]ethynyl]piperidin-1-yl]-4-oxobutoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide	COC1=C(OCCCC(=O)N2CCCC(C#CC3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4)C2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C52H45F4N7O10	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-URIK96	WO2022253283A1_89	N-[4-[7-[4-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]carbamoyl]-6-azaspiro[2.5]octan-6-yl]-4-oxobutoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide	COC1=C(OCCCC(=O)N2CCC3(CC2)CC3C(=O)NC2=CC=C3C(=O)N(C4CCC(=O)NC4=O)CC3=C2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C53H48F4N8O11	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-FYTUV5	WO2022253283A1_90	.	COC1=C(OCCCC(=O)N2CCN(CC(=O)NC3=CC=C4C(=O)N(C5CCC(=O)NC5=O)CC4=C3)CC2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C51H47F4N9O11	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-ESWPR9	SCHEMBL30002770	N-[4-[7-[4-[4-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]amino]ethyl]piperidin-1-yl]-4-oxobutoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide	COC1=C(OCCCC(=O)N2CCC(CCNC3=CC=C4C(=O)N(C5CCC(=O)NC5=O)CC4=C3)CC2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C52H50F4N8O10	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-6DE47M	SCHEMBL30002192	N-[4-[7-[4-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]amino]-2-oxoethyl]-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-5-yl]-4-oxobutoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide	COC1=C(OCCCC(=O)N2CC3CN(CC(=O)NC4=CC=C5C(=O)N(C6CCC(=O)NC6=O)CC5=C4)CC3C2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C53H49F4N9O11	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-EZAEKG	WO2022253283A1_93	.	COC1=C(OCCCC(=O)N2C3CCC2CN(CC(=O)NC2=CC=C4C(=O)N(C5CCC(=O)NC5=O)CC4=C2)C3)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C53H49F4N9O11	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-BVMJYM	WO2022253283A1_94	N-[4-[7-[4-[3-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]amino]-2-oxoethyl]-3,6-diazabicyclo[3.1.1]heptan-6-yl]-4-oxobutoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide	COC1=C(OCCCC(=O)N2C3CC2CN(CC(=O)NC2=CC=C4C(=O)N(C5CCC(=O)NC5=O)CC4=C2)C3)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C52H47F4N9O11	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-UY5LVR	WO2022253283A1_95	N-[4-[7-[4-[[4-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]amino]-2-oxoethyl]piperazin-1-yl]amino]-4-oxobutoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide	COC1=C(OCCCC(=O)NN2CCN(CC(=O)NC3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4)CC2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C51H48F4N10O11	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-OMVLB1	SCHEMBL24737255	N-[4-[7-[4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]carbamoylamino]piperazin-1-yl]-4-oxobutoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide; SCHEMBL30002060	COC1=C(OCCCC(=O)N2CCN(NC(=O)NC3=CC=C4C(=O)N(C5CCC(=O)NC5=O)CC4=C3)CC2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C50H46F4N10O11	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-UIAUDH	WO2022253283A1_97	N-[4-[7-[4-[9-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]amino]-2-oxoethyl]-3,9-diazaspiro[5.5]undecan-3-yl]-4-oxobutoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide	COC1=C(OCCCC(=O)N2CCC3(CCN(CC(=O)NC4=CC=C5C(=O)N(C6CCC(=O)NC6=O)CC5=C4)CC3)CC2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C56H55F4N9O11	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-71DGJV	WO2022253283A1_98	N-[4-[7-[4-[8-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]amino]-2-oxoethyl]-3,8-diazabicyclo[3.2.1]octan-3-yl]-4-oxobutoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide	COC1=C(OCCCC(=O)N2CC3CCC(C2)N3CC(=O)NC2=CC=C3C(=O)N(C4CCC(=O)NC4=O)CC3=C2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C53H49F4N9O11	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-B220G6	WO2022253283A1_99	N-[4-[7-[4-[6-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]amino]-2-oxoethyl]-3,6-diazabicyclo[3.1.1]heptan-3-yl]-4-oxobutoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide	COC1=C(OCCCC(=O)N2CC3CC(C2)N3CC(=O)NC2=CC=C3C(=O)N(C4CCC(=O)NC4=O)CC3=C2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C52H47F4N9O11	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-R9RV4A	WO2022253283A1_100	N-[4-[7-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindole-5-carbonyl]-2,8-diazaspiro[4.5]decan-8-yl]-4-oxobutoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide	COC1=C(OCCCC(=O)N2CCC3(CC2)CCN(C(=O)C2=CC=C4C(=O)N(C5CCC(=O)NC5=O)CC4=C2)C3)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C54H50F4N8O11	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-L76OP4	WO2022253283A1_101	.	COC1=C(OCCCC(=O)N2CCC(CNC(=O)C3=CC=C4C(=O)N(C5CCC(=O)NC5=O)CC4=C3)CC2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C52H48F4N8O11	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-A3ANKS	WO2022253283A1_102	N-[4-[7-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindole-5-carbonyl]-2,7-diazaspiro[3.5]nonan-7-yl]-4-oxobutoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide	COC1=C(OCCCC(=O)N2CCC3(CC2)CN(C(=O)C2=CC=C4C(=O)N(C5CCC(=O)NC5=O)CC4=C2)C3)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C53H48F4N8O11	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-3XN9WE	WO2022253283A1_103	N-[4-[7-[4-[7-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindole-5-carbonyl]-2,7-diazaspiro[3.5]nonan-2-yl]-4-oxobutoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide	COC1=C(OCCCC(=O)N2CC3(CCN(C(=O)C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)CC5=C4)CC3)C2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C53H48F4N8O11	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-FLIPPC	WO2022253283A1_104	N-[4-[7-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindole-5-carbonyl]-2,6-diazaspiro[3.3]heptan-6-yl]-4-oxobutoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide	COC1=C(OCCCC(=O)N2CC3(C2)CN(C(=O)C2=CC=C4C(=O)N(C5CCC(=O)NC5=O)CC4=C2)C3)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C51H44F4N8O11	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-YYP0NA	SCHEMBL30002798	N-[4-[7-[4-[3-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindole-5-carbonyl]-3,9-diazaspiro[5.5]undecan-9-yl]-4-oxobutoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide	COC1=C(OCCCC(=O)N2CCC3(CC2)CCN(C(=O)C2=CC=C4C(=O)N(C5CCC(=O)NC5=O)CC4=C2)CC3)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C55H52F4N8O11	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-M1J15I	SCHEMBL30001925	N-[4-[7-[4-[4-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]-2-oxoethyl]piperidin-1-yl]-4-oxobutoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide	COC1=C(OCCCC(=O)N2CCC(CC(=O)NC3=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)CC2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C52H48F4N8O11	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-AQ99J8	SCHEMBL24737823	N-[4-[7-[4-[4-[2-[[2-(2,6-dioxopiperidin-3-yl)-3-oxo-1H-isoindol-5-yl]amino]-2-oxoethyl]piperidin-1-yl]-4-oxobutoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide; SCHEMBL30002692	COC1=C(OCCCC(=O)N2CCC(CC(=O)NC3=CC4=C(C=C3)CN(C3CCC(=O)NC3=O)C4=O)CC2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C52H48F4N8O11	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-KGP3YE	SCHEMBL24737824	N-[4-[7-[4-[[4-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]carbamoyl]cyclohexyl]methylamino]-4-oxobutoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide; SCHEMBL30002080	COC1=C(OCCCC(=O)NCC2CCC(C(=O)NC3=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)CC2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C53H50F4N8O11	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-QTA3PX	SCHEMBL30002036	N-[4-[7-[1-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]acetyl]piperidin-4-yl]oxy-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide	COC1=C(OC2CCN(C(=O)CC3CCN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5)CC3)CC2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C53H50F4N8O10	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-SJVRFO	WO2022253283A1_110	N-[4-[7-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidine-4-carbonyl]piperidin-4-yl]oxy-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide	COC1=C(OC2CCN(C(=O)C3CCN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5)CC3)CC2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C52H48F4N8O10	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-BLCKHN	WO2022253283A1_111	N-[4-[7-[[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidine-4-carbonyl]piperidin-4-yl]methoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide	COC1=C(OCC2CCN(C(=O)C3CCN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5)CC3)CC2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C53H50F4N8O10	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-WX9QZJ	WO2022253283A1_112	N-[4-[7-[1-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]azetidin-3-yl]acetyl]piperidin-4-yl]oxy-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide	COC1=C(OC2CCN(C(=O)CC3CN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5)C3)CC2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C51H46F4N8O10	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-P4IF91	SCHEMBL30002094	N-[4-[7-[[1-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]azetidin-3-yl]acetyl]piperidin-4-yl]methoxy]-6-methoxyquinazolin-4-yl]oxy-3-fluorophenyl]-1,2-dimethyl-4-oxo-6-(trifluoromethoxy)quinoline-3-carboxamide	COC1=C(OCC2CCN(C(=O)CC3CN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5)C3)CC2)C=C2N=CN=C(OC3=C(F)C=C(NC(=O)C4=C(C)N(C)C5=C(C=C(OC(F)(F)F)C=C5)C4=O)C=C3)C2=C1	C52H48F4N8O10	AXL;FLT3	P30530/P36888	CRBN	WO-2022253283-A1
TPD-26585G	CHEMBL5270107	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[2-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyacetyl]amino]ethylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide; BDBM50615074	CC1(C)CCC(CN2CCN(c3ccc(C(=O)NS(=O)(=O)c4ccc(NCCNC(=O)COc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6=O)c([N+](=O)[O-])c4)c(Oc4cnc5[nH]ccc5c4)c3)CC2)=C(c2ccc(Cl)cc2)C1	C56H55ClN10O12S	BCL-2	P10415	CRBN	WO-2022266491-A1
TPD-Q1FSPC	CHEMBL5279723	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[2-[2-[2-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyacetyl]amino]ethoxy]ethoxy]ethylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide; BDBM50615075	CC1(C)CCC(CN2CCN(c3ccc(C(=O)NS(=O)(=O)c4ccc(NCCOCCOCCNC(=O)COc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6=O)c([N+](=O)[O-])c4)c(Oc4cnc5[nH]ccc5c4)c3)CC2)=C(c2ccc(Cl)cc2)C1	C60H63ClN10O14S	BCL-2	P10415	CRBN	WO-2022266491-A1
TPD-8D8KF9	CHEMBL5276934	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[2-[2-[2-[3-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyacetyl]amino]propanoylamino]ethoxy]ethoxy]ethylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide; BDBM50615073	CC1(C)CCC(CN2CCN(c3ccc(C(=O)NS(=O)(=O)c4ccc(NCCOCCOCCNC(=O)CCNC(=O)COc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6=O)c([N+](=O)[O-])c4)c(Oc4cnc5[nH]ccc5c4)c3)CC2)=C(c2ccc(Cl)cc2)C1	C63H68ClN11O15S	BCL-2	P10415	CRBN	WO-2022266491-A1
TPD-X774TC	CHEMBL5268884	(2R,3S,4R,5S)-3-(3-chloro-2-fluorophenyl)-4-(4-chloro-2-fluorophenyl)-N-[4-[2-[4-[[4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzoyl]sulfamoyl]-2-nitroanilino]ethylcarbamoyl]-2-methoxyphenyl]-4-cyano-5-(2,2-dimethylpropyl)pyrrolidine-2-carboxamide; BDBM50615072	COc1cc(C(=O)NCCNc2ccc(S(=O)(=O)NC(=O)c3ccc(N4CCN(CC5=C(c6ccc(Cl)cc6)CC(C)(C)CC5)CC4)cc3Oc3cnc4[nH]ccc4c3)cc2[N+](=O)[O-])ccc1NC(=O)[C@@H]1N[C@@H](CC(C)(C)C)[C@](C#N)(c2ccc(Cl)cc2F)[C@H]1c1cccc(Cl)c1F	C72H72Cl3F2N11O9S	BCL-2	P10415	VHL	WO-2022266491-A1
TPD-6E4V3J	CHEMBL5283597	(2R,3S,4R,5S)-3-(3-chloro-2-fluorophenyl)-4-(4-chloro-2-fluorophenyl)-N-[4-[2-[2-[2-[4-[[4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzoyl]sulfamoyl]-2-nitroanilino]ethoxy]ethoxy]ethylcarbamoyl]-2-methoxyphenyl]-4-cyano-5-(2,2-dimethylpropyl)pyrrolidine-2-carboxamide; BDBM50615076	COc1cc(C(=O)NCCOCCOCCNc2ccc(S(=O)(=O)NC(=O)c3ccc(N4CCN(CC5=C(c6ccc(Cl)cc6)CC(C)(C)CC5)CC4)cc3Oc3cnc4[nH]ccc4c3)cc2[N+](=O)[O-])ccc1NC(=O)[C@@H]1N[C@@H](CC(C)(C)C)[C@](C#N)(c2ccc(Cl)cc2F)[C@H]1c1cccc(Cl)c1F	C76H80Cl3F2N11O11S	BCL-2	P10415	VHL	WO-2022266491-A1
TPD-RZ36A0	WO2022266491A1_SF-8-150	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCC(=O)N2CCN(c3ccc(S(=O)(=O)NC(=O)c4ccc(N5CCN(CC6=C(c7ccc(Cl)cc7)CC(C)(C)CC6)CC5)cc4Oc4cnc5[nH]ccc5c4)cc3[N+](=O)[O-])CC2)C(C)(C)C)cc1	C69H79ClN12O11S2	BCL-2	P10415	VHL	WO-2022266491-A1
TPD-0W4KC1	WO2022266491A1_SF-8-156	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCC(=O)NCCC(=O)N2CCN(c3ccc(S(=O)(=O)NC(=O)c4ccc(N5CCN(CC6=C(c7ccc(Cl)cc7)CC(C)(C)CC6)CC5)cc4Oc4cnc5[nH]ccc5c4)cc3[N+](=O)[O-])CC2)C(C)(C)C)cc1	C72H84ClN13O12S2	BCL-2	P10415	VHL	WO-2022266491-A1
TPD-FA0DS3	WO2022266491A1_SF-8-157	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCC(=O)NCCCCCCC(=O)N2CCN(c3ccc(S(=O)(=O)NC(=O)c4ccc(N5CCN(CC6=C(c7ccc(Cl)cc7)CC(C)(C)CC6)CC5)cc4Oc4cnc5[nH]ccc5c4)cc3[N+](=O)[O-])CC2)C(C)(C)C)cc1	C76H92ClN13O12S2	BCL-2	P10415	VHL	WO-2022266491-A1
TPD-0V4VKA	SCHEMBL24953105	N-[2-[6-[7-[4-(dimethylcarbamoyl)-3-methylphenyl]-5H-pyrrolo[2,3-b]pyrazin-2-yl]-8-methyl-3,4-dihydro-1H-isoquinolin-2-yl]ethyl]-1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidine-4-carboxamide; SCHEMBL30215932	CC1=CC(C2=NC3=C(N=C2)NC=C3C2=CC(C)=C(C(=O)N(C)C)C=C2)=CC2=C1CN(CCNC(=O)C1CCN(C3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC1)CC2	C47H49N9O6	HPK1	Q92918	CRBN	WO-2023006063-A1
TPD-EAO44C	SCHEMBL24954315	4-[2-[2-[3-[[1-[4-(2,6-dioxopiperidin-3-yl)phenyl]piperidin-4-yl]methylamino]-3-oxopropyl]-8-methyl-3,4-dihydro-1H-isoquinolin-6-yl]-5H-pyrrolo[2,3-b]pyrazin-7-yl]-N,N,2-trimethylbenzamide	CC1=CC(C2=NC3=C(N=C2)NC=C3C2=CC(C)=C(C(=O)N(C)C)C=C2)=CC2=C1CN(CCC(=O)NCC1CCN(C3=CC=C(C4CCC(=O)NC4=O)C=C3)CC1)CC2	C46H52N8O4	HPK1	Q92918	CRBN	WO-2023006063-A1
TPD-BHL4W5	PROTAC HPK1 Degrader-2	PROTAC HPK1 Degrader-2; orb2564376; SCHEMBL24954314; HY-162544; CS-1097493; 2893885-31-7	CC1=CC(C2=NC3=C(N=C2)NC=C3C2=CC(C)=C(C(=O)N(C)C)C=C2)=CC2=C1CN(CCC(=O)N1CCN(C3=CC=C(N4CCC(=O)NC4=O)C=C3)CC1)CC2	C43H47N9O4	HPK1	Q92918	CRBN	WO-2023006063-A1
TPD-B3TKH2	SCHEMBL24953100	4-[2-[2-[3-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]amino]-3-oxopropyl]-8-methyl-3,4-dihydro-1H-isoquinolin-6-yl]-5H-pyrrolo[2,3-b]pyrazin-7-yl]-N,N,2-trimethylbenzamide	CC1=CC(C2=NC3=C(N=C2)NC=C3C2=CC(C)=C(C(=O)N(C)C)C=C2)=CC2=C1CN(CCC(=O)NC1CCN(C3=CC=C(N4CCC(=O)NC4=O)C=C3)CC1)CC2	C44H49N9O4	HPK1	Q92918	CRBN	WO-2023006063-A1
TPD-FR0RWM	SCHEMBL24954306	4-[2-[2-[3-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperazin-1-yl]-3-oxopropyl]-8-methyl-3,4-dihydro-1H-isoquinolin-6-yl]-5H-pyrrolo[2,3-b]pyrazin-7-yl]-N,N-dimethylbenzamide	CC1=C2CN(CCC(=O)N3CCN(C4=CC=C(N5CCC(=O)NC5=O)C=C4)CC3)CCC2=CC(C2=NC3=C(N=C2)NC=C3C2=CC=C(C(=O)N(C)C)C=C2)=C1	C42H45N9O4	HPK1	Q92918	CRBN	WO-2023006063-A1
TPD-1KMTZL	SCHEMBL24954304	4-[5-[2-[3-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperazin-1-yl]-3-oxopropyl]-8-methyl-3,4-dihydro-1H-isoquinolin-6-yl]-1H-pyrrolo[2,3-b]pyridin-3-yl]-N,N-dimethylbenzamide	CC1=C2CN(CCC(=O)N3CCN(C4=CC=C(N5CCC(=O)NC5=O)C=C4)CC3)CCC2=CC(C2=CC3=C(N=C2)NC=C3C2=CC=C(C(=O)N(C)C)C=C2)=C1	C43H46N8O4	HPK1	Q92918	CRBN	WO-2023006063-A1
TPD-4X399D	SCHEMBL24954307	4-[2-[2-[3-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperazin-1-yl]-3-oxopropyl]-8-methyl-3,4-dihydro-1H-isoquinolin-6-yl]-5H-pyrrolo[2,3-b]pyrazin-7-yl]-N-[(2S)-2-hydroxypropyl]-N-methylbenzamide; SCHEMBL30215927	CC1=CC(C2=NC3=C(N=C2)NC=C3C2=CC=C(C(=O)N(C)C[C@H](C)O)C=C2)=CC2=C1CN(CCC(=O)N1CCN(C3=CC=C(N4CCC(=O)NC4=O)C=C3)CC1)CC2	C44H49N9O5	HPK1	Q92918	CRBN	WO-2023006063-A1
TPD-W4G8X1	SCHEMBL24954308	4-[2-[2-[2-[[2-[1-[4-(2,6-dioxopiperidin-3-yl)phenyl]piperidin-4-yl]acetyl]amino]ethyl]-8-methyl-3,4-dihydro-1H-isoquinolin-6-yl]-5H-pyrrolo[2,3-b]pyrazin-7-yl]-N,N,2-trimethylbenzamide	CC1=CC(C2=NC3=C(N=C2)NC=C3C2=CC(C)=C(C(=O)N(C)C)C=C2)=CC2=C1CN(CCNC(=O)CC1CCN(C3=CC=C(C4CCC(=O)NC4=O)C=C3)CC1)CC2	C46H52N8O4	HPK1	Q92918	CRBN	WO-2023006063-A1
TPD-FH5650	SCHEMBL24954305	4-[5-[2-[3-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperazin-1-yl]-3-oxopropyl]-8-methyl-3,4-dihydro-1H-isoquinolin-6-yl]-1H-pyrrolo[2,3-b]pyridin-3-yl]-N-[(2S)-2-hydroxypropyl]-N-methylbenzamide; SCHEMBL30215946	CC1=CC(C2=CC3=C(N=C2)NC=C3C2=CC=C(C(=O)N(C)C[C@H](C)O)C=C2)=CC2=C1CN(CCC(=O)N1CCN(C3=CC=C(N4CCC(=O)NC4=O)C=C3)CC1)CC2	C45H50N8O5	HPK1	Q92918	CRBN	WO-2023006063-A1
TPD-KG07G6	WO2023039081A2_1	.	CC(=O)C1=C(C)C2=C(N=C(NC3=NC=C(N4CCN(CC5CCCN(C6=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)C5)CC4)C=C3)N=C2)N(C2CCCC2)C1=O	C43H48N10O6	CDK4;CDK6	P11802/Q00534	CRBN	WO-2023039081-A2
TPD-BFBAU4	WO2023039081A2_2	.	CC(=O)C1=C(C)C2=C(N=C(NC3=NC=C(N4CCN(CC5(C)CCN(C6=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)CC5)CC4)C=C3)N=C2)N(C2CCCC2)C1=O	C44H50N10O6	CDK4;CDK6	P11802/Q00534	CRBN	WO-2023039081-A2
TPD-702MP5	WO2023039081A2_3	4-[3-[[4-[6-[(6-Acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]methyl]pyrrolidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CC(=O)C1=C(C)C2=C(N=C(NC3=NC=C(N4CCN(CC5CCN(C6=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)C5)CC4)C=C3)N=C2)N(C2CCCC2)C1=O	C42H46N10O6	CDK4;CDK6	P11802/Q00534	CRBN	WO-2023039081-A2
TPD-BSLOKW	SCHEMBL30338562	4-[[3-[2-[4-[6-[(6-Acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]ethyl]cyclobutyl]methylamino]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CC(=O)C1=C(C)C2=C(N=C(NC3=NC=C(N4CCN(CCC5CC(CNC6=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)C5)CC4)C=C3)N=C2)N(C2CCCC2)C1=O	C44H50N10O6	CDK4;CDK6	P11802/Q00534	CRBN	WO-2023039081-A2
TPD-YBTCKF	WO2023039081A2_5	.	CC(=O)C1=C(C)C2=C(N=C(NC3=NC=C(N4CCN(CCC5CCCCN5C5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)CC4)C=C3)N=C2)N(C2CCCC2)C1=O	C44H50N10O6	CDK4;CDK6	P11802/Q00534	CRBN	WO-2023039081-A2
TPD-HYZ1J4	WO2023039081A2_6	.	CC(=O)C1=C(C)C2=C(N=C(NC3=NC=C(N4CCN(CCCC5CCN(C6=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)CC5)CC4)C=C3)N=C2)N(C2CCCC2)C1=O	C45H52N10O6	CDK4;CDK6	P11802/Q00534	CRBN	WO-2023039081-A2
TPD-WYNU2V	SCHEMBL30339069	4-[4-[2-[4-[6-[(6-Acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]ethyl]piperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CC(=O)C1=C(C)C2=C(N=C(NC3=NC=C(N4CCN(CCC5CCN(C6=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)CC5)CC4)C=C3)N=C2)N(C2CCCC2)C1=O	C44H50N10O6	CDK4;CDK6	P11802/Q00534	CRBN	WO-2023039081-A2
TPD-MP534J	SCHEMBL30338413	5-[3-[[4-[6-[(6-Acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]methyl]piperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CC(=O)C1=C(C)C2=CN=C(NC3=NC=C(N4CCN(CC5CCCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C3)N=C2N(C2CCCC2)C1=O	C43H48N10O6	CDK4;CDK6	P11802/Q00534	CRBN	WO-2023039081-A2
TPD-B1EI9G	SCHEMBL25403625	5-[4-[2-[4-[6-[(6-Acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]ethyl]piperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CC(=O)C1=C(C)C2=C(N=C(NC3=NC=C(N4CCN(CCC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C=C3)N=C2)N(C2CCCC2)C1=O	C44H50N10O6	CDK4;CDK6	P11802/Q00534	CRBN	WO-2023039081-A2
TPD-M97AYN	WO2023039081A2_10	.	CC(=O)C1=C(C)C2=C(N=C(NC3=NC=C(N4CCN(CCC5CCCCN5C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)C=C3)N=C2)N(C2CCCC2)C1=O	C44H50N10O6	CDK4;CDK6	P11802/Q00534	CRBN	WO-2023039081-A2
TPD-VJ587W	WO2023039081A2_11	.	CC(=O)C1=C(C)C2=C(N=C(NC3=NC=C(N4CCN(CC5(C)CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C=C3)N=C2)N(C2CCCC2)C1=O	C44H50N10O6	CDK4;CDK6	P11802/Q00534	CRBN	WO-2023039081-A2
TPD-0X71BM	WO2023039081A2_12	.	CC(=O)C1=C(C)C2=CN=C(NC3=NC=C(N4CCN(C[C@@H]5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C3)N=C2N(C2CCCC2)C1=O	C42H46N10O6	CDK4;CDK6	P11802/Q00534	CRBN	WO-2023039081-A2
TPD-FXW6BK	WO2023039081A2_13	.	CC(=O)C1=C(C)C2=CN=C(NC3=NC=C(N4CCN(C[C@H]5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C3)N=C2N(C2CCCC2)C1=O	C42H46N10O6	CDK4;CDK6	P11802/Q00534	CRBN	WO-2023039081-A2
TPD-66RLD4	WO2023039081A2_14	.	CC(=O)C1=C(C)C2=CN=C(NC3=NC=C(N4CCN(C[C@@H]5CCN(C6=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)C5)CC4)C=C3)N=C2N(C2CCCC2)C1=O	C42H46N10O6	CDK4;CDK6	P11802/Q00534	CRBN	WO-2023039081-A2
TPD-9TH4TX	WO2023039081A2_15	.	CC(=O)C1=C(C)C2=CN=C(NC3=NC=C(N4CCN(C[C@H]5CCN(C6=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)C5)CC4)C=C3)N=C2N(C2CCCC2)C1=O	C42H46N10O6	CDK4;CDK6	P11802/Q00534	CRBN	WO-2023039081-A2
TPD-4AZVIH	WO2023039081A2_16	.	CC(=O)C1=C(C)C2=CN=C(NC3=NC=C(N4CCN(CC5CCCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C=C3)N=C2N(C2CCCC2)C1=O	C44H50N10O6	CDK4;CDK6	P11802/Q00534	CRBN	WO-2023039081-A2
TPD-CSJK88	WO2023039081A2_17	.	CC(=O)C1=C(C)C2=CN=C(NC3=NC=C(N4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)N(C)C8=O)C(=O)C7=C6)CC5)CC4)C=C3)N=C2N(C2CCCC2)C1=O	C44H50N10O6	CDK4;CDK6	P11802/Q00534	CRBN	WO-2023039081-A2
TPD-RPPS9O	SCHEMBL25401799	4-[4-[[4-[6-[(6-Acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]methyl]piperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione; SCHEMBL30672763	CC(=O)C1=C(C)C2=CN=C(NC3=NC=C(N4CCN(CC5CCN(C6=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)CC5)CC4)C=C3)N=C2N(C2CCCC2)C1=O	C43H48N10O6	CDK4;CDK6	P11802/Q00534	CRBN	WO-2023039081-A2
TPD-0EPB5P	WO2023039081A2_19	.	CC(=O)C1=C(C)C2=CN=C(NC3=NC=C(N4CCN(CC5(F)CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C=C3)N=C2N(C2CCCC2)C1=O	C43H47FN10O6	CDK4;CDK6	P11802/Q00534	CRBN	WO-2023039081-A2
TPD-S9DMA1	SCHEMBL25403511	3-[6-[4-[[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CC(=O)C1=C(C)C2=CN=C(NC3=NC=C(N4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)CC5)CC4)C=C3)N=C2N(C2CCCC2)C1=O	C43H50N10O5	CDK4;CDK6	P11802/Q00534	CRBN	WO-2023039081-A2
TPD-Y9NRCC	WO2023039081A2_21	.	CC(=O)C1=C(C)C2=CN=C(NC3=NC=C(N4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)N(C)C8=O)C(=O)C7=C6)CC5(F)F)CC4)C=C3)N=C2N(C2CCCC2)C1=O	C44H48F2N10O6	CDK4;CDK6	P11802/Q00534	CRBN	WO-2023039081-A2
TPD-HUGDNU	WO2023039081A2_22	.	CC(=O)C1=C(C)C2=CN=C(NC3=NC=C(N4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5(F)F)CC4)C=C3)N=C2N(C2CCCC2)C1=O	C43H46F2N10O6	CDK4;CDK6	P11802/Q00534	CRBN	WO-2023039081-A2
TPD-5NLOBS	WO2023039081A2_23	.	CC(=O)C1=C(C)C2=CN=C(NC3=NC=C(N4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5F)CC4)C=C3)N=C2N(C2CCCC2)C1=O	C43H47FN10O6	CDK4;CDK6	P11802/Q00534	CRBN	WO-2023039081-A2
TPD-SV24B6	WO2023039081A2_25	.	CC(=O)C1=C(C)C2=CN=C(NC3=NC=C(N4CCN(CC5(F)CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C3)N=C2N(C2CCCC2)C1=O	C42H45FN10O6	CDK4;CDK6	P11802/Q00534	CRBN	WO-2023039081-A2
TPD-6UQ8ZX	WO2023039081A2_26	.	CC(=O)C1=C(C)C2=CN=C(NC3=NC=C(N4CCN(CC5CCCN(C6=CC=C7C(=O)N(C8CCC(=O)N(C)C8=O)C(=O)C7=C6)CC5)CC4)C=C3)N=C2N(C2CCCC2)C1=O	C45H52N10O6	CDK4;CDK6	P11802/Q00534	CRBN	WO-2023039081-A2
TPD-KI2IWN	SCHEMBL21635227	N-[3-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]propyl]-2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyacetamide; SCHEMBL30338600; PD142094	CC(=O)C1=C(C)C2=CN=C(NC3=NC=C(N4CCN(CCCNC(=O)COC5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)CC4)C=C3)N=C2N(C2CCCC2)C1=O	C42H46N10O8	CDK4;CDK6	P11802/Q00534	CRBN	WO-2023039081-A2
TPD-XGRKMK	CHEMBL5415770	5-[4-[[4-[6-[(6-Acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]methyl]piperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione; SCHEMBL25403182	CC(=O)C1=C(C)C2=CN=C(NC3=NC=C(N4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C=C3)N=C2N(C2CCCC2)C1=O	C43H48N10O6	CDK4;CDK6	P11802/Q00534	CRBN	WO-2023039081-A2
TPD-FQAXS8	SCHEMBL25403271	5-[3-[[4-[6-[(6-Acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]methyl]azetidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CC(=O)C1=C(C)C2=CN=C(NC3=NC=C(N4CCN(CC5CN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C3)N=C2N(C2CCCC2)C1=O	C41H44N10O6	CDK4;CDK6	P11802/Q00534	CRBN	WO-2023039081-A2
TPD-PVNBXK	WO2023039081A2_33	.	CC(=O)C1=C(C)C2=CN=C(NC3=NC=C(N4CCN(CC(=O)NCCOCCOCCOCCC(=O)NC(C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=C(C)N=CS6)C=C5)C(C)(C)C)CC4)C=C3)N=C2N(C2CCCC2)C1=O	C58H78N12O10S	CDK4;CDK6	P11802/Q00534	VHL	WO-2023039081-A2
TPD-5VYGP2	WO2023039081A2_34	.	CC(=O)C1=C(C)C2=CN=C(NC3=NC=C(N4CCN(CCCCC(=O)NC(C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=C(C)N=CS6)C=C5)C(C)(C)C)CC4)C=C3)N=C2N(C2CCCC2)C1=O	C52H67N11O6S	CDK4;CDK6	P11802/Q00534	VHL	WO-2023039081-A2
TPD-8W9X2M	WO2023039081A2_35	.	CC(=O)C1=C(C)C2=CN=C(NC3=NC=C(N4CCN(CCCC(=O)NC(C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=C(C)N=CS6)C=C5)C(C)(C)C)CC4)C=C3)N=C2N(C2CCCC2)C1=O	C51H65N11O6S	CDK4;CDK6	P11802/Q00534	VHL	WO-2023039081-A2
TPD-WVVYQ4	WO2023039081A2_36	.	CC(=O)C1=C(C)C2=CN=C(NC3=NC=C(N4CCN(CCCCC(=O)NC(C(=O)N5C[C@@H](O)CC5C(=O)N[C@@H](C)C5=CC=C(C6=C(C)N=CS6)C=C5)C(C)(C)C)CC4)C=C3)N=C2N(C2CCCC2)C1=O	C52H67N11O6S	CDK4;CDK6	P11802/Q00534	VHL	WO-2023039081-A2
TPD-U0QN7V	SCHEMBL30291287	2-[2,3-difluoro-6-(2-morpholin-4-yl-1,3-thiazol-4-yl)phenoxy]-N-[4-[[3-(2,6-dioxopiperidin-3-yl)-4-oxo-1,2,3-benzotriazin-6-yl]amino]butyl]acetamide	O=C(COc1c(-c2csc(N3CCOCC3)n2)ccc(F)c1F)NCCCCNc1ccc2nnn(C3CCC(=O)NC3=O)c(=O)c2c1	C31H32F2N8O6S	AR-V7	P10275-3	CRBN	WO-2023039603-A2
TPD-MBAR2Z	SCHEMBL30291423	2-[2,3-difluoro-6-(2-morpholin-4-yl-1,3-thiazol-4-yl)phenoxy]-N-[6-[[3-(2,6-dioxopiperidin-3-yl)-4-oxo-1,2,3-benzotriazin-6-yl]amino]hexyl]acetamide	O=C(COc1c(-c2csc(N3CCOCC3)n2)ccc(F)c1F)NCCCCCCNc1ccc2nnn(C3CCC(=O)NC3=O)c(=O)c2c1	C33H36F2N8O6S	AR-V7	P10275-3	CRBN	WO-2023039603-A2
TPD-GBVHHR	SCHEMBL30291245	3-[6-[2-[2-[2-[2,3-Difluoro-6-(2-morpholin-4-yl-1,3-thiazol-4-yl)phenoxy]ethoxy]ethoxy]ethylamino]-4-oxo-1,2,3-benzotriazin-3-yl]piperidine-2,6-dione	O=C1CCC(n2nnc3ccc(NCCOCCOCCOc4c(-c5csc(N6CCOCC6)n5)ccc(F)c4F)cc3c2=O)C(=O)N1	C31H33F2N7O7S	AR-V7	P10275-3	CRBN	WO-2023039603-A2
TPD-70NS3Y	SCHEMBL30291298	2-[2,3-difluoro-6-(2-morpholin-4-yl-1,3-thiazol-4-yl)phenoxy]-N-[10-[[3-(2,6-dioxopiperidin-3-yl)-4-oxo-1,2,3-benzotriazin-6-yl]amino]decyl]acetamide	O=C(COc1c(-c2csc(N3CCOCC3)n2)ccc(F)c1F)NCCCCCCCCCCNc1ccc2nnn(C3CCC(=O)NC3=O)c(=O)c2c1	C37H44F2N8O6S	AR-V7	P10275-3	CRBN	WO-2023039603-A2
TPD-R04CDL	SCHEMBL31142843	3-[6-[2-[2-[2-[2-[2,3-Difluoro-6-(2-morpholin-4-yl-1,3-thiazol-4-yl)phenoxy]ethoxy]ethoxy]ethoxy]ethylamino]-4-oxo-1,2,3-benzotriazin-3-yl]piperidine-2,6-dione	O=C1CCC(n2nnc3ccc(NCCOCCOCCOCCOc4c(-c5csc(N6CCOCC6)n5)ccc(F)c4F)cc3c2=O)C(=O)N1	C33H37F2N7O8S	AR-V7	P10275-3	CRBN	WO-2023039603-A2
TPD-1JL9NN	SCHEMBL31142834	3-[6-[2-[2-[2-[2-[2-[2,3-Difluoro-6-(2-morpholin-4-yl-1,3-thiazol-4-yl)phenoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethylamino]-4-oxo-1,2,3-benzotriazin-3-yl]piperidine-2,6-dione	O=C1CCC(n2nnc3ccc(NCCOCCOCCOCCOCCOc4c(-c5csc(N6CCOCC6)n5)ccc(F)c4F)cc3c2=O)C(=O)N1	C35H41F2N7O9S	AR-V7	P10275-3	CRBN	WO-2023039603-A2
TPD-4017JC	WO2023039603A2_7	.	O=C1CCC(n2nnc3ccc(NCCCCCCCNCCCCCOc4c(-c5csc(N6CCOCC6)n5)ccc(F)c4F)cc3c2=O)C(=O)N1	C37H46F2N8O5S	AR-V7	P10275-3	CRBN	WO-2023039603-A2
TPD-8PI103	SCHEMBL31142808	3-[6-[8-[5-[2,3-Difluoro-6-(2-morpholin-4-yl-1,3-thiazol-4-yl)phenoxy]pentylamino]octylamino]-4-oxo-1,2,3-benzotriazin-3-yl]piperidine-2,6-dione	O=C1CCC(n2nnc3ccc(NCCCCCCCCNCCCCCOc4c(-c5csc(N6CCOCC6)n5)ccc(F)c4F)cc3c2=O)C(=O)N1	C38H48F2N8O5S	AR-V7	P10275-3	CRBN	WO-2023039603-A2
TPD-VY03T7	WO2023039603A2_9	.	O=C1CCC(n2nnc3ccc(NCCCCCCCCCNCCCCOc4c(-c5csc(N6CCOCC6)n5)ccc(F)c4F)cc3c2=O)C(=O)N1	C38H48F2N8O5S	AR-V7	P10275-3	CRBN	WO-2023039603-A2
TPD-F1KWNT	SCHEMBL31142796	3-[6-[8-[2-[2,3-Difluoro-6-(2-morpholin-4-yl-1,3-thiazol-4-yl)phenoxy]ethylamino]octylamino]-4-oxo-1,2,3-benzotriazin-3-yl]piperidine-2,6-dione	O=C1CCC(n2nnc3ccc(NCCCCCCCCNCCOc4c(-c5csc(N6CCOCC6)n5)ccc(F)c4F)cc3c2=O)C(=O)N1	C35H42F2N8O5S	AR-V7	P10275-3	CRBN	WO-2023039603-A2
TPD-8PV8YO	SCHEMBL31142798	3-[6-[10-[2-[2,3-Difluoro-6-(2-morpholin-4-yl-1,3-thiazol-4-yl)phenoxy]ethylamino]decylamino]-4-oxo-1,2,3-benzotriazin-3-yl]piperidine-2,6-dione	O=C1CCC(n2nnc3ccc(NCCCCCCCCCCNCCOc4c(-c5csc(N6CCOCC6)n5)ccc(F)c4F)cc3c2=O)C(=O)N1	C37H46F2N8O5S	AR-V7	P10275-3	CRBN	WO-2023039603-A2
TPD-U9BYNW	SCHEMBL31142807	2-[2,3-difluoro-6-[2-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)-1,3-thiazol-4-yl]phenoxy]-N-[6-[[3-(2,6-dioxopiperidin-3-yl)-4-oxo-1,2,3-benzotriazin-6-yl]amino]hexyl]acetamide	O=C(COc1c(-c2csc(N3CC4CCC(C3)O4)n2)ccc(F)c1F)NCCCCCCNc1ccc2nnn(C3CCC(=O)NC3=O)c(=O)c2c1	C35H38F2N8O6S	AR-V7	P10275-3	CRBN	WO-2023039603-A2
TPD-U1QHPV	SCHEMBL31142820	2-[2,3-difluoro-6-[2-(3-oxa-8-azabicyclo[3.2.1]octan-8-yl)-1,3-thiazol-4-yl]phenoxy]-N-[6-[[3-(2,6-dioxopiperidin-3-yl)-4-oxo-1,2,3-benzotriazin-6-yl]amino]hexyl]acetamide	O=C(COc1c(-c2csc(N3C4CCC3COC4)n2)ccc(F)c1F)NCCCCCCNc1ccc2nnn(C3CCC(=O)NC3=O)c(=O)c2c1	C35H38F2N8O6S	AR-V7	P10275-3	CRBN	WO-2023039603-A2
TPD-N3VDJT	SCHEMBL31142809	3-[6-[2-[4-[2-[2,3-Difluoro-6-(2-morpholin-4-yl-1,3-thiazol-4-yl)phenoxy]acetyl]piperazin-1-yl]ethylamino]-4-oxo-1,2,3-benzotriazin-3-yl]piperidine-2,6-dione	O=C1CCC(n2nnc3ccc(NCCN4CCN(C(=O)COc5c(-c6csc(N7CCOCC7)n6)ccc(F)c5F)CC4)cc3c2=O)C(=O)N1	C33H35F2N9O6S	AR-V7	P10275-3	CRBN	WO-2023039603-A2
TPD-O6YWVA	SCHEMBL31142816	2-[2,3-difluoro-6-(2-morpholin-4-yl-1,3-thiazol-4-yl)phenoxy]-N-[1-[4-[[3-(2,6-dioxopiperidin-3-yl)-4-oxo-1,2,3-benzotriazin-6-yl]amino]butanoyl]piperidin-3-yl]acetamide	O=C1CCC(n2nnc3ccc(NCCCC(=O)N4CCCC(NC(=O)COc5c(-c6csc(N7CCOCC7)n6)ccc(F)c5F)C4)cc3c2=O)C(=O)N1	C36H39F2N9O7S	AR-V7	P10275-3	CRBN	WO-2023039603-A2
TPD-P5O2V4	SCHEMBL31142803	3-[6-[4-[5-[2-[2,3-Difluoro-6-(2-morpholin-4-yl-1,3-thiazol-4-yl)phenoxy]ethyl]triazol-1-yl]butylamino]-4-oxo-1,2,3-benzotriazin-3-yl]piperidine-2,6-dione	O=C1CCC(n2nnc3ccc(NCCCCn4nncc4CCOc4c(-c5csc(N6CCOCC6)n5)ccc(F)c4F)cc3c2=O)C(=O)N1	C33H34F2N10O5S	AR-V7	P10275-3	CRBN	WO-2023039603-A2
TPD-PHKA2S	SCHEMBL31142805	N-[3-[2,3-difluoro-6-(2-morpholin-4-yl-1,3-thiazol-4-yl)phenoxy]cyclobutyl]-4-[[3-(2,6-dioxopiperidin-3-yl)-4-oxo-1,2,3-benzotriazin-6-yl]amino]butanamide	O=C1CCC(n2nnc3ccc(NCCCC(=O)N[C@H]4C[C@H](Oc5c(-c6csc(N7CCOCC7)n6)ccc(F)c5F)C4)cc3c2=O)C(=O)N1	C33H34F2N8O6S	AR-V7	P10275-3	CRBN	WO-2023039603-A2
TPD-FN69NU	WO2023045978A1_1	2-[2-(cyclopropylmethylamino)pyridin-4-yl]-N-[3-(difluoromethyl)-1-[4-[[4-[2-[[3-(2,6-dioxopiperidin-3-yl)-1-benzofuran-5-yl]amino]-2-oxoethyl]piperazin-1-yl]methyl]cyclohexyl]pyrazol-4-yl]-1,3-oxazole-4-carboxamide	O=C1CCC(c2coc3ccc(NC(=O)CN4CCN(C[C@H]5CC[C@H](n6cc(NC(=O)c7coc(-c8ccnc(NCC9CC9)c8)n7)c(C(F)F)n6)CC5)CC4)cc23)C(=O)N1	C43H48F2N10O6	IRAK4	Q9NWZ3	CRBN	WO-2023045978-A1
TPD-MWCE6Q	WO2023045978A1_2	.	O=C1CCC(c2coc3cc(NC(=O)CN4CCN(C[C@H]5CC[C@H](n6cc(NC(=O)c7coc(-c8ccnc(NCC9CC9)c8)n7)c(C(F)F)n6)CC5)CC4)ccc23)C(=O)N1	C43H48F2N10O6	IRAK4	Q9NWZ3	CRBN	WO-2023045978-A1
TPD-ALMY1U	WO2023045978A1_4	.	CN(CCCOCCCc1ccc2occ(C3CCC(=O)NC3=O)c2c1)C[C@H]1CC[C@H](N2C=C(NC(=O)c3coc(-c4ccnc(NCC5CC5)c4)n3)C(C(F)F)N2)CC1	C44H54F2N8O6	IRAK4	Q9NWZ3	CRBN	WO-2023045978-A1
TPD-DKV4EK	WO2023045978A1_7	.	O=C1CCC(C2=CCc3ccc4cc(NC(=O)CN5CCN(C[C@H]6CC[C@H](n7cc(NC(=O)c8coc(-c9ccnc(NCC%10CC%10)c9)n8)c(C(F)F)n7)CC6)CC5)ccc4c32)C(=O)N1	C48H52F2N10O5	IRAK4	Q9NWZ3	CRBN	WO-2023045978-A1
TPD-5Q1MKT	WO2023045978A1_8	.	CN(CCCOCCCc1ccc2c(ccc3occ(C4CCC(=O)NC4=O)c32)c1)C[C@H]1CC[C@H](N2C=C(NC(=O)c3coc(-c4ccnc(NCC5CC5)c4)n3)C(C(F)F)N2)CC1	C48H56F2N8O6	IRAK4	Q9NWZ3	CRBN	WO-2023045978-A1
TPD-2R3DF6	WO2023045978A1_10	.	CN(CCCOCCCc1cccc2c1ccc1occ(C3CCC(=O)NC3=O)c12)C[C@H]1CC[C@H](n2cc(NC(=O)c3coc(-c4ccnc(NCC5CC5)c4)n3)c(C(F)F)n2)CC1	C48H54F2N8O6	IRAK4	Q9NWZ3	CRBN	WO-2023045978-A1
TPD-51ZWFR	WO2023045978A1_11	.	O=C1CCC(c2coc3ccc4c(NC(=O)CN5CCN(C[C@H]6CC[C@H](n7cc(NC(=O)c8coc(-c9ccnc(NCC%10CC%10)c9)n8)c(C(F)F)n7)CC6)CC5)cccc4c23)C(=O)N1	C47H50F2N10O6	IRAK4	Q9NWZ3	CRBN	WO-2023045978-A1
TPD-GWW5I3	WO2023045978A1_13	.	CN(CCCOCCCc1cccc2c1ccc1onc(C3CCC(=O)NC3=O)c12)C[C@H]1CC[C@H](n2cc(NC(=O)c3coc(-c4ccnc(NCC5CC5)c4)n3)c(C(F)F)n2)CC1	C47H53F2N9O6	IRAK4	Q9NWZ3	CRBN	WO-2023045978-A1
TPD-OVD6IG	WO2023045978A1_14	2-[2-(cyclopropylmethylamino)pyridin-4-yl]-N-[3-(difluoromethyl)-1-[4-[[4-[2-[[1-(2,6-dioxopiperidin-3-yl)benzo[e][1,2]benzoxazol-6-yl]amino]-2-oxoethyl]piperazin-1-yl]methyl]cyclohexyl]pyrazol-4-yl]-1,3-oxazole-4-carboxamide	O=C1CCC(c2noc3ccc4c(NC(=O)CN5CCN(C[C@H]6CC[C@H](n7cc(NC(=O)c8coc(-c9ccnc(NCC%10CC%10)c9)n8)c(C(F)F)n7)CC6)CC5)cccc4c23)C(=O)N1	C46H49F2N11O6	IRAK4	Q9NWZ3	CRBN	WO-2023045978-A1
TPD-IANANS	WO2023045978A1_15	.	O=C1CCC(c2noc3ccc4cc(NC(=O)CN5CCN(C[C@H]6CC[C@H](n7cc(NC(=O)c8coc(-c9ccnc(NCC%10CC%10)c9)n8)c(C(F)F)n7)CC6)CC5)ccc4c23)C(=O)N1	C46H49F2N11O6	IRAK4	Q9NWZ3	CRBN	WO-2023045978-A1
TPD-VE74ZR	WO2023045978A1_16	.	CN(CCCOCCCc1ccc2c(ccc3onc(C4CCC(=O)NC4=O)c32)c1)C[C@H]1CC[C@H](n2cc(NC(=O)c3coc(-c4ccnc(NCC5CC5)c4)n3)c(C(F)F)n2)CC1	C47H53F2N9O6	IRAK4	Q9NWZ3	CRBN	WO-2023045978-A1
TPD-EAJUJA	WO2023045978A1_17	.	CC(C)(O)c1cc2nc([C@H]3CC[C@H](CN4CCN(CC(=O)Nc5cccc6c5ccc5onc(C7CCC(=O)NC7=O)c56)CC4)CC3)sc2cc1NC(=O)c1cccc(C(F)(F)F)n1	C46H47F3N8O6S	IRAK4	Q9NWZ3	CRBN	WO-2023045978-A1
TPD-NUOUQ2	WO2023045978A1_18	.	O=C1CCC(c2noc3ccc4c(NC(=O)C(F)(F)C5CCN(C[C@H]6CC[C@H](n7cc(NC(=O)c8coc(-c9ccnc(NCC%10CC%10)c9)n8)c(C(F)F)n7)CC6)CC5)cccc4c23)C(=O)N1	C47H48F4N10O6	IRAK4	Q9NWZ3	CRBN	WO-2023045978-A1
TPD-G3KLMG	WO2023045978A1_19	N-[2-[4-[[4-[2-[[1-(2,6-dioxopiperidin-3-yl)benzo[e][1,2]benzoxazol-6-yl]amino]-1,1-difluoro-2-oxoethyl]piperidin-1-yl]methyl]cyclohexyl]-5-(2-hydroxypropan-2-yl)-1,3-benzothiazol-6-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	CC(C)(O)c1cc2nc([C@H]3CC[C@H](CN4CCC(C(F)(F)C(=O)Nc5cccc6c5ccc5onc(C7CCC(=O)NC7=O)c56)CC4)CC3)sc2cc1NC(=O)c1cccc(C(F)(F)F)n1	C47H46F5N7O6S	IRAK4	Q9NWZ3	CRBN	WO-2023045978-A1
TPD-KVQXDU	WO2023045978A1_20	.	CC(C)(O)c1cc2c(cc1NC(=O)c1cccc(C(F)(F)F)n1)SC([C@H]1CC[C@H](CN3CCN(CC(=O)Nc4ccc5c(ccc6onc(C7CCC(=O)NC7=O)c65)c4)CC3)CC1)N2	C46H49F3N8O6S	IRAK4	Q9NWZ3	CRBN	WO-2023045978-A1
TPD-OAXDJU	WO2023045978A1_21	.	CNC(c1c(O)ccc2cc(NCCC3CC4(C3)CN(C[C@H]3CC[C@H](c5nc6cc(C(C)(C)O)c(NC(=O)c7cccc(C(F)(F)F)n7)cc6s5)CC3)C4)ccc12)C1CCC(=O)NC1=O	C49H56F3N7O5S	IRAK4	Q9NWZ3	CRBN	WO-2023045978-A1
TPD-6E08RN	WO2023045978A1_23	N-[2-[4-[[4-[2-[[3-(2,6-dioxopiperidin-3-yl)-1,2-benzoxazol-7-yl]amino]-1,1-difluoro-2-oxoethyl]piperidin-1-yl]methyl]cyclohexyl]-5-(2-hydroxypropan-2-yl)-1,3-benzothiazol-6-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	CC(C)(O)c1cc2nc([C@H]3CC[C@H](CN4CCC(C(F)(F)C(=O)Nc5cccc6c(C7CCC(=O)NC7=O)noc56)CC4)CC3)sc2cc1NC(=O)c1cccc(C(F)(F)F)n1	C43H44F5N7O6S	IRAK4	Q9NWZ3	CRBN	WO-2023045978-A1
TPD-DEAYNW	WO2023045978A1_24	.	CN(/C=C(/NC(=O)c1coc(-c2ccnc(NCC3CC3)c2)n1)C(=N)C(F)F)[C@H]1CC[C@H](CN2CCC(C(F)(F)C(=O)Nc3cccc4c(C5CCC(=O)NC5=O)noc34)CC2)CC1	C44H50F4N10O6	IRAK4	Q9NWZ3	CRBN	WO-2023045978-A1
TPD-CG7KXQ	WO2023045978A1_25	.	CC(F)c1nn([C@H]2CC[C@H](CN3CCN(CC(=O)Nc4ccc5c(C6CCC(=O)NC6=O)noc5c4)CC3)CC2)cc1NC(=O)c1coc(-c2ccnc(NCC3CC3)c2)c1	C44H51FN10O6	IRAK4	Q9NWZ3	CRBN	WO-2023045978-A1
TPD-17C4OW	WO2023045978A1_26	.	CC(C)(O)c1cc2nc([C@H]3CC[C@H](CN4CCN(CC(=O)Nc5ccc6c(C7CCC(=O)NC7=O)noc6c5)CC4)CC3)sc2cc1NC(=O)c1cccc(C(F)(F)F)n1	C42H45F3N8O6S	IRAK4	Q9NWZ3	CRBN	WO-2023045978-A1
TPD-GOSO2T	WO2023045978A1_28	.	O=C1CCC(c2noc3c(NC(=O)CN4CCN(C[C@H]5CC[C@H](N6C=C(NC(=O)c7coc(-c8ccnc(NCC9CC9)c8)n7)C(C(F)F)N6)CC5)CC4)cccc23)C(=O)N1	C42H49F2N11O6	IRAK4	Q9NWZ3	CRBN	WO-2023045978-A1
TPD-4713ZU	WO2023045978A1_29	N-[2-[4-[[4-[2-[[3-(2,6-dioxopiperidin-3-yl)-1,2-benzoxazol-7-yl]amino]-2-oxoethyl]piperazin-1-yl]methyl]cyclohexyl]-5-(2-hydroxypropan-2-yl)-1,3-benzothiazol-6-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	CC(C)(O)c1cc2nc([C@H]3CC[C@H](CN4CCN(CC(=O)Nc5cccc6c(C7CCC(=O)NC7=O)noc56)CC4)CC3)sc2cc1NC(=O)c1cccc(C(F)(F)F)n1	C42H45F3N8O6S	IRAK4	Q9NWZ3	CRBN	WO-2023045978-A1
TPD-Y0ZLJN	WO2023045978A1_30	.	O=C1CC[C@H](c2noc3ccc4c(NC(=O)CN5CCN(C[C@H]6CC[C@H](n7cc(NC(=O)c8coc(-c9ccnc(NCC%10CC%10)c9)n8)c(C(F)F)n7)CC6)CC5)cccc4c23)C(=O)N1	C46H49F2N11O6	IRAK4	Q9NWZ3	CRBN	WO-2023045978-A1
TPD-GS7WPR	WO2023045978A1_31	.	O=C1CC[C@@H](C2NOc3ccc4c(NC(=O)CN5CCN(CC6CCC(n7cc(NC(=O)C8=COC(c9ccnc(NCC%10CC%10)c9)N8)c(C(F)F)n7)CC6)CC5)cccc4c32)C(=O)N1	C46H53F2N11O6	IRAK4	Q9NWZ3	CRBN	WO-2023045978-A1
TPD-RVPLQG	CHEMBL5416036	2-cyclopentyl-4-[7-[11-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-11-oxoundecoxy]quinazolin-4-yl]benzoic acid; SCHEMBL31513492; BDBM50631197; PD216520	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCCCCCOc2ccc3c(-c4ccc(C(=O)O)c(C5CCCC5)c4)ncnc3c2)C(C)(C)C)cc1	C53H66N6O7S	CAMKK2	Q96RR4	VHL	WO-2023059873-A1
TPD-5QEL39	2922675-91-8	2-cyclopentyl-4-{7-[(9-{[(2S)-1-[(2S,4R)-4-hydroxy-2-({[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl}carbamoyl)pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]carbamoyl}nonyl)oxy]quinazolin-4-yl}benzoic acid; 2-cyclopentyl-4-(7-((9-(((2S)-1-((2S,4R)-4-hydroxy-2-(((4-(4-methyl-1,3-thiazol-5-yl)phenyl)methyl)carbamoyl)pyrrolidin-1-yl)-3,3-dimethyl-1-oxobutan-2-yl)carbamoyl)nonyl)oxy)quinazolin-4-yl)benzoic acid; 2-cyclopentyl-4-{7-[(9-{[(2S)-1-[(2S,4R)-4-hydroxy-2-({[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl}carbamoyl)pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]carbamoyl}nonyl)oxy]quinazolin-4-yl}benzoic acid; 978-230-4; CC-3240; CHEMBL5422255; orb2566661; SCHEMBL30267807; OXICLXLJBMPGTO-LMIZGRGHSA-N; GLXC-27975; EX-A8394; BDBM50631192; HY-163064; CS-0910136; 2-Cyclopentyl-4-(7-((10-(((S)-1-((2S,4R)-4-hydroxy-2-((4-(4-methylthiazol-5-yl)benzyl)carbamoyl)pyrrolidin-1-yl)-3,3-dimethyl-1-oxobutan-2-yl)amino)-10-oxodecyl)oxy)quinazolin-4-yl)benzoic acid	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCCCCOc2ccc3c(-c4ccc(C(=O)O)c(C5CCCC5)c4)ncnc3c2)C(C)(C)C)cc1	C52H64N6O7S	CAMKK2	Q96RR4	VHL	WO-2023059873-A1
TPD-YORBYO	WO2023059873A1_4	.	Cc1ncsc1-c1ccc(CNC(=O)C2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCCCOc2ccc3c(-c4ccc(C(=O)O)c(C5CCCC5)c4)ncnc3c2)C(C)(C)C)cc1	C51H62N6O7S	CAMKK2	Q96RR4	VHL	WO-2023059873-A1
TPD-0VF0FM	CHEMBL5394508	2-cyclopentyl-4-[7-[8-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-8-oxooctoxy]quinazolin-4-yl]benzoic acid; BDBM50631195; PD216516	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCCOc2ccc3c(-c4ccc(C(=O)O)c(C5CCCC5)c4)ncnc3c2)C(C)(C)C)cc1	C50H60N6O7S	CAMKK2	Q96RR4	VHL	WO-2023059873-A1
TPD-KKV5D8	CHEMBL5395520	2-cyclopentyl-4-[7-[7-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-7-oxoheptoxy]quinazolin-4-yl]benzoic acid; SCHEMBL30267854; BDBM50631194; PD216514	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCOc2ccc3c(-c4ccc(C(=O)O)c(C5CCCC5)c4)ncnc3c2)C(C)(C)C)cc1	C49H58N6O7S	CAMKK2	Q96RR4	VHL	WO-2023059873-A1
TPD-U4JWQH	SCHEMBL25468997	5-[3-[3-[3-[4-Amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]azetidin-1-yl]azetidin-1-yl]azetidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	Nc1ncnc2c1c(-c1ccc(Oc3ccccc3)cc1)nn2C1CN(C2CN(C3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)C2)C1	C39H36N10O5	BTK	Q06187	CRBN	WO-2023072270-A1
TPD-2YUTN9	WO2023072270A1_3	.	Nc1ncnc2c1c(-c1ccc(Oc3ccccc3)cc1)nn2C1CCC(C(=O)N2CCN(C3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)CC2)CC1	C44H44N10O6	BTK	Q06187	CRBN	WO-2023072270-A1
TPD-JXRRIS	SCHEMBL26477467	1-[4-[4-[[[3-[4-[4-Amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidine-1-carbonyl]cyclobutyl]-methylamino]methyl]piperidine-1-carbonyl]phenyl]-1,3-diazinane-2,4-dione	CN(CC1CCN(C(=O)c2ccc(N3CCC(=O)NC3=O)cc2)CC1)C1CC(C(=O)N2CCC(n3nc(-c4ccc(Oc5ccccc5)cc4)c4c(N)ncnc43)CC2)C1	C45H50N10O5	BTK	Q06187	CRBN	WO-2023072270-A1
TPD-BZZ8IQ	SCHEMBL26479931	5-[3-[4-[4-[4-Amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]cyclohexyl]piperazin-1-yl]azetidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	Nc1ncnc2c1c(-c1ccc(Oc3ccccc3)cc1)nn2C1CCC(N2CCN(C3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)CC2)CC1	C43H44N10O5	BTK	Q06187	CRBN	WO-2023072270-A1
TPD-Q0DKYW	SCHEMBL26477446	6-[3-[4-[4-Amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]bicyclo[1.1.1]pentane-1-carbonyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	Nc1ncnc2c1c(-c1ccc(Oc3ccccc3)cc1)nn2C1CCN(C23CC(C(=O)N4Cc5cc6c(cc5C4)C(=O)N(C4CCC(=O)NC4=O)C6=O)(C2)C3)CC1	C43H39N9O6	BTK	Q06187	CRBN	WO-2023072270-A1
TPD-DNSYE4	SCHEMBL24697748	5-[3-[3-[5-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]-3,3a,4,5,6,6a-hexahydro-1H-cyclopenta[c]pyrrol-2-yl]azetidin-1-yl]azetidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	Nc1ncnc2c1c(-c1ccc(Oc3ccccc3)cc1)nn2C1CC2CN(C3CN(C4CN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)C3)CC2C1	C43H42N10O5	BTK	Q06187	CRBN	WO-2023072270-A1
TPD-WTBIRT	SCHEMBL26477441	5-[3-[3-[4-[4-Amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]azepan-1-yl]azetidin-1-yl]azetidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	Nc1ncnc2c1c(-c1ccc(Oc3ccccc3)cc1)nn2C1CCCN(C2CN(C3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)C2)CC1	C42H42N10O5	BTK	Q06187	CRBN	WO-2023072270-A1
TPD-U023BW	WO2023072270A1_9	.	COc1cccc(Oc2ccc(-c3nn(C4CCC(C(=O)N5CC(N6Cc7cc8c(cc7C6)C(=O)N(C6CCC(=O)NC6=O)C8=O)C5)CC4)c4c(OC)cncc34)cc2)c1F	C45H42FN7O8	BTK	Q06187	CRBN	WO-2023072270-A1
TPD-QG37PF	SCHEMBL26477449	3-[4-[3-[3-[4-[4-Amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]azetidin-1-yl]azetidin-1-yl]-3-fluoroanilino]piperidine-2,6-dione	Nc1ncnc2c1c(-c1ccc(Oc3ccccc3)cc1)nn2C1CCN(C2CN(C3CN(c4ccc(NC5CCC(=O)NC5=O)cc4F)C3)C2)CC1	C39H41FN10O3	BTK	Q06187	CRBN	WO-2023072270-A1
TPD-1DTX9E	SCHEMBL26477955	6-[3-[4-[4-Amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]cyclobutanecarbonyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	Nc1ncnc2c1c(-c1ccc(Oc3ccccc3)cc1)nn2C1CCN(C2CC(C(=O)N3Cc4cc5c(cc4C3)C(=O)N(C3CCC(=O)NC3=O)C5=O)C2)CC1	C42H39N9O6	BTK	Q06187	CRBN	WO-2023072270-A1
TPD-6A98IE	SCHEMBL26477806	5-[3-[3-[4-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]azetidin-1-yl]azetidin-1-yl]-N-(2,6-dioxopiperidin-3-yl)pyridine-2-carboxamide	Nc1ncnc2c1c(-c1ccc(Oc3ccccc3)cc1)nn2C1CCN(C2CN(C3CN(c4ccc(C(=O)NC5CCC(=O)NC5=O)nc4)C3)C2)CC1	C39H41N11O4	BTK	Q06187	CRBN	WO-2023072270-A1
TPD-1X80OI	SCHEMBL26106437	5-[3-[1-[4-[4-Amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]cyclohexyl]azetidin-3-yl]azetidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	Nc1ncnc2c1c(-c1ccc(Oc3ccccc3)cc1)nn2C1CCC(N2CC(C3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)C2)CC1	C42H41N9O5	BTK	Q06187	CRBN	WO-2023072270-A1
TPD-JR5VLP	SCHEMBL26477958	5-[3-[3-[5-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]-3,3a,4,5,6,6a-hexahydro-1H-cyclopenta[c]pyrrol-2-yl]azetidin-1-yl]pyrrolidin-1-yl]-N-(2,6-dioxopiperidin-3-yl)pyridine-2-carboxamide	Nc1ncnc2c1c(-c1ccc(Oc3ccccc3)cc1)nn2C1CC2CN(C3CN(C4CCN(c5ccc(C(=O)NC6CCC(=O)NC6=O)nc5)C4)C3)CC2C1	C42H45N11O4	BTK	Q06187	CRBN	WO-2023072270-A1
TPD-65AJ2R	SCHEMBL26477959	3-[4-[3-[3-[5-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]-3,3a,4,5,6,6a-hexahydro-1H-cyclopenta[c]pyrrol-2-yl]azetidin-1-yl]pyrrolidin-1-yl]-3-fluoroanilino]piperidine-2,6-dione	Nc1ncnc2c1c(-c1ccc(Oc3ccccc3)cc1)nn2C1CC2CN(C3CN(C4CCN(c5ccc(NC6CCC(=O)NC6=O)cc5F)C4)C3)CC2C1	C42H45FN10O3	BTK	Q06187	CRBN	WO-2023072270-A1
TPD-OU1BKC	SCHEMBL26477960	5-[3-[[3-[5-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]-3,3a,4,5,6,6a-hexahydro-1H-cyclopenta[c]pyrrol-2-yl]azetidin-1-yl]methyl]pyrrolidin-1-yl]-N-(2,6-dioxopiperidin-3-yl)pyridine-2-carboxamide	Nc1ncnc2c1c(-c1ccc(Oc3ccccc3)cc1)nn2C1CC2CN(C3CN(CC4CCN(c5ccc(C(=O)NC6CCC(=O)NC6=O)nc5)C4)C3)CC2C1	C43H47N11O4	BTK	Q06187	CRBN	WO-2023072270-A1
TPD-P429Z8	SCHEMBL26104846	5-[3-[3-[5-[4-amino-3-[4-(2-fluoro-3-methoxyphenoxy)phenyl]pyrazolo[3,4-d]pyrimidin-1-yl]-3,3a,4,5,6,6a-hexahydro-1H-cyclopenta[c]pyrrol-2-yl]azetidin-1-yl]azetidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)-6-fluoroisoindole-1,3-dione	COc1cccc(Oc2ccc(-c3nn(C4CC5CN(C6CN(C7CN(c8cc9c(cc8F)C(=O)N(C8CCC(=O)NC8=O)C9=O)C7)C6)CC5C4)c4ncnc(N)c34)cc2)c1F	C44H42F2N10O6	BTK	Q06187	CRBN	WO-2023072270-A1
TPD-9RLR2B	SCHEMBL26477964	5-[3-[[5-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]-3,3a,4,5,6,6a-hexahydro-1H-cyclopenta[c]pyrrol-2-yl]methyl]pyrrolidin-1-yl]-N-(2,6-dioxopiperidin-3-yl)pyridine-2-carboxamide; SCHEMBL30301985	Nc1ncnc2c1c(-c1ccc(Oc3ccccc3)cc1)nn2C1CC2CN(CC3CCN(c4ccc(C(=O)NC5CCC(=O)NC5=O)nc4)C3)CC2C1	C40H42N10O4	BTK	Q06187	CRBN	WO-2023072270-A1
TPD-QTDOTG	SCHEMBL26477965	5-[3-[[4-[4-[4-Amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]cyclohexyl]piperazin-1-yl]methyl]pyrrolidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	Nc1ncnc2c1c(-c1ccc(Oc3ccccc3)cc1)nn2C1CCC(N2CCN(CC3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)CC2)CC1	C45H48N10O5	BTK	Q06187	CRBN	WO-2023072270-A1
TPD-16CLT8	SCHEMBL26478123	5-[3-[4-[4-[4-amino-3-[4-(2-fluoro-3-methoxyphenoxy)phenyl]pyrazolo[3,4-d]pyrimidin-1-yl]cyclohexanecarbonyl]piperazin-1-yl]azetidin-1-yl]-N-(2,6-dioxopiperidin-3-yl)pyridine-2-carboxamide	COc1cccc(Oc2ccc(-c3nn(C4CCC(C(=O)N5CCN(C6CN(c7ccc(C(=O)NC8CCC(=O)NC8=O)nc7)C6)CC5)CC4)c4ncnc(N)c34)cc2)c1F	C43H46FN11O6	BTK	Q06187	CRBN	WO-2023072270-A1
TPD-Y798LW	SCHEMBL26478132	N-(2,6-dioxopiperidin-3-yl)-5-[3-[3-[4-[3-[4-(2-fluoro-3-methoxyphenoxy)phenyl]-7-methoxypyrazolo[4,3-c]pyridin-1-yl]piperidin-1-yl]azetidin-1-yl]azetidin-1-yl]pyridine-2-carboxamide	COc1cccc(Oc2ccc(-c3nn(C4CCN(C5CN(C6CN(c7ccc(C(=O)NC8CCC(=O)NC8=O)nc7)C6)C5)CC4)c4c(OC)cncc34)cc2)c1F	C42H44FN9O6	BTK	Q06187	CRBN	WO-2023072270-A1
TPD-IKUWQ0	SCHEMBL26478129	6-[[3-[4-[4-Amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]cyclobutyl]methyl]-2-(2,6-dioxopiperidin-3-yl)-5,7-dihydropyrrolo[3,4-f]isoindole-1,3-dione	Nc1ncnc2c1c(-c1ccc(Oc3ccccc3)cc1)nn2C1CCN(C2CC(CN3Cc4cc5c(cc4C3)C(=O)N(C3CCC(=O)NC3=O)C5=O)C2)CC1	C42H41N9O5	BTK	Q06187	CRBN	WO-2023072270-A1
TPD-THHD7V	SCHEMBL26478133	5-[4-[[4-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]cyclohexyl]methyl]piperazin-1-yl]-N-(2,6-dioxopiperidin-3-yl)pyridine-2-carboxamide	Nc1ncnc2c1c(-c1ccc(Oc3ccccc3)cc1)nn2C1CCC(CN2CCN(c3ccc(C(=O)NC4CCC(=O)NC4=O)nc3)CC2)CC1	C39H42N10O4	BTK	Q06187	CRBN	WO-2023072270-A1
TPD-QFK67L	SCHEMBL26478137	N-(2,6-dioxopiperidin-3-yl)-5-[3-[3-[5-[3-[4-(2-fluoro-3-methoxyphenoxy)phenyl]-7-methoxypyrazolo[4,3-c]pyridin-1-yl]-3,3a,4,5,6,6a-hexahydro-1H-cyclopenta[c]pyrrol-2-yl]azetidin-1-yl]azetidin-1-yl]pyridine-2-carboxamide	COc1cccc(Oc2ccc(-c3nn(C4CC5CN(C6CN(C7CN(c8ccc(C(=O)NC9CCC(=O)NC9=O)nc8)C7)C6)CC5C4)c4c(OC)cncc34)cc2)c1F	C44H46FN9O6	BTK	Q06187	CRBN	WO-2023072270-A1
TPD-DPFGZD	SCHEMBL26480234	5-[3-[3-[5-[4-amino-3-[4-(2-fluoro-3-methoxyphenoxy)phenyl]pyrazolo[3,4-d]pyrimidin-1-yl]-3,3a,4,5,6,6a-hexahydro-1H-cyclopenta[c]pyrrol-2-yl]azetidin-1-yl]azetidin-1-yl]-N-(2,6-dioxopiperidin-3-yl)pyridine-2-carboxamide	COc1cccc(Oc2ccc(-c3nn(C4CC5CN(C6CN(C7CN(c8ccc(C(=O)NC9CCC(=O)NC9=O)nc8)C7)C6)CC5C4)c4ncnc(N)c34)cc2)c1F	C42H44FN11O5	BTK	Q06187	CRBN	WO-2023072270-A1
TPD-59VEBW	SCHEMBL26480245	5-[4-[1-[4-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]cyclohexyl]azetidin-3-yl]piperazin-1-yl]-N-(2,6-dioxopiperidin-3-yl)pyridine-2-carboxamide	Nc1ncnc2c1c(-c1ccc(Oc3ccccc3)cc1)nn2C1CCC(N2CC(N3CCN(c4ccc(C(=O)NC5CCC(=O)NC5=O)nc4)CC3)C2)CC1	C41H45N11O4	BTK	Q06187	CRBN	WO-2023072270-A1
TPD-8HOEB1	SCHEMBL26478148	4-[3-[3-[5-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]-3,3a,4,5,6,6a-hexahydro-1H-cyclopenta[c]pyrrol-2-yl]azetidin-1-yl]azetidin-1-yl]-N-(2,6-dioxopiperidin-3-yl)-2-methoxybenzamide	COc1cc(N2CC(N3CC(N4CC5CC(n6nc(-c7ccc(Oc8ccccc8)cc7)c7c(N)ncnc76)CC5C4)C3)C2)ccc1C(=O)NC1CCC(=O)NC1=O	C43H46N10O5	BTK	Q06187	CRBN	WO-2023072270-A1
TPD-78JMRB	SCHEMBL26478151	5-[3-[3-[5-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]-3,3a,4,5,6,6a-hexahydro-1H-cyclopenta[c]pyrrol-2-yl]azetidin-1-yl]azetidin-1-yl]-N-(2,6-dioxopiperidin-3-yl)pyridine-2-carboxamide	Nc1ncnc2c1c(-c1ccc(Oc3ccccc3)cc1)nn2C1CC2CN(C3CN(C4CN(c5ccc(C(=O)NC6CCC(=O)NC6=O)nc5)C4)C3)CC2C1	C41H43N11O4	BTK	Q06187	CRBN	WO-2023072270-A1
TPD-3W14WY	SCHEMBL26102459	5-[3-[4-[4-[4-Amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]cyclohexyl]piperazin-1-yl]azetidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)-6-fluoroisoindole-1,3-dione; SCHEMBL26103645; SCHEMBL30301988; SCHEMBL30301994	Nc1ncnc2c1c(-c1ccc(Oc3ccccc3)cc1)nn2C1CCC(N2CCN(C3CN(c4cc5c(cc4F)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)CC2)CC1	C43H43FN10O5	BTK	Q06187	CRBN	WO-2023072270-A1
TPD-LQ4P76	SCHEMBL26477804	5-[3-[4-[4-[4-Amino-3-[4-(2-fluoro-3-methoxyphenoxy)phenyl]pyrazolo[3,4-d]pyrimidin-1-yl]cyclohexyl]piperazin-1-yl]azetidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	COc1cccc(Oc2ccc(-c3nn(C4CCC(N5CCN(C6CN(c7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)C6)CC5)CC4)c4ncnc(N)c34)cc2)c1F	C44H45FN10O6	BTK	Q06187	CRBN	WO-2023072270-A1
TPD-X272KJ	SCHEMBL26478153	5-[3-[4-[4-[4-amino-3-[4-(2-fluoro-3-methoxyphenoxy)phenyl]pyrazolo[3,4-d]pyrimidin-1-yl]cyclohexyl]piperazin-1-yl]azetidin-1-yl]-N-(2,6-dioxopiperidin-3-yl)pyridine-2-carboxamide	COc1cccc(Oc2ccc(-c3nn(C4CCC(N5CCN(C6CN(c7ccc(C(=O)NC8CCC(=O)NC8=O)nc7)C6)CC5)CC4)c4ncnc(N)c34)cc2)c1F	C42H46FN11O5	BTK	Q06187	CRBN	WO-2023072270-A1
TPD-DSSYWE	SCHEMBL26478306	5-[3-[4-[4-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]cyclohexyl]piperazin-1-yl]azetidin-1-yl]-N-(2,6-dioxopiperidin-3-yl)pyridine-2-carboxamide	Nc1ncnc2c1c(-c1ccc(Oc3ccccc3)cc1)nn2C1CCC(N2CCN(C3CN(c4ccc(C(=O)NC5CCC(=O)NC5=O)nc4)C3)CC2)CC1	C41H45N11O4	BTK	Q06187	CRBN	WO-2023072270-A1
TPD-W5CC9K	WO2023072270A1_33	.	COc1cccc(Oc2ccc(-c3nn(C4CCC(N5CCN(C6CN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)C6)CC5)CC4)c4ncnc(N)c34)cc2)c1F	C44H44F2N10O6	BTK	Q06187	CRBN	WO-2023072270-A1
TPD-WMM0F2	WO2023072270A1_36	.	Nc1ncnc2c1c(-c1ccc(Oc3ccccc3)cc1)nn2[C@H]1CC[C@H](N2CCN(C3CN(c4cc5c(cc4F)C(=O)N([C@H]4CCC(=O)NC4=O)C5=O)C3)CC2)CC1	C43H43FN10O5	BTK	Q06187	CRBN	WO-2023072270-A1
TPD-LQRHPP	WO2023072270A1_37	.	Nc1ncnc2c1c(-c1ccc(Oc3ccccc3)cc1)nn2[C@H]1CC[C@H](N2CCN(C3CN(c4cc5c(cc4F)C(=O)N([C@@H]4CCC(=O)NC4=O)C5=O)C3)CC2)CC1	C43H43FN10O5	BTK	Q06187	CRBN	WO-2023072270-A1
TPD-Y4KSIY	WO2023072270A1_38	.	Nc1ncnc2c1c(-c1ccc(Oc3ccccc3)cc1)nn2[C@H]1CC[C@@H](N2CCN(C3CN(c4cc5c(cc4F)C(=O)N([C@H]4CCC(=O)NC4=O)C5=O)C3)CC2)CC1	C43H43FN10O5	BTK	Q06187	CRBN	WO-2023072270-A1
TPD-TX9RJA	WO2023072270A1_39	.	Nc1ncnc2c1c(-c1ccc(Oc3ccccc3)cc1)nn2[C@H]1CC[C@@H](N2CCN(C3CN(c4cc5c(cc4F)C(=O)N([C@@H]4CCC(=O)NC4=O)C5=O)C3)CC2)CC1	C43H43FN10O5	BTK	Q06187	CRBN	WO-2023072270-A1
TPD-3QD15V	WO2023072270A1_40	.	Nc1ncnc2c1c(-c1ccc(Oc3ccccc3)cc1)nn2[C@H]1CC[C@H](N2CCN(C3CN(c4ccc5c(c4)C(=O)N([C@H]4CCC(=O)NC4=O)C5=O)C3)CC2)CC1	C43H44N10O5	BTK	Q06187	CRBN	WO-2023072270-A1
TPD-155KW7	WO2023072270A1_41	.	Nc1ncnc2c1c(-c1ccc(Oc3ccccc3)cc1)nn2[C@H]1CC[C@H](N2CCN(C3CN(c4ccc5c(c4)C(=O)N([C@@H]4CCC(=O)NC4=O)C5=O)C3)CC2)CC1	C43H44N10O5	BTK	Q06187	CRBN	WO-2023072270-A1
TPD-WPCX9F	WO2023072270A1_42	.	Nc1ncnc2c1c(-c1ccc(Oc3ccccc3)cc1)nn2[C@H]1CC[C@@H](N2CCN(C3CN(c4ccc5c(c4)C(=O)N([C@H]4CCC(=O)NC4=O)C5=O)C3)CC2)CC1	C43H44N10O5	BTK	Q06187	CRBN	WO-2023072270-A1
TPD-Y9BUOH	WO2023072270A1_43	.	Nc1ncnc2c1c(-c1ccc(Oc3ccccc3)cc1)nn2[C@H]1CC[C@@H](N2CCN(C3CN(c4ccc5c(c4)C(=O)N([C@@H]4CCC(=O)NC4=O)C5=O)C3)CC2)CC1	C43H44N10O5	BTK	Q06187	CRBN	WO-2023072270-A1
TPD-VVNVP0	CHEMBL5410660	(1S,2R)-2-[(1S)-5-chloro-8-[[1-[2-[[2-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]acetyl]amino]ethyl]-5-methyltriazol-4-yl]methoxy]-1-[(6-oxo-5-azaspiro[2.4]heptan-5-yl)methyl]-3,4-dihydro-1H-isoquinoline-2-carbonyl]-1-methylcyclohexane-1-carboxylic acid; SCHEMBL26105647; SCHEMBL30372063	CC1=NN=C2[C@H](CC(=O)NCC(=O)NCCN3N=NC(COC4=CC=C(Cl)C5=C4[C@@H](CN4CC6(CC6)CC4=O)N(C(=O)[C@@H]4CCCC[C@]4(C)C(=O)O)CC5)=C3C)N=C(C3=CC=C(Cl)C=C3)C3=C(SC(C)=C3C)N12	C52H59Cl2N11O7S	BRD4	O60885	KEAP1	WO-2023073364-A1
TPD-XKI8AI	SCHEMBL30372342	(1S,2R)-2-[(1S)-5-chloro-8-[[1-[2-[[2-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]acetyl]amino]ethyl]-5-methyltriazol-4-yl]methoxy]-1-[(6-oxo-5-azaspiro[2.4]heptan-5-yl)methyl]-3,4-dihydro-1H-isoquinoline-2-carbonyl]-N,1-dimethylcyclohexane-1-carboxamide	CNC(=O)[C@@]1(C)CCCC[C@H]1C(=O)N1CCC2=C(C(OCC3=C(C)N(CCNC(=O)CNC(=O)C[C@@H]4N=C(C5=CC=C(Cl)C=C5)C5=C(SC(C)=C5C)N5C(C)=NN=C45)N=N3)=CC=C2Cl)[C@H]1CN1CC2(CC2)CC1=O	C53H62Cl2N12O6S	BRD4	O60885	KEAP1	WO-2023073364-A1
TPD-LGM3IQ	SCHEMBL26101684	(1S,2R)-2-[(1S)-5-chloro-8-[[5-[2-[[2-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]acetyl]amino]ethoxymethyl]-1-methyltriazol-4-yl]methoxy]-1-[(6-oxo-5-azaspiro[2.4]heptan-5-yl)methyl]-3,4-dihydro-1H-isoquinoline-2-carbonyl]-1-methylcyclohexane-1-carboxylic acid; SCHEMBL30372075	CC1=NN=C2[C@H](CC(=O)NCC(=O)NCCOCC3=C(COC4=CC=C(Cl)C5=C4[C@@H](CN4CC6(CC6)CC4=O)N(C(=O)[C@@H]4CCCC[C@]4(C)C(=O)O)CC5)N=NN3C)N=C(C3=CC=C(Cl)C=C3)C3=C(SC(C)=C3C)N12	C53H61Cl2N11O8S	BRD4	O60885	KEAP1	WO-2023073364-A1
TPD-NFFALL	SCHEMBL26104043	(1S,2R)-2-[(1S)-5-chloro-8-[[5-[2-[3-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]propanoylamino]ethoxymethyl]-1-methyltriazol-4-yl]methoxy]-1-[(6-oxo-5-azaspiro[2.4]heptan-5-yl)methyl]-3,4-dihydro-1H-isoquinoline-2-carbonyl]-1-methylcyclohexane-1-carboxylic acid; SCHEMBL30372512	CC1=NN=C2[C@H](CC(=O)NCCC(=O)NCCOCC3=C(COC4=CC=C(Cl)C5=C4[C@@H](CN4CC6(CC6)CC4=O)N(C(=O)[C@@H]4CCCC[C@]4(C)C(=O)O)CC5)N=NN3C)N=C(C3=CC=C(Cl)C=C3)C3=C(SC(C)=C3C)N12	C54H63Cl2N11O8S	BRD4	O60885	KEAP1	WO-2023073364-A1
TPD-QVHBZE	SCHEMBL26103396	(1S,2R)-2-[(1S)-5-chloro-8-[[5-[2-[3-[2-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]ethoxy]propanoylamino]ethoxymethyl]-1-methyltriazol-4-yl]methoxy]-1-[(6-oxo-5-azaspiro[2.4]heptan-5-yl)methyl]-3,4-dihydro-1H-isoquinoline-2-carbonyl]-1-methylcyclohexane-1-carboxylic acid; SCHEMBL30372155	CC1=NN=C2[C@H](CC(=O)NCCOCCC(=O)NCCOCC3=C(COC4=CC=C(Cl)C5=C4[C@@H](CN4CC6(CC6)CC4=O)N(C(=O)[C@@H]4CCCC[C@]4(C)C(=O)O)CC5)N=NN3C)N=C(C3=CC=C(Cl)C=C3)C3=C(SC(C)=C3C)N12	C56H67Cl2N11O9S	BRD4	O60885	KEAP1	WO-2023073364-A1
TPD-K66W06	SCHEMBL26101542	(1S,2R)-2-[(1S)-5-chloro-8-[(3S)-1-[2-[2-[[2-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]acetyl]amino]ethoxy]acetyl]pyrrolidin-3-yl]oxy-1-[(6-oxo-5-azaspiro[2.4]heptan-5-yl)methyl]-3,4-dihydro-1H-isoquinoline-2-carbonyl]-1-methylcyclohexane-1-carboxylic acid; SCHEMBL30372347	CC1=NN=C2[C@H](CC(=O)NCC(=O)NCCOCC(=O)N3CC[C@H](OC4=CC=C(Cl)C5=C4[C@@H](CN4CC6(CC6)CC4=O)N(C(=O)[C@@H]4CCCC[C@]4(C)C(=O)O)CC5)C3)N=C(C3=CC=C(Cl)C=C3)C3=C(SC(C)=C3C)N12	C54H63Cl2N9O9S	BRD4	O60885	KEAP1	WO-2023073364-A1
TPD-5703K5	SCHEMBL26101832	(1S,2R)-2-[(1S)-5-chloro-8-[(1,5-dimethyltriazol-4-yl)methoxy]-1-[(6-oxo-5-azaspiro[2.4]heptan-5-yl)methyl]-3,4-dihydro-1H-isoquinoline-2-carbonyl]-N-[2-[[2-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]acetyl]amino]ethyl]-1-methylcyclohexane-1-carboxamide; SCHEMBL30372630	CC1=NN=C2[C@H](CC(=O)NCC(=O)NCCNC(=O)[C@@]3(C)CCCC[C@H]3C(=O)N3CCC4=C(C(OCC5=C(C)N(C)N=N5)=CC=C4Cl)[C@H]3CN3CC4(CC4)CC3=O)N=C(C3=CC=C(Cl)C=C3)C3=C(SC(C)=C3C)N12	C53H62Cl2N12O6S	BRD4	O60885	KEAP1	WO-2023073364-A1
TPD-72Z4L1	SCHEMBL26103474	(1S,2R)-2-[(1S)-5-chloro-8-[(1,5-dimethyltriazol-4-yl)methoxy]-1-[(6-oxo-5-azaspiro[2.4]heptan-5-yl)methyl]-3,4-dihydro-1H-isoquinoline-2-carbonyl]-N-[2-[2-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]ethoxy]ethyl]-1-methylcyclohexane-1-carboxamide; SCHEMBL30372186	CC1=NN=C2[C@H](CC(=O)NCCOCCNC(=O)[C@@]3(C)CCCC[C@H]3C(=O)N3CCC4=C(C(OCC5=C(C)N(C)N=N5)=CC=C4Cl)[C@H]3CN3CC4(CC4)CC3=O)N=C(C3=CC=C(Cl)C=C3)C3=C(SC(C)=C3C)N12	C53H63Cl2N11O6S	BRD4	O60885	KEAP1	WO-2023073364-A1
TPD-A4TBDS	SCHEMBL26102307	(1S,2R)-2-[(1S)-5-chloro-8-[(1,5-dimethyltriazol-4-yl)methoxy]-1-[(6-oxo-5-azaspiro[2.4]heptan-5-yl)methyl]-3,4-dihydro-1H-isoquinoline-2-carbonyl]-N-[2-[2-[2-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]ethoxy]ethoxy]ethyl]-1-methylcyclohexane-1-carboxamide; SCHEMBL30372184	CC1=NN=C2[C@H](CC(=O)NCCOCCOCCNC(=O)[C@@]3(C)CCCC[C@H]3C(=O)N3CCC4=C(C(OCC5=C(C)N(C)N=N5)=CC=C4Cl)[C@H]3CN3CC4(CC4)CC3=O)N=C(C3=CC=C(Cl)C=C3)C3=C(SC(C)=C3C)N12	C55H67Cl2N11O7S	BRD4	O60885	KEAP1	WO-2023073364-A1
TPD-L2QWD7	SCHEMBL31536434	6-[2-[(6-cyanoquinolin-4-yl)amino]ethyl]-N-[3-[3-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethoxy]propanoylamino]propyl]-N-methylnaphthalene-2-carboxamide	CN(CCCNC(=O)CCOCCOCCOCCOCCNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O)C(=O)c1ccc2cc(CCNc3ccnc4ccc(C#N)cc34)ccc2c1	C51H56N8O10	CDK8;CDK19	P49336/Q9BWU1	CRBN	WO-2023081452-A1
TPD-CAPOGP	WO2023081452A1_23b	.	N#Cc1ccc2nccc(NCCc3ccc4cc(C(=O)N5CCN(CCCNC(=O)CCOCCOCCOCCOCCNc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)ccc4c3)c2c1	C54H61N9O10	CDK8;CDK19	P49336/Q9BWU1	CRBN	WO-2023081452-A1
TPD-3KZVOK	SCHEMBL25415881	4-[2-[6-[4-[3-[2-[2-[[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]propanoyl]piperazine-1-carbonyl]naphthalen-2-yl]ethylamino]quinoline-6-carbonitrile; SCHEMBL30369538	N#Cc1ccc2nccc(NCCc3ccc4cc(C(=O)N5CCN(C(=O)CCOCCOCCNc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)ccc4c3)c2c1	C47H46N8O8	CDK8;CDK19	P49336/Q9BWU1	CRBN	WO-2023081452-A1
TPD-S4XIFK	SCHEMBL31536427	4-[2-[6-[4-[3-[2-[2-[2-[[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]propanoyl]piperazine-1-carbonyl]naphthalen-2-yl]ethylamino]quinoline-6-carbonitrile	N#Cc1ccc2nccc(NCCc3ccc4cc(C(=O)N5CCN(C(=O)CCOCCOCCOCCNc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)ccc4c3)c2c1	C49H50N8O9	CDK8;CDK19	P49336/Q9BWU1	CRBN	WO-2023081452-A1
TPD-7E1YBL	SCHEMBL25414417	4-[2-[6-[4-[3-[2-[2-[2-[2-[[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethoxy]propanoyl]piperazine-1-carbonyl]naphthalen-2-yl]ethylamino]quinoline-6-carbonitrile; SCHEMBL31536431	N#Cc1ccc2nccc(NCCc3ccc4cc(C(=O)N5CCN(C(=O)CCOCCOCCOCCOCCNc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)ccc4c3)c2c1	C51H54N8O10	CDK8;CDK19	P49336/Q9BWU1	CRBN	WO-2023081452-A1
TPD-5AZM18	SCHEMBL25416824	4-[2-[6-[4-[3-[2-[2-[2-[2-[2-[[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]propanoyl]piperazine-1-carbonyl]naphthalen-2-yl]ethylamino]quinoline-6-carbonitrile; SCHEMBL30369681	N#Cc1ccc2nccc(NCCc3ccc4cc(C(=O)N5CCN(C(=O)CCOCCOCCOCCOCCOCCNc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)ccc4c3)c2c1	C53H58N8O11	CDK8;CDK19	P49336/Q9BWU1	CRBN	WO-2023081452-A1
TPD-J9TMAB	SCHEMBL25415122	4-[2-[6-[4-[3-[2-[2-[2-[2-[2-[2-[[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]propanoyl]piperazine-1-carbonyl]naphthalen-2-yl]ethylamino]quinoline-6-carbonitrile; SCHEMBL30369934	N#Cc1ccc2nccc(NCCc3ccc4cc(C(=O)N5CCN(C(=O)CCOCCOCCOCCOCCOCCOCCNc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)ccc4c3)c2c1	C55H62N8O12	CDK8;CDK19	P49336/Q9BWU1	CRBN	WO-2023081452-A1
TPD-4JKM68	SCHEMBL25417125	3-Amino-4-[4-[4-[3-[3-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]propanoylamino]propyl-methylcarbamoyl]phenyl]-1,4-diazepan-1-yl]thieno[2,3-b]pyridine-2-carboxamide; SCHEMBL30369768	CN(CCCNC(=O)CCOCCOCCNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O)C(=O)c1ccc(N2CCCN(c3ccnc4sc(C(N)=O)c(N)c34)CC2)cc1	C44H52N10O9S	CDK8;CDK19	P49336/Q9BWU1	CRBN	WO-2023081452-A1
TPD-EOO8WB	SCHEMBL25416166	3-Amino-4-[4-[4-[3-[3-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]propanoylamino]propyl-methylcarbamoyl]phenyl]-1,4-diazepan-1-yl]thieno[2,3-b]pyridine-2-carboxamide; SCHEMBL30369981	CN(CCCNC(=O)CCOCCOCCOCCNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O)C(=O)c1ccc(N2CCCN(c3ccnc4sc(C(N)=O)c(N)c34)CC2)cc1	C46H56N10O10S	CDK8;CDK19	P49336/Q9BWU1	CRBN	WO-2023081452-A1
TPD-XQSVZH	WO2023081452A1_24c	.	CN(CCCNC(=O)CCOCCOCCOCCOCCNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O)C(=O)c1ccc(N2CCCN(c3ccnc4sc(C(N)=O)c(N)c34)CC2)cc1	C48H60N10O11S	CDK8;CDK19	P49336/Q9BWU1	CRBN	WO-2023081452-A1
TPD-P14Z8R	SCHEMBL25415595	3-Amino-4-[4-[4-[3-[3-[2-[2-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]propanoylamino]propyl-methylcarbamoyl]phenyl]-1,4-diazepan-1-yl]thieno[2,3-b]pyridine-2-carboxamide; SCHEMBL30369572	CN(CCCNC(=O)CCOCCOCCOCCOCCOCCOCCNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O)C(=O)c1ccc(N2CCCN(c3ccnc4sc(C(N)=O)c(N)c34)CC2)cc1	C52H68N10O13S	CDK8;CDK19	P49336/Q9BWU1	CRBN	WO-2023081452-A1
TPD-FB0XL2	SCHEMBL30369569	(2S,4R)-1-[(2S)-2-[3-[2-[2-[2-[3-[4-[6-[2-[(6-cyanoquinolin-4-yl)amino]ethyl]naphthalene-2-carbonyl]piperazin-1-yl]-3-oxopropoxy]ethoxy]ethoxy]ethoxy]propanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCOCCOCCOCCOCCC(=O)N2CCN(C(=O)c3ccc4cc(CCNc5ccnc6ccc(C#N)cc56)ccc4c3)CC2)C(C)(C)C)cc1	C61H73N9O10S	CDK8;CDK19	P49336/Q9BWU1	CRBN	WO-2023081452-A1
TPD-PZWGJP	SCHEMBL25434782	N-[3-[4-[6-[2-[(6-cyanoquinolin-4-yl)amino]ethyl]naphthalene-2-carbonyl]piperazin-1-yl]-3-oxopropyl]-3-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]propanamide; SCHEMBL30369455	N#Cc1ccc2nccc(NCCc3ccc4cc(C(=O)N5CCN(C(=O)CCNC(=O)CCOCCOCCOCCNc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)ccc4c3)c2c1	C52H55N9O10	CDK8;CDK19	P49336/Q9BWU1	CRBN	WO-2023081452-A1
TPD-1XCC8B	SCHEMBL25173857	N-[3-[4-[6-[2-[(6-cyanoquinolin-4-yl)amino]ethyl]naphthalene-2-carbonyl]piperazin-1-yl]-3-oxopropyl]-3-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethoxy]propanamide; SCHEMBL30369631	N#Cc1ccc2nccc(NCCc3ccc4cc(C(=O)N5CCN(C(=O)CCNC(=O)CCOCCOCCOCCOCCNc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)ccc4c3)c2c1	C54H59N9O11	CDK8;CDK19	P49336/Q9BWU1	CRBN	WO-2023081452-A1
TPD-CXRXKR	SCHEMBL25417253	4-[2-[6-[4-[3-[2-[2-[2-[2-[[2-(1-Methyl-2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethoxy]propanoyl]piperazine-1-carbonyl]naphthalen-2-yl]ethylamino]quinoline-6-carbonitrile; SCHEMBL30369634	CN1C(=O)CCC(N2C(=O)c3cccc(NCCOCCOCCOCCOCCC(=O)N4CCN(C(=O)c5ccc6cc(CCNc7ccnc8ccc(C#N)cc78)ccc6c5)CC4)c3C2=O)C1=O	C52H56N8O10	CDK8;CDK19	P49336/Q9BWU1	CRBN	WO-2023081452-A1
TPD-9QQ30V	SCHEMBL25417129	N-[2-[2-[2-[3-[4-[6-[2-[(6-cyanoquinolin-4-yl)amino]ethyl]naphthalene-2-carbonyl]piperazin-1-yl]-3-oxopropoxy]ethoxy]ethoxy]ethyl]-3-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]propanamide; SCHEMBL30369852	N#Cc1ccc2nccc(NCCc3ccc4cc(C(=O)N5CCN(C(=O)CCOCCOCCOCCNC(=O)CCNc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)ccc4c3)c2c1	C52H55N9O10	CDK8;CDK19	P49336/Q9BWU1	CRBN	WO-2023081452-A1
TPD-PSQ2LR	SCHEMBL31536423	N-[9-[4-[6-[2-[(6-cyanoquinolin-4-yl)amino]ethyl]naphthalene-2-carbonyl]piperazin-1-yl]-9-oxononyl]-3-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]propanamide	N#Cc1ccc2nccc(NCCc3ccc4cc(C(=O)N5CCN(C(=O)CCCCCCCCNC(=O)CCOCCNc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)ccc4c3)c2c1	C54H59N9O8	CDK8;CDK19	P49336/Q9BWU1	CRBN	WO-2023081452-A1
TPD-SPZXGX	SCHEMBL31536422	10-[4-[6-[2-[(6-cyanoquinolin-4-yl)amino]ethyl]naphthalene-2-carbonyl]piperazin-1-yl]-N-[5-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]pentyl]-10-oxodecanamide	N#Cc1ccc2nccc(NCCc3ccc4cc(C(=O)N5CCN(C(=O)CCCCCCCCC(=O)NCCCCCNc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)ccc4c3)c2c1	C55H61N9O7	CDK8;CDK19	P49336/Q9BWU1	CRBN	WO-2023081452-A1
TPD-KQDO8X	WO2023081452A1_48	.	Cc1ncsc1-c1ccc(CNC(=O)C2C[C@@H](O)CN2C(=O)C(NC(=O)CCCCCCCCC(=O)N2CCN(C(=O)c3ccc4cc(CCNc5ccnc6ccc(C#N)cc56)ccc4c3)CC2)C(C)(C)C)cc1	C59H69N9O6S	CDK8;CDK19	P49336/Q9BWU1	CRBN	WO-2023081452-A1
TPD-SC5ZF5	SCHEMBL30370005	N-[9-[4-[6-[2-[(6-cyanoquinolin-4-yl)amino]ethyl]naphthalene-2-carbonyl]piperazin-1-yl]-9-oxononyl]-5-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]pentanamide	N#Cc1ccc2nccc(NCCc3ccc4cc(C(=O)N5CCN(C(=O)CCCCCCCCNC(=O)CCCCNc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)ccc4c3)c2c1	C54H59N9O7	CDK8;CDK19	P49336/Q9BWU1	CRBN	WO-2023081452-A1
TPD-ZDWAAO	SCHEMBL25439171	N-[10-[4-[6-[2-[(6-cyanoquinolin-4-yl)amino]ethyl]naphthalene-2-carbonyl]piperazin-1-yl]-10-oxodecyl]-6-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]hexanamide; SCHEMBL30369882	N#Cc1ccc2nccc(NCCc3ccc4cc(C(=O)N5CCN(C(=O)CCCCCCCCCNC(=O)CCCCCNc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)ccc4c3)c2c1	C56H63N9O7	CDK8;CDK19	P49336/Q9BWU1	CRBN	WO-2023081452-A1
TPD-6X7YVU	SCHEMBL25438687	N-[9-[4-[6-[2-[(6-cyanoquinolin-4-yl)amino]ethyl]naphthalene-2-carbonyl]piperazin-1-yl]-9-oxononyl]-6-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]hexanamide; SCHEMBL31536437	N#Cc1ccc2nccc(NCCc3ccc4cc(C(=O)N5CCN(C(=O)CCCCCCCCNC(=O)CCCCCNc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)ccc4c3)c2c1	C55H61N9O7	CDK8;CDK19	P49336/Q9BWU1	CRBN	WO-2023081452-A1
TPD-654H4I	WO2023081452A1_49d	.	N#Cc1ccc2nccc(NCCc3ccc4cc(C(=O)N5CCN(C(=O)CCCCCCCCCCNC(=O)CCCNc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)ccc4c3)c2c1	C55H61N9O7	CDK8;CDK19	P49336/Q9BWU1	CRBN	WO-2023081452-A1
TPD-IAYS32	SCHEMBL31536419	N-[12-[4-[6-[2-[(6-cyanoquinolin-4-yl)amino]ethyl]naphthalene-2-carbonyl]piperazin-1-yl]-12-oxododecyl]-3-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]propanamide	N#Cc1ccc2nccc(NCCc3ccc4cc(C(=O)N5CCN(C(=O)CCCCCCCCCCCNC(=O)CCNc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)ccc4c3)c2c1	C55H61N9O7	CDK8;CDK19	P49336/Q9BWU1	CRBN	WO-2023081452-A1
TPD-C4J6S4	SCHEMBL25437264	N-[10-[4-[6-[2-[(6-cyanoquinolin-4-yl)amino]ethyl]naphthalene-2-carbonyl]piperazin-1-yl]-10-oxodecyl]-5-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]pentanamide; SCHEMBL30369633	N#Cc1ccc2nccc(NCCc3ccc4cc(C(=O)N5CCN(C(=O)CCCCCCCCCNC(=O)CCCCNc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)ccc4c3)c2c1	C55H61N9O7	CDK8;CDK19	P49336/Q9BWU1	CRBN	WO-2023081452-A1
TPD-MYY4AI	SCHEMBL25414729	N-[11-[4-[6-[2-[(6-cyanoquinolin-4-yl)amino]ethyl]naphthalene-2-carbonyl]piperazin-1-yl]-11-oxoundecyl]-4-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]butanamide; SCHEMBL31536426	N#Cc1ccc2nccc(NCCc3ccc4cc(C(=O)N5CCN(C(=O)CCCCCCCCCCNC(=O)CCCNc6cccc7c6CN(C6CCC(=O)NC6=O)C7=O)CC5)ccc4c3)c2c1	C55H63N9O6	CDK8;CDK19	P49336/Q9BWU1	CRBN	WO-2023081452-A1
TPD-NKK7SV	SCHEMBL25415117	N-[11-[4-[6-[2-[(6-cyanoquinolin-4-yl)amino]ethyl]naphthalene-2-carbonyl]piperazin-1-yl]-11-oxoundecyl]-4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]amino]butanamide; SCHEMBL31536420	N#Cc1ccc2nccc(NCCc3ccc4cc(C(=O)N5CCN(C(=O)CCCCCCCCCCNC(=O)CCCNc6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)ccc4c3)c2c1	C55H61N9O7	CDK8;CDK19	P49336/Q9BWU1	CRBN	WO-2023081452-A1
TPD-OYQB88	SCHEMBL25416881	2-[[1-(2-chloroacetyl)-3,4-dihydro-2H-quinolin-6-yl]oxy]-N-[10-[4-[6-[2-[(6-cyanoquinolin-4-yl)amino]ethyl]naphthalene-2-carbonyl]piperazin-1-yl]-10-oxodecyl]acetamide; SCHEMBL30369241	N#Cc1ccc2nccc(NCCc3ccc4cc(C(=O)N5CCN(C(=O)CCCCCCCCCNC(=O)COc6ccc7c(c6)CCCN7C(=O)CCl)CC5)ccc4c3)c2c1	C50H56ClN7O5	CDK8;CDK19	P49336/Q9BWU1	CRBN	WO-2023081452-A1
TPD-KXF92U	WO2023081452A1_67	.	O=C1CCC(N2C(=O)c3cccc(NCCOCCOCCOCCOCCC(=O)N4CCN(C(=O)Cn5cc(C6=CCC(c7cncc8ccccc78)C=C6)cn5)CC4)c3C2=O)C(=O)N1	C48H54N8O10	CDK8;CDK19	P49336/Q9BWU1	CRBN	WO-2023081452-A1
TPD-MCDH50	SNX7886	4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]-N-[11-[4-[2-[4-(4-isoquinolin-4-ylphenyl)pyrazol-1-yl]acetyl]piperazin-1-yl]-11-oxoundecyl]butanamide; 2924557-42-4; orb1943627; SCHEMBL25438359; SCHEMBL31536417; EX-A8703; BP-42145; DA-57956; HY-156366; CS-0899748	O=C(CCCNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O)NCCCCCCCCCCC(=O)N1CCN(C(=O)Cn2cc(-c3ccc(-c4cncc5ccccc45)cc3)cn2)CC1	C52H59N9O7	CDK8;CDK19	P49336/Q9BWU1	CRBN	WO-2023081452-A1
TPD-A7HGUM	SCHEMBL30369534	N-[2-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethyl]-2-[4-(4-isoquinolin-4-ylphenyl)pyrazol-1-yl]acetamide	O=C(Cn1cc(-c2ccc(-c3cncc4ccccc34)cc2)cn1)NCCOCCOCCOCCOCCNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O	C43H45N7O9	CDK8;CDK19	P49336/Q9BWU1	CRBN	WO-2023081452-A1
TPD-OWZ8YS	SCHEMBL25418151	3-Amino-4-[4-[4-[4-[3-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethoxy]propanoyl]piperazine-1-carbonyl]phenyl]-1,4-diazepan-1-yl]thieno[2,3-b]pyridine-2-carboxamide; SCHEMBL30369600	NC(=O)c1sc2nccc(N3CCCN(c4ccc(C(=O)N5CCN(C(=O)CCOCCOCCOCCOCCNc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)cc4)CC3)c2c1N	C48H58N10O11S	CDK8;CDK19	P49336/Q9BWU1	CRBN	WO-2023081452-A1
TPD-MR2OE4	WO2023081452A1_81	.	CC(C)(C)C(=O)OCN1C(=O)CCC(N2C(=O)c3cccc(NCCCC(=O)NCCCCCCCCCCC(=O)N4CCN(C(=O)Cn5cc(-c6ccc(-c7cccc8cnccc78)cc6)cn5)CC4)c3C2=O)C1=O	C58H69N9O9	CDK8;CDK19	P49336/Q9BWU1	CRBN	WO-2023081452-A1
TPD-ZHOM2Q	SCHEMBL25417230	2-(2,6-Dioxopiperidin-3-yl)-4-[2-[2-[2-[3-[4-[2-[4-(4-isoquinolin-4-ylphenyl)pyrazol-1-yl]acetyl]piperazin-1-yl]-3-oxopropoxy]ethoxy]ethoxy]ethylamino]isoindole-1,3-dione; SCHEMBL30369920	O=C1CCC(N2C(=O)c3cccc(NCCOCCOCCOCCC(=O)N4CCN(C(=O)Cn5cc(-c6ccc(-c7cncc8ccccc78)cc6)cn5)CC4)c3C2=O)C(=O)N1	C46H48N8O9	CDK8;CDK19	P49336/Q9BWU1	CRBN	WO-2023081452-A1
TPD-HEHUFW	SCHEMBL30369836	2-(2,6-Dioxopiperidin-3-yl)-4-[[5-[4-[2-[4-(4-isoquinolin-4-ylphenyl)pyrazol-1-yl]acetyl]piperazin-1-yl]-5-oxopentyl]amino]isoindole-1,3-dione	O=C1CCC(N2C(=O)c3cccc(NCCCCC(=O)N4CCN(C(=O)Cn5cc(-c6ccc(-c7cncc8ccccc78)cc6)cn5)CC4)c3C2=O)C(=O)N1	C42H40N8O6	CDK8;CDK19	P49336/Q9BWU1	CRBN	WO-2023081452-A1
TPD-XO0SNC	SCHEMBL26160087	3-[4-[1-[2-[4-[4-[(4-Anilino-5-chloropyrimidin-2-yl)amino]-3-methoxyphenyl]piperazin-1-yl]-2-oxoethyl]piperidin-4-yl]anilino]piperidine-2,6-dione	COC1=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=CC=C1NC1=NC=C(Cl)C(NC2=CC=CC=C2)=N1	C39H44ClN9O4	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-SH25BM	SCHEMBL26160088	3-[4-[1-[2-[4-[4-[[4-Anilino-5-(trifluoromethyl)pyrimidin-2-yl]amino]-3-methoxyphenyl]piperazin-1-yl]-2-oxoethyl]piperidin-4-yl]anilino]piperidine-2,6-dione	COC1=C(NC2=NC=C(C(F)(F)F)C(NC3=CC=CC=C3)=N2)C=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C40H44F3N9O4	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-BQZF3O	SCHEMBL26160089	3-[4-[1-[2-[4-[4-[[5-Chloro-4-(4-fluoroanilino)pyrimidin-2-yl]amino]-3-methoxyphenyl]piperazin-1-yl]-2-oxoethyl]piperidin-4-yl]anilino]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=CC=C(F)C=C3)=N2)C=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C39H43ClFN9O4	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-DMJN9K	SCHEMBL26160090	3-[4-[1-[2-[4-[4-[(4-Anilino-5-chloropyrimidin-2-yl)amino]-3-methoxyphenyl]piperazin-1-yl]-2-oxoethyl]piperidin-4-yl]-3-fluoroanilino]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=CC=CC=C3)=N2)C=CC(N2CCN(C(=O)CN3CCC(C4=C(F)C=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C39H43ClFN9O4	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-AN0S8N	SCHEMBL26160092	N-[5-[(4-anilino-5-chloropyrimidin-2-yl)amino]-2-[4-[2-[4-[4-[(2,6-dioxopiperidin-3-yl)amino]phenyl]piperidin-1-yl]acetyl]piperazin-1-yl]-4-methoxyphenyl]acetamide	COC1=C(NC2=NC=C(Cl)C(NC3=CC=CC=C3)=N2)C=C(NC(C)=O)C(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C41H47ClN10O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-1KD55J	SCHEMBL26160093	N-[5-[(4-anilino-5-chloropyrimidin-2-yl)amino]-2-[4-[2-[4-[4-[(2,6-dioxopiperidin-3-yl)amino]phenyl]piperidin-1-yl]acetyl]piperazin-1-yl]-4-methoxyphenyl]propanamide	CCC(=O)NC1=CC(NC2=NC=C(Cl)C(NC3=CC=CC=C3)=N2)=C(OC)C=C1N1CCN(C(=O)CN2CCC(C3=CC=C(NC4CCC(=O)NC4=O)C=C3)CC2)CC1	C42H49ClN10O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-W0N5FG	SCHEMBL26160094	3-[4-[1-[2-[4-[1-[4-[(4-Anilino-5-chloropyrimidin-2-yl)amino]-3-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]-2-oxoethyl]piperidin-4-yl]anilino]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=CC=CC=C3)=N2)C=CC(N2CCC(N3CCN(C(=O)CN4CCC(C5=CC=C(NC6CCC(=O)NC6=O)C=C5)CC4)CC3)CC2)=C1	C44H53ClN10O4	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-VNRVQA	SCHEMBL26160133	3-[4-[1-[2-[4-[4-[[5-Chloro-4-(3-fluoroanilino)pyrimidin-2-yl]amino]-3-methoxyphenyl]piperazin-1-yl]-2-oxoethyl]piperidin-4-yl]anilino]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=CC(F)=CC=C3)=N2)C=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C39H43ClFN9O4	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-U8B7E1	SCHEMBL26160137	3-[4-[1-[2-[4-[4-[[5-Chloro-4-(2-fluoroanilino)pyrimidin-2-yl]amino]-3-methoxyphenyl]piperazin-1-yl]-2-oxoethyl]piperidin-4-yl]anilino]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C(F)C=CC=C3)=N2)C=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C39H43ClFN9O4	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-8VDG04	SCHEMBL26160575	3-[[5-[4-[2-[4-[4-[[4-(2-Acetylanilino)-5-chloropyrimidin-2-yl]amino]-3-methoxyphenyl]piperazin-1-yl]-2-oxoethyl]piperazin-1-yl]pyridin-2-yl]amino]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C(C(C)=O)C=CC=C3)=N2)C=CC(N2CCN(C(=O)CN3CCN(C4=CC=C(NC5CCC(=O)NC5=O)N=C4)CC3)CC2)=C1	C39H44ClN11O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-BIBRX5	SCHEMBL26160658	3-[6-[4-[2-[4-[4-[[4-(2-acetylanilino)-5-chloropyrimidin-2-yl]amino]-3-methoxyphenyl]piperazin-1-yl]-2-oxoethyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C(C(C)=O)C=CC=C3)=N2)C=CC(N2CCN(C(=O)CN3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)CC5=C4)CC3)CC2)=C1	C42H45ClN10O6	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-B56I59	SCHEMBL26160140	3-[4-[1-[2-[4-[4-[[5-Chloro-4-(3-chloro-4-fluoroanilino)pyrimidin-2-yl]amino]-3-methoxyphenyl]piperazin-1-yl]-2-oxoethyl]piperidin-4-yl]anilino]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=CC(Cl)=C(F)C=C3)=N2)C=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C39H42Cl2FN9O4	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-SBDLGP	SCHEMBL26160143	3-[4-[1-[2-[4-[4-[[4-(2-Acetylanilino)-5-chloropyrimidin-2-yl]amino]-3-methoxyphenyl]piperazin-1-yl]-2-oxoethyl]piperidin-4-yl]anilino]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C(C(C)=O)C=CC=C3)=N2)C=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C41H46ClN9O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-IJ8SDH	WO2023088385A1_T-121	.	COC1=C(NC2=NC=C(Cl)C(NC3=C(C(C)=O)C=CC=C3)=N2)C=CC(N2CCC(N3CCN(C(=O)CN4CCC(C5=CC=C(NC6CCC(=O)NC6=O)C=C5)CC4)CC3)CC2)=C1	C46H55ClN10O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-VC4NE7	SCHEMBL26160605	3-[4-[1-[2-[4-[4-[(4-Anilino-5-chloropyrimidin-2-yl)amino]-3-methoxyphenyl]-3-methylpiperazin-1-yl]-2-oxoethyl]piperidin-4-yl]anilino]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=CC=CC=C3)=N2)C=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2C)=C1	C40H46ClN9O4	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-A4DCGA	SCHEMBL26160606	3-[4-[1-[2-[4-[4-[(4-Anilino-5-chloropyrimidin-2-yl)amino]-3-methoxyphenyl]-2-methylpiperazin-1-yl]-2-oxoethyl]piperidin-4-yl]anilino]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=CC=CC=C3)=N2)C=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)C(C)C2)=C1	C40H46ClN9O4	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-KRHMUV	SCHEMBL26160607	3-[4-[1-[2-[3-[4-[[4-(2-Acetylanilino)-5-chloropyrimidin-2-yl]amino]-3-methoxyphenyl]-3,6-diazabicyclo[3.1.1]heptan-6-yl]-2-oxoethyl]piperidin-4-yl]anilino]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C(C(C)=O)C=CC=C3)=N2)C=CC(N2CC3CC(C2)N3C(=O)CN2CCC(C3=CC=C(NC4CCC(=O)NC4=O)C=C3)CC2)=C1	C42H46ClN9O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-DXC7TN	SCHEMBL26160608	3-[4-[1-[2-[6-[4-[(4-Anilino-5-chloropyrimidin-2-yl)amino]-3-methoxyphenyl]-2,6-diazaspiro[3.3]heptan-2-yl]-2-oxoethyl]piperidin-4-yl]anilino]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=CC=CC=C3)=N2)C=CC(N2CC3(CN(C(=O)CN4CCC(C5=CC=C(NC6CCC(=O)NC6=O)C=C5)CC4)C3)C2)=C1	C40H44ClN9O4	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-B35J2A	SCHEMBL26160628	3-[4-[1-[2-[4-[4-[(4-Anilino-5-chloropyrimidin-2-yl)amino]-3-methoxyphenyl]piperidin-1-yl]-2-oxoethyl]piperidin-4-yl]anilino]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=CC=CC=C3)=N2)C=CC(C2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C40H45ClN8O4	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-I1YTTU	SCHEMBL26160144	3-[4-[1-[2-[4-[4-[[5-Chloro-4-(2-dimethylphosphorylanilino)pyrimidin-2-yl]amino]-3-methoxyphenyl]piperazin-1-yl]-2-oxoethyl]piperidin-4-yl]anilino]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C(P(C)(C)=O)C=CC=C3)=N2)C=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C41H49ClN9O5P	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-STHG1J	SCHEMBL26160631	3-[4-[1-[4-[[4-(2-Acetylanilino)-5-chloropyrimidin-2-yl]amino]-3-methoxybenzoyl]piperidin-4-yl]anilino]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C(C(C)=O)C=CC=C3)=N2)C=CC(C(=O)N2CCC(C3=CC=C(NC4CCC(=O)NC4=O)C=C3)CC2)=C1	C36H36ClN7O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-1A6H38	SCHEMBL26160632	3-[4-[1-[2-[4-[4-[[4-(2,4-Difluoroanilino)-5-(trifluoromethyl)pyrimidin-2-yl]amino]-3-methoxyphenyl]piperazin-1-yl]-2-oxoethyl]piperidin-4-yl]anilino]piperidine-2,6-dione	COC1=C(NC2=NC=C(C(F)(F)F)C(NC3=C(F)C=C(F)C=C3)=N2)C=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C40H42F5N9O4	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-JXNIZF	SCHEMBL26160633	3-[4-[1-[2-[4-[4-[[5-Chloro-4-(2,5-difluoroanilino)pyrimidin-2-yl]amino]-3-methoxyphenyl]piperazin-1-yl]-2-oxoethyl]piperidin-4-yl]anilino]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C(F)C=CC(F)=C3)=N2)C=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C39H42ClF2N9O4	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-BZWPDT	SCHEMBL26160634	3-[4-[1-[2-[4-[4-[[4-(3-Acetylanilino)-5-chloropyrimidin-2-yl]amino]-3-methoxyphenyl]piperazin-1-yl]-2-oxoethyl]piperidin-4-yl]anilino]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=CC(C(C)=O)=CC=C3)=N2)C=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C41H46ClN9O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-VYIGTM	WO2023088385A1_T-134	.	COC1=C(NC2=NC=C(Cl)C(NC3=CC(C#N)=CC=C3)=N2)C=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C40H43ClN10O4	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-2NI4LH	WO2023088385A1_T-135	.	COC1=C(NC2=NC=C(C(F)(F)F)C(C3=CN(C)C4=CC=CC=C34)=N2)C=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C43H46F3N9O4	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-6D31Z4	WO2023088385A1_T-136	.	COC1=C(NC2=NC=CC(C3=CN(C)C4=CC=CC=C34)=N2)C=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C42H47N9O4	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-L59YIB	WO2023088385A1_T-137	.	COC1=C(NC2=NC=C(Cl)C(OC3=CC=CC=C3)=N2)C=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C39H43ClN8O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-GJQC98	WO2023088385A1_T-138	.	COC1=C(NC2=NC=C(Cl)C(NC3=CC=CC=N3)=N2)C=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C38H43ClN10O4	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-TEMP5P	SCHEMBL26160636	2-[[5-Chloro-2-[4-[4-[2-[4-[4-[(2,6-dioxopiperidin-3-yl)amino]phenyl]piperidin-1-yl]acetyl]piperazin-1-yl]-2-methoxyanilino]pyrimidin-4-yl]amino]benzonitrile	COC1=C(NC2=NC=C(Cl)C(NC3=C(C#N)C=CC=C3)=N2)C=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C40H43ClN10O4	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-DPY0Q6	SCHEMBL26160145	1-[6-[1-[2-[4-[4-[(4-Anilino-5-chloropyrimidin-2-yl)amino]-3-methoxyphenyl]piperazin-1-yl]-2-oxoethyl]piperidin-4-yl]-1-methylindazol-3-yl]-1,3-diazinane-2,4-dione	COC1=C(NC2=NC=C(Cl)C(NC3=CC=CC=C3)=N2)C=CC(N2CCN(C(=O)CN3CCC(C4=CC=C5C(=C4)N(C)N=C5N4CCC(=O)NC4=O)CC3)CC2)=C1	C40H44ClN11O4	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-WAZ5Q0	SCHEMBL26160146	3-[6-[4-[2-[4-[4-[(4-anilino-5-chloropyrimidin-2-yl)amino]-3-methoxyphenyl]piperazin-1-yl]-2-oxoethyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=CC=CC=C3)=N2)C=CC(N2CCN(C(=O)CN3CCN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5)CC3)CC2)=C1	C40H43ClN10O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-PK4E41	SCHEMBL26161769	N-[(3R)-1-[4-[[4-(2-acetylanilino)-5-chloropyrimidin-2-yl]amino]-3-methoxyphenyl]piperidin-3-yl]-2-[4-[4-[(2,6-dioxopiperidin-3-yl)amino]phenyl]piperidin-1-yl]acetamide	COC1=C(NC2=NC=C(Cl)C(NC3=C(C(C)=O)C=CC=C3)=N2)C=CC(N2CCC[C@@H](NC(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)C2)=C1	C42H48ClN9O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-JDUF4N	WO2023088385A1_T-166	.	COC1=C(NC2=NC=C(Cl)C(NC3=C(C(C)=O)C=CC=C3)=N2)C=CC(N2CCC[C@H](NC(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)C2)=C1	C42H48ClN9O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-W69GVS	WO2023088385A1_T-167	.	COC1=C(NC2=NC=C(Cl)C(NC3=C(C(C)=O)C=CC=C3)=N2)C=CC(N2CCC[C@H](N(C)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)C2)=C1	C42H50ClN9O4	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-B917T4	WO2023088385A1_T-168	.	COC1=C(NC2=NC=C(Cl)C(NC3=C(C(C)=O)C=CC=C3)=N2)C=CC(N2CCC[C@@H](N(C)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)C2)=C1	C42H50ClN9O4	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-N905L5	SCHEMBL26160725	N-[1-[4-[[4-(2-acetylanilino)-5-chloropyrimidin-2-yl]amino]-3-methoxyphenyl]azetidin-3-yl]-2-[4-[4-[(2,6-dioxopiperidin-3-yl)amino]phenyl]piperidin-1-yl]acetamide	COC1=C(NC2=NC=C(Cl)C(NC3=C(C(C)=O)C=CC=C3)=N2)C=CC(N2CC(NC(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)C2)=C1	C40H44ClN9O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-1ZD2YU	SCHEMBL26161771	N-[1-[4-[[4-(2-acetylanilino)-5-chloropyrimidin-2-yl]amino]-3-methoxyphenyl]azetidin-3-yl]-2-[4-[4-[(2,6-dioxopiperidin-3-yl)amino]phenyl]piperidin-1-yl]-N-methylacetamide	COC1=C(NC2=NC=C(Cl)C(NC3=C(C(C)=O)C=CC=C3)=N2)C=CC(N2CC(N(C)C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)C2)=C1	C41H46ClN9O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-OHSBBQ	SCHEMBL26160727	N-[(3R)-1-[4-[[4-(2-acetylanilino)-5-chloropyrimidin-2-yl]amino]-3-methoxyphenyl]pyrrolidin-3-yl]-2-[4-[4-[(2,6-dioxopiperidin-3-yl)amino]phenyl]piperidin-1-yl]-N-methylacetamide	COC1=C(NC2=NC=C(Cl)C(NC3=C(C(C)=O)C=CC=C3)=N2)C=CC(N2CC[C@@H](N(C)C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)C2)=C1	C42H48ClN9O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-QNY0UN	WO2023088385A1_T-172	.	COC1=C(NC2=NC=C(Cl)C(NC3=C(C(C)=O)C=CC=C3)=N2)C=CC(N2CC[C@H](N(C)C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)C2)=C1	C42H48ClN9O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-OJS24J	SCHEMBL26160729	N-[(3R)-1-[4-[[4-(2-acetylanilino)-5-chloropyrimidin-2-yl]amino]-3-methoxyphenyl]pyrrolidin-3-yl]-2-[4-[4-[(2,6-dioxopiperidin-3-yl)amino]phenyl]piperidin-1-yl]acetamide	COC1=C(NC2=NC=C(Cl)C(NC3=C(C(C)=O)C=CC=C3)=N2)C=CC(N2CC[C@@H](NC(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)C2)=C1	C41H46ClN9O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-X9J9EP	SCHEMBL26160730	N-[(3S)-1-[4-[[4-(2-acetylanilino)-5-chloropyrimidin-2-yl]amino]-3-methoxyphenyl]pyrrolidin-3-yl]-2-[4-[4-[(2,6-dioxopiperidin-3-yl)amino]phenyl]piperidin-1-yl]acetamide	COC1=C(NC2=NC=C(Cl)C(NC3=C(C(C)=O)C=CC=C3)=N2)C=CC(N2CC[C@H](NC(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)C2)=C1	C41H46ClN9O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-BSEJD0	SCHEMBL26160732	3-[4-[1-[2-[6-[4-[[4-(2-Acetylanilino)-5-chloropyrimidin-2-yl]amino]-3-methoxyphenyl]-3,6-diazabicyclo[3.1.1]heptan-3-yl]-2-oxoethyl]piperidin-4-yl]anilino]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C(C(C)=O)C=CC=C3)=N2)C=CC(N2C3CC2CN(C(=O)CN2CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC2)C3)=C1	C42H46ClN9O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-H6S3UU	SCHEMBL26160328	3-[4-[1-[2-[4-[4-[[4-(2-Acetylanilino)-5-(trifluoromethyl)pyrimidin-2-yl]amino]-3-methoxyphenyl]piperazin-1-yl]-2-oxoethyl]piperidin-4-yl]anilino]piperidine-2,6-dione	COC1=C(NC2=NC=C(C(F)(F)F)C(NC3=C(C(C)=O)C=CC=C3)=N2)C=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C42H46F3N9O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-67Y1VR	SCHEMBL26160751	3-[4-[4-[2-[4-[4-[[4-(2-Acetylanilino)-5-chloropyrimidin-2-yl]amino]-3-methoxyphenyl]piperazin-1-yl]-2-oxoethyl]piperidin-1-yl]anilino]piperidine-2,6-dione	COC1=C(NC2=NC(NC3=CC=CC=C3C(C)=O)=C(Cl)C=N2)C=CC(N2CCN(C(=O)CC3CCN(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C41H46ClN9O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-GM0UB7	SCHEMBL26160752	3-[4-[1-[2-[4-[4-[[4-(2-Acetylanilino)-5-chloropyrimidin-2-yl]amino]-3-propan-2-yloxyphenyl]piperazin-1-yl]-2-oxoethyl]piperidin-4-yl]anilino]piperidine-2,6-dione	CC(=O)C1=C(NC2=NC(NC3=C(OC(C)C)C=C(N4CCN(C(=O)CN5CCC(C6=CC=C(NC7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)=NC=C2Cl)C=CC=C1	C43H50ClN9O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-T27EKT	SCHEMBL26160702	N-[5-[[4-anilino-5-(trifluoromethyl)pyrimidin-2-yl]amino]-2-[4-[2-[4-[4-[(2,6-dioxopiperidin-3-yl)amino]phenyl]piperidin-1-yl]acetyl]piperazin-1-yl]-4-methoxyphenyl]prop-2-enamide	C=CC(=O)NC1=CC(NC2=NC=C(C(F)(F)F)C(NC3=CC=CC=C3)=N2)=C(OC)C=C1N1CCN(C(=O)CN2CCC(C3=CC=C(NC4CCC(=O)NC4=O)C=C3)CC2)CC1	C43H47F3N10O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-QOPFH9	SCHEMBL26160754	3-[3-[1-[2-[4-[4-[[4-(2-Acetylanilino)-5-chloropyrimidin-2-yl]amino]-3-methoxyphenyl]piperazin-1-yl]-2-oxoethyl]piperidin-4-yl]anilino]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C(C(C)=O)C=CC=C3)=N2)C=CC(N2CCN(C(=O)CN3CCC(C4=CC(NC5CCC(=O)NC5=O)=CC=C4)CC3)CC2)=C1	C41H46ClN9O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-986BZU	SCHEMBL26160755	3-[4-[1-[2-[4-[4-[[4-(2-Acetylanilino)-5-chloropyrimidin-2-yl]amino]-3-methoxyphenyl]piperazin-1-yl]ethyl]piperidin-4-yl]anilino]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C(C(C)=O)C=CC=C3)=N2)C=CC(N2CCN(CCN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C41H48ClN9O4	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-O7NEXN	SCHEMBL26160756	3-[4-[1-[3-[4-[4-[[4-(2-Acetylanilino)-5-chloropyrimidin-2-yl]amino]-3-methoxyphenyl]piperazin-1-yl]propyl]piperidin-4-yl]anilino]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C(C(C)=O)C=CC=C3)=N2)C=CC(N2CCN(CCCN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C42H50ClN9O4	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-HUFL7N	SCHEMBL26160757	2-[[5-chloro-2-[4-[4-[2-[4-[4-[(2,6-dioxopiperidin-3-yl)amino]phenyl]piperidin-1-yl]acetyl]piperazin-1-yl]-2-methoxyanilino]pyrimidin-4-yl]amino]-N-methylbenzamide	CNC(=O)C1=C(NC2=NC(NC3=C(OC)C=C(N4CCN(C(=O)CN5CCC(C6=CC=C(NC7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)=NC=C2Cl)C=CC=C1	C41H47ClN10O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-4919AF	SCHEMBL26160758	2-[[5-bromo-2-[4-[4-[2-[4-[4-[(2,6-dioxopiperidin-3-yl)amino]phenyl]piperidin-1-yl]acetyl]piperazin-1-yl]-2-methoxyanilino]pyrimidin-4-yl]amino]-N-methylbenzamide	CNC(=O)C1=C(NC2=NC(NC3=C(OC)C=C(N4CCN(C(=O)CN5CCC(C6=CC=C(NC7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)=NC=C2Br)C=CC=C1	C41H47BrN10O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-4MHE0J	SCHEMBL26160759	2-[[2-[4-[4-[2-[4-[4-[(2,6-dioxopiperidin-3-yl)amino]phenyl]piperidin-1-yl]acetyl]piperazin-1-yl]-2-methoxyanilino]-5-(trifluoromethyl)pyrimidin-4-yl]amino]-N-methylbenzamide	CNC(=O)C1=C(NC2=NC(NC3=C(OC)C=C(N4CCN(C(=O)CN5CCC(C6=CC=C(NC7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)=NC=C2C(F)(F)F)C=CC=C1	C42H47F3N10O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-DL157I	SCHEMBL26160760	3-[4-[4-[2-[4-[4-[[4-(2-Acetylanilino)-5-chloropyrimidin-2-yl]amino]-3-methoxyphenyl]piperazin-1-yl]-2-oxoethyl]-2-oxopiperazin-1-yl]anilino]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C(C(C)=O)C=CC=C3)=N2)C=CC(N2CCN(C(=O)CN3CCN(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)C(=O)C3)CC2)=C1	C40H43ClN10O6	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-9JGZTI	WO2023088385A1_T-188	.	COC1=C(NC2=NC=C(Cl)C(NC3=C(C(C)=O)C=CC=C3)=N2)C=CC(N2CC3CN(C(=O)CN4CCC(C5=CC=C(NC6CCC(=O)NC6=O)C=C5)CC4)CC3C2)=C1	C43H48ClN9O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-O0F3EK	SCHEMBL26160781	3-[4-[4-[2-[(3aR,6aS)-2-[4-[[4-(2-acetylanilino)-5-chloropyrimidin-2-yl]amino]-3-methoxyphenyl]-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-5-yl]-2-oxoethyl]piperazin-1-yl]anilino]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C(C(C)=O)C=CC=C3)=N2)C=CC(N2C[C@H]3CN(C(=O)CN4CCN(C5=CC=C(NC6CCC(=O)NC6=O)C=C5)CC4)C[C@H]3C2)=C1	C42H47ClN10O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-Z7G1CS	WO2023088385A1_T-190	.	COC1=C(NC2=NC=[C]([Cr])C(NC3=C(C(=O)C(C)C)C=CC=C3)=N2)C=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C43H50CrN9O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-NY8ZQF	WO2023088385A1_T-191	.	COC1=C(NC2=NC=C(Cl)C(NC3=C(C(C)=O)C=CC=C3)=N2)C=CC(N2C3CCC2CN(C(=O)CN2CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC2)C3)=C1	C43H48ClN9O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-2KVO1E	SCHEMBL26160782	3-[4-[1-[2-[4-[6-[[4-(2-Acetylanilino)-5-chloropyrimidin-2-yl]amino]pyridin-3-yl]piperazin-1-yl]-2-oxoethyl]piperidin-4-yl]anilino]piperidine-2,6-dione	CC(=O)C1=C(NC2=NC(NC3=NC=C(N4CCN(C(=O)CN5CCC(C6=CC=C(NC7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)=NC=C2Cl)C=CC=C1	C39H43ClN10O4	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-G9815Y	SCHEMBL26160783	3-[2-[1-[2-[4-[4-[[4-(2-Acetylanilino)-5-chloropyrimidin-2-yl]amino]-3-methoxyphenyl]piperazin-1-yl]-2-oxoethyl]piperidin-4-yl]anilino]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C(C(C)=O)C=CC=C3)=N2)C=CC(N2CCN(C(=O)CN3CCC(C4=C(NC5CCC(=O)NC5=O)C=CC=C4)CC3)CC2)=C1	C41H46ClN9O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-TW5NOK	WO2023088385A1_T-194	.	COC(=O)C1=C(NC2=NC(NC3=C(OC)C=C(N4CCN(C(=O)CN5CCC(C6=CC=C(NC7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)=NC=C2Cl)C=CC=C1	C41H46ClN9O6	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-KQ0CCU	WO2023088385A1_T-195	.	COC1=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=CC=C1NC1=NC(NC2=C(NC(C)=O)C=CC=C2)=C(Cl)C=N1	C41H47ClN10O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-Q561ND	SCHEMBL26160784	3-[4-[1-[2-[4-[4-[[5-Chloro-4-[2-(2-hydroxypropan-2-yl)anilino]pyrimidin-2-yl]amino]-3-methoxyphenyl]piperazin-1-yl]-2-oxoethyl]piperidin-4-yl]anilino]piperidine-2,6-dione	COC1=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=CC=C1NC1=NC(NC2=CC=CC=C2C(C)(C)O)=C(Cl)C=N1	C42H50ClN9O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-9SXV4Z	WO2023088385A1_T-197	.	COC1=C(NC2=NC=C(Cl)C(NC3=C(C(C)=O)C=CC=C3)=N2)C=CC(N2CCN(C(=O)CCCCN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C44H52ClN9O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-VB7A1I	WO2023088385A1_T-198	.	COC1=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=CC=C1NC1=NC(NC2=C(C(=O)N(C)C)C=CC=C2)=C(Cl)C=N1	C42H49ClN10O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-UMD8U1	SCHEMBL26160787	3-[4-[1-[2-[4-[4-[[5-Chloro-4-[4-fluoro-2-(2-hydroxypropan-2-yl)anilino]pyrimidin-2-yl]amino]-3-methoxyphenyl]piperazin-1-yl]-2-oxoethyl]piperidin-4-yl]anilino]piperidine-2,6-dione	COC1=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=CC=C1NC1=NC(NC2=CC=C(F)C=C2C(C)(C)O)=C(Cl)C=N1	C42H49ClFN9O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-86L7AX	SCHEMBL26160788	3-[4-[1-[2-[4-[4-[[5-Chloro-4-(2-methoxyanilino)pyrimidin-2-yl]amino]-3-methoxyphenyl]piperazin-1-yl]-2-oxoethyl]piperidin-4-yl]anilino]piperidine-2,6-dione	COC1=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=CC=C1NC1=NC(NC2=C(OC)C=CC=C2)=C(Cl)C=N1	C40H46ClN9O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-WFZIKL	SCHEMBL26160816	5-[4-[2-[4-[4-[[4-(2-Acetylanilino)-5-chloropyrimidin-2-yl]amino]-3-methoxyphenyl]piperazin-1-yl]-2-oxoethyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C(C(C)=O)C=CC=C3)=N2)C=CC(N2CCN(C(=O)CN3CCN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)=C1	C42H43ClN10O7	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-1GLBF9	SCHEMBL26160817	3-[4-[1-[2-[4-[4-[[5-Chloro-4-[(2-oxo-1,4-dihydro-3,1-benzoxazin-8-yl)amino]pyrimidin-2-yl]amino]-3-methoxyphenyl]piperazin-1-yl]-2-oxoethyl]piperidin-4-yl]anilino]piperidine-2,6-dione	COC1=C(NC2=NC(NC3=CC=CC4=C3NC(=O)OC4)=C(Cl)C=N2)C=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C41H45ClN10O6	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-UEVLC3	SCHEMBL26160818	3-[4-[1-[2-[4-[5-[[5-Chloro-4-(2-dimethylphosphorylanilino)pyrimidin-2-yl]amino]-6-methoxypyridin-2-yl]piperazin-1-yl]-2-oxoethyl]piperidin-4-yl]anilino]piperidine-2,6-dione	COC1=NC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=CC=C1NC1=NC=C(Cl)C(NC2=CC=CC=C2P(C)(C)=O)=N1	C40H48ClN10O5P	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-WNXYU3	WO2023088385A1_T-204	.	COC1=C(NC2=NC=C(Cl)C(NC3=C(C(C)=O)C=CC=C3)=N2)C=CC(N2CCN(C(=O)C3CCN(CC4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)CC2)=C1	C48H53ClN10O7	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-8RK3XI	WO2023088385A1_T-205	.	COC1=C(NC2=NC=C(Cl)C(NC3=C(C(C)=O)C=CC=C3)=N2)C=CC(N2CCN(C(=O)C3CCN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)=C1	C42H42ClN9O7	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-RJPJBX	SCHEMBL26160822	1-[4-[1-[2-[4-[4-[[4-(2-Acetylanilino)-5-chloropyrimidin-2-yl]amino]-3-methoxyphenyl]piperazin-1-yl]-2-oxoethyl]piperidin-4-yl]phenyl]-1,3-diazinane-2,4-dione	COC1=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(N5CCC(=O)NC5=O)C=C4)CC3)CC2)=CC=C1NC1=NC(NC2=CC=CC=C2C(C)=O)=C(Cl)C=N1	C40H44ClN9O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-JCDLQE	SCHEMBL26160823	3-[4-[1-[2-[4-[5-[[4-(2-Acetylanilino)-5-chloropyrimidin-2-yl]amino]-6-methoxypyridin-2-yl]piperazin-1-yl]-2-oxoethyl]piperidin-4-yl]anilino]piperidine-2,6-dione	COC1=NC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=CC=C1NC1=NC=C(Cl)C(NC2=CC=CC=C2C(C)=O)=N1	C40H45ClN10O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-LIJAB1	WO2023088385A1_T-211	.	COC1=CC(N2CCC(N3CCN(C(=O)CN4CCC(C5=CC=C(NC6CCC(=O)NC6=O)C=C5)CC4)CC3)CC2)=CC=C1NC1=NC=C(Cl)C(NC2=CC=CC=C2N(C)S(C)(=O)=O)=N1	C46H58ClN11O6S	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-SAPTVA	SCHEMBL26160826	5-[4-[2-[4-[4-[[4-(2-Acetylanilino)-5-chloropyrimidin-2-yl]amino]-3-methoxyphenyl]piperazin-1-yl]ethyl]piperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C(C(C)=O)C=CC=C3)=N2)C=CC(N2CCN(CCC3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)=C1	C43H46ClN9O6	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-8J0OAN	SCHEMBL26161787	3-[4-[1-[2-[4-[4-[[4-(2-Acetylanilino)-5-chloropyrimidin-2-yl]amino]-3-methoxyphenoxy]piperidin-1-yl]-2-oxoethyl]piperidin-4-yl]anilino]piperidine-2,6-dione	COC1=CC(OC2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=CC=C1NC1=NC=C(Cl)C(NC2=CC=CC=C2C(C)=O)=N1	C42H47ClN8O6	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-ROQWNJ	WO2023088385A1_T-215	.	COC1=C(NC2=NC=C(Cl)C(NC3=C(C(C)=O)C=CC=C3)=N2)C=CC(N2CCN(C(=O)C3CCN(CC4CCN(C5=CC=C(NC6CCC(=O)NC6=O)C=C5)CC4)CC3)CC2)=C1	C46H55ClN10O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-HIXD6U	SCHEMBL26160847	5-[4-[5-[4-[4-[[4-(2-Acetylanilino)-5-chloropyrimidin-2-yl]amino]-3-methoxyphenyl]piperazin-1-yl]-5-oxopentyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	COC1=C(NC2=NC(NC3=C(C(C)=O)C=CC=C3)=C(Cl)C=N2)C=CC(N2CCN(C(=O)CCCCN3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)=C1	C45H49ClN10O7	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-E5I3KE	SCHEMBL26160848	1-[3-[1-[2-[4-[4-[[4-(2-Acetylanilino)-5-chloropyrimidin-2-yl]amino]-3-methoxyphenyl]piperazin-1-yl]-2-oxoethyl]piperidin-4-yl]phenyl]-1,3-diazinane-2,4-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C(C(C)=O)C=CC=C3)=N2)C=CC(N2CCN(C(=O)CN3CCC(C4=CC(N5CCC(=O)NC5=O)=CC=C4)CC3)CC2)=C1	C40H44ClN9O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-3NU6ZY	SCHEMBL26160870	N-[2-[[5-chloro-2-[4-[4-[2-[4-[4-[(2,6-dioxopiperidin-3-yl)amino]phenyl]piperidin-1-yl]acetyl]piperazin-1-yl]-2-methoxyanilino]pyrimidin-4-yl]amino]phenyl]-N-methylmethanesulfonamide	COC1=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=CC=C1NC1=NC=C(Cl)C(NC2=CC=CC=C2N(C)S(C)(=O)=O)=N1	C41H49ClN10O6S	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-SOLSB9	WO2023088385A1_T-219	.	C=CC(=O)NC1=CC(NC2=NC(C3=CN(C)C4C=CC=CC34)=CC=N2)=C(OC)C=C1N(C)CCN(C)C(=O)CN1CCC(C2=CC=C(NC3CCC(=O)NC3=O)C=C2)CC1	C45H54N10O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-QRWY0M	WO2023088385A1_T-220	.	COC1=C(NC2=NC(NC3=C(N(C)S(C)(=O)=O)C=CC=C3)=C(Cl)C=N2)C=CC(N2CCC(N3CCN(C(=O)CCCCN4CCC(C5=CC=C(NC6CCC(=O)NC6=O)C=C5)CC4)CC3)CC2)=C1	C49H64ClN11O6S	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-TV8ANV	WO2023088385A1_T-221	.	COC1=C(NC2=NC(NC3=CC=CC=C3C(C)=O)=C(Cl)C=N2)C=CC(N2CCC(N3CCN(C(=O)CCCCN4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)CC2)=C1	C50H58ClN11O7	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-XANHKN	WO2023088385A1_T-222	.	COC1=C(NC2=NC(NC3=C(N(C)C(C)=O)C=CC=C3)=C(Cl)C=N2)C=CC(N2CCC(N3CCN(C(=O)CN4CCC(C5=CC=C(NC6CCC(=O)NC6=O)C=C5)CC4)CC3)CC2)=C1	C47H58ClN11O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-6M5B2X	SCHEMBL26160851	N-[1-[4-[[4-(2-acetylanilino)-5-(trifluoromethyl)pyrimidin-2-yl]amino]-3-methoxyphenyl]piperidin-4-yl]-2-[4-[4-[(2,6-dioxopiperidin-3-yl)amino]phenyl]piperidin-1-yl]-N-methylacetamide	COC1=C(NC2=NC=C(C(F)(F)F)C(NC3=C(C(C)=O)C=CC=C3)=N2)C=CC(N2CCC(N(C)C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C44H50F3N9O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-7HN6EK	SCHEMBL26160868	5-[4-[[1-[4-[[4-(2-Acetylanilino)-5-chloropyrimidin-2-yl]amino]-3-methoxyphenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	COC1=C(NC2=NC=C(Cl)C(NC3=CC=CC=C3C(C)=O)=N2)C=CC(N2CCC(CN3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)=C1	C42H44ClN9O6	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-H6ZQDO	WO2023088385A1_T-226	.	COC1=C(NC2=NC=C(Cl)C(NC3=CC=CC=C3C(C)=O)=N2)C=CC(N2CCN(CC3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)=C1	C42H44ClN9O6	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-IBRYHV	WO2023088385A1_T-228	.	COC1=C(NC2=NC(NC3=C(C(C)=O)C=CC=C3)=C(Cl)C=N2)C=CC(N2CCC(N(C)C(=O)C3CCN(CC4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)CC2)=C1	C50H57ClN10O7	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-VV8M9A	SCHEMBL26160871	3-[4-[1-[2-[4-[4-[[4-(2-Acetylanilino)-5-chloropyrimidin-2-yl]amino]-3-methoxybenzoyl]piperazin-1-yl]-2-oxoethyl]piperidin-4-yl]anilino]piperidine-2,6-dione	COC1=CC(C(=O)N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=CC=C1NC1=NC=C(Cl)C(NC2=CC=CC=C2C(C)=O)=N1	C42H46ClN9O6	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-G6SRHG	SCHEMBL26160872	5-[[2-[4-[4-[[4-(2-Acetylanilino)-5-chloropyrimidin-2-yl]amino]-3-methoxyphenyl]piperazin-1-yl]-2-oxoethyl]amino]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	COC1=C(NC2=NC(NC3=CC=CC=C3C(C)=O)=C(Cl)C=N2)C=CC(N2CCN(C(=O)CNC3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)=C1	C38H36ClN9O7	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-UFUZ7P	SCHEMBL26160873	5-[4-[2-[4-[4-[[4-(2-Acetylanilino)-5-chloropyrimidin-2-yl]amino]-3-methoxyphenyl]piperazin-1-yl]-2-oxoethyl]piperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	COC1=C(NC2=NC(NC3=CC=CC=C3C(C)=O)=C(Cl)C=N2)C=CC(N2CCN(C(=O)CC3CCN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)=C1	C43H44ClN9O7	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-7QT4OK	SCHEMBL26160874	3-[4-[4-[4-[4-[[4-(2-Acetylanilino)-5-chloropyrimidin-2-yl]amino]-3-methoxyphenyl]piperazine-1-carbonyl]piperidine-1-carbonyl]anilino]piperidine-2,6-dione	COC1=CC(N2CCN(C(=O)C3CCN(C(=O)C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=CC=C1NC1=NC(NC2=CC=CC=C2C(C)=O)=C(Cl)C=N1	C41H44ClN9O6	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-IPCHNI	WO2023088385A1_T-233	.	COC1=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C(C2=CN(C)N=C2)C=C1NC1=NC=C(Cl)C(NC2=CC=CC=C2C(C)=O)=N1	C45H50ClN11O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-WXLE5K	WO2023088385A1_T-237	.	C=CC(=O)NC1=CC(NC2=NC(C3=CN(C)C4=C3C=CC=C4)=CC=N2)=C(OC)C=C1N1CCN(CC(=O)N2CCC(C3=CC=C(NC4CCC(=O)NC4=O)C=C3)CC2)CC1	C45H50N10O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-QCVCP1	WO2023088385A1_T-239	.	COC1=C(NC(=O)CN2CCC(C3=CC=C(NC4CCC(=O)NC4=O)C=C3)CC2)C=NC(N2CCN(C3=CC=C(Cl)C(NC4=CC=CC=C4C(C)=O)=N3)CC2)=C1	C41H46ClN9O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-Z64QHT	WO2023088385A1_T-240	.	COC1=C(NC2=NC=C(Cl)C(NC3=C(C(C)=O)C=CC=C3)=N2)C=CC(N2CCN(C(=O)C3CCN(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C40H44ClN9O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-ZYWH8Q	SCHEMBL26160893	2-[[5-chloro-2-[4-[4-[2-[4-[4-[(2,6-dioxopiperidin-3-yl)amino]phenyl]piperidin-1-yl]acetyl]piperazin-1-yl]-2-methoxy-5-methylanilino]pyrimidin-4-yl]amino]-N,N-dimethylbenzamide	COC1=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C(C)C=C1NC1=NC(NC2=C(C(=O)N(C)C)C=CC=C2)=C(Cl)C=N1	C43H51ClN10O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-6RZGTW	SCHEMBL26162025	3-[4-[1-[2-[4-[4-[[4-(2-Acetylanilino)-5-chloropyrimidin-2-yl]amino]-3-methoxyphenyl]piperazin-1-yl]-2-oxoethyl]pyrrolidin-3-yl]anilino]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C(C(C)=O)C=CC=C3)=N2)C=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)C3)CC2)=C1	C40H44ClN9O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-8SWKJ2	SCHEMBL26160896	3-[4-[1-[2-[4-[4-[[5-Chloro-4-[4-chloro-2-(2-hydroxypropan-2-yl)anilino]pyrimidin-2-yl]amino]-3-methoxyphenyl]piperazin-1-yl]-2-oxoethyl]piperidin-4-yl]anilino]piperidine-2,6-dione	COC1=C(NC2=NC(NC3=CC=C(Cl)C=C3C(C)(C)O)=C(Cl)C=N2)C=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C42H49Cl2N9O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-32Z097	SCHEMBL26160897	3-[4-[1-[2-[4-[5-[[4-(2-Acetylanilino)-5-chloropyrimidin-2-yl]amino]-4-methoxypyridin-2-yl]piperazin-1-yl]-2-oxoethyl]piperidin-4-yl]anilino]piperidine-2,6-dione	COC1=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=NC=C1NC1=NC=C(Cl)C(NC2=CC=CC=C2C(C)=O)=N1	C40H45ClN10O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-BIW6X2	SCHEMBL26160968	3-[4-[1-[2-[4-[4-[[4-(2-Acetyl-4-methoxyanilino)-5-chloropyrimidin-2-yl]amino]-3-methoxyphenyl]piperazin-1-yl]-2-oxoethyl]piperidin-4-yl]anilino]piperidine-2,6-dione	COC1=CC=C(NC2=C(Cl)C=NC(NC3=C(OC)C=C(N4CCN(C(=O)CN5CCC(C6=CC=C(NC7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)=N2)C(C(C)=O)=C1	C42H48ClN9O6	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-T2YD7R	SCHEMBL26160972	2-[[2-[4-[4-[2-[4-[4-[(2,6-dioxopiperidin-3-yl)amino]phenyl]piperidin-1-yl]acetyl]piperazin-1-yl]-2-methoxyanilino]-5-(trifluoromethyl)pyrimidin-4-yl]amino]-N,N-dimethylbenzamide	COC1=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=CC=C1NC1=NC(NC2=C(C(=O)N(C)C)C=CC=C2)=C(C(F)(F)F)C=N1	C43H49F3N10O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-UYNNSL	SCHEMBL26160973	2-[[5-chloro-2-[4-[4-[2-[4-[4-[(2,6-dioxopiperidin-3-yl)amino]phenyl]piperidin-1-yl]acetyl]piperazin-1-yl]-2-methoxy-5-methylanilino]pyrimidin-4-yl]amino]-N-methylbenzamide	CNC(=O)C1=C(NC2=NC(NC3=C(OC)C=C(N4CCN(C(=O)CN5CCC(C6=CC=C(NC7CCC(=O)NC7=O)C=C6)CC5)CC4)C(C)=C3)=NC=C2Cl)C=CC=C1	C42H49ClN10O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-0SPTE9	WO2023088385A1_T-258	.	COC1=C(NC2=NC=C(Cl)C(NC3=C(P(C)(C)=O)C=CC=C3)=N2)C=NC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C40H48ClN10O5P	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-K90FYA	SCHEMBL26160977	2-[[5-chloro-2-[4-[4-[2-[4-[4-[(2,6-dioxopiperidin-3-yl)amino]phenyl]piperidin-1-yl]acetyl]piperazin-1-yl]-2-methoxyanilino]pyrimidin-4-yl]amino]-N-propan-2-ylbenzamide	COC1=C(NC2=NC(NC3=C(C(=O)NC(C)C)C=CC=C3)=C(Cl)C=N2)C=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C43H51ClN10O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-1AYRHD	SCHEMBL26161091	2-[[2-[4-[4-[2-[4-[4-[(2,6-dioxopiperidin-3-yl)amino]phenyl]piperidin-1-yl]acetyl]piperazin-1-yl]-2-methoxyanilino]-5-(trifluoromethyl)pyrimidin-4-yl]amino]-N-phenylbenzamide	COC1=C(NC2=NC(NC3=C(C(=O)NC4=CC=CC=C4)C=CC=C3)=C(C(F)(F)F)C=N2)C=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C47H49F3N10O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-3BK4TG	SCHEMBL26161195	2-[[5-chloro-2-[4-[4-[3-[4-[(2,6-dioxopiperidin-3-yl)amino]phenyl]cyclobutanecarbonyl]piperazin-1-yl]-2-methoxyanilino]pyrimidin-4-yl]amino]-N-methylbenzamide	CNC(=O)C1=C(NC2=NC(NC3=C(OC)C=C(N4CCN(C(=O)C5CC(C6=CC=C(NC7CCC(=O)NC7=O)C=C6)C5)CC4)C=C3)=NC=C2Cl)C=CC=C1	C39H42ClN9O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-EKO8T6	SCHEMBL26161210	5-[[4-(2-Acetylanilino)-5-chloropyrimidin-2-yl]amino]-2-[4-[2-[4-[4-[(2,6-dioxopiperidin-3-yl)amino]phenyl]piperidin-1-yl]acetyl]piperazin-1-yl]-4-methoxybenzonitrile	COC1=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C(C#N)C=C1NC1=NC=C(Cl)C(NC2=CC=CC=C2C(C)=O)=N1	C42H45ClN10O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-7BVJMJ	SCHEMBL26161401	3-[5-[4-[2-[4-[4-[[4-Anilino-5-(trifluoromethyl)pyrimidin-2-yl]amino]-3-methoxyphenyl]piperazin-1-yl]-2-oxoethyl]piperazin-1-yl]indazol-1-yl]piperidine-2,6-dione	COC1=C(NC2=NC=C(C(F)(F)F)C(NC3=CC=CC=C3)=N2)C=CC(N2CCN(C(=O)CN3CCN(C4=CC5=C(C=C4)N(C4CCC(=O)NC4=O)N=C5)CC3)CC2)=C1	C40H42F3N11O4	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-JNR66H	SCHEMBL26161404	3-[5-[1-[2-[4-[4-[(4-Anilino-5-chloropyrimidin-2-yl)amino]-3-methoxyphenyl]piperazin-1-yl]-2-oxoethyl]piperidin-4-yl]indazol-1-yl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=CC=CC=C3)=N2)C=CC(N2CCN(C(=O)CN3CCC(C4=CC5=C(C=C4)N(C4CCC(=O)NC4=O)N=C5)CC3)CC2)=C1	C40H43ClN10O4	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-S50RRD	WO2023088385A1_T-327	.	COC1=C(NC2=NC=C(Cl)C(NC3=C(P(C)(C)=O)C=CC=C3)=N2)C=C(C)C(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C42H51ClN9O5P	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-W411GC	SCHEMBL26161405	3-[4-[1-[2-[4-[4-[(4-Anilino-5-chloropyrimidin-2-yl)amino]-3-chlorophenyl]piperazin-1-yl]-2-oxoethyl]piperidin-4-yl]anilino]piperidine-2,6-dione	O=C1CCC(NC2=CC=C(C3CCN(CC(=O)N4CCN(C5=CC(Cl)=C(NC6=NC=C(Cl)C(NC7=CC=CC=C7)=N6)C=C5)CC4)CC3)C=C2)C(=O)N1	C38H41Cl2N9O3	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-84RMTP	SCHEMBL26161406	3-[4-[1-[2-[4-[4-[[5-Chloro-4-(2-dimethylphosphorylanilino)pyrimidin-2-yl]amino]-3-methoxybenzoyl]piperazin-1-yl]-2-oxoethyl]piperidin-4-yl]anilino]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C(P(C)(C)=O)C=CC=C3)=N2)C=CC(C(=O)N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C42H49ClN9O6P	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-DMC8YK	SCHEMBL26161407	3-[4-[1-[2-[4-[3-Chloro-4-[[5-chloro-4-(2-dimethylphosphorylanilino)pyrimidin-2-yl]amino]phenyl]piperazin-1-yl]-2-oxoethyl]piperidin-4-yl]anilino]piperidine-2,6-dione	CP(C)(=O)C1=C(NC2=NC(NC3=C(Cl)C=C(N4CCN(C(=O)CN5CCC(C6=CC=C(NC7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)=NC=C2Cl)C=CC=C1	C40H46Cl2N9O4P	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-5MNCNI	SCHEMBL26161408	3-[4-[1-[2-[4-[4-[[5-Chloro-4-(2-dimethylphosphorylanilino)pyrimidin-2-yl]amino]-3-methoxyphenyl]piperidin-1-yl]-2-oxoethyl]piperidin-4-yl]anilino]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C(P(C)(C)=O)C=CC=C3)=N2)C=CC(C2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C42H50ClN8O5P	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-BTH6I1	SCHEMBL26162033	1-[[4-[1-[2-[4-[4-[[4-(2-Acetylanilino)-5-chloropyrimidin-2-yl]amino]-3-methoxyphenyl]piperazin-1-yl]-2-oxoethyl]piperidin-4-yl]phenyl]methyl]pyrimidine-2,4-dione	COC1=C(NC2=NC(NC3=C(C(C)=O)C=CC=C3)=C(Cl)C=N2)C=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(CN5C=CC(=O)NC5=O)C=C4)CC3)CC2)=C1	C41H44ClN9O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-OU8G96	SCHEMBL26161423	3-[4-[1-[2-[4-[4-[[4-(2-Acetylanilino)-5-chloropyrimidin-2-yl]amino]-3-chlorophenyl]piperazin-1-yl]-2-oxoethyl]piperidin-4-yl]anilino]piperidine-2,6-dione	CC(=O)C1=C(NC2=NC(NC3=C(Cl)C=C(N4CCN(C(=O)CN5CCC(C6=CC=C(NC7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)=NC=C2Cl)C=CC=C1	C40H43Cl2N9O4	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-7CBOPT	SCHEMBL26160392	3-[4-[1-[2-[4-[4-[[4-(2-Acetylanilino)-5-chloropyrimidin-2-yl]amino]-3-methoxyphenyl]piperidin-1-yl]-2-oxoethyl]piperidin-4-yl]anilino]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C(C(C)=O)C=CC=C3)=N2)C=CC(C2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C42H47ClN8O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-9NUGQN	SCHEMBL26161712	N-[5-[(4-anilino-5-chloropyrimidin-2-yl)amino]-2-[4-[2-[4-[4-[(2,6-dioxopiperidin-3-yl)amino]phenyl]piperidin-1-yl]acetyl]piperazin-1-yl]-4-methoxyphenyl]prop-2-enamide	C=CC(=O)NC1=CC(NC2=NC=C(Cl)C(NC3=CC=CC=C3)=N2)=C(OC)C=C1N1CCN(C(=O)CN2CCC(C3=CC=C(NC4CCC(=O)NC4=O)C=C3)CC2)CC1	C42H47ClN10O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-P2JFHP	SCHEMBL26161425	N-[1-[4-[[4-(2-acetylanilino)-5-chloropyrimidin-2-yl]amino]-3-methoxyphenyl]piperidin-4-yl]-2-[4-[4-[(2,6-dioxopiperidin-3-yl)amino]phenyl]piperidin-1-yl]acetamide	COC1=C(NC2=NC=C(Cl)C(NC3=C(C(C)=O)C=CC=C3)=N2)C=CC(N2CCC(NC(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C42H48ClN9O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-MSUOFI	SCHEMBL26161426	1-[[4-[1-[2-[4-[4-[[4-(2-Acetylanilino)-5-chloropyrimidin-2-yl]amino]-3-methoxyphenyl]piperazin-1-yl]-2-oxoethyl]piperidin-4-yl]phenyl]methyl]-1,3-diazinane-2,4-dione	COC1=C(NC2=NC(NC3=C(C(C)=O)C=CC=C3)=C(Cl)C=N2)C=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(CN5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C41H46ClN9O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-PB6U5V	SCHEMBL26161427	3-[4-[1-[2-[4-[4-[[4-(2-Acetylanilino)-5-chloropyrimidin-2-yl]amino]-3-methoxyphenyl]piperazin-1-yl]acetyl]piperidin-4-yl]anilino]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C(C(C)=O)C=CC=C3)=N2)C=CC(N2CCN(CC(=O)N3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C41H46ClN9O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-M43OQ2	SCHEMBL26161429	methyl N-[2-[[5-chloro-2-[4-[4-[2-[4-[4-[(2,6-dioxopiperidin-3-yl)amino]phenyl]piperidin-1-yl]acetyl]piperazin-1-yl]-2-methoxyanilino]pyrimidin-4-yl]amino]phenyl]carbamate	COC(=O)NC1=C(NC2=NC(NC3=C(OC)C=C(N4CCN(C(=O)CN5CCC(C6=CC=C(NC7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)=NC=C2Cl)C=CC=C1	C41H47ClN10O6	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-8JD4KI	SCHEMBL26161430	2-[[5-chloro-2-[4-[4-[2-[4-[4-[(2,6-dioxopiperidin-3-yl)amino]phenyl]piperidin-1-yl]acetyl]piperazin-1-yl]-2-methoxyanilino]pyrimidin-4-yl]amino]-N-cyclopentylbenzamide	COC1=C(NC2=NC(NC3=C(C(=O)NC4CCCC4)C=CC=C3)=C(Cl)C=N2)C=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C45H53ClN10O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-4BP2WY	WO2023088385A1_T-344	.	COC1=C(NC2=NC=C(Cl)C(NC3=CC=CC=C3)=N2)C=CC(N2CCN(C(=O)N3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)CC5=C4)CC3)CC2)=C1	C39H41ClN10O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-FYWBFC	SCHEMBL26162077	3-[6-[4-[4-[4-[[4-anilino-5-(trifluoromethyl)pyrimidin-2-yl]amino]-3-methoxyphenyl]piperazine-1-carbonyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	COC1=C(NC2=NC=C(C(F)(F)F)C(NC3=CC=CC=C3)=N2)C=CC(N2CCN(C(=O)N3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)CC5=C4)CC3)CC2)=C1	C40H41F3N10O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-5TNTFY	SCHEMBL26161448	3-[4-[1-[2-[4-[4-[(4-Anilino-5-chloropyrimidin-2-yl)amino]-3-methoxyphenyl]piperazin-1-yl]-2-oxoethyl]piperidin-4-yl]-2-fluoroanilino]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=CC=CC=C3)=N2)C=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C(F)=C4)CC3)CC2)=C1	C39H43ClFN9O4	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-23KEK4	SCHEMBL26161449	3-[4-[1-[2-[4-[4-[(4-Anilinopyrimidin-2-yl)amino]-3-methoxyphenyl]piperazin-1-yl]-2-oxoethyl]piperidin-4-yl]anilino]piperidine-2,6-dione	COC1=C(NC2=NC=CC(NC3=CC=CC=C3)=N2)C=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C39H45N9O4	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-ANB8CV	SCHEMBL26161450	3-[4-[1-[2-[4-[4-[[4-Anilino-5-(trifluoromethyl)pyrimidin-2-yl]amino]-3-methoxyphenyl]piperazin-1-yl]-2-oxoethyl]piperidin-4-yl]-2-fluoroanilino]piperidine-2,6-dione	COC1=C(NC2=NC=C(C(F)(F)F)C(NC3=CC=CC=C3)=N2)C=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C(F)=C4)CC3)CC2)=C1	C40H43F4N9O4	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-GYDXIL	SCHEMBL26161451	3-[[2-[4-[4-[2-[4-[4-[(2,6-Dioxopiperidin-3-yl)amino]phenyl]piperidin-1-yl]acetyl]piperazin-1-yl]-2-methoxyanilino]-5-(trifluoromethyl)pyrimidin-4-yl]amino]benzonitrile	COC1=C(NC2=NC=C(C(F)(F)F)C(NC3=CC(C#N)=CC=C3)=N2)C=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C41H43F3N10O4	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-8MHSVP	WO2023088385A1_T-350	.	COC1=C(NC2=NC=C(C(F)(F)F)C(OC3=CC=CC=C3)=N2)C=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C40H43F3N8O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-HN5CXD	SCHEMBL26161453	3-[5-[4-[2-[4-[4-[[4-Anilino-5-(trifluoromethyl)pyrimidin-2-yl]amino]-3-methoxyphenyl]piperazin-1-yl]-2-oxoethyl]piperazin-1-yl]indazol-2-yl]piperidine-2,6-dione	COC1=C(NC2=NC=C(C(F)(F)F)C(NC3=CC=CC=C3)=N2)C=CC(N2CCN(C(=O)CN3CCN(C4=CC5=CN(C6CCC(=O)NC6=O)N=C5C=C4)CC3)CC2)=C1	C40H42F3N11O4	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-S3HN9Q	SCHEMBL26161454	3-[4-[1-[2-[4-[4-[[4-(2-Acetylanilino)-5-(trifluoromethyl)pyrimidin-2-yl]amino]-3-methoxyphenyl]piperazin-1-yl]-2-oxoethyl]piperidin-4-yl]anilino]-1-methylpiperidine-2,6-dione	COC1=C(NC2=NC=C(C(F)(F)F)C(NC3=C(C(C)=O)C=CC=C3)=N2)C=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)N(C)C5=O)C=C4)CC3)CC2)=C1	C43H48F3N9O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-5DL59M	SCHEMBL26161455	N-[1-[4-[[4-(2-acetylanilino)-5-chloropyrimidin-2-yl]amino]-3-methoxyphenyl]piperidin-4-yl]-2-[4-[4-[(2,6-dioxopiperidin-3-yl)amino]phenyl]piperidin-1-yl]-N-methylacetamide	COC1=C(NC2=NC=C(Cl)C(NC3=C(C(C)=O)C=CC=C3)=N2)C=CC(N2CCC(N(C)C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C43H50ClN9O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-O2VYLN	SCHEMBL26161513	[2-[[5-chloro-2-[4-[4-[2-[4-[4-[(2,6-dioxopiperidin-3-yl)amino]phenyl]piperidin-1-yl]acetyl]piperazin-1-yl]-2-methoxyanilino]pyrimidin-4-yl]amino]phenyl] N,N-dimethylcarbamate	COC1=C(NC2=NC=C(Cl)C(NC3=C(OC(=O)N(C)C)C=CC=C3)=N2)C=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C42H49ClN10O6	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-Z0BR5Z	SCHEMBL26160270	1-[6-[1-[2-[4-[4-[[4-Anilino-5-(trifluoromethyl)pyrimidin-2-yl]amino]-3-methoxyphenyl]piperazin-1-yl]-2-oxoethyl]piperidin-4-yl]-1-methylindazol-3-yl]-1,3-diazinane-2,4-dione	COC1=C(NC2=NC=C(C(F)(F)F)C(NC3=CC=CC=C3)=N2)C=CC(N2CCN(C(=O)CN3CCC(C4=CC=C5C(=C4)N(C)N=C5N4CCC(=O)NC4=O)CC3)CC2)=C1	C41H44F3N11O4	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-FSBO4T	SCHEMBL26160271	3-[4-[1-[2-[4-[4-[[4-(2-Dimethylphosphorylanilino)-5-(trifluoromethyl)pyrimidin-2-yl]amino]-3-methoxyphenyl]piperazin-1-yl]-2-oxoethyl]piperidin-4-yl]anilino]piperidine-2,6-dione	COC1=C(NC2=NC=C(C(F)(F)F)C(NC3=C(P(C)(C)=O)C=CC=C3)=N2)C=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C42H49F3N9O5P	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-PIEKFX	SCHEMBL26160329	3-[4-[1-[2-[4-[4-[[4-(3-Acetylanilino)-5-(trifluoromethyl)pyrimidin-2-yl]amino]-3-methoxyphenyl]piperazin-1-yl]-2-oxoethyl]piperidin-4-yl]anilino]piperidine-2,6-dione	COC1=C(NC2=NC=C(C(F)(F)F)C(NC3=CC(C(C)=O)=CC=C3)=N2)C=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C42H46F3N9O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-EZU7UZ	SCHEMBL26160332	3-[4-[1-[2-[4-[4-[[4-(3-Chloro-4-fluoroanilino)-5-(trifluoromethyl)pyrimidin-2-yl]amino]-3-methoxyphenyl]piperazin-1-yl]-2-oxoethyl]piperidin-4-yl]anilino]piperidine-2,6-dione	COC1=C(NC2=NC=C(C(F)(F)F)C(NC3=CC(Cl)=C(F)C=C3)=N2)C=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C40H42ClF4N9O4	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-0K5RTQ	SCHEMBL26160339	3-[4-[1-[2-[4-[4-[[4-(4-Fluoroanilino)-5-(trifluoromethyl)pyrimidin-2-yl]amino]-3-methoxyphenyl]piperazin-1-yl]-2-oxoethyl]piperidin-4-yl]anilino]piperidine-2,6-dione	COC1=C(NC2=NC=C(C(F)(F)F)C(NC3=CC=C(F)C=C3)=N2)C=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C40H43F4N9O4	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-X8YBBO	SCHEMBL26160340	3-[4-[1-[2-[4-[1-[4-[[4-Anilino-5-(trifluoromethyl)pyrimidin-2-yl]amino]-3-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]-2-oxoethyl]piperidin-4-yl]anilino]piperidine-2,6-dione	COC1=C(NC2=NC=C(C(F)(F)F)C(NC3=CC=CC=C3)=N2)C=CC(N2CCC(N3CCN(C(=O)CN4CCC(C5=CC=C(NC6CCC(=O)NC6=O)C=C5)CC4)CC3)CC2)=C1	C45H53F3N10O4	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-4M604I	SCHEMBL26160343	N-[5-[[4-anilino-5-(trifluoromethyl)pyrimidin-2-yl]amino]-2-[4-[2-[4-[4-[(2,6-dioxopiperidin-3-yl)amino]phenyl]piperidin-1-yl]acetyl]piperazin-1-yl]-4-methoxyphenyl]acetamide	COC1=C(NC2=NC=C(C(F)(F)F)C(NC3=CC=CC=C3)=N2)C=C(NC(C)=O)C(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C42H47F3N10O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-JWXYZN	SCHEMBL26160346	3-[4-[1-[2-[4-[4-[[4-(2-Acetylanilino)-5-chloropyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperazin-1-yl]-2-oxoethyl]piperidin-4-yl]anilino]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C(C(C)=O)C=CC=C3)=N2)C=C(C)C(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C42H48ClN9O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-CZLTHQ	WO2023088385A1_T-58	.	COC1=C(NC2=NC=C(C(F)(F)F)C(NC3=C(C(C)=O)C=CC=C3)=N2)C=C(C)C(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C43H48F3N9O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-3GBLOE	SCHEMBL26160381	3-[4-[1-[2-[4-[4-[[4-(2-Acetylanilino)-5-bromopyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperazin-1-yl]-2-oxoethyl]piperidin-4-yl]anilino]piperidine-2,6-dione	COC1=C(NC2=NC=C(Br)C(NC3=C(C(C)=O)C=CC=C3)=N2)C=C(C)C(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C42H48BrN9O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-1FLQU6	SCHEMBL26160383	3-[4-[1-[2-[4-[4-[[4-(2-Acetylanilino)-5-chloropyrimidin-2-yl]amino]-3-methoxyphenyl]-3-methylpiperazin-1-yl]-2-oxoethyl]piperidin-4-yl]anilino]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C(C(C)=O)C=CC=C3)=N2)C=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2C)=C1	C42H48ClN9O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-40TZ59	WO2023088385A1_T-63	.	COC1=C(NC2=NC=C(Cl)C(NC3=C(C(C)=O)C=CC=C3)=N2)C=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)C(C)C2)=C1	C42H48ClN9O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-NN8AJI	WO2023088385A1_T-66	.	COC1=C(NC2=NC=C(Cl)C(NC3=C(C(C)=O)C=CC=C3)=N2)C=CC(N2CC3(CN(C(=O)CN4CCC(C5=CC=C(NC6CCC(=O)NC6=O)C=C5)CC4)C3)C2)=C1	C42H46ClN9O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-WZ9DRS	WO2023088385A1_T-72	.	COC1=C(NC2=NC=C(Cl)C(NC3=C(C(C)=O)C=CC=C3)=N2)C=CC(N2CCC(CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C41H47ClN8O4	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-B1YYHG	SCHEMBL26160473	3-[4-[1-[4-[4-[[4-(2-Acetylanilino)-5-chloropyrimidin-2-yl]amino]-3-methoxyphenyl]piperazine-1-carbonyl]piperidin-4-yl]anilino]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C(C(C)=O)C=CC=C3)=N2)C=CC(N2CCN(C(=O)N3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C40H44ClN9O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-QJOTQA	SCHEMBL26160475	3-[4-[4-[2-[4-[4-[[4-(2-Acetylanilino)-5-chloropyrimidin-2-yl]amino]-3-methoxyphenyl]piperazin-1-yl]-2-oxoethyl]piperazin-1-yl]anilino]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=C(C(C)=O)C=CC=C3)=N2)C=CC(N2CCN(C(=O)CN3CCN(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C40H45ClN10O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-6QGC74	SCHEMBL26160477	3-[4-[4-[2-[4-[4-[[4-(2-Acetylanilino)-5-bromopyrimidin-2-yl]amino]-3-methoxyphenyl]piperazin-1-yl]-2-oxoethyl]piperazin-1-yl]anilino]piperidine-2,6-dione	COC1=C(NC2=NC=C(Br)C(NC3=C(C(C)=O)C=CC=C3)=N2)C=CC(N2CCN(C(=O)CN3CCN(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C40H45BrN10O5	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-GC6A8T	SCHEMBL26161838	3-[4-[4-[[4-[4-[[4-(2-Acetylanilino)-5-chloropyrimidin-2-yl]amino]-3-methoxyphenyl]piperazin-1-yl]methyl]piperidin-1-yl]anilino]piperidine-2,6-dione	COC1=C(NC2=NC(NC3=C(C(C)=O)C=CC=C3)=C(Cl)C=N2)C=CC(N2CCN(CC3CCN(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C40H46ClN9O4	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-UQNOZT	WO2023088385A1_T-91	.	C=CC(=O)NC1=CC(NC2=NC=C(Cl)C(NC3=C(C(C)=O)C=CC=C3)=N2)=C(OC)C=C1N1CCN(C(=O)CN2CCC(C3=CC=C(NC4CCC(=O)NC4=O)C=C3)CC2)CC1	C44H49ClN10O6	EGFR	P00533	CRBN	WO-2023088385-A1
TPD-S2642V	SCHEMBL26158196	(2S,4R)-1-[(2S)-2-[[2-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCC(N4N=C(N)C5=C4C=C(C4=C(O)C=CC=C4)N=N5)CC3)C(C)(C)C)C=C2)SC=N1	C41H50N10O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-RXGU1J	SCHEMBL26157696	3-[4-[3-[4-[2-[4-[3-Amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]pyrimidin-5-yl]piperidin-1-yl]propyl]pyrido[2,3-b]indol-9-yl]piperidine-2,6-dione	NC1=NN(C2CCN(C3=NC=C(C4CCN(CCCC5=C6C(=NC=C5)N(C5CCC(=O)NC5=O)C5=C6C=CC=C5)CC4)C=N3)CC2)C2=C1N=NC(C1=C(O)C=CC=C1)=C2	C44H46N12O3	SMARCA2	P51531	CRBN	WO-2023093728-A1
TPD-QVBKCX	SCHEMBL25209496	3-[4-[3-[4-[2-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]pyrimidin-5-yl]-3,6-dihydro-2H-pyridin-1-yl]propyl]pyrido[2,3-b]indol-9-yl]piperidine-2,6-dione	NC1=NN(C2CCN(C3=NC=C(C4=CCN(CCCC5=C6C(=NC=C5)N(C5CCC(=O)NC5=O)C5=C6C=CC=C5)CC4)C=N3)CC2)C2=C1N=NC(C1=C(O)C=CC=C1)=C2	C44H44N12O3	SMARCA2	P51531	CRBN	WO-2023093728-A1
TPD-5XH0EA	WO2023093728A1_004-1	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)[C@H]3CC[C@@H](C4=CN=C(N5CCC(N6N=C(N)C7=C6C=C(C6=C(O)C=CC=C6)N=N7)CC5)N=C4)CC3)C(C)(C)C)C=C2)SC=N1	C50H60N12O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-3XHHTX	WO2023093728A1_004	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)[C@H]3CC[C@H](C4=CN=C(N5CCC(N6N=C(N)C7=C6C=C(C6=C(O)C=CC=C6)N=N7)CC5)N=C4)CC3)C(C)(C)C)C=C2)SC=N1	C50H60N12O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-BOY65K	SCHEMBL26157689	(2S,4R)-1-[(2S)-2-[[4-[2-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]pyrimidin-5-yl]cyclohex-3-ene-1-carbonyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3CC=C(C4=CN=C(N5CCC(N6N=C(N)C7=C6C=C(C6=C(O)C=CC=C6)N=N7)CC5)N=C4)CC3)C(C)(C)C)C=C2)SC=N1	C50H58N12O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-CXR516	SCHEMBL26157697	(2S,4R)-1-[2-[3-[9-[2-[4-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]pyridin-2-yl]oxyethyl]-3,9-diazaspiro[5.5]undecan-3-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCC5(CCN(CCOC6=NC=CC(N7CCC(N8N=C(N)C9=C8C=C(C8=C(O)C=CC=C8)N=N9)CC7)=C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C57H69N13O6S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-E99Z4L	SCHEMBL26157698	(2S,4R)-N-[(1S)-3-[4-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]piperidin-1-yl]-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]-3-oxopropyl]-4-hydroxy-1-[3-methyl-2-(3-methyl-1,2-oxazol-5-yl)butanoyl]pyrrolidine-2-carboxamide	CC1=NOC(C(C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](CC(=O)N2CCC(N3CCC(N4N=C(N)C5=C4C=C(C4=C(O)C=CC=C4)N=N5)CC3)CC2)C2=CC=C(C3=C(C)N=CS3)C=C2)C(C)C)=C1	C48H57N11O6S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-0WKJEJ	SCHEMBL25201037	(2S,4R)-N-[(1S)-3-[4-[2-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]pyrimidin-5-yl]piperidin-1-yl]-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]-3-oxopropyl]-4-hydroxy-1-[3-methyl-2-(3-methyl-1,2-oxazol-5-yl)butanoyl]pyrrolidine-2-carboxamide	CC1=NOC(C(C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](CC(=O)N2CCC(C3=CN=C(N4CCC(N5N=C(N)C6=C5C=C(C5=C(O)C=CC=C5)N=N6)CC4)N=C3)CC2)C2=CC=C(C3=C(C)N=CS3)C=C2)C(C)C)=C1	C52H59N13O6S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-2LA86T	WO2023093728A1_010	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(OCCN4CCC(C5=CN=C(N6CCC(N7N=C(N)C8=C7C=C(C7=C(O)C=CC=C7)N=N8)CC6)N=C5)CC4)=NO3)C(C)C)C=C2)SC=N1	C52H61N13O6S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-XYL4L5	WO2023093728A1_011	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCC(CN5CCC(N6N=C(N)C7=C6C=C(C6C=CC=CC6O)N=N7)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C47H59N11O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-KXITQY	WO2023093728A1_012	.	CC1=C(C2=NC=C(C(C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3CCC(C4=CN=C(N5CCC(N6N=C(N)C7=C6C=C(C6=C(O)C=CC=C6)N=N7)CC5)N=C4)CC3)C(C)(C)C)N=C2)SC=N1	C48H58N14O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-ZZN4BE	SCHEMBL26157711	(2S,4R)-1-[(2S)-2-[[4-[2-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]pyrimidin-5-yl]cyclohexanecarbonyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[1-[2-(4-methyl-1,3-thiazol-5-yl)pyrimidin-5-yl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=NC=C(C(C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3CCC(C4=CN=C(N5CCC(N6N=C(N)C7=C6C=C(C6=C(O)C=CC=C6)N=N7)CC5)N=C4)CC3)C(C)(C)C)C=N2)SC=N1	C48H58N14O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-KKZOW0	SCHEMBL26158424	(2S,4R)-1-[2-[3-[2-[4-[3-[4-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]ethoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[5-(4-methyl-1,3-thiazol-5-yl)pyrazin-2-yl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=NC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(OCCN4CCC(O[C@H]5C[C@H](OC6=CC(N7CCC(N8N=C(N)C9=C8C=C(C8=C(O)C=CC=C8)N=N9)CC7)=CC=N6)C5)CC4)=NO3)C(C)C)N=C2)SC=N1	C55H66N14O8S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-GFA97Y	WO2023093728A1_015	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3CCN(CC4=CN=C(N5CCC(N6N=C(N)C7=C6C=C(C6=C(O)C=CC=C6)N=N7)CC5)N=C4)CC3)C(C)(C)C)C=C2)SC=N1	C50H61N13O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-EH2I6I	SCHEMBL25236460	1-[2-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]pyrimidine-5-carbonyl]-N-[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]piperidine-4-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3CCN(C(=O)C4=CN=C(N5CCC(N6N=C(N)C7=C6C=C(C6=C(O)C=CC=C6)N=N7)CC5)N=C4)CC3)C(C)(C)C)C=C2)SC=N1	C50H59N13O6S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-PTSXGR	SCHEMBL26158461	(2S,4R)-1-[(2S)-2-[[2-[4-[2-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]pyrimidin-5-yl]piperidin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCC(C4=CN=C(N5CCC(N6N=C(N)C7=C6C=C(C6=C(O)C=CC=C6)N=N7)CC5)N=C4)CC3)C(C)(C)C)C=C2)SC=N1	C50H61N13O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-UVUWNJ	SCHEMBL25199322	(2S,4R)-1-[2-[3-[2-[2-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]ethoxy]ethoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(OCCOCCN4CCC(N5N=C(N)C6=C5C=C(C5=C(O)C=CC=C5)N=N6)CC4)=NO3)C(C)C)C=C2)SC=N1	C45H54N10O7S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-6OVBDR	SCHEMBL25224306	(2S,4R)-1-[(2S)-2-[8-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]octanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCN3CCC(N4N=C(N)C5=C4C=C(C4=C(O)C=CC=C4)N=N5)CC3)C(C)(C)C)C=C2)SC=N1	C47H62N10O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-NCNXCU	SCHEMBL25237915	(2S,4R)-1-[(2S)-2-[4-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]butanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCN3CCC(N4N=C(N)C5=C4C=C(C4=C(O)C=CC=C4)N=N5)CC3)C(C)(C)C)C=C2)SC=N1	C43H54N10O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-4879XC	SCHEMBL26157731	(2S,4R)-1-[(2S)-2-[10-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]decanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCCCN3CCC(N4N=C(N)C5=C4C=C(C4=C(O)C=CC=C4)N=N5)CC3)C(C)(C)C)C=C2)SC=N1	C49H66N10O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-KR9P9M	SCHEMBL26157742	(2S,4R)-1-[(2S)-2-[12-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]dodecanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCCCCCN3CCC(N4N=C(N)C5=C4C=C(C4=C(O)C=CC=C4)N=N5)CC3)C(C)(C)C)C=C2)SC=N1	C51H70N10O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-JYK5KB	SCHEMBL26157743	(2S,4R)-1-[(2S)-2-[9-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]nonanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCCN3CCC(N4N=C(N)C5=C4C=C(C4=C(O)C=CC=C4)N=N5)CC3)C(C)(C)C)C=C2)SC=N1	C48H64N10O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-U22MOO	SCHEMBL25237864	(2S,4R)-1-[2-[3-[3-[4-[1-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]ethyl]phenyl]propoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(OCCCC4=CC=C(C(C)N5CCC(N6N=C(N)C7=C6C=C(C6=C(O)C=CC=C6)N=N7)CC5)C=C4)=NO3)C(C)C)C=C2)SC=N1	C52H60N10O6S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-6RC7TJ	SCHEMBL26157744	(2S,4R)-1-[2-[3-[4-[[4-[4-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]pyridin-2-yl]oxypiperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCC(CN5CCC(OC6=NC=CC(N7CCC(N8N=C(N)C9=C8C=C(C8=C(O)C=CC=C8)N=N9)CC7)=C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C57H69N13O6S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-E5H24U	SCHEMBL25201735	(2S,4R)-1-[2-[3-[4-[[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCC(CN5CCC(N6N=C(N)C7=C6C=C(C6=C(O)C=CC=C6)N=N7)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C47H57N11O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-Z68HVD	SCHEMBL25228596	(2S,4R)-1-[2-[3-[4-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidine-1-carbonyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCC(C(=O)N5CCC(N6N=C(N)C7=C6C=C(C6=C(O)C=CC=C6)N=N7)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C47H55N11O6S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-KQH4VJ	SCHEMBL25196730	(2S,4R)-1-[(2S)-2-[11-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]undecanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCCCCN3CCC(N4N=C(N)C5=C4C=C(C4=C(O)C=CC=C4)N=N5)CC3)C(C)(C)C)C=C2)SC=N1	C50H68N10O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-5WWEEV	WO2023093728A1_030	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(OCCN4CCC(N5N=C(N)C6N=NC(C7=C(O)C=CC=C7)=CC65)CC4)=NO3)C(C)C)C=C2)SC=N1	C43H52N10O6S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-8VZ8W0	SCHEMBL25194967	(2S,4R)-1-[2-[3-[7-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]heptoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(OCCCCCCCN4CCC(N5N=C(N)C6=C5C=C(C5=C(O)C=CC=C5)N=N6)CC4)=NO3)C(C)C)C=C2)SC=N1	C48H60N10O6S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-X46UUY	SCHEMBL26157766	(2S,4R)-1-[(2S)-2-[3-[9-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]nonoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3=CC(OCCCCCCCCCN4CCC(N5N=C(N)C6=C5C=C(C5=C(O)C=CC=C5)N=N6)CC4)=NO3)C(C)C)C=C2)SC=N1	C50H64N10O6S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-K10R7M	SCHEMBL25212374	(2S,4R)-1-[(2R)-2-[3-[9-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]nonoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(OCCCCCCCCCN4CCC(N5N=C(N)C6=C5C=C(C5=C(O)C=CC=C5)N=N6)CC4)=NO3)C(C)C)C=C2)SC=N1	C50H64N10O6S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-ZVZT53	WO2023093728A1_033-1	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)[C@H]3CC[C@@H](C4=CN=C(N5CCC(N6N=C(N)C7=C6C=C(C6=C(O)C=CC=C6)N=N7)CC5)N=C4)CC3)C(C)(C)C)C=N2)SC=N1	C49H59N13O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-YC7P0P	WO2023093728A1_033	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)[C@H]3CC[C@H](C4=CN=C(N5CCC(N6N=C(N)C7=C6C=C(C6=C(O)C=CC=C6)N=N7)CC5)N=C4)CC3)C(C)(C)C)C=N2)SC=N1	C49H59N13O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-BFOEKU	WO2023093728A1_034	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCN3CCC(N4N=C(N)C5N=NC(C6=C(O)C=CC=C6)=CC54)CC3)C(C)(C)C)C=C2)SC=N1	C44H58N10O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-TY5RTH	SCHEMBL26157769	(2S,4R)-1-[(2S)-2-[6-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]hexanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCN3CCC(N4N=C(N)C5=C4C=C(C4=C(O)C=CC=C4)N=N5)CC3)C(C)(C)C)C=C2)SC=N1	C45H58N10O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-S86ANV	SCHEMBL25208536	(2S,4R)-1-[2-[3-[8-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]octoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(OCCCCCCCCN4CCC(N5N=C(N)C6=C5C=C(C5=C(O)C=CC=C5)N=N6)CC4)=NO3)C(C)C)C=C2)SC=N1	C49H62N10O6S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-3QR5A8	SCHEMBL25195490	(2S,4R)-1-[2-[3-[4-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]butoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(OCCCCN4CCC(N5N=C(N)C6=C5C=C(C5=C(O)C=CC=C5)N=N6)CC4)=NO3)C(C)C)C=C2)SC=N1	C45H54N10O6S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-RG4ZJU	SCHEMBL26159010	(2S,4R)-1-[(2S)-2-[7-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]heptanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCN3CCC(N4N=C(N)C5=C4C=C(C4=C(O)C=CC=C4)N=N5)CC3)C(C)(C)C)C=C2)SC=N1	C46H60N10O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-9MOVR9	SCHEMBL26157782	(2S,4R)-1-[(2S)-2-[13-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]tridecanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCCCCCCN3CCC(N4N=C(N)C5=C4C=C(C4=C(O)C=CC=C4)N=N5)CC3)C(C)(C)C)C=C2)SC=N1	C52H72N10O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-B9SZSM	SCHEMBL26157783	(2S,4R)-1-[2-[3-[3-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]propoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(OCCCN4CCC(N5N=C(N)C6=C5C=C(C5=C(O)C=CC=C5)N=N6)CC4)=NO3)C(C)C)C=C2)SC=N1	C44H52N10O6S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-IPCFG2	WO2023093728A1_041	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(OCCN4CCC(N5N=C(N)C6=C5C=C(C5C=CC=CC5O)N=N6)CC4)=NO3)C(C)C)C=C2)SC=N1	C43H52N10O6S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-XSRCBA	WO2023093728A1_042	.	CC1=C(C2=CC=C([C@H](C)NC(=O)C3C[C@@H](O)CN3C(=O)C(C3=CC(OCCCCCN4CCC(N5N=C(N)C6=C5C=C(C5=C(O)C=CC=C5)N=N6)CC4)=NO3)C(C)C)C=C2)SC=N1	C46H56N10O6S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-4UVSI4	SCHEMBL25228437	(2S,4R)-1-[2-[3-[6-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]hexoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(OCCCCCCN4CCC(N5N=C(N)C6=C5C=C(C5=C(O)C=CC=C5)N=N6)CC4)=NO3)C(C)C)C=C2)SC=N1	C47H58N10O6S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-QMGNA4	SCHEMBL26157806	(2S,4R)-1-[(2S)-2-[3-[10-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]decoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3=CC(OCCCCCCCCCCN4CCC(N5N=C(N)C6=C5C=C(C5=C(O)C=CC=C5)N=N6)CC4)=NO3)C(C)C)C=C2)SC=N1	C51H66N10O6S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-MM48PT	SCHEMBL25195448	(2S,4R)-1-[(2R)-2-[3-[10-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]decoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(OCCCCCCCCCCN4CCC(N5N=C(N)C6=C5C=C(C5=C(O)C=CC=C5)N=N6)CC4)=NO3)C(C)C)C=C2)SC=N1	C51H66N10O6S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-TAX1UU	SCHEMBL26157808	(2S,4R)-1-[(2S)-2-[3-[11-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]undecoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3=CC(OCCCCCCCCCCCN4CCC(N5N=C(N)C6=C5C=C(C5=C(O)C=CC=C5)N=N6)CC4)=NO3)C(C)C)C=C2)SC=N1	C52H68N10O6S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-2OH7NP	SCHEMBL25219300	(2S,4R)-1-[(2R)-2-[3-[11-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]undecoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(OCCCCCCCCCCCN4CCC(N5N=C(N)C6=C5C=C(C5=C(O)C=CC=C5)N=N6)CC4)=NO3)C(C)C)C=C2)SC=N1	C52H68N10O6S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-H1Z8GE	SCHEMBL25207259	(2S,4R)-1-[2-[3-[2-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]-2-oxoethoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(OCC(=O)N4CCC(N5N=C(N)C6=C5C=C(C5=C(O)C=CC=C5)N=N6)CC4)=NO3)C(C)C)C=C2)SC=N1	C43H48N10O7S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-V2CC7W	WO2023093728A1_047	.	CNC1=NN(C2CCN(CCOC3=NOC(C(C(=O)N4C[C@H](O)C[C@H]4C(=O)N[C@@H](C)C4=CC=C(C5=C(C)N=CS5)C=C4)C(C)C)=C3)CC2)C2=C1N=NC(C1=C(O)C=CC=C1)=C2	C44H52N10O6S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-PJZAU4	WO2023093728A1_048	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(OCCN4CCC(N5N=C(N)C6=C5C=C(C5=C(O)C=CC=C5)N=N6)C4)=NO3)C(C)C)C=C2)SC=N1	C42H48N10O6S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-QWTYYQ	SCHEMBL25213728	(2S,4R)-1-[2-[3-[2-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]ethoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-N-[(1S)-1-[2-fluoro-4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]-4-hydroxypyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(OCCN4CCC(N5N=C(N)C6=C5C=C(C5=C(O)C=CC=C5)N=N6)CC4)=NO3)C(C)C)C(F)=C2)SC=N1	C43H49FN10O6S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-YWKWSR	SCHEMBL25210110	(2S,4R)-1-[2-[3-[2-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]ethoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[5-(4-methyl-1,3-thiazol-5-yl)pyridin-2-yl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(OCCN4CCC(N5N=C(N)C6=C5C=C(C5=C(O)C=CC=C5)N=N6)CC4)=NO3)C(C)C)N=C2)SC=N1	C42H49N11O6S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-ROTBMJ	SCHEMBL26157823	(2S,4R)-1-[2-[3-[2-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]ethoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[6-(4-methyl-1,3-thiazol-5-yl)pyridin-3-yl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(OCCN4CCC(N5N=C(N)C6=C5C=C(C5=C(O)C=CC=C5)N=N6)CC4)=NO3)C(C)C)C=N2)SC=N1	C42H49N11O6S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-U7B8JD	WO2023093728A1_052	.	CC1=C(C2=NC=C(C(C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(OCCN4CCC(N5N=C(N)C6=C5C=C(C5=C(O)C=CC=C5)N=N6)CC4)=NO3)C(C)C)N=C2)SC=N1	C41H48N12O6S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-BWDB5O	SCHEMBL26159078	(2S,4R)-1-[2-[3-[2-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]ethoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(OCCN4CCC(N5N=C(N)C6=C5C=C(C5=C(O)C=CC=C5)N=N6)CC4)=NO3)C(C)C)C=C2)SC=N1	C43H50N10O6S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-9KSXH2	WO2023093728A1_054	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(OCCN4C5CCC4CC(N4N=C(N)C6=C4C=C(C4=C(O)C=CC=C4)N=N6)C5)=NO3)C(C)C)C=C2)SC=N1	C45H52N10O6S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-FXZ0QA	WO2023093728A1_055	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(OCCN4CCC(CN5N=C(N)C6=C5C=C(C5=C(O)C=CC=C5)N=N6)CC4)=NO3)C(C)C)C=C2)SC=N1	C44H52N10O6S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-EVTVIV	SCHEMBL26157837	(2S,4R)-1-[2-[3-[1-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]propan-2-yloxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(OC(C)CN4CCC(N5N=C(N)C6=C5C=C(C5=C(O)C=CC=C5)N=N6)CC4)=NO3)C(C)C)C=C2)SC=N1	C44H52N10O6S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-YZPGTV	SCHEMBL25210214	(2S,4R)-1-[(2S)-2-[[2-[2-[3-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]-8-azabicyclo[3.2.1]octan-8-yl]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCN3C4CCC3CC(N3N=C(N)C5=C3C=C(C3=C(O)C=CC=C3)N=N5)C4)C(C)(C)C)C=C2)SC=N1	C45H56N10O6S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-BCYN0V	SCHEMBL25198970	(2S,4R)-1-[2-[3-[3-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]azetidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CC(N5CCC(N6N=C(N)C7=C6C=C(C6=C(O)C=CC=C6)N=N7)CC5)C4)=NO3)C(C)C)C=C2)SC=N1	C44H51N11O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-Z8WTMN	SCHEMBL26157839	(2S,4R)-4-hydroxy-1-[(2S)-2-[6-[4-[6-(2-hydroxyphenyl)-3-(methylamino)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]hexanoylamino]-3,3-dimethylbutanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CNC1=NN(C2CCN(CCCCCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](C)C3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)CC2)C2=C1N=NC(C1=C(O)C=CC=C1)=C2	C46H60N10O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-4ZHN4Y	SCHEMBL26157869	(2S,4R)-1-[(2S)-2-[[2-[2-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]pyrimidin-5-yl]oxyacetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COC3=CN=C(N4CCC(N5N=C(N)C6=C5C=C(C5=C(O)C=CC=C5)N=N6)CC4)N=C3)C(C)(C)C)C=C2)SC=N1	C45H52N12O6S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-AUK5P8	SCHEMBL26159461	(2S,4R)-1-[(2S)-2-[[2-[4-[[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCC(CN4CCC(N5N=C(N)C6=C5C=C(C5=C(O)C=CC=C5)N=N6)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C47H61N11O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-XZ7535	SCHEMBL26157860	(2S,4R)-4-hydroxy-1-[2-[3-[4-[[4-[6-(2-hydroxyphenyl)-3-(methylamino)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CNC1=NN(C2CCN(CC3CCN(C4=NOC(C(C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=C(C)N=CS6)C=C5)C(C)C)=C4)CC3)CC2)C2=C1N=NC(C1=CC=CC=C1O)=C2	C48H59N11O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-XE1QKE	SCHEMBL25208646	(2S,4R)-4-hydroxy-1-[2-[3-[2-[3-[6-(2-hydroxyphenyl)-3-(methylamino)pyrazolo[4,3-c]pyridazin-1-yl]pyrrolidin-1-yl]ethoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CNC1=NN(C2CCN(CCOC3=NOC(C(C(=O)N4C[C@H](O)C[C@H]4C(=O)N[C@@H](C)C4=CC=C(C5=C(C)N=CS5)C=C4)C(C)C)=C3)C2)C2=C1N=NC(C1=C(O)C=CC=C1)=C2	C43H50N10O6S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-H71B5B	SCHEMBL26157861	(2S,4R)-4-hydroxy-1-[2-[3-[2-[4-[2-[4-[6-(2-hydroxyphenyl)-3-(methylamino)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]pyrimidin-5-yl]piperidin-1-yl]ethoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CNC1=NN(C2CCN(C3=NC=C(C4CCN(CCOC5=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C5)CC4)C=N3)CC2)C2=C1N=NC(C1=C(O)C=CC=C1)=C2	C53H63N13O6S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-55QU5L	SCHEMBL26157862	(2S,4R)-1-[2-[3-[2-[4-[2-[3-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]-8-azabicyclo[3.2.1]octan-8-yl]pyrimidin-5-yl]piperidin-1-yl]ethoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(OCCN4CCC(C5=CN=C(N6C7CCC6CC(N6N=C(N)C8=C6C=C(C6=C(O)C=CC=C6)N=N8)C7)N=C5)CC4)=NO3)C(C)C)C=C2)SC=N1	C54H63N13O6S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-ZRCJK3	SCHEMBL26157863	(2S,4R)-4-hydroxy-1-[2-[3-[2-[4-[6-(2-hydroxyphenyl)-3-(methylamino)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]ethyl-methylamino]-1,2-oxazol-5-yl]-3-methylbutanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CNC1=NN(C2CCN(CCN(C)C3=NOC(C(C(=O)N4C[C@H](O)C[C@H]4C(=O)N[C@@H](C)C4=CC=C(C5=C(C)N=CS5)C=C4)C(C)C)=C3)CC2)C2=C1N=NC(C1=C(O)C=CC=C1)=C2	C45H55N11O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-DNZCPR	SCHEMBL26157864	(2S,4R)-1-[2-[3-[4-[[4-[3-(ethylamino)-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CCNC1=NN(C2CCN(CC3CCN(C4=NOC(C(C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=C(C)N=CS6)C=C5)C(C)C)=C4)CC3)CC2)C2=C1N=NC(C1=C(O)C=CC=C1)=C2	C49H61N11O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-0LREBG	SCHEMBL26157838	(2S,4R)-4-hydroxy-1-[2-[3-[4-[[4-[6-(2-hydroxyphenyl)-3-(propylamino)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CCCNC1=NN(C2CCN(CC3CCN(C4=NOC(C(C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=C(C)N=CS6)C=C5)C(C)C)=C4)CC3)CC2)C2=C1N=NC(C1=C(O)C=CC=C1)=C2	C50H63N11O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-5UN166	orb2802138	(2S,4R)-4-hydroxy-1-[2-[3-[4-[[4-[6-(2-hydroxyphenyl)-3-(propan-2-ylamino)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL26157849; 2933125-05-2	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCC(CN5CCC(N6N=C(NC(C)C)C7=C6C=C(C6=C(O)C=CC=C6)N=N7)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C50H63N11O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-IEAAD5	SCHEMBL26157840	(2S,4R)-1-[2-[3-[4-[[4-[3-(cyclopropanecarbonylamino)-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCC(CN5CCC(N6N=C(NC(=O)C7CC7)C7=C6C=C(C6=C(O)C=CC=C6)N=N7)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C51H61N11O6S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-I4KLIN	SCHEMBL26157850	(2S,4R)-1-[2-[3-[4-[[4-[3-amino-6-(3-chloro-2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCC(CN5CCC(N6N=C(N)C7=C6C=C(C6=C(O)C(Cl)=CC=C6)N=N7)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C47H56ClN11O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-QBLMXE	WO2023093728A1_308	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCC(CN5CCC(N6N=C(NC(=O)C7CC7)C7=C6C=C(C6=C(O)C(Cl)=CC=C6)N=N7)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C51H60ClN11O6S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-TP75OG	SCHEMBL26157865	(2S,4R)-4-hydroxy-1-[(2S)-2-[[2-[4-[[4-[6-(2-hydroxyphenyl)-3-(methylamino)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CNC1=NN(C2CCN(CC3CCN(CC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)N[C@@H](C)C4=CC=C(C5=C(C)N=CS5)C=C4)C(C)(C)C)CC3)CC2)C2=C1N=NC(C1=C(O)C=CC=C1)=C2	C48H63N11O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-DN09UB	SCHEMBL26157841	(2S,4R)-1-[2-[3-[4-[[4-[3-(cyclopropylamino)-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCC(CN5CCC(N6N=C(NC7CC7)C7=C6C=C(C6=C(O)C=CC=C6)N=N7)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C50H61N11O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-UZSGEC	SCHEMBL26157847	(2S,4R)-4-hydroxy-1-[2-[3-[4-[[4-[6-(2-hydroxyphenyl)-3-(2,2,2-trifluoroethylamino)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCC(CN5CCC(N6N=C(NCC(F)(F)F)C7=C6C=C(C6=C(O)C=CC=C6)N=N7)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C49H58F3N11O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-NA4EQC	WO2023093728A1_318-1	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCC(CN5CCC(C6=CN=C(N7C8CCC7CC(N7N=C(N)C9=C7C=C(C7=C(O)C=CC=C7)N=N9)C8)N=C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C58H70N14O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-Z3Z1Z9	SCHEMBL26157853	(2S,4R)-4-hydroxy-1-[2-[3-[4-[[4-[2-[4-[6-(2-hydroxyphenyl)-3-(methylamino)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]pyrimidin-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CNC1=NN(C2CCN(C3=NC=C(C4CCN(CC5CCN(C6=NOC(C(C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)C)=C6)CC5)CC4)C=N3)CC2)C2=C1N=NC(C1=C(O)C=CC=C1)=C2	C57H70N14O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-4W3D30	WO2023093728A1_322	.	CNC1=NN(C2CCN(C3=NC=C(C4CCN(CC5CCN(C6=NOC(C(C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)C)=C6)CC5)CC4)C=C3)CC2)C2=C1N=NC(C1=C(O)C=CC=C1)=C2	C58H71N13O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-ETEC69	SCHEMBL26157859	(2S,4R)-4-hydroxy-1-[2-[3-[4-[[4-[2-[4-[6-(2-hydroxyphenyl)-3-(propan-2-ylamino)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]pyrimidin-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCC(CN5CCC(C6=CN=C(N7CCC(N8N=C(NC(C)C)C9=C8C=C(C8=C(O)C=CC=C8)N=N9)CC7)N=C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C59H74N14O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-XKO3BX	SCHEMBL26159965	(2S,4R)-1-[2-[3-[4-[[4-[3-[4-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCC(CN5CCC(O[C@H]6C[C@H](OC7=CC(N8CCC(N9N=C(N)C%10=C9C=C(C9=C(O)C=CC=C9)N=N%10)CC8)=CC=N7)C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C61H75N13O7S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-NGOHQ3	SCHEMBL26157870	(2S,4R)-1-[2-[3-[4-[[4-[3-[2-[3-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]-8-azabicyclo[3.2.1]octan-8-yl]pyrimidin-5-yl]oxycyclobutyl]oxypiperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCC(CN5CCC(O[C@H]6C[C@H](OC7=CN=C(N8C9CCC8CC(N8N=C(N)C%10=C8C=C(C8=C(O)C=CC=C8)N=N%10)C9)N=C7)C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C62H76N14O7S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-RWARID	WO2023093728A1_333	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCC(CN5CCC(O[C@H]6C[C@H](OC7=CC=C(N8C9CCC8CC(N8N=C(N)C%10=C8C=C(C8=C(O)C=CC=C8)N=N%10)C9)N=C7)C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C63H77N13O7S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-B1VDSA	WO2023093728A1_334-1	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCC(CN5CCC(O[C@H]6C[C@H](OC7=CC(N8C9CCC8CC(N8N=C(N)C%10=C8C=C(C8=C(O)C=CC=C8)N=N%10)C9)=CC=N7)C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C63H77N13O7S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-0CVG3E	SCHEMBL26157875	(2S,4R)-1-[2-[3-[4-[[4-[3-[2-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]pyrimidin-5-yl]oxycyclobutyl]oxypiperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCC(CN5CCC(O[C@H]6C[C@H](OC7=CN=C(N8CCC(N9N=C(N)C%10=C9C=C(C9=C(O)C=CC=C9)N=N%10)CC8)N=C7)C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C60H74N14O7S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-JLNENU	SCHEMBL26157876	(2S,4R)-4-hydroxy-1-[2-[3-[4-[[4-[3-[2-[4-[6-(2-hydroxyphenyl)-3-(propan-2-ylamino)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]pyrimidin-5-yl]oxycyclobutyl]oxypiperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCC(CN5CCC(O[C@H]6C[C@H](OC7=CN=C(N8CCC(N9N=C(NC(C)C)C%10=C9C=C(C9=C(O)C=CC=C9)N=N%10)CC8)N=C7)C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C63H80N14O7S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-AB1B3H	SCHEMBL26157877	(2S,4R)-4-hydroxy-1-[2-[3-[4-[[4-[3-[4-[4-[6-(2-hydroxyphenyl)-3-(propan-2-ylamino)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCC(CN5CCC(O[C@H]6C[C@H](OC7=NC=CC(N8CCC(N9N=C(NC(C)C)C%10=C9C=C(C9=C(O)C=CC=C9)N=N%10)CC8)=C7)C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C64H81N13O7S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-Y16MKP	WO2023093728A1_375	.	CC1=C(C2C=CC([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(OCCN4CCC(N5N=C(NC6CC6)C6=C5C=C(C5C=CC=CC5O)N=N6)CC4)=NO3)C(C)C)=CC2)SC=N1	C46H58N10O6S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-WGIG32	WO2023093728A1_378	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCC(CN5CCC(N6N=C(NC(C)C)C7=C6C=C(C6=C(O)C(Cl)=CC=C6)N=N7)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C50H62ClN11O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-C5X9UG	WO2023093728A1_386	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCC(CN5CCC(C6=CC(N7CCC(N8N=C(N)C9=C8C=C(C8=C(O)C=CC=C8)N=N9)CC7)=CC=N6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C57H69N13O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-Y1N81B	SCHEMBL26157884	4-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]-N-[[1-[[1-[5-[1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]-1,2-oxazol-3-yl]piperidin-4-yl]methyl]piperidin-4-yl]methyl]pyridine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCC(CN5CCC(CNC(=O)C6=CC(N7CCC(N8N=C(N)C9=C8C=C(C8=C(O)C=CC=C8)N=N9)CC7)=CC=N6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C59H72N14O6S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-99ZEJA	WO2023093728A1_398	.	CCNC1=NN(C2CCN(CC3CCN(CC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)N[C@@H](C)C4=CC=C(C5=C(C)N=CS5)C=C4)C(C)(C)C)CC3)CC2)C2=C1N=NC(C1=C(O)C=CC=C1)=C2	C49H65N11O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-S406R2	SCHEMBL26157887	(2S,4R)-4-hydroxy-1-[(2S)-2-[[2-[4-[[4-[6-(2-hydroxyphenyl)-3-(propylamino)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CCCNC1=NN(C2CCN(CC3CCN(CC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)N[C@@H](C)C4=CC=C(C5=C(C)N=CS5)C=C4)C(C)(C)C)CC3)CC2)C2=C1N=NC(C1=C(O)C=CC=C1)=C2	C50H67N11O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-8MACRJ	SCHEMBL26157889	(2S,4R)-4-hydroxy-1-[(2S)-2-[[2-[4-[[4-[6-(2-hydroxyphenyl)-3-(propan-2-ylamino)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCC(CN4CCC(N5N=C(NC(C)C)C6=C5C=C(C5=C(O)C=CC=C5)N=N6)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C50H67N11O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-K2YUNM	WO2023093728A1_409	.	CC1=C(C2=CCC([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCC(CN5CCC(N6N=C(NC(C)C)C7=C6C=C(C6=C(O)C(F)=CC=C6)N=N7)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C50H64FN11O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-1YOFBE	WO2023093728A1_410	.	CC1=C(C2=CCC([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCC(CN5CCC(N6N=C(NC(C)C)C7=C6C=C(C6=C(O)C=CC(F)=C6)N=N7)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C50H64FN11O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-GOBNPI	WO2023093728A1_412	.	CC1=C(C2=CCC([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCC(CN5CCC(N6N=C(NCC(C)(C)O)C7=C6C=C(C6=C(O)C=CC=C6)N=N7)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C51H67N11O6S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-2QFODT	SCHEMBL26157893	(2S,4R)-1-[2-[3-[4-[[4-[2-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]pyrimidin-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCC(CN5CCN(C6=CN=C(N7CCC(N8N=C(N)C9=C8C=C(C8=C(O)C=CC=C8)N=N9)CC7)N=C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C55H67N15O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-NUMPB4	SCHEMBL26157894	(2S,4R)-1-[2-[3-[4-[[4-[2-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]pyrimidin-5-yl]cyclohexyl]methyl]piperazin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCN(CC5CCC(C6=CN=C(N7CCC(N8N=C(N)C9=C8C=C(C8=C(O)C=CC=C8)N=N9)CC7)N=C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C56H68N14O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-UGAAEO	SCHEMBL26157899	(2S,4R)-1-[2-[3-[4-[[4-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCC(CN5CCC(N6CCC(N7N=C(N)C8=C7C=C(C7=C(O)C=CC=C7)N=N8)CC6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C52H66N12O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-OXPBIJ	SCHEMBL26157900	(2S,4R)-4-hydroxy-1-[2-[3-[4-[[4-[[4-[6-(2-hydroxyphenyl)-3-(propan-2-ylamino)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCC(CN5CCC(CN6CCC(N7N=C(NC(C)C)C8=C7C=C(C7=C(O)C=CC=C7)N=N8)CC6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C56H74N12O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-KK018M	SCHEMBL26157901	(2S,4R)-1-[2-[3-[4-[2-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]pyrimidin-5-yl]oxypiperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCC(OC5=CN=C(N6CCC(N7N=C(N)C8=C7C=C(C7=C(O)C=CC=C7)N=N8)CC6)N=C5)CC4)=NO3)C(C)C)C=C2)SC=N1	C50H57N13O6S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-PZYHR4	SCHEMBL26157902	(2S,4R)-1-[2-[3-[4-[[2-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]pyrimidin-5-yl]methyl]piperazin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCN(CC5=CN=C(N6CCC(N7N=C(N)C8=C7C=C(C7=C(O)C=CC=C7)N=N8)CC6)N=C5)CC4)=NO3)C(C)C)C=C2)SC=N1	C50H58N14O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-SIQA6C	SCHEMBL26157903	(2S,4R)-1-[2-[3-[4-[[4-[2-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]pyrimidin-4-yl]piperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCC(CN5CCC(C6=NC(N7CCC(N8N=C(N)C9=C8C=C(C8=C(O)C=CC=C8)N=N9)CC7)=NC=C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C56H68N14O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-Q9RG8Y	SCHEMBL26157905	(2S,4R)-1-[2-[3-[4-[[4-[2-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]pyrimidin-4-yl]piperazin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCC(CN5CCN(C6=NC(N7CCC(N8N=C(N)C9=C8C=C(C8=C(O)C=CC=C8)N=N9)CC7)=NC=C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C55H67N15O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-3AKBJX	SCHEMBL26157906	(2S,4R)-1-[(2S)-2-[[4-[[4-[3-(ethylamino)-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]methyl]cyclohexanecarbonyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CCNC1=NN(C2CCN(C[C@H]3CC[C@H](C(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)N[C@@H](C)C4=CC=C(C5=C(C)N=CS5)C=C4)C(C)(C)C)CC3)CC2)C2=C1N=NC(C1=C(O)C=CC=C1)=C2	C49H64N10O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-818V6D	SCHEMBL26157907	(2S,4R)-1-[2-[3-[4-[[4-[6-(3-fluoro-2-hydroxyphenyl)-3-(propylamino)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CCCNC1=NN(C2CCN(CC3CCN(C4=NOC(C(C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=C(C)N=CS6)C=C5)C(C)C)=C4)CC3)CC2)C2=C1N=NC(C1=C(O)C(F)=CC=C1)=C2	C50H62FN11O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-ET27IU	SCHEMBL26157908	(2S,4R)-1-[2-[3-[4-[[4-[6-(3-fluoro-2-hydroxyphenyl)-3-[(2-hydroxy-2-methylpropyl)amino]pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCC(CN5CCC(N6N=C(NCC(C)(C)O)C7=C6C=C(C6=C(O)C(F)=CC=C6)N=N7)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C51H64FN11O6S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-V9LOTK	SCHEMBL26157909	(2S,4R)-1-[2-[3-[4-[[4-[2-[4-[3-amino-6-(3-fluoro-2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]pyrimidin-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCC(CN5CCC(C6=CN=C(N7CCC(N8N=C(N)C9=C8C=C(C8=C(O)C(F)=CC=C8)N=N9)CC7)N=C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C56H67FN14O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-YLK6HT	SCHEMBL26157912	(2S,4R)-1-[2-[3-[4-[[4-[3-amino-6-(3-fluoro-2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCC(CN5CCC(N6N=C(N)C7=C6C=C(C6=C(O)C(F)=CC=C6)N=N7)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C47H56FN11O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-74P2QK	SCHEMBL26157913	(2S,4R)-1-[2-[3-[4-[[4-[3-amino-6-(5-fluoro-2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCC(CN5CCC(N6N=C(N)C7=C6C=C(C6=C(O)C=CC(F)=C6)N=N7)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C47H56FN11O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-3MB0TH	SCHEMBL26157914	(2S,4R)-1-[2-[3-[4-[[3-[2-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]pyrimidin-5-yl]oxyazetidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCC(CN5CC(OC6=CN=C(N7CCC(N8N=C(N)C9=C8C=C(C8=C(O)C=CC=C8)N=N9)CC7)N=C6)C5)CC4)=NO3)C(C)C)C=C2)SC=N1	C54H64N14O6S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-LNMTSO	WO2023093728A1_453	.	CCNC1=NN(C2CCN(CC3CC4(C3)CN(C(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](C)C3=CC=C(C5=C(C)N=CS5)C=C3)C(C)(C)C)C4)CC2)C2=C1N=NC(C1=C(O)C=CC=C1)=C2	C49H63N11O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-CZ52XK	SCHEMBL26157916	(2S,4R)-1-[2-[3-[4-[[4-[6-(5-fluoro-2-hydroxyphenyl)-3-[(2-hydroxy-2-methylpropyl)amino]pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCC(CN5CCC(N6N=C(NCC(C)(C)O)C7=C6C=C(C6=C(O)C=CC(F)=C6)N=N7)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C51H64FN11O6S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-ALQ6EY	SCHEMBL26157917	(2S,4R)-1-[2-[3-[4-[[4-[2-[4-[3-amino-6-(5-fluoro-2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]pyrimidin-5-yl]piperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCC(CN5CCC(C6=CN=C(N7CCC(N8N=C(N)C9=C8C=C(C8=C(O)C=CC(F)=C8)N=N9)CC7)N=C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C56H67FN14O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-MLNZSL	SCHEMBL26157918	(2S,4R)-1-[2-[3-[4-[[3-[2-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]pyrimidin-5-yl]-8-azabicyclo[3.2.1]octan-8-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCC(CN5C6CCC5CC(C5=CN=C(N7CCC(N8N=C(N)C9=C8C=C(C8=C(O)C=CC=C8)N=N9)CC7)N=C5)C6)CC4)=NO3)C(C)C)C=C2)SC=N1	C58H70N14O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-DAIGN6	SCHEMBL26157919	(2S,4R)-4-hydroxy-1-[2-[3-[4-[[4-[4-[6-(2-hydroxyphenyl)-3-(propylamino)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CCCNC1=NN(C2CCN(C3CCN(CC4CCN(C5=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C5)CC4)CC3)CC2)C2=C1N=NC(C1=C(O)C=CC=C1)=C2	C55H72N12O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-BW4NQB	SCHEMBL26157920	(2S,4R)-1-[2-[3-[4-[[4-[6-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]pyridin-3-yl]piperazin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCC(CN5CCN(C6=CC=C(N7CCC(N8N=C(N)C9=C8C=C(C8=C(O)C=CC=C8)N=N9)CC7)N=C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C56H68N14O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-K9AZ63	SCHEMBL26157921	(2S,4R)-1-[2-[3-[4-[[4-[6-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]pyridin-3-yl]piperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCC(CN5CCC(C6=CC=C(N7CCC(N8N=C(N)C9=C8C=C(C8=C(O)C=CC=C8)N=N9)CC7)N=C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C57H69N13O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-35WOIH	WO2023093728A1_494	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCC(CN5CCC(C6=NN=C(N7CCC(N8N=C(N)C9=C8C=C(C8=C(O)C=CC=C8)N=N9)CC7)C=C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C56H68N14O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-3R8FFG	SCHEMBL26157922	(2S,4R)-1-[2-[3-[4-[[4-[5-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]pyrazin-2-yl]piperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCC(CN5CCC(C6=CN=C(N7CCC(N8N=C(N)C9=C8C=C(C8=C(O)C=CC=C8)N=N9)CC7)C=N6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C56H68N14O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-EPYBXF	WO2023093728A1_496	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCC(CN5CCC(C6=CN=C(N7CCC(N8N=C(N)C9=C8C=C(C8=C(O)C=CC=C8)N=N9)CC7)S6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C55H67N13O5S2	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-N5BGTO	WO2023093728A1_499	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCN(CCN5CCC(N6N=C(NCC(C)(C)O)C7=C6C=C(C6=C(O)C=CC=C6)N=N7)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C51H66N12O6S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-TOQX9H	SCHEMBL26157934	(2S,4R)-1-[2-[3-[4-[[4-[6-(4-fluoro-2-hydroxyphenyl)-3-[(2-hydroxy-2-methylpropyl)amino]pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCC(CN5CCC(N6N=C(NCC(C)(C)O)C7=C6C=C(C6=C(O)C=C(F)C=C6)N=N7)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C51H64FN11O6S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-0Z478W	WO2023093728A1_515	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCC(CN5CCC(OC6=CN=C(N7CCC(N8N=C(N)C9=C8C=C(C8=C(O)C=CC=C8)N=N9)CC7)N=C6)CC5)CC4)=[SH]O3)C(C)C)C=C2)SC=N1	C56H69N13O6S2	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-757YAK	SCHEMBL26157936	(2S,4R)-1-[2-[3-[4-[[3-[2-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]pyrimidin-5-yl]oxypyrrolidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCC(CN5CCC(OC6=CN=C(N7CCC(N8N=C(N)C9=C8C=C(C8=C(O)C=CC=C8)N=N9)CC7)N=C6)C5)CC4)=NO3)C(C)C)C=C2)SC=N1	C55H66N14O6S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-W51OQJ	SCHEMBL26157937	(2S,4R)-1-[2-[3-[4-[[4-[5-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]pyrazin-2-yl]piperazin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCC(CN5CCN(C6=NC=C(N7CCC(N8N=C(N)C9=C8C=C(C8=C(O)C=CC=C8)N=N9)CC7)N=C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C55H67N15O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-AQG3FB	SCHEMBL26157938	(2S,4R)-1-[2-[3-[4-[[4-[6-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]pyridazin-3-yl]piperazin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCC(CN5CCN(C6=CC=C(N7CCC(N8N=C(N)C9=C8C=C(C8=C(O)C=CC=C8)N=N9)CC7)N=N6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C55H67N15O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-X7H2UF	SCHEMBL26157939	2-[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]-N-[[1-[[1-[5-[1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]-1,2-oxazol-3-yl]piperidin-4-yl]methyl]piperidin-4-yl]methyl]pyrimidine-5-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCC(CN5CCC(CNC(=O)C6=CN=C(N7CCC(N8N=C(N)C9=C8C=C(C8=C(O)C=CC=C8)N=N9)CC7)N=C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C58H71N15O6S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-P0UYNI	SCHEMBL26157940	(2S,4R)-4-hydroxy-1-[(2S)-2-[[2-[4-[[4-[6-(2-hydroxyphenyl)-3-(methylamino)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]methyl]cyclohexyl]acetyl]amino]-3,3-dimethylbutanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CNC1=NN(C2CCN(CC3CCC(CC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)N[C@@H](C)C4=CC=C(C5=C(C)N=CS5)C=C4)C(C)(C)C)CC3)CC2)C2=C1N=NC(C1=C(O)C=CC=C1)=C2	C49H64N10O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-LN3R3J	SCHEMBL26157941	(2S,4R)-1-[2-[3-[4-[[4-[[4-[3-amino-6-(2-hydroxyphenyl)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCC(CN5CCC(CN6CCC(N7N=C(N)C8=C7C=C(C7=C(O)C=CC=C7)N=N8)CC6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C53H68N12O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-H64L67	SCHEMBL26157943	N-[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]-7-[[4-[6-(2-hydroxyphenyl)-3-(methylamino)pyrazolo[4,3-c]pyridazin-1-yl]piperidin-1-yl]methyl]-2-azaspiro[3.5]nonane-2-carboxamide	CNC1=NN(C2CCN(CC3CCC4(CC3)CN(C(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](C)C3=CC=C(C5=C(C)N=CS5)C=C3)C(C)(C)C)C4)CC2)C2=CC(C3=C(O)C=CC=C3)=NN=C21	C50H65N11O5S	SMARCA2	P51531	VHL	WO-2023093728-A1
TPD-B7WX40	SCHEMBL25267812	4-[4-[1-[4-[(3S)-2-(3-chloro-4-cyanophenyl)-3-methyl-2,8-diazaspiro[4.5]decan-8-yl]benzoyl]piperidin-4-yl]piperazin-1-yl]-N-(2,6-dioxopiperidin-3-yl)-2-fluorobenzamide; SCHEMBL30525366	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(N5CCN(c6ccc(C(=O)NC7CCC(=O)NC7=O)c(F)c6)CC5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H50ClFN8O4	AR	P10275	CRBN	WO-2023093845-A1
TPD-FS5MG0	SCHEMBL25268666	2-chloro-4-[(3S)-8-[4-[4-[4-[3-[(2,6-dioxopiperidin-3-yl)amino]phenyl]piperazin-1-yl]piperidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(N5CCN(c6cccc(NC7CCC(=O)NC7=O)c6)CC5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H51ClN8O3	AR	P10275	CRBN	WO-2023093845-A1
TPD-EKY3SB	SCHEMBL25634326	2-chloro-4-[(3S)-8-[4-[4-[[4-[3-[[(3S)-2,6-dioxopiperidin-3-yl]amino]phenyl]piperazin-1-yl]methyl]piperidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL30525359	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(CN5CCN(c6cccc(N[C@H]7CCC(=O)NC7=O)c6)CC5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H53ClN8O3	AR	P10275	CRBN	WO-2023093845-A1
TPD-R7VBPK	SCHEMBL25629496	2-chloro-4-[(3S)-8-[4-[4-[[4-[3-[[(3R)-2,6-dioxopiperidin-3-yl]amino]phenyl]piperazin-1-yl]methyl]piperidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL30525341	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(CN5CCN(c6cccc(N[C@@H]7CCC(=O)NC7=O)c6)CC5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H53ClN8O3	AR	P10275	CRBN	WO-2023093845-A1
TPD-J7AREZ	SCHEMBL25220352	2-chloro-4-[(3S)-8-[4-[4-[[4-[3-[(2,6-dioxopiperidin-3-yl)amino]phenyl]piperazin-1-yl]methyl]piperidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(CN5CCN(c6cccc(NC7CCC(=O)NC7=O)c6)CC5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H53ClN8O3	AR	P10275	CRBN	WO-2023093845-A1
TPD-VCLXJ3	WO2023093845A1_12-1	.	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(CN5CCN(c6cccc(N[C@H]7CCC(=O)NC7=O)c6)CC5)CC4)nc3)CC2)CC1c1ccc(C#N)c(Cl)c1	C44H53ClN8O3	AR	P10275	CRBN	WO-2023093845-A1
TPD-FBWFT4	SCHEMBL25629559	2-chloro-4-[(3S)-8-[6-[4-[[4-[3-[[(3R)-2,6-dioxopiperidin-3-yl]amino]phenyl]piperazin-1-yl]methyl]piperidine-1-carbonyl]pyridin-3-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL30525386	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(CN5CCN(c6cccc(N[C@@H]7CCC(=O)NC7=O)c6)CC5)CC4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H52ClN9O3	AR	P10275	CRBN	WO-2023093845-A1
TPD-YPHSA9	SCHEMBL25268696	2-chloro-4-[(3S)-8-[6-[4-[[4-[3-[(2,6-dioxopiperidin-3-yl)amino]phenyl]piperazin-1-yl]methyl]piperidine-1-carbonyl]pyridazin-3-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL30525369	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(CN5CCN(c6cccc(NC7CCC(=O)NC7=O)c6)CC5)CC4)nn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H51ClN10O3	AR	P10275	CRBN	WO-2023093845-A1
TPD-VQB4NH	SCHEMBL25263424	2-chloro-4-[(3S)-8-[4-[3-[[4-[3-[(2,6-dioxopiperidin-3-yl)amino]phenyl]piperazin-1-yl]methyl]azetidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CC(CN5CCN(c6cccc(NC7CCC(=O)NC7=O)c6)CC5)C4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H49ClN8O3	AR	P10275	CRBN	WO-2023093845-A1
TPD-NPNFQX	SCHEMBL25629677	2-chloro-4-[(3S)-8-[4-[4-[[4-[3-[[(3S)-2,6-dioxopiperidin-3-yl]amino]phenyl]piperazin-1-yl]methyl]piperidine-1-carbonyl]-2-fluorophenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL31230771	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(CN5CCN(c6cccc(N[C@H]7CCC(=O)NC7=O)c6)CC5)CC4)cc3F)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H52ClFN8O3	AR	P10275	CRBN	WO-2023093845-A1
TPD-GALFI5	SCHEMBL25629676	2-chloro-4-[(3S)-8-[4-[4-[[4-[3-[[(3R)-2,6-dioxopiperidin-3-yl]amino]phenyl]piperazin-1-yl]methyl]piperidine-1-carbonyl]-2-fluorophenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL31230798	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(CN5CCN(c6cccc(N[C@@H]7CCC(=O)NC7=O)c6)CC5)CC4)cc3F)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H52ClFN8O3	AR	P10275	CRBN	WO-2023093845-A1
TPD-JPANGK	WO2023093845A1_15	.	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(CN5CCN(c6cccc(NC7CCC(=O)NC7=O)c6)CC5)CC4)cc3F)CC2)CC1c1ccc(C#N)c(Cl)c1	C45H53ClFN7O3	AR	P10275	CRBN	WO-2023093845-A1
TPD-II8NVP	SCHEMBL25262676	2-chloro-4-[(3S)-8-[4-[4-[[4-[3-[(2,6-dioxopiperidin-3-yl)amino]phenyl]piperazin-1-yl]methyl]piperidine-1-carbonyl]-3-fluorophenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(CN5CCN(c6cccc(NC7CCC(=O)NC7=O)c6)CC5)CC4)c(F)c3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H52ClFN8O3	AR	P10275	CRBN	WO-2023093845-A1
TPD-FEZE1I	SCHEMBL25220104	2-chloro-4-[(3S)-8-[5-[4-[[4-[3-[(2,6-dioxopiperidin-3-yl)amino]phenyl]piperazin-1-yl]methyl]piperidine-1-carbonyl]pyrazin-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL30525302	C[C@H]1CC2(CCN(c3cnc(C(=O)N4CCC(CN5CCN(c6cccc(NC7CCC(=O)NC7=O)c6)CC5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C42H51ClN10O3	AR	P10275	CRBN	WO-2023093845-A1
TPD-9E87TE	SCHEMBL25224212	2-chloro-4-[(3S)-8-[5-[4-[[4-[3-[(2,6-dioxopiperidin-3-yl)amino]phenyl]piperazin-1-yl]methyl]piperidine-1-carbonyl]pyridin-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(CN5CCN(c6cccc(NC7CCC(=O)NC7=O)c6)CC5)CC4)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H52ClN9O3	AR	P10275	CRBN	WO-2023093845-A1
TPD-UXOJBS	SCHEMBL25220290	2-chloro-4-[(3S)-8-[4-[4-[[4-[3-[(2,6-dioxopiperidin-3-yl)amino]phenyl]piperidin-1-yl]methyl]piperidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(CN5CCC(c6cccc(NC7CCC(=O)NC7=O)c6)CC5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H54ClN7O3	AR	P10275	CRBN	WO-2023093845-A1
TPD-08F4E4	SCHEMBL25220326	5-[4-[1-[4-[(3S)-2-(3-chloro-4-cyanophenyl)-3-methyl-2,8-diazaspiro[4.5]decan-8-yl]benzoyl]piperidin-4-yl]piperazin-1-yl]-N-(2,6-dioxopiperidin-3-yl)pyridine-2-carboxamide; SCHEMBL30525299	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(N5CCN(c6ccc(C(=O)NC7CCC(=O)NC7=O)nc6)CC5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H50ClN9O4	AR	P10275	CRBN	WO-2023093845-A1
TPD-09N7H8	WO2023093845A1_20	.	C[C@H]1CC2(CCN(C3=CC=C(C(=O)N4CCC(CN5CCC(c6cccc(NC7CCC(=O)NC7=O)c6)CC5)CC4)NN3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H54ClN9O3	AR	P10275	CRBN	WO-2023093845-A1
TPD-OEC2EB	SCHEMBL25260462	2-chloro-4-[(3S)-8-[6-[3-[[4-[3-[(2,6-dioxopiperidin-3-yl)amino]phenyl]piperidin-1-yl]methyl]azetidine-1-carbonyl]pyridazin-3-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL30525412	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CC(CN5CCC(c6cccc(NC7CCC(=O)NC7=O)c6)CC5)C4)nn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C41H48ClN9O3	AR	P10275	CRBN	WO-2023093845-A1
TPD-AP24CN	SCHEMBL25273437	2-chloro-4-[(3S)-8-[6-[3-[[4-[3-[(2,6-dioxopiperidin-3-yl)amino]phenyl]piperazin-1-yl]methyl]azetidine-1-carbonyl]pyridazin-3-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL30525306	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CC(CN5CCN(c6cccc(NC7CCC(=O)NC7=O)c6)CC5)C4)nn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C40H47ClN10O3	AR	P10275	CRBN	WO-2023093845-A1
TPD-ORVYFN	SCHEMBL25267421	2-chloro-4-[(3S)-8-[4-[4-[[4-[5-[(2,6-dioxopiperidin-3-yl)amino]-2-fluorophenyl]piperazin-1-yl]methyl]piperidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(CN5CCN(c6cc(NC7CCC(=O)NC7=O)ccc6F)CC5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H52ClFN8O3	AR	P10275	CRBN	WO-2023093845-A1
TPD-D0XJ4H	SCHEMBL25222835	2-chloro-4-[(3S)-8-[4-[4-[[4-[4-[(2,6-dioxopiperidin-3-yl)amino]pyridin-2-yl]piperazin-1-yl]methyl]piperidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(CN5CCN(c6cc(NC7CCC(=O)NC7=O)ccn6)CC5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H52ClN9O3	AR	P10275	CRBN	WO-2023093845-A1
TPD-9PMRMT	SCHEMBL25221165	2-chloro-4-[(3S)-8-[4-[4-[[4-[4-[(2,6-dioxopiperidin-3-yl)amino]phenyl]piperazin-1-yl]methyl]piperidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(CN5CCN(c6ccc(NC7CCC(=O)NC7=O)cc6)CC5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H53ClN8O3	AR	P10275	CRBN	WO-2023093845-A1
TPD-7AG1D2	SCHEMBL25256339	2-chloro-4-[(3S)-8-[4-[4-[[4-[4-[(2,6-dioxopiperidin-3-yl)amino]-2-fluorophenyl]piperidin-1-yl]methyl]piperidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(CN5CCC(c6ccc(NC7CCC(=O)NC7=O)cc6F)CC5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H53ClFN7O3	AR	P10275	CRBN	WO-2023093845-A1
TPD-ZRSBAZ	SCHEMBL25269249	2-chloro-4-[(3S)-8-[4-[2-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperazin-1-yl]-7-azaspiro[3.5]nonane-7-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC5(CC4)CC(N4CCN(c6ccc(N7CCC(=O)NC7=O)cc6)CC4)C5)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H53ClN8O3	AR	P10275	CRBN	WO-2023093845-A1
TPD-4JKLAK	SCHEMBL25267816	2-chloro-4-[(3S)-8-[4-[9-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperazin-1-yl]-3-azaspiro[5.5]undecane-3-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC5(CCC(N6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C47H57ClN8O3	AR	P10275	CRBN	WO-2023093845-A1
TPD-52BDBQ	SCHEMBL25220287	4-[4-[[1-[4-[(3S)-2-(3-chloro-4-cyanophenyl)-3-methyl-2,8-diazaspiro[4.5]decan-8-yl]benzoyl]piperidin-4-yl]methyl]piperazin-1-yl]-N-(2,6-dioxopiperidin-3-yl)-2-fluorobenzamide; SCHEMBL30525371	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(CN5CCN(c6ccc(C(=O)NC7CCC(=O)NC7=O)c(F)c6)CC5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H52ClFN8O4	AR	P10275	CRBN	WO-2023093845-A1
TPD-MQ9KOB	SCHEMBL25630557	2-chloro-4-[(3S)-8-[4-[2-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperazin-1-yl]-7-azaspiro[3.5]nonane-7-carbonyl]-2-fluorophenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL30525396	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC5(CC4)CC(N4CCN(c6ccc(N7CCC(=O)NC7=O)cc6)CC4)C5)cc3F)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H52ClFN8O3	AR	P10275	CRBN	WO-2023093845-A1
TPD-TMUMCR	SCHEMBL25634669	2-chloro-4-[(3S)-8-[4-[2-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperazin-1-yl]-7-azaspiro[3.5]nonane-7-carbonyl]-3-fluorophenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL30525345	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC5(CC4)CC(N4CCN(c6ccc(N7CCC(=O)NC7=O)cc6)CC4)C5)c(F)c3)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H52ClFN8O3	AR	P10275	CRBN	WO-2023093845-A1
TPD-JGSA3L	SCHEMBL25630560	2-chloro-4-[(3S)-8-[6-[2-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperazin-1-yl]-7-azaspiro[3.5]nonane-7-carbonyl]pyridin-3-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL31230697	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC5(CC4)CC(N4CCN(c6ccc(N7CCC(=O)NC7=O)cc6)CC4)C5)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H52ClN9O3	AR	P10275	CRBN	WO-2023093845-A1
TPD-NTYJ8I	SCHEMBL25634708	2-chloro-4-[(3S)-8-[5-[2-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperazin-1-yl]-7-azaspiro[3.5]nonane-7-carbonyl]pyridin-2-yl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL31230727	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC5(CC4)CC(N4CCN(c6ccc(N7CCC(=O)NC7=O)cc6)CC4)C5)cn3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H52ClN9O3	AR	P10275	CRBN	WO-2023093845-A1
TPD-4VVE88	SCHEMBL25217026	2-chloro-4-[(3S)-8-[4-[2-[4-[4-(2,6-dioxopiperidin-3-yl)phenyl]piperazin-1-yl]-7-azaspiro[3.5]nonane-7-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC5(CC4)CC(N4CCN(c6ccc(C7CCC(=O)NC7=O)cc6)CC4)C5)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C46H54ClN7O3	AR	P10275	CRBN	WO-2023093845-A1
TPD-VRTJP6	SCHEMBL25224983	2-chloro-4-[(3S)-8-[4-[2-[4-[3-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperazin-1-yl]-7-azaspiro[3.5]nonane-7-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC5(CC4)CC(N4CCN(c6cccc(N7CCC(=O)NC7=O)c6)CC4)C5)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H53ClN8O3	AR	P10275	CRBN	WO-2023093845-A1
TPD-WET8LU	SCHEMBL25634745	2-chloro-4-[(3S)-8-[4-[2-[4-[3-[(2,6-dioxopiperidin-3-yl)amino]phenyl]piperazin-1-yl]-7-azaspiro[3.5]nonane-7-carbonyl]-2-fluorophenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL30525315	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC5(CC4)CC(N4CCN(c6cccc(NC7CCC(=O)NC7=O)c6)CC4)C5)cc3F)CC2)CN1c1ccc(C#N)c(Cl)c1	C46H54ClFN8O3	AR	P10275	CRBN	WO-2023093845-A1
TPD-MK3J4I	SCHEMBL25220842	2-chloro-4-[(3S)-8-[4-[4-[[1-[3-[(2,6-dioxopiperidin-3-yl)amino]phenyl]piperidin-4-yl]methyl]piperazine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(CC5CCN(c6cccc(NC7CCC(=O)NC7=O)c6)CC5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H53ClN8O3	AR	P10275	CRBN	WO-2023093845-A1
TPD-05FFW0	SCHEMBL25269424	2-Chloro-4-[8-[4-[4-[[4-[3-[(2,6-dioxopiperidin-3-yl)amino]phenyl]piperazin-1-yl]methyl]piperidine-1-carbonyl]phenyl]-2,8-diazaspiro[4.5]decan-2-yl]-3-methylbenzonitrile	Cc1c(N2CCC3(CCN(c4ccc(C(=O)N5CCC(CN6CCN(c7cccc(NC8CCC(=O)NC8=O)c7)CC6)CC5)cc4)CC3)C2)ccc(C#N)c1Cl	C44H53ClN8O3	AR	P10275	CRBN	WO-2023093845-A1
TPD-43KBBU	SCHEMBL25260475	2-chloro-4-[(3S)-8-[4-[4-[[4-[2-[(2,6-dioxopiperidin-3-yl)amino]phenyl]piperazin-1-yl]methyl]piperidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL30525339	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(CN5CCN(c6ccccc6NC6CCC(=O)NC6=O)CC5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H53ClN8O3	AR	P10275	CRBN	WO-2023093845-A1
TPD-FW80DE	SCHEMBL25269228	5-[4-[[1-[4-[(3S)-2-(3-chloro-4-cyanophenyl)-3-methyl-2,8-diazaspiro[4.5]decan-8-yl]benzoyl]piperidin-4-yl]methyl]piperazin-1-yl]-N-(2,6-dioxopiperidin-3-yl)pyridine-2-carboxamide; SCHEMBL30525356	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(CN5CCN(c6ccc(C(=O)NC7CCC(=O)NC7=O)nc6)CC5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H52ClN9O4	AR	P10275	CRBN	WO-2023093845-A1
TPD-DSUJ5W	SCHEMBL25222787	2-chloro-4-[(3S)-8-[4-[4-[[4-[3-[(2,6-dioxopiperidin-3-yl)amino]phenyl]-3-oxopiperazin-1-yl]methyl]piperidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(CN5CCN(c6cccc(NC7CCC(=O)NC7=O)c6)C(=O)C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C44H51ClN8O4	AR	P10275	CRBN	WO-2023093845-A1
TPD-0RCF9L	SCHEMBL25221947	4-[(3S)-8-[4-[4-[[4-[3-[(2,6-dioxopiperidin-3-yl)amino]phenyl]piperazin-1-yl]methyl]piperidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]-2-(trifluoromethyl)benzonitrile; SCHEMBL31230807	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(CN5CCN(c6cccc(NC7CCC(=O)NC7=O)c6)CC5)CC4)cc3)CC2)CN1c1ccc(C#N)c(C(F)(F)F)c1	C45H53F3N8O3	AR	P10275	CRBN	WO-2023093845-A1
TPD-I6LXEJ	SCHEMBL25273442	2-[4-[4-[(3S)-2-(3-chloro-4-cyanophenyl)-3-methyl-2,8-diazaspiro[4.5]decan-8-yl]benzoyl]piperazin-1-yl]-N-[3-[(2,6-dioxopiperidin-3-yl)amino]phenyl]acetamide; SCHEMBL31230622	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCN(CC(=O)Nc5cccc(NC6CCC(=O)NC6=O)c5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C40H45ClN8O4	AR	P10275	CRBN	WO-2023093845-A1
TPD-C2U45H	SCHEMBL25267779	4-[4-[[1-[4-[(3S)-2-(3-chloro-4-cyanophenyl)-3-methyl-2,8-diazaspiro[4.5]decan-8-yl]benzoyl]piperidin-4-yl]methyl]piperazin-1-yl]-N-(2,6-dioxopiperidin-3-yl)benzamide; SCHEMBL30525381	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(CN5CCN(c6ccc(C(=O)NC7CCC(=O)NC7=O)cc6)CC5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H53ClN8O4	AR	P10275	CRBN	WO-2023093845-A1
TPD-RQ7U7F	WO2023093845A1_5	.	C[C@H]1CC2(CCC(C(=O)c3ccc(SC4CCN(C5CN(c6ccc(C(=O)NC7CCC(=O)NC7=O)c(F)c6)C5)CC4)nc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C43H47ClFN7O4S	AR	P10275	CRBN	WO-2023093845-A1
TPD-2ZZX4K	SCHEMBL25268698	2-chloro-4-[(3S)-8-[4-[4-[4-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperazin-1-yl]piperidin-1-yl]piperidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(N5CCC(N6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C47H58ClN9O3	AR	P10275	CRBN	WO-2023093845-A1
TPD-05GZ1I	SCHEMBL25634187	2-chloro-4-[(3S)-8-[4-[4-[3-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperazin-1-yl]azetidin-1-yl]piperidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(N5CC(N6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H54ClN9O3	AR	P10275	CRBN	WO-2023093845-A1
TPD-6C35LE	SCHEMBL25634194	2-chloro-4-[(3S)-8-[4-[4-[[3-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperazin-1-yl]azetidin-1-yl]methyl]piperidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL31230642	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(CN5CC(N6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C46H56ClN9O3	AR	P10275	CRBN	WO-2023093845-A1
TPD-SPHYFH	SCHEMBL25629380	2-chloro-4-[(3S)-8-[4-[4-[[4-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperazin-1-yl]piperidin-1-yl]methyl]piperidine-1-carbonyl]phenyl]-3-methyl-2,8-diazaspiro[4.5]decan-2-yl]benzonitrile; SCHEMBL31230753	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(CN5CCC(N6CCN(c7ccc(N8CCC(=O)NC8=O)cc7)CC6)CC5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C48H60ClN9O3	AR	P10275	CRBN	WO-2023093845-A1
TPD-EK1K4G	SCHEMBL25206128	N-(2-chloro-6-methylphenyl)-2-[[6-[4-[6-[2-[2-[6-[4-(2,6-dioxopiperidin-3-yl)anilino]-6-oxohexoxy]ethoxy]ethoxy]hexyl]piperazin-1-yl]-2-methylpyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide; SCHEMBL30429932	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCCCCOCCOCCOCCCCCC(=O)Nc3ccc(C4CCC(=O)NC4=O)cc3)CC2)n1	C47H62ClN9O7S	LCK	P06239	CRBN	WO-2023096995-A1
TPD-KPYTNK	SCHEMBL25208376	N-(2-chloro-6-methylphenyl)-2-[[6-[4-[6-[2-[2-[6-[3-(2,6-dioxopiperidin-3-yl)anilino]-6-oxohexoxy]ethoxy]ethoxy]hexyl]piperazin-1-yl]-2-methylpyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide; SCHEMBL30429716	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCCCCOCCOCCOCCCCCC(=O)Nc3cccc(C4CCC(=O)NC4=O)c3)CC2)n1	C47H62ClN9O7S	LCK	P06239	CRBN	WO-2023096995-A1
TPD-A3B9FN	SCHEMBL25205474	N-(2-chloro-6-methylphenyl)-2-[[6-[4-[6-[2-[2-[4-(2,6-dioxopiperidin-3-yl)anilino]-2-oxoethoxy]ethoxy]hexyl]piperazin-1-yl]-2-methylpyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide; SCHEMBL30429688	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCCCCOCCOCC(=O)Nc3ccc(C4CCC(=O)NC4=O)cc3)CC2)n1	C41H50ClN9O6S	LCK	P06239	CRBN	WO-2023096995-A1
TPD-SDGG3V	SCHEMBL25205845	N-(2-chloro-6-methylphenyl)-2-[[6-[4-[6-[2-[2-[3-(2,6-dioxopiperidin-3-yl)anilino]-2-oxoethoxy]ethoxy]hexyl]piperazin-1-yl]-2-methylpyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide; SCHEMBL30429744	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCCCCOCCOCC(=O)Nc3cccc(C4CCC(=O)NC4=O)c3)CC2)n1	C41H50ClN9O6S	LCK	P06239	CRBN	WO-2023096995-A1
TPD-E1TLSX	SCHEMBL25209230	N-(2-chloro-6-methylphenyl)-2-[[6-[4-[6-[2-[2-[2-[2-[2-[2-[4-(2,6-dioxopiperidin-3-yl)anilino]-2-oxoethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]hexyl]piperazin-1-yl]-2-methylpyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide; SCHEMBL30430017	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCCCCOCCOCCOCCOCCOCCOCC(=O)Nc3ccc(C4CCC(=O)NC4=O)cc3)CC2)n1	C49H66ClN9O10S	LCK	P06239	CRBN	WO-2023096995-A1
TPD-UTPUCD	SCHEMBL25232980	N-(2-chloro-6-methylphenyl)-2-[[6-[4-[6-[2-[2-[2-[2-[2-[2-[3-(2,6-dioxopiperidin-3-yl)anilino]-2-oxoethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]hexyl]piperazin-1-yl]-2-methylpyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide; SCHEMBL30429729	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCCCCOCCOCCOCCOCCOCCOCC(=O)Nc3cccc(C4CCC(=O)NC4=O)c3)CC2)n1	C49H66ClN9O10S	LCK	P06239	CRBN	WO-2023096995-A1
TPD-PS6S6O	SCHEMBL25227536	N-(2-chloro-6-methylphenyl)-2-[[6-[4-[6-[4-(2,6-dioxopiperidin-3-yl)anilino]-6-oxohexyl]piperazin-1-yl]-2-methylpyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide; SCHEMBL30429842	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCCCC(=O)Nc3ccc(C4CCC(=O)NC4=O)cc3)CC2)n1	C37H42ClN9O4S	LCK	P06239	CRBN	WO-2023096995-A1
TPD-9RIX0C	SCHEMBL25244012	N-(2-chloro-6-methylphenyl)-2-[[6-[4-[6-[3-(2,6-dioxopiperidin-3-yl)anilino]-6-oxohexyl]piperazin-1-yl]-2-methylpyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide; SCHEMBL30429237	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCCCC(=O)Nc3cccc(C4CCC(=O)NC4=O)c3)CC2)n1	C37H42ClN9O4S	LCK	P06239	CRBN	WO-2023096995-A1
TPD-SC764K	orb1979943	N-(2-chloro-6-methylphenyl)-2-[[6-[4-[3-[[2-[4-(2,6-dioxopiperidin-3-yl)phenoxy]acetyl]amino]propyl]piperazin-1-yl]-2-methylpyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide; CHEMBL5270900; SCHEMBL25208355; SCHEMBL30428950; NSC836838; NSC-836838; SJ11646	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCNC(=O)COc3ccc(C4CCC(=O)NC4=O)cc3)CC2)n1	C36H40ClN9O5S	LCK	P06239	CRBN	WO-2023096995-A1
TPD-AMX2ME	SCHEMBL25207489	N-(2-chloro-6-methylphenyl)-2-[[6-[4-[3-[[2-[3-(2,6-dioxopiperidin-3-yl)phenoxy]acetyl]amino]propyl]piperazin-1-yl]-2-methylpyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide; SCHEMBL30429263	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCNC(=O)COc3cccc(C4CCC(=O)NC4=O)c3)CC2)n1	C36H40ClN9O5S	LCK	P06239	CRBN	WO-2023096995-A1
TPD-PRQPM9	WO2023096995A1_11	.	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2C[C@@H](C)N(CCCNC(=O)COc3ccc(C4CCC(=O)NC4=O)cc3)C[C@H]2C)n1	C38H44ClN9O5S	LCK	P06239	CRBN	WO-2023096995-A1
TPD-OF2RUB	WO2023096995A1_12	.	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCCCCOCCOCCOCCCCCC(=O)Nc3cccc4c3C(=O)C(C3CCC(=O)N(C)C3=O)C4=O)CC2)n1	C51H64ClN9O9S	LCK	P06239	CRBN	WO-2023096995-A1
TPD-CUV3XJ	WO2023096995A1_13	.	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCCCCOCCOCCOCCCCCC(=O)Nc3cccc4c3C(=O)C(C3CCC(=O)NC3=O)C4=O)CC2)n1	C50H62ClN9O9S	LCK	P06239	CRBN	WO-2023096995-A1
TPD-DWY2O1	CHEMBL5268757	N-(2-chloro-6-methylphenyl)-2-[[6-[4-[3-[[2-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenoxy]acetyl]amino]propyl]piperazin-1-yl]-2-methylpyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide; SCHEMBL25206192; SCHEMBL30428919; SJ34739	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCNC(=O)COc3ccc(N4CCC(=O)NC4=O)cc3)CC2)n1	C35H39ClN10O5S	LCK	P06239	CRBN	WO-2023096995-A1
TPD-B8SCGH	SCHEMBL25209192	N-(2-chloro-6-methylphenyl)-2-[[6-[4-[5-[5-[4-(2,6-dioxopiperidin-3-yl)phenyl]-2,5-diazabicyclo[2.2.1]heptan-2-yl]-5-oxopentyl]piperazin-1-yl]-2-methylpyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide; SCHEMBL30429681	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCCC(=O)N3CC4CC3CN4c3ccc(C4CCC(=O)NC4=O)cc3)CC2)n1	C41H47ClN10O4S	LCK	P06239	CRBN	WO-2023096995-A1
TPD-ZNGP23	SCHEMBL25239181	N-(2-chloro-6-methylphenyl)-2-[[6-[4-[5-[5-[4-(2,6-dioxopiperidin-3-yl)phenyl]-2,5-diazabicyclo[2.2.2]octan-2-yl]-5-oxopentyl]piperazin-1-yl]-2-methylpyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide; SCHEMBL30429260	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCCC(=O)N3CC4CCC3CN4c3ccc(C4CCC(=O)NC4=O)cc3)CC2)n1	C42H49ClN10O4S	LCK	P06239	CRBN	WO-2023096995-A1
TPD-CHAXHT	SCHEMBL25203775	N-(2-chloro-6-methylphenyl)-2-[[6-[4-[5-[8-[4-(2,6-dioxopiperidin-3-yl)phenyl]-3,8-diazabicyclo[3.2.1]octan-3-yl]-5-oxopentyl]piperazin-1-yl]-2-methylpyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide; SCHEMBL30429374	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCCC(=O)N3CC4CCC(C3)N4c3ccc(C4CCC(=O)NC4=O)cc3)CC2)n1	C42H49ClN10O4S	LCK	P06239	CRBN	WO-2023096995-A1
TPD-AUFME0	SCHEMBL25206738	N-(2-chloro-6-methylphenyl)-2-[[6-[4-[4-[5-[4-(2,6-dioxopiperidin-3-yl)phenyl]-2,5-diazabicyclo[2.2.1]heptan-2-yl]-4-oxobutyl]piperazin-1-yl]-2-methylpyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide; SCHEMBL30429543	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCC(=O)N3CC4CC3CN4c3ccc(C4CCC(=O)NC4=O)cc3)CC2)n1	C40H45ClN10O4S	LCK	P06239	CRBN	WO-2023096995-A1
TPD-8R1J3E	SCHEMBL25239049	N-(2-chloro-6-methylphenyl)-2-[[6-[4-[4-[5-[4-(2,6-dioxopiperidin-3-yl)phenyl]-2,5-diazabicyclo[2.2.2]octan-2-yl]-4-oxobutyl]piperazin-1-yl]-2-methylpyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide; SCHEMBL30429696	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCC(=O)N3CC4CCC3CN4c3ccc(C4CCC(=O)NC4=O)cc3)CC2)n1	C41H47ClN10O4S	LCK	P06239	CRBN	WO-2023096995-A1
TPD-L3DJF2	SCHEMBL25235798	N-(2-chloro-6-methylphenyl)-2-[[6-[4-[4-[8-[4-(2,6-dioxopiperidin-3-yl)phenyl]-3,8-diazabicyclo[3.2.1]octan-3-yl]-4-oxobutyl]piperazin-1-yl]-2-methylpyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide; SCHEMBL30430182	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCC(=O)N3CC4CCC(C3)N4c3ccc(C4CCC(=O)NC4=O)cc3)CC2)n1	C41H47ClN10O4S	LCK	P06239	CRBN	WO-2023096995-A1
TPD-8HGPOG	SCHEMBL25206733	N-(2-chloro-6-methylphenyl)-2-[[6-[4-[4-[9-[4-(2,6-dioxopiperidin-3-yl)phenyl]-3,9-diazaspiro[5.5]undecan-3-yl]-4-oxobutyl]piperazin-1-yl]-2-methylpyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide; SCHEMBL30428942	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCC(=O)N3CCC4(CC3)CCN(c3ccc(C5CCC(=O)NC5=O)cc3)CC4)CC2)n1	C44H53ClN10O4S	LCK	P06239	CRBN	WO-2023096995-A1
TPD-9HBJG3	SCHEMBL25207515	N-(2-chloro-6-methylphenyl)-2-[[6-[4-[4-[8-[4-(2,6-dioxopiperidin-3-yl)phenyl]-2,8-diazaspiro[4.5]decan-2-yl]-4-oxobutyl]piperazin-1-yl]-2-methylpyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide; SCHEMBL30429710	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCC(=O)N3CCC4(CCN(c5ccc(C6CCC(=O)NC6=O)cc5)CC4)C3)CC2)n1	C43H51ClN10O4S	LCK	P06239	CRBN	WO-2023096995-A1
TPD-3FKZDS	SCHEMBL25205852	N-(2-chloro-6-methylphenyl)-2-[[6-[4-[4-[6-[4-(2,6-dioxopiperidin-3-yl)phenyl]-2,6-diazaspiro[3.3]heptan-2-yl]-4-oxobutyl]piperazin-1-yl]-2-methylpyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide; SCHEMBL30430735	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCC(=O)N3CC4(C3)CN(c3ccc(C5CCC(=O)NC5=O)cc3)C4)CC2)n1	C40H45ClN10O4S	LCK	P06239	CRBN	WO-2023096995-A1
TPD-H2BLPR	SCHEMBL25232367	N-(2-chloro-6-methylphenyl)-2-[[6-[4-[5-[9-[4-(2,6-dioxopiperidin-3-yl)phenyl]-3,9-diazaspiro[5.5]undecan-3-yl]-5-oxopentyl]piperazin-1-yl]-2-methylpyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide; SCHEMBL30429375	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCCC(=O)N3CCC4(CC3)CCN(c3ccc(C5CCC(=O)NC5=O)cc3)CC4)CC2)n1	C45H55ClN10O4S	LCK	P06239	CRBN	WO-2023096995-A1
TPD-XLGIZP	SCHEMBL25204595	N-(2-chloro-6-methylphenyl)-2-[[6-[4-[5-[8-[4-(2,6-dioxopiperidin-3-yl)phenyl]-2,8-diazaspiro[4.5]decan-2-yl]-5-oxopentyl]piperazin-1-yl]-2-methylpyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide; SCHEMBL30428961	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCCC(=O)N3CCC4(CCN(c5ccc(C6CCC(=O)NC6=O)cc5)CC4)C3)CC2)n1	C44H53ClN10O4S	LCK	P06239	CRBN	WO-2023096995-A1
TPD-ZDYUCT	SCHEMBL25225299	N-(2-chloro-6-methylphenyl)-2-[[6-[4-[5-[6-[4-(2,6-dioxopiperidin-3-yl)phenyl]-2,6-diazaspiro[3.3]heptan-2-yl]-5-oxopentyl]piperazin-1-yl]-2-methylpyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide; SCHEMBL30429735	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCCC(=O)N3CC4(C3)CN(c3ccc(C5CCC(=O)NC5=O)cc3)C4)CC2)n1	C41H47ClN10O4S	LCK	P06239	CRBN	WO-2023096995-A1
TPD-7E2TTE	CHEMBL5276245	N-(2-chloro-6-methylphenyl)-2-[[6-[4-[4-[4-[4-(2,6-dioxopiperidin-3-yl)phenyl]piperazin-1-yl]-4-oxobutyl]piperazin-1-yl]-2-methylpyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide; SCHEMBL25226200; SCHEMBL30429986; SJ34769	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCC(=O)N3CCN(c4ccc(C5CCC(=O)NC5=O)cc4)CC3)CC2)n1	C39H45ClN10O4S	LCK	P06239	CRBN	WO-2023096995-A1
TPD-24ROLB	SCHEMBL25207030	N-(2-chloro-6-methylphenyl)-2-[[6-[4-[5-[4-[4-(2,6-dioxopiperidin-3-yl)phenyl]piperazin-1-yl]-5-oxopentyl]piperazin-1-yl]-2-methylpyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide; SCHEMBL30429755	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCCC(=O)N3CCN(c4ccc(C5CCC(=O)NC5=O)cc4)CC3)CC2)n1	C40H47ClN10O4S	LCK	P06239	CRBN	WO-2023096995-A1
TPD-VEFD4W	WO2023096995A1_29	.	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2C[C@@H](C)N(CCCNC(=O)COc3ccc(N4CCC(=O)NC4=O)cc3)C[C@H]2C)n1	C37H43ClN10O5S	LCK	P06239	CRBN	WO-2023096995-A1
TPD-AZQZMK	WO2023096995A1_30	N-(2-chloro-6-methylphenyl)-2-[[2-methyl-6-[4-[3-[[2-[4-(1-methyl-2,6-dioxopiperidin-3-yl)phenoxy]acetyl]amino]propyl]piperazin-1-yl]pyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCNC(=O)COc3ccc(C4CCC(=O)N(C)C4=O)cc3)CC2)n1	C37H42ClN9O5S	LCK	P06239	CRBN	WO-2023096995-A1
TPD-2Q4592	SCHEMBL25564453	N-(2-chloro-6-methylphenyl)-2-[[6-[(1S,4S)-5-[4-[5-[4-(2,6-dioxopiperidin-3-yl)phenyl]-2,5-diazabicyclo[2.2.1]heptan-2-yl]-4-oxobutyl]-2,5-diazabicyclo[2.2.1]heptan-2-yl]-2-methylpyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2C[C@@H]3C[C@H]2CN3CCCC(=O)N2CC3CC2CN3c2ccc(C3CCC(=O)NC3=O)cc2)n1	C41H45ClN10O4S	LCK	P06239	CRBN	WO-2023096995-A1
TPD-F1S9AI	SCHEMBL25208339	N-(2-chloro-6-methylphenyl)-2-[[6-[4-[4-[4-[[4-[4-(2,6-dioxopiperidin-3-yl)phenyl]piperazin-1-yl]methyl]piperidin-1-yl]-4-oxobutyl]piperazin-1-yl]-2-methylpyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide; SCHEMBL30429900	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCC(=O)N3CCC(CN4CCN(c5ccc(C6CCC(=O)NC6=O)cc5)CC4)CC3)CC2)n1	C45H56ClN11O4S	LCK	P06239	CRBN	WO-2023096995-A1
TPD-7GKJDD	SCHEMBL25203231	N-(2-chloro-6-methylphenyl)-2-[[6-[4-[3-[4-[4-(2,6-dioxopiperidin-3-yl)phenyl]piperazin-1-yl]propyl]piperazin-1-yl]-2-methylpyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide; SCHEMBL30429847	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCN3CCN(c4ccc(C5CCC(=O)NC5=O)cc4)CC3)CC2)n1	C38H45ClN10O3S	LCK	P06239	CRBN	WO-2023096995-A1
TPD-HKIFF8	SCHEMBL25206718	N-(2-chloro-6-methylphenyl)-2-[[6-[4-[4-[4-[4-(2,6-dioxopiperidin-3-yl)phenyl]piperazin-1-yl]butanoyl]piperazin-1-yl]-2-methylpyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide; SCHEMBL30429946	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(C(=O)CCCN3CCN(c4ccc(C5CCC(=O)NC5=O)cc4)CC3)CC2)n1	C39H45ClN10O4S	LCK	P06239	CRBN	WO-2023096995-A1
TPD-8GTRXM	SCHEMBL25209210	N-(2-chloro-6-methylphenyl)-2-[[6-[4-[4-[5-[4-(2,6-dioxopiperidin-3-yl)phenyl]-2,5-diazabicyclo[2.2.1]heptan-2-yl]butanoyl]piperazin-1-yl]-2-methylpyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide; SCHEMBL30429752	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(C(=O)CCCN3CC4CC3CN4c3ccc(C4CCC(=O)NC4=O)cc3)CC2)n1	C40H45ClN10O4S	LCK	P06239	CRBN	WO-2023096995-A1
TPD-3Z3RPC	SCHEMBL25206743	2-[[6-[4-[4-[(3aR,6aS)-2-[4-(2,6-dioxopiperidin-3-yl)phenyl]-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-5-yl]-4-oxobutyl]piperazin-1-yl]-2-methylpyrimidin-4-yl]amino]-N-(2-chloro-6-methylphenyl)-1,3-thiazole-5-carboxamide; SCHEMBL30429228	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCC(=O)N3C[C@@H]4CN(c5ccc(C6CCC(=O)NC6=O)cc5)C[C@@H]4C3)CC2)n1	C41H47ClN10O4S	LCK	P06239	CRBN	WO-2023096995-A1
TPD-UCOFRI	SCHEMBL25206196	N-(2-chloro-6-methylphenyl)-2-[[6-[4-[3-[[2-[4-(2,4-dioxopyrimidin-1-yl)phenoxy]acetyl]amino]propyl]piperazin-1-yl]-2-methylpyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide; SCHEMBL30429292	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCNC(=O)COc3ccc(-n4ccc(=O)[nH]c4=O)cc3)CC2)n1	C35H37ClN10O5S	LCK	P06239	CRBN	WO-2023096995-A1
TPD-CVLBAG	SCHEMBL25215651	N-(2-chloro-6-methylphenyl)-2-[[6-[4-[3-[[2-[4-(2,4-dioxo-1,3-diazinan-1-yl)-2,5-difluorophenoxy]acetyl]amino]propyl]piperazin-1-yl]-2-methylpyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide; SCHEMBL30429525	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCNC(=O)COc3cc(F)c(N4CCC(=O)NC4=O)cc3F)CC2)n1	C35H37ClF2N10O5S	LCK	P06239	CRBN	WO-2023096995-A1
TPD-Y0OFLI	SCHEMBL25205860	N-(2-chloro-6-methylphenyl)-2-[[6-[4-[3-[[2-[4-(2,4-dioxo-1,3-diazinan-1-yl)-3-fluorophenoxy]acetyl]amino]propyl]piperazin-1-yl]-2-methylpyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide; SCHEMBL30429666	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCNC(=O)COc3ccc(N4CCC(=O)NC4=O)c(F)c3)CC2)n1	C35H38ClFN10O5S	LCK	P06239	CRBN	WO-2023096995-A1
TPD-SX3Z7M	SCHEMBL25208396	N-(2-chloro-6-methylphenyl)-2-[[6-[4-[3-[[2-[4-(2,4-dioxo-1,3-diazinan-1-yl)-2-fluorophenoxy]acetyl]amino]propyl]piperazin-1-yl]-2-methylpyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide; SCHEMBL30429774	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCNC(=O)COc3ccc(N4CCC(=O)NC4=O)cc3F)CC2)n1	C35H38ClFN10O5S	LCK	P06239	CRBN	WO-2023096995-A1
TPD-5B8XOV	SCHEMBL25564628	N-(2-chloro-6-methylphenyl)-2-[[6-[4-[4-[(1S,4S)-5-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]-2,5-diazabicyclo[2.2.1]heptan-2-yl]-4-oxobutyl]piperazin-1-yl]-2-methylpyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCC(=O)N3C[C@@H]4C[C@H]3CN4c3ccc(N4CCC(=O)NC4=O)cc3)CC2)n1	C39H44ClN11O4S	LCK	P06239	CRBN	WO-2023096995-A1
TPD-OWWJWQ	SCHEMBL25217093	N-(2-chloro-6-methylphenyl)-2-[[6-[4-[3-[[2-[4-(2,6-dioxopiperidin-3-yl)-2-(trifluoromethyl)phenoxy]acetyl]amino]propyl]piperazin-1-yl]-2-methylpyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide; SCHEMBL30428984	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCNC(=O)COc3ccc(C4CCC(=O)NC4=O)cc3C(F)(F)F)CC2)n1	C37H39ClF3N9O5S	LCK	P06239	CRBN	WO-2023096995-A1
TPD-RPQUQC	SCHEMBL25235908	N-(2-chloro-6-methylphenyl)-2-[[6-[4-[3-[[2-[4-(2,6-dioxopiperidin-3-yl)-3-(trifluoromethyl)phenoxy]acetyl]amino]propyl]piperazin-1-yl]-2-methylpyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide; SCHEMBL30429658	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCNC(=O)COc3ccc(C4CCC(=O)NC4=O)c(C(F)(F)F)c3)CC2)n1	C37H39ClF3N9O5S	LCK	P06239	CRBN	WO-2023096995-A1
TPD-W4EEAY	SCHEMBL25233950	N-(2-chloro-6-methylphenyl)-2-[[6-[4-[3-[[2-[4-(2,6-dioxopiperidin-3-yl)-3,5-difluorophenoxy]acetyl]amino]propyl]piperazin-1-yl]-2-methylpyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide; SCHEMBL30429731	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCNC(=O)COc3cc(F)c(C4CCC(=O)NC4=O)c(F)c3)CC2)n1	C36H38ClF2N9O5S	LCK	P06239	CRBN	WO-2023096995-A1
TPD-YP1OBQ	SCHEMBL25564634	N-(2-chloro-6-methylphenyl)-2-[[6-[(1S,4S)-5-[3-[4-[4-(2,6-dioxopiperidin-3-yl)phenyl]piperazin-1-yl]propyl]-2,5-diazabicyclo[2.2.1]heptan-2-yl]-2-methylpyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2C[C@@H]3C[C@H]2CN3CCCN2CCN(c3ccc(C4CCC(=O)NC4=O)cc3)CC2)n1	C39H45ClN10O3S	LCK	P06239	CRBN	WO-2023096995-A1
TPD-V5KN1E	SCHEMBL25207555	N-(2-chloro-6-methylphenyl)-2-[[6-[4-[3-[5-[4-(2,6-dioxopiperidin-3-yl)phenyl]-2,5-diazabicyclo[2.2.1]heptan-2-yl]propyl]piperazin-1-yl]-2-methylpyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide; SCHEMBL30429527	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCN3CC4CC3CN4c3ccc(C4CCC(=O)NC4=O)cc3)CC2)n1	C39H45ClN10O3S	LCK	P06239	CRBN	WO-2023096995-A1
TPD-QVB13G	SJ43489	N-(2-Chloro-6-methylphenyl)-2-((6-(4-(4-(4-(4-(2,4-dioxotetrahydropyrimidin-1(2H)-yl)phenyl)piperazin-1-yl)-4-oxobutyl)piperazin-1-yl)-2-methylpyrimidin-4-yl)amino)thiazole-5-carboxamide; orb2813962; CHEMBL5283559; SCHEMBL25229621; SCHEMBL30429912; GLXC-26781; SJ-43489; N-(2-Chloro-6-methylphenyl)-2-((6-(4-(4-(4-(4-(2,4-dioxotetrahydropyrimidin-1(2H)-yl)phenyl)piperazin-1-yl)-4-oxobutyl)piperazin-1-yl)-2-methylpyrimidin-4-yl)amino)thiazole-5-carboxamide	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCC(=O)N3CCN(c4ccc(N5CCC(=O)NC5=O)cc4)CC3)CC2)n1	C38H44ClN11O4S	LCK	P06239	CRBN	WO-2023096995-A1
TPD-93RBJ1	SCHEMBL25207500	N-(2-chloro-6-methylphenyl)-2-[[6-[4-[3-[(1R,4R)-5-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]-2,5-diazabicyclo[2.2.1]heptan-2-yl]propyl]piperazin-1-yl]-2-methylpyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide; SCHEMBL30429709	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCN3C[C@H]4C[C@@H]3CN4c3ccc(N4CCC(=O)NC4=O)cc3)CC2)n1	C38H44ClN11O3S	LCK	P06239	CRBN	WO-2023096995-A1
TPD-RXG75T	SCHEMBL25206957	N-(2-chloro-6-methylphenyl)-2-[[2-methyl-6-[4-[3-[[2-[4-(3-methyl-2,4-dioxo-1,3-diazinan-1-yl)phenoxy]acetyl]amino]propyl]piperazin-1-yl]pyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide; SCHEMBL30429391	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCNC(=O)COc3ccc(N4CCC(=O)N(C)C4=O)cc3)CC2)n1	C36H41ClN10O5S	LCK	P06239	CRBN	WO-2023096995-A1
TPD-1KVSNH	SCHEMBL25243728	N-(2-chloro-6-methylphenyl)-2-[[6-[4-[3-[4-[[4-[4-(2,6-dioxopiperidin-3-yl)phenyl]piperazin-1-yl]methyl]piperidin-1-yl]propyl]piperazin-1-yl]-2-methylpyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide; SCHEMBL30429534	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCN3CCC(CN4CCN(c5ccc(C6CCC(=O)NC6=O)cc5)CC4)CC3)CC2)n1	C44H56ClN11O3S	LCK	P06239	CRBN	WO-2023096995-A1
TPD-F5UQ3V	SCHEMBL25211280	N-(2-chloro-6-methylphenyl)-2-[[6-[4-[3-[4-[3-(2,6-dioxopiperidin-3-yl)phenyl]piperazin-1-yl]propyl]piperazin-1-yl]-2-methylpyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide; SCHEMBL30429722	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCN3CCN(c4cccc(C5CCC(=O)NC5=O)c4)CC3)CC2)n1	C38H45ClN10O3S	LCK	P06239	CRBN	WO-2023096995-A1
TPD-GXXYEY	SCHEMBL25205383	N-(2-chloro-6-methylphenyl)-2-[[6-[4-[3-[4-[3-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperazin-1-yl]propyl]piperazin-1-yl]-2-methylpyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide; SCHEMBL30429727	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCN3CCN(c4cccc(N5CCC(=O)NC5=O)c4)CC3)CC2)n1	C37H44ClN11O3S	LCK	P06239	CRBN	WO-2023096995-A1
TPD-29V7GP	SCHEMBL25202413	N-(2-chloro-6-methylphenyl)-2-[[6-[4-[3-[5-[4-(2,6-dioxopiperidin-3-yl)phenyl]-2,5-diazabicyclo[2.2.2]octan-2-yl]propyl]piperazin-1-yl]-2-methylpyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide; SCHEMBL30429281	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCN3CC4CCC3CN4c3ccc(C4CCC(=O)NC4=O)cc3)CC2)n1	C40H47ClN10O3S	LCK	P06239	CRBN	WO-2023096995-A1
TPD-ZPST33	SCHEMBL25209157	N-(2-chloro-6-methylphenyl)-2-[[6-[4-[2-[(1R,4R)-5-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]-2,5-diazabicyclo[2.2.1]heptan-2-yl]ethyl]piperazin-1-yl]-2-methylpyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide; SCHEMBL30429569	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCN3C[C@H]4C[C@@H]3CN4c3ccc(N4CCC(=O)NC4=O)cc3)CC2)n1	C37H42ClN11O3S	LCK	P06239	CRBN	WO-2023096995-A1
TPD-COJU0A	SCHEMBL25202405	N-(2-chloro-6-methylphenyl)-2-[[6-[4-[3-[3-[4-(2,6-dioxopiperidin-3-yl)phenyl]-3,9-diazaspiro[5.5]undecan-9-yl]propyl]piperazin-1-yl]-2-methylpyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide; SCHEMBL30429935	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCN3CCC4(CC3)CCN(c3ccc(C5CCC(=O)NC5=O)cc3)CC4)CC2)n1	C43H53ClN10O3S	LCK	P06239	CRBN	WO-2023096995-A1
TPD-3QZ01W	SCHEMBL25209197	N-(2-chloro-6-methylphenyl)-2-[[6-[4-[3-[4-[4-(2,6-dioxopiperidin-3-yl)phenyl]piperidin-1-yl]propyl]piperazin-1-yl]-2-methylpyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide; SCHEMBL30430137	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCN3CCC(c4ccc(C5CCC(=O)NC5=O)cc4)CC3)CC2)n1	C39H46ClN9O3S	LCK	P06239	CRBN	WO-2023096995-A1
TPD-7RD7WC	SCHEMBL25245789	N-(2-chloro-6-methylphenyl)-2-[[6-[4-[3-[4-[[4-(2,6-dioxopiperidin-3-yl)phenyl]methyl]piperazin-1-yl]propyl]piperazin-1-yl]-2-methylpyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide; SCHEMBL30430361	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCCN3CCN(Cc4ccc(C5CCC(=O)NC5=O)cc4)CC3)CC2)n1	C39H47ClN10O3S	LCK	P06239	CRBN	WO-2023096995-A1
TPD-VG2GNZ	WO2023097031A1_1	.	CC(C)[C@H](C(=O)N1C[C@H](O)CC1C(=O)N[C@@H](C)C1=CC=C(C#N)C=C1)C1=CC(O[C@H]2C[C@@H](CN3CCC(O[C@H]4C[C@H](OC5=CC(N6C7CCC6CN(C6=C(N)N=NC(C8=C(O)C=CC=C8)=C6)C7)=CC=N5)C4)CC3)C2)=NO1	C57H69N11O8	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-6B276H	SCHEMBL25634620	(2S,4R)-1-[(2S)-2-[3-[4-[[4-[3-[4-[4-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]piperazin-1-yl]pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(2-methylpyrazol-3-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL31409047	CC(C)[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(N2CCC(CN3CCC(O[C@H]4C[C@H](OC5=CC(N6CCN(C7=C(N)N=NC(C8=C(O)C=CC=C8)=C7)CC6)=CC=N5)C4)CC3)CC2)=NO1	C59H75N13O7	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-7CHQKE	SCHEMBL21673728	(2S,4R)-1-[(2R)-2-[3-[4-[[4-[3-[4-[3-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-N-[(1S)-1-(4-cyano-2,5-difluorophenyl)ethyl]-4-hydroxypyrrolidine-2-carboxamide	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC(F)=C(C#N)C=C1F)C1=CC(N2CCC(CN3CCC(O[C@H]4C[C@H](OC5=CC(N6C7CCC6CN(C6=C(N)N=NC(C8=C(O)C=CC=C8)=C6)C7)=CC=N5)C4)CC3)CC2)=NO1	C58H70F2N12O7	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-ZBJ15A	SCHEMBL25634988	(2S,4R)-1-[(2R)-2-[3-[4-[[4-[3-[4-[3-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-N-[1-(4-cyano-3-fluorophenyl)ethyl]-4-hydroxypyrrolidine-2-carboxamide	CC(NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](C1=CC(N2CCC(CN3CCC(OC4CC(OC5=CC(N6C7CCC6CN(C6=C(N)N=NC(C8=C(O)C=CC=C8)=C6)C7)=CC=N5)C4)CC3)CC2)=NO1)C(C)C)C1=CC=C(C#N)C(F)=C1	C58H71FN12O7	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-I9E2TC	SCHEMBL25635038	(2S,4R)-1-[(2S)-2-[3-[4-[[4-[3-[4-[3-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-N-[(1S)-1-[2-amino-4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]-4-hydroxypyrrolidine-2-carboxamide	CC1=C(C2=CC(N)=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3=CC(N4CCC(CN5CCC(O[C@H]6C[C@H](OC7=CC(N8C9CCC8CN(C8=C(N)N=NC(C%10=C(O)C=CC=C%10)=C8)C9)=CC=N7)C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C61H77N13O7S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-8M7W91	WO2023097031A1_6	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCC(O[C@H]6C[C@H](N7CCC([C@@H](C)N8C=C(C9=C(N)N=NC(C%10=CC=CC=C%10O)=C9)C=N8)CC7)C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C60H78N12O6S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-9IOJW9	WO2023097031A1_7	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCC(O[C@H]6C[C@@H](N7CCC([C@@H](C)N8C=C(C9=C(N)N=NC(C%10=CC=CC=C%10O)=C9)C=N8)CC7)C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C60H78N12O6S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-8UO8W9	WO2023097031A1_8	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCC(O[C@H]6C[C@H](N7CCC([C@H](C)N8C=C(C9=C(N)N=NC(C%10=CC=CC=C%10O)=C9)C=N8)CC7)C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C60H78N12O6S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-6JOMTX	WO2023097031A1_9	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCC(OC6CC(N7CCC([C@H](C)N8C=C(C9=C(N)N=NC(C%10=CC=CC=C%10O)=C9)C=N8)CC7)C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C60H78N12O6S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-3GECMO	WO2023097031A1_10	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCC(N[C@H]6C[C@H](OC7=NC=CC(N8C9CCC8CN(C8=C(N)N=NC(C%10=C(O)C=CC=C%10)=C8)C9)=C7)C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C61H77N13O6S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-P2T5KS	WO2023097031A1_11	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCC(OC6CC(N7CCC(O)(CN8C9CC8CN(C8=C(N)N=NC(C%10=C(O)C=CC=C%10)=C8)C9)CC7)C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C61H82N12O7S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-6GUO9N	SCHEMBL21673727	(2S,4R)-1-[(2R)-2-[3-[4-[4-[[4-[3-[4-[3-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]methyl]imidazol-1-yl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(N5C=NC(CN6CCC(OC7CC(OC8=CC(N9C%10CCC9CN(C9=C(N)N=NC(C%11=C(O)C=CC=C%11)=C9)C%10)=CC=N8)C7)CC6)=C5)CC4)=NO3)C(C)C)C=C2)SC=N1	C64H78N14O7S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-6SMNSQ	SCHEMBL25631782	(2S,4R)-1-[(2S)-2-[3-[4-[1-[4-[3-[4-[3-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]cyclopropyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3=CC(N4CCC(C5(N6CCC(O[C@H]7C[C@H](OC8=CC(N9C%10CCC9CN(C9=C(N)N=NC(C%11=C(O)C=CC=C%11)=C9)C%10)=CC=N8)C7)CC6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C63H78N12O7S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-0D2NGD	SCHEMBL25626558	(2S,4R)-1-[(2R)-2-[3-[4-[[4-[3-[4-[3-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3,9-diazabicyclo[4.2.1]nonan-9-yl]pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-N-[(1S)-1-(4-cyanophenyl)ethyl]-4-hydroxypyrrolidine-2-carboxamide	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C#N)C=C1)C1=CC(N2CCC(CN3CCC(O[C@H]4C[C@H](OC5=CC(N6C7CCC6CN(C6=C(N)N=NC(C8=C(O)C=CC=C8)=C6)CC7)=CC=N5)C4)CC3)CC2)=NO1	C59H74N12O7	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-NSH27W	SCHEMBL25631790	(2S,4R)-1-[(2R)-2-[3-[4-[[4-[3-[4-[8-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3,8-diazabicyclo[3.2.1]octan-3-yl]pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-N-[(1S)-1-(4-cyanophenyl)ethyl]-4-hydroxypyrrolidine-2-carboxamide	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C#N)C=C1)C1=CC(N2CCC(CN3CCC(OC4CC(OC5=CC(N6CC7CCC(C6)N7C6=C(N)N=NC(C7=C(O)C=CC=C7)=C6)=CC=N5)C4)CC3)CC2)=NO1	C58H72N12O7	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-45AFBG	SCHEMBL21673502	(2S,4R)-1-[(2R)-2-[3-[4-[[4-[3-[4-[3-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-N-[(1S)-1-(4-cyanophenyl)ethyl]-4-hydroxypyrrolidine-2-carboxamide	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C#N)C=C1)C1=CC(N2CCC(CN3CCC(OC4CC(OC5=CC(N6C7CCC6CN(C6=C(N)N=NC(C8=C(O)C=CC=C8)=C6)C7)=CC=N5)C4)CC3)CC2)=NO1	C58H72N12O7	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-DU0YSJ	SCHEMBL25631793	(2S,4R)-1-[(2R)-2-[3-[4-[[4-[3-[4-[3-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3,6-diazabicyclo[3.1.1]heptan-6-yl]pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-N-[(1S)-1-(4-cyanophenyl)ethyl]-4-hydroxypyrrolidine-2-carboxamide	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C#N)C=C1)C1=CC(N2CCC(CN3CCC(O[C@H]4C[C@H](OC5=CC(N6C7CC6CN(C6=C(N)N=NC(C8=C(O)C=CC=C8)=C6)C7)=CC=N5)C4)CC3)CC2)=NO1	C57H70N12O7	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-Z8K8N5	SCHEMBL25635048	(2S,4R)-1-[(2S)-2-[3-[3-[[4-[3-[4-[3-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]methyl]-8-azabicyclo[3.2.1]octan-8-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3=CC(N4C5CCC4CC(CN4CCC(OC6CC(OC7=CC(N8C9CCC8CN(C8=C(N)N=NC(C%10=C(O)C=CC=C%10)=C8)C9)=CC=N7)C6)CC4)C5)=NO3)C(C)C)C=C2)SC=N1	C63H78N12O7S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-SI5W5I	SCHEMBL25631834	(2S,4R)-1-[(2R)-2-[3-[4-[[4-[2-[3-[4-[3-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]pyridin-2-yl]oxycyclobutyl]ethynyl]-4-hydroxypiperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCC(O)(C#CC6CC(OC7=CC(N8C9CCC8CN(C8=CC(C%10=C(O)C=CC=C%10)=NN=C8N)C9)=CC=N7)C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C63H76N12O7S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-6B425C	WO2023097031A1_20	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCC(OC6CC(N7CCC(C#N)(CN8C9CC8CN(C8=C(N)N=NC(C%10=C(O)C=CC=C%10)=C8)C9)CC7)C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C62H81N13O6S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-V4AMV8	SCHEMBL25635210	(2S,4R)-1-[(2R)-2-[3-[3-[[4-[3-[4-[3-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]methyl]-8-azabicyclo[3.2.1]octan-8-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4C5CCC4CC(CN4CCC(O[C@H]6C[C@@H](OC7=CC(N8C9CCC8CN(C8=C(N)N=NC(C%10=C(O)C=CC=C%10)=C8)C9)=CC=N7)C6)CC4)C5)=NO3)C(C)C)C=C2)SC=N1	C63H78N12O7S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-QAYYN7	WO2023097031A1_22	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCC(OC6CC(N7CCC(C(C)(C)N8C9CC8CN(C8=C(N)N=NC(C%10=C(O)C=CC=C%10)=C8)C9)CC7)C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C63H86N12O6S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-GEKBP4	SCHEMBL25631878	(2S,4R)-1-[(2R)-2-[3-[4-[[4-[3-[(2S)-2-[[3-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]methyl]morpholin-4-yl]cyclobutyl]oxypiperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCC(OC6CC(N7CCO[C@H](CN8C9CCC8CN(C8=C(N)N=NC(C%10=C(O)C=CC=C%10)=C8)C9)C7)C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C61H82N12O7S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-7EHRSF	SCHEMBL25626840	(2S,4R)-1-[(2R)-2-[3-[4-[[4-[3-[[4-[3-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]piperidin-1-yl]methyl]cyclobutyl]oxypiperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCC(O[C@H]6C[C@H](CN7CCC(N8C9CCC8CN(C8=C(N)N=NC(C%10=C(O)C=CC=C%10)=C8)C9)CC7)C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C62H84N12O6S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-88U1TW	SCHEMBL25626865	(2S,4R)-1-[(2R)-2-[3-[4-[[4-[3-[4-[3-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3,8-diazabicyclo[3.2.1]octane-8-carbonyl]piperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCC(OC6CC(N7CCC(C(=O)N8C9CCC8CN(C8=C(N)N=NC(C%10=C(O)C=CC=C%10)=C8)C9)CC7)C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C62H82N12O7S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-5ZFNLK	WO2023097031A1_27	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCC(OC6CC(N7CCC(F)(CN8C9CC8CN(C8=C(N)N=NC(C%10=C(O)C=CC=C%10)=C8)C9)CC7)C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C61H81FN12O6S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-XR9D6F	SCHEMBL25631927	(2S,4R)-1-[(2R)-2-[3-[4-[[4-[3-[9-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl]cyclobutyl]oxypiperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(2-methylpyrazol-3-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL31409087	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(N2CCC(CN3CCC(O[C@H]4C[C@@H](N5CCOC6(CCN(C7=C(N)N=NC(C8=CC=CC=C8O)=C7)CC6)C5)C4)CC3)CC2)=NO1	C58H78N12O7	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-YIIFSA	WO2023097031A1_29	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCC6(CC5)CC(OC5=NC(N7C8CCC7CN(C7=C(N)N=NC(C9=C(O)C=CC=C9)=C7)C8)=CC=N5)C6)CC4)=NO3)C(C)C)C=C2)SC=N1	C59H73N13O6S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-QNFHO8	SCHEMBL25634654	(2S,4R)-1-[(2R)-2-[3-[4-[[4-[3-[4-[(E)-2-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]ethenyl]pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(2-methylpyrazol-3-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL31409098	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(N2CCC(CN3CCC(OC4CC(OC5=CC(/C=C/C6=C(N)N=NC(C7=C(O)C=CC=C7)=C6)=CC=N5)C4)CC3)CC2)=NO1	C57H69N11O7	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-GMPMQQ	SCHEMBL25627183	(2S,4R)-1-[(2R)-2-[3-[4-[[4-[[2-[4-[1-[4-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]pyrazol-1-yl]ethyl]piperidin-1-yl]-7-azaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL31409021	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCC(CN6CCC7(CC6)CC(N6CCC(C(C)N8C=C(C9=C(N)N=NC(C%10=C(O)C=CC=C%10)=C9)C=N8)CC6)C7)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C65H87N13O5S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-AP7RHE	WO2023097031A1_32	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCC6(CC5)CC(CN5CCC(OC7=NC=CC(N8C9CCC8CN(C8=C(N)N=NC(C%10=C(O)C=CC=C%10)=C8)C9)=C7)CC5)C6)CC4)=NO3)C(C)C)C=C2)SC=N1	C66H85N13O6S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-LFYMNF	SCHEMBL25627695	(2S,4R)-1-[(2R)-2-[3-[4-[[4-[[2-[4-[3-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]pyridin-2-yl]oxy-7-azaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(2-methylpyrazol-3-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL31409008	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(N2CCC(CN3CCC(CN4CCC5(CC4)CC(OC4=CC(N6C7CCC6CN(C6=C(N)N=NC(C8=C(O)C=CC=C8)=C6)C7)=CC=N4)C5)CC3)CC2)=NO1	C66H86N14O6	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-ZUKNF3	SCHEMBL25631979	(2S,4R)-1-[2-[3-[3-[5-[3-[4-[4-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]piperazin-1-yl]pyridin-2-yl]oxycyclobutyl]oxypyrimidin-2-yl]prop-2-ynoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(2-methylpyrazol-3-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL31409116	CC(C)C(C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCC#CC2=NC=C(O[C@H]3C[C@H](OC4=CC(N5CCN(C6=CC(C7=C(O)C=CC=C7)=NN=C6N)CC5)=CC=N4)C3)C=N2)=NO1	C55H59N13O8	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-JDJ0S8	SCHEMBL25627345	(2S,4R)-1-[(2R)-2-[3-[4-[[2-[(2S)-2-[[3-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]methyl]morpholin-4-yl]-7-azaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL31408979	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCC6(CC5)CC(N5CCO[C@H](CN7C8CCC7CN(C7=C(N)N=NC(C9=CC=CC=C9O)=C7)C8)C5)C6)CC4)=NO3)C(C)C)C=C2)SC=N1	C60H80N12O6S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-B6K6O4	SCHEMBL25632027	(2S,4R)-1-[(2R)-2-[3-[4-[[2-[3-[4-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]pyrazol-1-yl]but-1-ynyl]-7-azaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL31408962	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCC6(CC5)CC(C#CC(C)N5C=C(C7=C(N)N=NC(C8=C(O)C=CC=C8)=C7)C=N5)C6)CC4)=NO3)C(C)C)C=C2)SC=N1	C56H67N11O5S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-0LTWMZ	SCHEMBL25632028	(2S,4R)-N-[(1S)-3-[4-[[4-[3-[4-[3-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]methyl]piperidin-1-yl]-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]-3-oxopropyl]-4-hydroxy-1-[(2R)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CC(=O)N3CCC(CN4CCC(OC5CC(OC6=CC(N7C8CCC7CN(C7=C(N)N=NC(C9=C(O)C=CC=C9)=C7)C8)=CC=N6)C5)CC4)CC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C=C2)SC=N1	C67H80N12O8S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-2N6N0Q	SCHEMBL25635275	(2S,4R)-N-[(1S)-3-[4-[[4-[3-[4-[3-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]methyl]piperidin-1-yl]-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]-3-oxopropyl]-4-hydroxy-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CC(=O)N3CCC(CN4CCC(OC5CC(OC6=CC(N7C8CCC7CN(C7=C(N)N=NC(C9=C(O)C=CC=C9)=C7)C8)=CC=N6)C5)CC4)CC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC=C4)C3=O)C=C2)SC=N1	C67H80N12O8S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-PV880P	SCHEMBL25627807	(2S,4R)-1-[(2R)-2-[3-[4-[[4-[3-[4-[4-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]piperazin-1-yl]pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-N-[(1S)-1-[4-(4-fluoro-2-methylpyrazol-3-yl)phenyl]ethyl]-4-hydroxypyrrolidine-2-carboxamide; SCHEMBL31408976	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=C(F)C=NN2C)C=C1)C1=CC(N2CCC(CN3CCC(O[C@H]4C[C@H](OC5=CC(N6CCN(C7=C(N)N=NC(C8=C(O)C=CC=C8)=C7)CC6)=CC=N5)C4)CC3)CC2)=NO1	C59H74FN13O7	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-0CXJZO	SCHEMBL25632082	(2S,4R)-1-[(2R)-2-[3-[4-[[4-[4-[4-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]piperazin-1-yl]pyridin-2-yl]oxypiperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(2-methylpyrazol-3-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(N2CCC(CN3CCC(OC4=CC(N5CCN(C6=CC(C7=C(O)C=CC=C7)=NN=C6N)CC5)=CC=N4)CC3)CC2)=NO1	C55H69N13O6	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-6SL8QF	WO2023097031A1_42	.	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(N2CCC(CN3CCC(OC4CC(N5CCC(C(C)N6C=NC(C#CC7=CC(C8=CC=CC=C8O)=NN=C7N)=C6)CC5)C4)CC3)CC2)=NO1	C62H79N13O6	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-9PUK7K	SCHEMBL25628143	(2S,4R)-1-[(2R)-2-[3-[4-[[4-[2-[4-[3-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]pyridin-2-yl]oxy-7-azaspiro[3.5]nonan-7-yl]piperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL31409002	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCC(N6CCC7(CC6)CC(OC6=CC(N8C9CCC8CN(C8=C(N)N=NC(C%10=C(O)C=CC=C%10)=C8)C9)=CC=N6)C7)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C65H83N13O6S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-S9HMIL	SCHEMBL25628239	(2S,4R)-1-[(2R)-2-[3-[4-[[4-[3-[2-[3-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]-7-azaspiro[3.5]nonan-7-yl]cyclobutyl]oxypiperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCC(OC6CC(N7CCC8(CC7)CC(N7C9CCC7CN(C7=C(N)N=NC(C%10=C(O)C=CC=C%10)=C7)C9)C8)C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C64H86N12O6S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-GZUK0T	SCHEMBL25628284	[3-[1-[[1-[5-[(2R)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]-1,2-oxazol-3-yl]piperidin-4-yl]methyl]piperidin-4-yl]oxycyclobutyl] 4-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]piperazine-1-carboxylate; SCHEMBL31409082	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCC(O[C@H]6C[C@H](OC(=O)N7CCN(C8=C(N)N=NC(C9=C(O)C=CC=C9)=C8)CC7)C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C55H71N11O8S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-LEZQ96	WO2023097031A1_46	.	CC(C)[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(Cl)C=C1)C1=CC(N2CCC(CN3CCC(OC4CC(OC5=CC(N6C7CCC6CN(C6=C(N)N=NC(C8=C(O)C=CC=C8)=C6)C7)=CC=N5)C4)CC3)CC2)=NO1	C57H72ClN11O7	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-7C6YWH	WO2023097031A1_47	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCC(OC6CC(N7CCN(CC8C9CC8CN(C8=C(N)N=NC(C%10=C(O)C=CC=C%10)=C8)C9)CC7)C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C61H82N12O6S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-3RA0SV	SCHEMBL25632119	(2S,4R)-1-[(2R)-2-[3-[4-[[4-[3-[4-[3-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-N-[(1S)-1-(4-chlorophenyl)ethyl]-4-hydroxypyrrolidine-2-carboxamide	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(Cl)C=C1)C1=CC(N2CCC(CN3CCC(OC4CC(OC5=NC=CC(N6C7CCC6CN(C6=C(N)N=NC(C8=C(O)C=CC=C8)=C6)C7)=C5)C4)CC3)CC2)=NO1	C57H72ClN11O7	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-CNUN15	SCHEMBL25628458	(2S,4R)-1-[(2R)-2-[3-[4-[[(3S,4R)-4-[4-[3-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]pyridin-2-yl]oxy-3-fluoropiperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL31408986	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CC[C@@H](OC6=CC(N7C8CCC7CN(C7=C(N)N=NC(C9=C(O)C=CC=C9)=C7)C8)=CC=N6)[C@@H](F)C5)CC4)=NO3)C(C)C)C=C2)SC=N1	C57H69FN12O6S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-SI3CI4	SCHEMBL25632177	(2S,4R)-1-[(2R)-2-[3-[4-[[(3R,4S)-4-[4-[3-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]pyridin-2-yl]oxy-3-fluoropiperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL31408996	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CC[C@H](OC6=CC(N7C8CCC7CN(C7=C(N)N=NC(C9=C(O)C=CC=C9)=C7)C8)=CC=N6)[C@H](F)C5)CC4)=NO3)C(C)C)C=C2)SC=N1	C57H69FN12O6S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-7KKO3P	WO2023097031A1_51	.	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(N2CCC(CN3CCC(O[C@H]4C[C@H](OC5=CC(/C=C(\F)C6=C(N)N=NC(C7=C(O)C=CC=C7)=C6)=CC=N5)C4)CC3)CC2)=NO1	C57H68FN11O7	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-60YR05	SCHEMBL25632179	(2S,4R)-1-[(2R)-2-[3-[4-[[4-[4-[(Z)-2-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-2-fluoroethenyl]pyridin-2-yl]oxypiperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(2-methylpyrazol-3-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(N2CCC(CN3CCC(OC4=CC(/C=C(\F)C5=C(N)N=NC(C6=C(O)C=CC=C6)=C5)=CC=N4)CC3)CC2)=NO1	C53H62FN11O6	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-8HEQWI	WO2023097031A1_53	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CC[C@@H](OC6=NC(N7C8CCC7CN(C7=C(N)N=NC(C9=C(O)C=CC=C9)=C7)C8)=CC=N6)C(F)(F)C5)CC4)=NO3)C(C)C)C=C2)SC=N1	C56H67F2N13O6S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-HMUNZ0	WO2023097031A1_54	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CC[C@H](OC6=NC(N7C8CCC7CN(C7=C(N)N=NC(C9=C(O)C=CC=C9)=C7)C8)=CC=N6)C(F)(F)C5)CC4)=NO3)C(C)C)C=C2)SC=N1	C56H67F2N13O6S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-HLDS2R	SCHEMBL25632226	(2S,4R)-1-[(2R)-2-[3-[4-[[4-[3-[9-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-2,2-difluoro-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl]cyclobutyl]oxypiperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL31408972	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCC(O[C@H]6C[C@@H](N7CC(F)(F)OC8(CCN(C9=C(N)N=NC(C%10=CC=CC=C%10O)=C9)CC8)C7)C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C58H75F2N11O7S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-3MMO6M	SCHEMBL25628556	(2S,4R)-1-[(2R)-2-[3-[4-[1-[[3-[9-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl]cyclobutyl]methyl]piperidin-4-yl]oxypiperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL31408987	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(OC5CCN(CC6CC(N7CCOC8(CCN(C9=C(N)N=NC(C%10=C(O)C=CC=C%10)=C9)CC8)C7)C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C58H77N11O7S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-CX8YHS	SCHEMBL25628609	(2S,4R)-1-[(2R)-2-[3-[4-[[4-[3-[4-[[1-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-4-hydroxypiperidin-4-yl]methyl]piperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL31409054	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCC(OC6CC(N7CCN(CC8(O)CCN(C9=C(N)N=NC(C%10=C(O)C=CC=C%10)=C9)CC8)CC7)C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C60H82N12O7S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-FELIUL	SCHEMBL25632233	(2S,4R)-1-[(2R)-2-[3-[4-[[2-[4-[3-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3,8-diazabicyclo[3.2.1]octane-8-carbonyl]piperidin-1-yl]-7-azaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL31409016	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCC6(CC5)CC(N5CCC(C(=O)N7C8CCC7CN(C7=C(N)N=NC(C9=C(O)C=CC=C9)=C7)C8)CC5)C6)CC4)=NO3)C(C)C)C=C2)SC=N1	C61H80N12O6S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-NBM2XO	SCHEMBL25632290	(2S,4R)-1-[(2R)-2-[3-[4-[[(3R,4R)-4-[4-[3-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]pyridin-2-yl]oxy-3-fluoropiperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL31409038	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CC[C@@H](OC6=CC(N7C8CCC7CN(C7=C(N)N=NC(C9=C(O)C=CC=C9)=C7)C8)=CC=N6)[C@H](F)C5)CC4)=NO3)C(C)C)C=C2)SC=N1	C57H69FN12O6S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-IAS91E	SCHEMBL25632291	(2S,4R)-1-[(2R)-2-[3-[4-[[(3S,4S)-4-[4-[3-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]pyridin-2-yl]oxy-3-fluoropiperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL31409006	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CC[C@H](OC6=CC(N7C8CCC7CN(C7=C(N)N=NC(C9=C(O)C=CC=C9)=C7)C8)=CC=N6)[C@@H](F)C5)CC4)=NO3)C(C)C)C=C2)SC=N1	C57H69FN12O6S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-9GFGOZ	SCHEMBL25632362	(2S,4R)-1-[(2R)-2-[3-[4-[[2-[(3S)-3-[[3-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]methyl]-3-hydroxypiperidin-1-yl]-7-azaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL31409059	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCC6(CC5)CC(N5CCC[C@@](O)(CN7C8CCC7CN(C7=C(N)N=NC(C9=C(O)C=CC=C9)=C7)C8)C5)C6)CC4)=NO3)C(C)C)C=C2)SC=N1	C61H82N12O6S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-8QRKFL	SCHEMBL25628730	(2S,4R)-1-[(2R)-2-[3-[4-[[2-[(2R)-2-[3-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3,8-diazabicyclo[3.2.1]octane-8-carbonyl]morpholin-4-yl]-7-azaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL31409049	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCC6(CC5)CC(N5CCO[C@@H](C(=O)N7C8CCC7CN(C7=C(N)N=NC(C9=C(O)C=CC=C9)=C7)C8)C5)C6)CC4)=NO3)C(C)C)C=C2)SC=N1	C60H78N12O7S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-OW8JHZ	SCHEMBL25628789	(2S,4R)-1-[(2R)-2-[3-[4-[[2-[4-[2-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]ethynyl]pyrazol-1-yl]-7-azaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL31409010	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCC6(CC5)CC(N5C=C(C#CC7=CC(C8=CC=CC=C8O)=NN=C7N)C=N5)C6)CC4)=NO3)C(C)C)C=C2)SC=N1	C54H63N11O5S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-AIR1IY	SCHEMBL25628898	[1-[2-[[5-[(2R)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]-1,2-oxazol-3-yl]oxy]ethyl]piperidin-4-yl] 4-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]piperazine-1-carboxylate; SCHEMBL31409083	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(OCCN4CCC(OC(=O)N5CCN(C6=C(N)N=NC(C7=C(O)C=CC=C7)=C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C47H58N10O8S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-53R9N7	SCHEMBL25628955	[1-[[1-[5-[(2R)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]-1,2-oxazol-3-yl]piperidin-4-yl]methyl]piperidin-4-yl] 4-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]piperazine-1-carboxylate; SCHEMBL31409084	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCC(OC(=O)N6CCN(C7=C(N)N=NC(C8=C(O)C=CC=C8)=C7)CC6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C51H65N11O7S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-ABBCY4	SCHEMBL25632328	(2S,4R)-1-[(2R)-2-[3-[2-[4-[2-[4-[3-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]pyridin-2-yl]oxyethyl]piperazin-1-yl]ethoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-N-[(1S)-1-(4-cyanophenyl)ethyl]-4-hydroxypyrrolidine-2-carboxamide; SCHEMBL31409108	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C#N)C=C1)C1=CC(OCCN2CCN(CCOC3=CC(N4C5CCC4CN(C4=C(N)N=NC(C6=C(O)C=CC=C6)=C4)C5)=CC=N3)CC2)=NO1	C51H62N12O7	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-IKTC4Z	SCHEMBL25632329	(2S,4R)-1-[(2S)-2-[3-[3-[[4-[3-[9-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl]cyclobutyl]oxypiperidin-1-yl]methyl]cyclobutyl]oxy-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL31409075	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3=CC(OC4CC(CN5CCC(O[C@H]6C[C@H](N7CCOC8(CCN(C9=C(N)N=NC(C%10=C(O)C=CC=C%10)=C9)CC8)C7)C6)CC5)C4)=NO3)C(C)C)C=C2)SC=N1	C57H74N10O8S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-NVIB93	SCHEMBL25629205	(2S,4R)-1-[(2R)-2-[3-[3-[[4-[3-[9-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl]cyclobutyl]oxypiperidin-1-yl]methyl]cyclobutyl]oxy-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL31409020	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(OC4CC(CN5CCC(O[C@H]6C[C@H](N7CCOC8(CCN(C9=C(N)N=NC(C%10=C(O)C=CC=C%10)=C9)CC8)C7)C6)CC5)C4)=NO3)C(C)C)C=C2)SC=N1	C57H74N10O8S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-IAHFPP	SCHEMBL25629280	(2S,4R)-1-[(2R)-2-[3-[4-[[4-[3-[4-[1-[4-[(E)-2-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]ethenyl]pyrazol-1-yl]ethyl]piperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCC(OC6CC(N7CCC(C(C)N8C=C(/C=C/C9=CC(C%10=CC=CC=C%10O)=NN=C9N)C=N8)CC7)C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C62H80N12O6S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-YTKW85	WO2023097031A1_70	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCC6(CC5)CC(N5CCC[C@H](CN7CC8CC7CN8C7=C(N)N=NC(C8=C(O)C=CC=C8)=C7)C5)C6)CC4)=NO3)C(C)C)C=C2)SC=N1	C60H80N12O5S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-0W744A	SCHEMBL25628696	(2S,4R)-1-[(2R)-2-[3-[4-[[2-[(3R)-3-[[3-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]methyl]-3-hydroxypiperidin-1-yl]-7-azaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL31409009	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCC6(CC5)CC(N5CCC[C@](O)(CN7C8CCC7CN(C7=C(N)N=NC(C9=C(O)C=CC=C9)=C7)C8)C5)C6)CC4)=NO3)C(C)C)C=C2)SC=N1	C61H82N12O6S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-9EDE2M	SCHEMBL25632363	(2S,4R)-N-[(1S)-1-[4-[4-[3-[2-[2-[2-[4-[3-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]pyridin-2-yl]oxyethoxy]ethoxy]ethoxy]prop-1-ynyl]-1,3-thiazol-5-yl]phenyl]ethyl]-4-hydroxy-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]pyrrolidine-2-carboxamide; SCHEMBL31409128	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=C(C#CCOCCOCCOCCOC3=CC(N4C5CCC4CN(C4=C(N)N=NC(C6=CC=CC=C6O)=C4)C5)=CC=N3)N=CS2)C=C1)N1CC2=C(C=CC=C2)C1=O	C59H66N10O9S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-VE8G6S	SCHEMBL25632366	(2S,4R)-1-[(2R)-2-[3-[4-[[2-[(2R,6R)-2-[[3-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]methyl]-6-methylmorpholin-4-yl]-7-azaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL31408967	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCC6(CC5)CC(N5C[C@H](CN7C8CCC7CN(C7=C(N)N=NC(C9=C(O)C=CC=C9)=C7)C8)O[C@H](C)C5)C6)CC4)=NO3)C(C)C)C=C2)SC=N1	C61H82N12O6S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-C7M8FD	SCHEMBL25629422	(2S,4R)-1-[(2R)-2-[3-[4-[[4-[3-[4-[(1R)-1-[1-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]pyrazol-4-yl]ethyl]piperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL31408982	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCC(OC6CC(N7CCC([C@@H](C)C8=CN(C9=C(N)N=NC(C%10=CC=CC=C%10O)=C9)N=C8)CC7)C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C60H78N12O6S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-WFR1JV	SCHEMBL25634770	(2S,4R)-1-[(2R)-2-[3-[4-[[4-[3-[4-[(1S)-1-[1-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]pyrazol-4-yl]ethyl]piperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL31409026	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCC(OC6CC(N7CCC([C@H](C)C8=CN(C9=C(N)N=NC(C%10=CC=CC=C%10O)=C9)N=C8)CC7)C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C60H78N12O6S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-1E2LLY	SCHEMBL25629503	(2S,4R)-1-[(2R)-2-[3-[4-[[4-[3-[4-[3-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]piperidine-1-carbonyl]cyclobutyl]oxypiperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCC(O[C@H]6C[C@H](C(=O)N7CCC(N8C9CCC8CN(C8=C(N)N=NC(C%10=C(O)C=CC=C%10)=C8)C9)CC7)C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C62H82N12O7S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-NTMV3M	WO2023097031A1_77	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCC(OC6CC(N7CCC(O[C@H]8CCN(C9=C(N)N=NC(C%10=CC=CC=C%10O)=C9)C8)CC7)C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C59H79N11O7S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-CAAR99	WO2023097031A1_78	.	CC(C)[C@@H](C(=O)N1C[C@H](O)CC1C(=O)N[C@@H](C)C1=CC=C(C#N)C=C1)C1=CC(N2CCC(CN3CCC(OC4CC(N5CCC(C(C)N6C=C(C#CC7=CC(C8=CC=CC=C8O)=NN=C7N)C=N6)CC5)C4)CC3)CC2)=NO1	C59H74N12O6	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-CRDALY	SCHEMBL25632431	(2S,4R)-1-[(2S)-2-[3-[4-[4-[4-[3-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]pyridin-2-yl]oxycyclohexyl]oxypiperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL25632769	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3=CC(N4CCC(O[C@H]5CC[C@@H](OC6=CC(N7C8CCC7CN(C7=C(N)N=NC(C9=C(O)C=CC=C9)=C7)C8)=CC=N6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C57H69N11O7S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-R46LA3	SCHEMBL25629620	(2S,4R)-1-[(2R)-2-[3-[4-[4-[4-[3-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]pyridin-2-yl]oxycyclohexyl]oxypiperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL25632770	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(OC5CCC(OC6=CC(N7C8CCC7CN(C7=C(N)N=NC(C9=C(O)C=CC=C9)=C7)C8)=CC=N6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C57H69N11O7S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-C1ADGQ	SCHEMBL25628352	[3-[1-[2-[[5-[(2R)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]-1,2-oxazol-3-yl]oxy]ethyl]piperidin-4-yl]oxycyclobutyl] 4-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]piperazine-1-carboxylate; SCHEMBL31409092	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(OCCN4CCC(O[C@H]5C[C@H](OC(=O)N6CCN(C7=C(N)N=NC(C8=C(O)C=CC=C8)=C7)CC6)C5)CC4)=NO3)C(C)C)C=C2)SC=N1	C51H64N10O9S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-GH5YLB	WO2023097031A1_82	.	CC(C)[C@@H](C(=O)N1C[C@H](O)CC1C(=O)N[C@@H](C)C1=CC=C(C2=C(C#CCOCCOCCOCCOCCOC3=CC(N4C5CCC4CN(C4=CC(C6=C(O)C=CC=C6)=NN=C4N)C5)=CC=N3)N=CS2)C=C1)N1CC2=C(C=CC=C2)C1=O	C61H70N10O10S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-0VV4SQ	SCHEMBL25632456	(2S,4R)-N-[(1S)-1-[4-[4-[3-[2-[2-[2-[2-[4-[3-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]pyridin-2-yl]oxyethoxy]ethoxy]ethoxy]ethoxy]prop-1-ynyl]-1,3-thiazol-5-yl]phenyl]ethyl]-4-hydroxy-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]pyrrolidine-2-carboxamide; SCHEMBL31409048	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=C(C#CCOCCOCCOCCOCCOC3=CC(N4C5CCC4CN(C4=CC(C6=C(O)C=CC=C6)=NN=C4N)C5)=CC=N3)N=CS2)C=C1)N1CC2=C(C=CC=C2)C1=O	C61H70N10O10S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-QTD8Y2	WO2023097031A1_84	.	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(N2CCC(CN3CCC(OC4CC(N5CCC(C(C)N6N=CC(C#CC7=CC(C8=CC=CC=C8O)=NN=C7N)=C6F)CC5)C4)CC3)CC2)=NO1	C62H78FN13O6	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-1BTVXI	SCHEMBL25629737	(2S,4R)-1-[(2R)-2-[3-[4-[[4-[3-[4-[1-[1-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]imidazol-4-yl]ethyl]piperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL25632457	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCC(O[C@H]6C[C@@H](N7CCC(C(C)C8=CN(C9=C(N)N=NC(C%10=CC=CC=C%10O)=C9)C=N8)CC7)C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C60H78N12O6S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-I0V819	SCHEMBL25632462	(2S,4R)-N-[(1S)-1-[4-[4-[3-[2-[2-[4-[3-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]pyridin-2-yl]oxyethoxy]ethoxy]prop-1-ynyl]-1,3-thiazol-5-yl]phenyl]ethyl]-4-hydroxy-1-[(2R)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]pyrrolidine-2-carboxamide; SCHEMBL31409029	CC(C)[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=C(C#CCOCCOCCOC3=CC(N4C5CCC4CN(C4=CC(C6=C(O)C=CC=C6)=NN=C4N)C5)=CC=N3)N=CS2)C=C1)N1CC2=C(C=CC=C2)C1=O	C57H62N10O8S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-BWCILW	SCHEMBL25629824	(2S,4R)-N-[(1S)-1-[4-[4-[3-[2-[2-[4-[3-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]pyridin-2-yl]oxyethoxy]ethoxy]prop-1-ynyl]-1,3-thiazol-5-yl]phenyl]ethyl]-4-hydroxy-1-[(2S)-3-methyl-2-(3-oxo-1H-isoindol-2-yl)butanoyl]pyrrolidine-2-carboxamide; SCHEMBL31408980	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=C(C#CCOCCOCCOC3=CC(N4C5CCC4CN(C4=CC(C6=C(O)C=CC=C6)=NN=C4N)C5)=CC=N3)N=CS2)C=C1)N1CC2=C(C=CC=C2)C1=O	C57H62N10O8S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-7I7AB1	SCHEMBL25632483	(2S,4R)-1-[(2R)-2-[3-[4-[[2-[(2S)-2-[1-[4-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]pyrazol-1-yl]ethyl]morpholin-4-yl]-7-azaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL31409019	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCC6(CC5)CC(N5CCO[C@H](C(C)N7C=C(C8=C(N)N=NC(C9=CC=CC=C9O)=C8)C=N7)C5)C6)CC4)=NO3)C(C)C)C=C2)SC=N1	C58H74N12O6S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-GB07OC	SCHEMBL25632485	(2S,4R)-1-[(2R)-2-[3-[4-[[2-[(2R)-2-[1-[4-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]pyrazol-1-yl]ethyl]morpholin-4-yl]-7-azaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL31409079	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCC6(CC5)CC(N5CCO[C@@H](C(C)N7C=C(C8=C(N)N=NC(C9=CC=CC=C9O)=C8)C=N7)C5)C6)CC4)=NO3)C(C)C)C=C2)SC=N1	C58H74N12O6S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-K2LLGQ	WO2023097031A1_90	.	CC1=NC=CN1C1=CC=C([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](C2=CC(N3CCC(CN4CCC(OC5CC(N6CCC(C(C)N7C=C(C#CC8=CC(C9=CC=CC=C9O)=NN=C8N)N=N7)CC6)C5)CC4)CC3)=NO2)C(C)C)C=C1	C61H78N14O6	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-XMDLJP	WO2023097031A1_91	.	CC1=NC=CN1C1=CC=C([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](C2=CC(N3CCC(CN4CCC(OC5CC(N6CCC(C(C)N7C=NC(C#CC8=CC(C9=CC=CC=C9O)=NN=C8N)=C7)CC6)C5)CC4)CC3)=NO2)C(C)C)C=C1	C62H79N13O6	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-7W5L3J	SCHEMBL25634792	(2S,4R)-1-[(2R)-2-[3-[4-[[4-[(2R)-2-[[3-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]methyl]morpholin-4-yl]piperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL31408994	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCC(N6CCO[C@@H](CN7C8CCC7CN(C7=C(N)N=NC(C9=C(O)C=CC=C9)=C7)C8)C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C57H76N12O6S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-6PDMRU	SCHEMBL25635516	(2S,4R)-1-[(2S)-2-[3-[3-[2-[4-[3-[4-[3-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]pyridin-2-yl]oxycyclobutyl]oxypiperidin-1-yl]propan-2-yl]cyclobutyl]oxy-1,2-oxazol-5-yl]-3-methylbutanoyl]-N-[(1S)-1-(4-cyanophenyl)ethyl]-4-hydroxypyrrolidine-2-carboxamide	CC(C)[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C#N)C=C1)C1=CC(O[C@H]2C[C@H](C(C)(C)N3CCC(O[C@H]4C[C@@H](OC5=CC(N6C7CCC6CN(C6=C(N)N=NC(C8=C(O)C=CC=C8)=C6)C7)=CC=N5)C4)CC3)C2)=NO1	C59H73N11O8	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-OBM1CJ	WO2023097031A1_94	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCC6(CC5)CC(N5CCO[C@H](C(C)(C)N7C8CC7CN(C7=C(N)N=NC(C9=C(O)C=CC=C9)=C7)C8)C5)C6)CC4)=NO3)C(C)C)C=C2)SC=N1	C61H82N12O6S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-EA22J0	WO2023097031A1_95	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCC6(CC5)CC(N5CCO[C@@H](C(C)(C)N7C8CC7CN(C7=C(N)N=NC(C9=C(O)C=CC=C9)=C7)C8)C5)C6)CC4)=NO3)C(C)C)C=C2)SC=N1	C61H82N12O6S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-IDSVVU	SCHEMBL25630101	(2S,4R)-1-[(2R)-2-[3-[4-[[2-[(2S)-2-[(1S)-1-[4-[2-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]ethynyl]pyrazol-1-yl]ethyl]morpholin-4-yl]-7-azaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL31409031	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCC6(CC5)CC(N5CCO[C@H]([C@H](C)N7C=C(C#CC8=CC(C9=CC=CC=C9O)=NN=C8N)C=N7)C5)C6)CC4)=NO3)C(C)C)C=C2)SC=N1	C60H74N12O6S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-FDT2J8	SCHEMBL25632532	(2S,4R)-1-[(2R)-2-[3-[4-[[2-[(2R)-2-[(1S)-1-[4-[2-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]ethynyl]pyrazol-1-yl]ethyl]morpholin-4-yl]-7-azaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL31409065	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCC6(CC5)CC(N5CCO[C@@H]([C@H](C)N7C=C(C#CC8=CC(C9=CC=CC=C9O)=NN=C8N)C=N7)C5)C6)CC4)=NO3)C(C)C)C=C2)SC=N1	C60H74N12O6S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-KW7XSH	SCHEMBL25632535	(2S,4R)-1-[(2R)-2-[3-[4-[[2-[(2R)-2-[(1R)-1-[4-[2-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]ethynyl]pyrazol-1-yl]ethyl]morpholin-4-yl]-7-azaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL31408963	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCC6(CC5)CC(N5CCO[C@@H]([C@@H](C)N7C=C(C#CC8=CC(C9=CC=CC=C9O)=NN=C8N)C=N7)C5)C6)CC4)=NO3)C(C)C)C=C2)SC=N1	C60H74N12O6S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-H3BSTJ	WO2023097031A1_100	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCC(OC6CC(N7CCC(C(C)N8N=CC(C9=C(N)N=NC(C%10=CC=CC=C%10O)=C9)=C8F)CC7)C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C60H77FN12O6S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-Y2IWSB	SCHEMBL25630128	[(3S,4R)-3-fluoro-1-[[1-[5-[(2R)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]-1,2-oxazol-3-yl]piperidin-4-yl]methyl]piperidin-4-yl] 4-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]piperazine-1-carboxylate; SCHEMBL31409096	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CC[C@@H](OC(=O)N6CCN(C7=C(N)N=NC(C8=C(O)C=CC=C8)=C7)CC6)[C@@H](F)C5)CC4)=NO3)C(C)C)C=C2)SC=N1	C51H64FN11O7S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-N6UOT7	SCHEMBL25632559	[(3R,4R)-3-fluoro-1-[[1-[5-[(2R)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]-1,2-oxazol-3-yl]piperidin-4-yl]methyl]piperidin-4-yl] 4-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]piperazine-1-carboxylate; SCHEMBL31409044	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CC[C@@H](OC(=O)N6CCN(C7=C(N)N=NC(C8=C(O)C=CC=C8)=C7)CC6)[C@H](F)C5)CC4)=NO3)C(C)C)C=C2)SC=N1	C51H64FN11O7S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-144VFG	SCHEMBL25632560	[(3R,4S)-3-fluoro-1-[[1-[5-[(2R)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]-1,2-oxazol-3-yl]piperidin-4-yl]methyl]piperidin-4-yl] 4-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]piperazine-1-carboxylate; SCHEMBL31409034	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CC[C@H](OC(=O)N6CCN(C7=C(N)N=NC(C8=C(O)C=CC=C8)=C7)CC6)[C@H](F)C5)CC4)=NO3)C(C)C)C=C2)SC=N1	C51H64FN11O7S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-12VB7D	SCHEMBL25632561	[(3S,4S)-3-fluoro-1-[[1-[5-[(2R)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]-1,2-oxazol-3-yl]piperidin-4-yl]methyl]piperidin-4-yl] 4-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]piperazine-1-carboxylate; SCHEMBL31409035	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CC[C@H](OC(=O)N6CCN(C7=C(N)N=NC(C8=C(O)C=CC=C8)=C7)CC6)[C@@H](F)C5)CC4)=NO3)C(C)C)C=C2)SC=N1	C51H64FN11O7S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-Q5RGQK	SCHEMBL25630183	(2S,4R)-1-[(2R)-2-[3-[4-[[4-[3-[4-[[1-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]pyrazol-4-yl]methyl]piperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL31408990	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCC(OC6CC(N7CCC(CC8=CN(C9=C(N)N=NC(C%10=CC=CC=C%10O)=C9)N=C8)CC7)C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C59H76N12O6S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-KEQQSZ	WO2023097031A1_106	.	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(N2CCC(CN3CCC4(CC3)CC(N3CCO[C@H](CN5C6CCC5CN(C5=C(N)N=NC(C7=CC=CC=C7O)=C5)C6)C3)C4)CC2)=NO1	C60H81N13O6	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-TZHY29	WO2023097031A1_107	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCN(C(=O)[C@H]5C[C@H](OC6=NC=CC(N7C8CCC7CN(C7=C(N)N=NC(C9=C(O)C=CC=C9)=C7)C8)=C6)C5)CC4)=NO3)C(C)C)C=C2)SC=N1	C55H64N12O7S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-SO808H	SCHEMBL25632600	(2S,4R)-1-[(2R)-2-[3-[4-[1-[[3-[(2R)-2-[[3-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]methyl]morpholin-4-yl]cyclobutyl]methyl]piperidin-4-yl]oxypiperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(OC5CCN(CC6CC(N7CCO[C@@H](CN8C9CCC8CN(C8=C(N)N=NC(C%10=C(O)C=CC=C%10)=C8)C9)C7)C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C61H82N12O7S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-WTDW5K	WO2023097031A1_109	.	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(N2CCC(OC3CCN(CC4CC(N5CCC([C@H](C)N6C=C(C#CC7=CC(C8=CC=CC=C8O)=NN=C7N)N=N6)CC5)C4)CC3)CC2)=NO1	C61H78N14O6	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-SXG1M1	SCHEMBL25630552	(2S,4R)-1-[(2R)-2-[3-[4-[1-[[3-[4-[(1R)-1-[4-[2-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]ethynyl]pyrazol-1-yl]ethyl]piperidin-1-yl]cyclobutyl]methyl]piperidin-4-yl]oxypiperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(2-methylpyrazol-3-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL31409076	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(N2CCC(OC3CCN(CC4CC(N5CCC([C@@H](C)N6C=C(C#CC7=CC(C8=CC=CC=C8O)=NN=C7N)C=N6)CC5)C4)CC3)CC2)=NO1	C62H79N13O6	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-HZ6XGN	WO2023097031A1_111	.	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(N2CCC(OC3CCN(CC4CC(N5CCC([C@H](C)N6C=C(C#CC7=CC(C8=CC=CC=C8O)=NN=C7N)C=N6)CC5)C4)CC3)CC2)=NO1	C62H79N13O6	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-ANX3PW	SCHEMBL25632627	(2S,4R)-1-[(2R)-2-[3-[4-[[2-[(2S)-2-[[[1-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]piperidin-4-yl]amino]methyl]morpholin-4-yl]-7-azaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL31409046	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCC6(CC5)CC(N5CCO[C@@H](CNC7CCN(C8=C(N)N=NC(C9=CC=CC=C9O)=C8)CC7)C5)C6)CC4)=NO3)C(C)C)C=C2)SC=N1	C59H80N12O6S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-HSGB66	WO2023097031A1_114	.	CC(C)[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(N2CCC(CN3CCC(O[C@H]4C[C@H](OC(=O)N5CCN(C6=C(N)N=NC(C7=C(O)C=CC=C7)=C6)CC5)C4)CC3)CC2)=NO1	C55H72N12O8	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-OAMKCR	SCHEMBL25632652	[3-[1-[[1-[5-[(2R)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(2-methylpyrazol-3-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]-1,2-oxazol-3-yl]piperidin-4-yl]methyl]piperidin-4-yl]oxycyclobutyl] 4-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]piperazine-1-carboxylate; SCHEMBL31408981	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(N2CCC(CN3CCC(O[C@H]4C[C@H](OC(=O)N5CCN(C6=C(N)N=NC(C7=C(O)C=CC=C7)=C6)CC5)C4)CC3)CC2)=NO1	C55H72N12O8	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-WQMDR5	SCHEMBL25630599	[1-[5-[(2R)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]-1,2-oxazol-3-yl]piperidin-4-yl] 4-[3-[4-[3-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]pyridin-2-yl]oxycyclobutyl]oxypiperidine-1-carboxylate	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(OC(=O)N5CCC(O[C@H]6C[C@H](OC7=CC(N8C9CCC8CN(C8=C(N)N=NC(C%10=C(O)C=CC=C%10)=C8)C9)=CC=N7)C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C61H74N12O9S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-6NB2PQ	SCHEMBL25632682	(2S,4R)-1-[(2S)-2-[3-[4-[3-[4-[3-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]pyridin-2-yl]oxycyclobutanecarbonyl]piperazin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3=CC(N4CCN(C(=O)[C@H]5C[C@H](OC6=NC=CC(N7C8CCC7CN(C7=C(N)N=NC(C9=C(O)C=CC=C9)=C7)C8)=C6)C5)CC4)=NO3)C(C)C)C=C2)SC=N1	C55H64N12O7S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-X0Q962	SCHEMBL25632684	(2S,4R)-1-[(2R)-2-[3-[4-[[2-[3-[[3-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]methyl]-4,4-difluoropiperidin-1-yl]-7-azaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL31409042	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCC6(CC5)CC(N5CCC(F)(F)C(CN7C8CCC7CN(C7=C(N)N=NC(C9=C(O)C=CC=C9)=C7)C8)C5)C6)CC4)=NO3)C(C)C)C=C2)SC=N1	C61H80F2N12O5S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-57TDPH	SCHEMBL25630744	(2S,4R)-1-[(2R)-2-[3-[4-[[2-[(2S)-2-[3-[4-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]pyrazol-1-yl]but-1-ynyl]morpholin-4-yl]-7-azaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL31409071	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCC6(CC5)CC(N5CCO[C@@H](C#CC(C)N7C=C(C8=C(N)N=NC(C9=C(O)C=CC=C9)=C8)C=N7)C5)C6)CC4)=NO3)C(C)C)C=C2)SC=N1	C60H74N12O6S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-ZHP4MA	SCHEMBL25632686	(2S,4R)-1-[(2R)-2-[3-[4-[[2-[4-[[1-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-4-hydroxypiperidin-4-yl]methyl]piperazin-1-yl]-7-azaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL31409005	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCC6(CC5)CC(N5CCN(CC7(O)CCN(C8=C(N)N=NC(C9=C(O)C=CC=C9)=C8)CC7)CC5)C6)CC4)=NO3)C(C)C)C=C2)SC=N1	C59H80N12O6S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-C8SVCU	WO2023097031A1_123	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCN(C(=O)N5CCC(O[C@H]6C[C@H](OC7=NC(N8C9CCC8CN(C8=C(N)N=NC(C%10=C(O)C=CC=C%10)=C8)C9)=CC=N7)C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C59H72N14O8S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-MF6CL0	WO2023097031A1_124	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3=CC(N4CCN(C(=O)N5CCC(O[C@H]6C[C@H](OC7=NC(N8C9CCC8CN(C8=C(N)N=NC(C%10=C(O)C=CC=C%10)=C8)C9)=CC=N7)C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C59H72N14O8S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-OGGYM3	SCHEMBL25631000	(2S,4R)-1-[(2R)-2-[3-[4-[[2-[2-[[3-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3-azabicyclo[3.2.1]octan-8-yl]methyl]-5-oxa-2,8-diazaspiro[3.5]nonan-8-yl]-7-azaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL31409121	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCC6(CC5)CC(N5CCOC7(CN(CC8C9CCC8CN(C8=C(N)N=NC(C%10=CC=CC=C%10O)=C8)C9)C7)C5)C6)CC4)=NO3)C(C)C)C=C2)SC=N1	C63H84N12O6S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-4BCV9K	SCHEMBL25631062	(2S,4R)-1-[(2R)-2-[3-[4-[[2-[2-[[3-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]methyl]-5-oxa-8-azaspiro[3.5]nonan-8-yl]-7-azaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL31409018	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCC6(CC5)CC(N5CCOC7(CC(CN8C9CCC8CN(C8=C(N)N=NC(C%10=CC=CC=C%10O)=C8)C9)C7)C5)C6)CC4)=NO3)C(C)C)C=C2)SC=N1	C63H84N12O6S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-5TEZWG	WO2023097031A1_127	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@H](O)CN3C(=O)[C@@H](C3=CC(OCCOC(=O)N4CCC(OC5CC(OC6=CC(N7C8CCC7CN(C7=C(N)N=NC(C9=C(O)C=CC=C9)=C7)C8)=CC=N6)C5)CC4)=NO3)C(C)C)C=C2)SC=N1	C58H69N11O10S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-013DLN	SCHEMBL25632738	[1-[5-[(2R)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]-1,2-oxazol-3-yl]piperidin-4-yl] 4-[4-[3-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]pyridin-2-yl]oxypiperidine-1-carboxylate; SCHEMBL31409011	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(OC(=O)N5CCC(OC6=NC=CC(N7C8CCC7CN(C7=C(N)N=NC(C9=C(O)C=CC=C9)=C7)C8)=C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C57H68N12O8S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-QJMG1U	SCHEMBL25632739	(2S,4R)-1-[(2R)-2-[3-[4-[3-[4-[3-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]pyridin-2-yl]oxyazetidine-1-carbonyl]piperazin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL31408974	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCN(C(=O)N5CC(OC6=CC(N7C8CCC7CN(C7=C(N)N=NC(C9=C(O)C=CC=C9)=C7)C8)=CC=N6)C5)CC4)=NO3)C(C)C)C=C2)SC=N1	C54H63N13O7S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-U06O6H	SCHEMBL25631409	(2S,4R)-1-[(2R)-2-[3-[4-[[4-[3-[4-[[1-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]imidazol-4-yl]methyl]piperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL31409105	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCC(OC6CC(N7CCC(CC8=CN(C9=C(N)N=NC(C%10=CC=CC=C%10O)=C9)C=N8)CC7)C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C59H76N12O6S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-IRYBWU	SCHEMBL25632741	[1-[5-[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]-1,2-oxazol-3-yl]piperidin-4-yl] 4-[4-[3-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]pyridin-2-yl]oxypiperidine-1-carboxylate; SCHEMBL31409037	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3=CC(N4CCC(OC(=O)N5CCC(OC6=NC=CC(N7C8CCC7CN(C7=C(N)N=NC(C9=C(O)C=CC=C9)=C7)C8)=C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C57H68N12O8S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-0PPBFJ	SCHEMBL25631474	(2S,4R)-1-[(2R)-2-[3-[4-[[2-[(3S)-3-[[3-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]methyl]-4-methylpiperazin-1-yl]-7-azaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL31409085	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCC6(CC5)CC(N5CCN(C)[C@H](CN7C8CCC7CN(C7=C(N)N=NC(C9=CC=CC=C9O)=C7)C8)C5)C6)CC4)=NO3)C(C)C)C=C2)SC=N1	C61H83N13O5S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-R9H567	SCHEMBL25635879	2-[[5-[(2R)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]-1,2-oxazol-3-yl]oxy]ethyl 4-[3-[4-[3-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]pyridin-2-yl]oxycyclobutyl]oxypiperidine-1-carboxylate	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(OCCOC(=O)N4CCC(OC5CC(OC6=CC(N7C8CCC7CN(C7=C(N)N=NC(C9=C(O)C=CC=C9)=C7)C8)=CC=N6)C5)CC4)=NO3)C(C)C)C=C2)SC=N1	C58H69N11O10S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-6KWEN3	SCHEMBL25636056	(2S,4R)-1-[(2S)-2-[3-[4-[4-[3-[4-[3-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]pyridin-2-yl]oxycyclobutyl]oxypiperidine-1-carbonyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-N-[(1S)-1-(4-cyanophenyl)ethyl]-4-hydroxypyrrolidine-2-carboxamide	CC(C)[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C#N)C=C1)C1=CC(N2CCC(C(=O)N3CCC(O[C@H]4C[C@@H](OC5=NC=CC(N6C7CCC6CN(C6=C(N)N=NC(C8=C(O)C=CC=C8)=C6)C7)=C5)C4)CC3)CC2)=NO1	C58H70N12O8	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-ZS4JX4	SCHEMBL25636059	(2S,4R)-1-[(2R)-2-[3-[4-[4-[3-[4-[3-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]pyridin-2-yl]oxycyclobutyl]oxypiperidine-1-carbonyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-N-[(1S)-1-(4-cyanophenyl)ethyl]-4-hydroxypyrrolidine-2-carboxamide	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C#N)C=C1)C1=CC(N2CCC(C(=O)N3CCC(O[C@H]4C[C@H](OC5=NC=CC(N6C7CCC6CN(C6=C(N)N=NC(C8=C(O)C=CC=C8)=C6)C7)=C5)C4)CC3)CC2)=NO1	C58H70N12O8	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-N74AWU	SCHEMBL25632791	(2S,4R)-1-[(2S)-2-[3-[4-[4-[3-[4-[3-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]pyridin-2-yl]oxycyclobutyl]oxypiperidine-1-carbonyl]piperazin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-N-[(1S)-1-(4-cyanophenyl)ethyl]-4-hydroxypyrrolidine-2-carboxamide	CC(C)[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C#N)C=C1)C1=CC(N2CCN(C(=O)N3CCC(O[C@H]4C[C@H](OC5=NC=CC(N6C7CCC6CN(C6=C(N)N=NC(C8=C(O)C=CC=C8)=C6)C7)=C5)C4)CC3)CC2)=NO1	C57H69N13O8	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-FDOKKC	WO2023097031A1_140	.	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C#N)C=C1)C1=CC(N2CCN(C(=O)N3CCC(O[C@H]4C[C@H](OC5=NC(N6C7CCC6CN(C6=C(N)N=NC(C8=C(O)C=CC=C8)=C6)C7)=CC=N5)C4)CC3)CC2)=NO1	C56H68N14O8	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-13B8QU	WO2023097031A1_141	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CC6(CC(N7CCO[C@H](CN8C9CCC8CN(C8=C(N)N=NC(C%10=CC=CC=C%10O)=C8)C9)C7)C6)C5)CC4)=NO3)C(C)C)C=C2)SC=N1	C58H76N12O6S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-J877W4	SCHEMBL25632807	(2S,4R)-1-[(2R)-2-[3-[4-[[2-[(2S)-2-[[3-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]methyl]morpholin-4-yl]-6-azaspiro[3.5]nonan-6-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL31408983	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCCC6(CC(N7CCO[C@H](CN8C9CCC8CN(C8=C(N)N=NC(C%10=CC=CC=C%10O)=C8)C9)C7)C6)C5)CC4)=NO3)C(C)C)C=C2)SC=N1	C60H80N12O6S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-F9FA2N	WO2023097031A1_143	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCC6(CCC6N6CCO[C@@H](CN7C8CCC7CN(C7=C(N)N=NC(C9=CC=CC=C9O)=C7)C8)C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C60H80N12O6S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-CD7E23	SCHEMBL25632809	[1-[5-[1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]-1,2-oxazol-3-yl]piperidin-4-yl] 4-[4-[4-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]piperazin-1-yl]pyridin-2-yl]oxypiperidine-1-carboxylate; SCHEMBL31409103	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCC(OC(=O)N5CCC(OC6=NC=CC(N7CCN(C8=C(N)N=NC(C9=C(O)C=CC=C9)=C8)CC7)=C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C55H66N12O8S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-L55IK1	WO2023097031A1_145	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCC(OC(=O)N5CCC(O[C@H]6C[C@H](OC7=NC=CC(N8CCN(C9=C(N)N=NC(C%10=C(O)C=CC=C%10)=C9)CC8)=C7)C6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C59H72N12O9S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-OOTOI7	WO2023097031A1_146	.	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C#N)C=C1)C1=CC(N2CCC(CN3CC[C@H](OC4=NC=CC(N5C6CCC5CN(C5=C(N)N=NC(C7=C(O)C=CC=C7)=C5)C6)=C4)C(F)(F)C3)CC2)=NO1	C54H64F2N12O6	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-EYBXM0	SCHEMBL25632845	(2S,4R)-1-[(2R)-2-[3-[4-[[(4R)-4-[4-[3-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]pyridin-2-yl]oxy-3,3-difluoropiperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-N-[(1S)-1-(4-cyanophenyl)ethyl]-4-hydroxypyrrolidine-2-carboxamide; SCHEMBL31408989	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C#N)C=C1)C1=CC(N2CCC(CN3CC[C@@H](OC4=NC=CC(N5C6CCC5CN(C5=C(N)N=NC(C7=C(O)C=CC=C7)=C5)C6)=C4)C(F)(F)C3)CC2)=NO1	C54H64F2N12O6	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-GZYPYK	WO2023097031A1_148	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(OCCN4CCN(CCOC5=NC=CC(N6C7CCC6CN(C6=C(N)N=NC(C8=C(O)C=CC(F)=C8)=C6)C7)=C5)[C@H](C)C4)=NO3)C(C)C)C=C2)SC=N1	C55H67FN12O7S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-3CW4M9	SCHEMBL25632848	(2S,4R)-1-[(2R)-2-[3-[2-[(3R)-4-[2-[4-[3-[3-amino-6-(3-hydroxypyridin-2-yl)pyridazin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]pyridin-2-yl]oxyethyl]-3-methylpiperazin-1-yl]ethoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL31408964	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(OCCN4CCN(CCOC5=NC=CC(N6C7CCC6CN(C6=C(N)N=NC(C8=C(O)C=CC=N8)=C6)C7)=C5)[C@H](C)C4)=NO3)C(C)C)C=C2)SC=N1	C54H67N13O7S	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-J5LES1	SCHEMBL25636203	(2S,4R)-1-[(2S)-2-[3-[4-[2-[4-[4-[3-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]pyridin-2-yl]oxypiperidin-1-yl]ethoxy]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-N-[(1S)-1-(4-cyanophenyl)ethyl]-4-hydroxypyrrolidine-2-carboxamide; SCHEMBL31408977	CC(C)[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C#N)C=C1)C1=CC(N2CCC(OCCN3CCC(OC4=CC(N5C6CCC5CN(C5=C(N)N=NC(C7=C(O)C=CC=C7)=C5)C6)=CC=N4)CC3)CC2)=NO1	C55H68N12O7	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-ITQ38R	SCHEMBL25632851	(2S,4R)-1-[(2R)-2-[3-[4-[2-[4-[4-[3-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]pyridin-2-yl]oxypiperidin-1-yl]ethoxy]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-N-[(1S)-1-(4-cyanophenyl)ethyl]-4-hydroxypyrrolidine-2-carboxamide; SCHEMBL31408993	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C#N)C=C1)C1=CC(N2CCC(OCCN3CCC(OC4=CC(N5C6CCC5CN(C5=C(N)N=NC(C7=C(O)C=CC=C7)=C5)C6)=CC=N4)CC3)CC2)=NO1	C55H68N12O7	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-2LWEY9	WO2023097031A1_152	.	CC(C)[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C#N)C=C1)C1=CC(N2CCC(OCCN3CCC(OC4CC(OC5=NC=CC(N6C7CCC6CN(C6=C(N)N=NC(C8=C(O)C=CC=C8)=C6)C7)=C5)C4)CC3)CC2)=NO1	C59H74N12O8	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-IHX8W2	WO2023097031A1_153	.	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C#N)C=C1)C1=CC(N2CCC(OCCN3CCC(OC4CC(OC5=NC=CC(N6C7CCC6CN(C6=C(N)N=NC(C8=C(O)C=CC=C8)=C6)C7)=C5)C4)CC3)CC2)=NO1	C59H74N12O8	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-6JMKW5	SCHEMBL25632886	(2S,4R)-1-[(2S)-2-[3-[4-[2-[4-[4-[4-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]piperazin-1-yl]pyridin-2-yl]oxypiperidin-1-yl]ethoxy]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-N-[(1S)-1-(4-cyanophenyl)ethyl]-4-hydroxypyrrolidine-2-carboxamide; SCHEMBL31409013	CC(C)[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C#N)C=C1)C1=CC(N2CCC(OCCN3CCC(OC4=CC(N5CCN(C6=C(N)N=NC(C7=C(O)C=CC=C7)=C6)CC5)=CC=N4)CC3)CC2)=NO1	C53H66N12O7	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-C7019M	SCHEMBL25632887	(2S,4R)-1-[(2R)-2-[3-[4-[2-[4-[4-[4-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]piperazin-1-yl]pyridin-2-yl]oxypiperidin-1-yl]ethoxy]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-N-[(1S)-1-(4-cyanophenyl)ethyl]-4-hydroxypyrrolidine-2-carboxamide; SCHEMBL31409097	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C#N)C=C1)C1=CC(N2CCC(OCCN3CCC(OC4=CC(N5CCN(C6=C(N)N=NC(C7=C(O)C=CC=C7)=C6)CC5)=CC=N4)CC3)CC2)=NO1	C53H66N12O7	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-ZIAF2P	SCHEMBL25632889	(2S,4R)-1-[(2R)-2-[3-[4-[[(3R,4S)-4-[4-[3-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]pyridin-2-yl]oxy-3-fluoropiperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-N-[(1S)-1-(4-cyanophenyl)ethyl]-4-hydroxypyrrolidine-2-carboxamide; SCHEMBL31408998	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C#N)C=C1)C1=CC(N2CCC(CN3CC[C@H](OC4=NC=CC(N5C6CCC5CN(C5=C(N)N=NC(C7=C(O)C=CC=C7)=C5)C6)=C4)[C@H](F)C3)CC2)=NO1	C54H65FN12O6	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-BLSD4Q	SCHEMBL25632941	(2S,4R)-1-[(2R)-2-[3-[4-[[(3S,4R)-4-[4-[3-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]pyridin-2-yl]oxy-3-fluoropiperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-N-[(1S)-1-(4-cyanophenyl)ethyl]-4-hydroxypyrrolidine-2-carboxamide; SCHEMBL31409069	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C#N)C=C1)C1=CC(N2CCC(CN3CC[C@@H](OC4=NC=CC(N5C6CCC5CN(C5=C(N)N=NC(C7=C(O)C=CC=C7)=C5)C6)=C4)[C@@H](F)C3)CC2)=NO1	C54H65FN12O6	SMARCA2	P51531	VHL	WO-2023097031-A1
TPD-POIBM4	WO2023116934A1_I-1	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CC4CCC(C1)N4)=NC(OC[C@]14CCCN1[C@@H](CNC(=O)CCNC1=CC=CC5=C1C(=O)N(C1CCC(=O)NC1=O)C5=O)CC4)=N3)=CC(O)=C2	C50H48F2N10O7	KRAS	P01116	CRBN	WO-2023116934-A1
TPD-37VY8C	WO2023116934A1_I-10	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CC4CCC(C1)N4)=NC(OC[C@]14CCCN1[C@H](CN(C)C(=O)CCCCCCNC1=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C1)CC4)=N3)=CC(O)=C2	C55H58F2N10O7	KRAS	P01116	CRBN	WO-2023116934-A1
TPD-KKALJT	WO2023116934A1_I-11	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CC4CCC(C1)N4)=NC(OC[C@]14CCCN1[C@H](CN(C)C(=O)CCCCCCCCCNC1=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C1)CC4)=N3)=CC(O)=C2	C58H64F2N10O7	KRAS	P01116	CRBN	WO-2023116934-A1
TPD-4I6VZQ	SCHEMBL25821102	N-[[(3S,8R)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl]-2-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperazin-1-yl]-N-methylacetamide	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CC4CCC(C1)N4)=NC(OC[C@]14CCCN1[C@H](CN(C)C(=O)CN1CCN(C5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC1)CC4)=N3)=CC(O)=C2	C59H64F2N12O7	KRAS	P01116	CRBN	WO-2023116934-A1
TPD-7H344A	WO2023116934A1_I-13	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CC4CCC(C1)N4)=NC(OC[C@]14CCCN1[C@H](CN(C)C(=O)CC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C5=C(C)N=CS5)C=C1)C(C)(C)C)CC4)=N3)=CC(O)=C2	C60H67F2N11O7S	KRAS	P01116	VHL	WO-2023116934-A1
TPD-Y9PANF	WO2023116934A1_I-14	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CC4CCC(C1)N4)=NC(OC[C@]14CCCN1[C@H](CN(C)C(=O)CCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C5=C(C)N=CS5)C=C1)C(C)(C)C)CC4)=N3)=CC(O)=C2	C61H69F2N11O7S	KRAS	P01116	VHL	WO-2023116934-A1
TPD-RHW7AC	WO2023116934A1_I-15	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CC4CCC(C1)N4)=NC(OC[C@]14CCCN1[C@H](CN(C)C(=O)CCCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C5=C(C)N=CS5)C=C1)C(C)(C)C)CC4)=N3)=CC(O)=C2	C62H71F2N11O7S	KRAS	P01116	VHL	WO-2023116934-A1
TPD-N56CF0	WO2023116934A1_I-16	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CC4CCC(C1)N4)=NC(OC[C@]14CCCN1[C@H](CN(C)C(=O)CCCCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C5=C(C)N=CS5)C=C1)C(C)(C)C)CC4)=N3)=CC(O)=C2	C63H73F2N11O7S	KRAS	P01116	VHL	WO-2023116934-A1
TPD-FIT8PY	WO2023116934A1_I-17	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CC4CCC(C1)N4)=NC(OC[C@]14CCCN1[C@H](CN(C)C(=O)CCCCCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C5=C(C)N=CS5)C=C1)C(C)(C)C)CC4)=N3)=CC(O)=C2	C64H75F2N11O7S	KRAS	P01116	VHL	WO-2023116934-A1
TPD-2ZWYTW	WO2023116934A1_I-18	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CC4CCC(C1)N4)=NC(OC[C@]14CCCN1[C@H](CN(C)C(=O)CCCCCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C5=C(C)N=CS5)C=C1)C(C)(C)C)CC4)=N3)=CC(O)=C2	C65H77F2N11O7S	KRAS	P01116	VHL	WO-2023116934-A1
TPD-25Z0DA	WO2023116934A1_I-19	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CC4CCC(C1)N4)=NC(OC[C@]14CCCN1[C@H](CN(C)C(=O)COCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C5=C(C)N=CS5)C=C1)C(C)(C)C)CC4)=N3)=CC(O)=C2	C61H69F2N11O8S	KRAS	P01116	VHL	WO-2023116934-A1
TPD-ZSS0RU	WO2023116934A1_I-2	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CC4CCC(C1)N4)=NC(OC[C@]14CCCN1[C@@H](CNC(=O)CCCNC1=CC=CC5=C1C(=O)N(C1CCC(=O)NC1=O)C5=O)CC4)=N3)=CC(O)=C2	C51H50F2N10O7	KRAS	P01116	VHL	WO-2023116934-A1
TPD-1WL41I	WO2023116934A1_I-20	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CC4CCC(C1)N4)=NC(OC[C@]14CCCN1[C@H](CN(C)C(=O)CCOCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C5=C(C)N=CS5)C=C1)C(C)(C)C)CC4)=N3)=CC(O)=C2	C62H71F2N11O8S	KRAS	P01116	VHL	WO-2023116934-A1
TPD-ZC1JG3	WO2023116934A1_I-21	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CC4CCC(C1)N4)=NC(OC[C@]14CCCN1[C@H](CN(C)C(=O)CCOCCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C5=C(C)N=CS5)C=C1)C(C)(C)C)CC4)=N3)=CC(O)=C2	C63H73F2N11O8S	KRAS	P01116	VHL	WO-2023116934-A1
TPD-2PXWME	WO2023116934A1_I-22	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CC4CCC(C1)N4)=NC(OC[C@]14CCCN1[C@H](CN(C)C(=O)CCOCCOCCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C5=C(C)N=CS5)C=C1)C(C)(C)C)CC4)=N3)=CC(O)=C2	C65H77F2N11O9S	KRAS	P01116	VHL	WO-2023116934-A1
TPD-DQF5BH	WO2023116934A1_I-3	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CC4CCC(C1)N4)=NC(OC[C@]14CCCN1[C@@H](CNC(=O)CCCCNC1=CC=CC5=C1C(=O)N(C1CCC(=O)NC1=O)C5=O)CC4)=N3)=CC(O)=C2	C52H52F2N10O7	KRAS	P01116	CRBN	WO-2023116934-A1
TPD-WGO9SP	WO2023116934A1_I-4	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CC4CCC(C1)N4)=NC(OC[C@]14CCCN1[C@@H](CNC(=O)CCCCCNC1=CC=CC5=C1C(=O)N(C1CCC(=O)NC1=O)C5=O)CC4)=N3)=CC(O)=C2	C53H54F2N10O7	KRAS	P01116	CRBN	WO-2023116934-A1
TPD-BP7FVB	WO2023116934A1_I-5	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CC4CCC(C1)N4)=NC(OC[C@]14CCCN1[C@@H](CNC(=O)CCCCCCNC1=CC=CC5=C1C(=O)N(C1CCC(=O)NC1=O)C5=O)CC4)=N3)=CC(O)=C2	C54H56F2N10O7	KRAS	P01116	CRBN	WO-2023116934-A1
TPD-X55LHP	WO2023116934A1_I-6	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CC4CCC(C1)N4)=NC(OC[C@]14CCCN1[C@H](CN(C)C(=O)CCNC1=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C1)CC4)=N3)=CC(O)=C2	C51H50F2N10O7	KRAS	P01116	CRBN	WO-2023116934-A1
TPD-N29VGR	WO2023116934A1_I-7	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CC4CCC(C1)N4)=NC(OC[C@]14CCCN1[C@H](CN(C)C(=O)CCCNC1=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C1)CC4)=N3)=CC(O)=C2	C52H52F2N10O7	KRAS	P01116	CRBN	WO-2023116934-A1
TPD-T7KUKR	WO2023116934A1_I-8	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CC4CCC(C1)N4)=NC(OC[C@]14CCCN1[C@H](CN(C)C(=O)CCCCNC1=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C1)CC4)=N3)=CC(O)=C2	C53H54F2N10O7	KRAS	P01116	CRBN	WO-2023116934-A1
TPD-T0GAPI	WO2023116934A1_I-9	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CC4CCC(C1)N4)=NC(OC[C@]14CCCN1[C@H](CN(C)C(=O)CCCCCNC1=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C1)CC4)=N3)=CC(O)=C2	C54H56F2N10O7	KRAS	P01116	CRBN	WO-2023116934-A1
TPD-OV1LN0	WO2023116934A1_II-1	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CC4CCC(C1)N4)=NC(OC[C@H]1CCCN1C(=O)CCNC1=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C1)=N3)=CC(O)=C2	C46H41F2N9O7	KRAS	P01116	CRBN	WO-2023116934-A1
TPD-M6ZD3R	WO2023116934A1_II-2	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CC4CCC(C1)N4)=NC(OC[C@H]1CCCN1C(=O)CCCNC1=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C1)=N3)=CC(O)=C2	C47H43F2N9O7	KRAS	P01116	CRBN	WO-2023116934-A1
TPD-PYJ7BZ	WO2023116934A1_II-3	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CC4CCC(C1)N4)=NC(OC[C@H]1CCCN1C(=O)CCCCNC1=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C1)=N3)=CC(O)=C2	C48H45F2N9O7	KRAS	P01116	CRBN	WO-2023116934-A1
TPD-WYX3Q5	WO2023116934A1_II-4	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CC4CCC(C1)N4)=NC(OC[C@H]1CCCN1C(=O)CCCCCNC1=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C1)=N3)=CC(O)=C2	C49H47F2N9O7	KRAS	P01116	CRBN	WO-2023116934-A1
TPD-NHCJHR	SCHEMBL25821381	4-[[7-[(2R)-2-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]pyrrolidin-1-yl]-7-oxoheptyl]amino]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CC4CCC(C1)N4)=NC(OC[C@H]1CCCN1C(=O)CCCCCCNC1=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C1)=N3)=CC(O)=C2	C50H49F2N9O7	KRAS	P01116	CRBN	WO-2023116934-A1
TPD-QXRJEL	YD23	1H-Isoindole-1,3(2H)-dione, 4-[[2-[2-[4-[[4-[3-amino-6-(2-hydroxyphenyl)-4-pyridazinyl]-1-piperazinyl]methyl]-2-fluorophenoxy]ethoxy]ethyl]amino]-2-(2,6-dioxo-3-piperidinyl)-; 2951015-29-3; 1H-Isoindole-1,3(2H)-dione, 4-[[2-[2-[4-[[4-[3-amino-6-(2-hydroxyphenyl)-4-pyridazinyl]-1-piperazinyl]methyl]-2-fluorophenoxy]ethoxy]ethyl]amino]-2-(2,6-dioxo-3-piperidinyl)-; orb2278977; SCHEMBL25815188; EX-A7830; AT45556; BP-42170; HY-153361	Nc1nnc(-c2ccccc2O)cc1N1CCN(Cc2ccc(OCCOCCNc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)c(F)c2)CC1	C38H39FN8O7	SMARCA2	P51531	CRBN	WO-2023129506-A1
TPD-GRUFP8	orb2695207	4-[2-[4-[4-[[4-[3-Amino-6-(2-hydroxyphenyl)pyridazin-4-yl]piperazin-1-yl]methyl]-2-fluorophenyl]piperazin-1-yl]ethoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione; YD54; SCHEMBL25816186; GTPL13901; 2951015-30-6; 4-[2-[4-[4-[[4-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]piperazin-1-yl]methyl]-2-fluorophenyl]piperazin-1-yl]ethoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	Nc1nnc(-c2ccccc2O)cc1N1CCN(Cc2ccc(N3CCN(CCOc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)c(F)c2)CC1	C40H42FN9O6	SMARCA2	P51531	CRBN	WO-2023129506-A1
TPD-CVJZZL	2951015-31-7	5-[4-[[1-[4-[[4-[3-Amino-6-(2-hydroxyphenyl)pyridazin-4-yl]piperazin-1-yl]methyl]-2-fluorophenyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione; YDR1; orb2695662; SCHEMBL25816414; EX-A13244	Nc1nnc(-c2ccccc2O)cc1N1CCN(Cc2ccc(N3CCC(CN4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)c(F)c2)CC1	C44H49FN10O5	SMARCA2	P51531	CRBN	WO-2023129506-A1
TPD-2V9IQZ	SCHEMBL25815260	4-[2-[2-[4-[[4-[3-Amino-6-(2-hydroxyphenyl)pyridazin-4-yl]piperazin-1-yl]methyl]-2,6-difluorophenoxy]ethoxy]ethylamino]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	Nc1nnc(-c2ccccc2O)cc1N1CCN(Cc2cc(F)c(OCCOCCNc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)c(F)c2)CC1	C38H38F2N8O7	SMARCA2	P51531	CRBN	WO-2023129506-A1
TPD-X2I7VH	SCHEMBL25815262	4-[2-[2-[4-[[4-[3-Amino-6-(2-hydroxyphenyl)pyridazin-4-yl]piperazin-1-yl]methyl]-2,3-difluorophenoxy]ethoxy]ethylamino]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	Nc1nnc(-c2ccccc2O)cc1N1CCN(Cc2ccc(OCCOCCNc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)c(F)c2F)CC1	C38H38F2N8O7	SMARCA2	P51531	CRBN	WO-2023129506-A1
TPD-IRTIHA	SCHEMBL25815278	4-[2-[2-[4-[[4-[3-Amino-6-(2-hydroxyphenyl)pyridazin-4-yl]piperazin-1-yl]methyl]-2,5-difluorophenoxy]ethoxy]ethylamino]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	Nc1nnc(-c2ccccc2O)cc1N1CCN(Cc2cc(F)c(OCCOCCNc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)cc2F)CC1	C38H38F2N8O7	SMARCA2	P51531	CRBN	WO-2023129506-A1
TPD-NKM15K	SCHEMBL25815933	4-[2-[2-[4-[[4-[3-Amino-6-(2-hydroxyphenyl)pyridazin-4-yl]piperazin-1-yl]methyl]-3,5-difluorophenoxy]ethoxy]ethylamino]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	Nc1nnc(-c2ccccc2O)cc1N1CCN(Cc2c(F)cc(OCCOCCNc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)cc2F)CC1	C38H38F2N8O7	SMARCA2	P51531	CRBN	WO-2023129506-A1
TPD-G2MNLA	SCHEMBL25815256	4-[2-[3-[4-[[4-[3-Amino-6-(2-hydroxyphenyl)pyridazin-4-yl]piperazin-1-yl]methyl]-2-fluorophenyl]propoxy]ethylamino]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	Nc1nnc(-c2ccccc2O)cc1N1CCN(Cc2ccc(CCCOCCNc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)c(F)c2)CC1	C39H41FN8O6	SMARCA2	P51531	CRBN	WO-2023129506-A1
TPD-NSPKPD	SCHEMBL30488311	5-[4-[[4-[[4-[[1-(3-Aminopropyl)-3-[4-(trifluoromethoxy)phenyl]indol-5-yl]methyl]piperazin-1-yl]methyl]phenyl]methyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	NCCCn1cc(-c2ccc(OC(F)(F)F)cc2)c2cc(CN3CCN(Cc4ccc(CN5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)cc4)CC3)ccc21	C48H51F3N8O5	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-D9SW7A	SCHEMBL25435573	4-amino-N-[3-[5-[[4-[[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]phenyl]methyl]piperazin-1-yl]methyl]-3-[4-(trifluoromethoxy)phenyl]indol-1-yl]propyl]piperidine-4-carboxamide	NC1(C(=O)NCCCn2cc(-c3ccc(OC(F)(F)F)cc3)c3cc(CN4CCN(Cc5ccc(CN6CCN(c7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)cc5)CC4)ccc32)CCNCC1	C54H61F3N10O6	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-LI42K3	SCHEMBL25438692	5-[4-[[4-[[1-(3-Aminopropyl)-3-[4-(trifluoromethoxy)phenyl]indol-5-yl]methyl]piperazin-1-yl]methyl]piperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	NCCCn1cc(-c2ccc(OC(F)(F)F)cc2)c2cc(CN3CCN(CC4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)ccc21	C42H46F3N7O5	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-OBZI76	SCHEMBL30488342	5-[4-[[4-[[1-(3-Aminopropyl)-3-(4-hydroxyphenyl)indol-5-yl]methyl]piperazin-1-yl]methyl]piperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	NCCCn1cc(-c2ccc(O)cc2)c2cc(CN3CCN(CC4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)ccc21	C41H47N7O5	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-ZOYRZX	SCHEMBL30488060	5-[4-[[1-[[1-(3-Aminopropyl)-3-(4-hydroxyphenyl)indol-5-yl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	NCCCn1cc(-c2ccc(O)cc2)c2cc(CN3CCC(CN4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)ccc21	C41H47N7O5	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-G11OBI	SCHEMBL25424686	5-[4-[[1-[[1-(3-Aminopropyl)-3-[4-(trifluoromethoxy)phenyl]indol-5-yl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	NCCCn1cc(-c2ccc(OC(F)(F)F)cc2)c2cc(CN3CCC(CN4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)ccc21	C42H46F3N7O5	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-RNZWLE	SCHEMBL30488046	5-[4-[[4-[[1-(3-Aminopropyl)-3-(4-fluorophenyl)indol-5-yl]methyl]piperazin-1-yl]methyl]piperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	NCCCn1cc(-c2ccc(F)cc2)c2cc(CN3CCN(CC4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)ccc21	C41H46FN7O4	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-FFH55M	SCHEMBL30488048	5-[4-[[1-(3-Aminopropyl)-3-[4-(trifluoromethoxy)phenyl]indol-5-yl]methyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	NCCCn1cc(-c2ccc(OC(F)(F)F)cc2)c2cc(CN3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)ccc21	C36H35F3N6O5	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-MPIBLG	SCHEMBL30488084	5-[4-[[4-[[1-(3-Aminopropyl)-3-(4-methoxyphenyl)indol-5-yl]methyl]piperazin-1-yl]methyl]piperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	COc1ccc(-c2cn(CCCN)c3ccc(CN4CCN(CC5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc23)cc1	C42H49N7O5	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-U3N2KA	SCHEMBL25421625	4-[1-(3-Aminopropyl)-5-[[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]methyl]indol-3-yl]benzonitrile	N#Cc1ccc(-c2cn(CCCN)c3ccc(CN4CCC(CN5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc23)cc1	C42H46N8O4	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-28XF5J	WO2023130012A1_12	.	COc1ccc(-c2cn(CCCN)c3ccc(CN4CCC(CN5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc23)cn1	C41H48N8O5	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-BSSSQL	SCHEMBL25422541	3-[1-(3-Aminopropyl)-5-[[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]methyl]indol-3-yl]benzonitrile; SCHEMBL30488047	N#Cc1cccc(-c2cn(CCCN)c3ccc(CN4CCC(CN5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc23)c1	C42H46N8O4	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-Q27B1D	SCHEMBL25426473	5-[4-[[1-[[1-(3-Aminopropyl)-3-[4-(trifluoromethoxy)phenyl]indol-7-yl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	NCCCn1cc(-c2ccc(OC(F)(F)F)cc2)c2cccc(CN3CCC(CN4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)c21	C42H46F3N7O5	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-BV0MW8	SCHEMBL30488332	5-[4-[[1-[[1-(3-Aminopropyl)-3-(2-fluoro-4-methoxyphenyl)indol-5-yl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	COc1ccc(-c2cn(CCCN)c3ccc(CN4CCC(CN5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc23)c(F)c1	C42H48FN7O5	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-FDS5K6	SCHEMBL30488349	5-[4-[[1-[[1-(3-Aminopropyl)-3-[4-(trifluoromethoxy)phenyl]indol-6-yl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	NCCCn1cc(-c2ccc(OC(F)(F)F)cc2)c2ccc(CN3CCC(CN4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)cc21	C42H46F3N7O5	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-V2G5E0	SCHEMBL30488370	5-[4-[[1-[[1-(3-Aminopropyl)-3-(2-methoxypyridin-3-yl)indol-5-yl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	COc1ncccc1-c1cn(CCCN)c2ccc(CN3CCC(CN4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)cc12	C41H48N8O5	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-AK97PZ	SCHEMBL25439709	5-[4-[[1-[[1-(3-Aminopropyl)-3-[4-(trifluoromethyl)phenyl]indol-5-yl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	NCCCn1cc(-c2ccc(C(F)(F)F)cc2)c2cc(CN3CCC(CN4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)ccc21	C42H46F3N7O4	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-OB83V9	SCHEMBL30488331	5-[4-[[1-[[1-(3-Aminopropyl)-3-[4-(trifluoromethoxy)phenyl]indol-4-yl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	NCCCn1cc(-c2ccc(OC(F)(F)F)cc2)c2c(CN3CCC(CN4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)cccc21	C42H46F3N7O5	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-EWJOFX	SCHEMBL25423185	4-[4-[[1-[[1-(3-Aminopropyl)-3-[4-(trifluoromethoxy)phenyl]indol-5-yl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione; SCHEMBL30488363	NCCCn1cc(-c2ccc(OC(F)(F)F)cc2)c2cc(CN3CCC(CN4CCN(c5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)ccc21	C42H46F3N7O5	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-HTOA42	SCHEMBL30488052	tert-butyl N-[3-[5-[[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]methyl]-3-[4-(trifluoromethoxy)phenyl]indol-1-yl]propyl]carbamate	CC(C)(C)OC(=O)NCCCn1cc(-c2ccc(OC(F)(F)F)cc2)c2cc(CN3CCC(CN4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)ccc21	C47H54F3N7O7	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-6JKJPB	SCHEMBL25422385	5-[3-[1-[[1-(3-Aminopropyl)-3-[4-(trifluoromethoxy)phenyl]indol-5-yl]methyl]piperidin-4-yl]oxyprop-1-ynyl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	NCCCn1cc(-c2ccc(OC(F)(F)F)cc2)c2cc(CN3CCC(OCC#Cc4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)ccc21	C40H38F3N5O6	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-666F1G	SCHEMBL25427046	5-[3-[1-[[1-(3-Aminopropyl)-3-[4-(trifluoromethoxy)phenyl]indol-5-yl]methyl]piperidin-4-yl]oxypropyl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	NCCCn1cc(-c2ccc(OC(F)(F)F)cc2)c2cc(CN3CCC(OCCCc4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)ccc21	C40H42F3N5O6	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-8237O2	SCHEMBL25423957	5-[4-[2-[4-[[1-(3-Aminopropyl)-3-[4-(trifluoromethoxy)phenyl]indol-5-yl]methyl]piperazin-1-yl]acetyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	NCCCn1cc(-c2ccc(OC(F)(F)F)cc2)c2cc(CN3CCN(CC(=O)N4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)ccc21	C42H45F3N8O6	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-JE0GJU	SCHEMBL25436285	5-[4-[[1-[[1-(3-Aminopropyl)-3-[3-(trifluoromethoxy)phenyl]indol-5-yl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	NCCCn1cc(-c2cccc(OC(F)(F)F)c2)c2cc(CN3CCC(CN4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)ccc21	C42H46F3N7O5	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-DTD9YP	SCHEMBL30488068	5-[4-[[1-[1-(3-Aminopropyl)-3-[4-(trifluoromethoxy)phenyl]indole-5-carbonyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	NCCCn1cc(-c2ccc(OC(F)(F)F)cc2)c2cc(C(=O)N3CCC(CN4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)ccc21	C42H44F3N7O6	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-C4IFOG	SCHEMBL30488325	5-[4-[[1-[[1-(3-Aminopropyl)-3-(3-hydroxynaphthalen-1-yl)indol-5-yl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	NCCCn1cc(-c2cc(O)cc3ccccc23)c2cc(CN3CCC(CN4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)ccc21	C45H49N7O5	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-16G5IO	SCHEMBL25437601	5-[4-[[1-[[1-(Azetidin-3-ylmethyl)-3-[4-(trifluoromethoxy)phenyl]indol-5-yl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	O=C1CCC(N2C(=O)c3ccc(N4CCN(CC5CCN(Cc6ccc7c(c6)c(-c6ccc(OC(F)(F)F)cc6)cn7CC6CNC6)CC5)CC4)cc3C2=O)C(=O)N1	C43H46F3N7O5	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-FJJPY5	WO2023130012A1_29	.	Cc1cc2[nH]ncc2c(-c2cn(CCCN)c3ccc(CN4CCC(CN5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc23)c1Cl	C43H48ClN9O4	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-JGKEYW	WO2023130012A1_31	.	Cc1ncsc1-c1ccc(CNC(=O)C2CC(O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)C)c(OCCCN2CCN(Cc3ccc4c(c3)c(-c3ccc(OC(F)(F)F)cc3)cn4CCCN)CC2)c1	C52H64F4N8O6S	KRAS	P01116	VHL	WO-2023130012-A1
TPD-IX5NQ3	SCHEMBL30488050	5-[4-[[1-[[1-(3-Aminopropyl)-3-[4-(trifluoromethoxy)phenyl]indol-5-yl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)-6-fluoroisoindole-1,3-dione	NCCCn1cc(-c2ccc(OC(F)(F)F)cc2)c2cc(CN3CCC(CN4CCN(c5cc6c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)ccc21	C42H45F4N7O5	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-BGLZ6F	SCHEMBL30488329	2-(2,6-Dioxopiperidin-3-yl)-5-[4-[[1-[[1-[3-(methylamino)propyl]-3-[4-(trifluoromethoxy)phenyl]indol-5-yl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]isoindole-1,3-dione	CNCCCn1cc(-c2ccc(OC(F)(F)F)cc2)c2cc(CN3CCC(CN4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)ccc21	C43H48F3N7O5	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-5PZCT9	SCHEMBL30488082	5-[7-[[1-(3-Aminopropyl)-3-[4-(trifluoromethoxy)phenyl]indol-5-yl]methyl]-2,7-diazaspiro[3.5]nonan-2-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	NCCCn1cc(-c2ccc(OC(F)(F)F)cc2)c2cc(CN3CCC4(CC3)CN(c3ccc5c(c3)C(=O)N(C3CCC(=O)NC3=O)C5=O)C4)ccc21	C39H39F3N6O5	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-UHP7PD	SCHEMBL30488061	5-[4-[[1-[[1-(3-Aminopropyl)-3-[2-fluoro-4-[(3-fluoropyridin-2-yl)methoxy]phenyl]indol-5-yl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	NCCCn1cc(-c2ccc(OCc3ncccc3F)cc2F)c2cc(CN3CCC(CN4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)ccc21	C47H50F2N8O5	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-WD4HWE	SCHEMBL30488069	5-[4-[1-[[1-(3-Aminopropyl)-3-[4-(trifluoromethoxy)phenyl]indol-5-yl]methyl]azetidin-3-yl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	NCCCn1cc(-c2ccc(OC(F)(F)F)cc2)c2cc(CN3CC(N4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C3)ccc21	C39H40F3N7O5	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-T8X8TP	SCHEMBL25437233	5-[4-[[1-[[1-[3-(Dimethylamino)propyl]-3-[4-(trifluoromethoxy)phenyl]indol-5-yl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN(C)CCCn1cc(-c2ccc(OC(F)(F)F)cc2)c2cc(CN3CCC(CN4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)ccc21	C44H50F3N7O5	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-58OZ6D	WO2023130012A1_38	.	NCCCCCn1cc(-c2ccc(OC(F)(F)F)cc2)c2cc(CN3CCC(CN4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)ccc21	C44H50F3N7O5	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-1G7CZ7	SCHEMBL30488076	5-[7-[[1-[[1-(3-Aminopropyl)-3-[4-(trifluoromethoxy)phenyl]indol-5-yl]methyl]piperidin-4-yl]methyl]-2,7-diazaspiro[3.5]nonan-2-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	NCCCn1cc(-c2ccc(OC(F)(F)F)cc2)c2cc(CN3CCC(CN4CCC5(CC4)CN(c4ccc6c(c4)C(=O)N(C4CCC(=O)NC4=O)C6=O)C5)CC3)ccc21	C45H50F3N7O5	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-QM36HU	SCHEMBL25425156	N-[3-[5-[[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]methyl]-3-[4-(trifluoromethoxy)phenyl]indol-1-yl]propyl]acetamide; SCHEMBL30488078	CC(=O)NCCCn1cc(-c2ccc(OC(F)(F)F)cc2)c2cc(CN3CCC(CN4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)ccc21	C44H48F3N7O6	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-LWM151	SCHEMBL25424176	4-[5-[[4-[[4-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]methyl]-3-[4-(trifluoromethoxy)phenyl]indol-1-yl]butanenitrile; SCHEMBL30488049	N#CCCCn1cc(-c2ccc(OC(F)(F)F)cc2)c2cc(CN3CCC(CN4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)ccc21	C43H44F3N7O5	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-HDU8KA	WO2023130012A1_42	.	Cn1cncc1Cn1cc(-c2ccc(OC(F)(F)F)cc2)c2cc(CN3CCC(CN4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)ccc21	C44H45F3N8O5	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-P5WAL7	SCHEMBL30488326	2-(2,6-Dioxopiperidin-3-yl)-5-[4-[[1-[[1-(3-methoxypropyl)-3-[4-(trifluoromethoxy)phenyl]indol-5-yl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]isoindole-1,3-dione	COCCCn1cc(-c2ccc(OC(F)(F)F)cc2)c2cc(CN3CCC(CN4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)ccc21	C43H47F3N6O6	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-AROEIR	SCHEMBL25437871	2-(2,6-Dioxopiperidin-3-yl)-5-[4-[[1-[[1-[3-(2,2,2-trifluoroethoxy)propyl]-3-[4-(trifluoromethoxy)phenyl]indol-5-yl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]isoindole-1,3-dione	O=C1CCC(N2C(=O)c3ccc(N4CCN(CC5CCN(Cc6ccc7c(c6)c(-c6ccc(OC(F)(F)F)cc6)cn7CCCOCC(F)(F)F)CC5)CC4)cc3C2=O)C(=O)N1	C44H46F6N6O6	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-D6BQN2	SCHEMBL25437395	N-[3-[5-[[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]methyl]-3-[4-(trifluoromethoxy)phenyl]indol-1-yl]propyl]-1H-pyrrole-2-carboxamide; SCHEMBL30488057	O=C1CCC(N2C(=O)c3ccc(N4CCN(CC5CCN(Cc6ccc7c(c6)c(-c6ccc(OC(F)(F)F)cc6)cn7CCCNC(=O)c6ccc[nH]6)CC5)CC4)cc3C2=O)C(=O)N1	C47H49F3N8O6	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-QZHAET	SCHEMBL25438857	3-[4-[1-[[1-(3-Aminopropyl)-3-[4-(trifluoromethoxy)phenyl]indol-5-yl]methyl]piperidin-4-yl]-3-fluoroanilino]piperidine-2,6-dione	NCCCn1cc(-c2ccc(OC(F)(F)F)cc2)c2cc(CN3CCC(c4ccc(NC5CCC(=O)NC5=O)cc4F)CC3)ccc21	C35H37F4N5O3	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-G41Y9B	WO2023130012A1_47	.	O=C1CCC(N2C(=O)c3ccc(N4CCN(CC5CCN(Cc6ccc7c(c6)c(-c6ccc(OC(F)(F)F)cc6)cn7CCCNC(=O)c6cccc(C(F)(F)F)c6)CC5)CC4)cc3C2=O)C(=O)N1	C50H49F6N7O6	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-G9B6NJ	SCHEMBL25427783	N-[3-[5-[[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]methyl]-3-[4-(trifluoromethoxy)phenyl]indol-1-yl]propyl]-4-fluorobenzamide; SCHEMBL30488044	O=C1CCC(N2C(=O)c3ccc(N4CCN(CC5CCN(Cc6ccc7c(c6)c(-c6ccc(OC(F)(F)F)cc6)cn7CCCNC(=O)c6ccc(F)cc6)CC5)CC4)cc3C2=O)C(=O)N1	C49H49F4N7O6	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-W0WZ8X	SCHEMBL25437402	3-[4-[4-[[1-[[1-(3-Aminopropyl)-3-[4-(trifluoromethoxy)phenyl]indol-5-yl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-fluoroanilino]piperidine-2,6-dione	NCCCn1cc(-c2ccc(OC(F)(F)F)cc2)c2cc(CN3CCC(CN4CCN(c5ccc(NC6CCC(=O)NC6=O)cc5F)CC4)CC3)ccc21	C40H47F4N7O3	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-LF384X	SCHEMBL30488065	5-[4-[[1-[[1-Butyl-3-[4-(trifluoromethoxy)phenyl]indol-5-yl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CCCCn1cc(-c2ccc(OC(F)(F)F)cc2)c2cc(CN3CCC(CN4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)ccc21	C43H47F3N6O5	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-VRY5VK	SCHEMBL30488075	2-(2,6-dioxopiperidin-3-yl)-5-[4-[[1-[[3-[4-(trifluoromethoxy)phenyl]-1H-indol-5-yl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]isoindole-1,3-dione	O=C1CCC(N2C(=O)c3ccc(N4CCN(CC5CCN(Cc6ccc7[nH]cc(-c8ccc(OC(F)(F)F)cc8)c7c6)CC5)CC4)cc3C2=O)C(=O)N1	C39H39F3N6O5	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-82B28C	WO2023130012A1_52	.	O=C1CCC(N2C(=O)c3ccc(N4CCN(CC5CCN(Cc6ccc7c(c6)c(-c6ccc(OC(F)(F)F)cc6)cn7CC6COc7ccccc7O6)CC5)CC4)cc3C2=O)C(=O)N1	C48H47F3N6O7	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-5OXU4U	SCHEMBL30488346	2-(2,6-Dioxopiperidin-3-yl)-5-[4-[[1-[[1-(pyridin-2-ylmethyl)-3-[4-(trifluoromethoxy)phenyl]indol-5-yl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]isoindole-1,3-dione	O=C1CCC(N2C(=O)c3ccc(N4CCN(CC5CCN(Cc6ccc7c(c6)c(-c6ccc(OC(F)(F)F)cc6)cn7Cc6ccccn6)CC5)CC4)cc3C2=O)C(=O)N1	C45H44F3N7O5	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-4FFP8K	SCHEMBL30488397	3-[4-[4-[1-[[1-(3-Aminopropyl)-3-[4-(trifluoromethoxy)phenyl]indol-5-yl]methyl]piperidin-4-yl]piperidin-1-yl]-3-fluoroanilino]piperidine-2,6-dione	NCCCn1cc(-c2ccc(OC(F)(F)F)cc2)c2cc(CN3CCC(C4CCN(c5ccc(NC6CCC(=O)NC6=O)cc5F)CC4)CC3)ccc21	C40H46F4N6O3	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-U6E20F	SCHEMBL25436618	3-[4-[4-[[1-[[1-Butyl-3-[4-(trifluoromethoxy)phenyl]indol-5-yl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-fluoroanilino]piperidine-2,6-dione	CCCCn1cc(-c2ccc(OC(F)(F)F)cc2)c2cc(CN3CCC(CN4CCN(c5ccc(NC6CCC(=O)NC6=O)cc5F)CC4)CC3)ccc21	C41H48F4N6O3	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-836LTU	SCHEMBL25424397	5-[4-[[1-[[1-(1,3-Dioxolan-2-ylmethyl)-3-[4-(trifluoromethoxy)phenyl]indol-5-yl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	O=C1CCC(N2C(=O)c3ccc(N4CCN(CC5CCN(Cc6ccc7c(c6)c(-c6ccc(OC(F)(F)F)cc6)cn7CC6OCCO6)CC5)CC4)cc3C2=O)C(=O)N1	C43H45F3N6O7	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-D3OZVL	WO2023130012A1_57	.	CC(C)CCCn1cc(-c2ccc(OC(F)(F)F)cc2)c2cc(CN3CCC(CN4CCN(c5ccc6c(c5)C(=O)C(C5CCC(=O)NC5=O)C6=O)CC4)CC3)ccc21	C46H52F3N5O5	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-9X1YLZ	SCHEMBL25426505	3-[4-[4-[[1-[[1-[3-(Dimethylamino)propyl]-3-[4-(trifluoromethoxy)phenyl]indol-5-yl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-fluoroanilino]piperidine-2,6-dione	CN(C)CCCn1cc(-c2ccc(OC(F)(F)F)cc2)c2cc(CN3CCC(CN4CCN(c5ccc(NC6CCC(=O)NC6=O)cc5F)CC4)CC3)ccc21	C42H51F4N7O3	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-8BC4TH	SCHEMBL30488064	5-[4-[1-[[1-(3-Aminopropyl)-3-[4-(trifluoromethoxy)phenyl]indol-5-yl]methyl]piperidin-4-yl]piperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	NCCCn1cc(-c2ccc(OC(F)(F)F)cc2)c2cc(CN3CCC(C4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)ccc21	C42H45F3N6O5	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-W86CGB	WO2023130012A1_60	.	CN(C)CCCn1cc(-c2ccc(OC(F)(F)F)cc2)c2cc(CN3CCC(C4CCN(c5ccc(NC6CCC(=O)NC6=O)cc5F)CC4)CC3)ccc21	C42H50F4N6O3	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-VOKHS2	SCHEMBL25422705	4-amino-N-[3-[5-[[4-[[4-[4-[(2,6-dioxopiperidin-3-yl)amino]-2-fluorophenyl]piperazin-1-yl]methyl]piperidin-1-yl]methyl]-3-[4-(trifluoromethoxy)phenyl]indol-1-yl]propyl]piperidine-4-carboxamide	NC1(C(=O)NCCCn2cc(-c3ccc(OC(F)(F)F)cc3)c3cc(CN4CCC(CN5CCN(c6ccc(NC7CCC(=O)NC7=O)cc6F)CC5)CC4)ccc32)CCNCC1	C46H57F4N9O4	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-K8H6HP	WO2023130012A1_62	.	CN(C)S(=O)(=O)n1cc(-c2ccc(OC(F)(F)F)cc2)c2cc(CN3CCC(CN4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)ccc21	C41H44F3N7O7S	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-L12WVQ	SCHEMBL25427389	3-[3-Fluoro-4-[4-[[1-[[1-(4-methylpentyl)-3-[4-(trifluoromethoxy)phenyl]indol-5-yl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]anilino]piperidine-2,6-dione; SCHEMBL30488055	CC(C)CCCn1cc(-c2ccc(OC(F)(F)F)cc2)c2cc(CN3CCC(CN4CCN(c5ccc(NC6CCC(=O)NC6=O)cc5F)CC4)CC3)ccc21	C43H52F4N6O3	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-8Y3A4W	WO2023130012A1_64	.	O=C1CCC(Nc2ccc(N3CCN(CC4CCN(Cc5ccc6[nH]cc(-c7ccc(OC(F)(F)F)cc7)c6c5)CC4)CC3)c(F)c2)C(=O)N1	C37H40F4N6O3	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-2KW4AP	SCHEMBL30488085	3-[3-fluoro-4-[4-[1-[[3-[4-(trifluoromethoxy)phenyl]-1H-indol-5-yl]methyl]piperidin-4-yl]piperidin-1-yl]anilino]piperidine-2,6-dione	O=C1CCC(Nc2ccc(N3CCC(C4CCN(Cc5ccc6[nH]cc(-c7ccc(OC(F)(F)F)cc7)c6c5)CC4)CC3)c(F)c2)C(=O)N1	C37H39F4N5O3	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-OVFSMD	SCHEMBL30488086	5-[2-[[1-(3-Aminopropyl)-3-[4-(trifluoromethoxy)phenyl]indol-5-yl]methyl]-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-5-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	NCCCn1cc(-c2ccc(OC(F)(F)F)cc2)c2cc(CN3CC4CN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4C3)ccc21	C38H37F3N6O5	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-QMSGH2	SCHEMBL25437406	3-[4-[2-[[1-(3-Aminopropyl)-3-[4-(trifluoromethoxy)phenyl]indol-5-yl]methyl]-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-5-yl]-3-fluoroanilino]piperidine-2,6-dione	NCCCn1cc(-c2ccc(OC(F)(F)F)cc2)c2cc(CN3CC4CN(c5ccc(NC6CCC(=O)NC6=O)cc5F)CC4C3)ccc21	C36H38F4N6O3	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-U30EXG	WO2023130012A1_68	.	COC(CCn1cc(-c2ccc(OC(F)(F)F)cc2)c2cc(CN3CCC(CN4CCN(c5ccc6c(c5)C(=O)N(C5=CCC(=O)NC5=O)C6=O)CC4)CC3)ccc21)OC	C44H47F3N6O7	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-KR89CB	SCHEMBL25425989	5-[2-[[1-[3-(Dimethylamino)propyl]-3-[4-(trifluoromethoxy)phenyl]indol-5-yl]methyl]-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-5-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN(C)CCCn1cc(-c2ccc(OC(F)(F)F)cc2)c2cc(CN3CC4CN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4C3)ccc21	C40H41F3N6O5	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-HVMU8E	SCHEMBL30488071	5-[3-[1-[[1-(3-Aminopropyl)-3-[4-(trifluoromethoxy)phenyl]indol-5-yl]methyl]azetidin-3-yl]azetidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	NCCCn1cc(-c2ccc(OC(F)(F)F)cc2)c2cc(CN3CC(C4CN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)C3)ccc21	C38H37F3N6O5	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-VNBACB	SCHEMBL30488059	5-[4-[1-[[1-[3-(Dimethylamino)propyl]-3-[4-(trifluoromethoxy)phenyl]indol-5-yl]methyl]piperidin-4-yl]piperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN(C)CCCn1cc(-c2ccc(OC(F)(F)F)cc2)c2cc(CN3CCC(C4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)ccc21	C44H49F3N6O5	KRAS	P01116	CRBN	WO-2023130012-A1
TPD-IGTKVZ	WO2023130012A1_72	.	Cc1ncsc1-c1ccc(C(C)NC(=O)C2C[C@@H](O)CN2C(=O)C(NC(=O)CN2CCN(CC3CCN(Cc4ccc5c(c4)c(-c4ccc(OC(F)(F)F)cc4)cn5CCCN)CC3)CC2)C(C)(C)C)cc1	C54H70F3N9O5S	KRAS	P01116	VHL	WO-2023130012-A1
TPD-D3G4BA	WO2023131118A1_BCL-03146	.	CC(=O)C1=C(NC[C@H]2CC[C@H](N3CCN(CC4=CC5=C(CN(C6CCC(=O)NC6=O)C5=O)C(Br)=C4)CC3)CC2)C=CC(S(=O)(=O)NC(=O)C2=CC=C(N3CCN(CC4=C(C5=CC=C(Cl)C=C5)CC(C)(C)CC4)CC3)C=C2OC2=CN=C3NC=CC3=C2)=C1	C66H74BrClN10O8S	BCL2L1	Q07817	CRBN	WO-2023131118-A1
TPD-EXME68	WO2023131118A1_BCL-03147	.	CC(=O)C1=C(NC[C@H]2CC[C@H](N3CCN(CC4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5)CC3)CC2)C=CC(S(=O)(=O)NC(=O)C2=CC=C(N3CCN(CC4=C(C5=CC=C(Cl)C=C5)CC(C)(C)CC4)CC3)C=C2OC2=CN=C3NC=CC3=C2)=C1	C66H75ClN10O8S	BCL2L1	Q07817	CRBN	WO-2023131118-A1
TPD-8MEOXO	WO2023131118A1_BCL-03148	.	CC(=O)C1=C(NC[C@H]2CC[C@@H](N3CCN(CC4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5)CC3)CC2)C=CC(S(=O)(=O)NC(=O)C2=CC=C(N3CCN(CC4=C(C5=CC=C(Cl)C=C5)CC(C)(C)CC4)CC3)C=C2OC2=CN=C3NC=CC3=C2)=C1	C66H75ClN10O8S	BCL2L1	Q07817	CRBN	WO-2023131118-A1
TPD-68OVTN	WO2023131118A1_BCL-03149	.	CC(=O)C1=C(NC[C@H]2CC[C@@H](N3CCN(CC4=CC5=C(CN(C6CCC(=O)NC6=O)C5=O)C(Br)=C4)CC3)CC2)C=CC(S(=O)(=O)NC(=O)C2=CC=C(N3CCN(CC4=C(C5=CC=C(Cl)C=C5)CC(C)(C)CC4)CC3)C=C2OC2=CN=C3NC=CC3=C2)=C1	C66H74BrClN10O8S	BCL2L1	Q07817	CRBN	WO-2023131118-A1
TPD-14LPQD	WO2023131118A1_BCL-03165	.	CC(=O)C1=C(NC[C@H]2CC[C@@H](N3CCN(CC4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5)[C@@H](C)C3)CC2)C=CC(S(=O)(=O)NC(=O)C2=CC=C(N3CCN(CC4=C(C5=CC=C(Cl)C=C5)CC(C)(C)CC4)CC3)C=C2OC2=CN=C3NC=CC3=C2)=C1	C67H77ClN10O8S	BCL2L1	Q07817	CRBN	WO-2023131118-A1
TPD-NZ51FX	WO2023131118A1_BCL-03166	.	CC(=O)C1=C(NC[C@H]2CC[C@H](N3CCN(CC4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5)[C@@H](C)C3)CC2)C=CC(S(=O)(=O)NC(=O)C2=CC=C(N3CCN(CC4=C(C5=CC=C(Cl)C=C5)CC(C)(C)CC4)CC3)C=C2OC2=CN=C3NC=CC3=C2)=C1	C67H77ClN10O8S	BCL2L1	Q07817	CRBN	WO-2023131118-A1
TPD-9RZI8D	WO2023131118A1_BCL-03167	.	CC(=O)C1=C(NC[C@H]2CC[C@@H](N3CCN(CC4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5)[C@H](C)C3)CC2)C=CC(S(=O)(=O)NC(=O)C2=CC=C(N3CCN(CC4=C(C5=CC=C(Cl)C=C5)CC(C)(C)CC4)CC3)C=C2OC2=CN=C3NC=CC3=C2)=C1	C67H77ClN10O8S	BCL2L1	Q07817	CRBN	WO-2023131118-A1
TPD-VP2KT6	WO2023131118A1_BCL-03168	.	CC(=O)C1=C(NC[C@H]2CC[C@H](N3CCN(CC4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5)[C@H](C)C3)CC2)C=CC(S(=O)(=O)NC(=O)C2=CC=C(N3CCN(CC4=C(C5=CC=C(Cl)C=C5)CC(C)(C)CC4)CC3)C=C2OC2=CN=C3NC=CC3=C2)=C1	C67H77ClN10O8S	BCL2L1	Q07817	CRBN	WO-2023131118-A1
TPD-CYC76Y	WO2023131118A1_BCL-03169	.	CC(=O)C1=C(NC[C@H]2CC[C@@H](N3CCN(CC4=CC5=C(CN(C6CCC(=O)NC6=O)C5=O)C(Br)=C4)[C@@H](C)C3)CC2)C=CC(S(=O)(=O)NC(=O)C2=CC=C(N3CCN(CC4=C(C5=CC=C(Cl)C=C5)CC(C)(C)CC4)CC3)C=C2OC2=CN=C3NC=CC3=C2)=C1	C67H76BrClN10O8S	BCL2L1	Q07817	CRBN	WO-2023131118-A1
TPD-D20P7Y	WO2023131118A1_BCL-03170	.	CC(=O)C1=C(NC[C@H]2CC[C@H](N3CCN(CC4=CC5=C(CN(C6CCC(=O)NC6=O)C5=O)C(Br)=C4)[C@@H](C)C3)CC2)C=CC(S(=O)(=O)NC(=O)C2=CC=C(N3CCN(CC4=C(C5=CC=C(Cl)C=C5)CC(C)(C)CC4)CC3)C=C2OC2=CN=C3NC=CC3=C2)=C1	C67H76BrClN10O8S	BCL2L1	Q07817	CRBN	WO-2023131118-A1
TPD-1EKCCO	WO2023131118A1_BCL-03171	.	CC(=O)C1=C(NC[C@H]2CC[C@@H](N3CCN(CC4=CC5=C(CN(C6CCC(=O)NC6=O)C5=O)C(Br)=C4)[C@H](C)C3)CC2)C=CC(S(=O)(=O)NC(=O)C2=CC=C(N3CCN(CC4=C(C5=CC=C(Cl)C=C5)CC(C)(C)CC4)CC3)C=C2OC2=CN=C3NC=CC3=C2)=C1	C67H76BrClN10O8S	BCL2L1	Q07817	CRBN	WO-2023131118-A1
TPD-NCCFBE	WO2023131118A1_BCL-03172	.	CC(=O)C1=C(NC[C@H]2CC[C@H](N3CCN(CC4=CC5=C(CN(C6CCC(=O)NC6=O)C5=O)C(Br)=C4)[C@H](C)C3)CC2)C=CC(S(=O)(=O)NC(=O)C2=CC=C(N3CCN(CC4=C(C5=CC=C(Cl)C=C5)CC(C)(C)CC4)CC3)C=C2OC2=CN=C3NC=CC3=C2)=C1	C67H76BrClN10O8S	BCL2L1	Q07817	CRBN	WO-2023131118-A1
TPD-UW6CCJ	SCHEMBL31202792	4-[4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[(2R)-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]methyl]piperazin-1-yl]-1-phenylsulfanylbutan-2-yl]amino]-3-(trifluoromethylsulfonyl)phenyl]sulfonylbenzamide	CC1(C)CCC(C2=CC=C(Cl)C=C2)=C(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC=C(N[C@H](CCN5CCN(CC6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)CC5)CSC5=CC=CC=C5)C(S(=O)(=O)C(F)(F)F)=C4)C=C3)CC2)C1	C61H68ClF3N8O8S3	BCL2L1	Q07817	CRBN	WO-2023131118-A1
TPD-8U767N	SCHEMBL25333338	N-[4-[[(2R)-4-[4-[[7-bromo-2-(2,6-dioxopiperidin-3-yl)-3-oxo-1H-isoindol-5-yl]methyl]piperazin-1-yl]-1-phenylsulfanylbutan-2-yl]amino]-3-(trifluoromethylsulfonyl)phenyl]sulfonyl-4-[4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]benzamide	CC1(C)CCC(C2=CC=C(Cl)C=C2)=C(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC=C(N[C@H](CCN5CCN(CC6=CC7=C(CN(C8CCC(=O)NC8=O)C7=O)C(Br)=C6)CC5)CSC5=CC=CC=C5)C(S(=O)(=O)C(F)(F)F)=C4)C=C3)CC2)C1	C61H67BrClF3N8O8S3	BCL2L1	Q07817	CRBN	WO-2023131118-A1
TPD-6315VK	SCHEMBL25331436	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]methyl]piperazin-1-yl]cyclohexyl]methylamino]-3-(trifluoromethylsulfonyl)phenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide; SCHEMBL25331454; SCHEMBL30484924	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC(S(=O)(=O)C(F)(F)F)=C(NC[C@H]5CC[C@H](N6CCN(CC7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8)CC6)CC5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C65H72ClF3N10O9S2	BCL2L1	Q07817	CRBN	WO-2023131118-A1
TPD-FI0Z1O	SCHEMBL31202892	4-[4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]methyl]piperazin-1-yl]cyclohexyl]methylamino]-3-(trifluoromethylsulfonyl)phenyl]sulfonylbenzamide	CC1(C)CCC(C2=CC=C(Cl)C=C2)=C(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC(S(=O)(=O)C(F)(F)F)=C(NC[C@H]5CC[C@H](N6CCN(CC7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8)CC6)CC5)C=C4)C=C3)CC2)C1	C58H68ClF3N8O8S2	BCL2L1	Q07817	CRBN	WO-2023131118-A1
TPD-NQ661A	SCHEMBL25333423	4-[4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]methyl]piperazin-1-yl]cyclohexyl]methylamino]-3-nitrophenyl]sulfonylbenzamide; SCHEMBL25333446; SCHEMBL30485141	CC1(C)CCC(C2=CC=C(Cl)C=C2)=C(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NC[C@H]5CC[C@H](N6CCN(CC7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8)CC6)CC5)C=C4)C=C3)CC2)C1	C57H68ClN9O8S	BCL2L1	Q07817	CRBN	WO-2023131118-A1
TPD-XJZ2O7	SCHEMBL25333891	N-[4-[[4-[4-[[7-bromo-2-(2,6-dioxopiperidin-3-yl)-3-oxo-1H-isoindol-5-yl]methyl]piperazin-1-yl]cyclohexyl]methylamino]-3-(trifluoromethylsulfonyl)phenyl]sulfonyl-4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide; SCHEMBL25333910; SCHEMBL30484936	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC(S(=O)(=O)C(F)(F)F)=C(NC[C@H]5CC[C@H](N6CCN(CC7=CC8=C(CN(C9CCC(=O)NC9=O)C8=O)C(Br)=C7)CC6)CC5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C65H71BrClF3N10O9S2	BCL2L1	Q07817	CRBN	WO-2023131118-A1
TPD-HV6H53	SCHEMBL31202699	N-[4-[[4-[4-[[7-bromo-2-(2,6-dioxopiperidin-3-yl)-3-oxo-1H-isoindol-5-yl]methyl]piperazin-1-yl]cyclohexyl]methylamino]-3-(trifluoromethylsulfonyl)phenyl]sulfonyl-4-[4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]benzamide	CC1(C)CCC(C2=CC=C(Cl)C=C2)=C(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC(S(=O)(=O)C(F)(F)F)=C(NC[C@H]5CC[C@H](N6CCN(CC7=CC8=C(CN(C9CCC(=O)NC9=O)C8=O)C(Br)=C7)CC6)CC5)C=C4)C=C3)CC2)C1	C58H67BrClF3N8O8S2	BCL2L1	Q07817	CRBN	WO-2023131118-A1
TPD-0RB0P0	SCHEMBL31202775	N-[4-[[4-[4-[[7-bromo-2-(2,6-dioxopiperidin-3-yl)-3-oxo-1H-isoindol-5-yl]methyl]piperazin-1-yl]cyclohexyl]methylamino]-3-nitrophenyl]sulfonyl-4-[4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]benzamide	CC1(C)CCC(C2=CC=C(Cl)C=C2)=C(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NC[C@H]5CC[C@H](N6CCN(CC7=CC8=C(CN(C9CCC(=O)NC9=O)C8=O)C(Br)=C7)CC6)CC5)C=C4)C=C3)CC2)C1	C57H67BrClN9O8S	BCL2L1	Q07817	CRBN	WO-2023131118-A1
TPD-95I4GE	SCHEMBL25333244	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]methyl]piperazin-1-yl]cyclohexyl]methylamino]-3-(trifluoromethylsulfonyl)phenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide; SCHEMBL25333265; SCHEMBL30484933	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC(S(=O)(=O)C(F)(F)F)=C(NC[C@H]5CC[C@H](N6CCN(CC7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C65H70ClF3N10O10S2	BCL2L1	Q07817	CRBN	WO-2023131118-A1
TPD-NUZXTF	SCHEMBL30484929	4-[4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]methyl]piperazin-1-yl]cyclohexyl]methylamino]-3-(trifluoromethylsulfonyl)phenyl]sulfonylbenzamide	CC1(C)CCC(C2=CC=C(Cl)C=C2)=C(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC(S(=O)(=O)C(F)(F)F)=C(NC[C@H]5CC[C@H](N6CCN(CC7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)C=C4)C=C3)CC2)C1	C58H66ClF3N8O9S2	BCL2L1	Q07817	CRBN	WO-2023131118-A1
TPD-T5SRF1	SCHEMBL25334675	4-[4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]methyl]piperazin-1-yl]cyclohexyl]methylamino]-3-nitrophenyl]sulfonylbenzamide; SCHEMBL30484948	CC1(C)CCC(C2=CC=C(Cl)C=C2)=C(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NC[C@H]5CC[C@H](N6CCN(CC7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)C=C4)C=C3)CC2)C1	C57H66ClN9O9S	BCL2L1	Q07817	CRBN	WO-2023131118-A1
TPD-M5ACCX	WO2023131118A1_BCL-03188	.	CC(=O)C1=C(NC[C@H]2CC[C@H](N3CCN(CC4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)C=CC(S(=O)(=O)NC(=O)C2=CC=C(N3CCN(CC4=C(C5=CC=C(Cl)C=C5)CC(C)(C)CC4)CC3)C=C2OC2=CN=C3NC=CC3=C2)=C1	C66H73ClN10O9S	BCL2L1	Q07817	CRBN	WO-2023131118-A1
TPD-XXP74O	SCHEMBL31202687	4-[4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[(2R)-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]methyl]piperazin-1-yl]-1-phenylsulfanylbutan-2-yl]amino]-3-(trifluoromethylsulfonyl)phenyl]sulfonylbenzamide	CC1(C)CCC(C2=CC=C(Cl)C=C2)=C(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC(S(=O)(=O)C(F)(F)F)=C(N[C@H](CCN5CCN(CC6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CSC5=CC=CC=C5)C=C4)C=C3)CC2)C1	C61H66ClF3N8O9S3	BCL2L1	Q07817	CRBN	WO-2023131118-A1
TPD-ER1A4Y	WO2023131118A1_BCL-03190	.	CC(=O)C1=C(NC[C@H]2CC[C@@H](N3CCN(CC4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)[C@@H](C)C3)CC2)C=CC(S(=O)(=O)NC(=O)C2=CC=C(N3CCN(CC4=C(C5=CC=C(Cl)C=C5)CC(C)(C)CC4)CC3)C=C2OC2=CN=C3NC=CC3=C2)=C1	C67H75ClN10O9S	BCL2L1	Q07817	CRBN	WO-2023131118-A1
TPD-F4M7CY	WO2023138524A1_1	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)CCCCCCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)NCc6ccc(-c7scnc7C)cc6)C(C)(C)C)CC5)nc4c3F)c12	C60H70F2N10O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-G1Z56S	WO2023138524A1_2	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCCN(C)CC2(COc3nc(N4CC5CCC(C4)N5)c4ccc(-c5cc(O)cc6ccccc56)c(F)c4n3)CC2)C(C)(C)C)cc1	C60H74FN9O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-L47RKZ	WO2023138524A1_3	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)CCCCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)NCc6ccc(-c7scnc7C)cc6)C(C)(C)C)CC5)nc4c3F)c12	C58H66F2N10O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-94BGAP	WO2023138524A1_4	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCOCCCN2CCC[C@H]2COc2nc(N3CC4CCC(C3)N4)c3ccc(-c4cc(O)cc5ccccc45)c(F)c3n2)C(C)(C)C)cc1	C57H68FN9O7S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-SS644U	WO2023138524A1_5	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)CCCCCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)NCc6ccc(-c7scnc7C)cc6)C(C)(C)C)CC5)nc4c3F)c12	C59H68F2N10O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-16SJ4L	WO2023138524A1_6	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)c2ccc(C(=O)N3CC4(CCN(CC5(COc6nc(N7CC8CCC(C7)N8)c7cnc(-c8cc(O)cc9ccc(F)c(F)c89)c(F)c7n6)CC5)CC4)C3)cc2)C(C)(C)C)cc1	C65H70F3N11O7S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-LVN80C	WO2023138524A1_7	.	C#Cc1cccc2cc(O)cc(-c3ccc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)CCCCCCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)NCc6ccc(-c7scnc7C)cc6)C(C)(C)C)CC5)nc4c3F)c12	C61H72FN9O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-X0HM62	WO2023138524A1_8	.	C#Cc1cccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)CCCCCCCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)NCc6ccc(-c7scnc7C)cc6)C(C)(C)C)CC5)nc4c3F)c12	C61H73FN10O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-RX06NR	WO2023138524A1_9	.	CCCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(C#CC5(CNCCCCCCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)NCc6ccc(-c7scnc7C)cc6)C(C)(C)C)CC5)nc4c3F)c12	C61H72F2N10O5S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-20NR5F	WO2023138524A1_10	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)CCCCCCCCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)NCc6ccc(-c7scnc7C)cc6)C(C)(C)C)CC5)nc4c3F)c12	C62H74F2N10O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-813U34	WO2023138524A1_11	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(C#CC5(CN(C)CCCCCCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)NCc6ccc(-c7scnc7C)cc6)C(C)(C)C)CC5)nc4c3F)c12	C61H72F2N10O5S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-EV0F8L	WO2023138524A1_12	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCCCN(C)CCCCCCC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)NCc5ccc(-c6scnc6C)cc5)C(C)(C)C)nc4c3F)c12	C58H68F2N10O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-DE9VNB	WO2023138524A1_13	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)CCCCCCNC(=O)C[C@H](NC(=O)[C@@H]6C[C@@H](O)CN6C(=O)[C@@H](NC(=O)C6(C#N)CC6)C(C)(C)C)c6ccc(-c7scnc7C)cc6)CC5)nc4c3F)c12	C66H76F2N12O7S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-BEVOYG	WO2023138524A1_14	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)CCCCc6ccc(C(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)NCc7ccc(-c8scnc8C)cc7)C(C)(C)C)cc6)CC5)nc4c3F)c12	C64H70F2N10O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-BLP2CL	WO2023138524A1_15	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)CCCNC(=O)C[C@H](NC(=O)[C@@H]6C[C@@H](O)CN6C(=O)[C@@H](NC(=O)C6(C#N)CC6)C(C)(C)C)c6ccc(-c7scnc7C)cc6)CC5)nc4c3F)c12	C63H70F2N12O7S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-ZGRRXX	WO2023138524A1_16	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(OCc7ccc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)NCc8ccc(-c9scnc9C)cc8)C(C)(C)C)cc7)CC6)CC5)nc4c3F)c12	C65H70F2N10O7S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-YFPTTE	WO2023138524A1_17	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)CCOCCOCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)NCc6ccc(-c7scnc7C)cc6)C(C)(C)C)CC5)nc4c3F)c12	C59H68F2N10O8S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-6FD2Z6	WO2023138524A1_18	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(Oc7ccc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)NCc8ccc(-c9scnc9C)cc8)C(C)(C)C)cc7)CC6)CC5)nc4c3F)c12	C64H68F2N10O7S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-LUSJ2N	WO2023138524A1_19	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCCCCCCCCCCC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)NCc5ccc(-c6scnc6C)cc5)C(C)(C)C)nc4c3F)c12	C58H67F2N9O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-4IGFNN	WO2023138524A1_20	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)CCCCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)c6ccc(-c7scnc7C)cc6)C(C)(C)C)CC5)nc4c3F)c12	C59H68F2N10O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-NNZGLR	WO2023138524A1_21	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)CCCCCNC(=O)C[C@H](NC(=O)[C@@H]6C[C@@H](O)CN6C(=O)[C@@H](NC(=O)C6(C#N)CC6)C(C)(C)C)c6ccc(-c7scnc7C)cc6)CC5)nc4c3F)c12	C65H74F2N12O7S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-2NXLPV	WO2023138524A1_22	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)CCCCCNC(=O)C[C@H](NC(=O)[C@@H]6C[C@@H](O)CN6C(=O)[C@@H](c6cc(C)no6)C(C)C)c6ccc(-c7scnc7C)cc6)CC5)nc4c3F)c12	C63H71F2N11O7S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-FPPQFE	WO2023138524A1_23	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)CCCCCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)c6ccc(-c7scnc7C)cc6)C(C)(C)C)CC5)nc4c3F)c12	C60H70F2N10O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-HGT9A3	WO2023138524A1_25	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)CCCCCCNC(=O)C[C@H](NC(=O)[C@@H]6C[C@@H](O)CN6C(=O)[C@@H](c6cc(C)no6)C(C)C)c6ccc(-c7scnc7C)cc6)CC5)nc4c3F)c12	C64H73F2N11O7S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-N6L5ID	WO2023138524A1_26	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)CCCCCCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)c6ccc(-c7scnc7C)cc6)C(C)(C)C)CC5)nc4c3F)c12	C61H72F2N10O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-QLNKEH	WO2023138524A1_27	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)CCCCCCCNC(=O)C[C@H](NC(=O)[C@@H]6C[C@@H](O)CN6C(=O)[C@@H](NC(=O)C6(C#N)CC6)C(C)(C)C)c6ccc(-c7scnc7C)cc6)CC5)nc4c3F)c12	C67H78F2N12O7S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-9GA2W9	WO2023138524A1_28	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)CCCCCCCNC(=O)C[C@H](NC(=O)[C@@H]6C[C@@H](O)CN6C(=O)[C@@H](c6cc(C)no6)C(C)C)c6ccc(-c7scnc7C)cc6)CC5)nc4c3F)c12	C65H75F2N11O7S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-UNCKK8	WO2023138524A1_29	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)CCCCCCCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)c6ccc(-c7scnc7C)cc6)C(C)(C)C)CC5)nc4c3F)c12	C62H74F2N10O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-63K0RG	WO2023138524A1_30	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)CCCCCCCCNC(=O)C[C@H](NC(=O)[C@@H]6C[C@@H](O)CN6C(=O)[C@@H](NC(=O)C6(C#N)CC6)C(C)(C)C)c6ccc(-c7scnc7C)cc6)CC5)nc4c3F)c12	C68H80F2N12O7S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-IIT3FZ	WO2023138524A1_31	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)CCCCCCCCNC(=O)C[C@H](NC(=O)[C@@H]6C[C@@H](O)CN6C(=O)[C@@H](c6cc(C)no6)C(C)C)c6ccc(-c7scnc7C)cc6)CC5)nc4c3F)c12	C66H77F2N11O7S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-OWQHXI	WO2023138524A1_32	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)CCCCCCCCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)c6ccc(-c7scnc7C)cc6)C(C)(C)C)CC5)nc4c3F)c12	C63H76F2N10O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-IF5HIJ	WO2023138524A1_33	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)CCCCCCCCCNC(=O)C[C@H](NC(=O)[C@@H]6C[C@@H](O)CN6C(=O)[C@@H](NC(=O)C6(C#N)CC6)C(C)(C)C)c6ccc(-c7scnc7C)cc6)CC5)nc4c3F)c12	C69H82F2N12O7S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-N4X39A	WO2023138524A1_34	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)CCCCCCCCCNC(=O)C[C@H](NC(=O)[C@@H]6C[C@@H](O)CN6C(=O)[C@@H](c6cc(C)no6)C(C)C)c6ccc(-c7scnc7C)cc6)CC5)nc4c3F)c12	C67H79F2N11O7S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-IWPG6B	WO2023138524A1_35	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)CCCCCCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)c6ccc(-c7scnc7C)cc6)C(C)C)CC5)nc4c3F)c12	C60H70F2N10O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-WW2DM5	WO2023138524A1_36	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)CCCCCCCCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)c6ccc(-c7scnc7C)cc6)C(C)C)CC5)nc4c3F)c12	C62H74F2N10O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-7TSALJ	WO2023138524A1_37	.	C#Cc1ccc([C@H](CC(=O)NCCCCCCCN(C)CC2(COc3nc(N4CC5CCC(C4)N5)c4cnc(-c5cc(O)cc6ccc(F)c(C#C)c56)c(F)c4n3)CC2)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](c2cc(C)no2)C(C)C)cc1	C63H72F2N10O7	KRAS	P01116	VHL	WO-2023138524-A1
TPD-Y54Y9K	WO2023138524A1_38	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)CCCCCCCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)c6ccc(-c7scnc7C)cc6)C(C)C)CC5)nc4c3F)c12	C61H72F2N10O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-WJZ2EO	WO2023138524A1_39	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)CCCCCCCNC(=O)C[C@H](NC(=O)[C@@H]6C[C@@H](O)CN6C(=O)[C@@H](c6cc(C)no6)C(C)C)c6ccc(C#N)cc6)CC5)nc4c3F)c12	C62H71F2N11O7	KRAS	P01116	VHL	WO-2023138524-A1
TPD-CB9R0M	WO2023138524A1_45	.	C#Cc1cccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)CCCCCCCNC(=O)C[C@H](NC(=O)[C@@H]6C[C@@H](O)CN6C(=O)[C@@H](c6cc(C)no6)C(C)C)c6ccc(-c7scnc7C)cc6)CC5)nc4c3F)c12	C65H76FN11O7S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-R9KCPU	WO2023138524A1_46	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCN(C)CC2(COc3nc(N4CC5CCC(C4)N5)c4cnc(-c5cc(O)cc6ccc(F)c(F)c56)c(F)c4n3)CC2)C(C)(C)C)cc1	C59H71F3N10O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-XFI7BH	WO2023138524A1_47	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCN(C)CC2(COc3nc(N4CC5CCC(C4)N5)c4cnc(-c5cc(O)cc6ccc(F)c(F)c56)c(F)c4n3)CC2)C(C)(C)C)cc1	C58H69F3N10O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-Z8C3LB	WO2023138524A1_48	.	Cc1ncsc1-c1ccc([C@H](CC(=O)NCCCCCCCN(C)CC2(COc3nc(N4CC5CCC(C4)N5)c4cnc(-c5cc(O)cc6ccc(F)c(F)c56)c(F)c4n3)CC2)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(C#N)CC2)C(C)(C)C)cc1	C65H77F3N12O7S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-47OZ57	WO2023138524A1_49	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCCN(C)CC2(COc3nc(N4CC5CCC(C4)N5)c4cnc(-c5cc(O)cc6ccc(F)c(F)c56)c(F)c4n3)CC2)C(C)(C)C)cc1	C60H73F3N10O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-CMLPH0	WO2023138524A1_50	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCCN(C)CC2(COc3nc(N4CC5CCC(C4)N5)c4cnc(-c5cc(O)cc6ccc(F)c(F)c56)c(F)c4n3)CC2)C(C)C)cc1	C59H71F3N10O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-LUU7DQ	WO2023138524A1_51	.	Cc1cc([C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](CC(=O)NCCCCCCCN(C)CC2(COc3nc(N4CC5CCC(C4)N5)c4cnc(-c5cc(O)cc6ccc(F)c(F)c56)c(F)c4n3)CC2)c2ccc(-c3scnc3C)cc2)C(C)C)on1	C63H74F3N11O7S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-V3R6UH	WO2023138524A1_52	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)CCCCCCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)c6ccc(-c7scnc7C)cc6)C(C)(C)C)CC5)nc4c3F)c12	C61H76F2N10O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-RIKP4B	WO2023138524A1_53	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)CCCCCCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)NCc6ccc(-c7scnc7C)cc6)C(C)(C)C)CC5)nc4c3F)c12	C60H74F2N10O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-M3VZ4O	WO2023138524A1_54	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)CCCCCCCNC(=O)C[C@H](NC(=O)[C@@H]6C[C@@H](O)CN6C(=O)[C@@H](NC(=O)C6(C#N)CC6)C(C)(C)C)c6ccc(-c7scnc7C)cc6)CC5)nc4c3F)c12	C67H82F2N12O7S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-QUSL8X	WO2023138524A1_55	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)CCCCCCCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)c6ccc(-c7scnc7C)cc6)C(C)(C)C)CC5)nc4c3F)c12	C62H78F2N10O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-03RGTP	WO2023138524A1_56	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)CCCCCCCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)c6ccc(-c7scnc7C)cc6)C(C)C)CC5)nc4c3F)c12	C61H76F2N10O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-JRUGTW	WO2023138524A1_57	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)CCCCCCCNC(=O)C[C@H](NC(=O)[C@@H]6C[C@@H](O)CN6C(=O)[C@@H](c6cc(C)no6)C(C)C)c6ccc(-c7scnc7C)cc6)CC5)nc4c3F)c12	C65H79F2N11O7S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-4S9ACT	WO2023138524A1_60	.	C#Cc1c(F)ccc2cc(O)cc(-c3ccc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)CCCCCCCNC(=O)C[C@H](NC(=O)[C@@H]6C[C@@H](O)CN6C(=O)[C@@H](NC(=O)C6(C#N)CC6)C(C)(C)C)c6ccc(-c7scnc7C)cc6)CC5)nc4c3F)c12	C68H79F2N11O7S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-RTPWPC	WO2023138524A1_61	.	C#Cc1c(F)ccc2cc(O)cc(-c3ccc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)CCCCCCCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)c6ccc(-c7scnc7C)cc6)C(C)(C)C)CC5)nc4c3F)c12	C63H75F2N9O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-QVG565	WO2023138524A1_62	.	C#Cc1c(F)ccc2cc(O)cc(-c3ccc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)CCCCCCCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)c6ccc(-c7scnc7C)cc6)C(C)C)CC5)nc4c3F)c12	C62H73F2N9O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-H9YNN1	WO2023138524A1_63	.	C#Cc1c(F)ccc2cc(O)cc(-c3ccc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)CCCCCCCNC(=O)C[C@H](NC(=O)[C@@H]6C[C@@H](O)CN6C(=O)[C@@H](c6cc(C)no6)C(C)C)c6ccc(-c7scnc7C)cc6)CC5)nc4c3F)c12	C66H76F2N10O7S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-6CVT8S	WO2023138524A1_64	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(C#CC5(CN(C)CCCCCCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)c6ccc(-c7scnc7C)cc6)C(C)(C)C)CC5)nc4c3F)c12	C62H70F2N10O5S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-XAOJG0	WO2023138524A1_65	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(C#CC5(CN(C)CCCCCCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)NCc6ccc(-c7scnc7C)cc6)C(C)(C)C)CC5)nc4c3F)c12	C61H68F2N10O5S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-LKIOTF	WO2023138524A1_66	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(C#CC5(CN(C)CCCCCCCNC(=O)C[C@H](NC(=O)[C@@H]6C[C@@H](O)CN6C(=O)[C@@H](NC(=O)C6(C#N)CC6)C(C)(C)C)c6ccc(-c7scnc7C)cc6)CC5)nc4c3F)c12	C68H76F2N12O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-IAZG09	WO2023138524A1_67	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(C#CC5(CN(C)CCCCCCCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)c6ccc(-c7scnc7C)cc6)C(C)(C)C)CC5)nc4c3F)c12	C63H72F2N10O5S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-EUCLR9	WO2023138524A1_68	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(C#CC5(CN(C)CCCCCCCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)c6ccc(-c7scnc7C)cc6)C(C)C)CC5)nc4c3F)c12	C62H70F2N10O5S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-NG67I3	WO2023138524A1_69	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(C#CC5(CN(C)CCCCCCCNC(=O)C[C@H](NC(=O)[C@@H]6C[C@@H](O)CN6C(=O)[C@@H](c6cc(C)no6)C(C)C)c6ccc(-c7scnc7C)cc6)CC5)nc4c3F)c12	C66H73F2N11O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-TTMVS5	WO2023138524A1_70	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCN(C)CC2(COc3nc(N4CC5CCC(C4)N5)c4cc(Cl)c(-c5ccc(F)c6sc(N)c(C#N)c56)c(F)c4n3)CC2)C(C)(C)C)cc1	C59H70ClF2N11O5S2	KRAS	P01116	VHL	WO-2023138524-A1
TPD-6RP6W0	WO2023138524A1_71	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCN(C)CC2(COc3nc(N4CC5CCC(C4)N5)c4cc(Cl)c(-c5ccc(F)c6sc(N)c(C#N)c56)c(F)c4n3)CC2)C(C)(C)C)cc1	C58H68ClF2N11O5S2	KRAS	P01116	VHL	WO-2023138524-A1
TPD-22G8UF	WO2023138524A1_72	.	Cc1ncsc1-c1ccc([C@H](CC(=O)NCCCCCCCN(C)CC2(COc3nc(N4CC5CCC(C4)N5)c4cc(Cl)c(-c5ccc(F)c6sc(N)c(C#N)c56)c(F)c4n3)CC2)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(C#N)CC2)C(C)(C)C)cc1	C65H76ClF2N13O6S2	KRAS	P01116	VHL	WO-2023138524-A1
TPD-WZZLEA	WO2023138524A1_73	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCCN(C)CC2(COc3nc(N4CC5CCC(C4)N5)c4cc(Cl)c(-c5ccc(F)c6sc(N)c(C#N)c56)c(F)c4n3)CC2)C(C)(C)C)cc1	C60H72ClF2N11O5S2	KRAS	P01116	VHL	WO-2023138524-A1
TPD-RZ25IV	WO2023138524A1_74	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCCN(C)CC2(COc3nc(N4CC5CCC(C4)N5)c4cc(Cl)c(-c5ccc(F)c6sc(N)c(C#N)c56)c(F)c4n3)CC2)C(C)C)cc1	C59H70ClF2N11O5S2	KRAS	P01116	VHL	WO-2023138524-A1
TPD-18OLIV	WO2023138524A1_75	.	Cc1cc([C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](CC(=O)NCCCCCCCN(C)CC2(COc3nc(N4CC5CCC(C4)N5)c4cc(Cl)c(-c5ccc(F)c6sc(N)c(C#N)c56)c(F)c4n3)CC2)c2ccc(-c3scnc3C)cc2)C(C)C)on1	C63H73ClF2N12O6S2	KRAS	P01116	VHL	WO-2023138524-A1
TPD-Q5YGZ8	WO2023138524A1_76	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCN(C)CC2(C#Cc3nc(N4CC5CCC(C4)N5)c4cc(Cl)c(-c5ccc(F)c6sc(N)c(C#N)c56)c(F)c4n3)CC2)C(C)(C)C)cc1	C60H68ClF2N11O4S2	KRAS	P01116	VHL	WO-2023138524-A1
TPD-CRKIDT	WO2023138524A1_77	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCN(C)CC2(C#Cc3nc(N4CC5CCC(C4)N5)c4cc(Cl)c(-c5ccc(F)c6sc(N)c(C#N)c56)c(F)c4n3)CC2)C(C)(C)C)cc1	C59H66ClF2N11O4S2	KRAS	P01116	VHL	WO-2023138524-A1
TPD-W5HLKB	WO2023138524A1_78	.	Cc1ncsc1-c1ccc([C@H](CC(=O)NCCCCCCCN(C)CC2(C#Cc3nc(N4CC5CCC(C4)N5)c4cc(Cl)c(-c5ccc(F)c6sc(N)c(C#N)c56)c(F)c4n3)CC2)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(C#N)CC2)C(C)(C)C)cc1	C66H74ClF2N13O5S2	KRAS	P01116	VHL	WO-2023138524-A1
TPD-95P9W4	WO2023138524A1_79	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCCN(C)CC2(C#Cc3nc(N4CC5CCC(C4)N5)c4cc(Cl)c(-c5ccc(F)c6sc(N)c(C#N)c56)c(F)c4n3)CC2)C(C)(C)C)cc1	C61H70ClF2N11O4S2	KRAS	P01116	VHL	WO-2023138524-A1
TPD-5H5U3W	WO2023138524A1_80	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCCN(C)CC2(C#Cc3nc(N4CC5CCC(C4)N5)c4cc(Cl)c(-c5ccc(F)c6sc(N)c(C#N)c56)c(F)c4n3)CC2)C(C)C)cc1	C60H68ClF2N11O4S2	KRAS	P01116	VHL	WO-2023138524-A1
TPD-V4B2TW	WO2023138524A1_81	.	Cc1cc([C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](CC(=O)NCCCCCCCN(C)CC2(C#Cc3nc(N4CC5CCC(C4)N5)c4cc(Cl)c(-c5ccc(F)c6sc(N)c(C#N)c56)c(F)c4n3)CC2)c2ccc(-c3scnc3C)cc2)C(C)C)on1	C64H71ClF2N12O5S2	KRAS	P01116	VHL	WO-2023138524-A1
TPD-MK1ET4	WO2023138524A1_82	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC[C@@H]5CCCN5CCCCCCC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)c5ccc(-c6scnc6C)cc5)C(C)(C)C)nc4c3F)c12	C60H70F2N10O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-UD1TNT	WO2023138524A1_83	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC[C@@H]5CCCN5CCCCCCC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)c5ccc(-c6scnc6C)cc5)C(C)C)nc4c3F)c12	C59H68F2N10O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-JMOWW2	WO2023138524A1_84	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC[C@@H]5CCCN5CCCCCCCNC(=O)C[C@H](NC(=O)[C@@H]5C[C@@H](O)CN5C(=O)[C@@H](NC(=O)C5(C#N)CC5)C(C)(C)C)c5ccc(-c6scnc6C)cc5)nc4c3F)c12	C66H76F2N12O7S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-1VMLSZ	WO2023138524A1_85	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC[C@@H]5CCCN5CCCCCCCC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)c5ccc(-c6scnc6C)cc5)C(C)(C)C)nc4c3F)c12	C61H72F2N10O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-HF5F9R	WO2023138524A1_86	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC[C@@H]5CCCN5CCCCCCCC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)c5ccc(-c6scnc6C)cc5)C(C)C)nc4c3F)c12	C60H70F2N10O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-R1Y21C	WO2023138524A1_87	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC[C@@H]5CCCN5CCCCCCCNC(=O)C[C@H](NC(=O)[C@@H]5C[C@@H](O)CN5C(=O)[C@@H](c5cc(C)no5)C(C)C)c5ccc(-c6scnc6C)cc5)nc4c3F)c12	C64H73F2N11O7S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-B6X7WB	WO2023138524A1_88	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(CCc7ccc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)NCc8ccc(-c9scnc9C)cc8)C(C)(C)C)cc7)CC6)CC5)nc4c3F)c12	C66H72F2N10O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-1C78YV	WO2023138524A1_89	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(NCc7ccc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)NCc8ccc(-c9scnc9C)cc8)C(C)(C)C)cc7)CC6)CC5)nc4c3F)c12	C65H71F2N11O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-HD605P	WO2023138524A1_90	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(N(C)Cc7ccc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)NCc8ccc(-c9scnc9C)cc8)C(C)(C)C)cc7)CC6)CC5)nc4c3F)c12	C66H73F2N11O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-HC1LG8	WO2023138524A1_91	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)CCCCOc6ccc(C(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)NCc7ccc(-c8scnc8C)cc7)C(C)(C)C)cc6)CC5)nc4c3F)c12	C64H70F2N10O7S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-R66TBE	WO2023138524A1_92	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(Cc7ccc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)NCc8ccc(-c9scnc9C)cc8)C(C)(C)C)cc7)CC6)CC5)nc4c3F)c12	C65H70F2N10O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-V128LZ	WO2023138524A1_93	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(Nc7ccc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)NCc8ccc(-c9scnc9C)cc8)C(C)(C)C)cc7)CC6)CC5)nc4c3F)c12	C64H69F2N11O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-0OAQRY	WO2023138524A1_94	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(N(C)c7ccc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)NCc8ccc(-c9scnc9C)cc8)C(C)(C)C)cc7)CC6)CC5)nc4c3F)c12	C65H71F2N11O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-ID8XUD	WO2023138524A1_95	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)CCCOc6ccc(C(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)NCc7ccc(-c8scnc8C)cc7)C(C)(C)C)cc6)CC5)nc4c3F)c12	C63H68F2N10O7S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-APQETG	WO2023138524A1_96	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)CCCCCc6ccc(C(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)NCc7ccc(-c8scnc8C)cc7)C(C)(C)C)cc6)CC5)nc4c3F)c12	C65H72F2N10O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-ZNV3U1	WO2023138524A1_97	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(CCCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)NCc7ccc(-c8scnc8C)cc7)C(C)(C)C)CC6)CC5)nc4c3F)c12	C64H76F2N10O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-7KVSRM	WO2023138524A1_98	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(CCC7CCN(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)NCc8ccc(-c9scnc9C)cc8)C(C)(C)C)CC7)CC6)CC5)nc4c3F)c12	C65H77F2N11O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-UPLN2Q	WO2023138524A1_99	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)CCN6CC7(CCN(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)NCc8ccc(-c9scnc9C)cc8)C(C)(C)C)CC7)C6)CC5)nc4c3F)c12	C63H74F2N12O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-D91ZT8	WO2023138524A1_100	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)CCCCCc6ccc(C(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)NCc7ccc(-c8scnc8C)cc7)C(C)(C)C)nc6)CC5)nc4c3F)c12	C64H71F2N11O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-EX63RO	WO2023138524A1_101	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)CCCCCc6ccc(C(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)NCc7ccc(-c8scnc8C)cc7)C(C)(C)C)cn6)CC5)nc4c3F)c12	C64H71F2N11O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-QO76FA	WO2023138524A1_102	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(CCN7CCC(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)NCc8ccc(-c9scnc9C)cc8)C(C)(C)C)CC7)CC6)CC5)nc4c3F)c12	C65H77F2N11O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-373P7V	WO2023138524A1_103	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)CCC6CN(c7ccc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)NCc8ccc(-c9scnc9C)cc8)C(C)(C)C)cc7)C6)CC5)nc4c3F)c12	C65H71F2N11O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-S1UVHC	WO2023138524A1_104	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)CCCCCc6cnc(C(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)NCc7ccc(-c8scnc8C)cc7)C(C)(C)C)n6C)CC5)nc4c3F)c12	C63H72F2N12O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-7GZPI2	WO2023138524A1_105	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)CCCCCc6cnc(C(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)NCc7ccc(-c8scnc8C)cc7)C(C)(C)C)s6)CC5)nc4c3F)c12	C62H69F2N11O6S2	KRAS	P01116	VHL	WO-2023138524-A1
TPD-W7B9RZ	WO2023138524A1_106	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)CCCCCc6cnc(C(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)NCc7ccc(-c8scnc8C)cc7)C(C)(C)C)o6)CC5)nc4c3F)c12	C62H69F2N11O7S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-R8R6XF	WO2023138524A1_107	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)CC6CN(c7ccc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)NCc8ccc(-c9scnc9C)cc8)C(C)(C)C)cc7)C6)CC5)nc4c3F)c12	C64H69F2N11O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-55TR00	WO2023138524A1_108	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC7(CC6)CN(c6ccc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)NCc8ccc(-c9scnc9C)cc8)C(C)(C)C)cc6)C7)CC5)nc4c3F)c12	C66H71F2N11O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-TX28IX	WO2023138524A1_109	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC7(CC6)CCN(c6ccc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)NCc8ccc(-c9scnc9C)cc8)C(C)(C)C)cc6)CC7)CC5)nc4c3F)c12	C68H75F2N11O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-K1AW2K	WO2023138524A1_110	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CC7(CCN(c8ccc(C(=O)N[C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)NCc9ccc(-c%10scnc%10C)cc9)C(C)(C)C)cc8)CC7)C6)CC5)nc4c3F)c12	C66H71F2N11O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-0KWG2T	WO2023138524A1_111	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC7(CC6)CCN(c6ccc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)NCc8ccc(-c9scnc9C)cc8)C(C)(C)C)nc6)CC7)CC5)nc4c3F)c12	C67H74F2N12O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-8E9RE4	WO2023138524A1_112	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC7(CC6)CN(c6ccc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)NCc8ccc(-c9scnc9C)cc8)C(C)(C)C)nc6)C7)CC5)nc4c3F)c12	C65H70F2N12O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-T86K6U	WO2023138524A1_113	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC7(CC6)CN(c6ccc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)NCc8ccc(-c9scnc9C)cc8)C(C)(C)C)cn6)C7)CC5)nc4c3F)c12	C65H70F2N12O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-1SMQG5	WO2023138524A1_114	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC7(CC6)CCN(c6ccc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)NCc8ccc(-c9scnc9C)cc8)C(C)(C)C)cn6)CC7)CC5)nc4c3F)c12	C67H74F2N12O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-PFIQFR	WO2023138524A1_115	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC7(CC6)CN(Cc6ccc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)NCc8ccc(-c9scnc9C)cc8)C(C)(C)C)cc6)C7)CC5)nc4c3F)c12	C67H73F2N11O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-RXWYIM	WO2023138524A1_116	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)Cc6ccc(N7CCC(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)NCc8ccc(-c9scnc9C)cc8)C(C)(C)C)CC7)cc6)CC5)nc4c3F)c12	C66H73F2N11O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-PD2LS4	WO2023138524A1_117	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)C6CCN(c7ccc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)NCc8ccc(-c9scnc9C)cc8)C(C)(C)C)cc7)CC6)CC5)nc4c3F)c12	C65H71F2N11O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-2NL1UW	WO2023138524A1_118	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)CC6CCN(c7ccc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)NCc8ccc(-c9scnc9C)cc8)C(C)(C)C)cc7)CC6)CC5)nc4c3F)c12	C66H73F2N11O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-5Q11HB	WO2023138524A1_119	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC7(CC6)CN(C(=O)c6ccc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)NCc8ccc(-c9scnc9C)cc8)C(C)(C)C)cc6)C7)CC5)nc4c3F)c12	C67H71F2N11O7S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-D2LUOG	WO2023138524A1_120	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)Cc6ccc(N7CCN(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)NCc8ccc(-c9scnc9C)cc8)C(C)(C)C)CC7)cc6)CC5)nc4c3F)c12	C65H72F2N12O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-KU8IN9	WO2023138524A1_121	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)Cc6ccc(N7CC(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)NCc8ccc(-c9scnc9C)cc8)C(C)(C)C)C7)cc6)CC5)nc4c3F)c12	C64H69F2N11O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-YSPT6S	WO2023138524A1_122	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)Cc6ccc(N7CCC(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)NCc8ccc(-c9scnc9C)cc8)C(C)(C)C)CC7)nc6)CC5)nc4c3F)c12	C65H72F2N12O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-SX9F64	WO2023138524A1_123	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)Cc6ccc(N7CCC(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)NCc8ccc(-c9scnc9C)cc8)C(C)(C)C)CC7)cn6)CC5)nc4c3F)c12	C65H72F2N12O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-R12YAU	WO2023138524A1_124	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)CC6CCN(c7cnc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)NCc8ccc(-c9scnc9C)cc8)C(C)(C)C)s7)CC6)CC5)nc4c3F)c12	C63H70F2N12O6S2	KRAS	P01116	VHL	WO-2023138524-A1
TPD-U9YVE4	WO2023138524A1_125	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)CC6CCN(c7csc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)NCc8ccc(-c9scnc9C)cc8)C(C)(C)C)n7)CC6)CC5)nc4c3F)c12	C63H70F2N12O6S2	KRAS	P01116	VHL	WO-2023138524-A1
TPD-GKOFD6	WO2023138524A1_126	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)C6CCC7(CC6)CN(c6ccc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)NCc8ccc(-c9scnc9C)cc8)C(C)(C)C)cc6)C7)CC5)nc4c3F)c12	C68H75F2N11O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-RY2ZMG	WO2023138524A1_127	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(OCc7ccc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)cc7)CC6)CC5)nc4c3F)c12	C66H72F2N10O7S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-X9ZTPH	WO2023138524A1_128	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)CC6CCN(c7cnc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)s7)CC6)CC5)nc4c3F)c12	C64H72F2N12O6S2	KRAS	P01116	VHL	WO-2023138524-A1
TPD-7ZHOU5	WO2023138524A1_129	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC7(CC6)CN(c6ccc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)cc6)C7)CC5)nc4c3F)c12	C67H73F2N11O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-1EL1DC	WO2023138524A1_130	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC7(CC6)CCN(c6ccc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)cc6)CC7)CC5)nc4c3F)c12	C69H77F2N11O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-UNPVHQ	WO2023138524A1_131	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)CC6CN(c7ccc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)cc7)C6)CC5)nc4c3F)c12	C65H71F2N11O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-HM6W6O	WO2023138524A1_132	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)Cc6ccc(N7CCC(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)CC7)cc6)CC5)nc4c3F)c12	C67H75F2N11O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-BJDZ82	WO2023138524A1_133	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)C6CCC7(CC6)CN(c6ccc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)cc6)C7)CC5)nc4c3F)c12	C69H77F2N11O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-6BAYX6	WO2023138524A1_134	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC7(CC6)CN(C(=O)c6ccc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)cc6)C7)CC5)nc4c3F)c12	C68H73F2N11O7S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-Z0MA3N	WO2023138524A1_135	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)c2ccc(COC3CCN(CC4(COc5nc(N6CC7CCC(C6)N7)c6cnc(-c7cc(O)cc8ccc(F)c(F)c78)c(F)c6n5)CC4)CC3)cc2)C(C)(C)C)cc1	C63H69F3N10O7S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-RCDPWR	WO2023138524A1_136	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)c2ncc(N3CCC(CN(C)CC4(COc5nc(N6CC7CCC(C6)N7)c6cnc(-c7cc(O)cc8ccc(F)c(F)c78)c(F)c6n5)CC4)CC3)s2)C(C)(C)C)cc1	C61H69F3N12O6S2	KRAS	P01116	VHL	WO-2023138524-A1
TPD-V1ULGF	WO2023138524A1_137	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)c2ccc(N3CC4(CCN(CC5(COc6nc(N7CC8CCC(C7)N8)c7cnc(-c8cc(O)cc9ccc(F)c(F)c89)c(F)c7n6)CC5)CC4)C3)cc2)C(C)(C)C)cc1	C64H70F3N11O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-ZLYEIG	WO2023138524A1_138	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)c2ccc(N3CCC4(CCN(CC5(COc6nc(N7CC8CCC(C7)N8)c7cnc(-c8cc(O)cc9ccc(F)c(F)c89)c(F)c7n6)CC5)CC4)CC3)cc2)C(C)(C)C)cc1	C66H74F3N11O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-NKV6FJ	WO2023138524A1_139	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)c2ccc(N3CC(CN(C)CC4(COc5nc(N6CC7CCC(C6)N7)c6cnc(-c7cc(O)cc8ccc(F)c(F)c78)c(F)c6n5)CC4)C3)cc2)C(C)(C)C)cc1	C62H68F3N11O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-INTQ9Y	WO2023138524A1_140	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCN(c3ccc(CN(C)CC4(COc5nc(N6CC7CCC(C6)N7)c6cnc(-c7cc(O)cc8ccc(F)c(F)c78)c(F)c6n5)CC4)cc3)CC2)C(C)(C)C)cc1	C64H72F3N11O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-BCYATJ	WO2023138524A1_141	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)c2ccc(N3CC4(CCC(N(C)CC5(COc6nc(N7CC8CCC(C7)N8)c7cnc(-c8cc(O)cc9ccc(F)c(F)c89)c(F)c7n6)CC5)CC4)C3)cc2)C(C)(C)C)cc1	C66H74F3N11O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-HQ3BJ0	WO2023138524A1_142	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCO[C@H]2CN3CCC[C@@]3(COc3nc(N4CC5CCC(C4)N5)c4cc(Cl)c(-c5ccc(F)c6sc(N)c(C#N)c56)c(F)c4n3)C2)C(C)(C)C)cc1	C61H72ClF2N11O6S2	KRAS	P01116	VHL	WO-2023138524-A1
TPD-UE753K	WO2023138524A1_143	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCO[C@H]2CN3CCC[C@@]3(COc3nc(N4CC5CCC(C4)N5)c4cc(Cl)c(-c5ccc(F)c6sc(N)c(C#N)c56)c(F)c4n3)C2)C(C)(C)C)cc1	C60H70ClF2N11O6S2	KRAS	P01116	VHL	WO-2023138524-A1
TPD-4QE8R3	WO2023138524A1_144	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCCC[C@H]2CC[C@@]3(COc4nc(N5CC6CCC(C5)N6)c5cc(Cl)c(-c6ccc(F)c7sc(N)c(C#N)c67)c(F)c5n4)CCCN23)C(C)(C)C)cc1	C63H76ClF2N11O5S2	KRAS	P01116	VHL	WO-2023138524-A1
TPD-QSXQH8	WO2023138524A1_145	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CC2CCN(C(=O)OC[C@H]3CC[C@@]4(COc5nc(N6CC7CCC(C6)N7)c6cc(Cl)c(-c7ccc(F)c8sc(N)c(C#N)c78)c(F)c6n5)CCCN34)CC2)C(C)(C)C)cc1	C63H73ClF2N12O7S2	KRAS	P01116	VHL	WO-2023138524-A1
TPD-PB7CVX	WO2023138524A1_146	.	Cc1ncsc1-c1ccc([C@H](CC(=O)NCCCCCCO[C@H]2CN3CCC[C@@]3(COc3nc(N4CC5CCC(C4)N5)c4cc(Cl)c(-c5ccc(F)c6sc(N)c(C#N)c56)c(F)c4n3)C2)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(C#N)CC2)C(C)(C)C)cc1	C66H76ClF2N13O7S2	KRAS	P01116	VHL	WO-2023138524-A1
TPD-5YR00W	WO2023138524A1_147	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCNC(=O)OC[C@H]2CC[C@@]3(COc4nc(N5CC6CCC(C5)N6)c5cc(Cl)c(-c6ccc(F)c7sc(N)c(C#N)c67)c(F)c5n4)CCCN23)C(C)(C)C)cc1	C61H71ClF2N12O7S2	KRAS	P01116	VHL	WO-2023138524-A1
TPD-JAMQBD	WO2023138524A1_148	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)c2ccc(OCC3CCN(CC4(COc5nc(N6CC7CCC(C6)N7)c6cc(Cl)c(-c7cccc8sc(N)c(C#N)c78)c(F)c6n5)CC4)CC3)cc2)C(C)(C)C)cc1	C64H71ClFN11O6S2	KRAS	P01116	VHL	WO-2023138524-A1
TPD-366O8K	WO2023138524A1_149	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](n2cc(C3CCN(C(=O)OC[C@H]4CC[C@@]5(COc6nc(N7CC8CCC(C7)N8)c7cc(Cl)c(-c8cccc9sc(N)c(C#N)c89)c(F)c7n6)CCCN45)CC3)nn2)C(C)(C)C)cc1	C63H72ClFN14O6S2	KRAS	P01116	VHL	WO-2023138524-A1
TPD-29T0MG	WO2023138524A1_150	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](n2cc(-c3ccc(NC(=O)OC[C@H]4CC[C@@]5(COc6nc(N7CC8CCC(C7)N8)c7cc(Cl)c(-c8cccc9sc(N)c(C#N)c89)c(F)c7n6)CCCN45)cc3)nn2)C(C)(C)C)cc1	C64H68ClFN14O6S2	KRAS	P01116	VHL	WO-2023138524-A1
TPD-0YUVIW	WO2023138524A1_151	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CC3(C2)CN(C(=O)OC[C@H]2CC[C@@]4(COc5nc(N6CC7CCC(C6)N7)c6cc(Cl)c(-c7cccc8sc(N)c(C#N)c78)c(F)c6n5)CCCN24)C3)C(C)(C)C)cc1	C63H72ClFN12O7S2	KRAS	P01116	VHL	WO-2023138524-A1
TPD-WPMMAJ	WO2023138524A1_152	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(COc7ccc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)NCc8ccc(-c9scnc9C)cc8)C(C)(C)C)cc7)CC6)CC5)nc4c3F)c12	C65H70F2N10O7S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-4BR8ES	WO2023138524A1_153	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCNC(=O)OC[C@H]2CC[C@@]3(COc4nc(N5CC6CCC(C5)N6)c5cc(Cl)c(-c6cccc7sc(N)c(C#N)c67)c(F)c5n4)CCCN23)C(C)(C)C)cc1	C62H74ClFN12O7S2	KRAS	P01116	VHL	WO-2023138524-A1
TPD-6M7BG8	WO2023138524A1_154	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCNC(=O)OC[C@H]2CC[C@@]3(COc4nc(N5CC6CCC(C5)N6)c5cc(Cl)c(-c6cccc7sc(N)c(C#N)c67)c(F)c5n4)CCCN23)C(C)(C)C)cc1	C60H70ClFN12O7S2	KRAS	P01116	VHL	WO-2023138524-A1
TPD-6LCM2Z	WO2023138524A1_155	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCCNC(=O)OC[C@H]2CC[C@@]3(COc4nc(N5CC6CCC(C5)N6)c5cc(Cl)c(-c6cccc7sc(N)c(C#N)c67)c(F)c5n4)CCCN23)C(C)(C)C)cc1	C64H78ClFN12O7S2	KRAS	P01116	VHL	WO-2023138524-A1
TPD-1JOUH8	WO2023138524A1_156	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CC3(CCN(C(=O)OC[C@H]4CC[C@@]5(COc6nc(N7CC8CCC(C7)N8)c7cc(Cl)c(-c8cccc9sc(N)c(C#N)c89)c(F)c7n6)CCCN45)CC3)C2)C(C)(C)C)cc1	C65H76ClFN12O7S2	KRAS	P01116	VHL	WO-2023138524-A1
TPD-F20NC8	WO2023138524A1_157	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CC2CCN(C(=O)OC[C@H]3CC[C@@]4(COc5nc(N6CC7CCC(C6)N7)c6cc(Cl)c(-c7cccc8sc(N)c(C#N)c78)c(F)c6n5)CCCN34)CC2)C(C)(C)C)cc1	C63H74ClFN12O7S2	KRAS	P01116	VHL	WO-2023138524-A1
TPD-WB8QYT	WO2023138524A1_158	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCN(C(=O)OC[C@H]3CC[C@@]4(COc5nc(N6CC7CCC(C6)N7)c6cc(Cl)c(-c7cccc8sc(N)c(C#N)c78)c(F)c6n5)CCCN34)CC2)C(C)(C)C)cc1	C62H72ClFN12O7S2	KRAS	P01116	VHL	WO-2023138524-A1
TPD-P6XBS9	WO2023138524A1_159	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](n2cc(C3CC4(CCN(C(=O)OC[C@H]5CC[C@@]6(COc7nc(N8CC9CCC(C8)N9)c8cc(Cl)c(-c9cccc%10sc(N)c(C#N)c9%10)c(F)c8n7)CCCN56)CC4)C3)nn2)C(C)(C)C)cc1	C66H76ClFN14O6S2	KRAS	P01116	VHL	WO-2023138524-A1
TPD-FCBUOW	WO2023138524A1_160	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](n2cc(C3CC4(CCN(C(=O)[C@H]5CC[C@@]6(COc7nc(N8CC9CCC(C8)N9)c8cc(Cl)c(-c9cccc%10sc(N)c(C#N)c9%10)c(F)c8n7)CCCN56)CC4)C3)nn2)C(C)(C)C)cc1	C65H74ClFN14O5S2	KRAS	P01116	VHL	WO-2023138524-A1
TPD-HW45LS	WO2023138524A1_161	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CC3(CCN(C(=O)[C@H]4CC[C@@]5(COc6nc(N7CC8CCC(C7)N8)c7cc(Cl)c(-c8cccc9sc(N)c(C#N)c89)c(F)c7n6)CCCN45)CC3)C2)C(C)(C)C)cc1	C64H74ClFN12O6S2	KRAS	P01116	VHL	WO-2023138524-A1
TPD-6G5Y2A	WO2023138524A1_162	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC[C@]56CCCN5[C@@H](COC(=O)N5CCC7(CC5)CC(C(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)c5ccc(-c8scnc8C)cc5)C(C)(C)C)C7)CC6)nc4c3F)c12	C67H77F2N11O8S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-K4N2GI	WO2023138524A1_163	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC[C@]56CCCN5[C@@H](COC(=O)N5CCC7(CC5)CC(C(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)c5ccc(-c8scnc8C)cc5)C(C)(C)C)C7)CC6)nc4c3F)c12	C67H81F2N11O8S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-FRRPWL	WO2023138524A1_165	.	CCn1nccc1-c1ccc([C@H](CO)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](C(C)C)n2cc(C3CC4(CCN(C(=O)OC[C@H]5CC[C@@]6(COc7nc(N8CC9CCC(C8)N9)c8cc(Cl)c(-c9cccc%10sc(N)c(C#N)c9%10)c(F)c8n7)CCCN56)CC4)C3)nn2)cc1	C66H77ClFN15O7S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-853IKS	WO2023138524A1_166	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCC3(CC2)CN(C(=O)OC[C@H]2CC[C@@]4(COc5nc(N6CC7CCC(C6)N7)c6cc(Cl)c(-c7cccc8sc(N)c(C#N)c78)c(F)c6n5)CCCN24)C3)C(C)(C)C)cc1	C65H76ClFN12O7S2	KRAS	P01116	VHL	WO-2023138524-A1
TPD-B7KGIF	WO2023138524A1_167	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](n2cc(-c3ccc(OC[C@H]4CC[C@@]5(COc6nc(N7CC8CCC(C7)N8)c7cc(Cl)c(-c8cccc9sc(N)c(C#N)c89)c(F)c7n6)CCCN45)nc3)nn2)C(C)(C)C)cc1	C62H66ClFN14O5S2	KRAS	P01116	VHL	WO-2023138524-A1
TPD-H4T2XN	WO2023138524A1_168	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)c2ccc(C3CN(C(=O)OC[C@H]4CC[C@@]5(COc6nc(N7CC8CCC(C7)N8)c7cc(Cl)c(-c8cccc9sc(N)c(C#N)c89)c(F)c7n6)CCCN45)C3)cc2)C(C)(C)C)cc1	C66H72ClFN12O7S2	KRAS	P01116	VHL	WO-2023138524-A1
TPD-VA8YJZ	WO2023138524A1_169	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)c2ccc(C3CCN(C(=O)OC[C@H]4CC[C@@]5(COc6nc(N7CC8CCC(C7)N8)c7cc(Cl)c(-c8cccc9sc(N)c(C#N)c89)c(F)c7n6)CCCN45)CC3)cc2)C(C)(C)C)cc1	C68H76ClFN12O7S2	KRAS	P01116	VHL	WO-2023138524-A1
TPD-ANKZYK	WO2023138524A1_170	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)c2ccc(C3CCN(C(=O)[C@H]4CC[C@@]5(COc6nc(N7CC8CCC(C7)N8)c7cc(Cl)c(-c8cccc9sc(N)c(C#N)c89)c(F)c7n6)CCCN45)CC3)cc2)C(C)(C)C)cc1	C67H74ClFN12O6S2	KRAS	P01116	VHL	WO-2023138524-A1
TPD-KEZDZZ	WO2023138524A1_171	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(CCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)NCc7ccc(-c8scnc8C)cc7)C(C)(C)C)CC6)CC5)nc4c3F)c12	C62H72F2N10O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-79X3KH	WO2023138524A1_172	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CC7(CCN(c8ccc(C(=O)N[C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)(C)C)cc8)CC7)C6)CC5)nc4c3F)c12	C67H73F2N11O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-Y988UK	WO2023138524A1_173	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC7(CC6)CN(c6ccc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)cn6)C7)CC5)nc4c3F)c12	C66H72F2N12O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-H5YY14	WO2023138524A1_174	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC7(CC6)CN(Oc6ccc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)cc6)C7)CC5)nc4c3F)c12	C67H73F2N11O7S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-N6OMXV	WO2023138524A1_175	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC7(CC6)CC(c6cn([C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)nn6)C7)CC5)nc4c3F)c12	C63H70F2N12O5S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-1Y6FMW	WO2023138524A1_176	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(c7ccc(-c8cn([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)(C)C)nn8)cc7)CC6)CC5)nc4c3F)c12	C66H70F2N12O5S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-7O6232	WO2023138524A1_177	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(COc7ccc(-c8cn([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)(C)C)nn8)cc7)CC6)CC5)nc4c3F)c12	C67H72F2N12O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-2BY7NO	WO2023138524A1_178	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC[C@]56CCCN5[C@@H](COC(=O)N5CCC7(CC5)CC(c5cn([C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)nn5)C7)CC6)nc4c3F)c12	C68H77F2N13O7S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-UT12FW	WO2023138524A1_179	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](n2cc(C3CC4(CCN(CC5(COc6nc(N7CC8CCC(C7)N8)c7cc(Cl)c(-c8cccc9sc(N)c(C#N)c89)c(F)c7n6)CC5)CC4)C3)nn2)C(C)(C)C)cc1	C61H69ClFN13O4S2	KRAS	P01116	VHL	WO-2023138524-A1
TPD-VV1Q36	WO2023138524A1_180	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(COc7ccc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)cc7)CC6)CC5)nc4c3F)c12	C66H76F2N10O7S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-7KXNSY	WO2023138524A1_181	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(COc7ccc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](CO)c8ccc(-c9ccnn9CC)cc8)C(C)(C)C)cc7)CC6)CC5)nc4c3F)c12	C67H79F2N11O8	KRAS	P01116	VHL	WO-2023138524-A1
TPD-XXN411	WO2023138524A1_182	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(COC78CCC(C(=O)N[C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)(C)C)(CC7)CC8)CC6)CC5)nc4c3F)c12	C68H80F2N10O7S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-XEGMG8	WO2023138524A1_183	.	C#Cc1c(F)ccc2cc(O)cc(-c3nc(OC)c4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(COc7ccc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)cc7)CC6)CC5)nc4c3F)c12	C67H74F2N10O8S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-85CB0O	WO2023138524A1_184	.	CCc1c(F)ccc2cc(O)cc(-c3nc(OC)c4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(COc7ccc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)cc7)CC6)CC5)nc4c3F)c12	C67H78F2N10O8S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-LWCEBJ	WO2023138524A1_185	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)c2ccc(OC3CC4(CCN(CC5(COc6nc(N7CC8CCC(C7)N8)c7cc(Cl)c(-c8ccc(F)c9sc(N)c(C#N)c89)c(F)c7n6)CC5)CC4)C3)cc2)C(C)(C)C)cc1	C66H72ClF2N11O6S2	KRAS	P01116	VHL	WO-2023138524-A1
TPD-XJ3ZX9	WO2023138524A1_187	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)CC6CC7(C6)CN(c6ccc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)cc6)C7)CC5)nc4c3F)c12	C68H75F2N11O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-ZNFO4E	WO2023138524A1_188	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)c2ccc(OCC3CCN(CC4(COc5nc(N6CC7CCC(C6)N7)c6cnc(-c7cc(O)cc8ccc(F)c(F)c78)c(F)c6n5)CC4)CC3)cc2)C(C)(C)C)cc1	C64H71F3N10O7S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-47BV24	WO2023138524A1_189	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)c2ccc(N3CC4(CCN(CC5(COc6nc(N7CC8CCC(C7)N8)c7cnc(-c8cc(O)cc9ccc(F)c(F)c89)c(F)c7n6)CC5)CC4)C3)cc2)C(C)(C)C)cc1	C65H72F3N11O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-GVUFF9	WO2023138524A1_190	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)Cc6ccc(OCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)NCc7ccc(-c8scnc8C)cc7)C(C)(C)C)nc6)CC5)nc4c3F)c12	C62H67F2N11O7S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-A226TO	WO2023138524A1_192	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(CN(C)c7ccc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)cc7)CC6)CC5)nc4c3F)c12	C67H75F2N11O6S	KRAS	P01116	VHL	WO-2023138524-A1
TPD-EZTNUF	SCHEMBL25926332	4-[4-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]butoxy]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	COc1cc(N2CCN(CCCCOc3ccc(C4CCN(c5ccc(C#N)c(C(F)(F)F)c5)CC4)cc3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C41H45F3N6O5	AR	P10275	CRBN	WO-2023139199-A1
TPD-58XF8R	SCHEMBL25926393	4-[4-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]butoxy]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(OCCCCN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)cc3)CC2)cc1C(F)(F)F	C40H43F3N6O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-DCVHGH	SCHEMBL25926573	2-cyclopropyl-4-[4-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]benzonitrile	COc1cc(N2CCN(CC3CCN(c4ccc(C5CCN(c6ccc(C#N)c(C7CC7)c6)CC5)cc4)CC3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C45H53N7O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-15M7HN	SCHEMBL25926628	4-[4-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	COc1cc(N2CCN(CC3CCN(c4ccc(C5CCN(c6ccc(C#N)c(C(F)(F)F)c6)CC5)cc4)CC3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C43H48F3N7O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-BCZ4LA	SCHEMBL25926737	4-[4-[4-[3-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]ethyl]cyclobutyl]oxyphenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	COc1cc(N2CCN(CCC3CC(Oc4ccc(C5CCN(c6ccc(C#N)c(C(F)(F)F)c6)CC5)cc4)C3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C43H47F3N6O5	AR	P10275	CRBN	WO-2023139199-A1
TPD-8TUQSZ	AZ'3137	4-[4-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-3-fluoro-2-(trifluoromethyl)benzonitrile; 2960179-55-7; orb2664298; EX-A9771; HY-162702	COc1cc(N2CCN(CC3CCN(c4ccc(C5CCN(c6ccc(C#N)c(C(F)(F)F)c6F)CC5)cc4)CC3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C43H47F4N7O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-W1VRTS	SCHEMBL25926899	4-[4-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]butoxy]phenyl]piperidin-1-yl]-3-fluoro-2-(trifluoromethyl)benzonitrile	COc1cc(N2CCN(CCCCOc3ccc(C4CCN(c5ccc(C#N)c(C(F)(F)F)c5F)CC4)cc3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C41H44F4N6O5	AR	P10275	CRBN	WO-2023139199-A1
TPD-3G4L1X	SCHEMBL25926985	4-[4-[5-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]butoxy]pyrimidin-2-yl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile; SCHEMBL30493334	COc1cc(N2CCN(CCCCOc3cnc(C4CCN(c5ccc(C#N)c(C(F)(F)F)c5)CC4)nc3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C39H43F3N8O5	AR	P10275	CRBN	WO-2023139199-A1
TPD-EXXH28	SCHEMBL25927277	4-[4-[4-[3-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]ethyl]azetidin-1-yl]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	COc1cc(N2CCN(CCC3CN(c4ccc(C5CCN(c6ccc(C#N)c(C(F)(F)F)c6)CC5)cc4)C3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C42H46F3N7O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-AW0DDM	SCHEMBL25927342	5-[4-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]butoxy]phenyl]piperidin-1-yl]-3-(trifluoromethyl)pyridine-2-carbonitrile	COc1cc(N2CCN(CCCCOc3ccc(C4CCN(c5cnc(C#N)c(C(F)(F)F)c5)CC4)cc3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C40H44F3N7O5	AR	P10275	CRBN	WO-2023139199-A1
TPD-3TB4GA	SCHEMBL25927406	4-[4-[4-[5-[4-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]-3,3-difluoropentoxy]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	COc1cc(N2CCN(CCC(F)(F)CCOc3ccc(C4CCN(c5ccc(C#N)c(C(F)(F)F)c5)CC4)cc3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C42H45F5N6O5	AR	P10275	CRBN	WO-2023139199-A1
TPD-UGBYID	SCHEMBL25927540	4-[4-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]propoxy]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	COc1cc(N2CCN(CCCOc3ccc(C4CCN(c5ccc(C#N)c(C(F)(F)F)c5)CC4)cc3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C40H43F3N6O5	AR	P10275	CRBN	WO-2023139199-A1
TPD-BCV2R8	SCHEMBL25927601	2-cyclopropyl-4-[4-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]butoxy]phenyl]piperidin-1-yl]benzonitrile	COc1cc(N2CCN(CCCCOc3ccc(C4CCN(c5ccc(C#N)c(C6CC6)c5)CC4)cc3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C43H50N6O5	AR	P10275	CRBN	WO-2023139199-A1
TPD-AGDU8H	SCHEMBL25927788	4-[4-[4-[4-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]ethyl]piperidin-1-yl]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	COc1cc(N2CCN(CCC3CCN(c4ccc(C5CCN(c6ccc(C#N)c(C(F)(F)F)c6)CC5)cc4)CC3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C44H50F3N7O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-CWB2LZ	SCHEMBL25927908	2-chloro-4-[4-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]butoxy]phenyl]piperidin-1-yl]benzonitrile	N#Cc1ccc(N2CCC(c3ccc(OCCCCN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)cc3)CC2)cc1Cl	C39H43ClN6O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-XZ9D8U	SCHEMBL25927933	4-[4-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]butoxy]phenyl]piperidin-1-yl]-2-methoxybenzonitrile	COc1cc(N2CCC(c3ccc(OCCCCN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)cc3)CC2)ccc1C#N	C40H46N6O5	AR	P10275	CRBN	WO-2023139199-A1
TPD-MDNC7S	SCHEMBL25928091	6-[4-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]butoxy]phenyl]piperidin-1-yl]-2-methylpyridine-3-carbonitrile	Cc1nc(N2CCC(c3ccc(OCCCCN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)cc3)CC2)ccc1C#N	C39H45N7O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-UE5IFX	SCHEMBL25928152	8-[4-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]butoxy]phenyl]piperidin-1-yl]quinoline-5-carbonitrile	N#Cc1ccc(N2CCC(c3ccc(OCCCCN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)cc3)CC2)c2ncccc12	C42H45N7O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-ELA06I	SCHEMBL25928303	4-[4-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-3-oxo-1H-isoindol-5-yl]piperazin-1-yl]butoxy]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(OCCCCN4CCN(c5cc6c(cc5F)CN(C5CCC(=O)NC5=O)C6=O)CC4)cc3)CC2)cc1C(F)(F)F	C40H42F4N6O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-XGQ3EI	SCHEMBL25928323	4-[4-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]butoxy]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(OCCCCN4CCN(c5cc6c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C6)CC4)cc3)CC2)cc1C(F)(F)F	C40H42F4N6O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-JR8VEV	SCHEMBL25928350	4-[4-[5-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]butoxy]pyrimidin-2-yl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ncc(OCCCCN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)cn3)CC2)cc1C(F)(F)F	C38H41F3N8O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-LYMSIW	WO2023139199A1_23	4-[4-[4-[4-[4-[2-(2,6-Dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]butoxy]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(OCCCCN4CCN(c5cc6c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)cc3)CC2)cc1C(F)(F)F	C40H40F4N6O5	AR	P10275	CRBN	WO-2023139199-A1
TPD-N6802I	SCHEMBL25928610	4-[(4S)-4-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]butoxy]phenyl]-3,3-dimethylpiperidin-1-yl]-2-(trifluoromethyl)benzonitrile	CC1(C)CN(c2ccc(C#N)c(C(F)(F)F)c2)CC[C@H]1c1ccc(OCCCCN2CCN(c3ccc4c(c3)CN(C3CCC(=O)NC3=O)C4=O)CC2)cc1	C42H47F3N6O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-3Z65CU	SCHEMBL25928670	4-[(4R)-4-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]butoxy]phenyl]-3,3-dimethylpiperidin-1-yl]-2-(trifluoromethyl)benzonitrile	CC1(C)CN(c2ccc(C#N)c(C(F)(F)F)c2)CC[C@@H]1c1ccc(OCCCCN2CCN(c3ccc4c(c3)CN(C3CCC(=O)NC3=O)C4=O)CC2)cc1	C42H47F3N6O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-J9CMRK	SCHEMBL25928746	4-[4-[4-[4-[4-[3-(2,6-Dioxopiperidin-3-yl)-2-oxo-1,3-benzoxazol-6-yl]piperazin-1-yl]butoxy]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(OCCCCN4CCN(c5ccc6c(c5)oc(=O)n6C5CCC(=O)NC5=O)CC4)cc3)CC2)cc1C(F)(F)F	C39H41F3N6O5	AR	P10275	CRBN	WO-2023139199-A1
TPD-1RFIX5	SCHEMBL25928891	4-[4-[4-[4-[[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(N4CCC(CN5CCN(CC6CCN(c7ccc8c(c7)CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)CC4)cc3)CC2)cc1C(F)(F)F	C48H57F3N8O3	AR	P10275	CRBN	WO-2023139199-A1
TPD-5H0CQ2	WO2023139199A1_28	.	CC(F)(F)c1cc(N2CCC(c3ccc(OCCC(F)(F)CCN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)cc3)CC2)ccc1C#N	C42H46F4N6O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-TQ6IIM	WO2023139199A1_29	4-[4-[4-[4-[4-[1-(2,6-Dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperazin-1-yl]butoxy]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	Cn1c(=O)n(C2CCC(=O)NC2=O)c2ccc(N3CCN(CCCCOc4ccc(C5CCN(c6ccc(C#N)c(C(F)(F)F)c6)CC5)cc4)CC3)cc21	C40H44F3N7O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-VS60RZ	WO2023139199A1_30	.	N#Cc1ccc(N2CCC(c3ccc(O[C@H]4C[C@H](CCN5CCN(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC5)C4)cc3)CC2)cc1C(F)(F)F	C42H45F3N6O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-E6QALQ	WO2023139199A1_31	4-[4-[4-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]butoxy]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(OCCCCC4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)cc3)CC2)cc1C(F)(F)F	C41H44F3N5O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-7DI8BB	WO2023139199A1_32	.	N#Cc1ccc(N2CCC(c3ccc(O[C@H]4C[C@@H](CCN5CCN(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC5)C4)cc3)CC2)cc1C(F)(F)F	C42H45F3N6O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-BUC3KM	SCHEMBL25929634	4-[4-[4-[4-[3-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-7-oxa-3,10-diazaspiro[5.6]dodecan-10-yl]butoxy]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(OCCCCN4CCOC5(CC4)CCN(c4ccc6c(c4)CN(C4CCC(=O)NC4=O)C6=O)CC5)cc3)CC2)cc1C(F)(F)F	C45H51F3N6O5	AR	P10275	CRBN	WO-2023139199-A1
TPD-EJVZAO	WO2023139199A1_34	4-[4-[4-[4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]oxy]piperidin-1-yl]butoxy]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(OCCCCN4CCC(Oc5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)cc3)CC2)cc1C(F)(F)F	C41H44F3N5O5	AR	P10275	CRBN	WO-2023139199-A1
TPD-I34YJC	WO2023139199A1_35	4-[4-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]butoxy]-3-fluorophenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(OCCCCN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)c(F)c3)CC2)cc1C(F)(F)F	C40H42F4N6O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-ZAG340	WO2023139199A1_36	.	N#Cc1ccc(N2CCC(c3ccc(OC[C@H]4C[C@H](CN5CCN(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC5)C4)cc3)CC2)cc1C(F)(F)F	C42H45F3N6O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-IWU8TU	WO2023139199A1_37	4-[4-[4-[4-[[4-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]oxy]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(N4CCC(CN5CCC(Oc6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3)CC2)cc1C(F)(F)F	C43H47F3N6O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-J63H8G	WO2023139199A1_38	4-[4-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]butoxy]-2-fluorophenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(OCCCCN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)cc3F)CC2)cc1C(F)(F)F	C40H42F4N6O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-K155N9	WO2023139199A1_39	.	N#Cc1ccc(N2CCC(c3ccc(OC[C@H]4C[C@@H](CN5CCN(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC5)C4)cc3)CC2)cc1C(F)(F)F	C42H45F3N6O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-MU4K24	WO2023139199A1_40	4-[4-[4-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperidin-4-yl]oxyphenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(OC4CCN(CC5CCN(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3)CC2)cc1C(F)(F)F	C43H47F3N6O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-GC8VTV	SCHEMBL25930799	4-[4-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]butoxy]-2-methylphenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	Cc1cc(OCCCCN2CCN(c3ccc4c(c3)CN(C3CCC(=O)NC3=O)C4=O)CC2)ccc1C1CCN(c2ccc(C#N)c(C(F)(F)F)c2)CC1	C41H45F3N6O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-WXZBA2	SCHEMBL25930869	2-cyclopropyl-4-[4-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]benzonitrile	N#Cc1ccc(N2CCC(c3ccc(N4CCC(CN5CCN(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3)CC2)cc1C1CC1	C44H51N7O3	AR	P10275	CRBN	WO-2023139199-A1
TPD-7WPKJK	SCHEMBL25930880	2-cyclopropyl-4-[4-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]butoxy]phenyl]piperidin-1-yl]benzonitrile	N#Cc1ccc(N2CCC(c3ccc(OCCCCN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)cc3)CC2)cc1C1CC1	C42H48N6O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-OTUXYE	SCHEMBL25930924	4-[4-[4-[3-[4-[2-(2,6-Dioxopiperidin-3-yl)-3-oxo-[1,2,4]triazolo[4,3-a]pyridin-7-yl]piperazin-1-yl]propoxy]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(OCCCN4CCN(c5ccn6c(=O)n(C7CCC(=O)NC7=O)nc6c5)CC4)cc3)CC2)cc1C(F)(F)F	C37H39F3N8O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-YTBCR4	SCHEMBL25930934	4-[4-[4-[4-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]ethyl]piperidin-1-yl]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(N4CCC(CCN5CCN(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3)CC2)cc1C(F)(F)F	C43H48F3N7O3	AR	P10275	CRBN	WO-2023139199-A1
TPD-5HVG2K	SCHEMBL25930967	4-[4-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-3-fluoro-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(N4CCC(CN5CCN(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3)CC2)c(F)c1C(F)(F)F	C42H45F4N7O3	AR	P10275	CRBN	WO-2023139199-A1
TPD-26EO5D	SCHEMBL25931004	4-[4-[4-[4-[[4-[2-(2,6-Dioxopiperidin-3-yl)-3-oxo-[1,2,4]triazolo[4,3-a]pyridin-7-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(N4CCC(CN5CCN(c6ccn7c(=O)n(C8CCC(=O)NC8=O)nc7c6)CC5)CC4)cc3)CC2)cc1C(F)(F)F	C40H44F3N9O3	AR	P10275	CRBN	WO-2023139199-A1
TPD-M7V4GI	SCHEMBL25931066	4-[(3S)-4-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]butoxy]phenyl]-3-methylpiperazin-1-yl]-2-(trifluoromethyl)benzonitrile	C[C@H]1CN(c2ccc(C#N)c(C(F)(F)F)c2)CCN1c1ccc(OCCCCN2CCN(c3ccc4c(c3)CN(C3CCC(=O)NC3=O)C4=O)CC2)cc1	C40H44F3N7O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-WA7FA7	SCHEMBL25931166	5-[4-[4-[5-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]pentoxy]phenyl]piperidin-1-yl]-3-(trifluoromethyl)pyridine-2-carbonitrile	N#Cc1ncc(N2CCC(c3ccc(OCCCCCN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)cc3)CC2)cc1C(F)(F)F	C40H44F3N7O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-GYQZWM	SCHEMBL25931233	4-[4-[4-[4-[4-[2-(2,6-Dioxopiperidin-3-yl)-3-oxo-[1,2,4]triazolo[4,3-a]pyrimidin-7-yl]piperazin-1-yl]butoxy]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(OCCCCN4CCN(c5ccn6c(=O)n(C7CCC(=O)NC7=O)nc6n5)CC4)cc3)CC2)cc1C(F)(F)F	C37H40F3N9O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-FNXEQL	WO2023139199A1_51	4-[4-[4-[5-[4-[2-(2,6-Dioxopiperidin-3-yl)-3-oxo-[1,2,4]triazolo[4,3-a]pyridin-7-yl]piperazin-1-yl]pentoxy]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(OCCCCCN4CCN(c5ccn6c(=O)n(C7CCC(=O)NC7=O)nc6c5)CC4)cc3)CC2)cc1C(F)(F)F	C39H43F3N8O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-E7ZWX1	SCHEMBL25931308	5-[4-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]butoxy]phenyl]piperidin-1-yl]-3-(trifluoromethyl)pyridine-2-carbonitrile	N#Cc1ncc(N2CCC(c3ccc(OCCCCN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)cc3)CC2)cc1C(F)(F)F	C39H42F3N7O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-BOVZG3	SCHEMBL25931334	4-[4-[4-[3-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]ethyl]pyrrolidin-1-yl]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(N4CCC(CCN5CCN(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC5)C4)cc3)CC2)cc1C(F)(F)F	C42H46F3N7O3	AR	P10275	CRBN	WO-2023139199-A1
TPD-C7UMZA	WO2023139199A1_54	4-[4-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]butoxy]phenyl]piperidin-1-yl]-3-fluoro-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(OCCCCN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)cc3)CC2)c(F)c1C(F)(F)F	C40H42F4N6O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-BMS3US	SCHEMBL25931412	4-[(3R)-4-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]butoxy]phenyl]-3-methylpiperazin-1-yl]-2-(trifluoromethyl)benzonitrile	C[C@@H]1CN(c2ccc(C#N)c(C(F)(F)F)c2)CCN1c1ccc(OCCCCN2CCN(c3ccc4c(c3)CN(C3CCC(=O)NC3=O)C4=O)CC2)cc1	C40H44F3N7O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-CRA36G	SCHEMBL25931721	4-[4-[6-[4-[4-[6-(2,6-dioxopiperidin-3-yl)-5-oxo-7H-pyrrolo[3,4-b]pyridin-2-yl]piperazin-1-yl]butoxy]pyridin-3-yl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(OCCCCN4CCN(c5ccc6c(n5)CN(C5CCC(=O)NC5=O)C6=O)CC4)nc3)CC2)cc1C(F)(F)F	C38H41F3N8O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-G6BBIO	SCHEMBL25931773	4-[4-[5-[4-[4-[6-(2,6-dioxopiperidin-3-yl)-5-oxo-7H-pyrrolo[3,4-b]pyridin-2-yl]piperazin-1-yl]butoxy]pyridin-2-yl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(OCCCCN4CCN(c5ccc6c(n5)CN(C5CCC(=O)NC5=O)C6=O)CC4)cn3)CC2)cc1C(F)(F)F	C38H41F3N8O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-J3QFWZ	WO2023139199A1_58	4-[4-[5-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]butoxy]pyridin-2-yl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(OCCCCN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)cn3)CC2)cc1C(F)(F)F	C39H42F3N7O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-BIZ13N	SCHEMBL25931846	4-[4-[4-[4-[4-[2-(2,6-Dioxopiperidin-3-yl)-1-oxo-3,4-dihydroisoquinolin-6-yl]piperazin-1-yl]butoxy]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(OCCCCN4CCN(c5ccc6c(c5)CCN(C5CCC(=O)NC5=O)C6=O)CC4)cc3)CC2)cc1C(F)(F)F	C41H45F3N6O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-J4R8W4	SCHEMBL25931924	4-[4-[4-[4-[4-[6-(2,6-dioxopiperidin-3-yl)-5-oxo-7H-pyrrolo[3,4-b]pyridin-2-yl]piperazin-1-yl]butoxy]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(OCCCCN4CCN(c5ccc6c(n5)CN(C5CCC(=O)NC5=O)C6=O)CC4)cc3)CC2)cc1C(F)(F)F	C39H42F3N7O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-NS3LPJ	SCHEMBL25932007	4-[4-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-3-oxo-1H-pyrrolo[3,4-c]pyridin-6-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(N4CCC(CN5CCN(c6cc7c(cn6)C(=O)N(C6CCC(=O)NC6=O)C7)CC5)CC4)cc3)CC2)cc1C(F)(F)F	C41H45F3N8O3	AR	P10275	CRBN	WO-2023139199-A1
TPD-JHSMZO	SCHEMBL25932015	4-[4-[4-[4-[4-[2-(2,6-Dioxopiperidin-3-yl)-3-oxo-[1,2,4]triazolo[4,3-a]pyridin-7-yl]piperazin-1-yl]butoxy]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(OCCCCN4CCN(c5ccn6c(=O)n(C7CCC(=O)NC7=O)nc6c5)CC4)cc3)CC2)cc1C(F)(F)F	C38H41F3N8O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-JOYP1W	SCHEMBL25932044	4-[4-[4-[4-[4-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]butoxy]phenyl]piperazin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCN(c3ccc(OCCCCN4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)cc3)CC2)cc1C(F)(F)F	C39H40F3N7O5	AR	P10275	CRBN	WO-2023139199-A1
TPD-GQJR7X	SCHEMBL25932128	4-[4-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]butoxy]phenyl]piperazin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCN(c3ccc(OCCCCN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)cc3)CC2)cc1C(F)(F)F	C39H42F3N7O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-O40NQO	SCHEMBL25932282	4-[(3R)-3-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]propoxy]phenyl]pyrrolidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CC[C@H](c3ccc(OCCCN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)cc3)C2)cc1C(F)(F)F	C38H39F3N6O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-306Z1J	SCHEMBL25932301	4-[4-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]piperidin-1-yl]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(N4CCC(N5CCN(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3)CC2)cc1C(F)(F)F	C41H44F3N7O3	AR	P10275	CRBN	WO-2023139199-A1
TPD-5LTCEY	SCHEMBL25932358	5-[4-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-3-(trifluoromethyl)pyridine-2-carbonitrile	N#Cc1ncc(N2CCC(c3ccc(N4CCC(CN5CCN(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3)CC2)cc1C(F)(F)F	C41H45F3N8O3	AR	P10275	CRBN	WO-2023139199-A1
TPD-OIAIOM	SCHEMBL25932378	4-[4-[5-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]pyridin-2-yl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(N4CCC(CN5CCN(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cn3)CC2)cc1C(F)(F)F	C41H45F3N8O3	AR	P10275	CRBN	WO-2023139199-A1
TPD-0318B6	SCHEMBL25932409	4-[(3R)-3-[4-[4-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]ethyl]piperidin-1-yl]phenyl]pyrrolidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CC[C@H](c3ccc(N4CCC(CCN5CCN(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3)C2)cc1C(F)(F)F	C42H46F3N7O3	AR	P10275	CRBN	WO-2023139199-A1
TPD-WT5ZK1	SCHEMBL25932438	4-[(3S)-3-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]propoxy]phenyl]pyrrolidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CC[C@@H](c3ccc(OCCCN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)cc3)C2)cc1C(F)(F)F	C38H39F3N6O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-0PGMC5	SCHEMBL25932461	4-[(3R)-3-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]pyrrolidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CC[C@H](c3ccc(N4CCC(CN5CCN(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3)C2)cc1C(F)(F)F	C41H44F3N7O3	AR	P10275	CRBN	WO-2023139199-A1
TPD-IW03GQ	SCHEMBL25932517	4-[4-[4-[4-[4-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]butyl-methylamino]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	CN(CCCCN1CCN(c2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)CC1)c1ccc(C2CCN(c3ccc(C#N)c(C(F)(F)F)c3)CC2)cc1	C41H44F3N7O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-MNPWVI	SCHEMBL25932606	4-[4-[4-[4-[[4-[6-(2,6-dioxopiperidin-3-yl)-5-oxo-7H-pyrrolo[3,4-b]pyridin-2-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(N4CCC(CN5CCN(c6ccc7c(n6)CN(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3)CC2)cc1C(F)(F)F	C41H45F3N8O3	AR	P10275	CRBN	WO-2023139199-A1
TPD-EF0FG6	SCHEMBL25932642	4-[4-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-1,4-diazepan-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(N4CCC(CN5CCCN(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3)CC2)cc1C(F)(F)F	C43H48F3N7O3	AR	P10275	CRBN	WO-2023139199-A1
TPD-KOCI3V	SCHEMBL25932698	4-[(3R)-3-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]butoxy]phenyl]pyrrolidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CC[C@H](c3ccc(OCCCCN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)cc3)C2)cc1C(F)(F)F	C39H41F3N6O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-QTFD73	SCHEMBL25932770	4-[4-[4-[[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]piperidin-1-yl]methyl]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(CN4CCC(N5CCN(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3)CC2)cc1C(F)(F)F	C42H46F3N7O3	AR	P10275	CRBN	WO-2023139199-A1
TPD-15WWFF	SCHEMBL25932786	4-[4-[4-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(OCCOCCOCCNc4cccc5c4CN(C4CCC(=O)NC4=O)C5=O)cc3)CC2)cc1C(F)(F)F	C38H40F3N5O6	AR	P10275	CRBN	WO-2023139199-A1
TPD-LIXMXB	SCHEMBL25932812	4-[3-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]pyrrolidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(N4CCC(CN5CCN(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3)C2)cc1C(F)(F)F	C41H44F3N7O3	AR	P10275	CRBN	WO-2023139199-A1
TPD-A09RBC	SCHEMBL25932834	4-[(3S)-3-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]butoxy]phenyl]pyrrolidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CC[C@@H](c3ccc(OCCCCN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)cc3)C2)cc1C(F)(F)F	C39H41F3N6O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-387CY9	WO2023139199A1_80	4-[4-[4-[4-[[(3aR,6aS)-5-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-2-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(N4CCC(CN5C[C@@H]6CN(c7ccc8c(c7)CN(C7CCC(=O)NC7=O)C8=O)C[C@@H]6C5)CC4)cc3)CC2)cc1C(F)(F)F	C44H48F3N7O3	AR	P10275	CRBN	WO-2023139199-A1
TPD-Q21RUP	WO2023139199A1_81	.	CCN(CCCc1ccc(N2CCC(CN3C[C@H]4C[C@@H]3CN4c3ccc4c(c3)CN(C3CCC(=O)NC3=O)C4=O)CC2)cc1)c1ccc(C#N)c(C(F)(F)F)c1	C43H48F3N7O3	AR	P10275	CRBN	WO-2023139199-A1
TPD-KMCGPU	SCHEMBL25933328	4-[4-[4-[4-[[3-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-3,9-diazaspiro[5.5]undecan-9-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(N4CCC(CN5CCC6(CC5)CCN(c5ccc7c(c5)CN(C5CCC(=O)NC5=O)C7=O)CC6)CC4)cc3)CC2)cc1C(F)(F)F	C47H54F3N7O3	AR	P10275	CRBN	WO-2023139199-A1
TPD-HYV64R	WO2023139199A1_83	.	N#Cc1ccc(N2CCC(c3ccc(N4CCC(CNC5CCN(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3)CC2)cc1C(F)(F)F	C43H48F3N7O3	AR	P10275	CRBN	WO-2023139199-A1
TPD-7BHO3C	SCHEMBL25933448	4-[4-[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(N4CCN(CC5CCN(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3)CC2)cc1C(F)(F)F	C42H46F3N7O3	AR	P10275	CRBN	WO-2023139199-A1
TPD-OKJTZM	SCHEMBL25933502	4-[4-[6-[4-[4-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]butoxy]pyridin-3-yl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(OCCCCN4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)nc3)CC2)cc1C(F)(F)F	C39H40F3N7O5	AR	P10275	CRBN	WO-2023139199-A1
TPD-JHMGPI	SCHEMBL25933590	4-[4-[6-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]butoxy]pyridin-3-yl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(OCCCCN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)nc3)CC2)cc1C(F)(F)F	C39H42F3N7O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-33QRW7	SCHEMBL25933606	4-[4-[4-[4-[[1-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(N4CCN(CC5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3)CC2)cc1C(F)(F)F	C42H44F3N7O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-JXGVXG	WO2023139199A1_88	.	N#Cc1ccc(N2CCC(C3=CC=C(OCCCCCN4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)NC3)CC2)cc1C(F)(F)F	C40H44F3N7O5	AR	P10275	CRBN	WO-2023139199-A1
TPD-I8O98K	SCHEMBL25933726	4-[4-[6-[5-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]pentoxy]pyridin-3-yl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(OCCCCCN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)nc3)CC2)cc1C(F)(F)F	C40H44F3N7O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-X1E41H	SCHEMBL25933803	4-[4-[6-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]propoxy]pyridin-3-yl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(OCCCN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)nc3)CC2)cc1C(F)(F)F	C38H40F3N7O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-HF29M7	SCHEMBL25933839	4-[4-[4-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]ethoxy]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(OCCN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)cc3)CC2)cc1C(F)(F)F	C38H39F3N6O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-SM414V	SCHEMBL25934057	2-Cyclopropyl-4-[4-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]propoxy]phenyl]piperidin-1-yl]benzonitrile	N#Cc1ccc(N2CCC(c3ccc(OCCCN4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)cc3)CC2)cc1C1CC1	C41H44N6O5	AR	P10275	CRBN	WO-2023139199-A1
TPD-QNIPCL	WO2023139199A1_93	2-(Difluoromethyl)-4-[4-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]propoxy]phenyl]piperidin-1-yl]benzonitrile	N#Cc1ccc(N2CCC(c3ccc(OCCCN4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)cc3)CC2)cc1C(F)F	C39H40F2N6O5	AR	P10275	CRBN	WO-2023139199-A1
TPD-NLX336	WO2023139199A1_94	.	CC(F)(F)C1=C(C#N)C=CC(N2CCC(c3ccc(N4CCC(CN5CCN(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC5)CC4)nc3)CC2)C1	C42H50F2N8O3	AR	P10275	CRBN	WO-2023139199-A1
TPD-LP1AHX	SCHEMBL25934158	4-[4-[4-[2-[4-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]ethoxy]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(OCCN4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)cc3)CC2)cc1C(F)(F)F	C38H37F3N6O5	AR	P10275	CRBN	WO-2023139199-A1
TPD-9LN0BF	WO2023139199A1_96	.	N#CC1=C(C(F)(F)F)CC(N2CCC(c3ccc(NCCN4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)cc3)CC2)C=C1	C38H40F3N7O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-XY1WL8	SCHEMBL25934286	4-[4-[4-[4-[2-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxyethyl]piperazin-1-yl]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(N4CCN(CCOc5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)cc3)CC2)cc1C(F)(F)F	C38H37F3N6O5	AR	P10275	CRBN	WO-2023139199-A1
TPD-W9MAOD	WO2023139199A1_98	4-[4-[4-[4-[1-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperazin-1-yl]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(N4CCN(C5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3)CC2)cc1C(F)(F)F	C41H42F3N7O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-PLFSD1	WO2023139199A1_99	4-[4-[4-[4-[4-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxybutyl]piperazin-1-yl]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(N4CCN(CCCCOc5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)cc3)CC2)cc1C(F)(F)F	C40H41F3N6O5	AR	P10275	CRBN	WO-2023139199-A1
TPD-J9011V	SCHEMBL25934489	4-[4-[4-[4-[3-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxypropyl]piperazin-1-yl]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(N4CCN(CCCOc5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)cc3)CC2)cc1C(F)(F)F	C39H39F3N6O5	AR	P10275	CRBN	WO-2023139199-A1
TPD-X7JF5L	WO2023139199A1_101	4-[4-[4-[5-[4-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]pentoxy]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(OCCCCCN4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)cc3)CC2)cc1C(F)(F)F	C41H43F3N6O5	AR	P10275	CRBN	WO-2023139199-A1
TPD-R84XN1	WO2023139199A1_102	4-[4-[4-[5-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]pentoxy]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(OCCCCCN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)cc3)CC2)cc1C(F)(F)F	C41H45F3N6O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-EK57B3	SCHEMBL25934743	4-[4-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]butylamino]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(NCCCCN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)cc3)CC2)cc1C(F)(F)F	C40H44F3N7O3	AR	P10275	CRBN	WO-2023139199-A1
TPD-3M71HR	WO2023139199A1_104	.	CC(F)(F)c1cc(N2CCC(c3ccc(OCCCCCCCN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)cc3)CC2)ccc1C#N	C44H52F2N6O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-GO96FT	SCHEMBL25934766	4-[4-[4-[4-[4-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]butoxy]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(OCCCCN4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)cc3)CC2)cc1C(F)(F)F	C40H41F3N6O5	AR	P10275	CRBN	WO-2023139199-A1
TPD-3ZL5OP	SCHEMBL25934775	4-[4-[4-[6-[4-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]hexoxy]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(OCCCCCCN4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)cc3)CC2)cc1C(F)(F)F	C42H45F3N6O5	AR	P10275	CRBN	WO-2023139199-A1
TPD-VKGE2S	WO2023139199A1_107	4-[4-[4-[2-[2-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]ethoxy]ethoxy]ethylamino]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(NCCOCCOCCN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)cc3)CC2)cc1C(F)(F)F	C42H48F3N7O5	AR	P10275	CRBN	WO-2023139199-A1
TPD-3DJYEW	SCHEMBL25934945	4-[4-[4-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]ethylamino]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(NCCN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)cc3)CC2)cc1C(F)(F)F	C38H40F3N7O3	AR	P10275	CRBN	WO-2023139199-A1
TPD-AP2AGK	SCHEMBL25935026	4-[4-[4-[6-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]hexoxy]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(OCCCCCCN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)cc3)CC2)cc1C(F)(F)F	C42H47F3N6O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-TJP7G3	SCHEMBL25935156	4-[4-[4-[6-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]hexylamino]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(NCCCCCCN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)cc3)CC2)cc1C(F)(F)F	C42H48F3N7O3	AR	P10275	CRBN	WO-2023139199-A1
TPD-7G5ZFK	SCHEMBL25935294	4-[4-[4-[5-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]pentylamino]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(NCCCCCN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)cc3)CC2)cc1C(F)(F)F	C41H46F3N7O3	AR	P10275	CRBN	WO-2023139199-A1
TPD-KGGCY5	SCHEMBL25935402	4-[4-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]propoxy]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(OCCCN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)cc3)CC2)cc1C(F)(F)F	C39H41F3N6O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-VPCUIH	SCHEMBL25935406	4-[4-[4-[3-[4-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]propoxy]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(OCCCN4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)cc3)CC2)cc1C(F)(F)F	C39H39F3N6O5	AR	P10275	CRBN	WO-2023139199-A1
TPD-RA7WON	SCHEMBL25935506	4-[4-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(N4CCC(CN5CCN(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3)CC2)cc1C(F)(F)F	C42H46F3N7O3	AR	P10275	CRBN	WO-2023139199-A1
TPD-E5301T	SCHEMBL25935629	4-[4-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]propylamino]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(NCCCN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)cc3)CC2)cc1C(F)(F)F	C39H42F3N7O3	AR	P10275	CRBN	WO-2023139199-A1
TPD-YKOPSV	SCHEMBL25935690	4-[4-[4-[4-[[4-[1-(2,6-Dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	Cn1c(=O)n(C2CCC(=O)NC2=O)c2ccc(N3CCN(CC4CCN(c5ccc(C6CCN(c7ccc(C#N)c(C(F)(F)F)c7)CC6)cc5)CC4)CC3)cc21	C42H47F3N8O3	AR	P10275	CRBN	WO-2023139199-A1
TPD-CNMPMP	WO2023139199A1_117	4-[4-[4-[4-[4-[6-(2,6-dioxopiperidin-3-yl)-4-methoxy-5-oxo-7H-pyrrolo[3,4-b]pyridin-2-yl]piperazin-1-yl]butoxy]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	COc1cc(N2CCN(CCCCOc3ccc(C4CCN(c5ccc(C#N)c(C(F)(F)F)c5)CC4)cc3)CC2)nc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C40H44F3N7O5	AR	P10275	CRBN	WO-2023139199-A1
TPD-JWJE4Q	WO2023139199A1_118	.	CC(F)(F)c1cc(N2CCC(c3ccc(N4CCC5(CCN(CC6CCN(c7ccc8c(c7)CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)CC4)cc3)CC2)ccc1C#N	C48H57F2N7O3	AR	P10275	CRBN	WO-2023139199-A1
TPD-B1RW7N	SCHEMBL30493381	4-[4-[4-[5-[4-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]pentoxy]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	COc1cc(N2CCN(CCCCCOc3ccc(C4CCN(c5ccc(C#N)c(C(F)(F)F)c5)CC4)cc3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C42H47F3N6O5	AR	P10275	CRBN	WO-2023139199-A1
TPD-EEVR2V	WO2023139199A1_120	4-[4-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-4-methoxy-3-oxo-1H-pyrrolo[3,4-c]pyridin-6-yl]piperazin-1-yl]butoxy]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	COc1nc(N2CCN(CCCCOc3ccc(C4CCN(c5ccc(C#N)c(C(F)(F)F)c5)CC4)cc3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C40H44F3N7O5	AR	P10275	CRBN	WO-2023139199-A1
TPD-KBGBXJ	SCHEMBL25427786	4-[4-[4-[4-[4-[4-chloro-2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]butoxy]-2-fluorophenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile; SCHEMBL30493234	COc1cc(N2CCN(CCCCOc3ccc(C4CCN(c5ccc(C#N)c(C(F)(F)F)c5)CC4)c(F)c3)CC2)c(Cl)c2c1C(=O)N(C1CCC(=O)NC1=O)C2	C41H43ClF4N6O5	AR	P10275	CRBN	WO-2023139199-A1
TPD-NJ26VH	SCHEMBL25430363	4-[4-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]butoxy]-2-fluorophenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile; SCHEMBL30493216	COc1cc(N2CCN(CCCCOc3ccc(C4CCN(c5ccc(C#N)c(C(F)(F)F)c5)CC4)c(F)c3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C41H44F4N6O5	AR	P10275	CRBN	WO-2023139199-A1
TPD-LD1H6Z	SCHEMBL25428302	4-[4-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]butoxy]-2-methylphenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile; SCHEMBL30493299; SCHEMBL30493300	COc1cc(N2CCN(CCCCOc3ccc(C4CCN(c5ccc(C#N)c(C(F)(F)F)c5)CC4)c(C)c3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C42H47F3N6O5	AR	P10275	CRBN	WO-2023139199-A1
TPD-6G9N5X	WO2023139199A1_124	4-[4-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]butyl]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(CCCCN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)cc3)CC2)cc1C(F)(F)F	C40H43F3N6O3	AR	P10275	CRBN	WO-2023139199-A1
TPD-3S177R	WO2023139199A1_125	.	COc1cc(N2CCN(C[C@H]3C[C@H](COc4ccc(C5CCN(c6ccc(C#N)c(C(F)(F)F)c6)CC5)cc4)C3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C43H47F3N6O5	AR	P10275	CRBN	WO-2023139199-A1
TPD-8LWC64	WO2023139199A1_126	.	COc1cc(N2CCN(C[C@H]3C[C@@H](COc4ccc(C5CCN(c6ccc(C#N)c(C(F)(F)F)c6)CC5)cc4)C3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C43H47F3N6O5	AR	P10275	CRBN	WO-2023139199-A1
TPD-15VUP4	SCHEMBL25936889	4-[4-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]butoxy]phenyl]azepan-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCCC(c3ccc(OCCCCN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)cc3)CC2)cc1C(F)(F)F	C41H45F3N6O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-G53YS7	SCHEMBL25937109	4-[4-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-3,6-dihydro-2H-pyridin-1-yl]butoxy]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(OCCCCN4CC=C(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)cc3)CC2)cc1C(F)(F)F	C41H42F3N5O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-RJ6SYA	SCHEMBL25937184	4-[4-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]butoxy]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(OCCCCN4CCC(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)cc3)CC2)cc1C(F)(F)F	C41H44F3N5O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-YD2SWH	SCHEMBL25937402	4-[4-[4-[4-[4-[7-chloro-2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]butoxy]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(OCCCCN4CCN(c5cc(Cl)c6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)cc3)CC2)cc1C(F)(F)F	C40H42ClF3N6O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-1RLJJ7	SCHEMBL25937595	4-[4-[4-[4-[4-[7-(difluoromethoxy)-2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]butoxy]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(OCCCCN4CCN(c5cc6c(c(OC(F)F)c5)C(=O)N(C5CCC(=O)NC5=O)C6)CC4)cc3)CC2)cc1C(F)(F)F	C41H43F5N6O5	AR	P10275	CRBN	WO-2023139199-A1
TPD-49ED3L	SCHEMBL25937730	4-[4-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-4-methoxy-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]butoxy]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	COc1c(N2CCN(CCCCOc3ccc(C4CCN(c5ccc(C#N)c(C(F)(F)F)c5)CC4)cc3)CC2)ccc2c1CN(C1CCC(=O)NC1=O)C2=O	C41H45F3N6O5	AR	P10275	CRBN	WO-2023139199-A1
TPD-5MBJ6Q	SCHEMBL25937811	4-[4-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-6-methoxy-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]butoxy]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	COc1cc2c(cc1N1CCN(CCCCOc3ccc(C4CCN(c5ccc(C#N)c(C(F)(F)F)c5)CC4)cc3)CC1)CN(C1CCC(=O)NC1=O)C2=O	C41H45F3N6O5	AR	P10275	CRBN	WO-2023139199-A1
TPD-NA74GP	SCHEMBL25937822	4-[4-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-4-methoxy-3-oxo-1H-pyrrolo[3,4-c]pyridin-6-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	COc1nc(N2CCN(CC3CCN(c4ccc(C5CCN(c6ccc(C#N)c(C(F)(F)F)c6)CC5)cc4)CC3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C42H47F3N8O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-NMZA9E	WO2023139199A1_136	4-[4-[4-[[3-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]-3-azaspiro[5.5]undecan-9-yl]oxy]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(OC4CCC5(CC4)CCN(CC4CCN(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC4)CC5)cc3)CC2)cc1C(F)(F)F	C48H55F3N6O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-0O5URK	WO2023139199A1_137	4-[4-[2-cyano-4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]butoxy]phenyl]piperidin-1-yl]-3-fluoro-2-(trifluoromethyl)benzonitrile	N#Cc1cc(OCCCCN2CCN(c3ccc4c(c3)CN(C3CCC(=O)NC3=O)C4=O)CC2)ccc1C1CCN(c2ccc(C#N)c(C(F)(F)F)c2F)CC1	C41H41F4N7O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-9HUKRO	WO2023139199A1_138	4-[4-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-4-methoxy-3-oxo-1H-pyrrolo[3,4-c]pyridin-6-yl]piperazin-1-yl]methyl]piperidin-1-yl]-2,6-difluorophenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	COc1nc(N2CCN(CC3CCN(c4cc(F)c(C5CCN(c6ccc(C#N)c(C(F)(F)F)c6)CC5)c(F)c4)CC3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C42H45F5N8O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-YLA3ZB	WO2023139199A1_139	4-[(3S)-4-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]-3-methylpiperazin-1-yl]-3-fluoro-2-(trifluoromethyl)benzonitrile	COc1cc(N2CCN(CC3CCN(c4ccc(N5CCN(c6ccc(C#N)c(C(F)(F)F)c6F)C[C@@H]5C)cc4)CC3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C43H48F4N8O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-LIGJN4	SCHEMBL25938448	4-[(2R)-4-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]-2-methylpiperazin-1-yl]-2-(trifluoromethyl)benzonitrile	COc1cc(N2CCN(CC3CCN(c4ccc(N5CCN(c6ccc(C#N)c(C(F)(F)F)c6)[C@H](C)C5)cc4)CC3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C43H49F3N8O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-GF9TLH	SCHEMBL25938457	4-[(2S)-4-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]-2-methylpiperazin-1-yl]-2-(trifluoromethyl)benzonitrile	COc1cc(N2CCN(CC3CCN(c4ccc(N5CCN(c6ccc(C#N)c(C(F)(F)F)c6)[C@@H](C)C5)cc4)CC3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C43H49F3N8O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-U7CJK6	WO2023139199A1_142	.	COc1cc(N2CCN(CC3CCN(c4ccc([C@H]5CCN(c6ccc(C#N)c(C(F)(F)F)c6F)C[C@H]5C)cc4)CC3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C44H49F4N7O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-2JM681	WO2023139199A1_143	.	COc1cc(N2CCN(CC3CCN(c4ccc(C5CCN(c6ccc(C#N)c(C(F)(F)F)c6F)C[C@@H]5C)cc4)CC3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C44H49F4N7O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-KZDQ6N	WO2023139199A1_144	4-[4-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-3-ethyl-2-(trifluoromethyl)benzonitrile	CCc1c(N2CCC(c3ccc(N4CCC(CN5CCN(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3)CC2)ccc(C#N)c1C(F)(F)F	C44H50F3N7O3	AR	P10275	CRBN	WO-2023139199-A1
TPD-BZTMYG	SCHEMBL25939107	4-[4-[4-[4-[4-[4-(2,4-Dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]butoxy]-2-fluorophenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(OCCCCN4CCC(n5ccc6c(N7CCC(=O)NC7=O)cccc65)CC4)cc3F)CC2)cc1C(F)(F)F	C40H42F4N6O3	AR	P10275	CRBN	WO-2023139199-A1
TPD-LKAOCG	SCHEMBL25939331	4-[4-[4-[4-[[4-[6-(2,4-Dioxo-1,3-diazinan-1-yl)-1-methylpyrrolo[3,2-b]pyridin-2-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-3-fluoro-2-(trifluoromethyl)benzonitrile	Cn1c(C2CCN(CC3CCN(c4ccc(C5CCN(c6ccc(C#N)c(C(F)(F)F)c6F)CC5)cc4)CC3)CC2)cc2ncc(N3CCC(=O)NC3=O)cc21	C42H46F4N8O2	AR	P10275	CRBN	WO-2023139199-A1
TPD-KKSBS8	SCHEMBL25939362	4-[4-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]-2,6-difluorophenyl]piperidin-1-yl]-3-fluoro-2-(trifluoromethyl)benzonitrile	COc1cc(N2CCN(CC3CCN(c4cc(F)c(C5CCN(c6ccc(C#N)c(C(F)(F)F)c6F)CC5)c(F)c4)CC3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C43H45F6N7O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-Y37Y2B	SCHEMBL25939458	4-[4-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]-2-fluorophenyl]piperidin-1-yl]-3-fluoro-2-(trifluoromethyl)benzonitrile	COc1cc(N2CCN(CC3CCN(c4ccc(C5CCN(c6ccc(C#N)c(C(F)(F)F)c6F)CC5)c(F)c4)CC3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C43H46F5N7O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-VW9FH3	SCHEMBL25939778	4-[4-[4-[4-[[4-[[1-(2,6-Dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-4-yl]methyl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-3-fluoro-2-(trifluoromethyl)benzonitrile	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(CN3CCN(CC4CCN(c5ccc(C6CCN(c7ccc(C#N)c(C(F)(F)F)c7F)CC6)cc5)CC4)CC3)c21	C43H48F4N8O3	AR	P10275	CRBN	WO-2023139199-A1
TPD-UEAOO8	WO2023139199A1_150	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C3CCN(CC4CCN(c5ccc(C6CCN(c7ccc(C#N)c(C(F)(F)F)c7F)CC6)cc5)CC4)CC3)c21	C43H47F4N7O3	AR	P10275	CRBN	WO-2023139199-A1
TPD-BDE4O5	SCHEMBL25940079	4-[4-[4-[[1-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]ethyl]azetidin-3-yl]methoxy]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(OCC4CN(CCN5CCN(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC5)C4)cc3)CC2)cc1C(F)(F)F	C42H46F3N7O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-LJAKH3	SCHEMBL25940139	4-[4-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-4-methoxy-3-oxo-1H-pyrrolo[3,4-c]pyridin-6-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-3-fluoro-2-(trifluoromethyl)benzonitrile	COc1nc(N2CCN(CC3CCN(c4ccc(C5CCN(c6ccc(C#N)c(C(F)(F)F)c6F)CC5)cc4)CC3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C42H46F4N8O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-3YBWUF	SCHEMBL25940465	4-[4-[4-[4-[[4-[6-(2,4-Dioxo-1,3-diazinan-1-yl)-1-methylindol-2-yl]piperidin-1-yl]methyl]piperidin-1-yl]-2,6-difluorophenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	Cn1c(C2CCN(CC3CCN(c4cc(F)c(C5CCN(c6ccc(C#N)c(C(F)(F)F)c6)CC5)c(F)c4)CC3)CC2)cc2ccc(N3CCC(=O)NC3=O)cc21	C43H46F5N7O2	AR	P10275	CRBN	WO-2023139199-A1
TPD-LQTPYE	SCHEMBL25940558	4-[4-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]-2,6-difluorophenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	COc1cc(N2CCN(CC3CCN(c4cc(F)c(C5CCN(c6ccc(C#N)c(C(F)(F)F)c6)CC5)c(F)c4)CC3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C43H46F5N7O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-TZ4HSQ	WO2023139199A1_155	.	Cc1c(N2CCC(c3ccc(N4CCC(CN5CCC(c6cc7ccc(N8CCC(=O)NC8=O)cc7n6C)CC5)CC4)cc3)CC2)ccc(C#N)c1C(F)(F)F	C44H50F3N7O2	AR	P10275	CRBN	WO-2023139199-A1
TPD-6US0ST	WO2023139199A1_156	4-[4-[4-[4-[[4-[6-(2,6-dioxopiperidin-3-yl)-5-oxo-7H-pyrrolo[3,4-b]pyridin-2-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-3-fluoro-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(N4CCC(CN5CCN(c6ccc7c(n6)CN(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3)CC2)c(F)c1C(F)(F)F	C41H44F4N8O3	AR	P10275	CRBN	WO-2023139199-A1
TPD-2TQYEL	SCHEMBL25941024	4-[4-[4-[4-[4-[6-(2,4-Dioxo-1,3-diazinan-1-yl)-1-methylindol-2-yl]piperidin-1-yl]butoxy]-2-fluorophenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	Cn1c(C2CCN(CCCCOc3ccc(C4CCN(c5ccc(C#N)c(C(F)(F)F)c5)CC4)c(F)c3)CC2)cc2ccc(N3CCC(=O)NC3=O)cc21	C41H44F4N6O3	AR	P10275	CRBN	WO-2023139199-A1
TPD-9J6MHQ	WO2023139199A1_158	4-[4-[4-[4-[4-[5-(2,4-Dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]butoxy]-2-fluorophenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(OCCCCN4CCC(n5ccc6cc(N7CCC(=O)NC7=O)ccc65)CC4)cc3F)CC2)cc1C(F)(F)F	C40H42F4N6O3	AR	P10275	CRBN	WO-2023139199-A1
TPD-PKWX16	SCHEMBL25941617	4-[4-[4-[3-[4-[6-(2,4-Dioxo-1,3-diazinan-1-yl)-4-fluoro-1-methylindol-2-yl]piperidin-1-yl]propoxy]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	Cn1c(C2CCN(CCCOc3ccc(C4CCN(c5ccc(C#N)c(C(F)(F)F)c5)CC4)cc3)CC2)cc2c(F)cc(N3CCC(=O)NC3=O)cc21	C40H42F4N6O3	AR	P10275	CRBN	WO-2023139199-A1
TPD-20JS7W	SCHEMBL25941676	4-[4-[4-[3-[4-[6-(2,4-Dioxo-1,3-diazinan-1-yl)-5-fluoro-1-methylindol-2-yl]piperidin-1-yl]propoxy]phenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	Cn1c(C2CCN(CCCOc3ccc(C4CCN(c5ccc(C#N)c(C(F)(F)F)c5)CC4)cc3)CC2)cc2cc(F)c(N3CCC(=O)NC3=O)cc21	C40H42F4N6O3	AR	P10275	CRBN	WO-2023139199-A1
TPD-IGAR4N	SCHEMBL25941691	4-[4-[4-[4-[4-[6-(2,6-dioxopiperidin-3-yl)-5-oxo-7H-pyrrolo[3,4-b]pyridin-2-yl]piperazin-1-yl]butoxy]-2-fluorophenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(OCCCCN4CCN(c5ccc6c(n5)CN(C5CCC(=O)NC5=O)C6=O)CC4)cc3F)CC2)cc1C(F)(F)F	C39H41F4N7O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-KXI6S3	WO2023139199A1_162	4-[4-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]butoxy]-2,6-difluorophenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3c(F)cc(OCCCCN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)cc3F)CC2)cc1C(F)(F)F	C40H41F5N6O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-X4ZL6G	WO2023139199A1_163	4-[4-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]butoxy]-2,6-difluorophenyl]piperidin-1-yl]-2-(trifluoromethyl)benzonitrile	COc1cc(N2CCN(CCCCOc3cc(F)c(C4CCN(c5ccc(C#N)c(C(F)(F)F)c5)CC4)c(F)c3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C41H43F5N6O5	AR	P10275	CRBN	WO-2023139199-A1
TPD-0FSCSW	SCHEMBL25942028	4-[4-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]butoxy]-2-fluorophenyl]piperidin-1-yl]-3-fluoro-2-(trifluoromethyl)benzonitrile	N#Cc1ccc(N2CCC(c3ccc(OCCCCN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)cc3F)CC2)c(F)c1C(F)(F)F	C40H41F5N6O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-94LRQ3	SCHEMBL25942182	4-[4-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]butoxy]-2-methylphenyl]piperidin-1-yl]-3-fluoro-2-(trifluoromethyl)benzonitrile	Cc1cc(OCCCCN2CCN(c3ccc4c(c3)CN(C3CCC(=O)NC3=O)C4=O)CC2)ccc1C1CCN(c2ccc(C#N)c(C(F)(F)F)c2F)CC1	C41H44F4N6O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-BSRWVA	WO2023139199A1_166	.	COc1cc(N2CCN(CCCCOc3ccc(C4CCN(c5ccc(C#N)c(C(C)(F)F)c5F)CC4)c(F)c3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C42H46F4N6O5	AR	P10275	CRBN	WO-2023139199-A1
TPD-6KQJQF	SCHEMBL25942408	2-cyclopropyl-4-[4-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]-2-fluorophenyl]piperidin-1-yl]benzonitrile	COc1cc(N2CCN(CC3CCN(c4ccc(C5CCN(c6ccc(C#N)c(C7CC7)c6)CC5)c(F)c4)CC3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C45H52FN7O4	AR	P10275	CRBN	WO-2023139199-A1
TPD-BXT69O	WO2023143384A1_1	.	NC1=C(C2=NC3=C(N=C(C4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C=C3)N2)C(=O)NC2=C1C=CS2	C37H37N9O5S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-RFG218	WO2023143384A1_2	.	NC1=C(C2=NC3=C(N=C(C4CCN(CC5CCN(C6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)CC5)CC4)C=C3)N2)C(=O)NC2=C1C=CS2	C42H46N10O5S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-C45HKZ	WO2023143384A1_3	.	NC1=C(C2=NC3=C(N=C(C4CCN(C5CCN(C6CN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)C6)CC5)CC4)C=C3)N2)C(=O)NC2=C1C=CS2	C39H40N10O5S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-XCVLMG	WO2023143384A1_4	.	NC1=C(C2=NC3=C(N=C(C4CCN(C5CCN(CC6CN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)C6)CC5)CC4)C=C3)N2)C(=O)NC2=C1C=CS2	C40H42N10O5S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-5J65L5	WO2023143384A1_5	.	NC1=C(C2=NC3C=CC(C4CCN(CCC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)=NC3N2)C(=O)NC2=C1C=CS2	C38H41N9O5S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-L59H6W	WO2023143384A1_6	.	NC1=C(C2=NC3=C(N=C(C4CCN(CC5CN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)C=C3)N2)C(=O)NC2=C1C=CS2	C35H33N9O5S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-VX0GO7	WO2023143384A1_7	.	NC1=C(C2=NC3=C(N=C(C4CCN(CC5CN(C6=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)C5)CC4)C=C3)N2)C(=O)NC2=C1C=CS2	C35H33N9O5S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-KIZOWY	WO2023143384A1_8	.	NC1=C(C2=NC3=C(N=C(C4CCN(CC5CN(C6=CC7=C(C=C6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)C=C3)N2)C(=O)NC2=C1C=CS2	C35H32FN9O5S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-8N31CZ	WO2023143384A1_9	.	NC1=C(C2=NC3=C(N=C(C4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C3)N2)C(=O)NC2=C1C=CS2	C36H35N9O5S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-OBE9ZO	WO2023143384A1_10	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=CC(CN3CCC(C4=NC5=C(C=C4)N=C(C4=C(N)C6=C(NC4=O)SC=C6)N5)CC3)=C21	C32H31N9O4S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-KULKHV	WO2023143384A1_11	.	NC1=C(C2=NC3=C(C=C(N4CCN(CC5CN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C3)N2)C(=O)NC2=C1[Se]C=C2	C35H33N9O5Se	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-G8K3JJ	WO2023143384A1_12	.	NC1=C(C2=NC3=C(N=C(C4CCN(CC5CN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C3)N2)C(=O)NC2=C1[Se]C=C2	C35H33N9O5Se	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-HP29PO	WO2023143384A1_13	.	CN1N=C(C2CCC(=O)NC2=O)C2=CC=CC(CN3CCC(C4=NC5=C(C=C4)N=C(C4=C(N)C6=C(NC4=O)SC=C6)N5)CC3)=C21	C32H31N9O3S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-8JKFP4	WO2023143384A1_14	.	NC1=C(C2=NC3=C(C=C(C4CCN(CC5CN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C3)N2)C(=O)NC2=C1C=CS2	C36H34N8O5S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-NK3PT3	WO2023143384A1_15	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=CC(CN3CC(CN4CCC(C5=NC6=C(C=C5)N=C(C5=C(N)C7=C(NC5=O)SC=C7)N6)CC4)C3)=C21	C36H38N10O4S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-L32AM1	WO2023143384A1_16	.	NC1=C(C2=NC3=C(C=C(N4CCC5(CC4)CN(C4=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C4)C5)C=C3)N2)C(=O)NC2=C1C=CS2	C34H30N8O5S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-ZAYW3E	WO2023143384A1_17	.	NC1=C(C2=NC3=C(N=C(C4CCN(CC5CN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C3)N2)C(=O)NC2=C1C1=C(CCC1)S2	C38H37N9O5S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-D91GE9	WO2023143384A1_18	.	NC1=C(C2=NC3=C(C=C(N4CCC5(CC4)CN(CC4=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C4)C5)C=C3)N2)C(=O)NC2=C1C=CS2	C35H32N8O5S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-WA9DQ4	WO2023143384A1_19	.	NC1=C(C2=NC3=C(C=C(N4CCC5(CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C=C3)N2)C(=O)NC2=C1C=CS2	C36H34N8O5S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-LGLZ3T	WO2023143384A1_20	.	NC1=C(C2=NC3=C(C=C(N4CCN(CC5CN(C6=CC=C(NC7CCC(=O)NC7=O)C=C6F)C5)CC4)C=C3)N2)C(=O)NC2=C1C=CS2	C33H34FN9O3S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-U2GONH	WO2023143384A1_21	.	O=C1CCC(N2C(=O)C3=CC=C(N4CC(CN5CCN(C6=CC7=C(C=C6)N=C(C6=CC8=C(C=CS8)NC6=O)N7)CC5)C4)C=C3C2=O)C(=O)N1	C35H32N8O5S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-H7UQZX	WO2023143384A1_22	.	NC1=C(C2=NC3=C(C=C(N4CCN(C5CC6(CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)C5)CC4)C=C3)N2)C(=O)NC2=C1C=CS2	C39H39N9O5S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-QM1CO5	WO2023143384A1_23	.	NC1=C(C2=NC3=C(C=C(N4CCN(CC5CN(C6=CC=C(C7CCC(=O)NC7=O)C=C6)C5)CC4)C=C3)N2)C(=O)NC2=C1C=CS2	C33H34N8O3S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-YN3151	WO2023143384A1_24	.	NC1=C(C2=NC3=C(C=C(N4CCN(CC5CN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C3)N2)C(=O)NC2=C1C=CS2	C35H33N9O5S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-BLGG5T	WO2023143384A1_25	.	NC1=C(C2=NC3=C(C=C(C4CCN(CC5CN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C3)N2)C(=O)NC2=C1[Se]C=C2	C36H34N8O5Se	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-CMYKZG	WO2023143384A1_26	.	NC1=C(C2=NC3=C(C=C(N4CCN(CCC5=CC(F)=C(C6CCC(=O)NC6=O)C(F)=C5)CC4)C=C3)N2)C(=O)NC2=C1C=CS2	C31H29F2N7O3S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-PAAQPK	WO2023143384A1_27	.	NC1=C(C2=NC3=C(N2)C(F)=C(N2CCN(CC4CN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC2)C(F)=C3)C(=O)NC2=C1C=CS2	C35H31F2N9O5S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-JNBQ1G	WO2023143384A1_28	.	NC1=C(C2=NC3=C(C=C(N4CCN(CC5CN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)C(F)=C3)N2)C(=O)NC2=C1[Se]C=C2	C35H32FN9O5Se	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-YR13PU	WO2023143384A1_29	.	NC1=C(C2=NC3=C(N=C(C4CCN(C5CN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C3)N2)C(=O)NC2=C1C=CS2	C34H31N9O5S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-IOIC1W	WO2023143384A1_30	.	NC1=C(C2=NC3=C(N=C(C4CCN(C5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)CC4)C=C3)N2)C(=O)NC2=C1C=CS2	C31H26N8O5S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-ABYYJD	WO2023143384A1_31	.	NC1=C(C2=NC3=C(N=C(C4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)C=C3)N2)C(=O)NC2=C1C=CS2	C31H26N8O5S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-RH0DTO	WO2023143384A1_32	.	NC1=C(C2=NC3=C(C=C(N4CCN(CC5CN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C3)N2)C(=O)NC2=C1SC=C2	C35H33N9O5S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-GZ9AVV	WO2023143384A1_33	.	NC1=C(C2=NC3=C(C=C(N4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C=C3)N2)C(=O)NC2=C1[Se]C=C2	C37H37N9O5Se	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-9U0JNK	WO2023143384A1_34	.	NC1=C(C2=NC3=C(C=C(N4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C=C3)N2)C(=O)NC2=C1C=CS2	C37H37N9O5S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-4BI8XQ	WO2023143384A1_35	.	NC1=C(C2=NC3=C(C=C(N4CCN(CC5CN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)N=CC7=C6)C5)CC4)C=C3)N2)C(=O)NC2=C1C=CS2	C35H34N10O4S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-EOEXQA	WO2023143384A1_36	.	NC1=C(C2=NC3=C(C=C(N4CCN(CC5CN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C(F)=C3)N2)C(=O)NC2=C1C=CS2	C35H32FN9O5S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-WB3L59	WO2023143384A1_37	.	NC1=C(C2=NC3=C(C=C(N4CCN(CC5CN(C6=CN=C(C(=O)NC7CCC(=O)NC7=O)CC6)C5)CC4)C=C3)N2)C(=O)NC2=C1C=CS2	C33H36N10O4S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-NJULRF	WO2023143384A1_38	.	NC1=C(C2=NC3=C(C=C(N4CCN(CC5CN(C6=CC=C(C7CCC(=O)NC7=O)C=C6F)C5)CC4)C=C3)N2)C(=O)NC2=C1C=CS2	C33H33FN8O3S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-LANFLY	WO2023143384A1_39	.	NC1=C(C2=NC3=C(C=C(N4CCN(CC5(F)CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C=C3)N2)C(=O)NC2=C1[Se]C=C2	C37H36FN9O5Se	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-ZZOI9X	WO2023143384A1_40	.	NC1=C(C2=NC3=C(C=C(N4CCN(CC5CN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)N=C3)N2)C(=O)NC2=C1C=CS2	C34H32N10O5S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-1R8RAB	WO2023143384A1_41	.	NC1=C(C2=NC3=C(C=C(N4CCN(CC5CN(C6=CC(F)=C(C7CCC(=O)NC7=O)C(F)=C6)C5)CC4)C=C3)N2)C(=O)NC2=C1C=CS2	C33H32F2N8O3S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-ZI4GZF	WO2023143384A1_42	.	NC1=C(C2=NC3=C(C=C(N4CCN(CC5CN(C6=C7OCOC7=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C3)N2)C(=O)NC2=C1C=CS2	C36H33N9O7S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-3TO4G0	WO2023143384A1_43	.	NC1=C(C2=NC3=C(C=C(N4CCN(C5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C=C3)N2)C(=O)NC2=C1C=CS2	C36H35N9O5S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-KO0WD0	WO2023143384A1_44	.	NC1=C(C2=NC3=C(C=C(N4CCN(C5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C3)N2)C(=O)NC2=C1C=CS2	C35H33N9O5S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-5H4Y6G	WO2023143384A1_45	.	NC1=C(C2=NC3=C(C=C(N4CCN(C5CC6(C5)CN(C5=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C5)C6)CC4)C=C3)N2)C(=O)NC2=C1C=CS2	C37H35N9O5S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-XSCZLR	WO2023143384A1_46	.	NC1=C(C2=NC3=C(C=C(N4CCN(C5CCC6(CC5)CN(C5=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C5)C6)CC4)C=C3)N2)C(=O)NC2=C1C=CS2	C39H39N9O5S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-0FZEP2	WO2023143384A1_47	.	NC1=C(C2=NC3=C(C=C(N4CCN(C5C[C@@H]6CN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)C[C@@H]6C5)CC4)C=C3)N2)C(=O)NC2=C1C=CS2	C38H37N9O5S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-2G6QXR	WO2023143384A1_48	.	NC1=C(C2=NC3=C(C=C(N4CCN(C5CCN(C6=CC=C(C7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)N2)C(=O)NC2=C1C=CS2	C34H36N8O3S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-1GAIMU	WO2023143384A1_49	.	NC1=C(C2=NC3=C(C=C(N4CCN(C5CC6(C5)CN(C5=CC=C(C7CCC(=O)NC7=O)C=C5)C6)CC4)C=C3)N2)C(=O)NC2=C1C=CS2	C35H36N8O3S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-87SLBO	WO2023143384A1_50	.	NC1=C(C2=NC3=C(C=C(N4CCN(C5CCC6(CC5)CN(C5=CC=C(C7CCC(=O)NC7=O)C=C5)C6)CC4)C=C3)N2)C(=O)NC2=C1C=CS2	C37H40N8O3S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-RT79NG	WO2023143384A1_51	.	NC1=C(C2=NC3=C(C=C(N4CCN(C5CCN(C6=C(F)C=C(NC7CCC(=O)NC7=O)C=C6)CC5(F)F)CC4)C=C3)N2)C(=O)NC2=C1C=CS2	C34H34F3N9O3S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-UFRLTR	WO2023143384A1_52	.	NC1=C(C2=NC3=C(C=C(N4CCN(C5CCN(C6=C(F)C=C(NC7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)N2)C(=O)NC2=C1C=CS2	C34H36FN9O3S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-2QCN31	WO2023143384A1_53	.	NC1=C(C2=NC3=C(C=C(N4CCN(C5CN(C6=C(F)C=C(NC7CCC(=O)NC7=O)C=C6)C5)CC4)C=C3)N2)C(=O)NC2=C1C=CS2	C32H32FN9O3S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-ZLY4N0	WO2023143384A1_54	.	NC1=C(C2=NC3=C(C=C(N4CCN(CC5CCN(C6=CC=C(C7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)N2)C(=O)NC2=C1C=CS2	C35H38N8O3S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-ROTUHS	WO2023143384A1_55	.	NC1=C(C2=NC3=C(C=C(N4CCN(CC5CCN(C6=CC=C(C7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)N2)C(=O)NC2=C1SC=C2	C35H38N8O3S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-J3JZ3U	WO2023143384A1_56	.	NC1=C(C2=NC3=C(C=C(N4CCN(CC5CCN(C6=CC=C(C7CCC(=O)NC7=O)C(F)=C6)CC5)CC4)C=C3)N2)C(=O)NC2=C1C=CS2	C35H37FN8O3S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-NFPSAW	WO2023143384A1_57	.	NC1=C(C2=NC3=C(C=C(N4CCN(CC5CCN(C6=CC=C(C7CCC(=O)NC7=O)C=N6)CC5)CC4)C=C3)N2)C(=O)NC2=C1C=CS2	C34H37N9O3S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-KEPWWV	WO2023143384A1_58	.	NC1=C(C2=NC3=C(C=C(N4CCN(CC5CN(C6=CC=C(C7CCC(=O)NC7=O)C=C6)C5)CC4)C=C3)N2)C(=O)NC2=C1SC=C2	C33H34N8O3S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-ZQB4ZI	WO2023143384A1_59	.	NC1=C(C2=NC3=C(C=C(N4CCN(CC5CCN(C6=CC(F)=C(C7CCC(=O)NC7=O)C(F)=C6)CC5)CC4)C=C3)N2)C(=O)NC2=C1C=CS2	C35H36F2N8O3S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-687WSX	WO2023143384A1_60	.	NC1=C(C2=NC3=C(C=C(N4CCN(CC5CCN(C6=CC=C(C7CCC(=O)NC7=O)C=C6F)CC5)CC4)C=C3)N2)C(=O)NC2=C1C=CS2	C35H37FN8O3S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-QQ9Z4W	WO2023143384A1_61	.	NC1=C(C2=NC3=C(C=C(N4CCN(CC5CCN(C6=CC=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)N2)C(=O)NC2=C1C=CS2	C34H37N9O3S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-RX9RE5	WO2023143384A1_62	.	NC1=C(C2=NC3=C(C=C(N4CCN(CC5CN(C6=CC=C(C7CCC(=O)NC7=O)C=C6)C5)CC4)C(C4CC4)=C3)N2)C(=O)NC2=C1C=CS2	C36H38N8O3S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-C0EJVU	WO2023143384A1_63	.	NC1=C(C2=NC3=C(C=C(N4CCN(CC5CCN(C6=CC=C(C7CCC(=O)NC7=O)C=C6)CC5)CC4)C(F)=C3)N2)C(=O)NC2=C1C=CS2	C35H37FN8O3S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-7AH1WD	WO2023143384A1_64	.	COC1=CC2=C(C=C1N1CCN(CC3CN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)C3)CC1)NC(C1=C(N)C3=C(NC1=O)SC=C3)=N2	C36H35N9O6S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-YE4TN1	WO2023143384A1_65	.	NC1=C(C2=NC3=C(C=C(N4CCN(CC#CC5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)C=C3)N2)C(=O)NC2=C1C=CS2	C34H28N8O5S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-SRV2RT	WO2023143384A1_66	.	NC1=C(C2=NC3=C(C=C(N4CCC5(CCCN(C6CN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)C6)C5)CC4)C=C3)N2)C(=O)NC2=C1C=CS2	C39H39N9O5S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-6K2XER	WO2023143384A1_67	.	NC1=C(C2=NC3=C(C=C(N4CCN(C(=O)C5CN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C3)N2)C(=O)NC2=C1C=CS2	C35H31N9O6S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-DXSAHR	WO2023143384A1_68	.	NC1=C(C2=NC3=C(C=C(N4CCN(C5CCN(C6=CC=C(C7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)N2)C(=O)NC2=C1[Se]C=C2	C34H36N8O3Se	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-RAPHAS	WO2023143384A1_69	.	NC1=C(C2=NC3=C(C=C(N4CCN(CC5CN(C6=C(F)C=C(C7CCC(=O)NC7=O)C=C6)C5)CC4)C=C3)N2)C(=O)NC2=C1[Se]C=C2	C33H33FN8O3Se	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-207437	WO2023143384A1_70	.	NC1=C(C2=NC3=C(C=C(N4CCN(CC5CCN(C6=C(F)C=C(N7CCC(=O)NC7=O)C=C6F)CC5)CC4)C=C3)N2)C(=O)NC2=C1C=CS2	C34H35F2N9O3S	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-T6KK8X	WO2023143384A1_71	.	NC1=C(C2=NC3=C(C=C(N4CCN(CC5CN(C6=CC(F)=C(C7CCC(=O)NC7=O)C(F)=C6)C5)CC4)C=C3)N2)C(=O)NC2=C1[Se]C=C2	C33H32F2N8O3Se	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-3YR30I	WO2023143384A1_72	.	NC1=C(C2=NC3=C(C=C(N4CCN(CC5CN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)C(C4CC4)=C3)N2)C(=O)NC2=C1[Se]C=C2	C38H37N9O5Se	HPK1	Q92918	CRBN	WO-2023143384-A1
TPD-RWF9EE	WO2023143494A1_1	.	COC(=O)c1ccc(N(C(=O)COCCOCCN2C(=O)c3cccc(F)c3C2=O)c2ccc([N+](=O)[O-])c3nonc23)c(-c2ccc(C)cc2)c1	C35H28FN5O10	c-Myc	P01106	CRBN	WO-2023143494-A1
TPD-2EVNZY	WO2023143494A1_2	.	COC(=O)c1ccc(N(C(=O)COCCOCCN2C(=O)c3cccc(F)c3C2=O)c2ccc([N+](=O)[O-])c3nonc23)c(-c2ccc(C(C)(C)C)cc2)c1	C38H34FN5O10	c-Myc	P01106	CRBN	WO-2023143494-A1
TPD-BO8DWH	WO2023143494A1_3	.	CC(=O)c1ccc(N(C(=O)COCCOCCN2C(=O)c3cccc(F)c3C2=O)c2ccc([N+](=O)[O-])c3nonc23)c(-c2ccc(C)cc2)c1	C35H28FN5O9	c-Myc	P01106	CRBN	WO-2023143494-A1
TPD-IBIFDL	WO2023143494A1_4	.	Cc1ccc(-c2cc(C(N)=O)ccc2N(C(=O)COCCOCCN2C(=O)c3cccc(F)c3C2=O)C2=CC=C([N+](=O)[O-])C3NON=C23)cc1	C34H29FN6O9	c-Myc	P01106	CRBN	WO-2023143494-A1
TPD-X0GEZ4	WO2023143494A1_5	.	O=C1c2cccc(F)c2C(=O)N1CCOCCOCC(=O)N(c1ccccc1-c1ccccc1)c1ccc(NOO)c2nonc12	C32H26FN5O8	c-Myc	P01106	CRBN	WO-2023143494-A1
TPD-BBZFVU	WO2023143494A1_6	.	Cc1ccc(-c2ccccc2N(C(=O)COCCOCCN2C(=O)c3cccc(F)c3C2=O)c2ccc(NOO)c3nonc23)cc1	C33H28FN5O8	c-Myc	P01106	CRBN	WO-2023143494-A1
TPD-QJ55WR	WO2023143494A1_7	.	Cc1ccc(-c2cc(C(=O)O)ccc2N(C(=O)COCCOCCN2C(=O)c3cccc(F)c3C2=O)c2ccc([N+](=O)[O-])c3nonc23)cc1	C34H26FN5O10	c-Myc	P01106	CRBN	WO-2023143494-A1
TPD-IND79J	WO2023143494A1_8	.	Cc1ccc(-c2cc(F)ccc2N(C(=O)COCCOCCN2C(=O)c3cccc(F)c3C2=O)c2ccc([N+](=O)[O-])c3nonc23)cc1	C33H25F2N5O8	c-Myc	P01106	CRBN	WO-2023143494-A1
TPD-HH0A3W	WO2023143494A1_9	.	O=C1c2cccc(F)c2C(=O)N1CCOCCOCC(=O)N(c1ccccc1Br)c1ccc([N+](=O)[O-])c2nonc12	C26H19BrFN5O8	c-Myc	P01106	CRBN	WO-2023143494-A1
TPD-O8B6ES	WO2023143494A1_10	.	O=C1c2cccc(F)c2C(=O)N1CCOCCOCC(=O)N(c1ccccc1F)c1ccc(NOO)c2nonc12	C26H21F2N5O8	c-Myc	P01106	CRBN	WO-2023143494-A1
TPD-1WBBHI	WO2023143494A1_11	.	O=C1c2cccc(F)c2C(=O)N1CCOCCOCC(=O)N(c1ccccc1-c1cccnc1)c1ccc([N+](=O)[O-])c2nonc12	C31H23FN6O8	c-Myc	P01106	CRBN	WO-2023143494-A1
TPD-WG9IUS	WO2023143494A1_12	.	O=C1c2cccc(F)c2C(=O)N1CCOCCOCC(=O)N(c1ccccc1-c1cccc(C(F)(F)F)c1)c1ccc([N+](=O)[O-])c2nonc12	C33H23F4N5O8	c-Myc	P01106	CRBN	WO-2023143494-A1
TPD-BKN68Q	WO2023143494A1_13	.	COC(=O)c1ccc(N(C(=O)COCCOCCN2C(=O)c3cccc(F)c3C2=O)c2ccc([N+](=O)[O-])c3nonc23)c(-c2ccc(C(C)C)cc2)c1	C37H32FN5O10	c-Myc	P01106	CRBN	WO-2023143494-A1
TPD-D8QJPM	WO2023143494A1_14	.	Cc1ccc(-c2cc(C#N)ccc2N(C(=O)COCCOCCN2C(=O)c3cccc(F)c3C2=O)c2ccc([N+](=O)[O-])c3nonc23)cc1	C34H25FN6O8	c-Myc	P01106	CRBN	WO-2023143494-A1
TPD-9G7O4H	WO2023143494A1_15	.	COC(=O)c1ccc(N(C(=O)COCCOCCN2C(=O)c3cccc(F)c3C2=O)c2ccc([N+](=O)[O-])c3nonc23)c(-c2ccc(C(F)(F)F)cc2)c1	C35H25F4N5O10	c-Myc	P01106	CRBN	WO-2023143494-A1
TPD-DM2IOO	WO2023143494A1_16	.	O=C1c2cccc(F)c2C(=O)N1CCOCCOCC(=O)N(c1ccc(C(F)(F)F)cc1C1CC1)c1ccc(NOO)c2nonc12	C30H25F4N5O8	c-Myc	P01106	CRBN	WO-2023143494-A1
TPD-K1GSHD	WO2023143494A1_17	.	O=C1c2cccc(F)c2C(=O)N1CCOCCOCC(=O)N(c1ccc(F)cc1C1CC1)c1ccc(NOO)c2nonc12	C29H25F2N5O8	c-Myc	P01106	CRBN	WO-2023143494-A1
TPD-WY4RHV	WO2023143494A1_18	.	COC(=O)c1ccc(N(C(=O)COCCOCCN2C(=O)c3cccc(N)c3C2=O)c2ccc(NOO)c3nonc23)c(-c2ccc(C)cc2)c1	C35H32N6O10	c-Myc	P01106	CRBN	WO-2023143494-A1
TPD-RD6VW0	WO2023143494A1_19	.	O=C1c2ccc(F)cc2C(=O)N1CCOCCOCC(=O)N(c1ccc(F)cc1C1CC1)c1ccc(NOO)c2nonc12	C29H25F2N5O8	c-Myc	P01106	CRBN	WO-2023143494-A1
TPD-MVFK58	WO2023143494A1_20	.	COC(=O)c1ccc(N(C(=O)COCCOCCN2C(=O)c3cccc(F)c3C2=O)c2ccc(S(=O)(=O)N(C)C)c3nonc23)c(-c2ccc(C)cc2)c1	C37H34FN5O10S	c-Myc	P01106	CRBN	WO-2023143494-A1
TPD-DEXBJ1	WO2023143494A1_21	.	O=C1c2cccc(F)c2C(=O)N1CCOCCOCC(=O)N(c1cccc(F)c1)c1ccc(NOO)c2nonc12	C26H21F2N5O8	c-Myc	P01106	CRBN	WO-2023143494-A1
TPD-UOLDU3	WO2023143494A1_22	.	O=C1c2cccc(F)c2C(=O)N1CCOCCOCC(=O)N(c1ccc(F)cc1)c1ccc(NOO)c2nonc12	C26H21F2N5O8	c-Myc	P01106	CRBN	WO-2023143494-A1
TPD-9ZHV33	WO2023143494A1_23	.	O=C1c2cccc(F)c2C(=O)N1CCOCCOCC(=O)N(c1ccc(F)cn1)c1ccc(NOO)c2nonc12	C25H20F2N6O8	c-Myc	P01106	CRBN	WO-2023143494-A1
TPD-USC7II	WO2023143494A1_24	.	COC(=O)c1ccc(N(C(=O)COCCOCCN2C(=O)c3cccc(F)c3C2=O)c2ccc(NOO)c3nonc23)cc1	C28H24FN5O10	c-Myc	P01106	CRBN	WO-2023143494-A1
TPD-X2K31J	WO2023143494A1_25	.	O=C(OCc1ccccc1)c1ccc(N(C(=O)COCCOCCN2C(=O)c3cccc(F)c3C2=O)c2ccc([N+](=O)[O-])c3nonc23)cc1	C34H26FN5O10	c-Myc	P01106	CRBN	WO-2023143494-A1
TPD-9NCTXB	WO2023143494A1_26	.	Cc1ccc(-c2ccc(CN(C(=O)COCCOCCN3C(=O)c4cccc(F)c4C3=O)c3ccc(NOO)c4nonc34)cc2)cc1	C34H30FN5O8	c-Myc	P01106	CRBN	WO-2023143494-A1
TPD-5BQRX1	WO2023143494A1_27	.	O=C1c2cccc(F)c2C(=O)N1CCOCCOCC(=O)N(Cc1ccc(F)cc1)c1ccc(NOO)c2nonc12	C27H23F2N5O8	c-Myc	P01106	CRBN	WO-2023143494-A1
TPD-RYQYHI	WO2023143494A1_28	.	Cc1cc(F)ccc1CN(C(=O)COCCOCCN1C(=O)c2cccc(F)c2C1=O)c1ccc(NOO)c2nonc12	C28H25F2N5O8	c-Myc	P01106	CRBN	WO-2023143494-A1
TPD-HOG5AT	WO2023143494A1_29	.	O=C1c2ccccc2C(=O)N1CCCCCCCCN(Cc1ccc(F)cc1)c1ccc([N+](=O)[O-])c2nonc12	C29H28FN5O5	c-Myc	P01106	CRBN	WO-2023143494-A1
TPD-OKH4PU	WO2023143494A1_30	.	O=C(COc1ccc(N2C(=O)c3cccc(F)c3C2=O)cc1)NCCN(Cc1ccc(F)cc1)c1ccc([N+](=O)[O-])c2nonc12	C31H22F2N6O7	c-Myc	P01106	CRBN	WO-2023143494-A1
TPD-RZ116C	WO2023143494A1_31	.	O=C(CN1CCC(N2C(=O)c3cccc(F)c3C2=O)CC1)NCCN(Cc1ccc(F)cc1)c1ccc([N+](=O)[O-])c2nonc12	C30H27F2N7O6	c-Myc	P01106	CRBN	WO-2023143494-A1
TPD-ZPHDJS	WO2023143494A1_32	.	O=C(CCCCN1C(=O)c2cccc(F)c2C1=O)NCCN(Cc1ccc(F)cc1)c1ccc([N+](=O)[O-])c2nonc12	C28H24F2N6O6	c-Myc	P01106	CRBN	WO-2023143494-A1
TPD-9MFPJK	WO2023143494A1_33	.	O=C(COCCOCCN1C(=O)c2cccc(F)c2C1=O)NCCN(Cc1ccc(F)cc1)c1ccc(NOO)c2nonc12	C29H28F2N6O8	c-Myc	P01106	CRBN	WO-2023143494-A1
TPD-BR7PWR	WO2023143494A1_34	.	O=C1CCC(N2C(=O)c3cccc(NCCOCCOCC(=O)N(c4ccccc4-c4ccccc4)c4ccc(NOO)c5nonc45)c3C2=O)C(=O)N1	C37H33N7O10	c-Myc	P01106	CRBN	WO-2023143494-A1
TPD-HFET2H	WO2023143494A1_35	.	O=C1CCC(N2C(=O)c3cccc(NCCOCCOCCOCCC(=O)N(c4ccccc4-c4ccccc4)c4ccc(NOO)c5nonc45)c3C2=O)C(=O)N1	C40H39N7O11	c-Myc	P01106	CRBN	WO-2023143494-A1
TPD-N46IAS	WO2023143494A1_36	.	O=C1CCC(N2C(=O)c3cccc(NCCOCCC(=O)N(c4ccccc4-c4ccccc4)c4ccc(NOO)c5nonc45)c3C2=O)C(=O)N1	C36H31N7O9	c-Myc	P01106	CRBN	WO-2023143494-A1
TPD-W0ZSEX	WO2023143494A1_37	.	O=C(CN1CCC(CN2C(=O)c3cccc(F)c3C2=O)CC1)NCCN(Cc1ccc(F)cc1)c1ccc(NOO)c2nonc12	C31H31F2N7O6	c-Myc	P01106	CRBN	WO-2023143494-A1
TPD-UTO5WB	WO2023143494A1_38	.	O=C1c2cccc(F)c2C(=O)N1CCCCCCCC(=O)N(c1ccc(F)cc1C1CC1)c1ccc(NOO)c2nonc12	C31H29F2N5O6	c-Myc	P01106	CRBN	WO-2023143494-A1
TPD-T4B7UR	WO2023143494A1_39	.	O=C1c2cccc(F)c2C(=O)N1CCCCCCCC(=O)N(Cc1ccc(F)cc1)c1ccc(NOO)c2nonc12	C29H27F2N5O6	c-Myc	P01106	CRBN	WO-2023143494-A1
TPD-FINO6K	WO2023143494A1_40	.	O=C1c2cccc(F)c2C(=O)N1CC1CCN(CC(=O)N(c2ccc(F)cc2C2CC2)c2ccc(NOO)c3nonc23)CC1	C31H28F2N6O6	c-Myc	P01106	CRBN	WO-2023143494-A1
TPD-7SMKTG	WO2023143494A1_41	.	O=C1c2cccc(F)c2C(=O)N1CC1CCN(CC(=O)N(Cc2ccc(F)cc2)c2ccc(NOO)c3nonc23)CC1	C29H26F2N6O6	c-Myc	P01106	CRBN	WO-2023143494-A1
TPD-A6KG63	WO2023143494A1_42	.	O=C1c2cccc(F)c2C(=O)N1CCCCn1cc(C(=O)N(c2ccc(F)cc2C2CC2)c2ccc(NOO)c3nonc23)nn1	C30H24F2N8O6	c-Myc	P01106	CRBN	WO-2023143494-A1
TPD-JN4UA5	WO2023143494A1_43	.	O=C1c2cccc(F)c2C(=O)N1CCCCn1cc(C(=O)N(c2ccc(F)cc2C2CC2)c2ccc(NOO)c3nonc23)cn1	C31H25F2N7O6	c-Myc	P01106	CRBN	WO-2023143494-A1
TPD-GHO0T1	WO2023143494A1_44	.	O=C(CN1CC(N2C(=O)c3cccc(F)c3C2=O)C1)N(c1ccc(F)cc1C1CC1)c1ccc(NOO)c2nonc12	C28H22F2N6O6	c-Myc	P01106	CRBN	WO-2023143494-A1
TPD-P3UK6T	WO2023143494A1_45	.	O=C1c2cccc(F)c2C(=O)N1CCN1CCN(CC(=O)N(c2ccc(F)cc2C2CC2)c2ccc(NOO)c3nonc23)CC1	C31H29F2N7O6	c-Myc	P01106	CRBN	WO-2023143494-A1
TPD-BTJSLN	WO2023143494A1_46	.	O=C1c2cccc(F)c2C(=O)N1CCN1CCC(CC(=O)N(c2ccc(F)cc2C2CC2)c2ccc(NOO)c3nonc23)CC1	C32H30F2N6O6	c-Myc	P01106	CRBN	WO-2023143494-A1
TPD-Z1HWXC	WO2023143494A1_47	.	O=C1c2cccc(F)c2C(=O)N1CCN1CCN(CC(=O)N(Cc2ccc(F)cc2)c2ccc(NOO)c3nonc23)CC1	C29H27F2N7O6	c-Myc	P01106	CRBN	WO-2023143494-A1
TPD-4VISU0	WO2023143494A1_48	.	O=C1c2cccc(F)c2C(=O)N1CCN1CCC(CC(=O)N(Cc2ccc(F)cc2)c2ccc(NOO)c3nonc23)CC1	C30H28F2N6O6	c-Myc	P01106	CRBN	WO-2023143494-A1
TPD-F3PMGW	WO2023143494A1_49	.	O=C1c2cccc(F)c2C(=O)N1CC1CCN(CCC(=O)N(Cc2ccc(F)cc2)c2ccc(NOO)c3nonc23)CC1	C30H28F2N6O6	c-Myc	P01106	CRBN	WO-2023143494-A1
TPD-6JJE5Y	WO2023143494A1_50	.	O=C(CN(Cc1ccc(F)cc1)c1ccc(NOO)c2nonc12)N1CCC(CN2C(=O)c3cccc(F)c3C2=O)CC1	C29H26F2N6O6	c-Myc	P01106	CRBN	WO-2023143494-A1
TPD-E6T2MJ	SCHEMBL25342439	N-(2-cyclopropyl-4-fluorophenyl)-2-[4-[(4,7-difluoro-1,3-dioxoisoindol-2-yl)methyl]piperidin-1-yl]-N-(4-nitro-2,1,3-benzoxadiazol-7-yl)acetamide; SCHEMBL30520863	O=C1c2c(F)ccc(F)c2C(=O)N1CC1CCN(CC(=O)N(c2ccc(F)cc2C2CC2)c2ccc([N+](=O)[O-])c3nonc23)CC1	C31H25F3N6O6	c-Myc	P01106	CRBN	WO-2023143494-A1
TPD-CH5OBX	SCHEMBL25342833	3-[1'-[4-[[9-chloro-7-(2-fluoro-6-methoxyphenyl)-5H-pyrimido[5,4-d][2]benzazepin-2-yl]amino]-2-methoxybenzoyl]-6-oxospiro[4,8-dihydro-3H-pyrano[3,2-f]isoindole-2,4'-piperidine]-7-yl]piperidine-2,6-dione; SCHEMBL30520479	COc1cc(Nc2ncc3c(n2)-c2ccc(Cl)cc2C(c2c(F)cccc2OC)=NC3)ccc1C(=O)N1CCC2(CCc3cc4c(cc3O2)CN(C2CCC(=O)NC2=O)C4=O)CC1	C47H41ClFN7O7	AURKA	O14965	CRBN	WO-2023143589-A1
TPD-DO9LXD	SCHEMBL25340528	3-[1'-[4-[[9-chloro-7-(2-fluoro-6-methoxyphenyl)-5H-pyrimido[5,4-d][2]benzazepin-2-yl]amino]-2-methoxybenzoyl]-8-oxospiro[2,6-dihydro-[1,4]dioxino[2,3-f]isoindole-3,4'-piperidine]-7-yl]piperidine-2,6-dione; SCHEMBL30520283	COc1cc(Nc2ncc3c(n2)-c2ccc(Cl)cc2C(c2c(F)cccc2OC)=NC3)ccc1C(=O)N1CCC2(CC1)COc1cc3c(cc1O2)CN(C1CCC(=O)NC1=O)C3=O	C46H39ClFN7O8	AURKA	O14965	CRBN	WO-2023143589-A1
TPD-JWXZNY	SCHEMBL25343337	3-[1'-[4-[[9-chloro-7-(2-fluoro-6-methoxyphenyl)-5H-pyrimido[5,4-d][2]benzazepin-2-yl]amino]-2-methoxybenzoyl]-6-oxospiro[4,8-dihydro-3H-pyrano[3,2-f]isoindole-2,3'-azetidine]-7-yl]piperidine-2,6-dione; SCHEMBL30520273	COc1cc(Nc2ncc3c(n2)-c2ccc(Cl)cc2C(c2c(F)cccc2OC)=NC3)ccc1C(=O)N1CC2(CCc3cc4c(cc3O2)CN(C2CCC(=O)NC2=O)C4=O)C1	C45H37ClFN7O7	AURKA	O14965	CRBN	WO-2023143589-A1
TPD-OUHNG7	SCHEMBL25342481	3-[1'-[4-[[9-chloro-7-(2-fluoro-6-methoxyphenyl)-5H-pyrimido[5,4-d][2]benzazepin-2-yl]amino]-2-methoxybenzoyl]-8-oxospiro[4,6-dihydro-3H-pyrano[2,3-f]isoindole-2,3'-azetidine]-7-yl]piperidine-2,6-dione; SCHEMBL30520488	COc1cc(Nc2ncc3c(n2)-c2ccc(Cl)cc2C(c2c(F)cccc2OC)=NC3)ccc1C(=O)N1CC2(CCc3cc4c(cc3O2)C(=O)N(C2CCC(=O)NC2=O)C4)C1	C45H37ClFN7O7	AURKA	O14965	CRBN	WO-2023143589-A1
TPD-AO5RK8	SCHEMBL25343377	4-[[9-chloro-7-(2-fluoro-6-methoxyphenyl)-5H-pyrimido[5,4-d][2]benzazepin-2-yl]amino]-N-[2-[3-[7-(2,6-dioxopiperidin-3-yl)-6,8-dioxospiro[3,4-dihydropyrano[3,2-f]isoindole-2,4'-piperidine]-1'-yl]-3-oxopropoxy]ethyl]-2-methoxybenzamide; SCHEMBL30520470	COc1cc(Nc2ncc3c(n2)-c2ccc(Cl)cc2C(c2c(F)cccc2OC)=NC3)ccc1C(=O)NCCOCCC(=O)N1CCC2(CCc3cc4c(cc3O2)C(=O)N(C2CCC(=O)NC2=O)C4=O)CC1	C52H48ClFN8O10	AURKA	O14965	CRBN	WO-2023143589-A1
TPD-HQ01VD	SCHEMBL25340707	4-[[9-chloro-7-(2-fluoro-6-methoxyphenyl)-5H-pyrimido[5,4-d][2]benzazepin-2-yl]amino]-N-[2-[3-[7-(2,6-dioxopiperidin-3-yl)-6,8-dioxospiro[2,4-dihydropyrano[3,2-f]isoindole-3,4'-piperidine]-1'-yl]-3-oxopropoxy]ethyl]-2-methoxybenzamide; SCHEMBL30520459	COc1cc(Nc2ncc3c(n2)-c2ccc(Cl)cc2C(c2c(F)cccc2OC)=NC3)ccc1C(=O)NCCOCCC(=O)N1CCC2(CC1)COc1cc3c(cc1C2)C(=O)N(C1CCC(=O)NC1=O)C3=O	C52H48ClFN8O10	AURKA	O14965	CRBN	WO-2023143589-A1
TPD-ZTNIFN	SCHEMBL25344345	4-[[9-chloro-7-(2-fluoro-6-methoxyphenyl)-5H-pyrimido[5,4-d][2]benzazepin-2-yl]amino]-N-[2-[3-[6-(2,6-dioxopiperidin-3-yl)-5,7-dioxospiro[2H-furo[3,2-f]isoindole-3,4'-piperidine]-1'-yl]-3-oxopropoxy]ethyl]-2-methoxybenzamide; SCHEMBL31169234	COc1cc(Nc2ncc3c(n2)-c2ccc(Cl)cc2C(c2c(F)cccc2OC)=NC3)ccc1C(=O)NCCOCCC(=O)N1CCC2(CC1)COc1cc3c(cc12)C(=O)N(C1CCC(=O)NC1=O)C3=O	C51H46ClFN8O10	AURKA	O14965	CRBN	WO-2023143589-A1
TPD-WWLFCG	WO2023143589A1_8	4-[[9-chloro-7-(2-fluoro-6-methoxyphenyl)-5H-pyrimido[5,4-d][2]benzazepin-2-yl]amino]-N-[2-[3-[7-(2,6-dioxopiperidin-3-yl)-6,8-dioxospiro[3,4-dihydropyrano[3,2-f]isoindole-2,3'-azetidine]-1'-yl]-3-oxopropoxy]ethyl]-2-methoxybenzamide	COc1cc(Nc2ncc3c(n2)-c2ccc(Cl)cc2C(c2c(F)cccc2OC)=NC3)ccc1C(=O)NCCOCCC(=O)N1CC2(CCc3cc4c(cc3O2)C(=O)N(C2CCC(=O)NC2=O)C4=O)C1	C50H44ClFN8O10	AURKA	O14965	CRBN	WO-2023143589-A1
TPD-5QCOGG	WO2023143589A1_9	.	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3C)s2)cc(N2CCN(CCOCCC(=O)N3CCC4(CCc5cc6c(cc5O4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)CC2)n1	C46H52N10O8S	BCR-ABL	Q16189	CRBN	WO-2023143589-A1
TPD-9NPOXV	SCHEMBL25339738	N-(2-chloro-6-methylphenyl)-2-[[6-[4-[2-[3-[7-(2,6-dioxopiperidin-3-yl)-6,8-dioxospiro[2,4-dihydropyrano[3,2-f]isoindole-3,4'-piperidine]-1'-yl]-3-oxopropoxy]ethyl]piperazin-1-yl]-2-methylpyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide; SCHEMBL30520420	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCOCCC(=O)N3CCC4(CC3)COc3cc5c(cc3C4)C(=O)N(C3CCC(=O)NC3=O)C5=O)CC2)n1	C45H49ClN10O8S	BCR-ABL	Q16189	CRBN	WO-2023143589-A1
TPD-VBUA47	SCHEMBL25342991	N-(2-chloro-6-methylphenyl)-2-[[6-[4-[2-[3-[7-(2,6-dioxopiperidin-3-yl)-6,8-dioxospiro[3,4-dihydropyrano[3,2-f]isoindole-2,3'-azetidine]-1'-yl]-3-oxopropoxy]ethyl]piperazin-1-yl]-2-methylpyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide; SCHEMBL30520277	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCOCCC(=O)N3CC4(CCc5cc6c(cc5O4)C(=O)N(C4CCC(=O)NC4=O)C6=O)C3)CC2)n1	C43H45ClN10O8S	BCR-ABL	Q16189	CRBN	WO-2023143589-A1
TPD-QISNF4	SCHEMBL25342506	N-(2-chloro-6-methylphenyl)-2-[[6-[4-[2-[3-[6-(2,6-dioxopiperidin-3-yl)-5,7-dioxospiro[2H-furo[3,2-f]isoindole-3,4'-piperidine]-1'-yl]-3-oxopropoxy]ethyl]piperazin-1-yl]-2-methylpyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide; SCHEMBL30521001	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCOCCC(=O)N3CCC4(CC3)COc3cc5c(cc34)C(=O)N(C3CCC(=O)NC3=O)C5=O)CC2)n1	C44H47ClN10O8S	BCR-ABL	Q16189	CRBN	WO-2023143589-A1
TPD-QH29Y4	WO2023143589A1_13	.	Cc1nc(NC2NC=C(C(=O)Nc3c(C)cccc3Cl)S2)cc(N2CCN(CCOCCC(=O)N3CCC4(CCc5cc6c(cc5O4)C(=O)N(C4CCC(=O)NC4=O)C6)CC3)CC2)n1	C45H53ClN10O7S	BCR-ABL	Q16189	CRBN	WO-2023143589-A1
TPD-G7FHZG	WO2023143589A1_14	.	Cc1cc(N2CCN(CCOCCC(=O)N3CC4(CCc5cc6c(cc5O4)C(=O)N(C4CCC(=O)NC4=O)C6)C3)CC2)cc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)n1	C44H48ClN9O7S	BCR-ABL	Q16189	CRBN	WO-2023143589-A1
TPD-4QNBIN	SCHEMBL25342861	N-(2-chloro-6-methylphenyl)-2-[[6-[4-[2-[3-[7-(2,6-dioxopiperidin-3-yl)-8-oxospiro[2,6-dihydro-[1,4]dioxino[2,3-f]isoindole-3,4'-piperidine]-1'-yl]-3-oxopropoxy]ethyl]piperazin-1-yl]-2-methylpyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide; SCHEMBL30520440	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCOCCC(=O)N3CCC4(CC3)COc3cc5c(cc3O4)CN(C3CCC(=O)NC3=O)C5=O)CC2)n1	C44H49ClN10O8S	BCR-ABL	Q16189	CRBN	WO-2023143589-A1
TPD-S4YXYL	SCHEMBL25342629	N-(2-chloro-6-methylphenyl)-2-[[6-[4-[2-[3-[7-(2,6-dioxopiperidin-3-yl)-6-oxospiro[4,8-dihydro-3H-pyrano[3,2-f]isoindole-2,3'-azetidine]-1'-yl]-3-oxopropoxy]ethyl]piperazin-1-yl]-2-methylpyrimidin-4-yl]amino]-1,3-thiazole-5-carboxamide; SCHEMBL30520455	Cc1nc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)s2)cc(N2CCN(CCOCCC(=O)N3CC4(CCc5cc6c(cc5O4)CN(C4CCC(=O)NC4=O)C6=O)C3)CC2)n1	C43H47ClN10O7S	BCR-ABL	Q16189	CRBN	WO-2023143589-A1
TPD-N1U9O7	SCHEMBL25342938	3-[1'-[3-[2-[4-[3-[4-(3-chloro-4-fluoroanilino)-7-methoxyquinazolin-6-yl]oxypropyl]piperazin-1-yl]ethoxy]propanoyl]-8-oxospiro[4,6-dihydro-3H-pyrano[2,3-f]isoindole-2,4'-piperidine]-7-yl]piperidine-2,6-dione; SCHEMBL30520474	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1OCCCN1CCN(CCOCCC(=O)N2CCC3(CCc4cc5c(cc4O3)C(=O)N(C3CCC(=O)NC3=O)C5)CC2)CC1	C47H54ClFN8O8	EGFR	P00533	CRBN	WO-2023143589-A1
TPD-SNJ99C	SCHEMBL25432408	3-[1'-[3-[2-[4-[3-[4-(3-Chloro-4-fluoroanilino)-7-methoxyquinazolin-6-yl]oxypropyl]piperazin-1-yl]ethoxy]propanoyl]-8-oxospiro[2,6-dihydro-[1,4]dioxino[2,3-f]isoindole-3,4'-piperidine]-7-yl]piperidine-2,6-dione; SCHEMBL30520359	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1OCCCN1CCN(CCOCCC(=O)N2CCC3(CC2)COc2cc4c(cc2O3)CN(C2CCC(=O)NC2=O)C4=O)CC1	C46H52ClFN8O9	EGFR	P00533	CRBN	WO-2023143589-A1
TPD-JOCU7X	WO2023143589A1_19	.	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1OCCCN1CCN(CCOCCC(=O)N(C)CC2(C)CCc3cc4c(cc3O2)C(=O)N(C2CCC(=O)NC2=O)C4)CC1	C46H54ClFN8O8	EGFR	P00533	CRBN	WO-2023143589-A1
TPD-XRI3NY	WO2023143589A1_20	.	COc1cc2c(cc1OCCCN1CCN(CCOCCC(=O)N3CC4(CCc5cc6c(cc5O4)CN(C4CCC(=O)NC4=O)C6=O)C3)CC1)=C(Nc1ccc(F)c(Cl)c1)NCN=2	C45H52ClFN8O8	EGFR	P00533	CRBN	WO-2023143589-A1
TPD-J3IO93	SCHEMBL25341756	1'-[3-[2-[4-[3-[4-(3-Chloro-4-fluoroanilino)-7-methoxyquinazolin-6-yl]oxypropyl]piperazin-1-yl]ethoxy]propanoyl]-7-(2,6-dioxopiperidin-3-yl)spiro[3,4-dihydropyrano[3,2-f]isoindole-2,4'-piperidine]-6,8-dione; SCHEMBL30520274	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1OCCCN1CCN(CCOCCC(=O)N2CCC3(CCc4cc5c(cc4O3)C(=O)N(C3CCC(=O)NC3=O)C5=O)CC2)CC1	C47H52ClFN8O9	EGFR	P00533	CRBN	WO-2023143589-A1
TPD-RUPS5D	SCHEMBL25344510	1'-[3-[2-[4-[3-[4-(3-Chloro-4-fluoroanilino)-7-methoxyquinazolin-6-yl]oxypropyl]piperazin-1-yl]ethoxy]propanoyl]-7-(2,6-dioxopiperidin-3-yl)spiro[2,4-dihydropyrano[3,2-f]isoindole-3,4'-piperidine]-6,8-dione; SCHEMBL31192126	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1OCCCN1CCN(CCOCCC(=O)N2CCC3(CC2)COc2cc4c(cc2C3)C(=O)N(C2CCC(=O)NC2=O)C4=O)CC1	C47H52ClFN8O9	EGFR	P00533	CRBN	WO-2023143589-A1
TPD-1KXZ1D	SCHEMBL25342551	1'-[3-[2-[4-[3-[4-(3-Chloro-4-fluoroanilino)-7-methoxyquinazolin-6-yl]oxypropyl]piperazin-1-yl]ethoxy]propanoyl]-7-(2,6-dioxopiperidin-3-yl)spiro[3,4-dihydropyrano[3,2-f]isoindole-2,3'-azetidine]-6,8-dione; SCHEMBL30520398	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1OCCCN1CCN(CCOCCC(=O)N2CC3(CCc4cc5c(cc4O3)C(=O)N(C3CCC(=O)NC3=O)C5=O)C2)CC1	C45H48ClFN8O9	EGFR	P00533	CRBN	WO-2023143589-A1
TPD-0WW2M5	SCHEMBL25343365	1'-[3-[2-[4-[3-[4-(3-chloro-4-fluoroanilino)-7-methoxyquinazolin-6-yl]oxypropyl]piperazin-1-yl]ethoxy]propanoyl]-6-(2,6-dioxopiperidin-3-yl)spiro[2H-furo[3,2-f]isoindole-3,4'-piperidine]-5,7-dione	COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1OCCCN1CCN(CCOCCC(=O)N2CCC3(CC2)COc2cc4c(cc23)C(=O)N(C2CCC(=O)NC2=O)C4=O)CC1	C46H50ClFN8O9	EGFR	P00533	CRBN	WO-2023143589-A1
TPD-3UYWTT	SCHEMBL25342746	3-[1'-[3-[2-[4-[4-[[5-chloro-4-(2-propan-2-ylsulfonylanilino)pyrimidin-2-yl]amino]-2-methyl-5-propan-2-yloxyphenyl]piperidin-1-yl]ethoxy]propanoyl]-6-oxospiro[4,8-dihydro-3H-pyrano[3,2-f]isoindole-2,4'-piperidine]-7-yl]piperidine-2,6-dione; SCHEMBL30520284	Cc1cc(Nc2ncc(Cl)c(Nc3ccccc3S(=O)(=O)C(C)C)n2)c(OC(C)C)cc1C1CCN(CCOCCC(=O)N2CCC3(CCc4cc5c(cc4O3)CN(C3CCC(=O)NC3=O)C5=O)CC2)CC1	C53H65ClN8O9S	ALK	Q9UM73	CRBN	WO-2023143589-A1
TPD-ZGVBVI	SCHEMBL25341673	3-[1'-[3-[2-[4-[4-[[5-chloro-4-(2-propan-2-ylsulfonylanilino)pyrimidin-2-yl]amino]-2-methyl-5-propan-2-yloxyphenyl]piperidin-1-yl]ethoxy]propanoyl]-8-oxospiro[4,6-dihydro-3H-pyrano[2,3-f]isoindole-2,4'-piperidine]-7-yl]piperidine-2,6-dione; SCHEMBL30520387	Cc1cc(Nc2ncc(Cl)c(Nc3ccccc3S(=O)(=O)C(C)C)n2)c(OC(C)C)cc1C1CCN(CCOCCC(=O)N2CCC3(CCc4cc5c(cc4O3)C(=O)N(C3CCC(=O)NC3=O)C5)CC2)CC1	C53H65ClN8O9S	ALK	Q9UM73	CRBN	WO-2023143589-A1
TPD-YC8CPZ	SCHEMBL25342966	3-[1'-[3-[2-[4-[4-[[5-chloro-4-(2-propan-2-ylsulfonylanilino)pyrimidin-2-yl]amino]-2-methyl-5-propan-2-yloxyphenyl]piperidin-1-yl]ethoxy]propanoyl]-6-oxospiro[4,8-dihydro-3H-pyrano[3,2-f]isoindole-2,3'-azetidine]-7-yl]piperidine-2,6-dione; SCHEMBL30520306	Cc1cc(Nc2ncc(Cl)c(Nc3ccccc3S(=O)(=O)C(C)C)n2)c(OC(C)C)cc1C1CCN(CCOCCC(=O)N2CC3(CCc4cc5c(cc4O3)CN(C3CCC(=O)NC3=O)C5=O)C2)CC1	C51H61ClN8O9S	ALK	Q9UM73	CRBN	WO-2023143589-A1
TPD-LMKZ6V	SCHEMBL25342871	3-[1'-[3-[2-[4-[4-[[5-chloro-4-(2-propan-2-ylsulfonylanilino)pyrimidin-2-yl]amino]-2-methyl-5-propan-2-yloxyphenyl]piperidin-1-yl]ethoxy]propanoyl]-8-oxospiro[4,6-dihydro-3H-pyrano[2,3-f]isoindole-2,3'-azetidine]-7-yl]piperidine-2,6-dione; SCHEMBL30520362	Cc1cc(Nc2ncc(Cl)c(Nc3ccccc3S(=O)(=O)C(C)C)n2)c(OC(C)C)cc1C1CCN(CCOCCC(=O)N2CC3(CCc4cc5c(cc4O3)C(=O)N(C3CCC(=O)NC3=O)C5)C2)CC1	C51H61ClN8O9S	ALK	Q9UM73	CRBN	WO-2023143589-A1
TPD-Q0NWB7	SCHEMBL25340633	1'-[3-[2-[4-[4-[[5-Chloro-4-(2-propan-2-ylsulfonylanilino)pyrimidin-2-yl]amino]-2-methyl-5-propan-2-yloxyphenyl]piperidin-1-yl]ethoxy]propanoyl]-7-(2,6-dioxopiperidin-3-yl)spiro[3,4-dihydropyrano[3,2-f]isoindole-2,4'-piperidine]-6,8-dione; SCHEMBL30520439	Cc1cc(Nc2ncc(Cl)c(Nc3ccccc3S(=O)(=O)C(C)C)n2)c(OC(C)C)cc1C1CCN(CCOCCC(=O)N2CCC3(CCc4cc5c(cc4O3)C(=O)N(C3CCC(=O)NC3=O)C5=O)CC2)CC1	C53H63ClN8O10S	ALK	Q9UM73	CRBN	WO-2023143589-A1
TPD-IJNCRS	SCHEMBL25342387	1'-[3-[2-[4-[4-[[5-Chloro-4-(2-propan-2-ylsulfonylanilino)pyrimidin-2-yl]amino]-2-methyl-5-propan-2-yloxyphenyl]piperidin-1-yl]ethoxy]propanoyl]-7-(2,6-dioxopiperidin-3-yl)spiro[2,4-dihydropyrano[3,2-f]isoindole-3,4'-piperidine]-6,8-dione; SCHEMBL30520347	Cc1cc(Nc2ncc(Cl)c(Nc3ccccc3S(=O)(=O)C(C)C)n2)c(OC(C)C)cc1C1CCN(CCOCCC(=O)N2CCC3(CC2)COc2cc4c(cc2C3)C(=O)N(C2CCC(=O)NC2=O)C4=O)CC1	C53H63ClN8O10S	ALK	Q9UM73	CRBN	WO-2023143589-A1
TPD-R7R0U6	SCHEMBL25341024	1'-[3-[2-[4-[4-[[5-chloro-4-(2-propan-2-ylsulfonylanilino)pyrimidin-2-yl]amino]-2-methyl-5-propan-2-yloxyphenyl]piperidin-1-yl]ethoxy]propanoyl]-6-(2,6-dioxopiperidin-3-yl)spiro[2H-furo[3,2-f]isoindole-3,4'-piperidine]-5,7-dione	Cc1cc(Nc2ncc(Cl)c(Nc3ccccc3S(=O)(=O)C(C)C)n2)c(OC(C)C)cc1C1CCN(CCOCCC(=O)N2CCC3(CC2)COc2cc4c(cc23)C(=O)N(C2CCC(=O)NC2=O)C4=O)CC1	C52H61ClN8O10S	ALK	Q9UM73	CRBN	WO-2023143589-A1
TPD-3RN39W	SCHEMBL25342278	1'-[3-[2-[(3R)-3-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]ethoxy]propanoyl]-7-(2,6-dioxopiperidin-3-yl)spiro[3,4-dihydropyrano[3,2-f]isoindole-2,4'-piperidine]-6,8-dione; SCHEMBL30520267	Nc1ncnc2c1c(-c1ccc(Oc3ccccc3)cc1)nn2[C@@H]1CCCN(CCOCCC(=O)N2CCC3(CCc4cc5c(cc4O3)C(=O)N(C3CCC(=O)NC3=O)C5=O)CC2)C1	C47H49N9O8	BTK	Q06187	CRBN	WO-2023143589-A1
TPD-H9CTW2	SCHEMBL25341657	1'-[3-[2-[(3R)-3-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]ethoxy]propanoyl]-7-(2,6-dioxopiperidin-3-yl)spiro[3,4-dihydropyrano[3,2-f]isoindole-2,3'-azetidine]-6,8-dione; SCHEMBL30520900	Nc1ncnc2c1c(-c1ccc(Oc3ccccc3)cc1)nn2[C@@H]1CCCN(CCOCCC(=O)N2CC3(CCc4cc5c(cc4O3)C(=O)N(C3CCC(=O)NC3=O)C5=O)C2)C1	C45H45N9O8	BTK	Q06187	CRBN	WO-2023143589-A1
TPD-P5MJV4	SCHEMBL30520452	1'-[3-[2-[(3R)-3-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]ethoxy]propanoyl]-7-(2,6-dioxopiperidin-3-yl)spiro[2,4-dihydropyrano[3,2-f]isoindole-3,4'-piperidine]-6,8-dione	Nc1ncnc2c1c(-c1ccc(Oc3ccccc3)cc1)nn2[C@@H]1CCCN(CCOCCC(=O)N2CCC3(CC2)COc2cc4c(cc2C3)C(=O)N(C2CCC(=O)NC2=O)C4=O)C1	C47H49N9O8	BTK	Q06187	CRBN	WO-2023143589-A1
TPD-4F2WVV	SCHEMBL25342493	3-[1'-[3-[2-[(3R)-3-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]ethoxy]propanoyl]-6-oxospiro[4,8-dihydro-3H-pyrano[3,2-f]isoindole-2,4'-piperidine]-7-yl]piperidine-2,6-dione; SCHEMBL30520358	Nc1ncnc2c1c(-c1ccc(Oc3ccccc3)cc1)nn2[C@@H]1CCCN(CCOCCC(=O)N2CCC3(CCc4cc5c(cc4O3)CN(C3CCC(=O)NC3=O)C5=O)CC2)C1	C47H51N9O7	BTK	Q06187	CRBN	WO-2023143589-A1
TPD-84KJUD	SCHEMBL25343004	3-[1'-[3-[2-[(3R)-3-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]ethoxy]propanoyl]-8-oxospiro[4,6-dihydro-3H-pyrano[2,3-f]isoindole-2,4'-piperidine]-7-yl]piperidine-2,6-dione; SCHEMBL30520419	Nc1ncnc2c1c(-c1ccc(Oc3ccccc3)cc1)nn2[C@@H]1CCCN(CCOCCC(=O)N2CCC3(CCc4cc5c(cc4O3)C(=O)N(C3CCC(=O)NC3=O)C5)CC2)C1	C47H51N9O7	BTK	Q06187	CRBN	WO-2023143589-A1
TPD-NN5VVG	SCHEMBL25342071	3-[1'-[3-[2-[(3R)-3-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]ethoxy]propanoyl]-8-oxospiro[2,6-dihydro-[1,4]dioxino[2,3-f]isoindole-3,4'-piperidine]-7-yl]piperidine-2,6-dione; SCHEMBL30520282	Nc1ncnc2c1c(-c1ccc(Oc3ccccc3)cc1)nn2[C@@H]1CCCN(CCOCCC(=O)N2CCC3(CC2)COc2cc4c(cc2O3)CN(C2CCC(=O)NC2=O)C4=O)C1	C46H49N9O8	BTK	Q06187	CRBN	WO-2023143589-A1
TPD-FVEW43	WO2023143589A1_38	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CCOCCC(=O)N5CCC6(CCc7cc8c(cc7O6)C(=O)N(C6CCC(=O)NC6=O)C8=O)CC5)CC4)cn3)nc2n(C2CCCC2)c1=O	C49H56N10O9	CDK4;CDK6	P11802/Q00534	CRBN	WO-2023143589-A1
TPD-YDC7C4	WO2023143589A1_39	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CCOCCC(=O)N5CC6(CCc7cc8c(cc7O6)C(=O)N(C6CCC(=O)NC6=O)C8=O)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H52N10O9	CDK4;CDK6	P11802/Q00534	CRBN	WO-2023143589-A1
TPD-HFV5ED	SCHEMBL25430286	1'-[3-[2-[4-[6-[(6-Acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]ethoxy]propanoyl]-7-(2,6-dioxopiperidin-3-yl)spiro[2,4-dihydropyrano[3,2-f]isoindole-3,4'-piperidine]-6,8-dione	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CCOCCC(=O)N5CCC6(CC5)COc5cc7c(cc5C6)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)cn3)nc2n(C2CCCC2)c1=O	C49H56N10O9	CDK4;CDK6	P11802/Q00534	CRBN	WO-2023143589-A1
TPD-BJRBA8	SCHEMBL25430026	1'-[3-[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]ethoxy]propanoyl]-6-(2,6-dioxopiperidin-3-yl)spiro[2H-furo[3,2-f]isoindole-3,4'-piperidine]-5,7-dione	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CCOCCC(=O)N5CCC6(CC5)COc5cc7c(cc56)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)cn3)nc2n(C2CCCC2)c1=O	C48H54N10O9	CDK4;CDK6	P11802/Q00534	CRBN	WO-2023143589-A1
TPD-8LL7YD	SCHEMBL25429276	3-[1'-[3-[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]ethoxy]propanoyl]-8-oxospiro[4,6-dihydro-3H-pyrano[2,3-f]isoindole-2,4'-piperidine]-7-yl]piperidine-2,6-dione	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CCOCCC(=O)N5CCC6(CCc7cc8c(cc7O6)C(=O)N(C6CCC(=O)NC6=O)C8)CC5)CC4)cn3)nc2n(C2CCCC2)c1=O	C49H58N10O8	CDK4;CDK6	P11802/Q00534	CRBN	WO-2023143589-A1
TPD-RIO69B	WO2023143589A1_43	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CCOCCC(=O)N5CCC6(CCc7cc8c(cc7O6)CN(C6CCC(=O)NC6=O)C8=O)CC5)CC4)cn3)nc2n(C2CCCC2)c1=O	C49H58N10O8	CDK4;CDK6	P11802/Q00534	CRBN	WO-2023143589-A1
TPD-Q9GJID	WO2023143589A1_44	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CCOCCC(=O)N5CC6(CCc7cc8c(cc7O6)C(=O)N(C6CCC(=O)NC6=O)C8)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H54N10O8	CDK4;CDK6	P11802/Q00534	CRBN	WO-2023143589-A1
TPD-9V2FTA	WO2023143589A1_45	.	CC(=O)c1c(C)c2cnc(Nc3ccc(N4CCN(CCOCCC(=O)N5CC6(CCc7cc8c(cc7O6)CN(C6CCC(=O)NC6=O)C8=O)C5)CC4)cn3)nc2n(C2CCCC2)c1=O	C47H54N10O8	CDK4;CDK6	P11802/Q00534	CRBN	WO-2023143589-A1
TPD-EXDI8Z	SCHEMBL25342748	3-[1'-[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]-6-oxospiro[4,8-dihydro-3H-pyrano[3,2-f]isoindole-2,3'-azetidine]-7-yl]piperidine-2,6-dione; SCHEMBL30520728	Cc1sc2c(c1C)C(c1ccc(Cl)cc1)=N[C@@H](CC(=O)N1CC3(CCc4cc5c(cc4O3)CN(C3CCC(=O)NC3=O)C5=O)C1)c1nnc(C)n1-2	C37H34ClN7O5S	BRD4	O60885	CRBN	WO-2023143589-A1
TPD-4AAWQ7	SCHEMBL25343870	3-[1'-[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]-6-oxospiro[4,8-dihydro-3H-pyrano[3,2-f]isoindole-2,4'-piperidine]-7-yl]piperidine-2,6-dione; SCHEMBL30520396	Cc1sc2c(c1C)C(c1ccc(Cl)cc1)=N[C@@H](CC(=O)N1CCC3(CCc4cc5c(cc4O3)CN(C3CCC(=O)NC3=O)C5=O)CC1)c1nnc(C)n1-2	C39H38ClN7O5S	BRD4	O60885	CRBN	WO-2023143589-A1
TPD-64PGTI	SCHEMBL25342250	3-[1'-[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]-8-oxospiro[4,6-dihydro-3H-pyrano[2,3-f]isoindole-2,4'-piperidine]-7-yl]piperidine-2,6-dione; SCHEMBL30520461	Cc1sc2c(c1C)C(c1ccc(Cl)cc1)=N[C@@H](CC(=O)N1CCC3(CCc4cc5c(cc4O3)C(=O)N(C3CCC(=O)NC3=O)C5)CC1)c1nnc(C)n1-2	C39H38ClN7O5S	BRD4	O60885	CRBN	WO-2023143589-A1
TPD-X75RQL	SCHEMBL30520476	3-[1'-[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]-8-oxospiro[2,6-dihydro-[1,4]dioxino[2,3-f]isoindole-3,4'-piperidine]-7-yl]piperidine-2,6-dione	Cc1sc2c(c1C)C(c1ccc(Cl)cc1)=N[C@@H](CC(=O)N1CCC3(CC1)COc1cc4c(cc1O3)CN(C1CCC(=O)NC1=O)C4=O)c1nnc(C)n1-2	C38H36ClN7O6S	BRD4	O60885	CRBN	WO-2023143589-A1
TPD-EAYABE	SCHEMBL31169253	1'-[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]-7-(2,6-dioxopiperidin-3-yl)spiro[3,4-dihydropyrano[3,2-f]isoindole-2,4'-piperidine]-6,8-dione	Cc1sc2c(c1C)C(c1ccc(Cl)cc1)=N[C@@H](CC(=O)N1CCC3(CCc4cc5c(cc4O3)C(=O)N(C3CCC(=O)NC3=O)C5=O)CC1)c1nnc(C)n1-2	C39H36ClN7O6S	BRD4	O60885	CRBN	WO-2023143589-A1
TPD-4AQTCJ	SCHEMBL31169206	1'-[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]-7-(2,6-dioxopiperidin-3-yl)spiro[3,4-dihydropyrano[3,2-f]isoindole-2,3'-azetidine]-6,8-dione	Cc1sc2c(c1C)C(c1ccc(Cl)cc1)=N[C@@H](CC(=O)N1CC3(CCc4cc5c(cc4O3)C(=O)N(C3CCC(=O)NC3=O)C5=O)C1)c1nnc(C)n1-2	C37H32ClN7O6S	BRD4	O60885	CRBN	WO-2023143589-A1
TPD-VSQPCU	WO2023143589A1_52	.	O=C1CCC(N2Cc3cc4c(cc3C2=O)CCC2(CN(C3CCC5(CC3)CCN(c3ccc([C@@H]6c7ccc(O)cc7CC[C@@H]6c6ccccc6)cc3)CC5)C2)O4)C(=O)N1	C50H54N4O5	ERα	P03372	CRBN	WO-2023143589-A1
TPD-CV4MIY	WO2023143589A1_53	.	O=C1CCC(N2Cc3cc4c(cc3C2=O)OC2(CC4)CN(C3CCC4(CC3)CN(c3ccc([C@@H]5c6ccc(O)cc6CC[C@@H]5c5ccccc5)cc3)C4)C2)C(=O)N1	C48H50N4O5	ERα	P03372	CRBN	WO-2023143589-A1
TPD-MM6A9W	SCHEMBL25342397	6-(2,6-dioxopiperidin-3-yl)-1'-[3-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-3-azaspiro[5.5]undecan-9-yl]spiro[2H-furo[3,2-f]isoindole-3,4'-piperidine]-5,7-dione	O=C1CCC(N2C(=O)c3cc4c(cc3C2=O)C2(CCN(C3CCC5(CC3)CCN(c3ccc([C@@H]6c7ccc(O)cc7CC[C@@H]6c6ccccc6)cc3)CC5)CC2)CO4)C(=O)N1	C51H54N4O6	ERα	P03372	CRBN	WO-2023143589-A1
TPD-165ONM	SCHEMBL25342089	3-[1'-[2-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-2-azaspiro[3.5]nonan-7-yl]-6-oxospiro[4,8-dihydro-3H-pyrano[3,2-f]isoindole-2,3'-azetidine]-7-yl]piperidine-2,6-dione; SCHEMBL30520381	O=C1CCC(N2Cc3cc4c(cc3C2=O)CCC2(CN(C3CCC5(CC3)CN(c3ccc([C@@H]6c7ccc(O)cc7CC[C@@H]6c6ccccc6)cc3)C5)C2)O4)C(=O)N1	C48H50N4O5	ERα	P03372	CRBN	WO-2023143589-A1
TPD-909EOJ	SCHEMBL25345073	3-[1'-[7-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-7-azaspiro[3.5]nonan-2-yl]-6-oxospiro[4,8-dihydro-3H-pyrano[3,2-f]isoindole-2,3'-azetidine]-7-yl]piperidine-2,6-dione; SCHEMBL30520395	O=C1CCC(N2Cc3cc4c(cc3C2=O)CCC2(CN(C3CC5(CCN(c6ccc([C@@H]7c8ccc(O)cc8CC[C@@H]7c7ccccc7)cc6)CC5)C3)C2)O4)C(=O)N1	C48H50N4O5	ERα	P03372	CRBN	WO-2023143589-A1
TPD-SHDMX0	SCHEMBL25343919	3-[1'-[7-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-7-azaspiro[3.5]nonan-2-yl]-6-oxospiro[4,8-dihydro-3H-pyrano[3,2-f]isoindole-2,4'-piperidine]-7-yl]piperidine-2,6-dione; SCHEMBL30520341	O=C1CCC(N2Cc3cc4c(cc3C2=O)CCC2(CCN(C3CC5(CCN(c6ccc([C@@H]7c8ccc(O)cc8CC[C@@H]7c7ccccc7)cc6)CC5)C3)CC2)O4)C(=O)N1	C50H54N4O5	ERα	P03372	CRBN	WO-2023143589-A1
TPD-IY8ROV	SCHEMBL25344014	3-[1'-[7-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-7-azaspiro[3.5]nonan-2-yl]-8-oxospiro[2,6-dihydro-[1,4]dioxino[2,3-f]isoindole-3,4'-piperidine]-7-yl]piperidine-2,6-dione; SCHEMBL30520429	O=C1CCC(N2Cc3cc4c(cc3C2=O)OCC2(CCN(C3CC5(CCN(c6ccc([C@@H]7c8ccc(O)cc8CC[C@@H]7c7ccccc7)cc6)CC5)C3)CC2)O4)C(=O)N1	C49H52N4O6	ERα	P03372	CRBN	WO-2023143589-A1
TPD-KDSJLS	WO2023143589A1_59	.	O=C1CCC(N2Cc3ccc4c(c3C2=O)OCC2(CCN(C3CCC5(CC3)CCN(c3ccc([C@@H]6c7ccc(O)cc7CC[C@@H]6c6ccccc6)cc3)CC5)CC2)C4)C(=O)N1	C52H58N4O5	ERα	P03372	CRBN	WO-2023143589-A1
TPD-ON69QL	WO2023143589A1_60	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CC6(CCc7cc8c(cc7O6)C(=O)N(C6CCC(=O)NC6=O)C8=O)C5)CC4)nn3)CC2)cc1Cl	C42H43ClN8O7	AR	P10275	CRBN	WO-2023143589-A1
TPD-NQC3OR	WO2023143589A1_61	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC5(CC4)CC(N4CCC6(CCc7cc8c(cc7O6)C(=O)N(C6CCC(=O)NC6=O)C8=O)CC4)C5)nn3)CC2)cc1Cl	C46H49ClN8O7	AR	P10275	CRBN	WO-2023143589-A1
TPD-Y0PD9R	WO2023143589A1_62	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CC(N5CCC6(CCc7cc8c(cc7O6)CN(C6CCC(=O)NC6=O)C8=O)CC5)C4)nn3)CC2)cc1Cl	C41H43ClN8O6	AR	P10275	CRBN	WO-2023143589-A1
TPD-W16FCW	WO2023143589A1_63	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC5(CC4)CC(N4CCC6(CC4)COc4cc7c(cc46)C(=O)N(C4CCC(=O)NC4=O)C7=O)C5)nn3)CC2)cc1Cl	C45H47ClN8O7	AR	P10275	CRBN	WO-2023143589-A1
TPD-K9SO30	SCHEMBL30520469	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[3-[7-(2,6-dioxopiperidin-3-yl)-6,8-dioxospiro[2,4-dihydropyrano[3,2-f]isoindole-3,4'-piperidine]-1'-yl]azetidin-1-yl]pyridazine-3-carboxamide	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CC(N5CCC6(CC5)COc5cc7c(cc5C6)C(=O)N(C5CCC(=O)NC5=O)C7=O)C4)nn3)CC2)cc1Cl	C41H41ClN8O7	AR	P10275	CRBN	WO-2023143589-A1
TPD-TULKL6	WO2023143589A1_65	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC6(CC5)COc5cc7c(cc5O6)CN(C5CCC(=O)NC5=O)C7=O)CC4)nn3)CC2)cc1Cl	C43H47ClN8O7	AR	P10275	CRBN	WO-2023143589-A1
TPD-LUY8W2	WO2023143589A1_66	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC6(CC5)Cc5cc7c(cc5O6)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)nn3)CC2)cc1Cl	C43H45ClN8O7	AR	P10275	CRBN	WO-2023143589-A1
TPD-OY5X99	WO2023143589A1_67	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CC(N5CCC6(CC5)Cc5cc7c(cc5O6)C(=O)N(C5CCC(=O)NC5=O)C7=O)C4)nn3)CC2)cc1Cl	C40H39ClN8O7	AR	P10275	CRBN	WO-2023143589-A1
TPD-2Y7XAW	WO2023143589A1_68	.	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=S)N1c1ccc(C(=O)N2CCC(F)(CN3CC4(CCc5cc6c(cc5O4)C(=O)N(C4CCC(=O)NC4=O)C6)C3)CC2)c(F)c1	C44H40F5N7O6S	AR	P10275	CRBN	WO-2023143589-A1
TPD-V8MMSD	WO2023143589A1_69	.	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=S)N1c1ccc(C(=O)N2CCC(CN3CCC4(CC3)COc3cc5c(cc3C4)C(=O)N(C3CCC(=O)NC3=O)C5=O)CC2)c(F)c1	C46H43F4N7O7S	AR	P10275	CRBN	WO-2023143589-A1
TPD-P94ZRY	WO2023143589A1_70	.	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=S)N1c1ccc(C(=O)N2CC[C@@H](CN3CCC4(CC3)COc3cc5c(cc3C4)C(=O)N(C3CCC(=O)NC3=O)C5=O)C2)c(F)c1	C45H41F4N7O7S	AR	P10275	CRBN	WO-2023143589-A1
TPD-PFLK0D	WO2023143589A1_71	.	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=S)N1c1ccc(C(=O)N2CC(CN3CCC4(CCc5cc6c(cc5O4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C2)c(F)c1	C44H39F4N7O7S	AR	P10275	CRBN	WO-2023143589-A1
TPD-F03UDH	WO2023143589A1_72	.	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=S)N1c1ccc(C(=O)N2CCC(CN3CCC4(CCc5cc6c(cc5O4)CN(C4CCC(=O)NC4=O)C6=O)CC3)CC2)c(F)c1	C46H45F4N7O6S	AR	P10275	CRBN	WO-2023143589-A1
TPD-D419OY	WO2023143589A1_73	.	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=S)N1c1ccc(C(=O)N2CC3(CCC(N4CCC5(CC4)COc4cc6c(cc4C5)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C2)c(F)c1	C48H45F4N7O7S	AR	P10275	CRBN	WO-2023143589-A1
TPD-PMSQBB	WO2023143589A1_74	.	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=S)N1c1ccc(C(=O)N2CCC3(CCC(N4CCC5(CC4)COc4cc6c(cc4C5)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C2)c(F)c1	C49H47F4N7O7S	AR	P10275	CRBN	WO-2023143589-A1
TPD-ZB3RCR	WO2023143589A1_75	.	COC1(CN2CC3(CCc4cc5c(cc4O3)C(=O)N(C3CCC(=O)NC3=O)C5=O)C2)CCN(C(=O)c2ccc(N3C(=S)N(c4ccc(C#N)c(C(F)(F)F)c4)C(=O)C3(C)C)cc2F)CC1	C45H41F4N7O8S	AR	P10275	CRBN	WO-2023143589-A1
TPD-JOEYTU	WO2023143589A1_76	.	COC1(CN2CC3(CCc4cc5c(cc4O3)CN(C3CCC(=O)NC3=O)C5=O)C2)CCN(C(=O)c2ccc(N3C(=S)N(c4ccc(C#N)c(C(F)(F)F)c4)C(=O)C3(C)C)cc2F)CC1	C45H43F4N7O7S	AR	P10275	CRBN	WO-2023143589-A1
TPD-SDX2ON	WO2023143589A1_77	.	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=S)N1c1ccc(C(=O)N2CC(N3CC4(CCc5cc6c(cc5O4)C(=O)N(C4CCC(=O)NC4=O)C6=O)C3)C2)c(F)c1	C41H33F4N7O7S	AR	P10275	CRBN	WO-2023143589-A1
TPD-2DU67U	WO2023143589A1_78	.	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=S)N1c1ccc(C(=O)N2CCC(N3CCC4(CC3)COc3cc5c(cc3C4)C(=O)N(C3CCC(=O)NC3=O)C5=O)CC2)c(F)c1	C45H41F4N7O7S	AR	P10275	CRBN	WO-2023143589-A1
TPD-G2R3RB	WO2023143589A1_79	.	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=S)N1c1ccc(C(=O)N2CC3(CC(N4CCC5(CC4)COc4cc6c(cc45)C(=O)N(C4CCC(=O)NC4=O)C6=O)C3)C2)c(F)c1	C45H39F4N7O7S	AR	P10275	CRBN	WO-2023143589-A1
TPD-I1SRO7	WO2023143589A1_80	.	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=S)N1c1ccc(C(=O)N2CCC(N3CCC4(CC3)COc3cc5c(cc34)C(=O)N(C3CCC(=O)NC3=O)C5=O)CC2)c(F)c1	C44H39F4N7O7S	AR	P10275	CRBN	WO-2023143589-A1
TPD-TRTK2K	WO2023143589A1_81	.	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=S)N1C1C=C(F)C(C(=O)N2CC(N3CCC4(CC3)COc3cc5c(cc34)C(=O)N(C3CCC(=O)NC3=O)C5=O)C2)=CC1	C42H37F4N7O7S	AR	P10275	CRBN	WO-2023143589-A1
TPD-K9OR6N	WO2023143589A1_82	.	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=S)N1c1ccc(C(=O)N2CCC(F)(CN3CCC4(CCc5cc6c(cc5O4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)CC2)c(F)c1	C46H42F5N7O7S	AR	P10275	CRBN	WO-2023143589-A1
TPD-4CG2UG	WO2023143589A1_83	.	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=S)N1c1ccc(C(=O)N2CCC3(CCC(N4CCC5(CCc6cc7c(cc6O5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)CC3)CC2)c(F)c1	C50H49F4N7O7S	AR	P10275	CRBN	WO-2023143589-A1
TPD-NV9PRO	WO2023143589A1_84	.	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=S)N1c1ccc(C(=O)N2CCC(CN3CCC4(CCc5cc6c(cc5O4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)CC2)c(F)c1	C46H43F4N7O7S	AR	P10275	CRBN	WO-2023143589-A1
TPD-Q8615W	WO2023143589A1_85	.	CC1C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=S)N1C1C=C(F)C(C(=O)N2CC3(CC(N4CCC5(CCc6cc7c(cc6O5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)C3)C2)=CC1	C45H41F4N7O7S	AR	P10275	CRBN	WO-2023143589-A1
TPD-2EIGGO	WO2023143589A1_86	.	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=S)N1C1=CCC(C(=O)N2CCC(N3CCC4(CCc5cc6c(cc5O4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)CC2)C(F)=C1	C45H43F4N7O7S	AR	P10275	CRBN	WO-2023143589-A1
TPD-UJY9AM	WO2023143589A1_87	.	CC1(C)C(=O)N(c2ccc(N=O)c(C(F)(F)F)c2)C(=S)N1c1ccc(C(=O)N2CC(N3CCC4(CCc5cc6c(cc5O4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C2)c(F)c1	C42H37F4N7O8S	AR	P10275	CRBN	WO-2023143589-A1
TPD-5X1ZDE	WO2023143589A1_88	.	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=S)N1C1C=C(F)C(C(=O)N2CCC3(CC2)CC(N2CCC4(CCc5cc6c(cc5O4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC2)C3)=CC1	C48H47F4N7O7S	AR	P10275	CRBN	WO-2023143589-A1
TPD-HIYCR5	WO2023143589A1_89	.	CC1(CN2CCC3(CCc4cc5c(cc4O3)CN(C3CCC(=O)NC3=O)C5=O)CC2)CCN(C(=O)c2ccc(N3C(=S)N(c4ccc(C#N)c(C(F)(F)F)c4)C(=O)C3(C)C)cc2F)CC1	C47H47F4N7O6S	AR	P10275	CRBN	WO-2023143589-A1
TPD-MRSVI8	WO2023143589A1_90	.	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=S)N1c1ccc(C(=O)N2CC(N3CCC4(CCc5cc6c(cc5O4)C(=O)N(C4CCC(=O)NC4=O)C6)CC3)C2)c(F)c1	C43H39F4N7O6S	AR	P10275	CRBN	WO-2023143589-A1
TPD-1T6S9V	WO2023143589A1_91	.	CC1(CN2CCC3(CCc4cc5c(cc4O3)C(=O)N(C3CCC(=O)NC3=O)C5=O)CC2)CCN(C(=O)c2ccc(N3C(=S)N(c4ccc(C#N)c(C(F)(F)F)c4)C(=O)C3(C)C)cc2F)CC1	C47H45F4N7O7S	AR	P10275	CRBN	WO-2023143589-A1
TPD-F2CQUX	WO2023143589A1_92	.	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=S)N1c1ccc(C(=O)N2CCC(CN3CCC4(CC3)COc3cc5c(cc34)C(=O)N(C3CCC(=O)NC3=O)C5=O)CC2)c(F)c1	C45H41F4N7O7S	AR	P10275	CRBN	WO-2023143589-A1
TPD-IKFHWP	WO2023143589A1_93	.	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=S)N1c1ccc(C(=O)N2CC(CN3CCC4(CC3)COc3cc5c(cc34)C(=O)N(C3CCC(=O)NC3=O)C5=O)C2)c(F)c1	C43H37F4N7O7S	AR	P10275	CRBN	WO-2023143589-A1
TPD-ZY0HBW	WO2023143589A1_94	.	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=S)N1c1ccc(C(=O)N2CCC(CN3CCC4(CC3)COc3cc5c(cc3O4)CN(C3CCC(=O)NC3=O)C5=O)CC2)c(F)c1	C45H43F4N7O7S	AR	P10275	CRBN	WO-2023143589-A1
TPD-KQUNU1	WO2023143589A1_95	.	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=S)N1c1ccc(C(=O)N2CC(N3CCC4(CC3)COc3cc5c(cc3C4)C(=O)N(C3CCC(=O)NC3=O)C5=O)C2)c(F)c1	C43H37F4N7O7S	AR	P10275	CRBN	WO-2023143589-A1
TPD-WQGHUF	WO2023143589A1_96	.	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=S)N1c1ccc(C(=O)N2CCC3(CCC(N4CCC5(CC4)COc4cc6c(cc4C5)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)CC2)c(F)c1	C50H49F4N7O7S	AR	P10275	CRBN	WO-2023143589-A1
TPD-9N4DVO	WO2023143589A1_97	.	CC1(CN2CCC3(CC2)COc2cc4c(cc2C3)C(=O)N(C2CCC(=O)NC2=O)C4=O)CCN(C(=O)c2ccc(N3C(=S)N(c4ccc(C#N)c(C(F)(F)F)c4)C(=O)C3(C)C)cc2F)CC1	C47H45F4N7O7S	AR	P10275	CRBN	WO-2023143589-A1
TPD-ZOVODR	WO2023143589A1_98	.	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=S)N1c1ccc(C(=O)N2CC3(CC(N4CCC5(CC4)COc4cc6c(cc4C5)C(=O)N(C4CCC(=O)NC4=O)C6=O)C3)C2)c(F)c1	C46H41F4N7O7S	AR	P10275	CRBN	WO-2023143589-A1
TPD-99JX7A	WO2023143589A1_99	.	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=S)N1c1ccc(C(=O)N2CCC(CN3CCC4(CCc5cc6c(cc5O4)C(=O)N(C4CCC(=O)NC4=O)C6)CC3)CC2)c(F)c1	C46H45F4N7O6S	AR	P10275	CRBN	WO-2023143589-A1
TPD-HEKC74	WO2023143589A1_100	.	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=S)N1c1ccc(C(=O)N2CC3(CCC(N4CCC5(CCC6=CC7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7C=C6O5)CC4)CC3)C2)c(F)c1	C48H47F4N7O7S	AR	P10275	CRBN	WO-2023143589-A1
TPD-1SV5QA	WO2023143589A1_101	.	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=S)N1c1ccc(C(=O)N2CCC(CN3CC4(CCc5cc6c(cc5O4)C(=O)N(C4CCC(=O)NC4=O)C6=O)C3)CC2)c(F)c1	C44H39F4N7O7S	AR	P10275	CRBN	WO-2023143589-A1
TPD-9PI9IE	WO2023143589A1_102	.	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=S)N1c1ccc(C(=O)N2CCC3(CCC(N4CCC5(CC4)COc4cc6c(cc45)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)CC2)c(F)c1	C49H47F4N7O7S	AR	P10275	CRBN	WO-2023143589-A1
TPD-5R4OGW	WO2023143589A1_103	.	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=S)N1c1ccc(C(=O)N2CC3(CCC(N4CCC5(CC4)COc4cc6c(cc45)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C2)c(F)c1	C47H43F4N7O7S	AR	P10275	CRBN	WO-2023143589-A1
TPD-EHOFWO	WO2023143589A1_104	.	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=S)N1C1=CCC(C(=O)N2CCC3(CC2)CC(N2CCC4(CC2)COc2cc5c(cc24)C(=O)N(C2CCC(=O)NC2=O)C5=O)C3)C(F)=C1	C47H45F4N7O7S	AR	P10275	CRBN	WO-2023143589-A1
TPD-2QS4QH	WO2023143589A1_105	.	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=S)N1c1ccc(C(=O)N2CCC3(CC2)CC(N2CCC4(CC2)COc2cc5c(cc2C4)C(=O)N(C2CCC(=O)NC2=O)C5=O)C3)c(F)c1	C48H45F4N7O7S	AR	P10275	CRBN	WO-2023143589-A1
TPD-83MZ7Q	WO2023143589A1_106	.	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=S)N1c1ccc(C(=O)N2CCC(CN3CC4(CCc5cc6c(cc5O4)CN(C4CCC(=O)NC4=O)C6=O)C3)CC2)c(F)c1	C44H41F4N7O6S	AR	P10275	CRBN	WO-2023143589-A1
TPD-ZPMH4F	WO2023143589A1_107	.	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=S)N1c1ccc(C(=O)N2CC[C@H](CN3CCC4(CC3)COc3cc5c(cc34)C(=O)N(C3CCC(=O)NC3=O)C5=O)C2)c(F)c1	C44H39F4N7O7S	AR	P10275	CRBN	WO-2023143589-A1
TPD-2KITBN	WO2023151113A1_11j	.	O=C1CCC(N2C(=O)c3cccc(NCc4cn(CCOCCOCCOCCOCCOCCOc5ccc(Cn6ccc7ccc(C(=O)NO)cc76)cc5)nn4)c3C2=O)C(=O)N1	C44H50N8O12	HDAC8	Q9BY41	CRBN	WO-2023151113-A1
TPD-SOA99Z	SCHEMBL30509127	4-[2-[2-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]butanoyl]-3,4-dihydro-1H-isoquinolin-6-yl]-5H-pyrrolo[2,3-b]pyrazin-7-yl]-N,N-dimethylbenzamide	CN(C)C(=O)c1ccc(-c2c[nH]c3ncc(-c4ccc5c(c4)CCN(C(=O)CCCNc4cccc6c4C(=O)N(C4CCC(=O)NC4=O)C6=O)C5)nc23)cc1	C41H38N8O6	HPK1	Q92918	CRBN	WO-2023151559-A1
TPD-5Q1DYD	WO2023151559A1_2	.	CN(C)C(=O)c1ccc(-c2c[nH]c3ncc(-c4ccc5c(c4)CCN(C(=O)CCCCCNc4cccc6c4C(=O)N(C4CCC(=O)NC4=O)C6=O)C5)nc23)cc1	C43H42N8O6	HPK1	Q92918	CRBN	WO-2023151559-A1
TPD-MLYFCY	WO2023151559A1_3	.	CN(C)C(=O)c1ccc(-c2c[nH]c3ncc(-c4ccc5c(c4)CCN(C(=O)CCCCCCNc4cccc6c4C(=O)N(C4CCC(=O)NC4=O)C6=O)C5)nc23)cc1	C44H44N8O6	HPK1	Q92918	CRBN	WO-2023151559-A1
TPD-I0M336	WO2023151559A1_4	.	CN(C)C(=O)c1ccc(-c2c[nH]c3ncc(-c4ccc5c(c4)CCN(C(=O)CCCCCCCNc4cccc6c4C(=O)N(C4CCC(=O)NC4=O)C6=O)C5)nc23)cc1	C45H46N8O6	HPK1	Q92918	CRBN	WO-2023151559-A1
TPD-4EV494	WO2023151559A1_5	.	CN(C)C(=O)c1ccc(-c2c[nH]c3ncc(-c4ccc5c(c4)CCN(C(=O)CCCCCCCCNc4cccc6c4C(=O)N(C4CCC(=O)NC4=O)C6=O)C5)nc23)cc1	C46H48N8O6	HPK1	Q92918	CRBN	WO-2023151559-A1
TPD-0MHL98	WO2023151559A1_6	.	CN(C)C(=O)c1ccc(-c2c[nH]c3ncc(-c4ccc5c(c4)CCN(C(=O)CCCCCCCCCNc4cccc6c4C(=O)N(C4CCC(=O)NC4=O)C6=O)C5)nc23)cc1	C47H50N8O6	HPK1	Q92918	CRBN	WO-2023151559-A1
TPD-9PYSME	WO2023151559A1_7	.	CN(C)C(=O)c1ccc(-c2c[nH]c3ncc(-c4ccc5c(c4)CCN(C(=O)CCCCCNc4ccc6c(c4)C(=O)N(C4CCC(=O)NC4=O)C6=O)C5)nc23)cc1	C43H42N8O6	HPK1	Q92918	CRBN	WO-2023151559-A1
TPD-BZC2K6	WO2023151559A1_8	.	CN(C)C(=O)c1ccc(-c2c[nH]c3ncc(-c4ccc5c(c4)CCN(C(=O)CCCCCCCNc4ccc6c(c4)C(=O)N(C4CCC(=O)NC4=O)C6=O)C5)nc23)cc1	C45H46N8O6	HPK1	Q92918	CRBN	WO-2023151559-A1
TPD-IY6LRG	WO2023151559A1_9	.	Cc1cc(-c2cnc3[nH]cc(-c4ccc(C(=O)N(C)C)cc4)c3n2)cc2c1CN(C(=O)CCCCCCCNc1cccc3c1C(=O)N(C1CCC(=O)NC1=O)C3=O)CC2	C46H48N8O6	HPK1	Q92918	CRBN	WO-2023151559-A1
TPD-6SYOGC	WO2023151559A1_10	.	CN(C)C(=O)c1ccc(-c2c[nH]c3ncc(-c4ccc5c(c4)CCN(C(=O)CCCCCC#Cc4cccc6c4C(=O)N(C4CCC(=O)NC4=O)C6=O)C5)nc23)cc1	C45H41N7O6	HPK1	Q92918	CRBN	WO-2023151559-A1
TPD-QIKYD7	WO2023151559A1_11	.	CN(C)C(=O)c1ccc(-c2c[nH]c3ncc(-c4ccc5c(c4)CCN(C(=O)CCCCCCC#Cc4cccc6c4C(=O)N(C4CCC(=O)NC4=O)C6=O)C5)nc23)cc1	C46H43N7O6	HPK1	Q92918	CRBN	WO-2023151559-A1
TPD-28S4P0	WO2023151559A1_12	.	CN(C)C(=O)c1ccc(-c2c[nH]c3ncc(-c4ccc5c(c4)CCN(C(=O)CCCCCCC#Cc4ccc6c(c4)C(=O)N(C4CCC(=O)NC4=O)C6=O)C5)nc23)cc1	C46H43N7O6	HPK1	Q92918	CRBN	WO-2023151559-A1
TPD-7WRM5J	WO2023151559A1_14	.	CN(C)C(=O)c1ccc(-c2c[nH]c3ncc(-c4ccc5c(c4)CCN(C(=O)CCCCCCCOc4cccc6c4C(=O)N(C4CCC(=O)NC4=O)C6=O)C5)nc23)cc1	C45H45N7O7	HPK1	Q92918	CRBN	WO-2023151559-A1
TPD-BZV368	WO2023151559A1_15	.	CN(C)C(=O)c1ccc(-c2c[nH]c3ncc(-c4ccc5c(c4)CN(C(=O)CCCCCCCNc4cccc6c4C(=O)N(C4CCC(=O)NC4=O)C6=O)CC5)nc23)cc1	C45H46N8O6	HPK1	Q92918	CRBN	WO-2023151559-A1
TPD-1QLGSF	WO2023151559A1_16	.	CN(C)C(=O)c1ccc(-c2c[nH]c3ncc(-c4ccc5c(c4)CN(C(=O)CCCCCC#Cc4cccc6c4C(=O)N(C4CCC(=O)NC4=O)C6=O)CC5)nc23)cc1	C45H41N7O6	HPK1	Q92918	CRBN	WO-2023151559-A1
TPD-UQW8M3	SCHEMBL30509131	4-[2-[2-[6-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]hexyl]-3,4-dihydro-1H-isoquinolin-6-yl]-5H-pyrrolo[2,3-b]pyrazin-7-yl]-N,N-dimethylbenzamide	CN(C)C(=O)c1ccc(-c2c[nH]c3ncc(-c4ccc5c(c4)CCN(CCCCCCNc4cccc6c4C(=O)N(C4CCC(=O)NC4=O)C6=O)C5)nc23)cc1	C43H44N8O5	HPK1	Q92918	CRBN	WO-2023151559-A1
TPD-VQ3UU8	SCHEMBL30509129	4-[2-[2-[6-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]hexyl]-3,4-dihydro-1H-isoquinolin-6-yl]-5H-pyrrolo[2,3-b]pyrazin-7-yl]-N,N-dimethylbenzamide	CN(C)C(=O)c1ccc(-c2c[nH]c3ncc(-c4ccc5c(c4)CCN(CCCCCCNc4cccc6c4CN(C4CCC(=O)NC4=O)C6=O)C5)nc23)cc1	C43H46N8O4	HPK1	Q92918	CRBN	WO-2023151559-A1
TPD-0NPJ7O	WO2023151559A1_19	4-[2-[2-[2-[3-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]propylamino]-2-oxoethyl]-3,4-dihydro-1H-isoquinolin-6-yl]-5H-pyrrolo[2,3-b]pyrazin-7-yl]-N,N-dimethylbenzamide	CN(C)C(=O)c1ccc(-c2c[nH]c3ncc(-c4ccc5c(c4)CCN(CC(=O)NCCCNc4cccc6c4C(=O)N(C4CCC(=O)NC4=O)C6=O)C5)nc23)cc1	C42H41N9O6	HPK1	Q92918	CRBN	WO-2023151559-A1
TPD-88OEOK	WO2023151559A1_20	.	CN(C)C(=O)c1ccc(-c2c[nH]c3ncc(-c4ccc5c(c4)CCN(CC(=O)NCCOCCNc4cccc6c4C(=O)N(C4CCC(=O)NC4=O)C6=O)C5)nc23)cc1	C43H43N9O7	HPK1	Q92918	CRBN	WO-2023151559-A1
TPD-8ZSX9E	WO2023151559A1_21	.	CN(C)C(=O)c1ccc(-c2c[nH]c3ncc(-c4ccc5c(c4)CCN(CC(=O)NCCOCCOCCNc4cccc6c4C(=O)N(C4CCC(=O)NC4=O)C6=O)C5)nc23)cc1	C45H47N9O8	HPK1	Q92918	CRBN	WO-2023151559-A1
TPD-BKNY3V	SCHEMBL30509130	N-[3-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]propyl]-N-methyl-4-[2-(2-methyl-3,4-dihydro-1H-isoquinolin-6-yl)-5H-pyrrolo[2,3-b]pyrazin-7-yl]benzamide	CN1CCc2cc(-c3cnc4[nH]cc(-c5ccc(C(=O)N(C)CCCNc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)cc5)c4n3)ccc2C1	C40H38N8O5	HPK1	Q92918	CRBN	WO-2023151559-A1
TPD-GKST9E	WO2023151559A1_23	.	CN1CCc2cc(-c3cnc4[nH]cc(-c5ccc(C(=O)N(C)CCCCCNc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)cc5)c4n3)ccc2C1	C42H42N8O5	HPK1	Q92918	CRBN	WO-2023151559-A1
TPD-WNEH03	WO2023151559A1_24	.	CN1CCc2cc(-c3cnc4[nH]cc(-c5ccc(C(=O)N(C)CCCCCCNc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)cc5)c4n3)ccc2C1	C43H44N8O5	HPK1	Q92918	CRBN	WO-2023151559-A1
TPD-MPIOG9	WO2023151559A1_25	.	CN1CCc2cc(-c3cnc4[nH]cc(-c5ccc(C(=O)N(C)CCCCCCCNc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)cc5)c4n3)ccc2C1	C44H46N8O5	HPK1	Q92918	CRBN	WO-2023151559-A1
TPD-VG9O7I	WO2023151559A1_26	.	CN1CCc2cc(-c3cnc4[nH]cc(-c5ccc(C(=O)N(C)CCCCCCCCNc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)cc5)c4n3)ccc2C1	C45H48N8O5	HPK1	Q92918	CRBN	WO-2023151559-A1
TPD-NDMDPU	WO2023151559A1_27	.	CN1CCc2cc(-c3cnc4[nH]cc(-c5ccc(C(=O)N(C)CCCCCCCCCNc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)cc5)c4n3)ccc2C1	C46H50N8O5	HPK1	Q92918	CRBN	WO-2023151559-A1
TPD-M54695	WO2023151559A1_28	.	Nc1c(-c2nc3ccc(N4CCN(C(=O)CCCCCNc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)cc3[nH]2)c(=O)[nH]c2ccsc12	C37H37N9O6S	HPK1	Q92918	CRBN	WO-2023151559-A1
TPD-OHCQDJ	SCHEMBL29036145	2-[4-[2-(7-amino-5-oxo-4H-thieno[3,2-b]pyridin-6-yl)-3H-benzimidazol-5-yl]piperazin-1-yl]-N-[3-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]propyl]acetamide	Nc1c(-c2nc3ccc(N4CCN(CC(=O)NCCCNc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)cc3[nH]2)c(=O)[nH]c2ccsc12	C36H36N10O6S	HPK1	Q92918	CRBN	WO-2023151559-A1
TPD-9E1DL7	WO2023151559A1_30	.	CN(C)C(=O)c1ccc(-c2c[nH]c3ncc(-c4ccc5c(c4)CCN(C(=O)COCCOCCNc4ccc6c(c4)C(=O)N(C4CCC(=O)NC4=O)C6=O)C5)nc23)cc1	C43H42N8O8	HPK1	Q92918	CRBN	WO-2023151559-A1
TPD-FTK4MT	WO2023151559A1_31	.	CN(C)C(=O)c1ccc(-c2c[nH]c3ncc(-c4ccc5c(c4)CCN(C(=O)CCCCCCCOc4ccc6c(c4)C(=O)N(C4CCC(=O)NC4=O)C6=O)C5)nc23)cc1	C45H45N7O7	HPK1	Q92918	CRBN	WO-2023151559-A1
TPD-CHW5GO	WO2023151559A1_32	.	COc1cc(-c2cnc3[nH]cc(-c4ccc(C(=O)N(C)C)cc4)c3n2)cc2c1CN(C(=O)CCCCCCCNc1cccc3c1C(=O)N(C1CCC(=O)NC1=O)C3=O)CC2	C46H48N8O7	HPK1	Q92918	CRBN	WO-2023151559-A1
TPD-S5W5WC	SCHEMBL25361571	2-(2,6-Dioxopiperidin-3-yl)-4-[5-[4-[1-[3-ethoxy-4-[(5-methyl-11-methylsulfonyl-6-oxopyrimido[4,5-b][1,4]benzodiazepin-2-yl)amino]benzoyl]piperidin-4-yl]piperazin-1-yl]pentyl]isoindole-1,3-dione; SCHEMBL30526062	CCOc1cc(C(=O)N2CCC(N3CCN(CCCCCc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)ccc1Nc1ncc2c(n1)N(S(C)(=O)=O)c1ccccc1C(=O)N2C	C49H56N10O9S	ERK5	Q13164	CRBN	WO-2023156791-A1
TPD-QXNJNB	SCHEMBL25362359	3-[7-[8-[4-[1-[3-ethoxy-4-[(5-methyl-11-methylsulfonyl-6-oxopyrimido[4,5-b][1,4]benzodiazepin-2-yl)amino]benzoyl]piperidin-4-yl]piperazin-1-yl]oct-1-ynyl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30526055	CCOc1cc(C(=O)N2CCC(N3CCN(CCCCCCC#Cc4cccc5c4CN(C4CCC(=O)NC4=O)C5=O)CC3)CC2)ccc1Nc1ncc2c(n1)N(S(C)(=O)=O)c1ccccc1C(=O)N2C	C52H60N10O8S	ERK5	Q13164	CRBN	WO-2023156791-A1
TPD-7BARLD	SCHEMBL25356654	3-[7-[9-[4-[1-[3-ethoxy-4-[(5-methyl-11-methylsulfonyl-6-oxopyrimido[4,5-b][1,4]benzodiazepin-2-yl)amino]benzoyl]piperidin-4-yl]piperazin-1-yl]non-1-ynyl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30526058	CCOc1cc(C(=O)N2CCC(N3CCN(CCCCCCCC#Cc4cccc5c4CN(C4CCC(=O)NC4=O)C5=O)CC3)CC2)ccc1Nc1ncc2c(n1)N(S(C)(=O)=O)c1ccccc1C(=O)N2C	C53H62N10O8S	ERK5	Q13164	CRBN	WO-2023156791-A1
TPD-EL09OR	SCHEMBL25356529	2-(2,6-Dioxopiperidin-3-yl)-4-[6-[4-[1-[3-ethoxy-4-[(5-methyl-11-methylsulfonyl-6-oxopyrimido[4,5-b][1,4]benzodiazepin-2-yl)amino]benzoyl]piperidin-4-yl]piperazin-1-yl]hexoxy]isoindole-1,3-dione; SCHEMBL30526060	CCOc1cc(C(=O)N2CCC(N3CCN(CCCCCCOc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)ccc1Nc1ncc2c(n1)N(S(C)(=O)=O)c1ccccc1C(=O)N2C	C50H58N10O10S	ERK5	Q13164	CRBN	WO-2023156791-A1
TPD-4R4O0N	SCHEMBL25359438	2-(2,6-Dioxopiperidin-3-yl)-4-[4-[4-[1-[3-ethoxy-4-[(5-methyl-11-methylsulfonyl-6-oxopyrimido[4,5-b][1,4]benzodiazepin-2-yl)amino]benzoyl]piperidin-4-yl]piperazin-1-yl]butoxy]isoindole-1,3-dione; SCHEMBL30526061	CCOc1cc(C(=O)N2CCC(N3CCN(CCCCOc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)ccc1Nc1ncc2c(n1)N(S(C)(=O)=O)c1ccccc1C(=O)N2C	C48H54N10O10S	ERK5	Q13164	CRBN	WO-2023156791-A1
TPD-LPQVHD	SCHEMBL25359609	3-[7-[10-[4-[1-[3-ethoxy-4-[(5-methyl-11-methylsulfonyl-6-oxopyrimido[4,5-b][1,4]benzodiazepin-2-yl)amino]benzoyl]piperidin-4-yl]piperazin-1-yl]dec-1-ynyl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30526054	CCOc1cc(C(=O)N2CCC(N3CCN(CCCCCCCCC#Cc4cccc5c4CN(C4CCC(=O)NC4=O)C5=O)CC3)CC2)ccc1Nc1ncc2c(n1)N(S(C)(=O)=O)c1ccccc1C(=O)N2C	C54H64N10O8S	ERK5	Q13164	CRBN	WO-2023156791-A1
TPD-UL91YG	WO2023156791A1_OS17	.	CCOc1cc(C(=O)N2CCC(N3CCN(CCCCCCCCOc4cccc5c4CN(C4CCC(=O)NC4=O)C5=O)CC3)CC2)ccc1Nc1ncc2c(n1)N(S(C)(=O)=O)c1ccccc1C(=O)N2C	C52H64N10O9S	ERK5	Q13164	CRBN	WO-2023156791-A1
TPD-YQ4T6Y	SCHEMBL25358383	3-[7-[5-[4-[1-[3-ethoxy-4-[(5-methyl-11-methylsulfonyl-6-oxopyrimido[4,5-b][1,4]benzodiazepin-2-yl)amino]benzoyl]piperidin-4-yl]piperazin-1-yl]pent-1-ynyl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30526052	CCOc1cc(C(=O)N2CCC(N3CCN(CCCC#Cc4cccc5c4CN(C4CCC(=O)NC4=O)C5=O)CC3)CC2)ccc1Nc1ncc2c(n1)N(S(C)(=O)=O)c1ccccc1C(=O)N2C	C49H54N10O8S	ERK5	Q13164	CRBN	WO-2023156791-A1
TPD-5RDEMJ	SCHEMBL25362026	3-[7-[4-[4-[1-[3-ethoxy-4-[(5-methyl-11-methylsulfonyl-6-oxopyrimido[4,5-b][1,4]benzodiazepin-2-yl)amino]benzoyl]piperidin-4-yl]piperazin-1-yl]but-1-ynyl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30526053	CCOc1cc(C(=O)N2CCC(N3CCN(CCC#Cc4cccc5c4CN(C4CCC(=O)NC4=O)C5=O)CC3)CC2)ccc1Nc1ncc2c(n1)N(S(C)(=O)=O)c1ccccc1C(=O)N2C	C48H52N10O8S	ERK5	Q13164	CRBN	WO-2023156791-A1
TPD-YW5WU1	SCHEMBL25358130	3-[7-[6-[4-[1-[3-ethoxy-4-[(5-methyl-11-methylsulfonyl-6-oxopyrimido[4,5-b][1,4]benzodiazepin-2-yl)amino]benzoyl]piperidin-4-yl]piperazin-1-yl]hex-1-ynyl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30526051	CCOc1cc(C(=O)N2CCC(N3CCN(CCCCC#Cc4cccc5c4CN(C4CCC(=O)NC4=O)C5=O)CC3)CC2)ccc1Nc1ncc2c(n1)N(S(C)(=O)=O)c1ccccc1C(=O)N2C	C50H56N10O8S	ERK5	Q13164	CRBN	WO-2023156791-A1
TPD-CLHW6J	SCHEMBL25356978	3-[7-[7-[4-[1-[3-ethoxy-4-[(5-methyl-11-methylsulfonyl-6-oxopyrimido[4,5-b][1,4]benzodiazepin-2-yl)amino]benzoyl]piperidin-4-yl]piperazin-1-yl]hept-1-ynyl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30526064	CCOc1cc(C(=O)N2CCC(N3CCN(CCCCCC#Cc4cccc5c4CN(C4CCC(=O)NC4=O)C5=O)CC3)CC2)ccc1Nc1ncc2c(n1)N(S(C)(=O)=O)c1ccccc1C(=O)N2C	C51H58N10O8S	ERK5	Q13164	CRBN	WO-2023156791-A1
TPD-JV4K9T	SCHEMBL25358120	2-(2,6-Dioxopiperidin-3-yl)-4-[6-[4-[1-[3-ethoxy-4-[(5-methyl-11-methylsulfonyl-6-oxopyrimido[4,5-b][1,4]benzodiazepin-2-yl)amino]benzoyl]piperidin-4-yl]piperazin-1-yl]hexylamino]isoindole-1,3-dione; SCHEMBL30526049	CCOc1cc(C(=O)N2CCC(N3CCN(CCCCCCNc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)ccc1Nc1ncc2c(n1)N(S(C)(=O)=O)c1ccccc1C(=O)N2C	C50H59N11O9S	ERK5	Q13164	CRBN	WO-2023156791-A1
TPD-BE39TQ	SCHEMBL25357853	3-[7-[3-[2-[2-[4-[1-[3-ethoxy-4-[(5-methyl-11-methylsulfonyl-6-oxopyrimido[4,5-b][1,4]benzodiazepin-2-yl)amino]benzoyl]piperidin-4-yl]piperazin-1-yl]ethoxy]ethoxy]prop-1-ynyl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30526050	CCOc1cc(C(=O)N2CCC(N3CCN(CCOCCOCC#Cc4cccc5c4CN(C4CCC(=O)NC4=O)C5=O)CC3)CC2)ccc1Nc1ncc2c(n1)N(S(C)(=O)=O)c1ccccc1C(=O)N2C	C51H58N10O10S	ERK5	Q13164	CRBN	WO-2023156791-A1
TPD-ATLMUF	SCHEMBL26116829	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[[4-[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]ethyl]piperidin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26116838; SCHEMBL30588381	CC(C1CCN(CC2CCN(c3ccc(C(=O)N[C@H]4CC[C@H](Oc5ccc(C#N)c(Cl)c5)CC4)nn3)CC2)CC1)n1ccc2c(N3CCC(=O)NC3=O)cccc21	C43H50ClN9O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-4LNMA3	WO2023180388A1_AR1	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-4-[1-[2-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]acetyl]piperidin-4-yl]benzamide	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(C4CCN(C(=O)CN5CCC(n6ccc7c(N8CCC(=O)NC8=O)cccc76)CC5)CC4)cc3)CC2)cc1Cl	C44H48ClN7O5	AR	P10275	CRBN	WO-2023180388-A1
TPD-T0VG8R	SCHEMBL26362432	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-2-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyrimidine-5-carboxamide	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCC(CN5CCC(n6ccc7c(N8CCC(=O)NC8=O)cccc76)CC5)CC4)nc3)CC2)cc1Cl	C41H46ClN9O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-K4MMN3	SCHEMBL26365051	4-[3-[4-[4-[2-[4-[4-(2,4-Dioxo-1,3-diazinan-1-yl)pyrrolo[2,3-c]pyridin-1-yl]piperidin-1-yl]ethyl]piperidin-1-yl]phenyl]-4,4-dimethyl-5-oxo-2-sulfanylideneimidazolidin-1-yl]-2-(trifluoromethyl)benzonitrile	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=S)N1c1ccc(N2CCC(CCN3CCC(n4ccc5c(N6CCC(=O)NC6=O)cncc54)CC3)CC2)cc1	C42H44F3N9O3S	AR	P10275	CRBN	WO-2023180388-A1
TPD-B52W1E	SCHEMBL26116990	4-[3-[4-[4-[[4-[4-(2,4-Dioxo-1,3-diazinan-1-yl)pyrrolo[2,3-c]pyridin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-4,4-dimethyl-5-oxo-2-sulfanylideneimidazolidin-1-yl]-2-(trifluoromethyl)benzonitrile; SCHEMBL30588362	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=S)N1c1ccc(N2CCC(CN3CCC(n4ccc5c(N6CCC(=O)NC6=O)cncc54)CC3)CC2)cc1	C41H42F3N9O3S	AR	P10275	CRBN	WO-2023180388-A1
TPD-EPG1SD	SCHEMBL26365091	4-[3-[4-[4-[4-[4-(2,4-Dioxo-1,3-diazinan-1-yl)pyrrolo[2,3-c]pyridin-1-yl]piperidin-1-yl]butoxy]phenyl]-4,4-dimethyl-5-oxo-2-sulfanylideneimidazolidin-1-yl]-2-(trifluoromethyl)benzonitrile	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=S)N1c1ccc(OCCCCN2CCC(n3ccc4c(N5CCC(=O)NC5=O)cncc43)CC2)cc1	C39H39F3N8O4S	AR	P10275	CRBN	WO-2023180388-A1
TPD-0ZAHDX	SCHEMBL26365103	4-[3-[4-[3-[4-[4-(2,4-Dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]propoxy]phenyl]-4,4-dimethyl-5-oxo-2-sulfanylideneimidazolidin-1-yl]-2-(trifluoromethyl)benzonitrile	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=S)N1c1ccc(OCCCN2CCC(n3ccc4c(N5CCC(=O)NC5=O)cccc43)CC2)cc1	C39H38F3N7O4S	AR	P10275	CRBN	WO-2023180388-A1
TPD-8S5AR2	SCHEMBL26112077	4-[3-[4-[3-[4-[4-(2,4-Dioxo-1,3-diazinan-1-yl)pyrrolo[2,3-c]pyridin-1-yl]piperidin-1-yl]propoxy]phenyl]-4,4-dimethyl-5-oxo-2-sulfanylideneimidazolidin-1-yl]-2-(trifluoromethyl)benzonitrile; SCHEMBL30588451	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=S)N1c1ccc(OCCCN2CCC(n3ccc4c(N5CCC(=O)NC5=O)cncc43)CC2)cc1	C38H37F3N8O4S	AR	P10275	CRBN	WO-2023180388-A1
TPD-7UN64Z	WO2023180388A1_AR105	.	CCC(CCN(C)c1ncc(NC(=O)N2C[C@H](C)N(c3ccc(C#N)c(Cl)c3)C[C@H]2C)cn1)CN1CCC(N2CCc3c(N4CCC(=O)NC4=O)cccc32)CC1	C42H54ClN11O3	AR	P10275	CRBN	WO-2023180388-A1
TPD-L87V7E	WO2023180388A1_AR106	.	C[C@@H]1CN(c2ccc(C#N)c(Cl)c2)[C@@H](C)CN1C(=O)Nc1cnc(N2CCC(CN3CCC(n4ccc5c(N6CCC(=O)NC6=O)cncc54)CC3)CC2)nc1	C40H47ClN12O3	AR	P10275	CRBN	WO-2023180388-A1
TPD-65X3F4	SCHEMBL26365346	(2R,5S)-4-(3-chloro-4-cyanophenyl)-N-[2-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)-1-propan-2-ylindole-6-carbonyl]piperazin-1-yl]methyl]piperidin-1-yl]pyrimidin-5-yl]-2,5-dimethylpiperazine-1-carboxamide	CC(C)n1ccc2c(N3CCC(=O)NC3=O)cc(C(=O)N3CCN(CC4CCN(c5ncc(NC(=O)N6C[C@H](C)N(c7ccc(C#N)c(Cl)c7)C[C@H]6C)cn5)CC4)CC3)cc21	C44H53ClN12O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-H33M4E	WO2023180388A1_AR108	(2R,5S)-4-(3-chloro-4-cyanophenyl)-N-[6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridin-3-yl]-2,5-dimethylpiperazine-1-carboxamide	C[C@@H]1CN(c2ccc(C#N)c(Cl)c2)[C@@H](C)CN1C(=O)Nc1ccc(N2CCC(CN3CCC(n4ccc5c(N6CCC(=O)NC6=O)cccc54)CC3)CC2)nc1	C42H49ClN10O3	AR	P10275	CRBN	WO-2023180388-A1
TPD-0M8HKA	SCHEMBL26365462	(2R,5S)-4-(3-chloro-4-cyanophenyl)-N-[6-[4-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]butoxy]pyridin-3-yl]-2,5-dimethylpiperazine-1-carboxamide	C[C@@H]1CN(c2ccc(C#N)c(Cl)c2)[C@@H](C)CN1C(=O)Nc1ccc(OCCCCN2CCC(n3ccc4c(N5CCC(=O)NC5=O)cccc43)CC2)nc1	C40H46ClN9O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-JTOIYR	WO2023180388A1_AR11	.	CC1(C)[C@H](NC(=O)c2cnc(N3CCC(CN4CCC(n5ccc6c(N7CCC(=O)NC7=O)cccc65)CC4)CC3)nc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C43H50ClN9O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-6XML5D	SCHEMBL26365539	(2R,5S)-4-(3-chloro-4-cyanophenyl)-N-[6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)pyrrolo[2,3-c]pyridin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridin-3-yl]-2,5-dimethylpiperazine-1-carboxamide	C[C@@H]1CN(c2ccc(C#N)c(Cl)c2)[C@@H](C)CN1C(=O)Nc1ccc(N2CCC(CN3CCC(n4ccc5c(N6CCC(=O)NC6=O)cncc54)CC3)CC2)nc1	C41H48ClN11O3	AR	P10275	CRBN	WO-2023180388-A1
TPD-GODK2A	WO2023180388A1_AR111	.	C[C@@H]1CN(c2ccc(C#N)c(Cl)c2)[C@@H](C)CN1C(=O)Nc1ccc(OCCCCN2CCC(n3ccc4c(N5CCC(=O)NC5=O)cncc43)CC2)nc1	C39H45ClN10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-PCERI7	WO2023180388A1_AR112	.	CC(C)n1ccc2c(N3CCC(=O)NC3=O)cc(C(=O)N3CCN(CC4CCN(c5ccc(NC(=O)N6C[C@H](C)N(c7ccc(C#N)c(Cl)c7)C[C@H]6C)cn5)CC4)CC3)cc21	C45H54ClN11O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-BVNGK7	WO2023180388A1_AR113	.	CC(C)n1ccc2c(N3CCC(=O)NC3=O)cc(C(=O)N3CCN(CCCCOc4ccc(NC(=O)N5C[C@H](C)N(c6ccc(C#N)c(Cl)c6)C[C@H]5C)cn4)CC3)cc21	C43H51ClN10O5	AR	P10275	CRBN	WO-2023180388-A1
TPD-F5FFJ9	WO2023180388A1_AR115	.	C[C@@H]1CN(c2ccc(C#N)c(Cl)c2)[C@@H](C)CN1C(=O)Nc1ccc(N2CCC(CCN3CCC(n4ccc5c(N6CCC(=O)NC6=O)cccc54)CC3)CC2)nc1	C43H51ClN10O3	AR	P10275	CRBN	WO-2023180388-A1
TPD-XJ9FPD	SCHEMBL26115740	(2S,5R)-4-(3-chloro-4-cyanophenyl)-N-[2-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyrimidin-5-yl]-2,5-dimethylpiperazine-1-carboxamide; SCHEMBL30588433	C[C@@H]1CN(C(=O)Nc2cnc(N3CCC(CN4CCC(n5ccc6c(N7CCC(=O)NC7=O)cccc65)CC4)CC3)nc2)[C@@H](C)CN1c1ccc(C#N)c(Cl)c1	C41H48ClN11O3	AR	P10275	CRBN	WO-2023180388-A1
TPD-FXF2FF	WO2023180388A1_AR118	.	CC(C)n1ccc2c(N3CCC(=O)NC3=O)cc(C(=O)N3CCN(CCC4CCN(c5ccc(NC(=O)N6C[C@H](C)N(c7ccc(C#N)c(Cl)c7)C[C@H]6C)cn5)CC4)CC3)cc21	C46H56ClN11O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-K6TTCF	SCHEMBL26116099	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)pyrrolo[2,3-d]pyrimidin-7-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26116106; SCHEMBL30588315	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC(n6ccc7c(N8CCC(=O)NC8=O)ncnc76)CC5)CC4)nn3)CC2)cc1Cl	C39H44ClN11O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-Y86YIK	SCHEMBL26362639	N-[4-[4-cyano-3-(trifluoromethyl)phenoxy]cyclohexyl]-6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridine-3-carboxamide	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC(n6ccc7c(N8CCC(=O)NC8=O)cccc76)CC5)CC4)nc3)CC2)cc1C(F)(F)F	C43H47F3N8O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-Z4ZKYN	SCHEMBL26115919	(2S,5R)-4-(3-chloro-4-cyanophenyl)-N-[6-[4-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]butoxy]pyridin-3-yl]-2,5-dimethylpiperazine-1-carboxamide; SCHEMBL30588491	C[C@@H]1CN(C(=O)Nc2ccc(OCCCCN3CCC(n4ccc5c(N6CCC(=O)NC6=O)cccc54)CC3)nc2)[C@@H](C)CN1c1ccc(C#N)c(Cl)c1	C40H46ClN9O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-WYQY0R	SCHEMBL26115984	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)pyrazolo[3,4-b]pyridin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26115996; SCHEMBL30588274	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC(n6ncc7c(N8CCC(=O)NC8=O)ccnc76)CC5)CC4)nn3)CC2)cc1Cl	C39H44ClN11O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-4X2IQG	SCHEMBL26113108	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[(2R)-2-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]morpholin-4-yl]pyridazine-3-carboxamide; SCHEMBL26365939; SCHEMBL30588188	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCO[C@H](CN5CCC(n6ccc7c(N8CCC(=O)NC8=O)cccc76)CC5)C4)nn3)CC2)cc1Cl	C40H44ClN9O5	AR	P10275	CRBN	WO-2023180388-A1
TPD-C5KLCE	SCHEMBL26112844	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[(2S)-2-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indazol-1-yl]piperidin-1-yl]methyl]morpholin-4-yl]pyridazine-3-carboxamide; SCHEMBL26365945; SCHEMBL30588536	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCO[C@@H](CN5CCC(n6ncc7c(N8CCC(=O)NC8=O)cccc76)CC5)C4)nn3)CC2)cc1Cl	C39H43ClN10O5	AR	P10275	CRBN	WO-2023180388-A1
TPD-MK2E99	SCHEMBL26116523	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[(2S)-2-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]morpholin-4-yl]pyridazine-3-carboxamide; SCHEMBL26365962; SCHEMBL30588513	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCO[C@@H](CN5CCC(n6ccc7c(N8CCC(=O)NC8=O)cccc76)CC5)C4)nn3)CC2)cc1Cl	C40H44ClN9O5	AR	P10275	CRBN	WO-2023180388-A1
TPD-AA3E6O	SCHEMBL26114507	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[(2R)-2-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indazol-1-yl]piperidin-1-yl]methyl]morpholin-4-yl]pyridazine-3-carboxamide; SCHEMBL26365973; SCHEMBL30588574	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCO[C@H](CN5CCC(n6ncc7c(N8CCC(=O)NC8=O)cccc76)CC5)C4)nn3)CC2)cc1Cl	C39H43ClN10O5	AR	P10275	CRBN	WO-2023180388-A1
TPD-AUT02F	SCHEMBL26110945	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indazol-1-yl]piperidin-1-yl]methyl]-4-fluoropiperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26110951; SCHEMBL30588471	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(F)(CN5CCC(n6ncc7c(N8CCC(=O)NC8=O)cccc76)CC5)CC4)nn3)CC2)cc1Cl	C40H44ClFN10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-B2ITNK	SCHEMBL26116034	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)pyrazolo[3,4-c]pyridin-1-yl]piperidin-1-yl]methyl]-4-fluoropiperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26116038; SCHEMBL30588359	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(F)(CN5CCC(n6ncc7c(N8CCC(=O)NC8=O)cncc76)CC5)CC4)nn3)CC2)cc1Cl	C39H43ClFN11O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-TS25AB	WO2023180388A1_AR13	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC(n6ccc7c(N8CCC(=O)NC8=O)cccc76)CC5)CC4)nc3)CC2)cc1Cl	C42H47ClN8O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-P67IAI	SCHEMBL26111997	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-4-[2-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]ethyl]benzamide; SCHEMBL26112003; SCHEMBL30588314	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(CCN4CCC(n5ccc6c(N7CCC(=O)NC7=O)cccc65)CC4)cc3)CC2)cc1Cl	C39H41ClN6O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-JQ6J58	SCHEMBL26119980	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[[3-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]azetidin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26119984; SCHEMBL30588335	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CC(n6ccc7c(N8CCC(=O)NC8=O)cccc76)C5)CC4)nn3)CC2)cc1Cl	C39H42ClN9O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-728DOM	SCHEMBL26115830	(2S,5R)-4-(3-chloro-4-cyanophenyl)-N-[6-[4-[2-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)pyrazolo[3,4-c]pyridin-1-yl]piperidin-1-yl]ethyl]piperidin-1-yl]pyridin-3-yl]-2,5-dimethylpiperazine-1-carboxamide	C[C@@H]1CN(C(=O)Nc2ccc(N3CCC(CCN4CCC(n5ncc6c(N7CCC(=O)NC7=O)cncc65)CC4)CC3)nc2)[C@@H](C)CN1c1ccc(C#N)c(Cl)c1	C41H49ClN12O3	AR	P10275	CRBN	WO-2023180388-A1
TPD-33Y1SY	SCHEMBL26113121	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[2-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]-2-oxoethyl]piperazin-1-yl]pyridazine-3-carboxamide; SCHEMBL26113124; SCHEMBL30588507	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCN(CC(=O)N5CCC(n6ccc7c(N8CCC(=O)NC8=O)cccc76)CC5)CC4)nn3)CC2)cc1Cl	C41H45ClN10O5	AR	P10275	CRBN	WO-2023180388-A1
TPD-YGB40H	WO2023180388A1_AR135	.	CC(C1CCN(c2ccc(C(=O)N[C@H]3CC[C@H](Oc4ccc(C#N)c(Cl)c4)CC3)nn2)CC1)N1CCC(n2ccc3c(N4CCC(=O)NC4=O)cccc32)CC1	C42H48ClN9O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-I1NUKQ	SCHEMBL26114026	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[(3R)-3-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indazol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26366052; SCHEMBL30588250	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC[C@H](CN5CCC(n6ncc7c(N8CCC(=O)NC8=O)cccc76)CC5)C4)nn3)CC2)cc1Cl	C40H45ClN10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-WBE93K	SCHEMBL26116249	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[(3S)-3-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indazol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26366065; SCHEMBL30588264	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC[C@@H](CN5CCC(n6ncc7c(N8CCC(=O)NC8=O)cccc76)CC5)C4)nn3)CC2)cc1Cl	C40H45ClN10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-A42VD0	SCHEMBL26118901	(2S,5R)-4-(3-chloro-4-cyanophenyl)-N-[6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indazol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridin-3-yl]-2,5-dimethylpiperazine-1-carboxamide	C[C@@H]1CN(C(=O)Nc2ccc(N3CCC(CN4CCC(n5ncc6c(N7CCC(=O)NC7=O)cccc65)CC4)CC3)nc2)[C@@H](C)CN1c1ccc(C#N)c(Cl)c1	C41H48ClN11O3	AR	P10275	CRBN	WO-2023180388-A1
TPD-AESAPF	SCHEMBL26115651	2-chloro-4-[(2S,5R)-4-[2-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)pyrazolo[3,4-c]pyridin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyrimidine-5-carbonyl]-2,5-dimethylpiperazin-1-yl]benzonitrile	C[C@@H]1CN(c2ccc(C#N)c(Cl)c2)[C@@H](C)CN1C(=O)c1cnc(N2CCC(CN3CCC(n4ncc5c(N6CCC(=O)NC6=O)cncc54)CC3)CC2)nc1	C39H45ClN12O3	AR	P10275	CRBN	WO-2023180388-A1
TPD-7ELGIF	SCHEMBL26362775	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-5-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)pyrrolo[2,3-c]pyridin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyrazine-2-carboxamide	CC1(C)[C@H](NC(=O)c2cnc(N3CCC(CN4CCC(n5ccc6c(N7CCC(=O)NC7=O)cncc65)CC4)CC3)cn2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C42H49ClN10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-0T06TK	SCHEMBL26113680	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)-5-fluoroindazol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26113695	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC(n6ncc7c(N8CCC(=O)NC8=O)c(F)ccc76)CC5)CC4)nn3)CC2)cc1Cl	C40H44ClFN10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-JESAKC	SCHEMBL26118842	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[[4-[4-(2,4-dioxopyrimidin-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26118852	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC(n6ccc7c(-n8ccc(=O)[nH]c8=O)cccc76)CC5)CC4)nn3)CC2)cc1Cl	C41H44ClN9O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-1QQ9TQ	SCHEMBL26119097	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[(3R)-3-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26366115; SCHEMBL30588540	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC[C@H](CN5CCC(n6ccc7c(N8CCC(=O)NC8=O)cccc76)CC5)C4)nn3)CC2)cc1Cl	C41H46ClN9O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-NF36AC	SCHEMBL26114958	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[(3S)-3-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26364670; SCHEMBL30588251	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC[C@@H](CN5CCC(n6ccc7c(N8CCC(=O)NC8=O)cccc76)CC5)C4)nn3)CC2)cc1Cl	C41H46ClN9O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-2HEBEU	SCHEMBL26112290	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[[(3R,4R)-4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]-3-fluoropiperidin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26112295; SCHEMBL30588517	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CC[C@@H](n6ccc7c(N8CCC(=O)NC8=O)cccc76)[C@H](F)C5)CC4)nn3)CC2)cc1Cl	C41H45ClFN9O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-R6UKB1	SCHEMBL26116083	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[[(3S,4S)-4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]-3-fluoropiperidin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26116088; SCHEMBL30588397	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CC[C@H](n6ccc7c(N8CCC(=O)NC8=O)cccc76)[C@@H](F)C5)CC4)nn3)CC2)cc1Cl	C41H45ClFN9O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-0P5NR6	WO2023180388A1_AR146	.	C[C@H]1CN(C(=O)c2ccc(N3CCC(CN4CCC(n5ncc6c(N7CCC(=O)NC7=O)cncc65)CC4)CC3)nn2)[C@H](I)CN1c1ccc(C#N)c(Cl)c1	C38H42ClIN12O3	AR	P10275	CRBN	WO-2023180388-A1
TPD-HJ84K6	SCHEMBL26116029	2-chloro-4-[(2S,5R)-4-[5-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)pyrrolo[2,3-c]pyridin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyrazine-2-carbonyl]-2,5-dimethylpiperazin-1-yl]benzonitrile; SCHEMBL30588582	C[C@@H]1CN(c2ccc(C#N)c(Cl)c2)[C@@H](C)CN1C(=O)c1cnc(N2CCC(CN3CCC(n4ccc5c(N6CCC(=O)NC6=O)cncc54)CC3)CC2)cn1	C40H46ClN11O3	AR	P10275	CRBN	WO-2023180388-A1
TPD-27OGFV	SCHEMBL26117670	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)pyrrolo[3,2-c]pyridin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26117684; SCHEMBL30588671	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC(n6ccc7c(N8CCC(=O)NC8=O)nccc76)CC5)CC4)nn3)CC2)cc1Cl	C40H45ClN10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-7PUXQA	SCHEMBL26113412	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)pyrrolo[2,3-b]pyridin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26113420; SCHEMBL30588384; SCHEMBL30588386	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC(n6ccc7c(N8CCC(=O)NC8=O)ccnc76)CC5)CC4)nn3)CC2)cc1Cl	C40H45ClN10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-JXBD7D	WO2023180388A1_AR15	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCC(CN5CCC(n6ccc7c(N8CCC(=O)NC8=O)cncc76)CC5)CC4)cn3)CC2)cc1C(F)(F)F	C41H45F3N10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-B77RAR	SCHEMBL26114945	2-chloro-4-[(2S,5R)-4-[5-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)pyrazolo[3,4-c]pyridin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyrazine-2-carbonyl]-2,5-dimethylpiperazin-1-yl]benzonitrile; SCHEMBL30588651	C[C@@H]1CN(c2ccc(C#N)c(Cl)c2)[C@@H](C)CN1C(=O)c1cnc(N2CCC(CN3CCC(n4ncc5c(N6CCC(=O)NC6=O)cncc54)CC3)CC2)cn1	C39H45ClN12O3	AR	P10275	CRBN	WO-2023180388-A1
TPD-74VVJS	WO2023180388A1_AR151	.	CN(CCCN1CCC(n2ccc3c(N4CCC(=O)NC4=O)cccc32)CC1)c1ccc(C(=O)N[C@H]2CC[C@H](Oc3ccc(C#N)c(Cl)c3)CC2)nn1	C39H44ClN9O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-CZIPWF	SCHEMBL26366299	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[3-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indazol-1-yl]piperidin-1-yl]methyl]pyrrolidin-1-yl]pyridazine-3-carboxamide	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC(n6ncc7c(N8CCC(=O)NC8=O)cccc76)CC5)C4)nn3)CC2)cc1Cl	C39H43ClN10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-Y6N6FK	SCHEMBL26366342	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[3-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indazol-1-yl]piperidin-1-yl]methyl]azetidin-1-yl]pyridazine-3-carboxamide	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CC(CN5CCC(n6ncc7c(N8CCC(=O)NC8=O)cccc76)CC5)C4)nn3)CC2)cc1Cl	C38H41ClN10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-STMY14	SCHEMBL26115055	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[[(3S,4R)-4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]-3-fluoropiperidin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26115058; SCHEMBL30588489	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CC[C@@H](n6ccc7c(N8CCC(=O)NC8=O)cccc76)[C@@H](F)C5)CC4)nn3)CC2)cc1Cl	C41H45ClFN9O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-7WU90F	SCHEMBL26112965	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[[(3R,4S)-4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]-3-fluoropiperidin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26112967; SCHEMBL30588408	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CC[C@H](n6ccc7c(N8CCC(=O)NC8=O)cccc76)[C@H](F)C5)CC4)nn3)CC2)cc1Cl	C41H45ClFN9O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-K18M3V	WO2023180388A1_AR157	.	CN(c1ccc(C#N)c(Cl)c1)[C@H]1CC[C@H](NC(=O)c2ccc(N3CCC(CN4C=CC(n5ccc6c(N7CCC(=O)NC7=O)cccc65)CC4)CC3)nn2)CC1	C42H47ClN10O3	AR	P10275	CRBN	WO-2023180388-A1
TPD-99SDZA	SCHEMBL26118911	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[2-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indazol-1-yl]piperidin-1-yl]-2-oxoethyl]piperazin-1-yl]pyridazine-3-carboxamide; SCHEMBL26118914; SCHEMBL30588283	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCN(CC(=O)N5CCC(n6ncc7c(N8CCC(=O)NC8=O)cccc76)CC5)CC4)nn3)CC2)cc1Cl	C40H44ClN11O5	AR	P10275	CRBN	WO-2023180388-A1
TPD-SYXJ8A	SCHEMBL26366505	N-[4-(4-chloro-3-cyanophenoxy)cyclohexyl]-6-[4-[[(3S)-3-[[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]methyl]-3-fluoropiperidin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide	N#Cc1cc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC[C@@](F)(Cn6ccc7c(N8CCC(=O)NC8=O)cccc76)C5)CC4)nn3)CC2)ccc1Cl	C42H47ClFN9O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-869T3E	WO2023180388A1_AR16	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCC(CN5CCC(n6ccc7c(N8CCC(=O)NC8=O)cncc76)CC5)CC4)cn3)CC2)cc1Cl	C40H45ClN10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-SPPRI5	SCHEMBL26114441	2-chloro-4-[(2S,5R)-4-[6-[4-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)pyrrolo[2,3-c]pyridin-1-yl]piperidin-1-yl]butoxy]pyridine-3-carbonyl]-2,5-dimethylpiperazin-1-yl]benzonitrile; SCHEMBL30588258	C[C@@H]1CN(c2ccc(C#N)c(Cl)c2)[C@@H](C)CN1C(=O)c1ccc(OCCCCN2CCC(n3ccc4c(N5CCC(=O)NC5=O)cncc43)CC2)nc1	C39H44ClN9O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-DT8PDL	SCHEMBL26116397	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]-3,3-difluoropiperidin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26116401; SCHEMBL30588287	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC(n6ccc7c(N8CCC(=O)NC8=O)cccc76)C(F)(F)C5)CC4)nn3)CC2)cc1Cl	C41H44ClF2N9O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-OALBDH	SCHEMBL26117188	2-chloro-4-[(2S,5R)-4-[6-[5-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)pyrazolo[3,4-c]pyridin-1-yl]piperidin-1-yl]pentoxy]pyridine-3-carbonyl]-2,5-dimethylpiperazin-1-yl]benzonitrile; SCHEMBL30588389	C[C@@H]1CN(c2ccc(C#N)c(Cl)c2)[C@@H](C)CN1C(=O)c1ccc(OCCCCCN2CCC(n3ncc4c(N5CCC(=O)NC5=O)cncc43)CC2)nc1	C39H45ClN10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-7WGMA6	SCHEMBL26117571	2-chloro-4-[(2S,5R)-4-[6-[5-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)pyrrolo[2,3-c]pyridin-1-yl]piperidin-1-yl]pentoxy]pyridine-3-carbonyl]-2,5-dimethylpiperazin-1-yl]benzonitrile; SCHEMBL30588348	C[C@@H]1CN(c2ccc(C#N)c(Cl)c2)[C@@H](C)CN1C(=O)c1ccc(OCCCCCN2CCC(n3ccc4c(N5CCC(=O)NC5=O)cncc43)CC2)nc1	C40H46ClN9O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-OX24RH	SCHEMBL26114991	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[1-[2-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]-2-oxoethyl]piperidin-4-yl]pyridazine-3-carboxamide; SCHEMBL26114994; SCHEMBL30588295	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(C4CCN(CC(=O)N5CCC(n6ccc7c(N8CCC(=O)NC8=O)cccc76)CC5)CC4)nn3)CC2)cc1Cl	C42H46ClN9O5	AR	P10275	CRBN	WO-2023180388-A1
TPD-NUZVIE	SCHEMBL26112383	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[[4-[[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]methyl]-4-fluoropiperidin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26112391; SCHEMBL30588257	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC(F)(Cn6ccc7c(N8CCC(=O)NC8=O)cccc76)CC5)CC4)nn3)CC2)cc1Cl	C42H47ClFN9O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-N7E2DA	SCHEMBL26114137	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-4-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]benzamide; SCHEMBL26114149; SCHEMBL30588273	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC(n6ccc7c(N8CCC(=O)NC8=O)cccc76)CC5)CC4)cc3)CC2)cc1Cl	C43H48ClN7O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-2AIC77	WO2023180388A1_AR17	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCC(CN5CCC(n6ccc7c(N8CCC(=O)NC8=O)cncc76)CC5)CC4)nc3)CC2)cc1C(F)(F)F	C41H45F3N10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-GDUC5P	SCHEMBL26117623	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)-5-fluoroindol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26117631	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC(n6ccc7c(N8CCC(=O)NC8=O)c(F)ccc76)CC5)CC4)nn3)CC2)cc1Cl	C41H45ClFN9O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-GEKFXG	SCHEMBL26116247	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[[(3S)-3-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]pyrrolidin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CC[C@H](n6ccc7c(N8CCC(=O)NC8=O)cccc76)C5)CC4)nn3)CC2)cc1Cl	C40H44ClN9O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-SS1PRT	SCHEMBL26115531	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[[(3R)-3-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]pyrrolidin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CC[C@@H](n6ccc7c(N8CCC(=O)NC8=O)cccc76)C5)CC4)nn3)CC2)cc1Cl	C40H44ClN9O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-3JBE6M	SCHEMBL26119139	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[[6-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]-2-azaspiro[3.3]heptan-2-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26119148; SCHEMBL30588240	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CC6(CC(n7ccc8c(N9CCC(=O)NC9=O)cccc87)C6)C5)CC4)nn3)CC2)cc1Cl	C42H46ClN9O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-8WM0HO	SCHEMBL26119663	2-chloro-4-[(2S,5R)-4-[6-[2-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)pyrazolo[3,4-c]pyridin-1-yl]piperidin-1-yl]ethoxy]pyridine-3-carbonyl]-2,5-dimethylpiperazin-1-yl]benzonitrile; SCHEMBL30588452	C[C@@H]1CN(c2ccc(C#N)c(Cl)c2)[C@@H](C)CN1C(=O)c1ccc(OCCN2CCC(n3ncc4c(N5CCC(=O)NC5=O)cncc43)CC2)nc1	C36H39ClN10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-T751AF	SCHEMBL26113013	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[[4-[2-chloro-4-(2,4-dioxo-1,3-diazinan-1-yl)pyrrolo[2,3-d]pyrimidin-7-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26113029	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC(n6ccc7c(N8CCC(=O)NC8=O)nc(Cl)nc76)CC5)CC4)nn3)CC2)cc1Cl	C39H43Cl2N11O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-1F4P3A	SCHEMBL26115691	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)-6-(trifluoromethyl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26115699; SCHEMBL30588228	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC(n6ccc7c(N8CCC(=O)NC8=O)cc(C(F)(F)F)cc76)CC5)CC4)nn3)CC2)cc1Cl	C42H45ClF3N9O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-XQ7RE5	SCHEMBL26117387	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[[4-[8-(2,4-dioxo-1,3-diazinan-1-yl)imidazo[1,5-a]pyridin-3-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26117397; SCHEMBL30588485	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC(c6ncc7c(N8CCC(=O)NC8=O)cccn67)CC5)CC4)nn3)CC2)cc1Cl	C40H45ClN10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-TVFR1C	SCHEMBL26118916	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[1-[2-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]acetyl]azetidin-3-yl]oxypyridazine-3-carboxamide; SCHEMBL26118921; SCHEMBL30588213	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(OC4CN(C(=O)CN5CCC(n6ccc7c(N8CCC(=O)NC8=O)cccc76)CC5)C4)nn3)CC2)cc1Cl	C40H42ClN9O6	AR	P10275	CRBN	WO-2023180388-A1
TPD-QZJXKV	SCHEMBL26367019	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[[4-[2-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]ethyl]piperidin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC(CCn6ccc7c(N8CCC(=O)NC8=O)cccc76)CC5)CC4)nn3)CC2)cc1Cl	C43H50ClN9O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-J31AQG	WO2023180388A1_AR18	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-2-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)pyrrolo[2,3-c]pyridin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyrimidine-5-carboxamide	CC1(C)[C@H](NC(=O)c2cnc(N3CCC(CN4CCC(n5ccc6c(N7CCC(=O)NC7=O)cncc65)CC4)CC3)nc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C42H49ClN10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-IN9AJS	SCHEMBL26110673	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]benzamide; SCHEMBL26110677; SCHEMBL30588334	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(CN4CCC(n5ccc6c(N7CCC(=O)NC7=O)cccc65)CC4)cc3)CC2)cc1Cl	C38H39ClN6O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-M77R0A	SCHEMBL26119372	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-5-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)pyrrolo[3,2-c]pyridin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyrazine-2-carboxamide; SCHEMBL26119387; SCHEMBL30588332	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCC(CN5CCC(n6ccc7c(N8CCC(=O)NC8=O)nccc76)CC5)CC4)cn3)CC2)cc1Cl	C40H45ClN10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-QV9K08	WO2023180388A1_AR183	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[[(3S)-3-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC[C@H](n6ccc7c(N8CCC(=O)NC8=O)cccc76)C5)CC4)nn3)CC2)cc1Cl	C41H46ClN9O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-9OHBZG	SCHEMBL26111694	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[[(3R)-3-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL30588330	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC[C@@H](n6ccc7c(N8CCC(=O)NC8=O)cccc76)C5)CC4)nn3)CC2)cc1Cl	C41H46ClN9O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-GVTWQ6	SCHEMBL26367106	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[[2-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]-7-azaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC6(CC5)CC(n5ccc7c(N8CCC(=O)NC8=O)cccc75)C6)CC4)nn3)CC2)cc1Cl	C44H50ClN9O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-12DODG	SCHEMBL26114360	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-5-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridine-2-carboxamide; SCHEMBL26114370; SCHEMBL30588217	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC(n6ccc7c(N8CCC(=O)NC8=O)cccc76)CC5)CC4)cn3)CC2)cc1Cl	C42H47ClN8O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-L30VQ5	SCHEMBL26113857	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-4-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]-2-fluorobenzamide; SCHEMBL26113868; SCHEMBL30588259	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC(n6ccc7c(N8CCC(=O)NC8=O)cccc76)CC5)CC4)cc3F)CC2)cc1Cl	C43H47ClFN7O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-T50J9C	SCHEMBL26111491	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[(3S)-1-[2-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]acetyl]pyrrolidin-3-yl]oxypyridazine-3-carboxamide; SCHEMBL26367155; SCHEMBL30588305	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(O[C@H]4CCN(C(=O)CN5CCC(n6ccc7c(N8CCC(=O)NC8=O)cccc76)CC5)C4)nn3)CC2)cc1Cl	C41H44ClN9O6	AR	P10275	CRBN	WO-2023180388-A1
TPD-4WIOQP	SCHEMBL26367165	N-[4-[4-cyano-3-(trifluoromethyl)phenoxy]cyclohexyl]-5-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)-5-fluoroindazol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyrazine-2-carboxamide	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCC(CN5CCC(n6ncc7c(N8CCC(=O)NC8=O)c(F)ccc76)CC5)CC4)cn3)CC2)cc1C(F)(F)F	C41H44F4N10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-M23T2V	WO2023180388A1_AR19	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC(n6ccc7c(N8CCC(=O)NC8=O)cncc76)CC5)CC4)cc3)CC2)cc1C(F)(F)F	C43H47F3N8O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-RM7QCH	SCHEMBL26367186	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-5-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)-5-fluoroindazol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyrazine-2-carboxamide	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCC(CN5CCC(n6ncc7c(N8CCC(=O)NC8=O)c(F)ccc76)CC5)CC4)cn3)CC2)cc1Cl	C40H44ClFN10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-GMXHD2	SCHEMBL26121792	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[2-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]-7-azaspiro[3.5]nonan-7-yl]pyridazine-3-carboxamide; SCHEMBL26121802; SCHEMBL30588417	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC5(CC4)CC(N4CCC(n6ccc7c(N8CCC(=O)NC8=O)cccc76)CC4)C5)nn3)CC2)cc1Cl	C43H48ClN9O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-7IVH11	WO2023180388A1_AR194	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCN(CC5CCC(n6ccc7c(N8CCC(=O)NC8=O)cccc76)CC5)CC4)nn3)CC2)cc1Cl	C41H46ClN9O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-44MJVF	SCHEMBL26367264	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-4-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)pyrrolo[2,3-d]pyrimidin-7-yl]piperidin-1-yl]methyl]piperidin-1-yl]benzamide	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC(n6ccc7c(N8CCC(=O)NC8=O)ncnc76)CC5)CC4)cc3)CC2)cc1Cl	C41H46ClN9O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-4F7GCD	SCHEMBL26367272	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-5-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)pyrrolo[2,3-d]pyrimidin-7-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyrazine-2-carboxamide	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCC(CN5CCC(n6ccc7c(N8CCC(=O)NC8=O)ncnc76)CC5)CC4)cn3)CC2)cc1Cl	C39H44ClN11O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-FP3ZLQ	WO2023180388A1_AR197	.	N#Cc1ccc(C[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC(n6ccc7c(N8CCC(=O)NC8=O)nccc76)CC5)CC4)cc3)CC2)cc1Cl	C43H49ClN8O3	AR	P10275	CRBN	WO-2023180388-A1
TPD-DWWORM	SCHEMBL26116011	N-[4-[4-cyano-3-(trifluoromethyl)phenoxy]cyclohexyl]-5-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)pyrrolo[2,3-d]pyrimidin-7-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyrazine-2-carboxamide; SCHEMBL26116028; SCHEMBL30588363	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCC(CN5CCC(n6ccc7c(N8CCC(=O)NC8=O)ncnc76)CC5)CC4)cn3)CC2)cc1C(F)(F)F	C40H44F3N11O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-YIQ4VW	SCHEMBL26116658	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-4-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)pyrazolo[4,3-c]pyridin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]benzamide; SCHEMBL26116665; SCHEMBL30588255	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC(n6ncc7c(N8CCC(=O)NC8=O)nccc76)CC5)CC4)cc3)CC2)cc1Cl	C41H46ClN9O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-49J026	WO2023180388A1_AR2	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-3-[1-[2-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]acetyl]piperidin-4-yl]oxybenzamide	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cccc(OC4CCN(C(=O)CN5CCC(n6ccc7c(N8CCC(=O)NC8=O)cccc76)CC5)CC4)c3)CC2)cc1Cl	C44H48ClN7O6	AR	P10275	CRBN	WO-2023180388-A1
TPD-ZM03WJ	WO2023180388A1_AR20	.	CC1(C)[C@H](NC(=O)c2ccc(N3CCC(CN4CCC(n5ccc6c5CNC=C6N5CCC(=O)NC5=O)CC4)CC3)nc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C43H52ClN9O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-HPO6US	SCHEMBL26367310	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-2-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)pyrrolo[2,3-d]pyrimidin-7-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyrimidine-5-carboxamide	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCC(CN5CCC(n6ccc7c(N8CCC(=O)NC8=O)ncnc76)CC5)CC4)nc3)CC2)cc1Cl	C39H44ClN11O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-YFLWNK	WO2023180388A1_AR201	N-[4-(3-chloro-4-cyano-N-methylanilino)cyclohexyl]-6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)-6-fluoroindol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide	CN(c1ccc(C#N)c(Cl)c1)[C@H]1CC[C@H](NC(=O)c2ccc(N3CCC(CN4CCC(n5ccc6c(N7CCC(=O)NC7=O)cc(F)cc65)CC4)CC3)nn2)CC1	C42H48ClFN10O3	AR	P10275	CRBN	WO-2023180388-A1
TPD-XW50J3	SCHEMBL26367335	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-5-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)-6-fluoroindol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyrazine-2-carboxamide	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCC(CN5CCC(n6ccc7c(N8CCC(=O)NC8=O)cc(F)cc76)CC5)CC4)cn3)CC2)cc1Cl	C41H45ClFN9O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-H9AUZO	SCHEMBL26367348	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-5-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)pyrazolo[4,3-c]pyridin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyrazine-2-carboxamide	N#Cc1ccc(OC2CCC(NC(=O)c3cnc(N4CCC(CN5CCC(n6ncc7c(N8CCC(=O)NC8=O)nccc76)CC5)CC4)cn3)CC2)cc1Cl	C39H44ClN11O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-S6OJ3O	SCHEMBL26115659	N-[4-[4-cyano-3-(trifluoromethyl)phenoxy]cyclohexyl]-6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)pyrrolo[3,2-c]pyridin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26115674; SCHEMBL30588571	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC(n6ccc7c(N8CCC(=O)NC8=O)nccc76)CC5)CC4)nn3)CC2)cc1C(F)(F)F	C41H45F3N10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-0HMPD3	SCHEMBL26119578	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-2-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)-6-fluoroindazol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyrimidine-5-carboxamide; SCHEMBL26119587; SCHEMBL30588548	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCC(CN5CCC(n6ncc7c(N8CCC(=O)NC8=O)cc(F)cc76)CC5)CC4)nc3)CC2)cc1Cl	C40H44ClFN10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-1V5Y7O	SCHEMBL26117577	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-4-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]-3-fluorobenzamide; SCHEMBL26117588; SCHEMBL30588328	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC(n6ccc7c(N8CCC(=O)NC8=O)cccc76)CC5)CC4)c(F)c3)CC2)cc1Cl	C43H47ClFN7O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-L5DJRJ	WO2023180388A1_AR207	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCN(C[C@H]5C[C@@H](n6ccc7c(N8CCC(=O)NC8=O)cccc76)C5)CC4)nn3)CC2)cc1Cl	C39H42ClN9O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-5UFZVK	WO2023180388A1_AR208	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCN(C[C@H]5C[C@H](n6ccc7c(N8CCC(=O)NC8=O)cccc76)C5)CC4)nn3)CC2)cc1Cl	C39H42ClN9O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-CMAEY7	SCHEMBL26120872	N-[4-[4-cyano-3-(trifluoromethyl)phenoxy]cyclohexyl]-6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)pyrazolo[4,3-c]pyridin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26120884; SCHEMBL30588484	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC(n6ncc7c(N8CCC(=O)NC8=O)nccc76)CC5)CC4)nn3)CC2)cc1C(F)(F)F	C40H44F3N11O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-X40B8P	SCHEMBL26363233	N-[4-[4-cyano-3-(trifluoromethyl)phenoxy]cyclohexyl]-5-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyrazine-2-carboxamide	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCC(CN5CCC(n6ccc7c(N8CCC(=O)NC8=O)cccc76)CC5)CC4)cn3)CC2)cc1C(F)(F)F	C42H46F3N9O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-UIQNGG	SCHEMBL26113075	N-[4-[4-cyano-3-(trifluoromethyl)phenoxy]cyclohexyl]-6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)pyrazolo[3,4-b]pyridin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26113094; SCHEMBL30588343	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC(n6ncc7c(N8CCC(=O)NC8=O)ccnc76)CC5)CC4)nn3)CC2)cc1C(F)(F)F	C40H44F3N11O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-BTE0ZU	SCHEMBL26367452	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-2-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)pyrrolo[3,2-c]pyridin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyrimidine-5-carboxamide	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCC(CN5CCC(n6ccc7c(N8CCC(=O)NC8=O)nccc76)CC5)CC4)nc3)CC2)cc1Cl	C40H45ClN10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-XSWC7Q	SCHEMBL26116548	N-[4-[4-cyano-3-(trifluoromethyl)phenoxy]cyclohexyl]-6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)pyrrolo[2,3-b]pyridin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26116562; SCHEMBL30588409	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC(n6ccc7c(N8CCC(=O)NC8=O)ccnc76)CC5)CC4)nn3)CC2)cc1C(F)(F)F	C41H45F3N10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-QDD7TM	SCHEMBL26121603	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]-4-methylpiperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26121612; SCHEMBL30588319	CC1(CN2CCC(n3ccc4c(N5CCC(=O)NC5=O)cccc43)CC2)CCN(c2ccc(C(=O)NC3CCC(Oc4ccc(C#N)c(Cl)c4)CC3)nn2)CC1	C42H48ClN9O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-28OTVP	WO2023180388A1_AR214	N-[4-(3-chloro-4-cyano-N-methylanilino)cyclohexyl]-6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)pyrrolo[2,3-d]pyrimidin-7-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide	CN(c1ccc(C#N)c(Cl)c1)[C@H]1CC[C@H](NC(=O)c2ccc(N3CCC(CN4CCC(n5ccc6c(N7CCC(=O)NC7=O)ncnc65)CC4)CC3)nn2)CC1	C40H47ClN12O3	AR	P10275	CRBN	WO-2023180388-A1
TPD-AT95XK	WO2023180388A1_AR215	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCN(C[C@H]5CC[C@H](n6ccc7c(N8CCC(=O)NC8=O)cccc76)CC5)CC4)nn3)CC2)cc1Cl	C41H46ClN9O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-6VOFP7	SCHEMBL26119680	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-2-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)pyrazolo[3,4-c]pyridin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyrimidine-5-carboxamide; SCHEMBL26119688; SCHEMBL30588234	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCC(CN5CCC(n6ncc7c(N8CCC(=O)NC8=O)cncc76)CC5)CC4)nc3)CC2)cc1Cl	C39H44ClN11O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-UMJOBB	SCHEMBL26367549	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-5-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)-6-fluoroindazol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyrazine-2-carboxamide	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCC(CN5CCC(n6ncc7c(N8CCC(=O)NC8=O)cc(F)cc76)CC5)CC4)cn3)CC2)cc1Cl	C40H44ClFN10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-GIGTLX	SCHEMBL26367677	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[7-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indazol-1-yl]piperidin-1-yl]methyl]-5-oxa-2-azaspiro[3.5]nonan-2-yl]pyridazine-3-carboxamide	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CC5(CCC(CN6CCC(n7ncc8c(N9CCC(=O)NC9=O)cccc87)CC6)CO5)C4)nn3)CC2)cc1Cl	C42H47ClN10O5	AR	P10275	CRBN	WO-2023180388-A1
TPD-FY248U	SCHEMBL26367821	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[1-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indazol-1-yl]piperidin-1-yl]methyl]-3-azabicyclo[3.1.1]heptan-3-yl]pyridazine-3-carboxamide	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CC5CC(CN6CCC(n7ncc8c(N9CCC(=O)NC9=O)cccc87)CC6)(C5)C4)nn3)CC2)cc1Cl	C41H45ClN10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-VZX6UI	WO2023180388A1_AR220	.	CN(CCCCCN1CCC(n2ncc3c(N4CCC(=O)NC4=O)cccc32)CC1)c1ccc(C(=O)N[C@H]2CC[C@H](Oc3ccc(C#N)c(Cl)c3)CC2)nn1	C40H47ClN10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-SD1NR0	WO2023180388A1_AR221	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(C#N)(CCN5CCC(n6ncc7c(N8CCC(=O)NC8=O)cccc76)CC5)CC4)nn3)CC2)cc1Cl	C42H46ClN11O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-3EUX7I	SCHEMBL26367895	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[3-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indazol-1-yl]piperidin-1-yl]methyl]-4,4-dimethylpiperidin-1-yl]pyridazine-3-carboxamide	CC1(C)CCN(c2ccc(C(=O)N[C@H]3CC[C@H](Oc4ccc(C#N)c(Cl)c4)CC3)nn2)CC1CN1CCC(n2ncc3c(N4CCC(=O)NC4=O)cccc32)CC1	C42H49ClN10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-MPJXCS	SCHEMBL26367896	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[5-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indazol-1-yl]piperidin-1-yl]methyl]-3,3-dimethylpiperidin-1-yl]pyridazine-3-carboxamide	CC1(C)CC(CN2CCC(n3ncc4c(N5CCC(=O)NC5=O)cccc43)CC2)CN(c2ccc(C(=O)N[C@H]3CC[C@H](Oc4ccc(C#N)c(Cl)c4)CC3)nn2)C1	C42H49ClN10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-4FVXMZ	WO2023180388A1_AR224	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CC5(CC(CN6CCC(n7ncc8c(N9CCC(=O)NC9=O)cccc87)CC6)C5)C4)nn3)CC2)cc1Cl	C41H45ClN10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-IUJXMD	SCHEMBL26367958	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[7-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indazol-1-yl]piperidin-1-yl]methyl]-2-azaspiro[3.5]nonan-2-yl]pyridazine-3-carboxamide	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CC5(CCC(CN6CCC(n7ncc8c(N9CCC(=O)NC9=O)cccc87)CC6)CC5)C4)nn3)CC2)cc1Cl	C43H49ClN10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-QOR06I	WO2023180388A1_AR226	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CC5CCC(C4)C5CN4CCC(n5ncc6c(N7CCC(=N)NC7=O)cccc65)CC4)nn3)CC2)cc1Cl	C42H48ClN11O3	AR	P10275	CRBN	WO-2023180388-A1
TPD-WAZXI4	SCHEMBL26368020	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[(3R,4R)-4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indazol-1-yl]piperidin-1-yl]methyl]-3-methylpiperidin-1-yl]pyridazine-3-carboxamide	C[C@H]1CN(c2ccc(C(=O)N[C@H]3CC[C@H](Oc4ccc(C#N)c(Cl)c4)CC3)nn2)CC[C@H]1CN1CCC(n2ncc3c(N4CCC(=O)NC4=O)cccc32)CC1	C41H47ClN10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-6LVCYM	SCHEMBL26368107	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[6-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indazol-1-yl]piperidin-1-yl]methyl]-3-azabicyclo[3.1.1]heptan-3-yl]pyridazine-3-carboxamide	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CC5CC(C4)C5CN4CCC(n5ncc6c(N7CCC(=O)NC7=O)cccc65)CC4)nn3)CC2)cc1Cl	C41H45ClN10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-JXMSHZ	SCHEMBL26368157	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indazol-1-yl]piperidin-1-yl]methyl]-2-methylpiperidin-1-yl]pyridazine-3-carboxamide	CC1CC(CN2CCC(n3ncc4c(N5CCC(=O)NC5=O)cccc43)CC2)CCN1c1ccc(C(=O)N[C@H]2CC[C@H](Oc3ccc(C#N)c(Cl)c3)CC2)nn1	C41H47ClN10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-GEXEQU	SCHEMBL26363374	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL30588277	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC(n6ccc7c(N8CCC(=O)NC8=O)cccc76)CC5)CC4)nn3)CC2)cc1Cl	C41H46ClN9O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-BDJJII	SCHEMBL26368160	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[3-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indazol-1-yl]piperidin-1-yl]methyl]-8-azabicyclo[3.2.1]octan-8-yl]pyridazine-3-carboxamide	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4C5CCC4CC(CN4CCC(n6ncc7c(N8CCC(=O)NC8=O)cccc76)CC4)C5)nn3)CC2)cc1Cl	C42H47ClN10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-8V3RLQ	WO2023180388A1_AR231	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(OCCN5CCC(n6ncc7c(N8CCC(=O)NC8=O)cccc76)CC5)CC4)nn3)CC2)cc1Cl	C41H47ClN10O5	AR	P10275	CRBN	WO-2023180388-A1
TPD-2IZVDJ	SCHEMBL26368240	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indazol-1-yl]piperidin-1-yl]methyl]-2-methylpyrrolidin-1-yl]pyridazine-3-carboxamide	CC1CC(CN2CCC(n3ncc4c(N5CCC(=O)NC5=O)cccc43)CC2)CN1c1ccc(C(=O)N[C@H]2CC[C@H](Oc3ccc(C#N)c(Cl)c3)CC2)nn1	C40H45ClN10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-0Z5I4T	SCHEMBL26368283	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[2-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indazol-1-yl]piperidin-1-yl]methyl]-6-azaspiro[3.4]octan-6-yl]pyridazine-3-carboxamide	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC5(CC(CN6CCC(n7ncc8c(N9CCC(=O)NC9=O)cccc87)CC6)C5)C4)nn3)CC2)cc1Cl	C42H47ClN10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-7OAIZ3	WO2023180388A1_AR234	.	CC1CN(c2ccc(C(=O)N[C@H]3CC[C@H](Oc4ccc(C#N)c(Cl)c4)CC3)nn2)CCC1CN1CCC(n2ncc3c(N4CCC(=O)NC4=O)cccc32)CC1	C41H47ClN10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-BETY0Y	SCHEMBL26368352	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[(1R,5S)-6-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indazol-1-yl]piperidin-1-yl]methyl]-3-azabicyclo[3.1.0]hexan-3-yl]pyridazine-3-carboxamide	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4C[C@@H]5[C@H](CN6CCC(n7ncc8c(N9CCC(=O)NC9=O)cccc87)CC6)[C@@H]5C4)nn3)CC2)cc1Cl	C40H43ClN10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-NYLH6Z	WO2023180388A1_AR236	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CC5(CCC5CN5CCC(n6ncc7c(N8CCC(=O)NC8=O)cccc76)CC5)C4)nn3)CC2)cc1Cl	C41H45ClN10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-ZZMZEV	SCHEMBL26368415	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[2-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indazol-1-yl]piperidin-1-yl]methyl]-7-azaspiro[3.5]nonan-7-yl]pyridazine-3-carboxamide	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC5(CC4)CC(CN4CCC(n6ncc7c(N8CCC(=O)NC8=O)cccc76)CC4)C5)nn3)CC2)cc1Cl	C43H49ClN10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-Q8DMB0	WO2023180388A1_AR238	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CC[C@H](CN5CCC(n6ncc7c(N8CCC(=O)NC8=O)cccc76)CC5)C4)nn3)CC2)cc1Cl	C39H43ClN10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-9NIV9W	SCHEMBL26368463	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[(3S)-3-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indazol-1-yl]piperidin-1-yl]methyl]pyrrolidin-1-yl]pyridazine-3-carboxamide	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CC[C@@H](CN5CCC(n6ncc7c(N8CCC(=O)NC8=O)cccc76)CC5)C4)nn3)CC2)cc1Cl	C39H43ClN10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-VMYNYC	SCHEMBL26121836	N-[4-[4-cyano-3-(trifluoromethyl)phenoxy]cyclohexyl]-6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26121846; SCHEMBL30588643	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC(n6ccc7c(N8CCC(=O)NC8=O)cccc76)CC5)CC4)nn3)CC2)cc1C(F)(F)F	C42H46F3N9O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-6N003O	SCHEMBL26368464	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[3-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indazol-1-yl]piperidin-1-yl]methyl]-3-methylazetidin-1-yl]pyridazine-3-carboxamide	CC1(CN2CCC(n3ncc4c(N5CCC(=O)NC5=O)cccc43)CC2)CN(c2ccc(C(=O)N[C@H]3CC[C@H](Oc4ccc(C#N)c(Cl)c4)CC3)nn2)C1	C39H43ClN10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-YKL4QF	SCHEMBL26368535	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[3-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indazol-1-yl]piperidin-1-yl]methyl]-3-methylpyrrolidin-1-yl]pyridazine-3-carboxamide	CC1(CN2CCC(n3ncc4c(N5CCC(=O)NC5=O)cccc43)CC2)CCN(c2ccc(C(=O)N[C@H]3CC[C@H](Oc4ccc(C#N)c(Cl)c4)CC3)nn2)C1	C40H45ClN10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-MSH3YZ	SCHEMBL26116422	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indazol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26116432; SCHEMBL30588303	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC(n6ncc7c(N8CCC(=O)NC8=O)cccc76)CC5)CC4)nn3)CC2)cc1Cl	C40H45ClN10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-O18NKN	SCHEMBL26368626	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[2-[2-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indazol-1-yl]piperidin-1-yl]ethyl]morpholin-4-yl]pyridazine-3-carboxamide	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCOC(CCN5CCC(n6ncc7c(N8CCC(=O)NC8=O)cccc76)CC5)C4)nn3)CC2)cc1Cl	C40H45ClN10O5	AR	P10275	CRBN	WO-2023180388-A1
TPD-FFEFZP	WO2023180388A1_AR244	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4C[C@]5(CN6CCC(n7ncc8c(N9CCC(=O)NC9=O)cccc87)CC6)C[C@]5(C(F)(F)F)C4)nn3)CC2)cc1Cl	C41H42ClF3N10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-NTCS5K	SCHEMBL26116244	(2S,5R)-4-(3-chloro-4-cyanophenyl)-N-[6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)pyrazolo[3,4-c]pyridin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridin-3-yl]-2,5-dimethylpiperazine-1-carboxamide; SCHEMBL30588629	C[C@@H]1CN(C(=O)Nc2ccc(N3CCC(CN4CCC(n5ncc6c(N7CCC(=O)NC7=O)cncc65)CC4)CC3)nc2)[C@@H](C)CN1c1ccc(C#N)c(Cl)c1	C40H47ClN12O3	AR	P10275	CRBN	WO-2023180388-A1
TPD-XW5RHT	SCHEMBL26118727	N-[3-(8-cyanoquinolin-5-yl)oxy-2,2,4,4-tetramethylcyclobutyl]-6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indazol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26118744; SCHEMBL30588242	CC1(C)[C@H](NC(=O)c2ccc(N3CCC(CN4CCC(n5ncc6c(N7CCC(=O)NC7=O)cccc65)CC4)CC3)nn2)C(C)(C)[C@H]1Oc1ccc(C#N)c2ncccc12	C45H51N11O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-0X2LYB	SCHEMBL26118937	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)pyrrolo[2,3-d]pyrimidin-7-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26118945; SCHEMBL30588351	CC1(C)[C@H](NC(=O)c2ccc(N3CCC(CN4CCC(n5ccc6c(N7CCC(=O)NC7=O)ncnc65)CC4)CC3)nn2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C41H48ClN11O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-VG00G2	SCHEMBL26119425	N-[3-(5-chloro-6-cyanopyridin-3-yl)oxy-2,2,4,4-tetramethylcyclobutyl]-6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indazol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26119438; SCHEMBL30588358	CC1(C)[C@H](NC(=O)c2ccc(N3CCC(CN4CCC(n5ncc6c(N7CCC(=O)NC7=O)cccc65)CC4)CC3)nn2)C(C)(C)[C@H]1Oc1cnc(C#N)c(Cl)c1	C41H48ClN11O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-P2LK80	SCHEMBL26114479	N-[3-(8-cyanoquinolin-5-yl)oxy-2,2,4,4-tetramethylcyclobutyl]-6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)pyrrolo[3,2-c]pyridin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26114491; SCHEMBL30588383	CC1(C)[C@H](NC(=O)c2ccc(N3CCC(CN4CCC(n5ccc6c(N7CCC(=O)NC7=O)nccc65)CC4)CC3)nn2)C(C)(C)[C@H]1Oc1ccc(C#N)c2ncccc12	C45H51N11O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-T6NRB3	SCHEMBL26118855	N-[3-(5-chloro-6-cyanopyridin-3-yl)oxy-2,2,4,4-tetramethylcyclobutyl]-2-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyrimidine-5-carboxamide; SCHEMBL26118865; SCHEMBL30588457	CC1(C)[C@H](NC(=O)c2cnc(N3CCC(CN4CCC(n5ccc6c(N7CCC(=O)NC7=O)cccc65)CC4)CC3)nc2)C(C)(C)[C@H]1Oc1cnc(C#N)c(Cl)c1	C42H49ClN10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-912LCW	SCHEMBL26117657	N-[3-(5-chloro-6-cyanopyridin-3-yl)oxy-2,2,4,4-tetramethylcyclobutyl]-2-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indazol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyrimidine-5-carboxamide; SCHEMBL26117665; SCHEMBL30588267	CC1(C)[C@H](NC(=O)c2cnc(N3CCC(CN4CCC(n5ncc6c(N7CCC(=O)NC7=O)cccc65)CC4)CC3)nc2)C(C)(C)[C@H]1Oc1cnc(C#N)c(Cl)c1	C41H48ClN11O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-3Z23QX	SCHEMBL26116075	N-[3-(5-chloro-6-cyanopyridin-3-yl)oxy-2,2,4,4-tetramethylcyclobutyl]-6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indazol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridine-3-carboxamide; SCHEMBL26116086; SCHEMBL30588503	CC1(C)[C@H](NC(=O)c2ccc(N3CCC(CN4CCC(n5ncc6c(N7CCC(=O)NC7=O)cccc65)CC4)CC3)nc2)C(C)(C)[C@H]1Oc1cnc(C#N)c(Cl)c1	C42H49ClN10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-O7ZW6Q	SCHEMBL26368835	N-[3-(5-chloro-6-cyanopyridin-3-yl)oxy-2,2,4,4-tetramethylcyclobutyl]-6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)pyrrolo[2,3-b]pyridin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridine-3-carboxamide; SCHEMBL31637046	CC1(C)[C@H](NC(=O)c2ccc(N3CCC(CN4CCC(n5ccc6c(N7CCC(=O)NC7=O)ccnc65)CC4)CC3)nc2)C(C)(C)[C@H]1Oc1cnc(C#N)c(Cl)c1	C42H49ClN10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-DTKCB0	SCHEMBL26368837	N-[3-(5-chloro-6-cyanopyridin-3-yl)oxy-2,2,4,4-tetramethylcyclobutyl]-6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)pyrazolo[3,4-b]pyridin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridine-3-carboxamide; SCHEMBL31637058	CC1(C)[C@H](NC(=O)c2ccc(N3CCC(CN4CCC(n5ncc6c(N7CCC(=O)NC7=O)ccnc65)CC4)CC3)nc2)C(C)(C)[C@H]1Oc1cnc(C#N)c(Cl)c1	C41H48ClN11O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-NILMRM	SCHEMBL26368879	N-[3-(5-chloro-6-cyanopyridin-3-yl)oxy-2,2,4,4-tetramethylcyclobutyl]-6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)pyrazolo[4,3-c]pyridin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridine-3-carboxamide; SCHEMBL31637020	CC1(C)[C@H](NC(=O)c2ccc(N3CCC(CN4CCC(n5ncc6c(N7CCC(=O)NC7=O)nccc65)CC4)CC3)nc2)C(C)(C)[C@H]1Oc1cnc(C#N)c(Cl)c1	C41H48ClN11O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-WWQBSC	SCHEMBL26368881	N-[3-(5-chloro-6-cyanopyridin-3-yl)oxy-2,2,4,4-tetramethylcyclobutyl]-6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)pyrrolo[2,3-d]pyrimidin-7-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridine-3-carboxamide; SCHEMBL31637053	CC1(C)[C@H](NC(=O)c2ccc(N3CCC(CN4CCC(n5ccc6c(N7CCC(=O)NC7=O)ncnc65)CC4)CC3)nc2)C(C)(C)[C@H]1Oc1cnc(C#N)c(Cl)c1	C41H48ClN11O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-BU1JT5	SCHEMBL26119512	N-[3-(5-chloro-6-cyanopyridin-3-yl)oxy-2,2,4,4-tetramethylcyclobutyl]-6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)pyrrolo[3,2-c]pyridin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridine-3-carboxamide; SCHEMBL26119522; SCHEMBL30588428	CC1(C)[C@H](NC(=O)c2ccc(N3CCC(CN4CCC(n5ccc6c(N7CCC(=O)NC7=O)nccc65)CC4)CC3)nc2)C(C)(C)[C@H]1Oc1cnc(C#N)c(Cl)c1	C42H49ClN10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-BNQCVI	SCHEMBL26363426	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[[4-[[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]methyl]piperidin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC(Cn6ccc7c(N8CCC(=O)NC8=O)cccc76)CC5)CC4)nn3)CC2)cc1Cl	C42H48ClN9O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-HZBEEB	SCHEMBL26116823	N-[3-(8-cyanoquinolin-5-yl)oxy-2,2,4,4-tetramethylcyclobutyl]-5-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)pyrazolo[3,4-b]pyridin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridine-2-carboxamide; SCHEMBL26116834; SCHEMBL30588324	CC1(C)[C@H](NC(=O)c2ccc(N3CCC(CN4CCC(n5ncc6c(N7CCC(=O)NC7=O)ccnc65)CC4)CC3)cn2)C(C)(C)[C@H]1Oc1ccc(C#N)c2ncccc12	C45H51N11O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-OC3Y0V	SCHEMBL26116350	N-[3-(8-cyanoquinolin-5-yl)oxy-2,2,4,4-tetramethylcyclobutyl]-6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indazol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridine-3-carboxamide; SCHEMBL26116362; SCHEMBL30588214	CC1(C)[C@H](NC(=O)c2ccc(N3CCC(CN4CCC(n5ncc6c(N7CCC(=O)NC7=O)cccc65)CC4)CC3)nc2)C(C)(C)[C@H]1Oc1ccc(C#N)c2ncccc12	C46H52N10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-HJ7ADY	SCHEMBL26113819	N-[3-(8-cyanoquinolin-5-yl)oxy-2,2,4,4-tetramethylcyclobutyl]-6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)pyrrolo[2,3-b]pyridin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26113829; SCHEMBL30588469	CC1(C)[C@H](NC(=O)c2ccc(N3CCC(CN4CCC(n5ccc6c(N7CCC(=O)NC7=O)ccnc65)CC4)CC3)nn2)C(C)(C)[C@H]1Oc1ccc(C#N)c2ncccc12	C45H51N11O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-KJWRYE	SCHEMBL26113534	N-[3-(5-chloro-6-cyanopyridin-3-yl)oxy-2,2,4,4-tetramethylcyclobutyl]-6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)pyrrolo[2,3-b]pyridin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26113545; SCHEMBL30588606	CC1(C)[C@H](NC(=O)c2ccc(N3CCC(CN4CCC(n5ccc6c(N7CCC(=O)NC7=O)ccnc65)CC4)CC3)nn2)C(C)(C)[C@H]1Oc1cnc(C#N)c(Cl)c1	C41H48ClN11O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-Y6T85M	SCHEMBL26114627	N-[3-(8-cyanoquinolin-5-yl)oxy-2,2,4,4-tetramethylcyclobutyl]-6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)pyrrolo[3,2-c]pyridin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridine-3-carboxamide; SCHEMBL26114645; SCHEMBL30588293	CC1(C)[C@H](NC(=O)c2ccc(N3CCC(CN4CCC(n5ccc6c(N7CCC(=O)NC7=O)nccc65)CC4)CC3)nc2)C(C)(C)[C@H]1Oc1ccc(C#N)c2ncccc12	C46H52N10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-PLMEHW	SCHEMBL26113790	N-[3-(8-cyanoquinolin-5-yl)oxy-2,2,4,4-tetramethylcyclobutyl]-6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)pyrazolo[3,4-b]pyridin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridine-3-carboxamide; SCHEMBL26113806; SCHEMBL30588783	CC1(C)[C@H](NC(=O)c2ccc(N3CCC(CN4CCC(n5ncc6c(N7CCC(=O)NC7=O)ccnc65)CC4)CC3)nc2)C(C)(C)[C@H]1Oc1ccc(C#N)c2ncccc12	C45H51N11O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-CTRLTR	SCHEMBL26114527	N-[3-(8-cyanoquinolin-5-yl)oxy-2,2,4,4-tetramethylcyclobutyl]-6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)pyrazolo[4,3-c]pyridin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridine-3-carboxamide; SCHEMBL26114548; SCHEMBL30588321	CC1(C)[C@H](NC(=O)c2ccc(N3CCC(CN4CCC(n5ncc6c(N7CCC(=O)NC7=O)nccc65)CC4)CC3)nc2)C(C)(C)[C@H]1Oc1ccc(C#N)c2ncccc12	C45H51N11O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-AF5CDZ	SCHEMBL26115580	N-[3-(5-chloro-6-cyanopyridin-3-yl)oxy-2,2,4,4-tetramethylcyclobutyl]-5-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indazol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyrimidine-2-carboxamide; SCHEMBL26115587; SCHEMBL30588508	CC1(C)[C@H](NC(=O)c2ncc(N3CCC(CN4CCC(n5ncc6c(N7CCC(=O)NC7=O)cccc65)CC4)CC3)cn2)C(C)(C)[C@H]1Oc1cnc(C#N)c(Cl)c1	C41H48ClN11O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-ZTNFSG	WO2023180388A1_AR269	.	CC1(C)[C@H](NC(=O)c2ccc(N3CCC(CN4CCC(n5ccc6c(N7CCC(=O)NC7=O)ccnc65)CC4)CC3)cn2)C(C)(C)[C@H]1Oc1cnc(C#N)c(Cl)c1	C42H49ClN10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-BN17J9	SCHEMBL26363456	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[4-[[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]methyl]piperidin-1-yl]piperidin-1-yl]pyridazine-3-carboxamide	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(N5CCC(Cn6ccc7c(N8CCC(=O)NC8=O)cccc76)CC5)CC4)nn3)CC2)cc1Cl	C41H46ClN9O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-L3J9PG	WO2023180388A1_AR270	.	CC1(C)[C@H](NCc2ncc(N3CCC(CN4CCC(n5ncc6c(N7CCC(=O)NC7=O)cccc65)CC4)CC3)cn2)C(C)(C)[C@H]1Oc1cnc(C#N)c(C(F)(F)F)c1	C42H50F3N11O3	AR	P10275	CRBN	WO-2023180388-A1
TPD-SLJTK2	WO2023180388A1_AR271	.	CC(F)(F)C1=C(C#N)NCC(O[C@H]2C(C)(C)[C@H](NC(=O)c3ncc(N4CCC(CN5CCC(n6ccc7c(N8CCC(=O)NC8=O)ccnc76)CC5)CC4)cn3)C2(C)C)=C1	C43H53F2N11O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-VT17OD	SCHEMBL26117240	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-5-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)pyrazolo[3,4-b]pyridin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyrimidine-2-carboxamide; SCHEMBL26117254; SCHEMBL30588365	CC1(C)[C@H](NC(=O)c2ncc(N3CCC(CN4CCC(n5ncc6c(N7CCC(=O)NC7=O)ccnc65)CC4)CC3)cn2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C41H48ClN11O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-5G3DFU	SCHEMBL26120702	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-5-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)pyrazolo[4,3-c]pyridin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyrimidine-2-carboxamide; SCHEMBL26120714; SCHEMBL30588447	CC1(C)[C@H](NC(=O)c2ncc(N3CCC(CN4CCC(n5ncc6c(N7CCC(=O)NC7=O)nccc65)CC4)CC3)cn2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C41H48ClN11O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-47LYLV	SCHEMBL26118730	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-4-[3-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]piperidin-1-yl]benzamide; SCHEMBL30588668	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCCC(N5CCC(n6ccc7c(N8CCC(=O)NC8=O)cccc76)CC5)C4)cc3)CC2)cc1Cl	C42H46ClN7O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-2GG9FE	WO2023180388A1_AR29	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridine-3-carboxamide	CC1(C)[C@H](NC(=O)c2ccc(N3CCC(CN4CCC(n5ccc6c(N7CCC(=O)NC7=O)cccc65)CC4)CC3)nc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C44H51ClN8O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-Q8D3H0	SCHEMBL26362116	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-3-[1-[2-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]acetyl]piperidin-4-yl]benzamide	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cccc(C4CCN(C(=O)CN5CCC(n6ccc7c(N8CCC(=O)NC8=O)cccc76)CC5)CC4)c3)CC2)cc1Cl	C44H48ClN7O5	AR	P10275	CRBN	WO-2023180388-A1
TPD-A2Y3TV	WO2023180388A1_AR30	.	CC1(F)CN(CC2CCN(c3ccc(C(=O)N[C@H]4CC[C@H](Oc5ccc(C#N)c(Cl)c5)CC4)nn3)CC2)CCC1n1ccc2c(N3CCC(=O)NC3=O)cccc21	C42H47ClFN9O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-M7HUR1	SCHEMBL26363530	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)-6-fluoroindol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC(n6ccc7c(N8CCC(=O)NC8=O)cc(F)cc76)CC5)CC4)nn3)CC2)cc1Cl	C41H45ClFN9O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-AOIT7K	SCHEMBL26118619	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[[4-[6-chloro-4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26118636; SCHEMBL30588424	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC(n6ccc7c(N8CCC(=O)NC8=O)cc(Cl)cc76)CC5)CC4)nn3)CC2)cc1Cl	C41H45Cl2N9O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-B7FR33	SCHEMBL26116486	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)-6-fluoroindazol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26116495; SCHEMBL30588751	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC(n6ncc7c(N8CCC(=O)NC8=O)cc(F)cc76)CC5)CC4)nn3)CC2)cc1Cl	C40H44ClFN10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-6LU6NQ	WO2023180388A1_AR34	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[[4-[6-chloro-4-(2,4-dioxo-1,3-diazinan-1-yl)indazol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide	N#Cc1ccc(O[C@H]2CC[C@@H](NC(=O)c3ccc(N4CCC(CN5CCC(n6ncc7c(N8CCC(=O)NC8=O)cc(Cl)cc76)CC5)CC4)nn3)CC2)cc1Cl	C40H44Cl2N10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-YNWWPZ	SCHEMBL26114741	1-[1-[[1-[6-[[4-(3-chloro-4-cyanophenoxy)cyclohexyl]carbamoyl]pyridazin-3-yl]piperidin-4-yl]methyl]piperidin-4-yl]-4-(2,4-dioxo-1,3-diazinan-1-yl)-N,N-dimethylindole-6-carboxamide; SCHEMBL26114752; SCHEMBL30588368	CN(C)C(=O)c1cc(N2CCC(=O)NC2=O)c2ccn(C3CCN(CC4CCN(c5ccc(C(=O)N[C@H]6CC[C@H](Oc7ccc(C#N)c(Cl)c7)CC6)nn5)CC4)CC3)c2c1	C44H51ClN10O5	AR	P10275	CRBN	WO-2023180388-A1
TPD-XIXAD0	WO2023180388A1_AR36	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCCC(CN5CCC(n6ncc7c(N8CCC(=O)NC8=O)cccc76)CC5)C4)nc3)CC2)cc1Cl	C41H46ClN9O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-4KI5R3	SCHEMBL26363743	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-5-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indazol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyrazine-2-carboxamide	CC1(C)[C@H](NC(=O)c2cnc(N3CCC(CN4CCC(n5ncc6c(N7CCC(=O)NC7=O)cccc65)CC4)CC3)cn2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C42H49ClN10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-D9XQH4	WO2023180388A1_AR38	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(C4CCC(CN5CCC(n6ncc7c(N8CCC(=O)NC8=O)cccc76)CC5)CC4)cn3)CC2)cc1C(F)(F)F	C42H46F3N9O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-I3WQJA	WO2023180388A1_AR39	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCC(CN5CCC(n6ncc7c(N8CCC(=O)NC8=O)cccc76)CC5)CC4)cn3)CC2)cc1CI	C41H47IN10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-UTXK1Y	WO2023180388A1_AR4	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc4c(c3)CN(C(=O)CN3CCC(n5ccc6c(N7CCC(=O)NC7=O)cccc65)CC3)CC4)CC2)cc1Cl	C42H44ClN7O5	AR	P10275	CRBN	WO-2023180388-A1
TPD-OGV15B	SCHEMBL26363818	N-[4-[4-cyano-3-(trifluoromethyl)phenoxy]cyclohexyl]-6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indazol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridine-3-carboxamide	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC(n6ncc7c(N8CCC(=O)NC8=O)cccc76)CC5)CC4)nc3)CC2)cc1C(F)(F)F	C42H46F3N9O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-CM69GY	WO2023180388A1_AR41	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indazol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridine-3-carboxamide	CC1(C)[C@H](NC(=O)c2ccc(N3CCC(CN4CCC(n5ncc6c(N7CCC(=O)NC7=O)cccc65)CC4)CC3)nc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C43H50ClN9O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-VAOD9L	SCHEMBL26363822	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indazol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridine-3-carboxamide	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC(n6ncc7c(N8CCC(=O)NC8=O)cccc76)CC5)CC4)nc3)CC2)cc1Cl	C41H46ClN9O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-SGR7LN	SCHEMBL26115599	N-[4-[4-cyano-3-(trifluoromethyl)phenoxy]cyclohexyl]-6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indazol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26115612; SCHEMBL30588632	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC(n6ncc7c(N8CCC(=O)NC8=O)cccc76)CC5)CC4)nn3)CC2)cc1C(F)(F)F	C41H45F3N10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-IRG8KK	SCHEMBL26116347	N-[4-[4-cyano-3-(trifluoromethyl)phenoxy]cyclohexyl]-6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)pyrrolo[2,3-c]pyridin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26116360; SCHEMBL30588388	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC(n6ccc7c(N8CCC(=O)NC8=O)cncc76)CC5)CC4)nn3)CC2)cc1C(F)(F)F	C41H45F3N10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-GUNXYD	SCHEMBL26116076	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)pyrrolo[2,3-c]pyridin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26116087; SCHEMBL30588480	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC(n6ccc7c(N8CCC(=O)NC8=O)cncc76)CC5)CC4)nn3)CC2)cc1Cl	C40H45ClN10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-8FJTWF	SCHEMBL26119796	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)pyrrolo[2,3-c]pyridin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridine-3-carboxamide; SCHEMBL26119809; SCHEMBL30588313	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC(n6ccc7c(N8CCC(=O)NC8=O)cncc76)CC5)CC4)nc3)CC2)cc1Cl	C41H46ClN9O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-2HFRA8	SCHEMBL26362122	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-2-[2-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]acetyl]-3,4-dihydro-1H-isoquinoline-6-carboxamide	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc4c(c3)CCN(C(=O)CN3CCC(n5ccc6c(N7CCC(=O)NC7=O)cccc65)CC3)C4)CC2)cc1Cl	C42H44ClN7O5	AR	P10275	CRBN	WO-2023180388-A1
TPD-6QU6MZ	SCHEMBL26114880	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)pyrazolo[4,3-c]pyridin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26114890; SCHEMBL30588497	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC(n6ncc7c(N8CCC(=O)NC8=O)nccc76)CC5)CC4)nn3)CC2)cc1Cl	C39H44ClN11O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-X4SQR7	SCHEMBL26364102	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)pyrazolo[3,4-c]pyridin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL30588268	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC(n6ncc7c(N8CCC(=O)NC8=O)cncc76)CC5)CC4)nn3)CC2)cc1Cl	C39H44ClN11O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-MXYPQH	SCHEMBL26115695	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-4-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]benzamide; SCHEMBL26115698; SCHEMBL30588717	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(n5ccc6c(N7CCC(=O)NC7=O)cccc65)CC4)cc3)CC2)cc1Cl	C37H37ClN6O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-IA7BH4	SCHEMBL26119942	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26119954; SCHEMBL30588501	CC1(C)[C@H](NC(=O)c2ccc(N3CCC(CN4CCC(n5ccc6c(N7CCC(=O)NC7=O)cccc65)CC4)CC3)nn2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C43H50ClN9O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-WCSVZ8	SCHEMBL26114040	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)pyrrolo[2,3-c]pyridin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26114048; SCHEMBL30588601	CC1(C)[C@H](NC(=O)c2ccc(N3CCC(CN4CCC(n5ccc6c(N7CCC(=O)NC7=O)cncc65)CC4)CC3)nn2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C42H49ClN10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-XG5QQO	SCHEMBL26117352	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[2-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]ethyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26117360; SCHEMBL30588467	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CCN5CCC(n6ccc7c(N8CCC(=O)NC8=O)cccc76)CC5)CC4)nn3)CC2)cc1Cl	C42H48ClN9O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-XTRA26	SCHEMBL26364234	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[2-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)-1-propan-2-ylindole-6-carbonyl]piperazin-1-yl]ethyl]piperidin-1-yl]pyridazine-3-carboxamide	CC(C)n1ccc2c(N3CCC(=O)NC3=O)cc(C(=O)N3CCN(CCC4CCN(c5ccc(C(=O)N[C@H]6CC[C@H](Oc7ccc(C#N)c(Cl)c7)CC6)nn5)CC4)CC3)cc21	C45H53ClN10O5	AR	P10275	CRBN	WO-2023180388-A1
TPD-ET81WY	WO2023180388A1_AR59	.	CC(C)n1ccc2c(N3CCC(=O)NC3=O)cc(C(=O)N3CCN(CCCOc4ccc(C(=O)N[C@H]5CC[C@H](Oc6ccc(C#N)c(Cl)c6)CC5)nc4)CC3)cc21	C42H47ClN8O6	AR	P10275	CRBN	WO-2023180388-A1
TPD-GCT9OF	WO2023180388A1_AR6	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-2-[2-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]acetyl]-1,3-dihydroisoindole-5-carboxamide	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc4c(c3)CN(C(=O)CN3CCC(n5ccc6c(N7CCC(=O)NC7=O)cccc65)CC3)C4)CC2)cc1Cl	C41H42ClN7O5	AR	P10275	CRBN	WO-2023180388-A1
TPD-39PZMU	SCHEMBL26364303	N-[1-[3-[6-[[4-(3-chloro-4-cyanophenoxy)cyclohexyl]carbamoyl]pyridin-3-yl]oxypropyl]piperidin-4-yl]-4-(2,4-dioxo-1,3-diazinan-1-yl)-N-methyl-1-propan-2-ylindole-6-carboxamide	CC(C)n1ccc2c(N3CCC(=O)NC3=O)cc(C(=O)N(C)C3CCN(CCCOc4ccc(C(=O)N[C@H]5CC[C@H](Oc6ccc(C#N)c(Cl)c6)CC5)nc4)CC3)cc21	C44H51ClN8O6	AR	P10275	CRBN	WO-2023180388-A1
TPD-92KLCB	SCHEMBL26364399	N-[[1-[3-[6-[[4-(3-chloro-4-cyanophenoxy)cyclohexyl]carbamoyl]pyridin-3-yl]oxypropyl]piperidin-4-yl]methyl]-4-(2,4-dioxo-1,3-diazinan-1-yl)-N-methyl-1-propan-2-ylindole-6-carboxamide	CC(C)n1ccc2c(N3CCC(=O)NC3=O)cc(C(=O)N(C)CC3CCN(CCCOc4ccc(C(=O)N[C@H]5CC[C@H](Oc6ccc(C#N)c(Cl)c6)CC5)nc4)CC3)cc21	C45H53ClN8O6	AR	P10275	CRBN	WO-2023180388-A1
TPD-W1RO0J	SCHEMBL26364401	N-[4-(4-chloro-3-cyanophenoxy)cyclohexyl]-5-[3-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]propoxy]pyridine-2-carboxamide	N#Cc1cc(O[C@H]2CC[C@H](NC(=O)c3ccc(OCCCN4CCC(n5ccc6c(N7CCC(=O)NC7=O)cccc65)CC4)cn3)CC2)ccc1Cl	C39H42ClN7O5	AR	P10275	CRBN	WO-2023180388-A1
TPD-W64LSX	SCHEMBL26364402	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-5-[4-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)-1-propan-2-ylindole-6-carbonyl]piperazin-1-yl]butoxy]pyridine-2-carboxamide	CC(C)n1ccc2c(N3CCC(=O)NC3=O)cc(C(=O)N3CCN(CCCCOc4ccc(C(=O)N[C@H]5CC[C@H](Oc6ccc(C#N)c(Cl)c6)CC5)nc4)CC3)cc21	C43H49ClN8O6	AR	P10275	CRBN	WO-2023180388-A1
TPD-J0HCK8	SCHEMBL26364502	N-[1-[4-[6-[[4-(3-chloro-4-cyanophenoxy)cyclohexyl]carbamoyl]pyridin-3-yl]oxybutyl]piperidin-4-yl]-4-(2,4-dioxo-1,3-diazinan-1-yl)-N-methyl-1-propan-2-ylindole-6-carboxamide	CC(C)n1ccc2c(N3CCC(=O)NC3=O)cc(C(=O)N(C)C3CCN(CCCCOc4ccc(C(=O)N[C@H]5CC[C@H](Oc6ccc(C#N)c(Cl)c6)CC5)nc4)CC3)cc21	C45H53ClN8O6	AR	P10275	CRBN	WO-2023180388-A1
TPD-OLQJ64	SCHEMBL26364504	N-[[1-[4-[6-[[4-(3-chloro-4-cyanophenoxy)cyclohexyl]carbamoyl]pyridin-3-yl]oxybutyl]piperidin-4-yl]methyl]-4-(2,4-dioxo-1,3-diazinan-1-yl)-N-methyl-1-propan-2-ylindole-6-carboxamide	CC(C)n1ccc2c(N3CCC(=O)NC3=O)cc(C(=O)N(C)CC3CCN(CCCCOc4ccc(C(=O)N[C@H]5CC[C@H](Oc6ccc(C#N)c(Cl)c6)CC5)nc4)CC3)cc21	C46H55ClN8O6	AR	P10275	CRBN	WO-2023180388-A1
TPD-65ZXO5	SCHEMBL26364506	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-5-[4-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]butoxy]pyridine-2-carboxamide	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(OCCCCN4CCC(n5ccc6c(N7CCC(=O)NC7=O)cccc65)CC4)cn3)CC2)cc1Cl	C40H44ClN7O5	AR	P10275	CRBN	WO-2023180388-A1
TPD-F49VTP	SCHEMBL26113649	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-2-[4-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidine-1-carbonyl]piperidin-1-yl]pyrimidine-5-carboxamide; SCHEMBL26113657; SCHEMBL30588545	CC1(C)[C@H](NC(=O)c2cnc(N3CCC(C(=O)N4CCC(n5ccc6c(N7CCC(=O)NC7=O)cccc65)CC4)CC3)nc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C43H48ClN9O5	AR	P10275	CRBN	WO-2023180388-A1
TPD-LJELP8	SCHEMBL26117961	N-[4-[4-cyano-3-(trifluoromethyl)phenoxy]cyclohexyl]-2-[4-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidine-1-carbonyl]piperidin-1-yl]pyrimidine-5-carboxamide; SCHEMBL26117967; SCHEMBL30588235	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCC(C(=O)N5CCC(n6ccc7c(N8CCC(=O)NC8=O)cccc76)CC5)CC4)nc3)CC2)cc1C(F)(F)F	C42H44F3N9O5	AR	P10275	CRBN	WO-2023180388-A1
TPD-HMW2BC	SCHEMBL26118465	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-2-[4-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidine-1-carbonyl]piperidin-1-yl]pyrimidine-5-carboxamide; SCHEMBL26118469; SCHEMBL30588205	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCC(C(=O)N5CCC(n6ccc7c(N8CCC(=O)NC8=O)cccc76)CC5)CC4)nc3)CC2)cc1Cl	C41H44ClN9O5	AR	P10275	CRBN	WO-2023180388-A1
TPD-6SO5C0	SCHEMBL26118993	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL30588201	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(N5CCC(n6ccc7c(N8CCC(=O)NC8=O)cccc76)CC5)CC4)nn3)CC2)cc1Cl	C40H44ClN9O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-YAFMIB	SCHEMBL26113542	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26113543; SCHEMBL30588427	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(n5ccc6c(N7CCC(=O)NC7=O)cccc65)CC4)nn3)CC2)cc1Cl	C35H35ClN8O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-IZXKD3	SCHEMBL26117462	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)pyrrolo[2,3-c]pyridin-1-yl]piperidin-1-yl]methyl]-4-fluoropiperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26117465; SCHEMBL30588372	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(F)(CN5CCC(n6ccc7c(N8CCC(=O)NC8=O)cncc76)CC5)CC4)nn3)CC2)cc1Cl	C40H44ClFN10O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-PSWE6A	SCHEMBL26364618	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[3-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]azetidin-1-yl]pyridazine-3-carboxamide	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CC(CN5CCC(n6ccc7c(N8CCC(=O)NC8=O)cccc76)CC5)C4)nn3)CC2)cc1Cl	C39H42ClN9O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-O56UT7	SCHEMBL26114973	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[3-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26118796; SCHEMBL31637051	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCCC(CN5CCC(n6ccc7c(N8CCC(=O)NC8=O)cccc76)CC5)C4)nn3)CC2)cc1Cl	C41H46ClN9O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-O7YFSX	SCHEMBL26114745	N-[3-[4-cyano-3-(trifluoromethyl)phenoxy]-2,2,4,4-tetramethylcyclobutyl]-4-[6-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]hexyl]benzamide; SCHEMBL26114757; SCHEMBL30588223	CC1(C)[C@H](NC(=O)c2ccc(CCCCCCN3CCC(n4ccc5c(N6CCC(=O)NC6=O)cccc54)CC3)cc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(C(F)(F)F)c1	C46H53F3N6O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-ADE2RW	SCHEMBL26119759	N-[2-[2-[4-[6-[[4-(3-chloro-4-cyanophenoxy)cyclohexyl]carbamoyl]pyridazin-3-yl]piperazin-1-yl]ethoxy]ethyl]-4-(2,4-dioxo-1,3-diazinan-1-yl)-1-propan-2-ylindole-6-carboxamide; SCHEMBL26119761; SCHEMBL30588401	CC(C)n1ccc2c(N3CCC(=O)NC3=O)cc(C(=O)NCCOCCN3CCN(c4ccc(C(=O)N[C@H]5CC[C@H](Oc6ccc(C#N)c(Cl)c6)CC5)nn4)CC3)cc21	C42H49ClN10O6	AR	P10275	CRBN	WO-2023180388-A1
TPD-JLP0AI	SCHEMBL26115872	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)-1-propan-2-ylindole-6-carbonyl]piperazin-1-yl]pyridazine-3-carboxamide; SCHEMBL26115877; SCHEMBL30588191	CC(C)n1ccc2c(N3CCC(=O)NC3=O)cc(C(=O)N3CCN(c4ccc(C(=O)N[C@H]5CC[C@H](Oc6ccc(C#N)c(Cl)c6)CC5)nn4)CC3)cc21	C38H40ClN9O5	AR	P10275	CRBN	WO-2023180388-A1
TPD-KZYSWF	SCHEMBL26119186	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)-1-propan-2-ylindole-6-carbonyl]piperazin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26119190; SCHEMBL30588380	CC(C)n1ccc2c(N3CCC(=O)NC3=O)cc(C(=O)N3CCN(CC4CCN(c5ccc(C(=O)N[C@H]6C(C)(C)[C@H](Oc7ccc(C#N)c(Cl)c7)C6(C)C)nn5)CC4)CC3)cc21	C46H55ClN10O5	AR	P10275	CRBN	WO-2023180388-A1
TPD-OOSUZ3	SCHEMBL26118174	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)-1-propan-2-ylindole-6-carbonyl]piperazin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide; SCHEMBL26118177; SCHEMBL30588566	CC(C)n1ccc2c(N3CCC(=O)NC3=O)cc(C(=O)N3CCN(CC4CCN(c5ccc(C(=O)N[C@H]6CC[C@H](Oc7ccc(C#N)c(Cl)c7)CC6)nn5)CC4)CC3)cc21	C44H51ClN10O5	AR	P10275	CRBN	WO-2023180388-A1
TPD-2Q8V2Z	SCHEMBL26362420	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-5-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyrazine-2-carboxamide	CC1(C)[C@H](NC(=O)c2cnc(N3CCC(CN4CCC(n5ccc6c(N7CCC(=O)NC7=O)cccc65)CC4)CC3)cn2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C43H50ClN9O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-2I7YTG	SCHEMBL26115067	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)-1-propan-2-ylindole-6-carbonyl]piperazin-1-yl]methyl]piperidin-1-yl]pyridine-3-carboxamide; SCHEMBL26115071; SCHEMBL30588230	CC(C)n1ccc2c(N3CCC(=O)NC3=O)cc(C(=O)N3CCN(CC4CCN(c5ccc(C(=O)N[C@H]6CC[C@H](Oc7ccc(C#N)c(Cl)c7)CC6)cn5)CC4)CC3)cc21	C45H52ClN9O5	AR	P10275	CRBN	WO-2023180388-A1
TPD-DCOKNP	SCHEMBL26114442	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-4-[[9-[4-(2,4-dioxo-1,3-diazinan-1-yl)-1-propan-2-ylindole-6-carbonyl]-2,9-diazaspiro[5.5]undecan-2-yl]methyl]benzamide; SCHEMBL26114446; SCHEMBL30588688	CC(C)n1ccc2c(N3CCC(=O)NC3=O)cc(C(=O)N3CCC4(CCCN(Cc5ccc(C(=O)N[C@H]6CC[C@H](Oc7ccc(C#N)c(Cl)c7)CC6)cc5)C4)CC3)cc21	C46H52ClN7O5	AR	P10275	CRBN	WO-2023180388-A1
TPD-1HX483	SCHEMBL26115295	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-4-[3-[9-[4-(2,4-dioxo-1,3-diazinan-1-yl)-1-propan-2-ylindole-6-carbonyl]-2,9-diazaspiro[5.5]undecan-2-yl]propyl]benzamide; SCHEMBL26115305; SCHEMBL30588425	CC(C)n1ccc2c(N3CCC(=O)NC3=O)cc(C(=O)N3CCC4(CCCN(CCCc5ccc(C(=O)N[C@H]6CC[C@H](Oc7ccc(C#N)c(Cl)c7)CC6)cc5)C4)CC3)cc21	C48H56ClN7O5	AR	P10275	CRBN	WO-2023180388-A1
TPD-RTGA3H	SCHEMBL26114363	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-4-[5-[9-[4-(2,4-dioxo-1,3-diazinan-1-yl)-1-propan-2-ylindole-6-carbonyl]-2,9-diazaspiro[5.5]undecan-2-yl]pentyl]benzamide; SCHEMBL26114373; SCHEMBL30588311	CC(C)n1ccc2c(N3CCC(=O)NC3=O)cc(C(=O)N3CCC4(CCCN(CCCCCc5ccc(C(=O)N[C@H]6CC[C@H](Oc7ccc(C#N)c(Cl)c7)CC6)cc5)C4)CC3)cc21	C50H60ClN7O5	AR	P10275	CRBN	WO-2023180388-A1
TPD-RK44IX	SCHEMBL26116615	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-4-[[3-[4-(2,4-dioxo-1,3-diazinan-1-yl)-1-propan-2-ylindole-6-carbonyl]-3,9-diazaspiro[5.5]undecan-9-yl]methyl]benzamide; SCHEMBL26116620; SCHEMBL30588260	CC(C)n1ccc2c(N3CCC(=O)NC3=O)cc(C(=O)N3CCC4(CCN(Cc5ccc(C(=O)N[C@H]6CC[C@H](Oc7ccc(C#N)c(Cl)c7)CC6)cc5)CC4)CC3)cc21	C46H52ClN7O5	AR	P10275	CRBN	WO-2023180388-A1
TPD-C6OEVB	SCHEMBL26118028	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-4-[3-[3-[4-(2,4-dioxo-1,3-diazinan-1-yl)-1-propan-2-ylindole-6-carbonyl]-3,9-diazaspiro[5.5]undecan-9-yl]propyl]benzamide; SCHEMBL26118042; SCHEMBL30588192	CC(C)n1ccc2c(N3CCC(=O)NC3=O)cc(C(=O)N3CCC4(CCN(CCCc5ccc(C(=O)N[C@H]6CC[C@H](Oc7ccc(C#N)c(Cl)c7)CC6)cc5)CC4)CC3)cc21	C48H56ClN7O5	AR	P10275	CRBN	WO-2023180388-A1
TPD-QVI0VZ	SCHEMBL26118939	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-4-[6-[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)-1-propan-2-ylindole-6-carbonyl]-1,8-diazaspiro[4.5]decan-8-yl]hexyl]benzamide; SCHEMBL26118953; SCHEMBL30588474	CC(C)n1ccc2c(N3CCC(=O)NC3=O)cc(C(=O)N3CCCC34CCN(CCCCCCc3ccc(C(=O)N[C@H]5CC[C@H](Oc6ccc(C#N)c(Cl)c6)CC5)cc3)CC4)cc21	C50H60ClN7O5	AR	P10275	CRBN	WO-2023180388-A1
TPD-TOGDHU	SCHEMBL26111807	N-[3-[4-cyano-3-(trifluoromethyl)phenoxy]-2,2,4,4-tetramethylcyclobutyl]-4-[6-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)-1-propan-2-ylindole-6-carbonyl]piperazin-1-yl]hexyl]benzamide; SCHEMBL26111808; SCHEMBL30588476	CC(C)n1ccc2c(N3CCC(=O)NC3=O)cc(C(=O)N3CCN(CCCCCCc4ccc(C(=O)N[C@H]5C(C)(C)[C@H](Oc6ccc(C#N)c(C(F)(F)F)c6)C5(C)C)cc4)CC3)cc21	C49H58F3N7O5	AR	P10275	CRBN	WO-2023180388-A1
TPD-B5NSS1	SCHEMBL26364845	N-[[1-[1-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]piperidin-4-yl]piperidin-4-yl]methyl]-4-(2,4-dioxo-1,3-diazinan-1-yl)-N-methyl-1-propan-2-ylindole-6-carboxamide	CC(C)n1ccc2c(N3CCC(=O)NC3=O)cc(C(=O)N(C)CC3CCN(C4CCN(c5ccc(N6C(=S)N(c7ccc(C#N)c(C(F)(F)F)c7)C(=O)C6(C)C)cc5)CC4)CC3)cc21	C47H52F3N9O4S	AR	P10275	CRBN	WO-2023180388-A1
TPD-R5HOOU	SCHEMBL26118147	N-[[1-[[1-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]piperidin-4-yl]methyl]piperidin-4-yl]methyl]-4-(2,4-dioxo-1,3-diazinan-1-yl)-N-methyl-1-propan-2-ylindole-6-carboxamide	CC(C)n1ccc2c(N3CCC(=O)NC3=O)cc(C(=O)N(C)CC3CCN(CC4CCN(c5ccc(N6C(=S)N(c7ccc(C#N)c(C(F)(F)F)c7)C(=O)C6(C)C)cc5)CC4)CC3)cc21	C48H54F3N9O4S	AR	P10275	CRBN	WO-2023180388-A1
TPD-S08V7F	SCHEMBL26362428	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-5-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyrazine-2-carboxamide	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCC(CN5CCC(n6ccc7c(N8CCC(=O)NC8=O)cccc76)CC5)CC4)cn3)CC2)cc1Cl	C41H46ClN9O4	AR	P10275	CRBN	WO-2023180388-A1
TPD-ZO78NQ	SCHEMBL26364864	N-[1-[[1-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]piperidin-4-yl]methyl]piperidin-4-yl]-4-(2,4-dioxo-1,3-diazinan-1-yl)-N-methyl-1-propan-2-ylindole-6-carboxamide	CC(C)n1ccc2c(N3CCC(=O)NC3=O)cc(C(=O)N(C)C3CCN(CC4CCN(c5ccc(N6C(=S)N(c7ccc(C#N)c(C(F)(F)F)c7)C(=O)C6(C)C)cc5)CC4)CC3)cc21	C47H52F3N9O4S	AR	P10275	CRBN	WO-2023180388-A1
TPD-5KA18R	SCHEMBL26116405	N-[[1-[2-[1-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenyl]piperidin-4-yl]ethyl]piperidin-4-yl]methyl]-4-(2,4-dioxo-1,3-diazinan-1-yl)-N-methyl-1-propan-2-ylindole-6-carboxamide	CC(C)n1ccc2c(N3CCC(=O)NC3=O)cc(C(=O)N(C)CC3CCN(CCC4CCN(c5ccc(N6C(=S)N(c7ccc(C#N)c(C(F)(F)F)c7)C(=O)C6(C)C)cc5)CC4)CC3)cc21	C49H56F3N9O4S	AR	P10275	CRBN	WO-2023180388-A1
TPD-1J6PCM	SCHEMBL26119295	4-[3-[4-[4-[4-[4-(2,4-Dioxo-1,3-diazinan-1-yl)-1-propan-2-ylindole-6-carbonyl]piperazin-1-yl]butoxy]phenyl]-4,4-dimethyl-5-oxo-2-sulfanylideneimidazolidin-1-yl]-2-(trifluoromethyl)benzonitrile	CC(C)n1ccc2c(N3CCC(=O)NC3=O)cc(C(=O)N3CCN(CCCCOc4ccc(N5C(=S)N(c6ccc(C#N)c(C(F)(F)F)c6)C(=O)C5(C)C)cc4)CC3)cc21	C43H45F3N8O5S	AR	P10275	CRBN	WO-2023180388-A1
TPD-5YP498	SCHEMBL26364904	N-[[1-[3-[4-[3-[4-cyano-3-(trifluoromethyl)phenyl]-5,5-dimethyl-4-oxo-2-sulfanylideneimidazolidin-1-yl]phenoxy]propyl]piperidin-4-yl]methyl]-4-(2,4-dioxo-1,3-diazinan-1-yl)-N-methyl-1-propan-2-ylindole-6-carboxamide	CC(C)n1ccc2c(N3CCC(=O)NC3=O)cc(C(=O)N(C)CC3CCN(CCCOc4ccc(N5C(=S)N(c6ccc(C#N)c(C(F)(F)F)c6)C(=O)C5(C)C)cc4)CC3)cc21	C45H49F3N8O5S	AR	P10275	CRBN	WO-2023180388-A1
TPD-KAA8BI	SCHEMBL26364927	4-[3-[4-[3-[4-[4-(2,4-Dioxo-1,3-diazinan-1-yl)-1-propan-2-ylindole-6-carbonyl]piperazin-1-yl]propoxy]phenyl]-4,4-dimethyl-5-oxo-2-sulfanylideneimidazolidin-1-yl]-2-(trifluoromethyl)benzonitrile	CC(C)n1ccc2c(N3CCC(=O)NC3=O)cc(C(=O)N3CCN(CCCOc4ccc(N5C(=S)N(c6ccc(C#N)c(C(F)(F)F)c6)C(=O)C5(C)C)cc4)CC3)cc21	C42H43F3N8O5S	AR	P10275	CRBN	WO-2023180388-A1
TPD-VNW6T7	SCHEMBL26116372	4-[3-[4-[4-[[4-[4-(2,4-Dioxo-1,3-diazinan-1-yl)indazol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-4,4-dimethyl-5-oxo-2-sulfanylideneimidazolidin-1-yl]-2-(trifluoromethyl)benzonitrile; SCHEMBL30588748	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=S)N1c1ccc(N2CCC(CN3CCC(n4ncc5c(N6CCC(=O)NC6=O)cccc54)CC3)CC2)cc1	C41H42F3N9O3S	AR	P10275	CRBN	WO-2023180388-A1
TPD-SWM7SZ	SCHEMBL26364960	4-[3-[4-[4-[4-[4-(2,4-Dioxo-1,3-diazinan-1-yl)pyrrolo[2,3-c]pyridin-1-yl]piperidin-1-yl]piperidin-1-yl]phenyl]-4,4-dimethyl-5-oxo-2-sulfanylideneimidazolidin-1-yl]-2-(trifluoromethyl)benzonitrile	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=S)N1c1ccc(N2CCC(N3CCC(n4ccc5c(N6CCC(=O)NC6=O)cncc54)CC3)CC2)cc1	C40H40F3N9O3S	AR	P10275	CRBN	WO-2023180388-A1
TPD-1WNZXF	SCHEMBL26364982	4-[3-[4-[4-[2-[4-[4-(2,4-Dioxo-1,3-diazinan-1-yl)pyrazolo[3,4-c]pyridin-1-yl]piperidin-1-yl]ethyl]piperidin-1-yl]phenyl]-4,4-dimethyl-5-oxo-2-sulfanylideneimidazolidin-1-yl]-2-(trifluoromethyl)benzonitrile	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=S)N1c1ccc(N2CCC(CCN3CCC(n4ncc5c(N6CCC(=O)NC6=O)cncc54)CC3)CC2)cc1	C41H43F3N10O3S	AR	P10275	CRBN	WO-2023180388-A1
TPD-TZNIL8	SCHEMBL26119417	4-[3-[4-[4-[[4-[4-(2,4-Dioxo-1,3-diazinan-1-yl)pyrazolo[3,4-c]pyridin-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-4,4-dimethyl-5-oxo-2-sulfanylideneimidazolidin-1-yl]-2-(trifluoromethyl)benzonitrile; SCHEMBL30588375	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=S)N1c1ccc(N2CCC(CN3CCC(n4ncc5c(N6CCC(=O)NC6=O)cncc54)CC3)CC2)cc1	C40H41F3N10O3S	AR	P10275	CRBN	WO-2023180388-A1
TPD-Y6RZPX	SCHEMBL26365037	4-[3-[4-[4-[[4-[4-(2,4-Dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-4,4-dimethyl-5-oxo-2-sulfanylideneimidazolidin-1-yl]-2-(trifluoromethyl)benzonitrile	CC1(C)C(=O)N(c2ccc(C#N)c(C(F)(F)F)c2)C(=S)N1c1ccc(N2CCC(CN3CCC(n4ccc5c(N6CCC(=O)NC6=O)cccc54)CC3)CC2)cc1	C42H43F3N8O3S	AR	P10275	CRBN	WO-2023180388-A1
TPD-Z7GNMT	SCHEMBL26546081	5-[2-[4-[4-[4-Amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidine-1-carbonyl]piperidin-1-yl]ethylamino]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	NC1=NC=NC2=C1C(C1=CC=C(OC3=CC=CC=C3)C=C1)=NN2C1CCN(C(=O)C2CCN(CCNC3=CC=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)CC2)CC1	C43H44N10O6	BTK;IKZF3	Q06187/Q9UKT9	CRBN	WO-2023184898-A1
TPD-KHA99P	SCHEMBL26546084	5-[2-[4-[4-[4-Amino-3-(2-fluoro-4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidine-1-carbonyl]piperidin-1-yl]ethylamino]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	NC1=C2C(C3=C(F)C=C(OC4=CC=CC=C4)C=C3)=NN(C3CCN(C(=O)C4CCN(CCNC5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)C2=NC=N1	C43H43FN10O6	BTK;IKZF3	Q06187/Q9UKT9	CRBN	WO-2023184898-A1
TPD-THB87U	SCHEMBL26546085	5-[2-[4-[4-[4-Amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]-3,3-difluoropiperidine-1-carbonyl]piperidin-1-yl]ethylamino]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	NC1=NC=NC2=C1C(C1=CC=C(OC3=CC=CC=C3)C=C1)=NN2C1CCN(C(=O)C2CCN(CCNC3=CC=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)CC2)CC1(F)F	C43H42F2N10O6	BTK;IKZF3	Q06187/Q9UKT9	CRBN	WO-2023184898-A1
TPD-FJIIQD	WO2023184898A1_4	.	NC1=C2C(C3=C(F)C=C(OC4=CC(F)=CC(F)=C4)C=C3)=NN(C3CCN(C(=O)C4CCN(CCNC5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)C2=NC=N1	C43H41F3N10O6	BTK;IKZF3	Q06187/Q9UKT9	CRBN	WO-2023184898-A1
TPD-UC6HTY	SCHEMBL26546086	5-[2-[4-[4-[4-Amino-3-[2-fluoro-4-(2,3,5,6-tetrafluorophenoxy)phenyl]pyrazolo[3,4-d]pyrimidin-1-yl]piperidine-1-carbonyl]piperidin-1-yl]ethylamino]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	NC1=C2C(C3=C(F)C=C(OC4=C(F)C(F)=CC(F)=C4F)C=C3)=NN(C3CCN(C(=O)C4CCN(CCNC5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)C2=NC=N1	C43H39F5N10O6	BTK;IKZF3	Q06187/Q9UKT9	CRBN	WO-2023184898-A1
TPD-OEYD1A	SCHEMBL26546087	5-[2-[4-[4-[4-Amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidine-1-carbonyl]piperidin-1-yl]propylamino]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CC(CNC1=CC=C2C(=O)N(C3CCC(=O)NC3=O)C(=O)C2=C1)N1CCC(C(=O)N2CCC(N3N=C(C4=CC=C(OC5=CC=CC=C5)C=C4)C4=C3N=CN=C4N)CC2)CC1	C44H46N10O6	BTK;IKZF3	Q06187/Q9UKT9	CRBN	WO-2023184898-A1
TPD-2UN1RU	WO2023185864A1_1	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(OCCOC5=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C60H69F2N9O8S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-HTS1UD	WO2023185864A1_10	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC5(CC4)CN(C4=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C4)C5)=NC3=C1F)=CC(O)=C2	C60H68F2N10O6S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-R3Y7L3	WO2023185864A1_100	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(OCC4(C)CCN(CCOC5=NC6=C(F)C(C7=CC(O)=CC(Cl)=C7C7CC7)=C(F)C=C6C(N6CC7CCC(C6)N7)=N5)CC4)=NO3)C(C)C)C=C2)SC=N1	C57H66ClF2N9O7S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-MQBQWG	WO2023185864A1_101	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(OCCOC4CCN(CCOC5=NC6=C(F)C(C7=CC(O)=CC(Cl)=C7C7CC7)=C(F)C=C6C(N6CC7CCC(C6)N7)=N5)CC4)=NO3)C(C)C)C=C2)SC=N1	C57H66ClF2N9O8S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-YLLPWW	WO2023185864A1_102	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CC5(CCN(CCOC6=NC7=C(F)C(C8=CC(O)=CC(Cl)=C8C8CC8)=C(F)C=C7C(N7CC8CCC(C7)N8)=N6)CC5)C4)=NO3)C(C)C)C=C2)SC=N1	C57H65ClF2N10O6S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-DW31Q4	WO2023185864A1_103	.	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCC2(F)CCN(CCOC3=NC4=C(F)C(C5=CC(O)=CC(Cl)=C5C5CC5)=C(F)C=C4C(N4CC5CCC(C4)N5)=N3)CC2)=NO1	C56H64ClF3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-OBBP83	WO2023185864A1_104	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(OCC4(C)CCN(CCOC5=NC6=C(F)C(C7=CC(O)=CC(Cl)=C7C7CC7)=C(F)C=C6C(N6CC7CCC(C6)N7)=N5)CC4)=NO3)C(C)C)C=C2)SC=N1	C57H66ClF2N9O7S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-I6ISCH	WO2023185864A1_105	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3=CC(OCCOC4CCN(CCOC5=NC6=C(F)C(C7=CC(O)=CC(Cl)=C7C7CC7)=C(F)C=C6C(N6CC7CCC(C6)N7)=N5)CC4)=NO3)C(C)C)C=C2)SC=N1	C57H66ClF2N9O8S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-CHOYPF	WO2023185864A1_106	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3=CC(N4CC5(CCN(CCOC6=NC7=C(F)C(C8=CC(O)=CC(Cl)=C8C8CC8)=C(F)C=C7C(N7CC8CCC(C7)N8)=N6)CC5)C4)=NO3)C(C)C)C=C2)SC=N1	C57H65ClF2N10O6S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-WTX6SY	WO2023185864A1_107	.	CC(C)[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCC2(F)CCN(CCOC3=NC4=C(F)C(C5=CC(O)=CC(Cl)=C5C5CC5)=C(F)C=C4C(N4CC5CCC(C4)N5)=N3)CC2)=NO1	C56H64ClF3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-LVLJJU	WO2023185864A1_108	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3=CC(OCC4(C)CCN(CCOC5=NC6=C(F)C(C7=CC(O)=CC(Cl)=C7C7CC7)=C(F)C=C6C(N6CC7CCC(C6)N7)=N5)CC4)=NO3)C(C)C)C=C2)SC=N1	C57H66ClF2N9O7S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-LEQK7T	WO2023185864A1_109	.	C#CC1=C(F)C=CC2=C1C(C1=NC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(OCCOC5=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C59H64F2N10O8S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-F3PKHK	WO2023185864A1_11	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(COC5=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C59H67F2N9O7S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-KZNVF8	WO2023185864A1_110	.	C#CC1=C(F)C=CC2=C1C(C1=NC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC5(CC4)CN(C4=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C4)C5)=NC3=C1F)=CC(O)=C2	C59H63F2N11O6S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-R038GM	WO2023185864A1_111	.	C#CC1=C(F)C=CC2=C1C(C1=NC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(F)(COC5=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C58H62F3N11O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-B75OG9	WO2023185864A1_112	.	C#CC1=C(F)C=CC2=C1C(C1=NC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(C)(COC5=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C59H64F2N10O7S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-FTYPUE	WO2023185864A1_113	.	C#CC1=C(F)C=CC2=C1C(C1=NC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(OCCOC5=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C59H64F2N10O8S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-74VZLU	SCHEMBL25307600	(2S,4R)-1-[(2R)-2-[3-[7-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]-2,7-diazaspiro[3.5]nonan-2-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL30960062	C#CC1=C(F)C=CC2=C1C(C1=NC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC5(CC4)CN(C4=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C4)C5)=NC3=C1F)=CC(O)=C2	C59H63F2N11O6S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-DT2OFM	WO2023185864A1_115	.	C#CC1=C(F)C=CC2=C1C(C1=NC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(F)(COC5=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C58H62F3N11O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-7YV92H	SCHEMBL25263245	(2S,4R)-1-[(2R)-2-[3-[[1-[2-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]-4-methylpiperidin-4-yl]methoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	C#CC1=C(F)C=CC2=C1C(C1=NC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(C)(COC5=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C59H64F2N10O7S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-8DE2DK	WO2023185864A1_117	.	C#CC1=C(F)C=CC2=C1C(C1=NC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(OCCOC5=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C59H64F2N10O8S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-HVX2CH	WO2023185864A1_118	.	C#CC1=C(F)C=CC2=C1C(C1=NC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC5(CC4)CN(C4=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C4)C5)=NC3=C1F)=CC(O)=C2	C59H63F2N11O6S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-M9ETRP	WO2023185864A1_119	.	C#CC1=C(F)C=CC2=C1C(C1=NC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(F)(COC5=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C58H62F3N11O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-EW05DO	WO2023185864A1_12	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(F)(COC5=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C59H67F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-YLTNZY	WO2023185864A1_120	.	C#CC1=C(F)C=CC2=C1C(C1=NC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(C)(COC5=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C59H64F2N10O7S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-6XOR18	WO2023185864A1_121	.	CCC1=C(F)C=CC2=C1C(C1=NC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC5(CC4)CN(C4=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C4)C5)=NC3=C1F)=CC(O)=C2	C59H67F2N11O6S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-JIY8V7	WO2023185864A1_122-1	.	CCC1=C(F)C=CC2=C1C(C1=NC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(F)(COC5=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C58H66F3N11O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-O5EQVM	WO2023185864A1_122-2	.	CCC1=C(F)C=CC2=C1C(C1=NC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(F)(COC5=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C58H66F3N11O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-S64PFQ	WO2023185864A1_122	.	CCC1=C(F)C=CC2=C1C(C1=NC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(F)(COC5=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C58H66F3N11O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-1XIT22	WO2023185864A1_123	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CC5(CCN(CCOC6=NC7=C(F)C(C8=CC(O)=CC9=C8C(Cl)=C(F)C=C9)=NC=C7C(N7CC8CCC(C7)N8)=N6)CC5)C4)=NO3)C(C)C)C=C2)SC=N1	C57H62ClF2N11O6S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-ESE1Y3	WO2023185864A1_124	.	CC(C)C(C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCC2(F)CCN(CCOC3=NC4=C(F)C(C5=CC(O)=CC(Cl)=C5C5CC5)=NC=C4C(N4CC5CCC(C4)N5)=N3)CC2)=NO1	C55H64ClF2N11O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-TRME1B	WO2023185864A1_125	.	C#CC1=C(F)C=CC2=C1C(C1=CN=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC5(CC4)CN(C4=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C4)C5)=NC3=C1F)=CC(O)=C2	C59H63F2N11O6S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-1DML3E	WO2023185864A1_126	.	CCC1=C(F)C=CC2=C1C(C1=CN=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(F)(COC5=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C58H66F3N11O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-ETGILY	WO2023185864A1_127	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CC5(CCN(CCOC6=NC7=C(F)C(C8=CC(O)=CC9=C8C(Cl)=C(F)C=C9)=CN=C7C(N7CC8CCC(C7)N8)=N6)CC5)C4)=NO3)C(C)C)C=C2)SC=N1	C57H62ClF2N11O6S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-WFG59F	WO2023185864A1_128	.	CC(C)C(C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCC2(F)CCN(CCOC3=NC4=C(F)C(C5=CC(O)=CC(Cl)=C5C5CC5)=CN=C4C(N4CC5CCC(C4)N5)=N3)CC2)=NO1	C55H64ClF2N11O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-Z5WKJF	WO2023185864A1_129	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(=N1)N=C(OCCN1CCC4(CC1)CN(C1=NOC(C(C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=C(C)N=CS6)C=C5)C(C)C)=C1)C4)N=C3N1CC3CCC(C1)N3)=CC(O)=C2	C59H63F2N11O6S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-HTA1QG	WO2023185864A1_13	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(C)(COC5=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C60H69F2N9O7S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-XTH3AD	WO2023185864A1_130	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(=N1)N=C(OCCN1CCC(F)(COC4=NOC(C(C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)CC1)N=C3N1CC3CCC(C1)N3)=CC(O)=C2	C58H66F3N11O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-UN8QLX	WO2023185864A1_131	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CC5(CCN(CCOC6=NC7=NC(C8=CC(O)=CC9=C8C(Cl)=C(F)C=C9)=C(F)C=C7C(N7CC8CCC(C7)N8)=N6)CC5)C4)=NO3)C(C)C)C=C2)SC=N1	C57H62ClF2N11O6S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-DIQUZH	WO2023185864A1_132	.	CC(C)C(C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCC2(F)CCN(CCOC3=NC4=NC(C5=CC(O)=CC(Cl)=C5C5CC5)=C(F)C=C4C(N4CC5CCC(C4)N5)=N3)CC2)=NO1	C55H64ClF2N11O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-A4EJPE	WO2023185864A1_133	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CC5(CCN(CCOC6=NC7=C(F)C(C8=CC(O)=CC9=C8C(C8CC8)=C(F)C=C9)=NC=C7C(N7CC8CCC(C7)N8)=N6)CC5)C4)=NO3)C(C)C)C=C2)SC=N1	C60H67F2N11O6S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-GF5NPQ	WO2023185864A1_134	.	CC(C)C(C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCC2(F)CCN(CCOC3=NC4=C(F)C(C5=CC(O)=CC6=C5C(C5CC5)=C(F)C=C6)=NC=C4C(N4CC5CCC(C4)N5)=N3)CC2)=NO1	C59H66F3N11O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-JK2ZL7	WO2023185864A1_135	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CC5(CCN(CCOC6=NC7=C(F)C(C8=CC(O)=CC9=C8C(C8CC8)=C(F)C=C9)=C(F)C=C7C(N7CC8CCC(C7)N8)=N6)CC5)C4)=NO3)C(C)C)C=C2)SC=N1	C61H67F3N10O6S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-702G2L	WO2023185864A1_136	.	CC(C)C(C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCC2(F)CCN(CCOC3=NC4=C(F)C(C5=CC(O)=CC6=C5C(C5CC5)=C(F)C=C6)=C(F)C=C4C(N4CC5CCC(C4)N5)=N3)CC2)=NO1	C60H66F4N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-YJMKOZ	WO2023185864A1_137	.	CC1=CC=CC(C)=C1C1=CC=C(O)C=C1C1=NC=C2C(N3CC4CCC(C3)N4)=NC(OCCN3CCC4(CC3)CN(C3=NOC(C(C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=C(C)N=CS6)C=C5)C(C)C)=C3)C4)=NC2=C1F	C61H70FN11O6S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-RXVNWL	WO2023185864A1_138	.	CC1=CC=CC(C)=C1C1=CC=C(O)C=C1C1=NC=C2C(N3CC4CCC(C3)N4)=NC(OCCN3CCC(F)(COC4=NOC(C(C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)CC3)=NC2=C1F	C60H69F2N11O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-4CZ3FG	WO2023185864A1_139	.	CC1=CC=CC(C)=C1C1=CC=C(O)C=C1C1=C(F)C=C2C(N3CC4CCC(C3)N4)=NC(OCCN3CCC4(CC3)CN(C3=NOC(C(C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=C(C)N=CS6)C=C5)C(C)C)=C3)C4)=NC2=C1F	C62H70F2N10O6S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-P9QY7L	WO2023185864A1_14	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCC45CCCN4C(COCCOC4=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C4)CC5)=NC3=C1F)=CC(O)=C2	C62H71F2N9O8S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-OWSL42	WO2023185864A1_140	.	CC1=CC=CC(C)=C1C1=CC=C(O)C=C1C1=C(F)C=C2C(N3CC4CCC(C3)N4)=NC(OCCN3CCC(F)(COC4=NOC(C(C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)CC3)=NC2=C1F	C61H69F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-VDX2SV	WO2023185864A1_141	.	CCN1C=CC(=O)C2=C1C(C1=NC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC5(CC4)CN(C4=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C4)C5)=NC3=C1F)=CC(O)=C2	C58H67FN12O7S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-1MQXEP	WO2023185864A1_142	.	CCN1C=CC(=O)C2=C1C(C1=NC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(F)(COC5=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C57H66F2N12O8	KRAS	P01116	VHL	WO-2023185864-A1
TPD-OUAA70	WO2023185864A1_143	.	CCN1C=CC(=O)C2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC5(CC4)CN(C4=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C4)C5)=NC3=C1F)=CC(O)=C2	C59H67F2N11O7S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-5U1R2F	WO2023185864A1_144	.	CCN1C=CC(=O)C2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(F)(COC5=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C58H66F3N11O8	KRAS	P01116	VHL	WO-2023185864-A1
TPD-EL410K	WO2023185864A1_145-1	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(COC5=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)(C(C)C)CC4)=NC3=C1F)=CC(O)=C2	C62H74F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-1HAI5J	WO2023185864A1_145-2	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(COC5=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)(C(C)C)CC4)=NC3=C1F)=CC(O)=C2	C62H74F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-OS3T1J	WO2023185864A1_145	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(COC5=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)(C(C)C)CC4)=NC3=C1F)=CC(O)=C2	C62H74F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-84CFUT	WO2023185864A1_146-1	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CC5CC(C4)C5COC4=NOC([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C60H68F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-UVZFOI	WO2023185864A1_146-2	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CC5CC(C4)C5COC4=NOC([C@@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C60H68F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-TVBT13	WO2023185864A1_146	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CC5CC(C4)C5COC4=NOC(C(C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C60H68F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-X0UHQZ	WO2023185864A1_147-1	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(C)(COC5=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)C(F)C4)=NC3=C1F)=CC(O)=C2	C60H69F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-FUZ80Q	WO2023185864A1_147-2	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(C)(COC5=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)C(F)C4)=NC3=C1F)=CC(O)=C2	C60H69F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-MDU194	WO2023185864A1_147	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(C)(COC5=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)C(F)C4)=NC3=C1F)=CC(O)=C2	C60H69F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-UNWBT2	WO2023185864A1_148-1	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCN(C(=O)OC5=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C58H65F2N11O8	KRAS	P01116	VHL	WO-2023185864-A1
TPD-75KJ3A	WO2023185864A1_148-2	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCN(C(=O)OC5=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C58H65F2N11O8	KRAS	P01116	VHL	WO-2023185864-A1
TPD-JR0JMI	WO2023185864A1_148	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCN(C(=O)OC5=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C58H65F2N11O8	KRAS	P01116	VHL	WO-2023185864-A1
TPD-0JA61O	WO2023185864A1_149-1	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC5(CC4)CC(OC4=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C4)C5)=NC3=C1F)=CC(O)=C2	C61H70F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-BHJIFX	WO2023185864A1_149-2	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC5(CC4)CC(OC4=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C4)C5)=NC3=C1F)=CC(O)=C2	C61H70F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-FBH3OH	WO2023185864A1_149	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC5(CC4)CC(OC4=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C4)C5)=NC3=C1F)=CC(O)=C2	C61H70F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-G23BOF	WO2023185864A1_15	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCC45CCCN4C(COC4=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C4)CC5)=NC3=C1F)=CC(O)=C2	C60H67F2N9O7S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-Z3GC6L	WO2023185864A1_150-1	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(F)(COC5=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)C4)=NC3=C1F)=CC(O)=C2	C58H65F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-HMTQSL	WO2023185864A1_150-2	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(F)(COC5=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)C4)=NC3=C1F)=CC(O)=C2	C58H65F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-QWT9EL	WO2023185864A1_150	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(F)(COC5=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)C4)=NC3=C1F)=CC(O)=C2	C58H65F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-JKA3BQ	WO2023185864A1_151-1	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CC(F)(COC5=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)C4)=NC3=C1F)=CC(O)=C2	C57H63F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-851E7L	WO2023185864A1_151-2	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CC(F)(COC5=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)C4)=NC3=C1F)=CC(O)=C2	C57H63F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-4X35DT	WO2023185864A1_151	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CC(F)(COC5=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)C4)=NC3=C1F)=CC(O)=C2	C57H63F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-C045YX	WO2023185864A1_152-1	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC5(COC6=NOC([C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=CC=NN8C)C=C7)C(C)C)=C6)CC5C4)=NC3=C1F)=CC(O)=C2	C60H68F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-5QP9ZN	WO2023185864A1_152-2	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC5(COC6=NOC([C@@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=CC=NN8C)C=C7)C(C)C)=C6)CC5C4)=NC3=C1F)=CC(O)=C2	C60H68F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-8S4D1Q	WO2023185864A1_152	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC5(COC6=NOC(C(C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=CC=NN8C)C=C7)C(C)C)=C6)CC5C4)=NC3=C1F)=CC(O)=C2	C60H68F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-JBVIPV	WO2023185864A1_153-1	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4C5CC(COC6=NOC([C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=CC=NN8C)C=C7)C(C)C)=C6)CC4C5)=NC3=C1F)=CC(O)=C2	C60H68F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-1TOHLB	WO2023185864A1_153-2	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4C5CC(COC6=NOC([C@@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=CC=NN8C)C=C7)C(C)C)=C6)CC4C5)=NC3=C1F)=CC(O)=C2	C60H68F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-B988KE	WO2023185864A1_153	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4C5CC(COC6=NOC(C(C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=CC=NN8C)C=C7)C(C)C)=C6)CC4C5)=NC3=C1F)=CC(O)=C2	C60H68F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-5XI827	WO2023185864A1_154-1	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CC5CCC(C4)C5COC4=NOC([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C61H70F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-MBUN8B	WO2023185864A1_154-2	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CC5CCC(C4)C5COC4=NOC([C@@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C61H70F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-9X0WWK	WO2023185864A1_154	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CC5CCC(C4)C5COC4=NOC(C(C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C61H70F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-4Q5T9I	WO2023185864A1_155-1	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CC5CCC4CC5COC4=NOC([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C61H70F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-NLZBVO	WO2023185864A1_155-2	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CC5CCC4CC5COC4=NOC([C@@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C61H70F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-6IJYQY	WO2023185864A1_155	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CC5CCC4CC5COC4=NOC(C(C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C61H70F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-SAD4TJ	WO2023185864A1_156-1	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4C5CCC4CC(COC4=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C4)C5)=NC3=C1F)=CC(O)=C2	C61H70F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-SXRXS8	WO2023185864A1_156-2	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4C5CCC4CC(COC4=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C4)C5)=NC3=C1F)=CC(O)=C2	C61H70F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-GRI4UM	WO2023185864A1_156	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4C5CCC4CC(COC4=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C4)C5)=NC3=C1F)=CC(O)=C2	C61H70F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-1JH8OV	WO2023185864A1_157-1	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CC5CC(C4)C5COC4=NOC([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C60H67F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-BGF65Y	WO2023185864A1_157-2	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CC5CC(C4)C5COC4=NOC([C@@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C60H67F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-2KF0I8	WO2023185864A1_157	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CC5CC(C4)C5COC4=NOC(C(C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C60H67F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-G9LS5H	WO2023185864A1_158	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CC5CCC(C4)N5COC4=NOC(C(C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C60H68F3N11O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-2B3ME8	WO2023185864A1_159	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CC5CCC4CN5COC4=NOC(C(C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C60H68F3N11O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-9WO22S	WO2023185864A1_16	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCC45CCCN4C(COC4=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C4)CC5)=NC3=C1F)=CC(O)=C2	C60H68F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-SNQIA3	WO2023185864A1_160	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCN4C5CC4CN(COC4=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C4)C5)=NC3=C1F)=CC(O)=C2	C59H66F3N11O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-0X2VT4	WO2023185864A1_161	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCN4C5CCC4CN(COC4=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C4)C5)=NC3=C1F)=CC(O)=C2	C60H68F3N11O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-I4SVJZ	WO2023185864A1_162	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CC5CC(C4)N5COC4=NOC(C(C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C59H66F3N11O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-ES0ZG1	WO2023185864A1_163-1	.	CCC1=C(F)C=CC2=C1C(C1=NC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CC5CC(C4)C5COC4=NOC([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C59H67F2N11O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-30WX96	WO2023185864A1_163-2	.	CCC1=C(F)C=CC2=C1C(C1=NC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CC5CC(C4)C5COC4=NOC([C@@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C59H67F2N11O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-2U24I4	WO2023185864A1_163	.	CCC1=C(F)C=CC2=C1C(C1=NC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CC5CC(C4)C5COC4=NOC(C(C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C59H67F2N11O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-YPFNIZ	WO2023185864A1_164-1	.	C#CC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CC5CC(C4)C5COC4=NOC([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C60H64F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-Z6KSBL	WO2023185864A1_164-2	.	C#CC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CC5CC(C4)C5COC4=NOC([C@@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C60H64F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-HXKLU9	WO2023185864A1_164	.	C#CC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CC5CC(C4)C5COC4=NOC(C(C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C60H64F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-NQWRXI	WO2023185864A1_165-1	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CC5CC(C4)C5COC4=NOC([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C60H63F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-DAM91Y	WO2023185864A1_165-2	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CC5CC(C4)C5COC4=NOC([C@@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C60H63F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-R9ATO2	WO2023185864A1_165	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CC5CC(C4)C5COC4=NOC(C(C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C60H63F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-EGPLTP	WO2023185864A1_166-1	.	C#CC1=C(F)C=CC2=C1C(C1=NC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CC5CC(C4)C5COC4=NOC([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C59H63F2N11O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-9FILZ6	WO2023185864A1_166-2	.	C#CC1=C(F)C=CC2=C1C(C1=NC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CC5CC(C4)C5COC4=NOC([C@@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C59H63F2N11O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-38JSXD	WO2023185864A1_166	.	C#CC1=C(F)C=CC2=C1C(C1=NC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CC5CC(C4)C5COC4=NOC(C(C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C59H63F2N11O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-AXFHLG	WO2023185864A1_167-1	.	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCC2C3CC2CN(CCOC2=NC4=C(F)C(C5=CC(O)=CC6=C5C(C5CC5)=C(F)C=C6)=NC=C4C(N4CC5CCC(C4)N5)=N2)C3)=NO1	C60H67F2N11O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-0SNOIZ	WO2023185864A1_167-2	.	CC(C)[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCC2C3CC2CN(CCOC2=NC4=C(F)C(C5=CC(O)=CC6=C5C(C5CC5)=C(F)C=C6)=NC=C4C(N4CC5CCC(C4)N5)=N2)C3)=NO1	C60H67F2N11O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-NSU9R1	WO2023185864A1_167	.	CC(C)C(C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCC2C3CC2CN(CCOC2=NC4=C(F)C(C5=CC(O)=CC6=C5C(C5CC5)=C(F)C=C6)=NC=C4C(N4CC5CCC(C4)N5)=N2)C3)=NO1	C60H67F2N11O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-PIAJZE	WO2023185864A1_168-1	.	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCC2C3CC2CN(CCOC2=NC4=C(F)C(C5=CC(O)=CC6=C5C(C5CC5)=C(F)C=C6)=CC=C4C(N4CC5CCC(C4)N5)=N2)C3)=NO1	C61H68F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-UJ26TZ	WO2023185864A1_168-2	.	CC(C)[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCC2C3CC2CN(CCOC2=NC4=C(F)C(C5=CC(O)=CC6=C5C(C5CC5)=C(F)C=C6)=CC=C4C(N4CC5CCC(C4)N5)=N2)C3)=NO1	C61H68F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-WBKC72	WO2023185864A1_168	.	CC(C)C(C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCC2C3CC2CN(CCOC2=NC4=C(F)C(C5=CC(O)=CC6=C5C(C5CC5)=C(F)C=C6)=CC=C4C(N4CC5CCC(C4)N5)=N2)C3)=NO1	C61H68F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-N59KAC	WO2023185864A1_169-1	.	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCC2C3CC2CN(CCOC2=NC4=C(F)C(C5=CC(O)=CC6=C5C(C5CC5)=C(F)C=C6)=C(F)C=C4C(N4CC5CCC(C4)N5)=N2)C3)=NO1	C61H67F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-0TFGBC	WO2023185864A1_169-2	.	CC(C)[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCC2C3CC2CN(CCOC2=NC4=C(F)C(C5=CC(O)=CC6=C5C(C5CC5)=C(F)C=C6)=C(F)C=C4C(N4CC5CCC(C4)N5)=N2)C3)=NO1	C61H67F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-COC0G9	WO2023185864A1_169	.	CC(C)C(C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCC2C3CC2CN(CCOC2=NC4=C(F)C(C5=CC(O)=CC6=C5C(C5CC5)=C(F)C=C6)=C(F)C=C4C(N4CC5CCC(C4)N5)=N2)C3)=NO1	C61H67F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-3Y8ONZ	WO2023185864A1_17	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(OCCOC5=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C60H69F2N9O8S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-7FIT2B	WO2023185864A1_170-1	.	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCC2C3CC2CN(CC2(COC4=NC5=C(F)C(C6=CC(O)=CC7=C6C(C6CC6)=C(F)C=C7)=CC=C5C(N5CC6CCC(C5)N6)=N4)CC2)C3)=NO1	C64H72F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-PVR2GX	WO2023185864A1_170-2	.	CC(C)[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCC2C3CC2CN(CC2(COC4=NC5=C(F)C(C6=CC(O)=CC7=C6C(C6CC6)=C(F)C=C7)=CC=C5C(N5CC6CCC(C5)N6)=N4)CC2)C3)=NO1	C64H72F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-2ND9JM	WO2023185864A1_170	.	CC(C)C(C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCC2C3CC2CN(CC2(COC4=NC5=C(F)C(C6=CC(O)=CC7=C6C(C6CC6)=C(F)C=C7)=CC=C5C(N5CC6CCC(C5)N6)=N4)CC2)C3)=NO1	C64H72F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-F5860X	WO2023185864A1_171-1	.	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCC2C3CC2CN(CC2(COC4=NC5=C(F)C(C6=CC(O)=CC7=C6C(C6CC6)=C(F)C=C7)=C(F)C=C5C(N5CC6CCC(C5)N6)=N4)CC2)C3)=NO1	C64H71F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-M4T684	WO2023185864A1_171-2	.	CC(C)[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCC2C3CC2CN(CC2(COC4=NC5=C(F)C(C6=CC(O)=CC7=C6C(C6CC6)=C(F)C=C7)=C(F)C=C5C(N5CC6CCC(C5)N6)=N4)CC2)C3)=NO1	C64H71F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-17UFIF	WO2023185864A1_171	.	CC(C)C(C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCC2C3CC2CN(CC2(COC4=NC5=C(F)C(C6=CC(O)=CC7=C6C(C6CC6)=C(F)C=C7)=C(F)C=C5C(N5CC6CCC(C5)N6)=N4)CC2)C3)=NO1	C64H71F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-N1XBPP	WO2023185864A1_172-1	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN5CC6CC(C5)C6COC5=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C63H72F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-ML42WX	WO2023185864A1_172-2	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN5CC6CC(C5)C6COC5=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C63H72F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-5BZ5RP	WO2023185864A1_172	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN5CC6CC(C5)C6COC5=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C63H72F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-T8R584	WO2023185864A1_173-1	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN5CC6CC(C5)C6COC5=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C63H71F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-3FX2QE	WO2023185864A1_173-2	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN5CC6CC(C5)C6COC5=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C63H71F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-H4X35P	WO2023185864A1_174-1	.	C#CC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN5CC6CC(C5)C6COC5=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C63H68F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-PO5FP8	WO2023185864A1_174-2	.	C#CC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN5CC6CC(C5)C6COC5=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C63H68F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-GWI4UK	WO2023185864A1_174	.	C#CC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN5CC6CC(C5)C6COC5=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C63H68F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-4RWTI1	WO2023185864A1_175-1	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN5CC6CC(C5)C6COC5=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C63H67F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-O72VIY	WO2023185864A1_175-2	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN5CC6CC(C5)C6COC5=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C63H67F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-95K8Y7	WO2023185864A1_175	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN5CC6CC(C5)C6COC5=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C63H67F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-DACLZE	WO2023185864A1_176-1	.	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCC2(F)CCN(CC3(COC4=NC5=C(F)C(C6=CC(O)=CC7=C6C(C6CC6)=C(F)C=C7)=CC=C5C(N5CC6CCC(C5)N6)=N4)CC3)CC2)=NO1	C63H71F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-GFSG9J	WO2023185864A1_176-2	.	CC(C)[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCC2(F)CCN(CC3(COC4=NC5=C(F)C(C6=CC(O)=CC7=C6C(C6CC6)=C(F)C=C7)=CC=C5C(N5CC6CCC(C5)N6)=N4)CC3)CC2)=NO1	C63H71F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-3UGEEU	WO2023185864A1_176	.	CC(C)C(C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCC2(F)CCN(CC3(COC4=NC5=C(F)C(C6=CC(O)=CC7=C6C(C6CC6)=C(F)C=C7)=CC=C5C(N5CC6CCC(C5)N6)=N4)CC3)CC2)=NO1	C63H71F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-N2LJCH	WO2023185864A1_177-1	.	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCC2(F)CCN(CC3(COC4=NC5=C(F)C(C6=CC(O)=CC7=C6C(C6CC6)=C(F)C=C7)=C(F)C=C5C(N5CC6CCC(C5)N6)=N4)CC3)CC2)=NO1	C63H70F4N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-4TYNVY	WO2023185864A1_177-2	.	CC(C)[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCC2(F)CCN(CC3(COC4=NC5=C(F)C(C6=CC(O)=CC7=C6C(C6CC6)=C(F)C=C7)=C(F)C=C5C(N5CC6CCC(C5)N6)=N4)CC3)CC2)=NO1	C63H70F4N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-8IMYPI	WO2023185864A1_177	.	CC(C)C(C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCC2(F)CCN(CC3(COC4=NC5=C(F)C(C6=CC(O)=CC7=C6C(C6CC6)=C(F)C=C7)=C(F)C=C5C(N5CC6CCC(C5)N6)=N4)CC3)CC2)=NO1	C63H70F4N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-0Z4BLZ	WO2023185864A1_178-1	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN5CCC(F)(COC6=NOC([C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=CC=NN8C)C=C7)C(C)C)=C6)CC5)CC4)=NC3=C1F)=CC(O)=C2	C62H71F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-ZHL9QU	WO2023185864A1_178-2	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN5CCC(F)(COC6=NOC([C@@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=CC=NN8C)C=C7)C(C)C)=C6)CC5)CC4)=NC3=C1F)=CC(O)=C2	C62H71F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-SPJ5Q0	WO2023185864A1_178	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN5CCC(F)(COC6=NOC(C(C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=CC=NN8C)C=C7)C(C)C)=C6)CC5)CC4)=NC3=C1F)=CC(O)=C2	C62H71F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-W4MXLI	WO2023185864A1_179-1	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN5CCC(F)(COC6=NOC([C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=CC=NN8C)C=C7)C(C)C)=C6)CC5)CC4)=NC3=C1F)=CC(O)=C2	C62H70F4N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-HNRM18	WO2023185864A1_179-2	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN5CCC(F)(COC6=NOC([C@@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=CC=NN8C)C=C7)C(C)C)=C6)CC5)CC4)=NC3=C1F)=CC(O)=C2	C62H70F4N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-3ZBXW1	WO2023185864A1_179	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN5CCC(F)(COC6=NOC(C(C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=CC=NN8C)C=C7)C(C)C)=C6)CC5)CC4)=NC3=C1F)=CC(O)=C2	C62H70F4N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-YQ1ZHB	WO2023185864A1_18	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC5(CC4)CN(C4=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C4)C5)=NC3=C1F)=CC(O)=C2	C60H68F2N10O6S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-17ATKP	WO2023185864A1_180-1	.	C#CC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN5CCC(F)(COC6=NOC([C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=CC=NN8C)C=C7)C(C)C)=C6)CC5)CC4)=NC3=C1F)=CC(O)=C2	C62H67F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-DRJ2IU	WO2023185864A1_180-2	.	C#CC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN5CCC(F)(COC6=NOC([C@@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=CC=NN8C)C=C7)C(C)C)=C6)CC5)CC4)=NC3=C1F)=CC(O)=C2	C62H67F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-661Q5O	WO2023185864A1_180	.	C#CC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN5CCC(F)(COC6=NOC(C(C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=CC=NN8C)C=C7)C(C)C)=C6)CC5)CC4)=NC3=C1F)=CC(O)=C2	C62H67F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-D7VN8L	WO2023185864A1_181-1	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN5CCC(F)(COC6=NOC([C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=CC=NN8C)C=C7)C(C)C)=C6)CC5)CC4)=NC3=C1F)=CC(O)=C2	C62H66F4N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-D1CK7G	WO2023185864A1_181-2	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN5CCC(F)(COC6=NOC([C@@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=CC=NN8C)C=C7)C(C)C)=C6)CC5)CC4)=NC3=C1F)=CC(O)=C2	C62H66F4N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-2MSHLZ	WO2023185864A1_181	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN5CCC(F)(COC6=NOC(C(C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=CC=NN8C)C=C7)C(C)C)=C6)CC5)CC4)=NC3=C1F)=CC(O)=C2	C62H66F4N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-PPR0EE	WO2023185864A1_182-1	.	C#CC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCCNCCOC4=NOC([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C56H60F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-J7QAA9	WO2023185864A1_182-2	.	C#CC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCCNCCOC4=NOC([C@@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C56H60F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-OJJJJN	WO2023185864A1_182	.	C#CC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCCNCCOC4=NOC(C(C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C56H60F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-G5Y9XX	WO2023185864A1_183-1	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCCNCCOC4=NOC([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C56H59F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-XY683Y	WO2023185864A1_183-2	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCCNCCOC4=NOC([C@@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C56H59F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-90WFCY	WO2023185864A1_183	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCCNCCOC4=NOC(C(C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C56H59F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-RGQIGQ	WO2023185864A1_184-1	.	C#CC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCCN(C)CCOC4=NOC([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C57H62F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-2HTKQX	WO2023185864A1_184-2	.	C#CC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCCN(C)CCOC4=NOC([C@@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C57H62F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-L5WPNJ	WO2023185864A1_184	.	C#CC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCCN(C)CCOC4=NOC(C(C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C57H62F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-LR8IOV	WO2023185864A1_185-1	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCCN(C)CCOC4=NOC([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C57H61F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-9CTUH5	WO2023185864A1_185-2	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCCN(C)CCOC4=NOC([C@@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C57H61F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-S1JNDC	WO2023185864A1_185	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCCN(C)CCOC4=NOC(C(C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C57H61F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-DVG153	WO2023185864A1_186-1	.	C#CC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCCN(CC)CCOC4=NOC([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C58H64F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-NN51YK	WO2023185864A1_186-2	.	C#CC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCCN(CC)CCOC4=NOC([C@@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C58H64F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-HMPW8P	WO2023185864A1_186	.	C#CC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCCN(CC)CCOC4=NOC(C(C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C58H64F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-L6CIDA	WO2023185864A1_187-1	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCCN(CC)CCOC4=NOC([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C58H63F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-70ZZH6	WO2023185864A1_187-2	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCCN(CC)CCOC4=NOC([C@@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C58H63F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-R1L5G4	WO2023185864A1_187	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCCN(CC)CCOC4=NOC(C(C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C58H63F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-DC32OF	WO2023185864A1_188-1	.	C#CC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCCN(CCOC4=NOC([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)C(C)C)=NC3=C1F)=CC(O)=C2	C59H66F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-ZK1BE2	WO2023185864A1_188-2	.	C#CC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCCN(CCOC4=NOC([C@@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)C(C)C)=NC3=C1F)=CC(O)=C2	C59H66F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-GN1H2F	WO2023185864A1_188	.	C#CC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCCN(CCOC4=NOC(C(C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)C(C)C)=NC3=C1F)=CC(O)=C2	C59H66F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-IYF8NE	WO2023185864A1_189-1	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCCN(CCOC4=NOC([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)C(C)C)=NC3=C1F)=CC(O)=C2	C59H65F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-QFYJGU	WO2023185864A1_189-2	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCCN(CCOC4=NOC([C@@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)C(C)C)=NC3=C1F)=CC(O)=C2	C59H65F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-6J5574	WO2023185864A1_189	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCCN(CCOC4=NOC(C(C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)C(C)C)=NC3=C1F)=CC(O)=C2	C59H65F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-J7MBSR	WO2023185864A1_19	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(COC5=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C59H67F2N9O7S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-PK5JM1	WO2023185864A1_190-1	.	C#CC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCCN(CCOC4=NOC([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)C4CC4)=NC3=C1F)=CC(O)=C2	C59H64F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-GSRQS9	WO2023185864A1_190-2	.	C#CC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCCN(CCOC4=NOC([C@@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)C4CC4)=NC3=C1F)=CC(O)=C2	C59H64F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-6XOU1Z	WO2023185864A1_190	.	C#CC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCCN(CCOC4=NOC(C(C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)C4CC4)=NC3=C1F)=CC(O)=C2	C59H64F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-UGUAO1	WO2023185864A1_191-1	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCCN(CCOC4=NOC([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)C4CC4)=NC3=C1F)=CC(O)=C2	C59H63F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-DH7YNX	WO2023185864A1_191-2	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCCN(CCOC4=NOC([C@@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)C4CC4)=NC3=C1F)=CC(O)=C2	C59H63F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-B9IDZW	WO2023185864A1_191	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCCN(CCOC4=NOC(C(C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)C4CC4)=NC3=C1F)=CC(O)=C2	C59H63F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-ZAV53P	WO2023185864A1_192-1	.	C#CC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CNCCOC5=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C58H62F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-A7H7UO	WO2023185864A1_192-2	.	C#CC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CNCCOC5=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C58H62F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-0ESXMS	WO2023185864A1_192	.	C#CC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CNCCOC5=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C58H62F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-V8MFZ4	WO2023185864A1_193-1	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CNCCOC5=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C58H61F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-DO0EK7	WO2023185864A1_193-2	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CNCCOC5=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C58H61F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-XXLGPE	WO2023185864A1_193	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CNCCOC5=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C58H61F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-GYAR44	WO2023185864A1_194-1	.	C#CC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN(C)CCOC5=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C59H64F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-UAOMCY	WO2023185864A1_194-2	.	C#CC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN(C)CCOC5=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C59H64F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-SJYML9	WO2023185864A1_194	.	C#CC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN(C)CCOC5=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C59H64F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-19RGLB	WO2023185864A1_195-1	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN(C)CCOC5=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C59H63F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-UK7UAO	WO2023185864A1_195-2	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN(C)CCOC5=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C59H63F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-D654CA	WO2023185864A1_195	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN(C)CCOC5=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C59H63F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-0G31RS	WO2023185864A1_196-1	.	C#CC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN(CC)CCOC5=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C60H66F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-OI0G99	WO2023185864A1_196-2	.	C#CC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN(CC)CCOC5=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C60H66F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-1O49SD	WO2023185864A1_196	.	C#CC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN(CC)CCOC5=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C60H66F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-1A8PU2	WO2023185864A1_197-1	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN(CC)CCOC5=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C60H65F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-BDJDHO	WO2023185864A1_197-2	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN(CC)CCOC5=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C60H65F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-GDK415	WO2023185864A1_197	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN(CC)CCOC5=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C60H65F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-TRN6FE	WO2023185864A1_198-1	.	C#CC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN(CCOC5=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)C(C)C)CC4)=NC3=C1F)=CC(O)=C2	C61H68F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-TY9MQR	WO2023185864A1_198-2	.	C#CC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN(CCOC5=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)C(C)C)CC4)=NC3=C1F)=CC(O)=C2	C61H68F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-979K6A	WO2023185864A1_198	.	C#CC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN(CCOC5=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)C(C)C)CC4)=NC3=C1F)=CC(O)=C2	C61H68F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-QB8020	WO2023185864A1_199-1	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN(CCOC5=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)C(C)C)CC4)=NC3=C1F)=CC(O)=C2	C61H67F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-TI5DM5	WO2023185864A1_199-2	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN(CCOC5=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)C(C)C)CC4)=NC3=C1F)=CC(O)=C2	C61H67F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-0631NB	WO2023185864A1_199	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN(CCOC5=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)C(C)C)CC4)=NC3=C1F)=CC(O)=C2	C61H67F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-KRMQCJ	WO2023185864A1_2	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC5(CC4)CN(C4=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C4)C5)=NC3=C1F)=CC(O)=C2	C60H68F2N10O6S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-I8DEMX	WO2023185864A1_20	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(F)(COC5=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C59H67F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-HM492L	WO2023185864A1_200-1	.	C#CC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN(CCOC5=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)C5CC5)CC4)=NC3=C1F)=CC(O)=C2	C61H66F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-FXWWVN	WO2023185864A1_200-2	.	C#CC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN(CCOC5=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)C5CC5)CC4)=NC3=C1F)=CC(O)=C2	C61H66F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-F1E5KR	WO2023185864A1_200	.	C#CC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN(CCOC5=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)C5CC5)CC4)=NC3=C1F)=CC(O)=C2	C61H66F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-B6WCOB	WO2023185864A1_201-1	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN(CCOC5=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)C5CC5)CC4)=NC3=C1F)=CC(O)=C2	C61H65F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-32838O	WO2023185864A1_201-2	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN(CCOC5=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)C5CC5)CC4)=NC3=C1F)=CC(O)=C2	C61H65F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-LK780C	WO2023185864A1_201	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN(CCOC5=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)C5CC5)CC4)=NC3=C1F)=CC(O)=C2	C61H65F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-K7JF4K	WO2023185864A1_202-1	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCCNCCOC4=NOC([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C56H64F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-NVMVIE	WO2023185864A1_202-2	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCCNCCOC4=NOC([C@@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C56H64F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-Y2JJ39	WO2023185864A1_202	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCCNCCOC4=NOC(C(C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C56H64F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-1EMXY9	WO2023185864A1_203-1	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCCNCCOC4=NOC([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C56H63F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-DB8B4U	WO2023185864A1_203-2	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCCNCCOC4=NOC([C@@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C56H63F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-93I6RM	WO2023185864A1_203	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCCNCCOC4=NOC(C(C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C56H63F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-GCR00U	WO2023185864A1_204-1	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCCN(C)CCOC4=NOC([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C57H66F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-H4OEBV	WO2023185864A1_204-2	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCCN(C)CCOC4=NOC([C@@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C57H66F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-05IU0E	WO2023185864A1_204	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCCN(C)CCOC4=NOC(C(C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C57H66F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-JSH6B0	WO2023185864A1_205-1	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCCN(C)CCOC4=NOC([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C57H65F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-VG2S16	WO2023185864A1_205-2	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCCN(C)CCOC4=NOC([C@@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C57H65F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-9W9KJA	WO2023185864A1_205	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCCN(C)CCOC4=NOC(C(C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C57H65F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-1II7LK	WO2023185864A1_206-1	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCCN(CC)CCOC4=NOC([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C58H68F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-WH4TIB	WO2023185864A1_206-2	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCCN(CC)CCOC4=NOC([C@@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C58H68F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-SUEXFC	WO2023185864A1_206	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCCN(CC)CCOC4=NOC(C(C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C58H68F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-YBBGML	WO2023185864A1_207-1	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCCN(CC)CCOC4=NOC([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C58H67F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-FRCSYL	WO2023185864A1_207-2	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCCN(CC)CCOC4=NOC([C@@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C58H67F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-ENW979	WO2023185864A1_207	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCCN(CC)CCOC4=NOC(C(C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)=NC3=C1F)=CC(O)=C2	C58H67F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-QIO0EI	WO2023185864A1_208-1	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCCN(CCOC4=NOC([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)C(C)C)=NC3=C1F)=CC(O)=C2	C59H70F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-FKEHCI	WO2023185864A1_208-2	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCCN(CCOC4=NOC([C@@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)C(C)C)=NC3=C1F)=CC(O)=C2	C59H70F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-8SI6RW	WO2023185864A1_208	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCCN(CCOC4=NOC(C(C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)C(C)C)=NC3=C1F)=CC(O)=C2	C59H70F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-0HT2MG	WO2023185864A1_209-1	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCCN(CCOC4=NOC([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)C(C)C)=NC3=C1F)=CC(O)=C2	C59H69F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-9YILXD	WO2023185864A1_209-2	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCCN(CCOC4=NOC([C@@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)C(C)C)=NC3=C1F)=CC(O)=C2	C59H69F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-NJ4ZB4	WO2023185864A1_209	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCCN(CCOC4=NOC(C(C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)C(C)C)=NC3=C1F)=CC(O)=C2	C59H69F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-BM997F	WO2023185864A1_21	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(C)(COC5=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C60H69F2N9O7S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-LBX3D0	WO2023185864A1_210-1	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCCN(CCOC4=NOC([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)C4CC4)=NC3=C1F)=CC(O)=C2	C59H68F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-1MK62N	WO2023185864A1_210-2	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCCN(CCOC4=NOC([C@@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)C4CC4)=NC3=C1F)=CC(O)=C2	C59H68F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-6PMMBK	WO2023185864A1_210	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCCN(CCOC4=NOC(C(C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)C4CC4)=NC3=C1F)=CC(O)=C2	C59H68F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-YIO80O	WO2023185864A1_211-1	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCCN(CCOC4=NOC([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)C4CC4)=NC3=C1F)=CC(O)=C2	C59H67F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-KCJFA3	WO2023185864A1_211-2	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCCN(CCOC4=NOC([C@@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)C4CC4)=NC3=C1F)=CC(O)=C2	C59H67F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-0P2YD6	WO2023185864A1_211	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCCN(CCOC4=NOC(C(C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=CC=NN6C)C=C5)C(C)C)=C4)C4CC4)=NC3=C1F)=CC(O)=C2	C59H67F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-KHABFT	WO2023185864A1_212-1	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CNCCOC5=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C58H66F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-3YQF1Z	WO2023185864A1_212-2	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CNCCOC5=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C58H66F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-G0AASP	WO2023185864A1_212	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CNCCOC5=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C58H66F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-B5XAUC	WO2023185864A1_213-1	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CNCCOC5=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C58H65F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-9704T1	WO2023185864A1_213-2	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CNCCOC5=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C58H65F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-BRWRH4	WO2023185864A1_213	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CNCCOC5=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C58H65F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-JPVT98	WO2023185864A1_214-1	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN(C)CCOC5=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C59H68F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-XJMGVU	WO2023185864A1_214-2	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN(C)CCOC5=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C59H68F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-WFGFXO	WO2023185864A1_214	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN(C)CCOC5=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C59H68F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-UKQNTL	WO2023185864A1_215-1	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN(C)CCOC5=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C59H67F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-GR7CI3	WO2023185864A1_215-2	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN(C)CCOC5=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C59H67F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-LQ0S5H	WO2023185864A1_215	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN(C)CCOC5=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C59H67F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-5IHYB0	WO2023185864A1_216-1	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN(CC)CCOC5=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C60H70F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-28XMDT	WO2023185864A1_216-2	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN(CC)CCOC5=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C60H70F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-OYJV07	WO2023185864A1_216	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN(CC)CCOC5=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C60H70F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-RX3K0U	WO2023185864A1_217-1	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN(CC)CCOC5=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C60H69F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-KXPSTP	WO2023185864A1_217-2	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN(CC)CCOC5=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C60H69F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-5CCUU2	WO2023185864A1_217	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN(CC)CCOC5=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C60H69F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-15ZS5C	WO2023185864A1_218-1	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN(CCOC5=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)C(C)C)CC4)=NC3=C1F)=CC(O)=C2	C61H72F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-6JACMD	WO2023185864A1_218-2	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN(CCOC5=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)C(C)C)CC4)=NC3=C1F)=CC(O)=C2	C61H72F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-LLMIWG	WO2023185864A1_218	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN(CCOC5=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)C(C)C)CC4)=NC3=C1F)=CC(O)=C2	C61H72F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-5Z8YFV	WO2023185864A1_219-1	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN(CCOC5=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)C(C)C)CC4)=NC3=C1F)=CC(O)=C2	C61H71F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-CCBX6W	WO2023185864A1_219-2	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN(CCOC5=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)C(C)C)CC4)=NC3=C1F)=CC(O)=C2	C61H71F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-GOM17T	WO2023185864A1_219	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN(CCOC5=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)C(C)C)CC4)=NC3=C1F)=CC(O)=C2	C61H71F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-E94TLJ	WO2023185864A1_22	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCC45CCCN4C(COCCOC4=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C4)CC5)=NC3=C1F)=CC(O)=C2	C62H71F2N9O8S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-CGTFZL	WO2023185864A1_220-1	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN(CCOC5=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)C5CC5)CC4)=NC3=C1F)=CC(O)=C2	C61H70F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-X8PNVZ	WO2023185864A1_220-2	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN(CCOC5=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)C5CC5)CC4)=NC3=C1F)=CC(O)=C2	C61H70F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-M0XMXW	WO2023185864A1_220	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN(CCOC5=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)C5CC5)CC4)=NC3=C1F)=CC(O)=C2	C61H70F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-JPWZG8	WO2023185864A1_221-1	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN(CCOC5=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)C5CC5)CC4)=NC3=C1F)=CC(O)=C2	C61H69F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-0P5ZXE	WO2023185864A1_221-2	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN(CCOC5=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)C5CC5)CC4)=NC3=C1F)=CC(O)=C2	C61H69F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-BTJAXR	WO2023185864A1_221	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCC4(CN(CCOC5=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)C5CC5)CC4)=NC3=C1F)=CC(O)=C2	C61H69F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-KJ0MY5	WO2023185864A1_222-1	.	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCCNCCCOC2=NC3=C(F)C(C4=CC(O)=CC5=C4C(C4CC4)=C(F)C=C5)=CC=C3C(N3CC4CCC(C3)N4)=N2)=NO1	C57H64F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-A6KP3V	WO2023185864A1_222-2	.	CC(C)[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCCNCCCOC2=NC3=C(F)C(C4=CC(O)=CC5=C4C(C4CC4)=C(F)C=C5)=CC=C3C(N3CC4CCC(C3)N4)=N2)=NO1	C57H64F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-INNET4	WO2023185864A1_222	.	CC(C)C(C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCCNCCCOC2=NC3=C(F)C(C4=CC(O)=CC5=C4C(C4CC4)=C(F)C=C5)=CC=C3C(N3CC4CCC(C3)N4)=N2)=NO1	C57H64F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-TLJ3A6	WO2023185864A1_223-1	.	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCCNCCCOC2=NC3=C(F)C(C4=CC(O)=CC5=C4C(C4CC4)=C(F)C=C5)=C(F)C=C3C(N3CC4CCC(C3)N4)=N2)=NO1	C57H63F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-1MY02W	WO2023185864A1_223-2	.	CC(C)[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCCNCCCOC2=NC3=C(F)C(C4=CC(O)=CC5=C4C(C4CC4)=C(F)C=C5)=C(F)C=C3C(N3CC4CCC(C3)N4)=N2)=NO1	C57H63F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-VTFJ6M	WO2023185864A1_223	.	CC(C)C(C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCCNCCCOC2=NC3=C(F)C(C4=CC(O)=CC5=C4C(C4CC4)=C(F)C=C5)=C(F)C=C3C(N3CC4CCC(C3)N4)=N2)=NO1	C57H63F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-K0VRZE	WO2023185864A1_224-1	.	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCCNCC2(COC3=NC4=C(F)C(C5=CC(O)=CC6=C5C(C5CC5)=C(F)C=C6)=CC=C4C(N4CC5CCC(C4)N5)=N3)CC2)=NO1	C59H66F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-IOBQJM	WO2023185864A1_224-2	.	CC(C)[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCCNCC2(COC3=NC4=C(F)C(C5=CC(O)=CC6=C5C(C5CC5)=C(F)C=C6)=CC=C4C(N4CC5CCC(C4)N5)=N3)CC2)=NO1	C59H66F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-3SEYWB	WO2023185864A1_224	.	CC(C)C(C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCCN(C)CCCOC2=NC3=C(F)C(C4=CC(O)=CC5=C4C(C4CC4)=C(F)C=C5)=CC=C3C(N3CC4CCC(C3)N4)=N2)=NO1	C58H66F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-C51VFG	WO2023185864A1_225-1	.	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCCNCC2(COC3=NC4=C(F)C(C5=CC(O)=CC6=C5C(C5CC5)=C(F)C=C6)=C(F)C=C4C(N4CC5CCC(C4)N5)=N3)CC2)=NO1	C59H65F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-7WWLXW	WO2023185864A1_225-2	.	CC(C)[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCCNCC2(COC3=NC4=C(F)C(C5=CC(O)=CC6=C5C(C5CC5)=C(F)C=C6)=C(F)C=C4C(N4CC5CCC(C4)N5)=N3)CC2)=NO1	C59H65F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-TV1DVF	WO2023185864A1_225	.	CC(C)C(C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCCNCC2(COC3=NC4=C(F)C(C5=CC(O)=CC6=C5C(C5CC5)=C(F)C=C6)=C(F)C=C4C(N4CC5CCC(C4)N5)=N3)CC2)=NO1	C59H65F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-QNDVOI	WO2023185864A1_226-1	.	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCCN(C)CC2(COC3=NC4=C(F)C(C5=CC(O)=CC6=C5C(C5CC5)=C(F)C=C6)=CC=C4C(N4CC5CCC(C4)N5)=N3)CC2)=NO1	C60H68F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-0DKYVT	WO2023185864A1_226-2	.	CC(C)[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCCN(C)CC2(COC3=NC4=C(F)C(C5=CC(O)=CC6=C5C(C5CC5)=C(F)C=C6)=CC=C4C(N4CC5CCC(C4)N5)=N3)CC2)=NO1	C60H68F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-1DLQU0	WO2023185864A1_226	.	CC(C)C(C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCCN(C)CC2(COC3=NC4=C(F)C(C5=CC(O)=CC6=C5C(C5CC5)=C(F)C=C6)=CC=C4C(N4CC5CCC(C4)N5)=N3)CC2)=NO1	C60H68F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-LL45F6	WO2023185864A1_227-1	.	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCCN(C)CC2(COC3=NC4=C(F)C(C5=CC(O)=CC6=C5C(C5CC5)=C(F)C=C6)=C(F)C=C4C(N4CC5CCC(C4)N5)=N3)CC2)=NO1	C60H67F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-EPWOTA	WO2023185864A1_227-2	.	CC(C)[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCCN(C)CC2(COC3=NC4=C(F)C(C5=CC(O)=CC6=C5C(C5CC5)=C(F)C=C6)=C(F)C=C4C(N4CC5CCC(C4)N5)=N3)CC2)=NO1	C60H67F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-F5KA1S	WO2023185864A1_227	.	CC(C)C(C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCCN(C)CC2(COC3=NC4=C(F)C(C5=CC(O)=CC6=C5C(C5CC5)=C(F)C=C6)=C(F)C=C4C(N4CC5CCC(C4)N5)=N3)CC2)=NO1	C60H67F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-CA8EDR	WO2023185864A1_228-1	.	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCCN(CCCOC2=NC3=C(F)C(C4=CC(O)=CC5=C4C(C4CC4)=C(F)C=C5)=CC=C3C(N3CC4CCC(C3)N4)=N2)C(C)C)=NO1	C60H70F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-8TNN9I	WO2023185864A1_228-2	.	CC(C)[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCCN(CCCOC2=NC3=C(F)C(C4=CC(O)=CC5=C4C(C4CC4)=C(F)C=C5)=CC=C3C(N3CC4CCC(C3)N4)=N2)C(C)C)=NO1	C60H70F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-ROR5T4	WO2023185864A1_228	.	CCN(CCOC1=NOC(C(C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=CC=NN3C)C=C2)C(C)C)=C1)CC1(COC2=NC3=C(F)C(C4=CC(O)=CC5=C4C(C4CC4)=C(F)C=C5)=CC=C3C(N3CC4CCC(C3)N4)=N2)CC1	C61H70F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-SQS2N8	WO2023185864A1_229-1	.	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCCN(CCCOC2=NC3=C(F)C(C4=CC(O)=CC5=C4C(C4CC4)=C(F)C=C5)=C(F)C=C3C(N3CC4CCC(C3)N4)=N2)C(C)C)=NO1	C60H69F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-55XRGI	WO2023185864A1_229-2	.	CC(C)[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCCN(CCCOC2=NC3=C(F)C(C4=CC(O)=CC5=C4C(C4CC4)=C(F)C=C5)=C(F)C=C3C(N3CC4CCC(C3)N4)=N2)C(C)C)=NO1	C60H69F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-KKSLFM	WO2023185864A1_229	.	CC(C)C(C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCCN(CCCOC2=NC3=C(F)C(C4=CC(O)=CC5=C4C(C4CC4)=C(F)C=C5)=C(F)C=C3C(N3CC4CCC(C3)N4)=N2)C(C)C)=NO1	C60H69F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-82YNID	WO2023185864A1_23	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCC45CCCN4C(COC4=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C4)CC5)=NC3=C1F)=CC(O)=C2	C60H67F2N9O7S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-P6A24D	WO2023185864A1_230-1	.	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCCN(CCCOC2=NC3=C(F)C(C4=CC(O)=CC5=C4C(C4CC4)=C(F)C=C5)=CC=C3C(N3CC4CCC(C3)N4)=N2)C2CC2)=NO1	C60H68F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-QIID6O	WO2023185864A1_230-2	.	CC(C)[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCCN(CCCOC2=NC3=C(F)C(C4=CC(O)=CC5=C4C(C4CC4)=C(F)C=C5)=CC=C3C(N3CC4CCC(C3)N4)=N2)C2CC2)=NO1	C60H68F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-UXIZXD	WO2023185864A1_230	.	CC(C)C(C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCCN(CCCOC2=NC3=C(F)C(C4=CC(O)=CC5=C4C(C4CC4)=C(F)C=C5)=CC=C3C(N3CC4CCC(C3)N4)=N2)C2CC2)=NO1	C60H68F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-25INLE	WO2023185864A1_231-1	.	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCCN(CCCOC2=NC3=C(F)C(C4=CC(O)=CC5=C4C(C4CC4)=C(F)C=C5)=C(F)C=C3C(N3CC4CCC(C3)N4)=N2)C2CC2)=NO1	C60H67F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-R5S2O6	WO2023185864A1_231-2	.	CC(C)[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCCN(CCCOC2=NC3=C(F)C(C4=CC(O)=CC5=C4C(C4CC4)=C(F)C=C5)=C(F)C=C3C(N3CC4CCC(C3)N4)=N2)C2CC2)=NO1	C60H67F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-4MEHWV	WO2023185864A1_231	.	CC(C)C(C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCCN(CCCOC2=NC3=C(F)C(C4=CC(O)=CC5=C4C(C4CC4)=C(F)C=C5)=C(F)C=C3C(N3CC4CCC(C3)N4)=N2)C2CC2)=NO1	C60H67F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-NM7LEA	WO2023185864A1_232	.	CC(C)C(C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCCNCC2(COC3=NC4=C(F)C(C5=CC(O)=CC6=C5C(C5CC5)=C(F)C=C6)=CC=C4C(N4CC5CCC(C4)N5)=N3)CC2)=NO1	C59H66F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-82EN1H	WO2023185864A1_236-1	.	CCN(CCOC1=NOC([C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=CC=NN3C)C=C2)C(C)C)=C1)CC1(COC2=NC3=C(F)C(C4=CC(O)=CC5=C4C(C4CC4)=C(F)C=C5)=CC=C3C(N3CC4CCC(C3)N4)=N2)CC1	C61H70F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-T1QLYD	WO2023185864A1_236-2	.	CCN(CCOC1=NOC([C@@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=CC=NN3C)C=C2)C(C)C)=C1)CC1(COC2=NC3=C(F)C(C4=CC(O)=CC5=C4C(C4CC4)=C(F)C=C5)=CC=C3C(N3CC4CCC(C3)N4)=N2)CC1	C61H70F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-5QSBF9	WO2023185864A1_237-1	.	CCN(CCOC1=NOC([C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=CC=NN3C)C=C2)C(C)C)=C1)CC1(COC2=NC3=C(F)C(C4=CC(O)=CC5=C4C(C4CC4)=C(F)C=C5)=C(F)C=C3C(N3CC4CCC(C3)N4)=N2)CC1	C61H69F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-FYHVEJ	WO2023185864A1_237-2	.	CCN(CCOC1=NOC([C@@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=CC=NN3C)C=C2)C(C)C)=C1)CC1(COC2=NC3=C(F)C(C4=CC(O)=CC5=C4C(C4CC4)=C(F)C=C5)=C(F)C=C3C(N3CC4CCC(C3)N4)=N2)CC1	C61H69F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-GA71RF	WO2023185864A1_237	.	CCN(CCOC1=NOC(C(C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=CC=NN3C)C=C2)C(C)C)=C1)CC1(COC2=NC3=C(F)C(C4=CC(O)=CC5=C4C(C4CC4)=C(F)C=C5)=C(F)C=C3C(N3CC4CCC(C3)N4)=N2)CC1	C61H69F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-96HXWL	WO2023185864A1_238-1	.	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCCN(CC2(COC3=NC4=C(F)C(C5=CC(O)=CC6=C5C(C5CC5)=C(F)C=C6)=CC=C4C(N4CC5CCC(C4)N5)=N3)CC2)C(C)C)=NO1	C62H72F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-ZQUI0D	WO2023185864A1_238-2	.	CC(C)[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCCN(CC2(COC3=NC4=C(F)C(C5=CC(O)=CC6=C5C(C5CC5)=C(F)C=C6)=CC=C4C(N4CC5CCC(C4)N5)=N3)CC2)C(C)C)=NO1	C62H72F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-CD7FM1	WO2023185864A1_238	.	CC(C)C(C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCCN(CC2(COC3=NC4=C(F)C(C5=CC(O)=CC6=C5C(C5CC5)=C(F)C=C6)=CC=C4C(N4CC5CCC(C4)N5)=N3)CC2)C(C)C)=NO1	C62H72F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-Q486YQ	WO2023185864A1_239-1	.	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCCN(CC2(COC3=NC4=C(F)C(C5=CC(O)=CC6=C5C(C5CC5)=C(F)C=C6)=C(F)C=C4C(N4CC5CCC(C4)N5)=N3)CC2)C(C)C)=NO1	C62H71F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-OZGCO1	WO2023185864A1_239-2	.	CC(C)[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCCN(CC2(COC3=NC4=C(F)C(C5=CC(O)=CC6=C5C(C5CC5)=C(F)C=C6)=C(F)C=C4C(N4CC5CCC(C4)N5)=N3)CC2)C(C)C)=NO1	C62H71F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-0OZWIR	WO2023185864A1_239	.	CC(C)C(C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCCN(CC2(COC3=NC4=C(F)C(C5=CC(O)=CC6=C5C(C5CC5)=C(F)C=C6)=C(F)C=C4C(N4CC5CCC(C4)N5)=N3)CC2)C(C)C)=NO1	C62H71F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-CF6NLE	WO2023185864A1_24	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCC45CCCN4C(COC4=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C4)CC5)=NC3=C1F)=CC(O)=C2	C60H68F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-IVY6DL	WO2023185864A1_240-1	.	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCCN(CC2(COC3=NC4=C(F)C(C5=CC(O)=CC6=C5C(C5CC5)=C(F)C=C6)=CC=C4C(N4CC5CCC(C4)N5)=N3)CC2)C2CC2)=NO1	C62H70F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-AN9G5P	WO2023185864A1_240-2	.	CC(C)[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCCN(CC2(COC3=NC4=C(F)C(C5=CC(O)=CC6=C5C(C5CC5)=C(F)C=C6)=CC=C4C(N4CC5CCC(C4)N5)=N3)CC2)C2CC2)=NO1	C62H70F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-PI24FL	WO2023185864A1_240	.	CC(C)C(C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCCN(CC2(COC3=NC4=C(F)C(C5=CC(O)=CC6=C5C(C5CC5)=C(F)C=C6)=CC=C4C(N4CC5CCC(C4)N5)=N3)CC2)C2CC2)=NO1	C62H70F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-SFJG6P	WO2023185864A1_241-1	.	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCCN(CC2(COC3=NC4=C(F)C(C5=CC(O)=CC6=C5C(C5CC5)=C(F)C=C6)=C(F)C=C4C(N4CC5CCC(C4)N5)=N3)CC2)C2CC2)=NO1	C62H69F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-I7Q6T4	WO2023185864A1_241-2	.	CC(C)[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCCN(CC2(COC3=NC4=C(F)C(C5=CC(O)=CC6=C5C(C5CC5)=C(F)C=C6)=C(F)C=C4C(N4CC5CCC(C4)N5)=N3)CC2)C2CC2)=NO1	C62H69F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-5NI479	WO2023185864A1_241	.	CC(C)C(C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCCN(CC2(COC3=NC4=C(F)C(C5=CC(O)=CC6=C5C(C5CC5)=C(F)C=C6)=C(F)C=C4C(N4CC5CCC(C4)N5)=N3)CC2)C2CC2)=NO1	C62H69F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-AA81CF	WO2023185864A1_242	.	C#CC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCC45CCCN4C(COC4=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C4)CC5)=NC3=C1F)=CC(O)=C2	C60H63F2N9O7S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-SAUU7K	WO2023185864A1_243	.	C#CC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCC45CCCN4C(COC4=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C4)CC5)=NC3=C1F)=CC(O)=C2	C60H64F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-199BJK	WO2023185864A1_244	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCC45CCCN4C(COC4=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C4)CC5)=NC3=C1F)=CC(O)=C2	C60H66F3N9O7S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-PRDBK4	WO2023185864A1_245	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCC45CCCN4C(COC4=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C4)CC5)=NC3=C1F)=CC(O)=C2	C60H67F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-1L3TSB	WO2023185864A1_246	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCC45CCCN4C(COC4=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C4)CC5)=NC3=C1F)=CC(O)=C2	C60H62F3N9O7S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-PM0D4B	WO2023185864A1_247	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCC45CCCN4C(COC4=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C4)CC5)=NC3=C1F)=CC(O)=C2	C60H63F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-98BV9X	WO2023185864A1_248	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCC45CCCN4C(COC(=O)N4C[C@H](O)C[C@H]4C(=O)N[C@@H](C)C4=CC=C(C6=C(C)N=CS6)C=C4)CC5)=NC3=C1F)=CC(O)=C2	C53H53F3N8O6S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-4W6XO0	WO2023185864A1_249	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCC45CCCN4C(COCCC(=O)N4C[C@H](O)C[C@H]4C(=O)N[C@@H](C)C4=CC=C(C6=C(C)N=CS6)C=C4)CC5)=NC3=C1F)=CC(O)=C2	C55H57F3N8O6S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-RDO6VD	WO2023185864A1_25	.	C#CC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(OCCOC5=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C60H65F2N9O8S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-FC2P4O	WO2023185864A1_250	.	C#CC1=C(F)C=CC2=C1C(C1=NC=C3C(N4CC5CCC(C4)N5)=NC(OCC45CCCN4C(COC4=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C4)CC5)=NC3=C1F)=CC(O)=C2	C59H63F2N11O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-0N8XEP	WO2023185864A1_251	.	CCC1=C(F)C=CC2=C1C(C1=NC=C3C(N4CC5CCC(C4)N5)=NC(OCC45CCCN4C(COC4=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C4)CC5)=NC3=C1F)=CC(O)=C2	C59H67F2N11O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-KHWMCC	WO2023185864A1_252	.	C#CC1=C(F)C=CC2=C1C(C1=NN=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(F)(COC5=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C57H61F3N12O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-T25EHD	WO2023185864A1_253	.	CCC1=C(F)C=CC2=C1C(C1=NN=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(F)(COC5=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C57H65F3N12O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-D9R6Y3	WO2023185864A1_26	.	C#CC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC5(CC4)CN(C4=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C4)C5)=NC3=C1F)=CC(O)=C2	C60H64F2N10O6S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-62JMMP	WO2023185864A1_27	.	C#CC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(F)(COC5=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C59H63F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-51XMTI	WO2023185864A1_28	.	C#CC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(C)(COC5=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C60H65F2N9O7S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-93W038	WO2023185864A1_29	.	C#CC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(OCCOC5=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C60H65F2N9O8S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-G5VJ0C	WO2023185864A1_3	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(COC5=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C59H67F2N9O7S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-J33YAH	WO2023185864A1_30	.	C#CC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC5(CC4)CN(C4=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C4)C5)=NC3=C1F)=CC(O)=C2	C60H64F2N10O6S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-1GUIKN	WO2023185864A1_31	.	C#CC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(F)(COC5=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C59H63F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-A4IPLO	WO2023185864A1_32	.	C#CC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(C)(COC5=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C60H65F2N9O7S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-1Z5STB	WO2023185864A1_33	.	C#CC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(OCCOC5=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C60H65F2N9O8S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-14ZU0Q	WO2023185864A1_34	.	C#CC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC5(CC4)CN(C4=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C4)C5)=NC3=C1F)=CC(O)=C2	C60H64F2N10O6S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-9I3GLF	WO2023185864A1_35	.	C#CC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(F)(COC5=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C59H63F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-SNRKMD	WO2023185864A1_36	.	C#CC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(C)(COC5=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C60H65F2N9O7S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-03VHG5	WO2023185864A1_37	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(OCCOC4CCN(CCOC5=NC6=C(F)C(C7=CC(O)=CC8=C7C(Cl)=C(F)C=C8)=CC=C6C(N6CC7CCC(C6)N7)=N5)CC4)=NO3)C(C)C)C=C2)SC=N1	C58H64ClF2N9O8S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-BNTPFR	WO2023185864A1_38	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CC5(CCN(CCOC6=NC7=C(F)C(C8=CC(O)=CC9=C8C(Cl)=C(F)C=C9)=CC=C7C(N7CC8CCC(C7)N8)=N6)CC5)C4)=NO3)C(C)C)C=C2)SC=N1	C58H63ClF2N10O6S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-0W7YJZ	WO2023185864A1_39	.	CC(C)C(C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCC2(F)CCN(CCOC3=NC4=C(F)C(C5=CC(O)=CC6=C5C(Cl)=C(F)C=C6)=CC=C4C(N4CC5CCC(C4)N5)=N3)CC2)=NO1	C57H62ClF3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-PKPKGM	WO2023185864A1_4	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(F)(COC5=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C59H67F3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-9OPFBQ	WO2023185864A1_40	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(OCC4(C)CCN(CCOC5=NC6=C(F)C(C7=CC(O)=CC8=C7C(Cl)=C(F)C=C8)=CC=C6C(N6CC7CCC(C6)N7)=N5)CC4)=NO3)C(C)C)C=C2)SC=N1	C58H64ClF2N9O7S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-3WIDBM	WO2023185864A1_41	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(OCCOC4CCN(CCOC5=NC6=C(F)C(C7=CC(O)=CC8=C7C(Cl)=C(F)C=C8)=CC=C6C(N6CC7CCC(C6)N7)=N5)CC4)=NO3)C(C)C)C=C2)SC=N1	C58H64ClF2N9O8S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-QMZ4U3	WO2023185864A1_42	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CC5(CCN(CCOC6=NC7=C(F)C(C8=CC(O)=CC9=C8C(Cl)=C(F)C=C9)=CC=C7C(N7CC8CCC(C7)N8)=N6)CC5)C4)=NO3)C(C)C)C=C2)SC=N1	C58H63ClF2N10O6S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-QSQUVY	WO2023185864A1_43	.	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCC2(F)CCN(CCOC3=NC4=C(F)C(C5=CC(O)=CC6=C5C(Cl)=C(F)C=C6)=CC=C4C(N4CC5CCC(C4)N5)=N3)CC2)=NO1	C57H62ClF3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-QOBV2D	WO2023185864A1_44	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(OCC4(C)CCN(CCOC5=NC6=C(F)C(C7=CC(O)=CC8=C7C(Cl)=C(F)C=C8)=CC=C6C(N6CC7CCC(C6)N7)=N5)CC4)=NO3)C(C)C)C=C2)SC=N1	C58H64ClF2N9O7S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-L43NP4	WO2023185864A1_45	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3=CC(OCCOC4CCN(CCOC5=NC6=C(F)C(C7=CC(O)=CC8=C7C(Cl)=C(F)C=C8)=CC=C6C(N6CC7CCC(C6)N7)=N5)CC4)=NO3)C(C)C)C=C2)SC=N1	C58H64ClF2N9O8S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-1K7VYN	WO2023185864A1_46	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3=CC(N4CC5(CCN(CCOC6=NC7=C(F)C(C8=CC(O)=CC9=C8C(Cl)=C(F)C=C9)=CC=C7C(N7CC8CCC(C7)N8)=N6)CC5)C4)=NO3)C(C)C)C=C2)SC=N1	C58H63ClF2N10O6S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-HIC2HH	WO2023185864A1_47	.	CC(C)[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCC2(F)CCN(CCOC3=NC4=C(F)C(C5=CC(O)=CC6=C5C(Cl)=C(F)C=C6)=CC=C4C(N4CC5CCC(C4)N5)=N3)CC2)=NO1	C57H62ClF3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-AMQVF4	WO2023185864A1_48	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3=CC(OCC4(C)CCN(CCOC5=NC6=C(F)C(C7=CC(O)=CC8=C7C(Cl)=C(F)C=C8)=CC=C6C(N6CC7CCC(C6)N7)=N5)CC4)=NO3)C(C)C)C=C2)SC=N1	C58H64ClF2N9O7S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-PRWOKY	WO2023185864A1_49	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(OCCOC4CCN(CCOC5=NC6=C(F)C(C7=CC(O)=CC(Cl)=C7C7CC7)=CC=C6C(N6CC7CCC(C6)N7)=N5)CC4)=NO3)C(C)C)C=C2)SC=N1	C57H67ClFN9O8S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-ZP71MA	WO2023185864A1_5	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(C)(COC5=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C60H69F2N9O7S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-MQ9IBV	WO2023185864A1_50	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CC5(CCN(CCOC6=NC7=C(F)C(C8=CC(O)=CC(Cl)=C8C8CC8)=CC=C7C(N7CC8CCC(C7)N8)=N6)CC5)C4)=NO3)C(C)C)C=C2)SC=N1	C57H66ClFN10O6S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-D6VG1U	WO2023185864A1_51	.	CC(C)C(C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCC2(F)CCN(CCOC3=NC4=C(F)C(C5=CC(O)=CC(Cl)=C5C5CC5)=CC=C4C(N4CC5CCC(C4)N5)=N3)CC2)=NO1	C56H65ClF2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-6H5PQB	WO2023185864A1_52	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(OCC4(C)CCN(CCOC5=NC6=C(F)C(C7=CC(O)=CC(Cl)=C7C7CC7)=CC=C6C(N6CC7CCC(C6)N7)=N5)CC4)=NO3)C(C)C)C=C2)SC=N1	C57H67ClFN9O7S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-ZLAE68	WO2023185864A1_53	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(OCCOC4CCN(CCOC5=NC6=C(F)C(C7=CC(O)=CC(Cl)=C7C7CC7)=CC=C6C(N6CC7CCC(C6)N7)=N5)CC4)=NO3)C(C)C)C=C2)SC=N1	C57H67ClFN9O8S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-QBK74V	WO2023185864A1_54	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CC5(CCN(CCOC6=NC7=C(F)C(C8=CC(O)=CC(Cl)=C8C8CC8)=CC=C7C(N7CC8CCC(C7)N8)=N6)CC5)C4)=NO3)C(C)C)C=C2)SC=N1	C57H66ClFN10O6S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-TXJ26X	WO2023185864A1_55	.	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCC2(F)CCN(CCOC3=NC4=C(F)C(C5=CC(O)=CC(Cl)=C5C5CC5)=CC=C4C(N4CC5CCC(C4)N5)=N3)CC2)=NO1	C56H65ClF2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-GIEUR0	WO2023185864A1_56	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(OCC4(C)CCN(CCOC5=NC6=C(F)C(C7=CC(O)=CC(Cl)=C7C7CC7)=CC=C6C(N6CC7CCC(C6)N7)=N5)CC4)=NO3)C(C)C)C=C2)SC=N1	C57H67ClFN9O7S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-A7ZIP8	WO2023185864A1_57	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3=CC(OCCOC4CCN(CCOC5=NC6=C(F)C(C7=CC(O)=CC(Cl)=C7C7CC7)=CC=C6C(N6CC7CCC(C6)N7)=N5)CC4)=NO3)C(C)C)C=C2)SC=N1	C57H67ClFN9O8S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-51FB5Y	WO2023185864A1_58	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3=CC(N4CC5(CCN(CCOC6=NC7=C(F)C(C8=CC(O)=CC(Cl)=C8C8CC8)=CC=C7C(N7CC8CCC(C7)N8)=N6)CC5)C4)=NO3)C(C)C)C=C2)SC=N1	C57H66ClFN10O6S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-RUY1BO	WO2023185864A1_59	.	CC(C)[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCC2(F)CCN(CCOC3=NC4=C(F)C(C5=CC(O)=CC(Cl)=C5C5CC5)=CC=C4C(N4CC5CCC(C4)N5)=N3)CC2)=NO1	C56H65ClF2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-59YIW0	WO2023185864A1_6	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCC45CCCN4C(COCCOC4=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C4)CC5)=NC3=C1F)=CC(O)=C2	C62H71F2N9O8S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-AIUI1A	WO2023185864A1_60	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3=CC(OCC4(C)CCN(CCOC5=NC6=C(F)C(C7=CC(O)=CC(Cl)=C7C7CC7)=CC=C6C(N6CC7CCC(C6)N7)=N5)CC4)=NO3)C(C)C)C=C2)SC=N1	C57H67ClFN9O7S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-JWMI8C	WO2023185864A1_61	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(OCCOC5=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C60H64F3N9O8S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-FKM149	WO2023185864A1_62	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC5(CC4)CN(C4=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C4)C5)=NC3=C1F)=CC(O)=C2	C60H63F3N10O6S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-MCTUFI	WO2023185864A1_63	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(F)(COC5=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C59H62F4N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-ZEY4LG	WO2023185864A1_64	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(C)(COC5=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C60H64F3N9O7S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-LDFMRV	WO2023185864A1_65	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(OCCOC5=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C60H64F3N9O8S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-LYU1O5	WO2023185864A1_66	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC5(CC4)CN(C4=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C4)C5)=NC3=C1F)=CC(O)=C2	C60H63F3N10O6S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-3CYAL2	WO2023185864A1_67	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(F)(COC5=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C59H62F4N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-3FHAC9	WO2023185864A1_68	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(C)(COC5=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C60H64F3N9O7S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-RVZVZO	WO2023185864A1_69	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(OCCOC5=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C60H64F3N9O8S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-KO2LDS	WO2023185864A1_7	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCC45CCCN4C(COC4=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C4)CC5)=NC3=C1F)=CC(O)=C2	C60H67F2N9O7S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-VE7YBY	WO2023185864A1_70	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC5(CC4)CN(C4=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C4)C5)=NC3=C1F)=CC(O)=C2	C60H63F3N10O6S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-TKE19X	WO2023185864A1_71	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(F)(COC5=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C59H62F4N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-UOJZP6	WO2023185864A1_72	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(C)(COC5=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C60H64F3N9O7S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-0R8QAX	WO2023185864A1_73	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(OCCOC5=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C60H68F3N9O8S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-P9US0D	WO2023185864A1_74	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC5(CC4)CN(C4=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C4)C5)=NC3=C1F)=CC(O)=C2	C60H67F3N10O6S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-Y3X40D	WO2023185864A1_75	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(F)(COC5=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C59H66F4N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-TA8OQ5	WO2023185864A1_76	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(C)(COC5=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C60H68F3N9O7S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-S0OMH5	WO2023185864A1_77	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(OCCOC5=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C60H68F3N9O8S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-S611ZB	WO2023185864A1_78	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC5(CC4)CN(C4=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C4)C5)=NC3=C1F)=CC(O)=C2	C60H67F3N10O6S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-UZ4EV6	WO2023185864A1_79	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(F)(COC5=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C59H66F4N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-SUSRB7	WO2023185864A1_8	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCC45CCCN4C(COC4=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C4)CC5)=NC3=C1F)=CC(O)=C2	C60H68F2N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-4KEPW1	WO2023185864A1_80	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(C)(COC5=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C60H68F3N9O7S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-SBZNCU	WO2023185864A1_81	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(OCCOC5=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C60H68F3N9O8S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-FMK58A	WO2023185864A1_82	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC5(CC4)CN(C4=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C4)C5)=NC3=C1F)=CC(O)=C2	C60H67F3N10O6S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-B7YXNO	WO2023185864A1_83	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(F)(COC5=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=CC=NN7C)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C59H66F4N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-SXMW44	WO2023185864A1_84	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(C)(COC5=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C60H68F3N9O7S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-CRYOSC	WO2023185864A1_85	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(OCCOC4CCN(CCOC5=NC6=C(F)C(C7=CC(O)=CC8=C7C(Cl)=C(F)C=C8)=C(F)C=C6C(N6CC7CCC(C6)N7)=N5)CC4)=NO3)C(C)C)C=C2)SC=N1	C58H63ClF3N9O8S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-3HR2Z5	WO2023185864A1_86	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CC5(CCN(CCOC6=NC7=C(F)C(C8=CC(O)=CC9=C8C(Cl)=C(F)C=C9)=C(F)C=C7C(N7CC8CCC(C7)N8)=N6)CC5)C4)=NO3)C(C)C)C=C2)SC=N1	C58H62ClF3N10O6S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-KMPMG9	WO2023185864A1_87	.	CC(C)C(C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCC2(F)CCN(CCOC3=NC4=C(F)C(C5=CC(O)=CC6=C5C(Cl)=C(F)C=C6)=C(F)C=C4C(N4CC5CCC(C4)N5)=N3)CC2)=NO1	C57H61ClF4N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-HQUHA7	WO2023185864A1_88	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(OCC4(C)CCN(CCOC5=NC6=C(F)C(C7=CC(O)=CC8=C7C(Cl)=C(F)C=C8)=C(F)C=C6C(N6CC7CCC(C6)N7)=N5)CC4)=NO3)C(C)C)C=C2)SC=N1	C58H63ClF3N9O7S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-YUKN2W	WO2023185864A1_89	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(OCCOC4CCN(CCOC5=NC6=C(F)C(C7=CC(O)=CC8=C7C(Cl)=C(F)C=C8)=C(F)C=C6C(N6CC7CCC(C6)N7)=N5)CC4)=NO3)C(C)C)C=C2)SC=N1	C58H63ClF3N9O8S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-VY5W9B	WO2023185864A1_9	.	CCC1=C(F)C=CC2=C1C(C1=CC=C3C(N4CC5CCC(C4)N5)=NC(OCCN4CCC(OCCOC5=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C5)CC4)=NC3=C1F)=CC(O)=C2	C60H69F2N9O8S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-DEADZL	WO2023185864A1_90	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CC5(CCN(CCOC6=NC7=C(F)C(C8=CC(O)=CC9=C8C(Cl)=C(F)C=C9)=C(F)C=C7C(N7CC8CCC(C7)N8)=N6)CC5)C4)=NO3)C(C)C)C=C2)SC=N1	C58H62ClF3N10O6S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-HBAEAK	WO2023185864A1_91	.	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCC2(F)CCN(CCOC3=NC4=C(F)C(C5=CC(O)=CC6=C5C(Cl)=C(F)C=C6)=C(F)C=C4C(N4CC5CCC(C4)N5)=N3)CC2)=NO1	C57H61ClF4N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-M1VYNH	WO2023185864A1_92	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(OCC4(C)CCN(CCOC5=NC6=C(F)C(C7=CC(O)=CC8=C7C(Cl)=C(F)C=C8)=C(F)C=C6C(N6CC7CCC(C6)N7)=N5)CC4)=NO3)C(C)C)C=C2)SC=N1	C58H63ClF3N9O7S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-9AH9MK	WO2023185864A1_93	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3=CC(OCCOC4CCN(CCOC5=NC6=C(F)C(C7=CC(O)=CC8=C7C(Cl)=C(F)C=C8)=C(F)C=C6C(N6CC7CCC(C6)N7)=N5)CC4)=NO3)C(C)C)C=C2)SC=N1	C58H63ClF3N9O8S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-7KPKNJ	WO2023185864A1_94	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3=CC(N4CC5(CCN(CCOC6=NC7=C(F)C(C8=CC(O)=CC9=C8C(Cl)=C(F)C=C9)=C(F)C=C7C(N7CC8CCC(C7)N8)=N6)CC5)C4)=NO3)C(C)C)C=C2)SC=N1	C58H62ClF3N10O6S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-QM8JGZ	WO2023185864A1_95	.	CC(C)[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCC2(F)CCN(CCOC3=NC4=C(F)C(C5=CC(O)=CC6=C5C(Cl)=C(F)C=C6)=C(F)C=C4C(N4CC5CCC(C4)N5)=N3)CC2)=NO1	C57H61ClF4N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-FMLHE9	WO2023185864A1_96	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3=CC(OCC4(C)CCN(CCOC5=NC6=C(F)C(C7=CC(O)=CC8=C7C(Cl)=C(F)C=C8)=C(F)C=C6C(N6CC7CCC(C6)N7)=N5)CC4)=NO3)C(C)C)C=C2)SC=N1	C58H63ClF3N9O7S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-IWQCI5	WO2023185864A1_97	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(OCCOC4CCN(CCOC5=NC6=C(F)C(C7=CC(O)=CC(Cl)=C7C7CC7)=C(F)C=C6C(N6CC7CCC(C6)N7)=N5)CC4)=NO3)C(C)C)C=C2)SC=N1	C57H66ClF2N9O8S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-BM0HWV	WO2023185864A1_98	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CC5(CCN(CCOC6=NC7=C(F)C(C8=CC(O)=CC(Cl)=C8C8CC8)=C(F)C=C7C(N7CC8CCC(C7)N8)=N6)CC5)C4)=NO3)C(C)C)C=C2)SC=N1	C57H65ClF2N10O6S	KRAS	P01116	VHL	WO-2023185864-A1
TPD-JOKGCB	WO2023185864A1_99	.	CC(C)C(C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CC=NN2C)C=C1)C1=CC(OCC2(F)CCN(CCOC3=NC4=C(F)C(C5=CC(O)=CC(Cl)=C5C5CC5)=C(F)C=C4C(N4CC5CCC(C4)N5)=N3)CC2)=NO1	C56H64ClF3N10O7	KRAS	P01116	VHL	WO-2023185864-A1
TPD-AUEVB5	SCHEMBL26110070	N-[4-[5-[6-(5-cyanoindol-1-yl)-4-(methylamino)pyridin-3-yl]-1,3,4-thiadiazol-2-yl]cyclohexyl]-2-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]acetamide; SCHEMBL26110076	CNC1=CC(N2C=CC3=C2C=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](NC(=O)CN3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)S1	C42H41N11O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-OB631U	SCHEMBL26111270	N-[4-[5-[6-(5-cyanopyrrolo[2,3-b]pyridin-1-yl)-4-(methylamino)pyridin-3-yl]-1,3,4-thiadiazol-2-yl]cyclohexyl]-2-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]acetamide; SCHEMBL26111275; SCHEMBL30569050	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](NC(=O)CN3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)S1	C41H40N12O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-H79607	SCHEMBL26112124	N-[4-[5-[6-(5-cyanopyrazolo[3,4-b]pyridin-1-yl)-4-(methylamino)pyridin-3-yl]-1,3,4-thiadiazol-2-yl]cyclohexyl]-2-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]acetamide; SCHEMBL26112127; SCHEMBL30569132	CNC1=CC(N2N=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](NC(=O)CN3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)S1	C40H39N13O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-G55UC3	SCHEMBL26109183	N-[3-[5-[6-(5-cyanopyrrolo[2,3-b]pyridin-1-yl)-4-(methylamino)pyridin-3-yl]-1,3,4-thiadiazol-2-yl]cyclobutyl]-2-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]acetamide; SCHEMBL26109186; SCHEMBL30569093	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2C[C@H](NC(=O)CN3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)C2)S1	C39H36N12O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-R46XZD	WO2023186069A1_5	.	CNC1=CC(N2C=CC3=C2N=CN=C3)=NC=C1C1=NN=C([C@H]2C[C@H](NC(=O)CN3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)C2)S1	C37H36N12O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-S1B05E	WO2023186069A1_6	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](NC(=O)CN3CCN(C4=CC=CC(N5CCC(=O)NC5=O)=C4)CC3)CC2)S1	C38H40N12O3S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-VC3FO3	SCHEMBL26111125	N-[4-[5-[6-(3-cyanopyrrolo[1,2-b]pyridazin-7-yl)-4-(methylamino)pyridin-3-yl]-1,3,4-thiadiazol-2-yl]cyclohexyl]-2-[8-(2,4-dioxo-1,3-diazinan-1-yl)-2,4,4a,5-tetrahydro-1H-pyrazino[2,1-c][1,4]benzoxazin-3-yl]acetamide	CNC1=CC(C2=CC=C3C=C(C#N)C=NN32)=NC=C1C1=NN=C([C@H]2CC[C@H](NC(=O)CN3CCN4C5=C(C=C(N6CCC(=O)NC6=O)C=C5)OCC4C3)CC2)S1	C39H40N12O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-OOCOQA	SCHEMBL26110625	N-[4-[5-[6-(5-cyanopyrrolo[2,3-b]pyridin-1-yl)-4-(methylamino)pyridin-3-yl]-1,3,4-thiadiazol-2-yl]cyclohexyl]-2-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperazin-1-yl]acetamide; SCHEMBL26110630; SCHEMBL30569053	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](NC(=O)CN3CCN(C4=CC=C(N5CCC(=O)NC5=O)C=C4)CC3)CC2)S1	C38H40N12O3S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-IKGLY6	WO2023186069A1_9	.	CNC1=CC(N2CCC3=C2C=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](NC(=O)CN3CCN(C4=CC=C(N5CCC(=O)NC5=O)C=C4)CC3)CC2)S1	C39H43N11O3S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-GJLVWA	WO2023186069A1_10	.	CNC1=CC(N2CCC3=C2N=CC(C#N)=C3)=NC=C1C1=CN=C([C@H]2CC[C@H](NC(=O)CN3CCN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)S1	C42H43N11O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-64CL3V	SCHEMBL26110573	N-[4-[5-[6-(5-cyanopyrrolo[2,3-b]pyridin-1-yl)-4-(methylamino)pyridin-3-yl]-1,3,4-thiadiazol-2-yl]cyclohexyl]-2-[4-[5-(2,4-dioxo-1,3-diazinan-1-yl)pyridin-2-yl]piperazin-1-yl]acetamide; SCHEMBL26110577; SCHEMBL30569038	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](NC(=O)CN3CCN(C4=NC=C(N5CCC(=O)NC5=O)C=C4)CC3)CC2)S1	C37H39N13O3S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-TITJYU	WO2023186069A1_12	.	CNC1=CC(N2CCC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C(C2CC3(C2)CN(C(=O)CN2CCN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC2)C3)S1	C41H40N12O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-69M8HQ	WO2023186069A1_13	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](NC(=O)CN3CCN(C4=C(F)C=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)S1	C41H39FN12O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-71WOH1	WO2023186069A1_14	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](NC(=O)N3CC4(CC(CCNC5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)C4)C3)CC2)S1	C44H44N12O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-AMNTPI	WO2023186069A1_15	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=CN=C(N2CCC(NC(=O)CN3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)S1	C41H40N12O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-ITH54Q	SCHEMBL26111651	N-[4-[5-[6-(5-cyanopyrrolo[2,3-b]pyridin-1-yl)-4-(methylamino)pyridin-3-yl]-1,3,4-thiadiazol-2-yl]cyclohexyl]-1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperidine-4-carboxamide; SCHEMBL30569092	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](NC(=O)C3CCN(C4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)CC2)S1	C41H39N11O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-AG1JC1	SCHEMBL26110285	N-[4-[5-[6-(5-cyanopyrrolo[2,3-b]pyridin-1-yl)-4-(methylamino)pyridin-3-yl]-1,3,4-thiadiazol-2-yl]cyclohexyl]-1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidine-4-carboxamide; SCHEMBL26110289; SCHEMBL30569131	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](NC(=O)C3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)S1	C41H39N11O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-C15TM2	WO2023186069A1_18	.	CC(C)NC1=CC(C2=C3N=CC(C#N)=CN3N=C2)=NC=C1C1=NN=C(N2CCN(C(=O)C3CCN(CC4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)S1	C41H41N13O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-33RYXD	WO2023186069A1_19	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C(C2CCN(C(=O)C3CCN(CC4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)S1	C41H39N11O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-MR7DAW	WO2023186069A1_20	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C(C2CCN(C(=O)C3CCN(CC4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)C2)S1	C40H37N11O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-95RXV9	WO2023186069A1_21	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C(C2CN(C(=O)C3CCN(CC4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)C2)S1	C39H35N11O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-HM4NO8	WO2023186069A1_22	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=CN=C([C@H]2CC[C@H](NC(=O)CN3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)S1	C42H41N11O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-1JVJ2E	WO2023186069A1_23	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=CN=C(C2CC3(C2)CN(C(=O)CN2CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC2)C3)S1	C42H39N11O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-HS9SSZ	WO2023186069A1_24	.	CNC1=CC(N2C=CC3=C2N=CC(C(N)=O)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](NC(=O)CN3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)S1	C41H42N12O6S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-RY8WUI	WO2023186069A1_25	.	CNC1=CC(N2C=NC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](NC(=O)CN3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)S1	C40H39N13O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-2KHBIQ	WO2023186069A1_26	.	CNC1=CC(C2=CN=C3C=C(C#N)C=NN23)=NC=C1C1=NN=C([C@H]2CC[C@H](NC(=O)CN3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)S1	C40H39N13O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-67NN4K	WO2023186069A1_27	.	CC(C)NC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C(N2CCN(C(=O)C3CCN(CC4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)S1	C42H42N12O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-MDEWGH	WO2023186069A1_28	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C(N2CCN(C3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)S1	C38H36N12O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-S3RVVT	WO2023186069A1_29	.	CNC1=CC(N2C=CC3=C2N=C(N)C(C(N)=O)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](NC(=O)CN3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)S1	C41H43N13O6S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-6802PU	WO2023186069A1_30	.	CNC1=CC(N2C=CC3=C2N=CN=C3)=NC=C1C1=NN=C([C@H]2C[C@H](NC(=O)CN3CCN(C4=C(F)C=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)C2)S1	C37H35FN12O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-5CLO3R	WO2023186069A1_31	.	CNC1=CC(C2=C3N=CC(C#N)=CN3N=C2)=NC=C1C1=NN=C([C@H]2CC[C@H](NC(=O)CN3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)S1	C40H39N13O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-ODN4HV	WO2023186069A1_32	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C(N2CCC3(CCN(C(=O)C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)S1	C39H35N11O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-ZG1C69	WO2023186069A1_33	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C(C2CC3(C2)CN(C(=O)C2=CC=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C2)C3)S1	C36H28N10O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-3MTC2U	WO2023186069A1_34	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C(C2CC3(C2)CN(C(=O)CN2CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC2)C3)S1	C41H38N12O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-Z590GY	WO2023186069A1_35	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](NC(=O)CN3CCN(C4=CC=C5C6=C4C=CC=C6C(=O)N5C4CCC(=O)NC4=O)CC3)CC2)S1	C44H42N12O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-0CRKS1	WO2023186069A1_36	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C(N2CCN(C(=O)C3CCN(CC4=CC=C5C6=C4C=CC=C6C(=O)N5C4CCC(=O)NC4=O)CC3)CC2)S1	C43H40N12O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-H8W9EY	WO2023186069A1_38	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](NC(=O)N3CCC(OCC#CC4=CC=C5C6=C4C=CC=C6C(=O)N5C4CCC(=O)NC4=O)CC3)CC2)S1	C47H43N11O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-6X71T2	WO2023186069A1_39	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](NC(=O)CN3CCN4C5=C(C=C(N6CCC(=O)NC6=O)C=C5)OCC4C3)CC2)S1	C39H40N12O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-GQ63T0	WO2023186069A1_40	.	CNC1=CC(C2=C3N=CC(C#N)=CN3N=C2)=NC=C1C1=NN=C([C@H]2CC[C@H](NC(=O)CN3CCN4C5=C(C=C(N6CCC(=O)NC6=O)C=C5)OCC4C3)CC2)S1	C38H39N13O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-UDF0C3	WO2023186069A1_41	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](NC(=O)CN3CCN(C4=CC=C5N=CC6=C(C5=C4)N(C4CCC(=O)NC4=O)C(=O)N6C)CC3)CC2)S1	C44H44N14O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-4H83SC	WO2023186069A1_42	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](NC(=O)CN3CCN(C4=CC=C5N=CC6=C(C5=C4)N(C)C(=O)N6C4CCC(=O)NC4=O)CC3)CC2)S1	C44H44N14O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-065KCZ	WO2023186069A1_43	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](NC(=O)CN3CCN(C4=C5C=CC6=C(C5=CC=C4)C(C4CCC(=O)NC4=O)=NO6)CC3)CC2)S1	C44H42N12O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-MRPO0J	WO2023186069A1_44	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](NC(=O)CN3CCN(C4=CC=C(N5N=CC(=O)NC5=O)C=C4)CC3)CC2)S1	C37H37N13O3S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-WRL5Q1	WO2023186069A1_45	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](NC(=O)CN3CCN(C4=C5OCOC5=C(N5CCC(=O)NC5=O)C=C4)CC3)CC2)S1	C39H40N12O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-SQZAJU	WO2023186069A1_47	.	CC(C)NC1=CC(C2=C3N=CC(C#N)=CN3N=C2)=NC=C1C1=NN=C(N2CCN(C(=O)C3CCN(C4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)CC2)S1	C40H39N13O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-BE7WOH	SCHEMBL26110785	N-[4-[5-[6-(5-cyanopyrrolo[2,3-b]pyridin-1-yl)-4-(methylamino)pyridin-3-yl]-1,3,4-thiadiazol-2-yl]cyclohexyl]-2-[4-[3-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-4-yl]prop-2-ynoxy]piperidin-1-yl]acetamide; SCHEMBL26110791; SCHEMBL30569065	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](NC(=O)CN3CCC(OCC#CC4=CC=CC5=C4N(C)C(=O)N5C4CCC(=O)NC4=O)CC3)CC2)S1	C45H46N12O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-ZL3BRW	WO2023186069A1_50	1-[5-[5-[2-[2-[4-[2-(2,6-Dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]acetyl]-2-azaspiro[3.3]heptan-6-yl]-1,3,4-thiadiazol-2-yl]-4-(methylamino)pyridin-2-yl]pyrrolo[2,3-b]pyridine-5-carbonitrile	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C(C2CC3(C2)CN(C(=O)CN2CCN(C4=CC5=C(C=C4F)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC2)C3)S1	C41H37FN12O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-QCOFHR	WO2023186069A1_51	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](NC(=O)CN3CCN(C(=O)C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)S1	C42H40N12O6S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-W189JT	SCHEMBL26109359	N-[4-[5-[6-(5-cyanopyrrolo[2,3-b]pyridin-1-yl)-4-(methylamino)pyridin-3-yl]-1,3,4-thiadiazol-2-yl]cyclohexyl]-2-[7-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-2,7-diazaspiro[3.5]nonan-2-yl]acetamide; SCHEMBL30569049	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](NC(=O)CN3CC4(CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)C3)CC2)S1	C44H44N12O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-2YZNY1	WO2023186069A1_53	.	CNC1=C(C2=NN=C(C3CCN(C(=O)CN4CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)S2)C=NC(N2C=CC3=C2N=CC(C#N)=C3)=C1	C40H38N12O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-H0AK6J	SCHEMBL26136006	N-[4-[5-[6-(5-cyanopyrrolo[2,3-b]pyridin-1-yl)-4-(methylamino)pyridin-3-yl]-1,3,4-thiadiazol-2-yl]cyclohexyl]-4-[3-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-4-yl]prop-2-ynoxy]piperidine-1-carboxamide; SCHEMBL26136009	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](NC(=O)N3CCC(OCC#CC4=CC=CC5=C4N(C)C(=O)N5C4CCC(=O)NC4=O)CC3)CC2)S1	C44H44N12O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-Z3MPCO	WO2023186069A1_55	.	CNC1=C(C2=CN=C(N3CCN(C(=O)C4CCN(C(=O)CN5CCN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)CC3)S2)C=NC(N2C=CC3=C2N=CC(C#N)=C3)=C1	C46H47N13O6S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-QZ5NO6	WO2023186069A1_56	.	CNC1=CC(N2CCC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C(C2CC3(C2)CN(C(=O)CN2CCN(C4=CC5=C(C=C4F)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC2)C3)S1	C41H39FN12O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-749VXJ	WO2023186069A1_57	.	CNC1=C(C2=NN=C(C3CCN(C(=O)CN4CCN(C5=CC6=C(C=C5F)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)S2)C=NC(N2C=CC3=C2N=CC(C#N)=C3)=C1	C40H37FN12O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-00UU6K	WO2023186069A1_58	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](NC(=O)C3CCN(C(=O)C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)S1	C42H39N11O6S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-OZAPYP	WO2023186069A1_59	.	CNC1=C(C2=NN=C(C3CCN(C(=O)CN4CCN(C5=NC=C(N6CCC(=O)NC6=O)C=C5)CC4)CC3)S2)C=NC(N2C=CC3=C2N=CC(C#N)=C3)=C1	C36H37N13O3S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-2GWWJJ	SCHEMBL26111395	1-[5-[5-[1-[2-[4-[[1-(2,6-Dioxopiperidin-3-yl)-2-oxobenzo[cd]indol-6-yl]methyl]piperazin-1-yl]acetyl]piperidin-4-yl]-1,3,4-thiadiazol-2-yl]-4-(methylamino)pyridin-2-yl]pyrrolo[2,3-b]pyridine-5-carbonitrile; SCHEMBL30569005	CNC1=C(C2=NN=C(C3CCN(C(=O)CN4CCN(CC5=C6C=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=C76)C=C5)CC4)CC3)S2)C=NC(N2C=CC3=C2N=CC(C#N)=C3)=C1	C44H42N12O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-2M0KZ5	WO2023186069A1_61	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](NCC3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)S1	C41H41N11O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-UKTJUU	WO2023186069A1_62	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](NC(=O)CN3CCN(C(=O)C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)CC5=C4)CC3)CC2)S1	C42H42N12O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-7ZRCH9	WO2023186069A1_63	.	CNC1=C(C2=NN=C(C3CCN(C(=O)C4CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)S2)C=NC(N2C=CC3=C2N=CC(C#N)=C3)=C1	C40H37N11O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-OSOQGN	WO2023186069A1_64	.	CNC1=C(C2=NN=C(C3CCN(CC4CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)S2)C=NC(N2C=CC3=C2N=CC(C#N)=C3)=C1	C40H39N11O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-M51XQN	WO2023186069A1_65	.	CNC1=CC(N2C=CC3=C2N=CC(N=O)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](NCC3CCN(C4=C(F)C=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)S1	C40H40FN11O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-UJI554	WO2023186069A1_66	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](NC(=O)CN3CCC4(CC3)CN(C3=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C3)C4)CC2)S1	C44H44N12O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-C09QU0	WO2023186069A1_67	.	CNC1=CC(N2C=CC3=C2N=CN=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](NC(=O)CN3CCC4(CC3)CN(C3=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C3)C4)CC2)S1	C42H44N12O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-3K46VR	WO2023186069A1_68	1-[5-[5-[1-[2-[4-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]acetyl]azetidin-3-yl]-1,3,4-thiadiazol-2-yl]-4-(methylamino)pyridin-2-yl]pyrrolo[2,3-b]pyridine-5-carbonitrile	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C(C2CN(C(=O)CN3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)C2)S1	C38H34N12O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-091OOY	SCHEMBL26112821	N-[4-[5-[6-(5-cyanopyrrolo[2,3-b]pyridin-1-yl)-4-(methylamino)pyridin-3-yl]-1,3,4-thiadiazol-2-yl]cyclohexyl]-1-[[1-(2,6-dioxopiperidin-3-yl)-2-oxobenzo[cd]indol-6-yl]methyl]piperidine-4-carboxamide; SCHEMBL26112825; SCHEMBL30569066	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](NC(=O)C3CCN(CC4=CC=C5C6=C4C=CC=C6C(=O)N5C4CCC(=O)NC4=O)CC3)CC2)S1	C45H43N11O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-ULLQ0J	WO2023186069A1_70	1-[5-[5-[4-[4-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindole-5-carbonyl]piperazin-1-yl]piperidin-1-yl]-1,3,4-thiadiazol-2-yl]-4-(methylamino)pyridin-2-yl]pyrrolo[2,3-b]pyridine-5-carbonitrile	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C(N2CCC(N3CCN(C(=O)C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)S1	C39H36N12O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-HQOU16	SCHEMBL26133555	N-[4-[5-[6-(5-cyanopyrrolo[2,3-b]pyridin-1-yl)-4-(methylamino)pyridin-3-yl]-1,3,4-thiadiazol-2-yl]cyclohexyl]-2-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]acetyl]piperazin-1-yl]acetamide; SCHEMBL26133557	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C(C2CCC(NC(=O)CN3CCN(C(=O)CC4=CC=C5C(=O)N(C6CCC(=O)NC6=O)CC5=C4)CC3)CC2)S1	C43H44N12O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-QBS0OS	WO2023186069A1_72	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C(C2CN(C(=O)CN3CCN(C(=O)C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)C2)S1	C39H34N12O6S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-HBJOLX	WO2023186069A1_73	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C(C2CN(C(=O)CN3CCN(C(=O)C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)CC5=C4)CC3)C2)S1	C39H36N12O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-TKBKNH	SCHEMBL26114923	1-[5-[5-[7-[2-[4-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]acetyl]-2,7-diazaspiro[3.5]nonan-2-yl]-1,3,4-thiadiazol-2-yl]-4-(methylamino)pyridin-2-yl]pyrrolo[2,3-b]pyridine-5-carbonitrile; SCHEMBL30569127	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C(N2CC3(CCN(C(=O)CN4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)C2)S1	C42H41N13O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-0XILTJ	WO2023186069A1_75	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](NCC3CCN(C(=O)C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)S1	C42H41N11O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-VJ2EYM	WO2023186069A1_76	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](NCC3CCN(C(=O)C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)CC5=C4)CC3)CC2)S1	C42H43N11O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-CRCNJO	WO2023186069A1_77	.	CNC1=C(C2=NN=C(C3CCN(C(=O)C4CCN(CC#CC5=CC=C6C(=O)N(C7CCC(=O)NC7=O)CC6=C5)CC4)CC3)S2)C=NC(N2C=CC3=C2N=CC(C#N)=C3)=C1	C43H41N11O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-FN11FF	WO2023186069A1_78	.	CNC1=C(C2=NN=C([C@H]3CC[C@H](NC(=O)C4CCN(CC#CC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6)CC4)CC3)S2)C=NC(N2C=CC3=C2C=CC(C#N)=C3)=C1	C45H44N10O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-PMJ9XF	WO2023186069A1_79	.	CNC1=C(C2=NN=C(C3CCN(CC4CCN(C5=C(F)C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)S2)C=NC(N2C=CC3=C2N=CC(C#N)=C3)=C1	C40H38FN11O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-G3PCH6	SCHEMBL30569121	1-[5-[5-[1-[[1-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]azetidin-3-yl]-1,3,4-thiadiazol-2-yl]-4-(methylamino)pyridin-2-yl]pyrrolo[2,3-b]pyridine-5-carbonitrile	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C(C2CN(CC3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)C2)S1	C38H35N11O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-1VAOXL	WO2023186069A1_81	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C(C2CN(CC3CCN(C4=CC=CC5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)C2)S1	C38H35N11O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-SHA66D	WO2023186069A1_82	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](NC(=O)CN3CCN4C5=C(C=C(N6CCC(=O)NC6=O)C=C5)OC[C@@H]4C3)CC2)S1	C39H40N12O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-7JNQYW	SCHEMBL26111463	2-[(4aR)-8-(2,4-dioxo-1,3-diazinan-1-yl)-2,4,4a,5-tetrahydro-1H-pyrazino[2,1-c][1,4]benzoxazin-3-yl]-N-[4-[5-[6-(5-cyanopyrrolo[2,3-b]pyridin-1-yl)-4-(methylamino)pyridin-3-yl]-1,3,4-thiadiazol-2-yl]cyclohexyl]acetamide	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](NC(=O)CN3CCN4C5=C(C=C(N6CCC(=O)NC6=O)C=C5)OC[C@H]4C3)CC2)S1	C39H40N12O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-EA2YAI	WO2023186069A1_84	1-[5-[5-[1-[1-[[1-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperidin-4-yl]methyl]piperidine-4-carbonyl]piperidin-4-yl]-1,3,4-thiadiazol-2-yl]-4-(methylamino)pyridin-2-yl]pyrrolo[2,3-b]pyridine-5-carbonitrile	CNC1=C(C2=NN=C(C3CCN(C(=O)C4CCN(CC5CCN(C6=CC=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)CC3)S2)C=NC(N2C=CC3=C2N=CC(C#N)=C3)=C1	C46H48N12O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-C7HLX8	WO2023186069A1_85	.	CNC1=C(C2=NN=C(C3CCN(C(=O)CN4CCN(C5=CC=C(N6CCC(=O)NC6=O)C=C5)CC4)CC3)S2)C=NC(N2C=CC3=C2N=CC(C#N)=C3)=C1	C37H38N12O3S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-81AXV0	WO2023186069A1_86	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C(C2CCN(C(=O)CN3CCN(C(=O)C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)C2)S1	C40H36N12O6S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-H8DL5E	WO2023186069A1_87	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](N(C)CC3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)S1	C42H43N11O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-6PJ7WF	WO2023186069A1_88	.	CNC1=CC(N2CCC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](NC(=O)CN3CCN4C5=C(C=C(N6CCC(=O)NC6=O)C=C5)OC[C@@H]4C3)CC2)S1	C39H42N12O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-YSPYXC	SCHEMBL26110706	2-[(4aR)-8-(2,4-dioxo-1,3-diazinan-1-yl)-2,4,4a,5-tetrahydro-1H-pyrazino[2,1-c][1,4]benzoxazin-3-yl]-N-[4-[5-[6-(5-cyano-2,3-dihydropyrrolo[2,3-b]pyridin-1-yl)-4-(methylamino)pyridin-3-yl]-1,3,4-thiadiazol-2-yl]cyclohexyl]acetamide	CNC1=CC(N2CCC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](NC(=O)CN3CCN4C5=C(C=C(N6CCC(=O)NC6=O)C=C5)OC[C@H]4C3)CC2)S1	C39H42N12O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-NQ8QWY	WO2023186069A1_90	.	CNC1=C(C2=NN=C([C@H]3CC[C@H](NC(=O)CN4CCN(C5=CC6=C(C=C5F)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)S2)C=NC(N2C=CC3=C2N=CC(C#N)=C3)=N1	C40H38FN13O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-QJOKDP	WO2023186069A1_91	.	CNC1=C(C2=NN=C([C@H]3CC[C@H](NC(=O)CN4CCN5C6=C(C=C(N7CCC(=O)NC7=O)C=C6)OC[C@@H]5C4)CC3)S2)C=NC(N2C=CC3=C2N=CC(C#N)=C3)=N1	C38H39N13O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-FN2E1W	WO2023186069A1_92	.	CNC1=C(C2=NN=C([C@H]3CC[C@H](NC(=O)CN4CCN5C6=C(C=C(N7CCC(=O)NC7=O)C=C6)OC[C@H]5C4)CC3)S2)C=NC(N2C=CC3=C2N=CC(C#N)=C3)=N1	C38H39N13O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-UBU0GC	SCHEMBL26110790	1-[5-[5-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindole-5-carbonyl]piperidin-4-yl]methyl-methylamino]cyclohexyl]-1,3,4-thiadiazol-2-yl]-4-(methylamino)pyridin-2-yl]pyrrolo[2,3-b]pyridine-5-carbonitrile; SCHEMBL30569062	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](N(C)CC3CCN(C(=O)C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)CC5=C4)CC3)CC2)S1	C43H45N11O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-5FD05O	WO2023186069A1_94	.	CNC1=C(C2=NN=C(C3CCN(C(=O)CN4CCN5C6=CC=C(N7CCC(=O)NC7=O)C=C6OC[C@@H]5C4)CC3)S2)C=NC(N2C=CC3=C2N=CC(C#N)=C3)=C1	C38H38N12O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-9K3J9F	WO2023186069A1_95	.	CNC1=C(C2=NN=C(C3CCN(C(=O)CN4CCN5C6=CC=C(N7CCC(=O)NC7=O)C=C6OC[C@H]5C4)CC3)S2)C=NC(N2C=CC3=C2N=CC(C#N)=C3)=C1	C38H38N12O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-UAZY3E	WO2023186069A1_96	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](N(C)CC3CCN(C4=C(F)C=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)S1	C42H42FN11O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-U14J3F	WO2023186069A1_97	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C(C2CC3(CCN(C(=O)CN4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)C2)S1	C43H42N12O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-GQ7OW3	WO2023186069A1_98	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C(C2CC3(CCN(C(=O)CN4CCN(C5=C(F)C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)C2)S1	C43H41FN12O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-8W43D4	WO2023186069A1_99	1-[5-[5-[1-[2-[4-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]acetyl]pyrrolidin-3-yl]-1,3,4-thiadiazol-2-yl]-4-(methylamino)pyridin-2-yl]pyrrolo[2,3-b]pyridine-5-carbonitrile	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C(C2CCN(C(=O)CN3CCN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)C2)S1	C39H36N12O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-J06IYX	WO2023186069A1_100	.	CNC1=NC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](NC(=O)CN3CCN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)S1	C40H39N13O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-UA49ZO	WO2023186069A1_101	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](NCC3CCN(C4=CC=C(N5CCC(=O)NC5=O)C=C4)CC3)CC2)S1	C38H41N11O2S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-VRVCKC	WO2023186069A1_102	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C(C2CC3(CC(NC(=O)CN4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)C3)C2)S1	C42H40N12O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-SL79BJ	WO2023186069A1_103	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C(C2CC3(C2)CN(C(=O)CN2CCN4C5=CC=C(N6CCC(=O)NC6=O)C=C5OC[C@@H]4C2)C3)S1	C39H38N12O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-QBVI1I	WO2023186069A1_104	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C(C2CC3(C2)CN(C(=O)CN2CCN4C5=CC=C(N6CCC(=O)NC6=O)C=C5OC[C@H]4C2)C3)S1	C39H38N12O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-THTEN8	WO2023186069A1_105	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C(C2CC3(CC(NC(=O)CN4CCN(C5=C(F)C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)C3)C2)S1	C42H39FN12O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-1BF68Z	WO2023186069A1_106	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](N(C)CC3CCN(C4=CC=C(N5CCC(=O)NC5=O)C=C4)CC3)CC2)S1	C39H43N11O2S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-GY8DOC	WO2023186069A1_107	.	CNC1=C(C2=NN=C([C@H]3CC[C@H](NC(=O)CN4CCN5C6=C(C=C(N7CCC(=O)NC7=O)C=C6)OC[C@@H]5C4)CC3)S2)C=NC(N2C=CC3=C2N=CC=C3C#N)=C1	C39H40N12O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-NZNH77	WO2023186069A1_108	.	CNC1=C(C2=NN=C([C@H]3CC[C@H](NC(=O)CN4CCN5C6=C(C=C(N7CCC(=O)NC7=O)C=C6)OC[C@H]5C4)CC3)S2)C=NC(N2C=CC3=C2N=CC=C3C#N)=C1	C39H40N12O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-9HP4UC	WO2023186069A1_109	.	CNC1=NC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](NCC3CCN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)S1	C40H40N12O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-Z2OD1E	SCHEMBL26135424	N-[4-[5-[6-(4-cyanopyrrolo[2,3-b]pyridin-1-yl)-4-(methylamino)pyridin-3-yl]-1,3,4-thiadiazol-2-yl]cyclohexyl]-2-[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]acetamide	CNC1=C(C2=NN=C([C@H]3CC[C@H](NC(=O)CN4CCN(C5=C(F)C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)S2)C=NC(N2C=CC3=C2N=CC=C3C#N)=C1	C41H39FN12O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-4AC7EQ	WO2023186069A1_111	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](CN3CCN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)S1	C40H39N11O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-GGDBMC	WO2023186069A1_112	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](CN3CCN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5)CC3)CC2)S1	C40H41N11O3S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-4TC1V0	WO2023186069A1_113	.	CNC1=CC(N2C=CC3=CC(C#N)=CN=C32)=NC=C1C1=NN=C([C@H]2CC[C@H](CN3CCN4C5=C(C=C(N6CCC(=O)NC6=O)C=C5)OC[C@@H]4C3)CC2)S1	C38H39N11O3S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-ZQYQ3W	WO2023186069A1_114	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](NC(=O)CN3CCN4C5=C(C=C(N6CCC(=O)NC6=O)C=C5F)OC[C@@H]4C3)CC2)S1	C39H39FN12O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-DED4GI	WO2023186069A1_115	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](NC(=O)CN3CCN4C5=C(C=C(N6CCC(=O)NC6=O)C=C5F)OC[C@H]4C3)CC2)S1	C39H39FN12O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-E2J6PC	WO2023186069A1_116	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](NC(=O)CN3CCN4C5=C(C=CC(N6CCC(=O)NC6=O)=C5)OC[C@@H]4C3)CC2)S1	C39H40N12O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-1VSM3G	WO2023186069A1_117	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](NC(=O)CN3CCN4C5=C(C=CC(N6CCC(=O)NC6=O)=C5)OC[C@H]4C3)CC2)S1	C39H40N12O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-A3UABG	WO2023186069A1_118	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](NC(=O)CN3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)CC5=C4)CC3)CC2)S1	C41H42N12O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-L6YO7M	WO2023186069A1_119	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C(C2CC3(C2)CN(C(=O)CN2CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)CC5=C4)CC2)C3)S1	C41H40N12O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-ZNEKRS	WO2023186069A1_120	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C(C2CC3(CCN(C(=O)CN4CCN5C6=C(C=C(N7CCC(=O)NC7=O)C=C6)OC[C@H]5C4)CC3)C2)S1	C41H42N12O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-ZK67P9	WO2023186069A1_121	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C(C2CC3(CCN(C(=O)CN4CCN5C6=C(C=C(N7CCC(=O)NC7=O)C=C6C)OC[C@H]5C4)CC3)C2)S1	C42H44N12O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-BQGRS6	WO2023186069A1_122	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C(C2CC3(CCN(C(=O)CN4CCN5C6=C(C=C(N7CCC(=O)NC7=O)C=C6C)OC[C@@H]5C4)CC3)C2)S1	C42H44N12O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-NXRUIL	SCHEMBL26111250	N-[1-[5-[6-(5-cyanopyrrolo[2,3-b]pyridin-1-yl)-4-(methylamino)pyridin-3-yl]-1,3,4-thiadiazol-2-yl]cyclopropyl]-2-[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]acetamide	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C(C2(NC(=O)CN3CCN(C4=CC5=C(C=C4F)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)S1	C38H33FN12O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-QDOTVU	WO2023186069A1_124	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C(C2(NC(=O)CN3CCN4C5=CC=C(N6CCC(=O)NC6=O)C=C5OC[C@H]4C3)CC2)S1	C36H34N12O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-Y3Z2KZ	WO2023186069A1_125	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C(N2CCC(NC(=O)CN3CCC(OCC#CC4=CC=CC5=C4N(C)C(=O)N5C4CCC(=O)NC4=O)CC3)CC2)S1	C44H45N13O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-HXNQ69	WO2023186069A1_126	.	CNC1=CC(N2C=CC3=CN=C(N4C[C@@H]5C[C@H]4CO5)N=C32)=NC=C1C1=NN=C([C@H]2CC[C@H](NC(=O)CN3CCN(C4=CC5=C(C=C4F)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)S1	C44H46FN13O6S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-CJF5LR	WO2023186069A1_127	.	CNC1=CC(N2C=CC3=CN=C(N4C[C@H]5C[C@@H]4CO5)N=C32)=NC=C1C1=NN=C([C@H]2CC[C@H](NC(=O)CN3CCN(C4=CC5=C(C=C4F)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)S1	C44H46FN13O6S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-MQ2B3N	WO2023186069A1_128	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C(C2(NC(=O)CN3CCN4C5=C(C)C=C(N6CCC(=O)NC6=O)C=C5OC[C@H]4C3)CC2)S1	C37H36N12O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-7BJHPV	WO2023186069A1_129	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C(C2CC3(C2)CC(N(C)CC2CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC2)C3)S1	C43H43N11O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-9KQSH8	WO2023186069A1_130	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C(C2CC3(CC(NC(=O)CN4CCN5C6=C(C=C(N7CCC(=O)NC7=O)C=C6C)OC[C@H]5C4)C3)C2)S1	C41H42N12O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-O9GFL6	WO2023186069A1_131	.	CNC1=CC(N2C=CC3=C2N=CC(C(N)=O)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](NC(=O)CN3CCN(C4=C(F)C=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)S1	C41H41FN12O6S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-CUHO3L	WO2023186069A1_132	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C(C2CC3(CC(NC(=O)CN4CCC(OCC#CC5=CC=CC6=C5N(C)C(=O)N6C5CCC(=O)NC5=O)CC4)C3)C2)S1	C46H46N12O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-QK3Y9S	WO2023186069A1_133	.	CNC1=C(C2=NN=C([C@H]3CC[C@H](NC(=O)CN4CCN(C5=NC=C(N6CCC(=O)NC6=O)C=N5)CC4)CC3)S2)C=NC(N2C=CC3=C2N=CC(C#N)=C3)=C1	C36H38N14O3S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-800IXZ	WO2023186069A1_134	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](N(C)C3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)S1	C41H41N11O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-J1EGD1	WO2023186069A1_135	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](C(=O)NC3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)S1	C41H39N11O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-APYM9X	WO2023186069A1_136	.	CNC1=C(C2=NN=C(C3CC[C@@H](NC(=O)CN4CCN(C5=C(F)C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CO3)S2)C=NC(N2C=CC3=C2N=CC(C#N)=C3)=C1	C40H37FN12O6S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-10FXBH	WO2023186069A1_137	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@@H]2CC[C@@H](NC(=O)CN3CCN4C5=C(C=C(N6CCC(=O)NC6=O)C=C5C)OC[C@H]4C3)CO2)S1	C39H40N12O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-4CJH95	WO2023186069A1_138	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](N(C)CC(=O)N3CCN4C5=C(C=C(N6CCC(=O)NC6=O)C=C5)OC[C@H]4C3)CC2)S1	C40H42N12O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-2QH2WK	WO2023186069A1_139	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@@H]2CC[C@@H](N(C)CC3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CO2)S1	C41H41N11O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-AVQ93V	WO2023186069A1_140	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C(C2CC3(C2)CC(N(C)C2CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC2)C3)S1	C42H41N11O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-BZP5SP	SCHEMBL26112989	2-[(4aR)-8-(2,4-dioxo-1,3-diazinan-1-yl)-10-propan-2-yl-2,4,4a,5-tetrahydro-1H-pyrazino[2,1-c][1,4]benzoxazin-3-yl]-N-[4-[5-[6-(5-cyanopyrrolo[2,3-b]pyridin-1-yl)-4-(methylamino)pyridin-3-yl]-1,3,4-thiadiazol-2-yl]cyclohexyl]acetamide	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](NC(=O)CN3CCN4C5=C(C=C(N6CCC(=O)NC6=O)C=C5C(C)C)OC[C@H]4C3)CC2)S1	C42H46N12O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-5A0C6B	WO2023186069A1_142	.	CNC1=CC(N2C=CC3=CC(C#N)=CN=C32)=NC=C1C1=NN=C([C@H]2CC[C@H](CN3CCN(C4=C(F)C=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)S1	C40H38FN11O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-HQ5Q3A	WO2023186069A1_143	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](CN(C)C3CCN(C4=CC=CC5=C4N(C)C(=O)N5C4CCC(=O)NC4=O)CC3)CC2)S1	C42H46N12O3S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-GPC91K	WO2023186069A1_144	.	CNC1=CC(N2C=CC3=CC(C#N)=CN=C32)=NC=C1C1=NN=C([C@H]2CC[C@H](CN3CCN4C5=CC=C(NC6CCC(=O)NC6=O)C=C5OC[C@H]4C3)CC2)S1	C39H41N11O3S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-JN5G65	WO2023186069A1_145	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C(C2CC3(C2)CN(C(=O)C2CCN(C4=C(F)C=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC2)C3)S1	C41H36FN11O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-SQ1EY6	WO2023186069A1_146	.	CNC1=CC(N2C=CC3=CC(C#N)=CN=C32)=NC=C1C1=NN=C([C@H]2CC[C@H](CN(C)C3CCN(C4=CC5=C(C=C4F)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)S1	C42H42FN11O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-SDB0U9	WO2023186069A1_147	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](CN3CCN4C5=C(C=CC(N6CCC(=O)NC6=O)=C5)OC[C@@H]4C3)CC2)S1	C38H39N11O3S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-XJSE6W	SCHEMBL26107878	1-[5-[5-[4-[[4-[1-(2,6-Dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-4-yl]piperazin-1-yl]methyl]cyclohexyl]-1,3,4-thiadiazol-2-yl]-4-(methylamino)pyridin-2-yl]pyrrolo[2,3-b]pyridine-5-carbonitrile; SCHEMBL30569044	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](CN3CCN(C4=CC=CC5=C4N(C)C(=O)N5C4CCC(=O)NC4=O)CC3)CC2)S1	C40H42N12O3S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-XAUYTV	WO2023186069A1_149	.	CNC1=C(C2=NN=C(C3CC4(C3)CN(C(=O)CN3CCN(C5=NC=C(N6CCC(=O)NC6=O)C=N5)CC3)C4)S2)C=NC(N2C=CC3=C2N=CC(C#N)=C3)=C1	C36H36N14O3S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-523Z99	WO2023186069A1_150	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C(C2CC3(CCN(CC4CCN(C5=CC6=C(C=C5F)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)C2)S1	C43H42FN11O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-F6O6AD	WO2023186069A1_151	.	CNC1=CC(N2C=CC3=CC(C#N)=CN=C32)=NC=C1C1=NN=C(C2CC3(C2)CN(C(=O)CN2CCN4C5=CC=C(NC6CCC(=O)NC6=O)C=C5OC[C@@H]4C2)C3)S1	C40H40N12O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-LIT45V	WO2023186069A1_152	.	CNC1=CC(N2C=CC3=CC(C#N)=CN=C32)=NC=C1C1=NN=C(C2CC3(C2)CN(C(=O)CN2CCN4C5=CC=C(NC6CCC(=O)NC6=O)C=C5OC[C@H]4C2)C3)S1	C40H40N12O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-4ZYHZW	WO2023186069A1_154	.	CC(C)NC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](NC(=O)CN3CCN(C4=C(F)C=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)S1	C43H43FN12O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-GLPXR0	WO2023186069A1_155	.	CC(C)NC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](N(C)CC3CCN(C4=C(F)C=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)S1	C44H46FN11O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-QIF5Y1	WO2023186069A1_156	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](CN(C)C3(C4CCN(C5=CC6=C(C=C5F)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)CC2)S1	C45H46FN11O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-L8ONOX	WO2023186069A1_157	.	O=NC1=CC2=C(N=C1)N(C1=NC=C(C3=NN=C([C@H]4CC[C@H](NC(=O)CN5CCN(C6=C(F)C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)S3)C(NC3CC3)=C1)C=C2	C42H41FN12O6S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-LUM1TR	WO2023186069A1_158	.	CN(CC1CCN(C2=C(F)C=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=C2)CC1)[C@H]1CC[C@H](C2=NN=C(C3=CN=C(N4C=CC5=C4N=CC(C#N)=C5)C=C3NC3CC3)S2)CC1	C44H44FN11O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-0B6DC7	WO2023186069A1_159	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](NC(=O)C3CCN(C4=C(F)C=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)S1	C41H38FN11O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-WDI4CR	WO2023186069A1_161	.	[H]C([H])([H])N(C(=O)CN1CCN(C2=C(F)C=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=C2)CC1)[C@H]1CC[C@H](C2=NN=C(C3=CN=C(N4C=CC5=C4N=CC(C#N)=C5)C=C3NC)S2)CC1	C42H41FN12O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-ZY9KK3	SCHEMBL30678688	N-[4-[5-[6-(5-cyanopyrrolo[2,3-b]pyridin-1-yl)-4-(propan-2-ylamino)pyridin-3-yl]-1,3,4-thiadiazol-2-yl]cyclohexyl]-1-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]methyl]piperidine-4-carboxamide	CC(C)NC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](NC(=O)C3CCN(CC4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)S1	C44H45N11O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-7NK6IX	WO2023186069A1_163	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C(C2CC3(C2)CN(C(=O)CN2CCN4C5=C(OC[C@H]4C2)C(C)=CC(N2CCC(=O)NC2=O)=C5)C3)S1	C40H40N12O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-WSFGY8	WO2023186069A1_165	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C(C2CC3(C2)CN(C(=O)C2CCN(C4=NC=C(N5CCC(=O)NC5=O)C=N4)CC2)C3)S1	C36H35N13O3S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-HDGWTF	WO2023186069A1_166	.	CNC1=CC(N2C=CC3=CC(C#N)=CN=C32)=NC=C1C1=NN=C([C@H]2CC[C@H](CN3CCC(C4(NC5=C(F)C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)CC2)S1	C44H44FN11O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-NYWZH0	WO2023186069A1_167	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](NC(=O)C3CCN(C4=C(F)C=C5C(=O)N(C6CCC(=O)NC6=O)CC5=C4)CC3)CC2)S1	C41H40FN11O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-RJXAY0	SCHEMBL26134335	N-[4-[5-[6-(3-chloro-5-cyanopyrrolo[2,3-b]pyridin-1-yl)-4-(methylamino)pyridin-3-yl]-1,3,4-thiadiazol-2-yl]cyclohexyl]-2-[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]acetamide; SCHEMBL30569125	CNC1=CC(N2C=C(Cl)C3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](NC(=O)CN3CCN(C4=C(F)C=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)S1	C41H38ClFN12O5S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-BDOVI2	WO2023186069A1_169	.	CNC1=CC(N2C=CC3=CC(C#N)=CN=C32)=NC=C1C1=NN=C([C@H]2CC[C@H](CN3CCN(C4=CC5=C(C=C4F)C(=O)N(C4CCC(=O)NC4=O)C5)CC3)CC2)S1	C40H40FN11O3S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-HTVBZG	WO2023186069A1_170	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](NCC3CCN(C4=NC=C(N5CCC(=O)NC5=O)C=N4)CC3)CC2)S1	C36H39N13O2S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-9610LT	WO2023186069A1_171	.	CNC1=C(C2=NN=C([C@H]3CC[C@H](NC(=O)CN4CCN(C5=C(F)C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)S2)C=NC(N2C=CC3=C2N=CC(C(C)=O)=C3)=C1	C42H42FN11O6S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-XDPDLU	WO2023186069A1_172	.	CNC1=CC(N2C=CC3=CC(C#N)=CN=C32)=NC=C1C1=NN=C([C@H]2CC[C@H](NCC3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)CC5=C4)CC3)CC2)S1	C41H43N11O3S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-GW0J79	WO2023186069A1_173	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](NC3CCN(C4=C(F)C=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)S1	C40H38FN11O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-VSP71Z	WO2023186069A1_174	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](N(C)C3CCN(C4=C(F)C=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)S1	C41H40FN11O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-XQTLPD	WO2023186069A1_175	.	CNC1=CC(N2C=CC3=CC(C#N)=CN=C32)=NC=C1C1=NN=C([C@H]2CC[C@H](N(C)CC3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)CC5=C4)CC3)CC2)S1	C42H45N11O3S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-4T2J9A	WO2023186069A1_176	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](N(C)CC3CC4(CCN(C5=C(F)C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)C3)CC2)S1	C45H46FN11O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-C0M6OU	WO2023186069A1_177	.	CNC1=CC(N2C=CC3=C2N=CC(C#N)=C3)=NC=C1C1=NN=C([C@H]2CC[C@H](CN3CCC4(CC3)CN(C3=CC5=C(C=C3F)C(=O)N(C3CCC(=O)NC3=O)C5=O)C4)CC2)S1	C43H42FN11O4S	IRAK4	Q9NWZ3	CRBN	WO-2023186069-A1
TPD-07GBTE	SCHEMBL26621444	3-[6-[[5-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-5-azaspiro[3.5]nonan-8-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661502	CN1N=C(C2CCC(=O)NC2=O)C2=C1C=C(NC1CCN(C3=NC(NC4=CC=C5C(=C4)CC(=O)N5C)=C(Cl)C=N3)C3(CCC3)C1)C=C2	C34H36ClN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-T54D9I	WO2023212147A1_2	.	CN1N=C(C2CCC(=O)NC2=O)C2=C1C=C(N1CCC(N(C)C3=NC(NC4C=C5CC(=O)N(C)C5=CC4)=C(Cl)C=N3)CC13CCC3)C=C2	C35H40ClN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-RLSV1X	WO2023212147A1_3	.	CN1N=C(C2CCC(=O)NC2=O)C2=C1C=C(N[C@H]1CC[C@H](N(C)C3=NC(NC4=CC5=C(C=C4)NC(=O)C5)=C(Cl)C=N3)CC1)C=C2	C32H34ClN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-P066CE	SCHEMBL26621426	3-[6-[(2R,4R)-4-[[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-methylamino]-2-methylpiperidin-1-yl]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661542	C[C@@H]1C[C@H](N(C)C2=NC(NC3=CC=C4C(=C3)CC(=O)N4C)=C(Cl)C=N2)CCN1C1=CC2=C(C=C1)C(C1CCC(=O)NC1=O)=NN2C	C33H36ClN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-41C3Q8	SCHEMBL26621430	3-[6-[4-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-2-methyl-6-oxopiperazin-1-yl]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661558	CC1CN(C2=NC=C(Cl)C(NC3=CC=C4C(=C3)CC(=O)N4C)=N2)CC(=O)N1C1=CC2=C(C=C1)C(C1CCC(=O)NC1=O)=NN2C	C31H30ClN9O4	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-SSKRBQ	WO2023212147A1_6	.	CN1N=C(C2CCC(=O)NC2=O)C2=CC=C(N3CCC(N(C)C4=NC=C(Cl)C(NC5=CC6=C(C=C5)NC(=O)C6)=N4)CC3)C=C21	C31H32ClN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-C4IDN8	SCHEMBL26621594	3-[6-[[1-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]piperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661506	CN1N=C(C2CCC(=O)NC2=O)C2=C1C=C(NC1CCN(C3=NC(NC4=CC=C5C(=C4)CC(=O)N5C)=C(Cl)C=N3)CC1)C=C2	C31H32ClN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-QVL0RN	SCHEMBL26752072	3-[6-[4-[[5-chloro-4-[[1-(3-hydroxy-3-methylbutyl)-2-oxo-3H-indol-6-yl]amino]pyrimidin-2-yl]amino]piperidin-1-yl]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL31444670	CN1N=C(C2CCC(=O)NC2=O)C2=C1C=C(N1CCC(NC3=NC=C(Cl)C(NC4=CC=C5CC(=O)N(CCC(C)(C)O)C5=C4)=N3)CC1)C=C2	C35H40ClN9O4	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-F60FNW	SCHEMBL26752227	3-[6-[[1-[5-chloro-4-[[1-(3-hydroxy-3-methylbutyl)-2-oxo-3H-indol-6-yl]amino]pyrimidin-2-yl]piperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL31444723	CN1N=C(C2CCC(=O)NC2=O)C2=C1C=C(NC1CCN(C3=NC=C(Cl)C(NC4=CC5=C(C=C4)CC(=O)N5CCC(C)(C)O)=N3)CC1)C=C2	C35H40ClN9O4	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-E8ODKV	SCHEMBL26752229	3-[6-[[1-[5-chloro-4-[[1-(3-hydroxy-3-methylbutyl)-2-oxo-3H-indol-6-yl]amino]pyrimidin-2-yl]piperidin-4-yl]-methylamino]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL31444696	CN1N=C(C2CCC(=O)NC2=O)C2=CC=C(N(C)C3CCN(C4=NC=C(Cl)C(NC5=CC=C6CC(=O)N(CCC(C)(C)O)C6=C5)=N4)CC3)C=C21	C36H42ClN9O4	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-K14DRE	SCHEMBL26752231	3-[6-[4-[[5-chloro-4-[[1-(3-hydroxy-3-methylbutyl)-2-oxo-3H-indol-6-yl]amino]pyrimidin-2-yl]-methylamino]piperidin-1-yl]-1-methylindazol-3-yl]piperidine-2,6-dione	CN1N=C(C2CCC(=O)NC2=O)C2=C1C=C(N1CCC(N(C)C3=NC=C(Cl)C(NC4=CC=C5CC(=O)N(CCC(C)(C)O)C5=C4)=N3)CC1)C=C2	C36H42ClN9O4	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-S5YX3X	SCHEMBL26752233	3-[6-[[(3R,4S)-1-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-3-methylpiperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione	C[C@@H]1CN(C2=NC=C(Cl)C(NC3=CC=C4C(=C3)CC(=O)N4C)=N2)CC[C@@H]1NC1=CC2=C(C=C1)C(C1CCC(=O)NC1=O)=NN2C	C32H34ClN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-W2WYJ0	SCHEMBL26752236	3-[6-[[(3S,4R)-1-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-3-methylpiperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione	C[C@H]1CN(C2=NC=C(Cl)C(NC3=CC=C4C(=C3)CC(=O)N4C)=N2)CC[C@H]1NC1=CC2=C(C=C1)C(C1CCC(=O)NC1=O)=NN2C	C32H34ClN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-WVOCNW	SCHEMBL26752240	3-[6-[[(3S,4S)-1-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-3-methylpiperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione	C[C@H]1CN(C2=NC=C(Cl)C(NC3=CC=C4C(=C3)CC(=O)N4C)=N2)CC[C@@H]1NC1=CC2=C(C=C1)C(C1CCC(=O)NC1=O)=NN2C	C32H34ClN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-FXVYI0	SCHEMBL26752243	3-[6-[3-[[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-methylamino]-8-azabicyclo[3.2.1]octan-8-yl]-1-methylindazol-3-yl]piperidine-2,6-dione	CN1N=C(C2CCC(=O)NC2=O)C2=C1C=C(N1C3CCC1CC(N(C)C1=NC(NC4=CC=C5C(=C4)CC(=O)N5C)=C(Cl)C=N1)C3)C=C2	C34H36ClN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-NBMB0L	SCHEMBL27071736	3-[6-[(1R,5S)-3-[[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-methylamino]-8-azabicyclo[3.2.1]octan-8-yl]-1-methylindazol-3-yl]piperidine-2,6-dione	CN1N=C(C2CCC(=O)NC2=O)C2=C1C=C(N1[C@@H]3CC[C@H]1C[C@@H](N(C)C1=NC(NC4=CC=C5C(=C4)CC(=O)N5C)=C(Cl)C=N1)C3)C=C2	C34H36ClN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-LQ4042	SCHEMBL27071737	3-[6-[[4-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]piperazin-1-yl]methyl]-1-methylindazol-3-yl]piperidine-2,6-dione	CN1N=C(C2CCC(=O)NC2=O)C2=C1C=C(CN1CCN(C3=NC(NC4=CC=C5C(=C4)CC(=O)N5C)=C(Cl)C=N3)CC1)C=C2	C31H32ClN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-RJBSYO	SCHEMBL27071738	3-[6-[[1-[5-chloro-4-[[2-oxo-1-(2,2,2-trifluoroethyl)-3H-indol-5-yl]amino]pyrimidin-2-yl]piperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione	CN1N=C(C2CCC(=O)NC2=O)C2=C1C=C(NC1CCN(C3=NC(NC4=CC=C5C(=C4)CC(=O)N5CC(F)(F)F)=C(Cl)C=N3)CC1)C=C2	C32H31ClF3N9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-6EQR31	SCHEMBL27071739	3-[6-[[(2S,4S)-1-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-2-methylpiperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione	C[C@H]1C[C@@H](NC2=CC3=C(C=C2)C(C2CCC(=O)NC2=O)=NN3C)CCN1C1=NC(NC2=CC=C3C(=C2)CC(=O)N3C)=C(Cl)C=N1	C32H34ClN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-XG2X40	SCHEMBL27071740	3-[6-[(2S,4S)-4-[[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-methylamino]-2-methylpiperidin-1-yl]-1-methylindazol-3-yl]piperidine-2,6-dione	C[C@H]1C[C@@H](N(C)C2=NC(NC3=CC=C4C(=C3)CC(=O)N4C)=C(Cl)C=N2)CCN1C1=CC2=C(C=C1)C(C1CCC(=O)NC1=O)=NN2C	C33H36ClN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-OAK10D	SCHEMBL27071741	3-[6-[[(2R,4R)-1-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-2-methylpiperidin-4-yl]-methylamino]-1-methylindazol-3-yl]piperidine-2,6-dione	C[C@@H]1C[C@H](N(C)C2=CC3=C(C=C2)C(C2CCC(=O)NC2=O)=NN3C)CCN1C1=NC(NC2=CC=C3C(=C2)CC(=O)N3C)=C(Cl)C=N1	C33H36ClN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-TWZLH2	SCHEMBL26752405	3-[6-[[(2R,4R)-1-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-2-methylpiperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione	C[C@@H]1C[C@H](NC2=CC3=C(C=C2)C(C2CCC(=O)NC2=O)=NN3C)CCN1C1=NC(NC2=CC=C3C(=C2)CC(=O)N3C)=C(Cl)C=N1	C32H34ClN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-YMG9SD	SCHEMBL26752406	3-[6-[[(2R,4S)-1-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-2-methylpiperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione	C[C@@H]1C[C@@H](NC2=CC3=C(C=C2)C(C2CCC(=O)NC2=O)=NN3C)CCN1C1=NC(NC2=CC=C3C(=C2)CC(=O)N3C)=C(Cl)C=N1	C32H34ClN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-BK39I9	SCHEMBL26752584	3-[6-[[(2S,4S)-1-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-2-methylpiperidin-4-yl]-methylamino]-1-methylindazol-3-yl]piperidine-2,6-dione	C[C@H]1C[C@@H](N(C)C2=CC3=C(C=C2)C(C2CCC(=O)NC2=O)=NN3C)CCN1C1=NC(NC2=CC=C3C(=C2)CC(=O)N3C)=C(Cl)C=N1	C33H36ClN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-ABHHLG	SCHEMBL26752587	3-[6-[[(2R,4S)-1-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-2-methylpiperidin-4-yl]-methylamino]-1-methylindazol-3-yl]piperidine-2,6-dione	C[C@@H]1C[C@@H](N(C)C2=CC3=C(C=C2)C(C2CCC(=O)NC2=O)=NN3C)CCN1C1=NC(NC2=CC=C3C(=C2)CC(=O)N3C)=C(Cl)C=N1	C33H36ClN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-ST2G09	SCHEMBL26752588	3-[6-[(2R,6S)-4-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-2,6-dimethylpiperazin-1-yl]-1-methylindazol-3-yl]piperidine-2,6-dione	C[C@@H]1CN(C2=NC=C(Cl)C(NC3=CC4=C(C=C3)N(C)C(=O)C4)=N2)C[C@H](C)N1C1=CC2=C(C=C1)C(C1CCC(=O)NC1=O)=NN2C	C32H34ClN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-FP3H5S	SCHEMBL26752594	3-[6-[(3R,5R)-4-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-3,5-dimethylpiperazin-1-yl]-1-methylindazol-3-yl]piperidine-2,6-dione	C[C@@H]1CN(C2=CC3=C(C=C2)C(C2CCC(=O)NC2=O)=NN3C)C[C@@H](C)N1C1=NC=C(Cl)C(NC2=CC3=C(C=C2)N(C)C(=O)C3)=N1	C32H34ClN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-77Q0D7	SCHEMBL26752596	3-[6-[(3S,5S)-4-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-3,5-dimethylpiperazin-1-yl]-1-methylindazol-3-yl]piperidine-2,6-dione	C[C@H]1CN(C2=CC3=C(C=C2)C(C2CCC(=O)NC2=O)=NN3C)C[C@H](C)N1C1=NC=C(Cl)C(NC2=CC3=C(C=C2)N(C)C(=O)C3)=N1	C32H34ClN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-QEK9DT	SCHEMBL26752598	3-[6-[(3R,5S)-4-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-3,5-dimethylpiperazin-1-yl]-1-methylindazol-3-yl]piperidine-2,6-dione	C[C@@H]1CN(C2=CC3=C(C=C2)C(C2CCC(=O)NC2=O)=NN3C)C[C@H](C)N1C1=NC=C(Cl)C(NC2=CC3=C(C=C2)N(C)C(=O)C3)=N1	C32H34ClN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-9925SQ	SCHEMBL26752778	3-[6-[[1-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]azepan-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione	CN1N=C(C2CCC(=O)NC2=O)C2=C1C=C(NC1CCCN(C3=NC=C(Cl)C(NC4=CC=C5C(=C4)CC(=O)N5C)=N3)CC1)C=C2	C32H34ClN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-FVB501	SCHEMBL26752780	3-[6-[4-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-1,4-diazepan-1-yl]-1-methylindazol-3-yl]piperidine-2,6-dione	CN1N=C(C2CCC(=O)NC2=O)C2=CC=C(N3CCCN(C4=NC=C(Cl)C(NC5=CC=C6C(=C5)CC(=O)N6C)=N4)CC3)C=C21	C31H32ClN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-AWOJ57	SCHEMBL26752782	3-[6-[[(3R,4R)-1-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-3-hydroxypiperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione	CN1N=C(C2CCC(=O)NC2=O)C2=CC=C(N[C@@H]3CCN(C4=NC(NC5=CC=C6C(=C5)CC(=O)N6C)=C(Cl)C=N4)C[C@H]3O)C=C21	C31H32ClN9O4	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-MCV9KL	SCHEMBL26752784	3-[6-[4-[5-Chloro-4-[(2-oxo-1,3-dihydroindol-5-yl)amino]pyrimidin-2-yl]piperazin-1-yl]-1-methylindazol-3-yl]piperidine-2,6-dione	CN1N=C(C2CCC(=O)NC2=O)C2=CC=C(N3CCN(C4=NC=C(Cl)C(NC5=CC6=C(C=C5)NC(=O)C6)=N4)CC3)C=C21	C29H28ClN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-N910AN	SCHEMBL26752786	3-[6-[4-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]piperazin-1-yl]-1-methylindazol-3-yl]piperidine-2,6-dione	CN1N=C(C2CCC(=O)NC2=O)C2=C1C=C(N1CCN(C3=NC=C(Cl)C(NC4=CC5=C(C=C4)N(C)C(=O)C5)=N3)CC1)C=C2	C30H30ClN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-QW4GCF	SCHEMBL26752789	2-[4-[[3-(2,6-dioxopiperidin-3-yl)-1-methylindazol-6-yl]amino]piperidin-1-yl]-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidine-5-carbonitrile	CN1N=C(C2CCC(=O)NC2=O)C2=C1C=C(NC1CCN(C3=NC=C(C#N)C(NC4=CC5=C(C=C4)N(C)C(=O)C5)=N3)CC1)C=C2	C32H32N10O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-DF8QQ9	SCHEMBL26753014	3-[6-[4-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-2-oxopiperazin-1-yl]-1-methylindazol-3-yl]piperidine-2,6-dione	CN1N=C(C2CCC(=O)NC2=O)C2=C1C=C(N1CCN(C3=NC(NC4=CC=C5C(=C4)CC(=O)N5C)=C(Cl)C=N3)CC1=O)C=C2	C30H28ClN9O4	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-3NXE89	SCHEMBL26753015	3-[6-[4-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-3-methyl-2-oxopiperazin-1-yl]-1-methylindazol-3-yl]piperidine-2,6-dione	CC1C(=O)N(C2=CC3=C(C=C2)C(C2CCC(=O)NC2=O)=NN3C)CCN1C1=NC=C(Cl)C(NC2=CC=C3C(=C2)CC(=O)N3C)=N1	C31H30ClN9O4	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-ZT2TNQ	SCHEMBL26753019	3-[6-[4-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-5-methyl-2-oxopiperazin-1-yl]-1-methylindazol-3-yl]piperidine-2,6-dione	CC1CN(C2=CC3=C(C=C2)C(C2CCC(=O)NC2=O)=NN3C)C(=O)CN1C1=NC=C(Cl)C(NC2=CC=C3C(=C2)CC(=O)N3C)=N1	C31H30ClN9O4	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-638NWK	SCHEMBL26753025	3-[6-[4-[[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]amino]piperidin-1-yl]-1-methylindazol-3-yl]piperidine-2,6-dione	CN1N=C(C2CCC(=O)NC2=O)C2=CC=C(N3CCC(NC4=NC=C(Cl)C(NC5=CC6=C(C=C5)N(C)C(=O)C6)=N4)CC3)C=C21	C31H32ClN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-A0AKX5	SCHEMBL26753026	3-[6-[[1-[5-chloro-4-[[1-(2-hydroxyethyl)-2-oxo-3H-indol-5-yl]amino]pyrimidin-2-yl]piperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione	CN1N=C(C2CCC(=O)NC2=O)C2=C1C=C(NC1CCN(C3=NC=C(Cl)C(NC4=CC5=C(C=C4)N(CCO)C(=O)C5)=N3)CC1)C=C2	C32H34ClN9O4	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-49OXW9	SCHEMBL26753027	3-[6-[[(3S,4S)-1-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-3-fluoropiperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione	CN1N=C(C2CCC(=O)NC2=O)C2=C1C=C(N[C@H]1CCN(C3=NC=C(Cl)C(NC4=CC5=C(C=C4)N(C)C(=O)C5)=N3)C[C@@H]1F)C=C2	C31H31ClFN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-3UIZZI	SCHEMBL26753028	3-[6-[[(3R,4S)-1-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-3-fluoropiperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione	CN1N=C(C2CCC(=O)NC2=O)C2=CC=C(N[C@H]3CCN(C4=NC=C(Cl)C(NC5=CC6=C(C=C5)N(C)C(=O)C6)=N4)C[C@H]3F)C=C21	C31H31ClFN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-A83X0R	SCHEMBL26753203	3-[6-[[(3S,4R)-1-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-3-fluoropiperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione	CN1N=C(C2CCC(=O)NC2=O)C2=CC=C(N[C@@H]3CCN(C4=NC=C(Cl)C(NC5=CC6=C(C=C5)N(C)C(=O)C6)=N4)C[C@@H]3F)C=C21	C31H31ClFN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-1Z6K7B	SCHEMBL26753204	3-[6-[[(3R,4R)-1-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-3-fluoropiperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione	CN1N=C(C2CCC(=O)NC2=O)C2=CC=C(N[C@@H]3CCN(C4=NC=C(Cl)C(NC5=CC6=C(C=C5)N(C)C(=O)C6)=N4)C[C@H]3F)C=C21	C31H31ClFN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-SU7L4B	SCHEMBL27033091	3-[6-[[(3R,4R)-1-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-3-fluoropiperidin-4-yl]-methylamino]-1-methylindazol-3-yl]piperidine-2,6-dione	CN1N=C(C2CCC(=O)NC2=O)C2=CC=C(N(C)[C@@H]3CCN(C4=NC=C(Cl)C(NC5=CC6=C(C=C5)N(C)C(=O)C6)=N4)C[C@H]3F)C=C21	C32H33ClFN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-5DPS33	SCHEMBL26753211	3-[6-[[1-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-5-methylazepan-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione	CC1CCN(C2=NC=C(Cl)C(NC3=CC=C4C(=C3)CC(=O)N4C)=N2)CCC1NC1=CC2=C(C=C1)C(C1CCC(=O)NC1=O)=NN2C	C33H36ClN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-4PEP2L	SCHEMBL26753212	3-[6-[[1-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-3-methylazepan-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione	CC1CN(C2=NC=C(Cl)C(NC3=CC=C4C(=C3)CC(=O)N4C)=N2)CCCC1NC1=CC2=C(C=C1)C(C1CCC(=O)NC1=O)=NN2C	C33H36ClN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-7A8IQY	SCHEMBL26621606	(3S)-3-[6-[[1-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]piperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione	CN1N=C([C@@H]2CCC(=O)NC2=O)C2=CC=C(NC3CCN(C4=NC=C(Cl)C(NC5=CC6=C(C=C5)N(C)C(=O)C6)=N4)CC3)C=C21	C31H32ClN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-34UAM2	SCHEMBL26621480	(3R)-3-[6-[[1-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]piperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661491	CN1N=C([C@H]2CCC(=O)NC2=O)C2=CC=C(NC3CCN(C4=NC=C(Cl)C(NC5=CC6=C(C=C5)N(C)C(=O)C6)=N4)CC3)C=C21	C31H32ClN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-WBEFIP	SCHEMBL26621412	3-[6-[[(3R,4R)-1-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-3-hydroxypiperidin-4-yl]amino]-1-methylpyrazolo[3,4-b]pyridin-3-yl]piperidine-2,6-dione; SCHEMBL30661663	CN1N=C(C2CCC(=O)NC2=O)C2=C1N=C(N[C@@H]1CCN(C3=NC=C(Cl)C(NC4=CC=C5C(=C4)CC(=O)N5C)=N3)C[C@H]1O)C=C2	C30H31ClN10O4	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-YQND6C	SCHEMBL26621613	3-[6-[[(3R,4R)-1-[5-chloro-4-[(3,3-difluoro-1-methyl-2-oxoindol-5-yl)amino]pyrimidin-2-yl]-3-methylpiperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661615	C[C@@H]1CN(C2=NC=C(Cl)C(NC3=CC=C4C(=C3)C(F)(F)C(=O)N4C)=N2)CC[C@H]1NC1=CC2=C(C=C1)C(C1CCC(=O)NC1=O)=NN2C	C32H32ClF2N9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-QUU4WK	SCHEMBL26621496	3-[6-[[(3S,4R)-1-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-3-(hydroxymethyl)piperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661471	CN1N=C(C2CCC(=O)NC2=O)C2=C1C=C(N[C@@H]1CCN(C3=NC(NC4=CC=C5C(=C4)CC(=O)N5C)=C(Cl)C=N3)C[C@@H]1CO)C=C2	C32H34ClN9O4	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-Y7IW8P	SCHEMBL26621722	3-[6-[[(3R,4S)-1-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-3-(hydroxymethyl)piperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661481	CN1N=C(C2CCC(=O)NC2=O)C2=C1C=C(N[C@H]1CCN(C3=NC(NC4=CC=C5C(=C4)CC(=O)N5C)=C(Cl)C=N3)C[C@H]1CO)C=C2	C32H34ClN9O4	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-SZYDNY	SCHEMBL26621420	3-[6-[4-[[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-methylamino]piperidin-1-yl]-1-methylpyrazolo[4,3-b]pyridin-3-yl]piperidine-2,6-dione; SCHEMBL30661472	CN1N=C(C2CCC(=O)NC2=O)C2=C1C=C(N1CCC(N(C)C3=NC(NC4=CC=C5C(=C4)CC(=O)N5C)=C(Cl)C=N3)CC1)C=N2	C31H33ClN10O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-ANWCIX	SCHEMBL26621407	3-[6-[4-[[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-methylamino]piperidin-1-yl]-1-methylpyrazolo[4,3-c]pyridin-3-yl]piperidine-2,6-dione; SCHEMBL30661504	CN1N=C(C2CCC(=O)NC2=O)C2=C1C=C(N1CCC(N(C)C3=NC(NC4=CC=C5C(=C4)CC(=O)N5C)=C(Cl)C=N3)CC1)N=C2	C31H33ClN10O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-DYENBY	SCHEMBL26621522	3-[6-[[(3R,4R)-1-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-6-yl)amino]pyrimidin-2-yl]-3-methylpiperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661598	C[C@@H]1CN(C2=NC(NC3=CC=C4CC(=O)N(C)C4=C3)=C(Cl)C=N2)CC[C@H]1NC1=CC2=C(C=C1)C(C1CCC(=O)NC1=O)=NN2C	C32H34ClN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-C9HWME	SCHEMBL26621640	3-[6-[[(3R,4R)-1-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-3-methylpiperidin-4-yl]amino]-1-methylpyrazolo[3,4-b]pyridin-3-yl]piperidine-2,6-dione; SCHEMBL30661606	C[C@@H]1CN(C2=NC=C(Cl)C(NC3=CC=C4C(=C3)CC(=O)N4C)=N2)CC[C@H]1NC1=NC2=C(C=C1)C(C1CCC(=O)NC1=O)=NN2C	C31H33ClN10O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-GJRVOF	SCHEMBL26621600	3-[6-[[1-[5-Chloro-4-[(2-oxo-1,3-dihydroindol-5-yl)amino]pyrimidin-2-yl]piperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661648	CN1N=C(C2CCC(=O)NC2=O)C2=CC=C(NC3CCN(C4=NC=C(Cl)C(NC5=CC6=C(C=C5)NC(=O)C6)=N4)CC3)C=C21	C30H30ClN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-YDJALG	SCHEMBL26621392	3-[6-[[1-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-3,3-difluoropiperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661623	CN1N=C(C2CCC(=O)NC2=O)C2=C1C=C(NC1CCN(C3=NC=C(Cl)C(NC4=CC5=C(C=C4)N(C)C(=O)C5)=N3)CC1(F)F)C=C2	C31H30ClF2N9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-QZT1OA	SCHEMBL26621547	1-[6-[[1-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-3,3-difluoropiperidin-4-yl]amino]-1-methylindazol-3-yl]-1,3-diazinane-2,4-dione; SCHEMBL30661656	CN1N=C(N2CCC(=O)NC2=O)C2=C1C=C(NC1CCN(C3=NC=C(Cl)C(NC4=CC5=C(C=C4)N(C)C(=O)C5)=N3)CC1(F)F)C=C2	C30H29ClF2N10O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-DD2B3V	SCHEMBL26621388	3-[6-[[(4R)-1-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-3,3-difluoropiperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661624	CN1N=C(C2CCC(=O)NC2=O)C2=C1C=C(N[C@@H]1CCN(C3=NC=C(Cl)C(NC4=CC5=C(C=C4)N(C)C(=O)C5)=N3)CC1(F)F)C=C2	C31H30ClF2N9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-MXX0J9	SCHEMBL26621395	3-[6-[[(4S)-1-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-3,3-difluoropiperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661516	CN1N=C(C2CCC(=O)NC2=O)C2=C1C=C(N[C@H]1CCN(C3=NC=C(Cl)C(NC4=CC5=C(C=C4)N(C)C(=O)C5)=N3)CC1(F)F)C=C2	C31H30ClF2N9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-3RGH5S	SCHEMBL26621586	3-[6-[4-[[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]amino]-3,3-difluoropiperidin-1-yl]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661560	CN1N=C(C2CCC(=O)NC2=O)C2=CC=C(N3CCC(NC4=NC=C(Cl)C(NC5=CC6=C(C=C5)N(C)C(=O)C6)=N4)C(F)(F)C3)C=C21	C31H30ClF2N9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-JGUHLC	SCHEMBL26621615	3-[6-[[(3R,4R)-1-[5-chloro-4-[(1-ethyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-3-methylpiperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661523	CCN1C(=O)CC2=CC(NC3=NC(N4CC[C@@H](NC5=CC6=C(C=C5)C(C5CCC(=O)NC5=O)=NN6C)[C@H](C)C4)=NC=C3Cl)=CC=C21	C33H36ClN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-SANNVD	BMS-986458	CID 169265594; 3005272-36-3; SCHEMBL26621427; SCHEMBL30661533; GTPL13838; EX-A12465; 3-[6-[[(3R,4R)-1-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-3-methylpiperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione	C[C@@H]1CN(C2=NC(NC3=CC=C4C(=C3)CC(=O)N4C)=C(Cl)C=N2)CC[C@H]1NC1=CC2=C(C=C1)C(C1CCC(=O)NC1=O)=NN2C	C32H34ClN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-6WRGKL	SCHEMBL26621693	(3R)-3-[6-[[(3R,4R)-1-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-3-methylpiperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661627	C[C@@H]1CN(C2=NC=C(Cl)C(NC3=CC=C4C(=C3)CC(=O)N4C)=N2)CC[C@H]1NC1=CC2=C(C=C1)C([C@H]1CCC(=O)NC1=O)=NN2C	C32H34ClN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-W4ENJT	SCHEMBL26621495	(3S)-3-[6-[[(3R,4R)-1-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-3-methylpiperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661550	C[C@@H]1CN(C2=NC=C(Cl)C(NC3=CC=C4C(=C3)CC(=O)N4C)=N2)CC[C@H]1NC1=CC2=C(C=C1)C([C@@H]1CCC(=O)NC1=O)=NN2C	C32H34ClN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-DZZG26	SCHEMBL26621605	3-[6-[[(3R,4R)-1-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-3-methylpiperidin-4-yl]-methylamino]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661626	C[C@@H]1CN(C2=NC=C(Cl)C(NC3=CC=C4C(=C3)CC(=O)N4C)=N2)CC[C@H]1N(C)C1=CC=C2C(=C1)N(C)N=C2C1CCC(=O)NC1=O	C33H36ClN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-ETRIAE	SCHEMBL26621571	3-[6-[[(3R,4R)-1-[5-chloro-4-[(1-methyl-2-oxo-3H-pyrrolo[2,3-b]pyridin-5-yl)amino]pyrimidin-2-yl]-3-methylpiperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661475	C[C@@H]1CN(C2=NC=C(Cl)C(NC3=CN=C4C(=C3)CC(=O)N4C)=N2)CC[C@H]1NC1=CC2=C(C=C1)C(C1CCC(=O)NC1=O)=NN2C	C31H33ClN10O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-5DDVBW	SCHEMBL26621393	3-[6-[[(3R,4R)-1-[5-chloro-4-[[1-(2-methoxyethyl)-2-oxo-3H-indol-5-yl]amino]pyrimidin-2-yl]-3-methylpiperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661485	COCCN1C(=O)CC2=CC(NC3=C(Cl)C=NC(N4CC[C@@H](NC5=CC6=C(C=C5)C(C5CCC(=O)NC5=O)=NN6C)[C@H](C)C4)=N3)=CC=C21	C34H38ClN9O4	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-05OTN0	SCHEMBL26621554	(3R)-3-[6-[[(3R,4R)-1-[5-chloro-4-[[1-(2-methoxyethyl)-2-oxo-3H-indol-5-yl]amino]pyrimidin-2-yl]-3-methylpiperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661580	COCCN1C(=O)CC2=CC(NC3=C(Cl)C=NC(N4CC[C@@H](NC5=CC6=C(C=C5)C([C@H]5CCC(=O)NC5=O)=NN6C)[C@H](C)C4)=N3)=CC=C21	C34H38ClN9O4	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-TN143D	SCHEMBL26621478	(3S)-3-[6-[[(3R,4R)-1-[5-chloro-4-[[1-(2-methoxyethyl)-2-oxo-3H-indol-5-yl]amino]pyrimidin-2-yl]-3-methylpiperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661474	COCCN1C(=O)CC2=CC(NC3=C(Cl)C=NC(N4CC[C@@H](NC5=CC6=C(C=C5)C([C@@H]5CCC(=O)NC5=O)=NN6C)[C@H](C)C4)=N3)=CC=C21	C34H38ClN9O4	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-OXLWQ9	SCHEMBL26621521	3-[6-[(2R,6R)-4-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-2,6-dimethylpiperazin-1-yl]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661492	C[C@@H]1CN(C2=NC=C(Cl)C(NC3=CC4=C(C=C3)N(C)C(=O)C4)=N2)C[C@@H](C)N1C1=CC2=C(C=C1)C(C1CCC(=O)NC1=O)=NN2C	C32H34ClN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-3TQ35X	SCHEMBL26621599	(3R)-3-[6-[(2R,6R)-4-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-2,6-dimethylpiperazin-1-yl]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661597	C[C@@H]1CN(C2=NC=C(Cl)C(NC3=CC4=C(C=C3)N(C)C(=O)C4)=N2)C[C@@H](C)N1C1=CC2=C(C=C1)C([C@H]1CCC(=O)NC1=O)=NN2C	C32H34ClN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-0YMV6K	SCHEMBL26621631	(3S)-3-[6-[(2R,6R)-4-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-2,6-dimethylpiperazin-1-yl]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661611	C[C@@H]1CN(C2=NC=C(Cl)C(NC3=CC4=C(C=C3)N(C)C(=O)C4)=N2)C[C@@H](C)N1C1=CC2=C(C=C1)C([C@@H]1CCC(=O)NC1=O)=NN2C	C32H34ClN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-BSV3IA	SCHEMBL26621467	3-[6-[[(2S,4R)-1-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-2-methylpiperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661659	C[C@H]1C[C@H](NC2=CC3=C(C=C2)C(C2CCC(=O)NC2=O)=NN3C)CCN1C1=NC(NC2=CC=C3C(=C2)CC(=O)N3C)=C(Cl)C=N1	C32H34ClN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-O4OA68	SCHEMBL26621649	(3R)-3-[6-[[(2S,4R)-1-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-2-methylpiperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661599	C[C@H]1C[C@H](NC2=CC3=C(C=C2)C([C@H]2CCC(=O)NC2=O)=NN3C)CCN1C1=NC(NC2=CC=C3C(=C2)CC(=O)N3C)=C(Cl)C=N1	C32H34ClN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-Y9XT6C	SCHEMBL26621549	(3S)-3-[6-[[(2S,4R)-1-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-2-methylpiperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661640	C[C@H]1C[C@H](NC2=CC3=C(C=C2)C([C@@H]2CCC(=O)NC2=O)=NN3C)CCN1C1=NC(NC2=CC=C3C(=C2)CC(=O)N3C)=C(Cl)C=N1	C32H34ClN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-8YV6IG	SCHEMBL26621635	3-[6-[[(2S,4R)-1-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-2-methylpiperidin-4-yl]-methylamino]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661524	C[C@H]1C[C@H](N(C)C2=CC3=C(C=C2)C(C2CCC(=O)NC2=O)=NN3C)CCN1C1=NC(NC2=CC=C3C(=C2)CC(=O)N3C)=C(Cl)C=N1	C33H36ClN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-S9XNS1	SCHEMBL26621655	3-[6-[[(3R,4R)-1-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-3-methylpiperidin-4-yl]amino]-1-methylindazol-3-yl]-3-methylpiperidine-2,6-dione; SCHEMBL30661571	C[C@@H]1CN(C2=NC(NC3=CC=C4C(=C3)CC(=O)N4C)=C(Cl)C=N2)CC[C@H]1NC1=CC=C2C(=C1)N(C)N=C2C1(C)CCC(=O)NC1=O	C33H36ClN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-RF9034	SCHEMBL26621692	3-[6-[[(3R,4R)-1-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-3-methylpiperidin-4-yl]amino]-1-methylpyrazolo[4,3-c]pyridin-3-yl]piperidine-2,6-dione; SCHEMBL30661583	C[C@@H]1CN(C2=NC=C(Cl)C(NC3=CC=C4C(=C3)CC(=O)N4C)=N2)CC[C@H]1NC1=CC2=C(C=N1)C(C1CCC(=O)NC1=O)=NN2C	C31H33ClN10O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-WFIAR6	SCHEMBL26621697	(3R)-3-[6-[[(2S,4R)-1-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-2-methylpiperidin-4-yl]-methylamino]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661467	C[C@H]1C[C@H](N(C)C2=CC3=C(C=C2)C([C@H]2CCC(=O)NC2=O)=NN3C)CCN1C1=NC(NC2=CC=C3C(=C2)CC(=O)N3C)=C(Cl)C=N1	C33H36ClN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-GSV6DB	SCHEMBL26621689	(3S)-3-[6-[[(2S,4R)-1-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-2-methylpiperidin-4-yl]-methylamino]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661618	C[C@H]1C[C@H](N(C)C2=CC3=C(C=C2)C([C@@H]2CCC(=O)NC2=O)=NN3C)CCN1C1=NC(NC2=CC=C3C(=C2)CC(=O)N3C)=C(Cl)C=N1	C33H36ClN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-B4JBE3	SCHEMBL26621440	3-[6-[[1-[5-chloro-4-[(1-ethyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]piperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661612	CCN1C(=O)CC2=CC(NC3=C(Cl)C=NC(N4CCC(NC5=CC6=C(C=C5)C(C5CCC(=O)NC5=O)=NN6C)CC4)=N3)=CC=C21	C32H34ClN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-KOJZ8S	SCHEMBL26621435	(3R)-3-[6-[[1-[5-chloro-4-[(1-ethyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]piperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661584	CCN1C(=O)CC2=CC(NC3=C(Cl)C=NC(N4CCC(NC5=CC6=C(C=C5)C([C@H]5CCC(=O)NC5=O)=NN6C)CC4)=N3)=CC=C21	C32H34ClN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-4FUWTM	SCHEMBL26621436	(3S)-3-[6-[[1-[5-chloro-4-[(1-ethyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]piperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661636	CCN1C(=O)CC2=CC(NC3=C(Cl)C=NC(N4CCC(NC5=CC6=C(C=C5)C([C@@H]5CCC(=O)NC5=O)=NN6C)CC4)=N3)=CC=C21	C32H34ClN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-6BIR3L	SCHEMBL26621403	3-[6-[[(3R,4R)-1-[5-chloro-4-[(6-fluoro-1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-3-methylpiperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661484	C[C@@H]1CN(C2=NC=C(Cl)C(NC3=CC4=C(C=C3F)N(C)C(=O)C4)=N2)CC[C@H]1NC1=CC2=C(C=C1)C(C1CCC(=O)NC1=O)=NN2C	C32H33ClFN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-8E88QX	SCHEMBL26621410	(3R)-3-[6-[[(3R,4R)-1-[5-chloro-4-[(6-fluoro-1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-3-methylpiperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661513	C[C@@H]1CN(C2=NC=C(Cl)C(NC3=CC4=C(C=C3F)N(C)C(=O)C4)=N2)CC[C@H]1NC1=CC2=C(C=C1)C([C@H]1CCC(=O)NC1=O)=NN2C	C32H33ClFN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-MDTODL	SCHEMBL26621401	(3S)-3-[6-[[(3R,4R)-1-[5-chloro-4-[(6-fluoro-1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-3-methylpiperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661546	C[C@@H]1CN(C2=NC=C(Cl)C(NC3=CC4=C(C=C3F)N(C)C(=O)C4)=N2)CC[C@H]1NC1=CC2=C(C=C1)C([C@@H]1CCC(=O)NC1=O)=NN2C	C32H33ClFN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-2ZG7WS	SCHEMBL26621402	3-[6-[[(3R,4R)-1-[5-chloro-4-[(7-fluoro-1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-3-methylpiperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661596	C[C@@H]1CN(C2=NC=C(Cl)C(NC3=CC(F)=C4C(=C3)CC(=O)N4C)=N2)CC[C@H]1NC1=CC2=C(C=C1)C(C1CCC(=O)NC1=O)=NN2C	C32H33ClFN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-AVWL5L	SCHEMBL26621414	(3R)-3-[6-[[(3R,4R)-1-[5-chloro-4-[(7-fluoro-1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-3-methylpiperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661607	C[C@@H]1CN(C2=NC=C(Cl)C(NC3=CC(F)=C4C(=C3)CC(=O)N4C)=N2)CC[C@H]1NC1=CC2=C(C=C1)C([C@H]1CCC(=O)NC1=O)=NN2C	C32H33ClFN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-4GYM55	SCHEMBL26621515	(3S)-3-[6-[[(3R,4R)-1-[5-chloro-4-[(7-fluoro-1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-3-methylpiperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661588	C[C@@H]1CN(C2=NC=C(Cl)C(NC3=CC(F)=C4C(=C3)CC(=O)N4C)=N2)CC[C@H]1NC1=CC2=C(C=C1)C([C@@H]1CCC(=O)NC1=O)=NN2C	C32H33ClFN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-AE2L52	SCHEMBL26621446	3-[6-[[(3R,4R)-1-[5-chloro-4-[(4-fluoro-1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-3-methylpiperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661528	C[C@@H]1CN(C2=NC=C(Cl)C(NC3=CC=C4C(=C3F)CC(=O)N4C)=N2)CC[C@H]1NC1=CC2=C(C=C1)C(C1CCC(=O)NC1=O)=NN2C	C32H33ClFN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-V2NQQ0	SCHEMBL26621680	(3R)-3-[6-[[(3R,4R)-1-[5-chloro-4-[(4-fluoro-1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-3-methylpiperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661639	C[C@@H]1CN(C2=NC=C(Cl)C(NC3=CC=C4C(=C3F)CC(=O)N4C)=N2)CC[C@H]1NC1=CC2=C(C=C1)C([C@H]1CCC(=O)NC1=O)=NN2C	C32H33ClFN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-EHSB8X	SCHEMBL26621441	(3S)-3-[6-[[(3R,4R)-1-[5-chloro-4-[(4-fluoro-1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-3-methylpiperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661566	C[C@@H]1CN(C2=NC=C(Cl)C(NC3=CC=C4C(=C3F)CC(=O)N4C)=N2)CC[C@H]1NC1=CC2=C(C=C1)C([C@@H]1CCC(=O)NC1=O)=NN2C	C32H33ClFN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-J1F07H	SCHEMBL26621454	3-[6-[[(3R,4R)-1-[5-chloro-4-[[1-(2-morpholin-4-ylethyl)-2-oxo-3H-indol-5-yl]amino]pyrimidin-2-yl]-3-methylpiperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661635	C[C@@H]1CN(C2=NC(NC3=CC=C4C(=C3)CC(=O)N4CCN3CCOCC3)=C(Cl)C=N2)CC[C@H]1NC1=CC2=C(C=C1)C(C1CCC(=O)NC1=O)=NN2C	C37H43ClN10O4	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-1ZOFYN	SCHEMBL26621603	(3R)-3-[6-[[(3R,4R)-1-[5-chloro-4-[[1-(2-morpholin-4-ylethyl)-2-oxo-3H-indol-5-yl]amino]pyrimidin-2-yl]-3-methylpiperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661569	C[C@@H]1CN(C2=NC(NC3=CC=C4C(=C3)CC(=O)N4CCN3CCOCC3)=C(Cl)C=N2)CC[C@H]1NC1=CC2=C(C=C1)C([C@H]1CCC(=O)NC1=O)=NN2C	C37H43ClN10O4	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-PH6546	SCHEMBL26621449	(3S)-3-[6-[[(3R,4R)-1-[5-chloro-4-[[1-(2-morpholin-4-ylethyl)-2-oxo-3H-indol-5-yl]amino]pyrimidin-2-yl]-3-methylpiperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661646	C[C@@H]1CN(C2=NC(NC3=CC=C4C(=C3)CC(=O)N4CCN3CCOCC3)=C(Cl)C=N2)CC[C@H]1NC1=CC2=C(C=C1)C([C@@H]1CCC(=O)NC1=O)=NN2C	C37H43ClN10O4	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-33ZI24	SCHEMBL26621481	3-[6-[[(3R,4R)-1-[5-chloro-4-[[1-[2-(methylamino)ethyl]-2-oxo-3H-indol-5-yl]amino]pyrimidin-2-yl]-3-methylpiperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661601	CNCCN1C(=O)CC2=CC(NC3=C(Cl)C=NC(N4CC[C@@H](NC5=CC6=C(C=C5)C(C5CCC(=O)NC5=O)=NN6C)[C@H](C)C4)=N3)=CC=C21	C34H39ClN10O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-F4X21C	SCHEMBL26621696	(3R)-3-[6-[[(3R,4R)-1-[5-chloro-4-[[1-[2-(methylamino)ethyl]-2-oxo-3H-indol-5-yl]amino]pyrimidin-2-yl]-3-methylpiperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661621	CNCCN1C(=O)CC2=CC(NC3=C(Cl)C=NC(N4CC[C@@H](NC5=CC6=C(C=C5)C([C@H]5CCC(=O)NC5=O)=NN6C)[C@H](C)C4)=N3)=CC=C21	C34H39ClN10O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-IMW1Y0	SCHEMBL26621661	(3S)-3-[6-[[(3R,4R)-1-[5-chloro-4-[[1-[2-(methylamino)ethyl]-2-oxo-3H-indol-5-yl]amino]pyrimidin-2-yl]-3-methylpiperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661489	CNCCN1C(=O)CC2=CC(NC3=C(Cl)C=NC(N4CC[C@@H](NC5=CC6=C(C=C5)C([C@@H]5CCC(=O)NC5=O)=NN6C)[C@H](C)C4)=N3)=CC=C21	C34H39ClN10O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-43QIDL	SCHEMBL26621683	3-[6-[[(3R,4R)-1-[5-chloro-4-[[1-(3-fluoro-3-methylbutyl)-2-oxo-3H-indol-5-yl]amino]pyrimidin-2-yl]-3-methylpiperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661507	C[C@@H]1CN(C2=NC(NC3=CC=C4C(=C3)CC(=O)N4CCC(C)(C)F)=C(Cl)C=N2)CC[C@H]1NC1=CC2=C(C=C1)C(C1CCC(=O)NC1=O)=NN2C	C36H41ClFN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-TEBLH2	SCHEMBL26621678	(3R)-3-[6-[[(3R,4R)-1-[5-chloro-4-[[1-(3-fluoro-3-methylbutyl)-2-oxo-3H-indol-5-yl]amino]pyrimidin-2-yl]-3-methylpiperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661595	C[C@@H]1CN(C2=NC(NC3=CC=C4C(=C3)CC(=O)N4CCC(C)(C)F)=C(Cl)C=N2)CC[C@H]1NC1=CC2=C(C=C1)C([C@H]1CCC(=O)NC1=O)=NN2C	C36H41ClFN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-G3QDDG	SCHEMBL26621698	(3S)-3-[6-[[(3R,4R)-1-[5-chloro-4-[[1-(3-fluoro-3-methylbutyl)-2-oxo-3H-indol-5-yl]amino]pyrimidin-2-yl]-3-methylpiperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661518	C[C@@H]1CN(C2=NC(NC3=CC=C4C(=C3)CC(=O)N4CCC(C)(C)F)=C(Cl)C=N2)CC[C@H]1NC1=CC2=C(C=C1)C([C@@H]1CCC(=O)NC1=O)=NN2C	C36H41ClFN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-M3BN7S	SCHEMBL26621501	3-[6-[[(3R,4R)-1-[5-chloro-4-[[1-(2,2-difluoropropyl)-2-oxo-3H-indol-5-yl]amino]pyrimidin-2-yl]-3-methylpiperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661529	C[C@@H]1CN(C2=NC(NC3=CC=C4C(=C3)CC(=O)N4CC(C)(F)F)=C(Cl)C=N2)CC[C@H]1NC1=CC2=C(C=C1)C(C1CCC(=O)NC1=O)=NN2C	C34H36ClF2N9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-J2LEOF	SCHEMBL26621709	(3R)-3-[6-[[(3R,4R)-1-[5-chloro-4-[[1-(2,2-difluoropropyl)-2-oxo-3H-indol-5-yl]amino]pyrimidin-2-yl]-3-methylpiperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661630	C[C@@H]1CN(C2=NC(NC3=CC=C4C(=C3)CC(=O)N4CC(C)(F)F)=C(Cl)C=N2)CC[C@H]1NC1=CC2=C(C=C1)C([C@H]1CCC(=O)NC1=O)=NN2C	C34H36ClF2N9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-RHA5L3	SCHEMBL26621716	(3S)-3-[6-[[(3R,4R)-1-[5-chloro-4-[[1-(2,2-difluoropropyl)-2-oxo-3H-indol-5-yl]amino]pyrimidin-2-yl]-3-methylpiperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661589	C[C@@H]1CN(C2=NC(NC3=CC=C4C(=C3)CC(=O)N4CC(C)(F)F)=C(Cl)C=N2)CC[C@H]1NC1=CC2=C(C=C1)C([C@@H]1CCC(=O)NC1=O)=NN2C	C34H36ClF2N9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-WSFYH1	SCHEMBL26754284	2-[(3R,4R)-4-[[3-(2,6-dioxopiperidin-3-yl)-1-methylindazol-6-yl]amino]-3-methylpiperidin-1-yl]-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidine-5-carbonitrile	C[C@@H]1CN(C2=NC=C(C#N)C(NC3=CC=C4C(=C3)CC(=O)N4C)=N2)CC[C@H]1NC1=CC=C2C(=C1)N(C)N=C2C1CCC(=O)NC1=O	C33H34N10O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-5NFYXF	SCHEMBL26754405	3-[6-[[(3R,4R)-1-[5-chloro-4-[(2-oxo-1,3-dihydroindol-5-yl)amino]pyrimidin-2-yl]-3-methylpiperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione	C[C@@H]1CN(C2=NC=C(Cl)C(NC3=CC=C4NC(=O)CC4=C3)=N2)CC[C@H]1NC1=CC2=C(C=C1)C(C1CCC(=O)NC1=O)=NN2C	C31H32ClN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-TJM27Q	SCHEMBL26754406	3-[6-[[(3R,4R)-1-[5-chloro-4-[(2-oxo-1-propan-2-yl-3H-indol-5-yl)amino]pyrimidin-2-yl]-3-methylpiperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione	CC(C)N1C(=O)CC2=CC(NC3=NC(N4CC[C@@H](NC5=CC6=C(C=C5)C(C5CCC(=O)NC5=O)=NN6C)[C@H](C)C4)=NC=C3Cl)=CC=C21	C34H38ClN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-SA3GZ9	SCHEMBL26754407	2-[(3R,4R)-4-[[3-(2,6-dioxopiperidin-3-yl)-1-methylindazol-6-yl]amino]-3-methylpiperidin-1-yl]-4-[(7-fluoro-1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidine-5-carbonitrile	C[C@@H]1CN(C2=NC(NC3=CC(F)=C4C(=C3)CC(=O)N4C)=C(C#N)C=N2)CC[C@H]1NC1=CC=C2C(=C1)N(C)N=C2C1CCC(=O)NC1=O	C33H33FN10O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-PQ02QS	SCHEMBL26754410	2-[(3R,4R)-4-[[3-(2,6-dioxopiperidin-3-yl)-1-methylindazol-6-yl]amino]-3-methylpiperidin-1-yl]-4-[(6-fluoro-1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidine-5-carbonitrile	C[C@@H]1CN(C2=NC(NC3=C(F)C=C4C(=C3)CC(=O)N4C)=C(C#N)C=N2)CC[C@H]1NC1=CC2=C(C=C1)C(C1CCC(=O)NC1=O)=NN2C	C33H33FN10O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-U20RTY	SCHEMBL26754412	2-[(3R,4R)-4-[[3-(2,6-dioxopiperidin-3-yl)-1-methylindazol-6-yl]amino]-3-methylpiperidin-1-yl]-4-[(4-fluoro-1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidine-5-carbonitrile	C[C@@H]1CN(C2=NC=C(C#N)C(NC3=CC=C4C(=C3F)CC(=O)N4C)=N2)CC[C@H]1NC1=CC2=C(C=C1)C(C1CCC(=O)NC1=O)=NN2C	C33H33FN10O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-XC062Z	SCHEMBL26754413	3-[6-[[(3R,4R)-1-[5-chloro-4-[[2-oxo-1-(4,4,4-trifluorobutyl)-3H-indol-5-yl]amino]pyrimidin-2-yl]-3-methylpiperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione	C[C@@H]1CN(C2=NC(NC3=CC=C4C(=C3)CC(=O)N4CCCC(F)(F)F)=C(Cl)C=N2)CC[C@H]1NC1=CC2=C(C=C1)C(C1CCC(=O)NC1=O)=NN2C	C35H37ClF3N9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-OJXRNV	SCHEMBL26754415	3-[6-[[(3R,4R)-1-[5-chloro-4-[[1-(3-hydroxy-3-methylbutyl)-2-oxo-3H-indol-6-yl]amino]pyrimidin-2-yl]-3-methylpiperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL31444695	C[C@@H]1CN(C2=NC(NC3=CC=C4CC(=O)N(CCC(C)(C)O)C4=C3)=C(Cl)C=N2)CC[C@H]1NC1=CC2=C(C=C1)C(C1CCC(=O)NC1=O)=NN2C	C36H42ClN9O4	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-YP4ZLY	SCHEMBL26754418	3-[6-[[(3R,4R)-1-[5-chloro-4-[[1-(2-fluoro-2-methylpropyl)-2-oxo-3H-indol-5-yl]amino]pyrimidin-2-yl]-3-methylpiperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione	C[C@@H]1CN(C2=NC(NC3=CC=C4C(=C3)CC(=O)N4CC(C)(C)F)=C(Cl)C=N2)CC[C@H]1NC1=CC2=C(C=C1)C(C1CCC(=O)NC1=O)=NN2C	C35H39ClFN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-PJCA2K	SCHEMBL27033171	3-[6-[[(3R,4R)-1-[5-chloro-4-methyl-6-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-3-methylpiperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione	CC1=C(Cl)C(NC2=CC=C3C(=C2)CC(=O)N3C)=NC(N2CC[C@@H](NC3=CC4=C(C=C3)C(C3CCC(=O)NC3=O)=NN4C)[C@H](C)C2)=N1	C33H36ClN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-6932HJ	SCHEMBL26754546	3-[6-[[(3R,4R)-1-[5-chloro-4-fluoro-6-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-3-methylpiperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione	C[C@@H]1CN(C2=NC(F)=C(Cl)C(NC3=CC4=C(C=C3)N(C)C(=O)C4)=N2)CC[C@H]1NC1=CC=C2C(=C1)N(C)N=C2C1CCC(=O)NC1=O	C32H33ClFN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-3UB0UO	SCHEMBL26621575	3-[6-[1-[5-Chloro-4-[(2-oxo-1,3-dihydroindol-5-yl)amino]pyrimidin-2-yl]piperidin-4-yl]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661526	CN1N=C(C2CCC(=O)NC2=O)C2=CC=C(C3CCN(C4=NC=C(Cl)C(NC5=CC6=C(C=C5)NC(=O)C6)=N4)CC3)C=C21	C30H29ClN8O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-MQGWL7	SCHEMBL26621702	3-[6-[1-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]piperidin-4-yl]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661478	CN1N=C(C2CCC(=O)NC2=O)C2=CC=C(C3CCN(C4=NC=C(Cl)C(NC5=CC6=C(C=C5)N(C)C(=O)C6)=N4)CC3)C=C21	C31H31ClN8O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-EH4MDN	SCHEMBL26621437	3-[6-[4-[[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]amino]-2-oxopiperidin-1-yl]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661568	CN1N=C(C2CCC(=O)NC2=O)C2=C1C=C(N1CCC(NC3=NC(NC4=CC=C5C(=C4)CC(=O)N5C)=C(Cl)C=N3)CC1=O)C=C2	C31H30ClN9O4	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-O6QMXR	SCHEMBL26621524	3-[6-[4-[[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-methylamino]-2-oxopiperidin-1-yl]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661561	CN1N=C(C2CCC(=O)NC2=O)C2=C1C=C(N1CCC(N(C)C3=NC(NC4=CC=C5C(=C4)CC(=O)N5C)=C(Cl)C=N3)CC1=O)C=C2	C32H32ClN9O4	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-NHH52B	SCHEMBL26621701	3-[6-[(4S)-4-[[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-methylamino]-2-oxopiperidin-1-yl]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661577	CN1N=C(C2CCC(=O)NC2=O)C2=C1C=C(N1CC[C@H](N(C)C3=NC(NC4=CC=C5C(=C4)CC(=O)N5C)=C(Cl)C=N3)CC1=O)C=C2	C32H32ClN9O4	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-Y9NA5P	SCHEMBL26621517	3-[6-[(4R)-4-[[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-methylamino]-2-oxopiperidin-1-yl]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661469	CN1N=C(C2CCC(=O)NC2=O)C2=C1C=C(N1CC[C@@H](N(C)C3=NC(NC4=CC=C5C(=C4)CC(=O)N5C)=C(Cl)C=N3)CC1=O)C=C2	C32H32ClN9O4	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-FEZGDI	SCHEMBL26621497	3-[6-[(3R,4S)-4-[[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-methylamino]-3-methyl-2-oxopiperidin-1-yl]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661540; SCHEMBL30661543	C[C@H]1C(=O)N(C2=CC3=C(C=C2)C(C2CCC(=O)NC2=O)=NN3C)CC[C@@H]1N(C)C1=NC(NC2=CC=C3C(=C2)CC(=O)N3C)=C(Cl)C=N1	C33H34ClN9O4	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-VI5Y5V	SCHEMBL26621694	3-[6-[(3S,4R)-4-[[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-methylamino]-3-methyl-2-oxopiperidin-1-yl]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661585	C[C@@H]1C(=O)N(C2=CC3=C(C=C2)C(C2CCC(=O)NC2=O)=NN3C)CC[C@H]1N(C)C1=NC(NC2=CC=C3C(=C2)CC(=O)N3C)=C(Cl)C=N1	C33H34ClN9O4	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-XO7EDJ	SCHEMBL26621731	2-[(3R,4R)-4-[[3-(2,4-dioxo-1,3-diazinan-1-yl)-1-methylindazol-6-yl]amino]-3-methylpiperidin-1-yl]-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidine-5-carbonitrile; SCHEMBL30661644	C[C@@H]1CN(C2=NC=C(C#N)C(NC3=CC=C4C(=C3)CC(=O)N4C)=N2)CC[C@H]1NC1=CC=C2C(=C1)N(C)N=C2N1CCC(=O)NC1=O	C32H33N11O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-FYK3ZT	SCHEMBL26621394	1-[6-[4-[[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]amino]piperidin-1-yl]-1-methylindazol-3-yl]-1,3-diazinane-2,4-dione; SCHEMBL30661622	CN1N=C(N2CCC(=O)NC2=O)C2=CC=C(N3CCC(NC4=NC=C(Cl)C(NC5=CC6=C(C=C5)N(C)C(=O)C6)=N4)CC3)C=C21	C30H31ClN10O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-6THABL	SCHEMBL26621616	1-[6-[1-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]piperidin-4-yl]-1-methylindazol-3-yl]-1,3-diazinane-2,4-dione; SCHEMBL30661582	CN1N=C(N2CCC(=O)NC2=O)C2=C1C=C(C1CCN(C3=NC=C(Cl)C(NC4=CC=C5C(=C4)CC(=O)N5C)=N3)CC1)C=C2	C30H30ClN9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-IJHPDC	SCHEMBL26621450	1-[6-[[1-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]piperidin-4-yl]amino]-1-methylindazol-3-yl]-1,3-diazinane-2,4-dione; SCHEMBL30661632	CN1N=C(N2CCC(=O)NC2=O)C2=C1C=C(NC1CCN(C3=NC(NC4=CC=C5C(=C4)CC(=O)N5C)=C(Cl)C=N3)CC1)C=C2	C30H31ClN10O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-1BYTS4	SCHEMBL26621657	1-[6-[[1-[5-chloro-4-[[2-oxo-1-(2,2,2-trifluoroethyl)-3H-indol-5-yl]amino]pyrimidin-2-yl]piperidin-4-yl]amino]-1-methylindazol-3-yl]-1,3-diazinane-2,4-dione; SCHEMBL30661512	CN1N=C(N2CCC(=O)NC2=O)C2=C1C=C(NC1CCN(C3=NC(NC4=CC=C5C(=C4)CC(=O)N5CC(F)(F)F)=C(Cl)C=N3)CC1)C=C2	C31H30ClF3N10O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-X9CDAI	SCHEMBL26621428	1-[6-[[1-[5-chloro-4-[[1-(2-hydroxyethyl)-2-oxo-3H-indol-5-yl]amino]pyrimidin-2-yl]piperidin-4-yl]amino]-1-methylindazol-3-yl]-1,3-diazinane-2,4-dione; SCHEMBL30661620	CN1N=C(N2CCC(=O)NC2=O)C2=C1C=C(NC1CCN(C3=NC(NC4=CC=C5C(=C4)CC(=O)N5CCO)=C(Cl)C=N3)CC1)C=C2	C31H33ClN10O4	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-D6KVMF	SCHEMBL26621705	2-[4-[[3-(2,4-dioxo-1,3-diazinan-1-yl)-1-methylindazol-6-yl]amino]piperidin-1-yl]-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidine-5-carbonitrile; SCHEMBL30661537	CN1N=C(N2CCC(=O)NC2=O)C2=C1C=C(NC1CCN(C3=NC(NC4=CC=C5C(=C4)CC(=O)N5C)=C(C#N)C=N3)CC1)C=C2	C31H31N11O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-55OQET	SCHEMBL26621445	1-[6-[[(3R,4R)-1-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-3-methylpiperidin-4-yl]amino]-1-methylindazol-3-yl]pyrimidine-2,4-dione; SCHEMBL30661631	C[C@@H]1CN(C2=NC=C(Cl)C(NC3=CC=C4C(=C3)CC(=O)N4C)=N2)CC[C@H]1NC1=CC2=C(C=C1)C(N1C=CC(=O)NC1=O)=NN2C	C31H31ClN10O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-03TJEJ	SCHEMBL26621608	1-[6-[[(3R,4R)-1-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-3-methylpiperidin-4-yl]amino]-1-methylindazol-3-yl]-5-fluoropyrimidine-2,4-dione; SCHEMBL30661551	C[C@@H]1CN(C2=NC=C(Cl)C(NC3=CC=C4C(=C3)CC(=O)N4C)=N2)CC[C@H]1NC1=CC2=C(C=C1)C(N1C=C(F)C(=O)NC1=O)=NN2C	C31H30ClFN10O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-S57YBU	SCHEMBL26754936	1-[6-[[(3R,4R)-1-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-3-methylpiperidin-4-yl]amino]-1-methylindazol-3-yl]-1,3-diazinane-2,4-dione	C[C@@H]1CN(C2=NC=C(Cl)C(NC3=CC=C4C(=C3)CC(=O)N4C)=N2)CC[C@H]1NC1=CC=C2C(=C1)N(C)N=C2N1CCC(=O)NC1=O	C31H33ClN10O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-TTPYW0	SCHEMBL26755005	1-[6-[[(3R,4R)-1-[5-chloro-4-[(4-fluoro-1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-3-methylpiperidin-4-yl]amino]-1-methylindazol-3-yl]-1,3-diazinane-2,4-dione	C[C@@H]1CN(C2=NC(NC3=CC=C4C(=C3F)CC(=O)N4C)=C(Cl)C=N2)CC[C@H]1NC1=CC2=C(C=C1)C(N1CCC(=O)NC1=O)=NN2C	C31H32ClFN10O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-KHHZSD	SCHEMBL26755006	1-[6-[[(3R,4R)-1-[5-chloro-4-[(1-methyl-2-oxo-3H-pyrrolo[2,3-b]pyridin-5-yl)amino]pyrimidin-2-yl]-3-methylpiperidin-4-yl]amino]-1-methylindazol-3-yl]-1,3-diazinane-2,4-dione	C[C@@H]1CN(C2=NC(NC3=CN=C4C(=C3)CC(=O)N4C)=C(Cl)C=N2)CC[C@H]1NC1=CC=C2C(=C1)N(C)N=C2N1CCC(=O)NC1=O	C30H32ClN11O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-6Y7F3U	SCHEMBL26755008	1-[6-[[1-[5-chloro-4-[(1-ethyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]piperidin-4-yl]amino]-1-methylindazol-3-yl]-1,3-diazinane-2,4-dione	CCN1C(=O)CC2=CC(NC3=C(Cl)C=NC(N4CCC(NC5=CC6=C(C=C5)C(N5CCC(=O)NC5=O)=NN6C)CC4)=N3)=CC=C21	C31H33ClN10O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-IFO2CH	SCHEMBL26621551	2-[(3R,4R)-4-[[3-(2,6-dioxopiperidin-3-yl)-1-methylindazol-6-yl]amino]-3-methoxypiperidin-1-yl]-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidine-5-carbonitrile; SCHEMBL30661575	CO[C@@H]1CN(C2=NC=C(C#N)C(NC3=CC4=C(C=C3)N(C)C(=O)C4)=N2)CC[C@H]1NC1=CC=C2C(=C1)N(C)N=C2C1CCC(=O)NC1=O	C33H34N10O4	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-P9BOF9	SCHEMBL26621626	3-[6-[[(3R,4R)-1-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-3-methoxypiperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661590	CO[C@@H]1CN(C2=NC=C(Cl)C(NC3=CC4=C(C=C3)N(C)C(=O)C4)=N2)CC[C@H]1NC1=CC=C2C(=C1)N(C)N=C2C1CCC(=O)NC1=O	C32H34ClN9O4	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-Q58NAG	SCHEMBL26755085	3-[6-[[(3R,4S)-1-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-3-(trifluoromethyl)piperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione	CN1N=C(C2CCC(=O)NC2=O)C2=C1C=C(N[C@H]1CCN(C3=NC(NC4=CC=C5C(=C4)CC(=O)N5C)=C(Cl)C=N3)C[C@H]1C(F)(F)F)C=C2	C32H31ClF3N9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-EIHW58	SCHEMBL26621682	3-[6-[[(3S,4R)-1-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-3-(trifluoromethyl)piperidin-4-yl]amino]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661565	CN1N=C(C2CCC(=O)NC2=O)C2=C1C=C(N[C@@H]1CCN(C3=NC(NC4=CC=C5C(=C4)CC(=O)N5C)=C(Cl)C=N3)C[C@@H]1C(F)(F)F)C=C2	C32H31ClF3N9O3	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-HLU46H	SCHEMBL26621421	3-[6-[(4R,5S)-4-[[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-methylamino]-5-methyl-2-oxopiperidin-1-yl]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661563	C[C@H]1CN(C2=CC=C3C(=C2)N(C)N=C3C2CCC(=O)NC2=O)C(=O)C[C@H]1N(C)C1=NC(NC2=CC3=C(C=C2)N(C)C(=O)C3)=C(Cl)C=N1	C33H34ClN9O4	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-2MVJJN	SCHEMBL26621757	3-[6-[(2R,4S)-4-[[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-methylamino]-2-methyl-6-oxopiperidin-1-yl]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661482	C[C@@H]1C[C@H](N(C)C2=NC(NC3=CC4=C(C=C3)N(C)C(=O)C4)=C(Cl)C=N2)CC(=O)N1C1=CC2=C(C=C1)C(C1CCC(=O)NC1=O)=NN2C	C33H34ClN9O4	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-CVVFHS	SCHEMBL26621641	3-[6-[(2R,4R)-4-[[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-methylamino]-2-methyl-6-oxopiperidin-1-yl]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661602	C[C@@H]1C[C@@H](N(C)C2=NC(NC3=CC4=C(C=C3)N(C)C(=O)C4)=C(Cl)C=N2)CC(=O)N1C1=CC2=C(C=C1)C(C1CCC(=O)NC1=O)=NN2C	C33H34ClN9O4	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-98323L	SCHEMBL26621660	3-[6-[(2S,4R)-4-[[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-methylamino]-2-methyl-6-oxopiperidin-1-yl]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661487	C[C@H]1C[C@@H](N(C)C2=NC(NC3=CC4=C(C=C3)N(C)C(=O)C4)=C(Cl)C=N2)CC(=O)N1C1=CC2=C(C=C1)C(C1CCC(=O)NC1=O)=NN2C	C33H34ClN9O4	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-N4VI01	SCHEMBL26621653	3-[6-[(2S,4S)-4-[[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-methylamino]-2-methyl-6-oxopiperidin-1-yl]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL30661637	C[C@H]1C[C@H](N(C)C2=NC(NC3=CC4=C(C=C3)N(C)C(=O)C4)=C(Cl)C=N2)CC(=O)N1C1=CC2=C(C=C1)C(C1CCC(=O)NC1=O)=NN2C	C33H34ClN9O4	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-EHU4PL	SCHEMBL26621573	3-[6-[[(3R,4R)-1-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-3-methoxypiperidin-4-yl]amino]-1-methylindazol-3-yl]-3-methylpiperidine-2,6-dione; SCHEMBL30661593	CO[C@@H]1CN(C2=NC=C(Cl)C(NC3=CC4=C(C=C3)N(C)C(=O)C4)=N2)CC[C@H]1NC1=CC=C2C(=C1)N(C)N=C2C1(C)CCC(=O)NC1=O	C33H36ClN9O4	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-M0SGX1	SCHEMBL26621533	2-[(3R,4R)-3-methoxy-4-[[1-methyl-3-(3-methyl-2,6-dioxopiperidin-3-yl)indazol-6-yl]amino]piperidin-1-yl]-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidine-5-carbonitrile; SCHEMBL30661633	CO[C@@H]1CN(C2=NC=C(C#N)C(NC3=CC4=C(C=C3)N(C)C(=O)C4)=N2)CC[C@H]1NC1=CC=C2C(=C1)N(C)N=C2C1(C)CCC(=O)NC1=O	C34H36N10O4	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-G0YHFA	SCHEMBL26621672	1-[6-[[(3R,4R)-1-[5-chloro-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-3-methoxypiperidin-4-yl]amino]-1-methylindazol-3-yl]-1,3-diazinane-2,4-dione	CO[C@@H]1CN(C2=NC=C(Cl)C(NC3=CC4=C(C=C3)N(C)C(=O)C4)=N2)CC[C@H]1NC1=CC=C2C(=C1)N(C)N=C2N1CCC(=O)NC1=O	C31H33ClN10O4	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-K90EP6	SCHEMBL26621559	2-[(3R,4R)-4-[[3-(2,4-dioxo-1,3-diazinan-1-yl)-1-methylindazol-6-yl]amino]-3-methoxypiperidin-1-yl]-4-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidine-5-carbonitrile; SCHEMBL30661547	CO[C@@H]1CN(C2=NC=C(C#N)C(NC3=CC4=C(C=C3)N(C)C(=O)C4)=N2)CC[C@H]1NC1=CC=C2C(=C1)N(C)N=C2N1CCC(=O)NC1=O	C32H33N11O4	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-FTP3XL	SCHEMBL26621728	1-[6-[[(3R,4R)-1-[5-chloro-4-fluoro-6-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-3-methoxypiperidin-4-yl]amino]-1-methylindazol-3-yl]-1,3-diazinane-2,4-dione; SCHEMBL30661496	CO[C@@H]1CN(C2=NC(F)=C(Cl)C(NC3=CC4=C(C=C3)N(C)C(=O)C4)=N2)CC[C@H]1NC1=CC=C2C(=C1)N(C)N=C2N1CCC(=O)NC1=O	C31H32ClFN10O4	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-3LXVGZ	SCHEMBL26621400	3-[6-[[(3R,4R)-1-[5-chloro-4-fluoro-6-[(1-methyl-2-oxo-3H-indol-5-yl)amino]pyrimidin-2-yl]-3-methoxypiperidin-4-yl]amino]-1-methylindazol-3-yl]-3-methylpiperidine-2,6-dione; SCHEMBL30661538	CO[C@@H]1CN(C2=NC(F)=C(Cl)C(NC3=CC4=C(C=C3)N(C)C(=O)C4)=N2)CC[C@H]1NC1=CC=C2C(=C1)N(C)N=C2C1(C)CCC(=O)NC1=O	C33H35ClFN9O4	BCL6	P41182	CRBN	WO-2023212147-A1
TPD-ELLJS1	SCHEMBL26625074	[4-[3-[4-[4-[3-[4-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]propyl]piperazin-1-yl]phenoxy]-6-hydroxy-1-benzothiophen-2-yl]phenyl]boronic acid; SCHEMBL30619776	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCCN5CCN(C6=CC=C(OC7=C(C8=CC=C(B(O)O)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C44H45BN6O8S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-RBV8SM	SCHEMBL26625228	[4-[3-[4-[4-[3-[4-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]propyl]piperazin-1-yl]benzoyl]-6-hydroxy-1-benzothiophen-2-yl]phenyl]boronic acid; SCHEMBL30619786	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCCN5CCN(C6=CC=C(C(=O)C7=C(C8=CC=C(B(O)O)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C45H45BN6O8S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-RDBUYP	SCHEMBL26625205	[4-[3-[4-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]propyl]piperazin-1-yl]phenoxy]-6-hydroxy-1-benzothiophen-2-yl]phenyl]boronic acid; SCHEMBL30619819	O=C1CCC(N2CC3=CC(N4CCN(CCCN5CCN(C6=CC=C(OC7=C(C8=CC=C(B(O)O)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C44H47BN6O7S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-TNFR3R	SCHEMBL26625090	[4-[3-[4-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]propyl]piperazin-1-yl]benzoyl]-6-hydroxy-1-benzothiophen-2-yl]phenyl]boronic acid; SCHEMBL30619762	O=C1CCC(N2CC3=CC(N4CCN(CCCN5CCN(C6=CC=C(C(=O)C7=C(C8=CC=C(B(O)O)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C45H47BN6O7S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-GXE0QU	SCHEMBL26625198	[3-[4-[4-[3-[4-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]propyl]piperazin-1-yl]phenoxy]-2-(4-fluorophenyl)-1-benzothiophen-6-yl]boronic acid; SCHEMBL30619820	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCCN5CCN(C6=CC=C(OC7=C(C8=CC=C(F)C=C8)SC8=C7C=CC(B(O)O)=C8)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C44H44BFN6O7S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-GTB72V	SCHEMBL26625129	[3-[4-[4-[3-[4-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]propyl]piperazin-1-yl]benzoyl]-2-(4-fluorophenyl)-1-benzothiophen-6-yl]boronic acid; SCHEMBL30619760	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCCN5CCN(C6=CC=C(C(=O)C7=C(C8=CC=C(F)C=C8)SC8=C7C=CC(B(O)O)=C8)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C45H44BFN6O7S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-BMJGPU	SCHEMBL26625159	[3-[4-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]propyl]piperazin-1-yl]phenoxy]-2-(4-fluorophenyl)-1-benzothiophen-6-yl]boronic acid; SCHEMBL30619711	O=C1CCC(N2CC3=CC(N4CCN(CCCN5CCN(C6=CC=C(OC7=C(C8=CC=C(F)C=C8)SC8=C7C=CC(B(O)O)=C8)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C44H46BFN6O6S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-W53QUT	SCHEMBL26625130	[3-[4-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]propyl]piperazin-1-yl]benzoyl]-2-(4-fluorophenyl)-1-benzothiophen-6-yl]boronic acid; SCHEMBL30619740	O=C1CCC(N2CC3=CC(N4CCN(CCCN5CCN(C6=CC=C(C(=O)C7=C(C8=CC=C(F)C=C8)SC8=C7C=CC(B(O)O)=C8)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C45H46BFN6O6S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-H2ERRZ	SCHEMBL26625034	2-(2,6-Dioxopiperidin-3-yl)-5-[4-[3-[4-[4-[[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenyl]piperazin-1-yl]propyl]piperazin-1-yl]isoindole-1,3-dione; SCHEMBL30619701	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCCN5CCN(C6=CC=C(OC7=C(C8=CC=C(F)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C44H43FN6O6S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-X5MSQ7	SCHEMBL26625046	2-(2,6-Dioxopiperidin-3-yl)-5-[4-[3-[4-[4-[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophene-3-carbonyl]phenyl]piperazin-1-yl]propyl]piperazin-1-yl]isoindole-1,3-dione; SCHEMBL30619706	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCCN5CCN(C6=CC=C(C(=O)C7=C(C8=CC=C(F)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C45H43FN6O6S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-8KI8WK	SCHEMBL26625295	3-[6-[4-[3-[4-[4-[[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenyl]piperazin-1-yl]propyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30619739	O=C1CCC(N2CC3=CC(N4CCN(CCCN5CCN(C6=CC=C(OC7=C(C8=CC=C(F)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C44H45FN6O5S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-0U8GYM	SCHEMBL26625051	3-[6-[4-[3-[4-[4-[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophene-3-carbonyl]phenyl]piperazin-1-yl]propyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30619788	O=C1CCC(N2CC3=CC(N4CCN(CCCN5CCN(C6=CC=C(C(=O)C7=C(C8=CC=C(F)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C45H45FN6O5S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-IYXWM8	SCHEMBL26625113	2-(2,6-Dioxopiperidin-3-yl)-5-[4-[3-[1-[4-[[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenyl]piperidin-4-yl]propyl]piperazin-1-yl]isoindole-1,3-dione; SCHEMBL30619694	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCCC5CCN(C6=CC=C(OC7=C(C8=CC=C(F)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C45H44FN5O6S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-9R7NGO	SCHEMBL26625137	2-(2,6-Dioxopiperidin-3-yl)-5-[4-[3-[1-[4-[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophene-3-carbonyl]phenyl]piperidin-4-yl]propyl]piperazin-1-yl]isoindole-1,3-dione; SCHEMBL30619697	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCCC5CCN(C6=CC=C(C(=O)C7=C(C8=CC=C(F)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C46H44FN5O6S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-FRE1SM	SCHEMBL26625042	3-[6-[4-[3-[1-[4-[[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenyl]piperidin-4-yl]propyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30619709	O=C1CCC(N2CC3=CC(N4CCN(CCCC5CCN(C6=CC=C(OC7=C(C8=CC=C(F)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C45H46FN5O5S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-KTNU7X	SCHEMBL26625292	3-[6-[4-[3-[1-[4-[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophene-3-carbonyl]phenyl]piperidin-4-yl]propyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30619728	O=C1CCC(N2CC3=CC(N4CCN(CCCC5CCN(C6=CC=C(C(=O)C7=C(C8=CC=C(F)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C46H46FN5O5S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-S3KCT7	SCHEMBL26625479	[4-[3-[4-[4-[3-[1-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]propyl]piperazin-1-yl]phenoxy]-6-hydroxy-1-benzothiophen-2-yl]phenyl]boronic acid; SCHEMBL30619747	O=C1CCC(N2C(=O)C3=CC=C(N4CCC(CCCN5CCN(C6=CC=C(OC7=C(C8=CC=C(B(O)O)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C45H46BN5O8S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-XOLYAU	WO2023212599A9_22	.	O=C1CCC(N2C(=O)C3=CC=C(N4CCC(CCCN5CCN(C6=CC=C(C(=O)C7=C(C8=CC=C(B(O)O)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C46H46BN5O8S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-V1WCHZ	SCHEMBL26625208	[4-[3-[4-[4-[3-[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]propyl]piperazin-1-yl]phenoxy]-6-hydroxy-1-benzothiophen-2-yl]phenyl]boronic acid	O=C1CCC(N2CC3=CC(N4CCC(CCCN5CCN(C6=CC=C(OC7=C(C8=CC=C(B(O)O)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C45H48BN5O7S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-OHNMD9	SCHEMBL26625174	[4-[3-[4-[4-[3-[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]propyl]piperazin-1-yl]benzoyl]-6-hydroxy-1-benzothiophen-2-yl]phenyl]boronic acid; SCHEMBL30619741	O=C1CCC(N2CC3=CC(N4CCC(CCCN5CCN(C6=CC=C(C(=O)C7=C(C8=CC=C(B(O)O)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C46H48BN5O7S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-QUSM35	WO2023212599A9_25	.	CC1=CC=C(C2=C(OC3=CC=C(N4CCN(CCCC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C=C3)C3=C(C=C(O)C=C3)S2)C=C1	C46H47N5O6S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-Y99JUC	SCHEMBL26625230	2-(2,6-Dioxopiperidin-3-yl)-5-[4-[3-[4-[4-[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophene-3-carbonyl]phenyl]piperazin-1-yl]propyl]piperidin-1-yl]isoindole-1,3-dione; SCHEMBL30619796	O=C1CCC(N2C(=O)C3=CC=C(N4CCC(CCCN5CCN(C6=CC=C(C(=O)C7=C(C8=CC=C(F)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C46H44FN5O6S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-1XGWDL	SCHEMBL26625329	3-[6-[4-[3-[4-[4-[[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenyl]piperazin-1-yl]propyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30619814	O=C1CCC(N2CC3=CC(N4CCC(CCCN5CCN(C6=CC=C(OC7=C(C8=CC=C(F)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C45H46FN5O5S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-7R6JNN	SCHEMBL26625182	3-[6-[4-[3-[4-[4-[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophene-3-carbonyl]phenyl]piperazin-1-yl]propyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30619705	O=C1CCC(N2CC3=CC(N4CCC(CCCN5CCN(C6=CC=C(C(=O)C7=C(C8=CC=C(F)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C46H46FN5O5S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-O4CAGX	SCHEMBL26625237	[4-[3-[4-[4-[2-[4-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]ethyl]piperazin-1-yl]phenoxy]-6-hydroxy-1-benzothiophen-2-yl]phenyl]boronic acid; SCHEMBL30619771	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCN5CCN(C6=CC=C(OC7=C(C8=CC=C(B(O)O)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C43H43BN6O8S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-K3JUPE	SCHEMBL26625211	[4-[3-[4-[4-[2-[4-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]ethyl]piperazin-1-yl]benzoyl]-6-hydroxy-1-benzothiophen-2-yl]phenyl]boronic acid; SCHEMBL30619721	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCN5CCN(C6=CC=C(C(=O)C7=C(C8=CC=C(B(O)O)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C44H43BN6O8S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-J4PTX7	SCHEMBL26625176	[4-[3-[4-[4-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]ethyl]piperazin-1-yl]phenoxy]-6-hydroxy-1-benzothiophen-2-yl]phenyl]boronic acid; SCHEMBL30619823	O=C1CCC(N2CC3=CC(N4CCN(CCN5CCN(C6=CC=C(OC7=C(C8=CC=C(B(O)O)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C43H45BN6O7S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-YEBK6H	SCHEMBL26625337	[4-[3-[4-[4-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]ethyl]piperazin-1-yl]benzoyl]-6-hydroxy-1-benzothiophen-2-yl]phenyl]boronic acid; SCHEMBL30619752	O=C1CCC(N2CC3=CC(N4CCN(CCN5CCN(C6=CC=C(C(=O)C7=C(C8=CC=C(B(O)O)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C44H45BN6O7S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-202M5X	SCHEMBL26625199	[3-[4-[4-[2-[4-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]ethyl]piperazin-1-yl]phenoxy]-2-(4-fluorophenyl)-1-benzothiophen-6-yl]boronic acid	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCN5CCN(C6=CC=C(OC7=C(C8=CC=C(F)C=C8)SC8=C7C=CC(B(O)O)=C8)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C43H42BFN6O7S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-WHZHZC	WO2023212599A9_34	.	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCN5CCN(C6=CC=C(C(=O)C7=C(C8=CC=C(F)C=C8)SC8=C7C=CC(B(O)O)=C8)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C44H42BFN6O7S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-ERNMAA	SCHEMBL30619736	[3-[4-[4-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]ethyl]piperazin-1-yl]phenoxy]-2-(4-fluorophenyl)-1-benzothiophen-6-yl]boronic acid	O=C1CCC(N2CC3=CC(N4CCN(CCN5CCN(C6=CC=C(OC7=C(C8=CC=C(F)C=C8)SC8=C7C=CC(B(O)O)=C8)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C43H44BFN6O6S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-44RY43	SCHEMBL26625206	[3-[4-[4-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]ethyl]piperazin-1-yl]benzoyl]-2-(4-fluorophenyl)-1-benzothiophen-6-yl]boronic acid; SCHEMBL30619723	O=C1CCC(N2CC3=CC(N4CCN(CCN5CCN(C6=CC=C(C(=O)C7=C(C8=CC=C(F)C=C8)SC8=C7C=CC(B(O)O)=C8)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C44H44BFN6O6S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-KD3I8V	SCHEMBL26625118	[4-[3-[4-[4-[2-[4-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]ethyl]piperidin-1-yl]phenoxy]-6-hydroxy-1-benzothiophen-2-yl]phenyl]boronic acid; SCHEMBL30619717	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCC5CCN(C6=CC=C(OC7=C(C8=CC=C(B(O)O)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C44H44BN5O8S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-3XJHKC	SCHEMBL26625186	[4-[3-[4-[4-[2-[4-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]ethyl]piperidin-1-yl]benzoyl]-6-hydroxy-1-benzothiophen-2-yl]phenyl]boronic acid; SCHEMBL30619707	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCC5CCN(C6=CC=C(C(=O)C7=C(C8=CC=C(B(O)O)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C45H44BN5O8S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-T5KXXQ	SCHEMBL26625114	[4-[3-[4-[4-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]ethyl]piperidin-1-yl]phenoxy]-6-hydroxy-1-benzothiophen-2-yl]phenyl]boronic acid; SCHEMBL30619712	O=C1CCC(N2CC3=CC(N4CCN(CCC5CCN(C6=CC=C(OC7=C(C8=CC=C(B(O)O)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C44H46BN5O7S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-JMKL5C	SCHEMBL26625080	[4-[3-[4-[4-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]ethyl]piperidin-1-yl]benzoyl]-6-hydroxy-1-benzothiophen-2-yl]phenyl]boronic acid; SCHEMBL30619763	O=C1CCC(N2CC3=CC(N4CCN(CCC5CCN(C6=CC=C(C(=O)C7=C(C8=CC=C(B(O)O)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C45H46BN5O7S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-RGS5TX	SCHEMBL26625254	[4-[3-[4-[4-[2-[1-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]ethyl]piperazin-1-yl]phenoxy]-6-hydroxy-1-benzothiophen-2-yl]phenyl]boronic acid	O=C1CCC(N2C(=O)C3=CC=C(N4CCC(CCN5CCN(C6=CC=C(OC7=C(C8=CC=C(B(O)O)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C44H44BN5O8S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-VAVAPP	SCHEMBL26625307	[4-[3-[4-[4-[2-[1-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]ethyl]piperazin-1-yl]benzoyl]-6-hydroxy-1-benzothiophen-2-yl]phenyl]boronic acid; SCHEMBL30619703	O=C1CCC(N2C(=O)C3=CC=C(N4CCC(CCN5CCN(C6=CC=C(C(=O)C7=C(C8=CC=C(B(O)O)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C45H44BN5O8S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-35O6IF	SCHEMBL30619750	[4-[3-[4-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]ethyl]piperazin-1-yl]phenoxy]-6-hydroxy-1-benzothiophen-2-yl]phenyl]boronic acid	O=C1CCC(N2CC3=CC(N4CCC(CCN5CCN(C6=CC=C(OC7=C(C8=CC=C(B(O)O)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C44H46BN5O7S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-3FMIN7	SCHEMBL26625082	[4-[3-[4-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]ethyl]piperazin-1-yl]benzoyl]-6-hydroxy-1-benzothiophen-2-yl]phenyl]boronic acid; SCHEMBL30619738	O=C1CCC(N2CC3=CC(N4CCC(CCN5CCN(C6=CC=C(C(=O)C7=C(C8=CC=C(B(O)O)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C45H46BN5O7S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-1HEXBC	SCHEMBL26625317	[4-[3-[4-[4-[2-[1-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]ethyl]piperidin-1-yl]phenoxy]-6-hydroxy-1-benzothiophen-2-yl]phenyl]boronic acid	O=C1CCC(N2C(=O)C3=CC=C(N4CCC(CCC5CCN(C6=CC=C(OC7=C(C8=CC=C(B(O)O)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C45H45BN4O8S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-XPCX6P	SCHEMBL26625218	[4-[3-[4-[4-[2-[1-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]ethyl]piperidin-1-yl]benzoyl]-6-hydroxy-1-benzothiophen-2-yl]phenyl]boronic acid	O=C1CCC(N2C(=O)C3=CC=C(N4CCC(CCC5CCN(C6=CC=C(C(=O)C7=C(C8=CC=C(B(O)O)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C46H45BN4O8S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-DPBY0U	SCHEMBL26625148	[4-[3-[4-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]ethyl]piperidin-1-yl]phenoxy]-6-hydroxy-1-benzothiophen-2-yl]phenyl]boronic acid	O=C1CCC(N2CC3=CC(N4CCC(CCC5CCN(C6=CC=C(OC7=C(C8=CC=C(B(O)O)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C45H47BN4O7S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-LKGR0A	SCHEMBL26625234	[4-[3-[4-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]ethyl]piperidin-1-yl]benzoyl]-6-hydroxy-1-benzothiophen-2-yl]phenyl]boronic acid; SCHEMBL30619764	O=C1CCC(N2CC3=CC(N4CCC(CCC5CCN(C6=CC=C(C(=O)C7=C(C8=CC=C(B(O)O)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C46H47BN4O7S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-CTVA4Y	SCHEMBL26625374	[4-[3-[4-[4-[[4-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenoxy]-6-hydroxy-1-benzothiophen-2-yl]phenyl]boronic acid	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CC5CCN(C6=CC=C(OC7=C(C8=CC=C(B(O)O)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C43H42BN5O8S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-JY0YLD	SCHEMBL26625031	[4-[3-[4-[4-[[4-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]benzoyl]-6-hydroxy-1-benzothiophen-2-yl]phenyl]boronic acid; SCHEMBL30619700	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CC5CCN(C6=CC=C(C(=O)C7=C(C8=CC=C(B(O)O)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C44H42BN5O8S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-KHP6HF	SCHEMBL26625308	[4-[3-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenoxy]-6-hydroxy-1-benzothiophen-2-yl]phenyl]boronic acid; SCHEMBL30619744	O=C1CCC(N2CC3=CC(N4CCN(CC5CCN(C6=CC=C(OC7=C(C8=CC=C(B(O)O)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C43H44BN5O7S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-SJJHIG	SCHEMBL26625009	[4-[3-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]benzoyl]-6-hydroxy-1-benzothiophen-2-yl]phenyl]boronic acid; SCHEMBL30619765	O=C1CCC(N2CC3=CC(N4CCN(CC5CCN(C6=CC=C(C(=O)C7=C(C8=CC=C(B(O)O)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C44H44BN5O7S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-21SEZP	SCHEMBL26625109	[4-[3-[4-[4-[[1-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]phenoxy]-6-hydroxy-1-benzothiophen-2-yl]phenyl]boronic acid; SCHEMBL30619803	O=C1CCC(N2C(=O)C3=CC=C(N4CCC(CN5CCN(C6=CC=C(OC7=C(C8=CC=C(B(O)O)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C43H42BN5O8S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-M8R4C4	SCHEMBL26625084	[4-[3-[4-[4-[[1-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]benzoyl]-6-hydroxy-1-benzothiophen-2-yl]phenyl]boronic acid; SCHEMBL30619775	O=C1CCC(N2C(=O)C3=CC=C(N4CCC(CN5CCN(C6=CC=C(C(=O)C7=C(C8=CC=C(B(O)O)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C44H42BN5O8S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-QFZHMZ	SCHEMBL30619722	[4-[3-[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]phenoxy]-6-hydroxy-1-benzothiophen-2-yl]phenyl]boronic acid	O=C1CCC(N2CC3=CC(N4CCC(CN5CCN(C6=CC=C(OC7=C(C8=CC=C(B(O)O)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C43H44BN5O7S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-AJAD6Q	SCHEMBL26625071	[4-[3-[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]benzoyl]-6-hydroxy-1-benzothiophen-2-yl]phenyl]boronic acid; SCHEMBL30619793	O=C1CCC(N2CC3=CC(N4CCC(CN5CCN(C6=CC=C(C(=O)C7=C(C8=CC=C(B(O)O)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C44H44BN5O7S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-3QWGH3	SCHEMBL26625272	[4-[3-[4-[[1-[3-[4-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]propyl]piperidin-4-yl]methoxy]phenoxy]-6-hydroxy-1-benzothiophen-2-yl]phenyl]boronic acid	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCCN5CCC(COC6=CC=C(OC7=C(C8=CC=C(B(O)O)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C46H48BN5O9S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-N287GP	SCHEMBL26624992	[4-[3-[4-[[1-[3-[4-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]propyl]piperidin-4-yl]methoxy]benzoyl]-6-hydroxy-1-benzothiophen-2-yl]phenyl]boronic acid	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCCN5CCC(COC6=CC=C(C(=O)C7=C(C8=CC=C(B(O)O)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C47H48BN5O9S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-JS80D8	SCHEMBL26625281	[4-[3-[4-[[1-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]propyl]piperidin-4-yl]methoxy]phenoxy]-6-hydroxy-1-benzothiophen-2-yl]phenyl]boronic acid	O=C1CCC(N2CC3=CC(N4CCN(CCCN5CCC(COC6=CC=C(OC7=C(C8=CC=C(B(O)O)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C46H50BN5O8S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-YGHJJ1	SCHEMBL26625142	[4-[3-[4-[[1-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]propyl]piperidin-4-yl]methoxy]benzoyl]-6-hydroxy-1-benzothiophen-2-yl]phenyl]boronic acid	O=C1CCC(N2CC3=CC(N4CCN(CCCN5CCC(COC6=CC=C(C(=O)C7=C(C8=CC=C(B(O)O)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C47H50BN5O8S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-90KTS8	SCHEMBL26625138	2-(2,6-Dioxopiperidin-3-yl)-5-[4-[3-[4-[[4-[[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]methyl]piperidin-1-yl]propyl]piperazin-1-yl]isoindole-1,3-dione; SCHEMBL30619756; SCHEMBL30619757	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCCN5CCC(COC6=CC=C(OC7=C(C8=CC=C(F)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C46H46FN5O7S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-JX8HBR	SCHEMBL26625293	2-(2,6-Dioxopiperidin-3-yl)-5-[4-[3-[4-[[4-[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophene-3-carbonyl]phenoxy]methyl]piperidin-1-yl]propyl]piperazin-1-yl]isoindole-1,3-dione; SCHEMBL30619698	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCCN5CCC(COC6=CC=C(C(=O)C7=C(C8=CC=C(F)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C47H46FN5O7S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-SRRADW	SCHEMBL26625348	3-[6-[4-[3-[4-[[4-[[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]methyl]piperidin-1-yl]propyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30619804	O=C1CCC(N2CC3=CC(N4CCN(CCCN5CCC(COC6=CC=C(OC7=C(C8=CC=C(F)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C46H48FN5O6S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-MPS2JC	SCHEMBL26625265	3-[6-[4-[3-[4-[[4-[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophene-3-carbonyl]phenoxy]methyl]piperidin-1-yl]propyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30619770	O=C1CCC(N2CC3=CC(N4CCN(CCCN5CCC(COC6=CC=C(C(=O)C7=C(C8=CC=C(F)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C47H48FN5O6S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-2NTY54	SCHEMBL26625215	2-(2,6-Dioxopiperidin-3-yl)-5-[4-[3-[4-[[4-[[6-hydroxy-2-(4-hydroxyphenyl)-1-benzothiophen-3-yl]oxy]phenoxy]methyl]piperidin-1-yl]propyl]piperazin-1-yl]isoindole-1,3-dione; SCHEMBL30619748	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCCN5CCC(COC6=CC=C(OC7=C(C8=CC=C(O)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C46H47N5O8S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-JH725M	SCHEMBL26625364	2-(2,6-Dioxopiperidin-3-yl)-5-[4-[3-[4-[[4-[6-hydroxy-2-(4-hydroxyphenyl)-1-benzothiophene-3-carbonyl]phenoxy]methyl]piperidin-1-yl]propyl]piperazin-1-yl]isoindole-1,3-dione; SCHEMBL30619751	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCCN5CCC(COC6=CC=C(C(=O)C7=C(C8=CC=C(O)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C47H47N5O8S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-7OF9OP	SCHEMBL26625127	3-[6-[4-[3-[4-[[4-[[6-hydroxy-2-(4-hydroxyphenyl)-1-benzothiophen-3-yl]oxy]phenoxy]methyl]piperidin-1-yl]propyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(N4CCN(CCCN5CCC(COC6=CC=C(OC7=C(C8=CC=C(O)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C46H49N5O7S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-R5DVI8	SCHEMBL26625092	3-[6-[4-[3-[4-[[4-[6-hydroxy-2-(4-hydroxyphenyl)-1-benzothiophene-3-carbonyl]phenoxy]methyl]piperidin-1-yl]propyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(N4CCN(CCCN5CCC(COC6=CC=C(C(=O)C7=C(C8=CC=C(O)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C47H49N5O7S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-P60614	SCHEMBL26625314	[4-[3-[4-[2-[4-[3-[4-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]propyl]piperazin-1-yl]ethoxy]phenoxy]-6-hydroxy-1-benzothiophen-2-yl]phenyl]boronic acid	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCCN5CCN(CCOC6=CC=C(OC7=C(C8=CC=C(B(O)O)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C46H49BN6O9S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-KLOMH0	SCHEMBL26625105	[4-[3-[4-[2-[4-[3-[4-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]propyl]piperazin-1-yl]ethoxy]benzoyl]-6-hydroxy-1-benzothiophen-2-yl]phenyl]boronic acid	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCCN5CCN(CCOC6=CC=C(C(=O)C7=C(C8=CC=C(B(O)O)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C47H49BN6O9S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-9RKUBO	SCHEMBL30619754	[4-[3-[4-[2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]propyl]piperazin-1-yl]ethoxy]phenoxy]-6-hydroxy-1-benzothiophen-2-yl]phenyl]boronic acid	O=C1CCC(N2CC3=CC(N4CCN(CCCN5CCN(CCOC6=CC=C(OC7=C(C8=CC=C(B(O)O)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C46H51BN6O8S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-EWS7G9	SCHEMBL26625263	[4-[3-[4-[2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]propyl]piperazin-1-yl]ethoxy]benzoyl]-6-hydroxy-1-benzothiophen-2-yl]phenyl]boronic acid	O=C1CCC(N2CC3=CC(N4CCN(CCCN5CCN(CCOC6=CC=C(C(=O)C7=C(C8=CC=C(B(O)O)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C47H51BN6O8S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-W029IW	SCHEMBL26625026	2-(2,6-Dioxopiperidin-3-yl)-5-[4-[3-[4-[2-[4-[[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperazin-1-yl]propyl]piperazin-1-yl]isoindole-1,3-dione; SCHEMBL30619730	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCCN5CCN(CCOC6=CC=C(OC7=C(C8=CC=C(F)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C46H47FN6O7S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-W7Z7C6	SCHEMBL26625192	2-(2,6-Dioxopiperidin-3-yl)-5-[4-[3-[4-[2-[4-[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophene-3-carbonyl]phenoxy]ethyl]piperazin-1-yl]propyl]piperazin-1-yl]isoindole-1,3-dione; SCHEMBL30619783	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCCN5CCN(CCOC6=CC=C(C(=O)C7=C(C8=CC=C(F)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C47H47FN6O7S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-4WBB1C	SCHEMBL26625017	3-[6-[4-[3-[4-[2-[4-[[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperazin-1-yl]propyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30619782	O=C1CCC(N2CC3=CC(N4CCN(CCCN5CCN(CCOC6=CC=C(OC7=C(C8=CC=C(F)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C46H49FN6O6S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-FAA9U5	SCHEMBL26625086	3-[6-[4-[3-[4-[2-[4-[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophene-3-carbonyl]phenoxy]ethyl]piperazin-1-yl]propyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30619818	O=C1CCC(N2CC3=CC(N4CCN(CCCN5CCN(CCOC6=CC=C(C(=O)C7=C(C8=CC=C(F)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C47H49FN6O6S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-TAHK9I	SCHEMBL26625249	[3-[4-[2-[4-[3-[4-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]propyl]piperazin-1-yl]ethoxy]phenoxy]-2-(4-fluorophenyl)-1-benzothiophen-6-yl]boronic acid	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCCN5CCN(CCOC6=CC=C(OC7=C(C8=CC=C(F)C=C8)SC8=CC(B(O)O)=CC=C87)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C46H48BFN6O8S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-RY9AHV	WO2023212599A9_78	.	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCCN5CCN(CCOC6=CC=C(C(=O)C7=C(C8=CC=C(F)C=C8)SC8=CC(B(O)O)=CC=C87)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C47H48BFN6O8S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-EAMDOK	SCHEMBL26625016	[3-[4-[2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]propyl]piperazin-1-yl]ethoxy]phenoxy]-2-(4-fluorophenyl)-1-benzothiophen-6-yl]boronic acid	O=C1CCC(N2CC3=CC(N4CCN(CCCN5CCN(CCOC6=CC=C(OC7=C(C8=CC=C(F)C=C8)SC8=CC(B(O)O)=CC=C87)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C46H50BFN6O7S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-GW3TOO	SCHEMBL26625207	[3-[4-[2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]propyl]piperazin-1-yl]ethoxy]benzoyl]-2-(4-fluorophenyl)-1-benzothiophen-6-yl]boronic acid	O=C1CCC(N2CC3=CC(N4CCN(CCCN5CCN(CCOC6=CC=C(C(=O)C7=C(C8=CC=C(F)C=C8)SC8=CC(B(O)O)=CC=C87)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C47H50BFN6O7S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-L3Y1PN	SCHEMBL26625241	2-(2,6-Dioxopiperidin-3-yl)-5-[4-[3-[4-[2-[4-[[6-hydroxy-2-(4-hydroxyphenyl)-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperazin-1-yl]propyl]piperazin-1-yl]isoindole-1,3-dione; SCHEMBL30619718	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCCN5CCN(CCOC6=CC=C(OC7=C(C8=CC=C(O)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C46H48N6O8S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-W69OW2	SCHEMBL26625376	2-(2,6-Dioxopiperidin-3-yl)-5-[4-[3-[4-[2-[4-[6-hydroxy-2-(4-hydroxyphenyl)-1-benzothiophene-3-carbonyl]phenoxy]ethyl]piperazin-1-yl]propyl]piperazin-1-yl]isoindole-1,3-dione; SCHEMBL30619735	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCCN5CCN(CCOC6=CC=C(C(=O)C7=C(C8=CC=C(O)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C47H48N6O8S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-R83M7Z	SCHEMBL26625146	3-[6-[4-[3-[4-[2-[4-[[6-hydroxy-2-(4-hydroxyphenyl)-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperazin-1-yl]propyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(N4CCN(CCCN5CCN(CCOC6=CC=C(OC7=C(C8=CC=C(O)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C46H50N6O7S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-4O7V7C	SCHEMBL26625415	3-[6-[4-[3-[4-[2-[4-[6-hydroxy-2-(4-hydroxyphenyl)-1-benzothiophene-3-carbonyl]phenoxy]ethyl]piperazin-1-yl]propyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(N4CCN(CCCN5CCN(CCOC6=CC=C(C(=O)C7=C(C8=CC=C(O)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C47H50N6O7S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-P460S3	SCHEMBL26625175	2-(2,6-Dioxopiperidin-3-yl)-5-[4-[3-[4-[4-[[6-hydroxy-2-(4-hydroxyphenyl)-1-benzothiophen-3-yl]oxy]phenyl]piperazin-1-yl]propyl]piperazin-1-yl]isoindole-1,3-dione; SCHEMBL30619713	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCCN5CCN(C6=CC=C(OC7=C(C8=CC=C(O)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C44H44N6O7S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-6JOFN1	SCHEMBL26625287	2-(2,6-Dioxopiperidin-3-yl)-5-[4-[3-[4-[4-[6-hydroxy-2-(4-hydroxyphenyl)-1-benzothiophene-3-carbonyl]phenyl]piperazin-1-yl]propyl]piperazin-1-yl]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCCN5CCN(C6=CC=C(C(=O)C7=C(C8=CC=C(O)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C45H44N6O7S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-DNJMG7	SCHEMBL26625332	3-[6-[4-[3-[4-[4-[[6-hydroxy-2-(4-hydroxyphenyl)-1-benzothiophen-3-yl]oxy]phenyl]piperazin-1-yl]propyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(N4CCN(CCCN5CCN(C6=CC=C(OC7=C(C8=CC=C(O)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C44H46N6O6S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-DEZZV3	SCHEMBL26625106	3-[6-[4-[3-[4-[4-[6-hydroxy-2-(4-hydroxyphenyl)-1-benzothiophene-3-carbonyl]phenyl]piperazin-1-yl]propyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(N4CCN(CCCN5CCN(C6=CC=C(C(=O)C7=C(C8=CC=C(O)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C45H46N6O6S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-52077I	SCHEMBL26625168	[3-[4-[[1-[3-[4-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]propyl]piperidin-4-yl]methoxy]phenoxy]-2-(4-fluorophenyl)-1-benzothiophen-6-yl]boronic acid	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCCN5CCC(COC6=CC=C(OC7=C(C8=CC=C(F)C=C8)SC8=CC(B(O)O)=CC=C87)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C46H47BFN5O8S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-HZS998	WO2023212599A9_98	.	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(CCCN5CCC(COC6=CC=C(C(=O)C7=C(C8=CC=C(F)C=C8)SC8=CC(B(O)O)=CC=C87)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C47H47BFN5O8S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-NHOVUS	SCHEMBL26625202	[3-[4-[[1-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]propyl]piperidin-4-yl]methoxy]phenoxy]-2-(4-fluorophenyl)-1-benzothiophen-6-yl]boronic acid	O=C1CCC(N2CC3=CC(N4CCN(CCCN5CCC(COC6=CC=C(OC7=C(C8=CC=C(F)C=C8)SC8=CC(B(O)O)=CC=C87)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C46H49BFN5O7S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-PKXGZZ	SCHEMBL26625325	[3-[4-[[1-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]propyl]piperidin-4-yl]methoxy]benzoyl]-2-(4-fluorophenyl)-1-benzothiophen-6-yl]boronic acid; SCHEMBL30619733	O=C1CCC(N2CC3=CC(N4CCN(CCCN5CCC(COC6=CC=C(C(=O)C7=C(C8=CC=C(F)C=C8)SC8=CC(B(O)O)=CC=C87)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C47H49BFN5O7S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-861RU6	SCHEMBL26625126	2-(2,6-Dioxopiperidin-3-yl)-5-[1-[3-[4-[4-[6-hydroxy-2-(4-hydroxyphenyl)-1-benzothiophene-3-carbonyl]phenyl]piperazin-1-yl]propyl]piperidin-4-yl]isoindole-1,3-dione; SCHEMBL30619824	O=C1CCC(N2C(=O)C3=CC=C(C4CCN(CCCN5CCN(C6=CC=C(C(=O)C7=C(C8=CC=C(O)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C46H45N5O7S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-NPZX65	WO2023212599A9_106	.	O=C1CCC(N2CC3=CC(C4CCN(CCCN5CCN(C6=CC=C(C(=O)C7=C(C8=CC=C(O)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C46H47N5O6S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-J955FL	SCHEMBL26625183	2-(2,6-Dioxopiperidin-3-yl)-5-[1-[3-[4-[4-[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophene-3-carbonyl]phenyl]piperazin-1-yl]propyl]piperidin-4-yl]isoindole-1,3-dione; SCHEMBL30619702	O=C1CCC(N2C(=O)C3=CC=C(C4CCN(CCCN5CCN(C6=CC=C(C(=O)C7=C(C8=CC=C(F)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C46H44FN5O6S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-O4D708	SCHEMBL26625023	3-[6-[1-[3-[4-[4-[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophene-3-carbonyl]phenyl]piperazin-1-yl]propyl]piperidin-4-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30619816	O=C1CCC(N2CC3=CC(C4CCN(CCCN5CCN(C6=CC=C(C(=O)C7=C(C8=CC=C(F)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C46H46FN5O5S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-FNUAYP	WO2023212599A9_109	.	O=C1CCC(N2C(=O)C3=CC=C(C4CCN(CCCN5CCN(C6=CC=C(C(=O)C7=C(C8=CC=C(B(O)O)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C46H46BN5O8S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-24I4GO	SCHEMBL26625224	[4-[3-[4-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]propyl]piperazin-1-yl]benzoyl]-6-hydroxy-1-benzothiophen-2-yl]phenyl]boronic acid	O=C1CCC(N2CC3=CC(C4CCN(CCCN5CCN(C6=CC=C(C(=O)C7=C(C8=CC=C(B(O)O)C=C8)SC8=C7C=CC(O)=C8)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C46H48BN5O7S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-TNQXA5	SCHEMBL26625200	[3-[4-[4-[3-[4-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-1-yl]propyl]piperazin-1-yl]benzoyl]-2-(4-fluorophenyl)-1-benzothiophen-6-yl]boronic acid	O=C1CCC(N2C(=O)C3=CC=C(C4CCN(CCCN5CCN(C6=CC=C(C(=O)C7=C(C8=CC=C(F)C=C8)SC8=C7C=CC(B(O)O)=C8)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C46H45BFN5O7S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-S7GN95	SCHEMBL30619720	[3-[4-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]propyl]piperazin-1-yl]benzoyl]-2-(4-fluorophenyl)-1-benzothiophen-6-yl]boronic acid	O=C1CCC(N2CC3=CC(C4CCN(CCCN5CCN(C6=CC=C(C(=O)C7=C(C8=CC=C(F)C=C8)SC8=C7C=CC(B(O)O)=C8)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C46H47BFN5O6S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-FLB22X	SCHEMBL26625185	2-(2,6-Dioxopiperidin-3-yl)-5-[1-[3-[4-[2-[4-[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophene-3-carbonyl]phenoxy]ethyl]piperazin-1-yl]propyl]piperidin-4-yl]isoindole-1,3-dione; SCHEMBL30619810	O=C1CCC(N2C(=O)C3=CC=C(C4CCN(CCCN5CCN(CCOC6=CC=C(C(=O)C7=C(C8=CC=C(F)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C48H48FN5O7S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-EKBK5K	SCHEMBL26625166	2-(2,6-Dioxopiperidin-3-yl)-5-[1-[3-[4-[2-[4-[[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperazin-1-yl]propyl]piperidin-4-yl]isoindole-1,3-dione; SCHEMBL30619724	O=C1CCC(N2C(=O)C3=CC=C(C4CCN(CCCN5CCN(CCOC6=CC=C(OC7=C(C8=CC=C(F)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C47H48FN5O7S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-MJRBPW	SCHEMBL26625020	3-[6-[1-[3-[4-[2-[4-[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophene-3-carbonyl]phenoxy]ethyl]piperazin-1-yl]propyl]piperidin-4-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30619784	O=C1CCC(N2CC3=CC(C4CCN(CCCN5CCN(CCOC6=CC=C(C(=O)C7=C(C8=CC=C(F)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C48H50FN5O6S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-C08ZN9	SCHEMBL26625300	3-[6-[1-[3-[4-[2-[4-[[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperazin-1-yl]propyl]piperidin-4-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30619836	O=C1CCC(N2CC3=CC(C4CCN(CCCN5CCN(CCOC6=CC=C(OC7=C(C8=CC=C(F)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C47H50FN5O6S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-SX1T3F	SCHEMBL26625172	[4-[3-[4-[2-[4-[3-[4-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-1-yl]propyl]piperazin-1-yl]ethoxy]benzoyl]-6-hydroxy-1-benzothiophen-2-yl]phenyl]boronic acid	O=C1CCC(N2C(=O)C3=CC=C(C4CCN(CCCN5CCN(CCOC6=CC=C(C(=O)C7=C(C8=CC=C(B(O)O)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C48H50BN5O9S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-4AZBKK	SCHEMBL26625299	[4-[3-[4-[2-[4-[3-[4-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-1-yl]propyl]piperazin-1-yl]ethoxy]phenoxy]-6-hydroxy-1-benzothiophen-2-yl]phenyl]boronic acid	O=C1CCC(N2C(=O)C3=CC=C(C4CCN(CCCN5CCN(CCOC6=CC=C(OC7=C(C8=CC=C(B(O)O)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C47H50BN5O9S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-PJN4PL	SCHEMBL26625187	[4-[3-[4-[2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]propyl]piperazin-1-yl]ethoxy]benzoyl]-6-hydroxy-1-benzothiophen-2-yl]phenyl]boronic acid	O=C1CCC(N2CC3=CC(C4CCN(CCCN5CCN(CCOC6=CC=C(C(=O)C7=C(C8=CC=C(B(O)O)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C48H52BN5O8S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-EIE1DJ	SCHEMBL26625225	[4-[3-[4-[2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]propyl]piperazin-1-yl]ethoxy]phenoxy]-6-hydroxy-1-benzothiophen-2-yl]phenyl]boronic acid	O=C1CCC(N2CC3=CC(C4CCN(CCCN5CCN(CCOC6=CC=C(OC7=C(C8=CC=C(B(O)O)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C47H52BN5O8S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-B70RJL	SCHEMBL26625171	[3-[4-[2-[4-[3-[4-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-1-yl]propyl]piperazin-1-yl]ethoxy]benzoyl]-2-(4-fluorophenyl)-1-benzothiophen-6-yl]boronic acid	O=C1CCC(N2C(=O)C3=CC=C(C4CCN(CCCN5CCN(CCOC6=CC=C(C(=O)C7=C(C8=CC=C(F)C=C8)SC8=CC(B(O)O)=CC=C87)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C48H49BFN5O8S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-LY0XN2	SCHEMBL26625248	[3-[4-[2-[4-[3-[4-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-1-yl]propyl]piperazin-1-yl]ethoxy]phenoxy]-2-(4-fluorophenyl)-1-benzothiophen-6-yl]boronic acid	O=C1CCC(N2C(=O)C3=CC=C(C4CCN(CCCN5CCN(CCOC6=CC=C(OC7=C(C8=CC=C(F)C=C8)SC8=CC(B(O)O)=CC=C87)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C47H49BFN5O8S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-TDS0UY	SCHEMBL26625213	[3-[4-[2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]propyl]piperazin-1-yl]ethoxy]benzoyl]-2-(4-fluorophenyl)-1-benzothiophen-6-yl]boronic acid	O=C1CCC(N2CC3=CC(C4CCN(CCCN5CCN(CCOC6=CC=C(C(=O)C7=C(C8=CC=C(F)C=C8)SC8=CC(B(O)O)=CC=C87)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C48H51BFN5O7S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-KE2ELD	WO2023212599A9_124	.	O=C1CCC(N2CC3=CC(C4CCN(CCCN5CCN(CCOC6=CC=C(OC7=C(C8=CC=C(F)C=C8)SC8=CC(B(O)O)=CC=C87)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C47H51BFN5O7S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-D0H2AF	SCHEMBL26625235	2-(2,6-Dioxopiperidin-3-yl)-5-[1-[3-[4-[2-[4-[6-hydroxy-2-(4-hydroxyphenyl)-1-benzothiophene-3-carbonyl]phenoxy]ethyl]piperazin-1-yl]propyl]piperidin-4-yl]isoindole-1,3-dione; SCHEMBL30619778	O=C1CCC(N2C(=O)C3=CC=C(C4CCN(CCCN5CCN(CCOC6=CC=C(C(=O)C7=C(C8=CC=C(O)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C48H49N5O8S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-VXAWFA	SCHEMBL26625032	2-(2,6-Dioxopiperidin-3-yl)-5-[1-[3-[4-[2-[4-[[6-hydroxy-2-(4-hydroxyphenyl)-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperazin-1-yl]propyl]piperidin-4-yl]isoindole-1,3-dione; SCHEMBL30619797	O=C1CCC(N2C(=O)C3=CC=C(C4CCN(CCCN5CCN(CCOC6=CC=C(OC7=C(C8=CC=C(O)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C47H49N5O8S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-8DBZ3B	SCHEMBL26625015	3-[6-[1-[3-[4-[2-[4-[6-hydroxy-2-(4-hydroxyphenyl)-1-benzothiophene-3-carbonyl]phenoxy]ethyl]piperazin-1-yl]propyl]piperidin-4-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(C4CCN(CCCN5CCN(CCOC6=CC=C(C(=O)C7=C(C8=CC=C(O)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C48H51N5O7S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-RFQXW5	SCHEMBL26625313	3-[6-[1-[3-[4-[2-[4-[[6-hydroxy-2-(4-hydroxyphenyl)-1-benzothiophen-3-yl]oxy]phenoxy]ethyl]piperazin-1-yl]propyl]piperidin-4-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(C4CCN(CCCN5CCN(CCOC6=CC=C(OC7=C(C8=CC=C(O)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C47H51N5O7S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-67NSE1	SCHEMBL26625240	2-(2,6-Dioxopiperidin-3-yl)-5-[1-[2-[4-[[4-[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophene-3-carbonyl]phenoxy]methyl]piperidin-1-yl]ethyl]piperidin-4-yl]isoindole-1,3-dione; SCHEMBL30619727	O=C1CCC(N2C(=O)C3=CC=C(C4CCN(CCN5CCC(COC6=CC=C(C(=O)C7=C(C8=CC=C(F)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C47H45FN4O7S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-4BT8BD	SCHEMBL26625246	2-(2,6-Dioxopiperidin-3-yl)-5-[1-[2-[4-[[4-[[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]methyl]piperidin-1-yl]ethyl]piperidin-4-yl]isoindole-1,3-dione; SCHEMBL30619780	O=C1CCC(N2C(=O)C3=CC=C(C4CCN(CCN5CCC(COC6=CC=C(OC7=C(C8=CC=C(F)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C46H45FN4O7S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-ZNTKIP	SCHEMBL30619746	3-[6-[1-[2-[4-[[4-[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophene-3-carbonyl]phenoxy]methyl]piperidin-1-yl]ethyl]piperidin-4-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(C4CCN(CCN5CCC(COC6=CC=C(C(=O)C7=C(C8=CC=C(F)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C47H47FN4O6S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-G2DRBK	SCHEMBL26624994	3-[6-[1-[2-[4-[[4-[[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]methyl]piperidin-1-yl]ethyl]piperidin-4-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30619699	O=C1CCC(N2CC3=CC(C4CCN(CCN5CCC(COC6=CC=C(OC7=C(C8=CC=C(F)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C46H47FN4O6S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-C095TX	WO2023212599A9_133	.	O=C1CCC(N2C(=O)C3=CC=C(C4CCN(CCN5CCC(COC6=CC=C(C(=O)C7=C(C8=CC=C(B(O)O)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C47H47BN4O9S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-FPEBFF	SCHEMBL26625072	[4-[3-[4-[[1-[2-[4-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-1-yl]ethyl]piperidin-4-yl]methoxy]phenoxy]-6-hydroxy-1-benzothiophen-2-yl]phenyl]boronic acid	O=C1CCC(N2C(=O)C3=CC=C(C4CCN(CCN5CCC(COC6=CC=C(OC7=C(C8=CC=C(B(O)O)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C46H47BN4O9S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-MCUL71	SCHEMBL26625095	[4-[3-[4-[[1-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]ethyl]piperidin-4-yl]methoxy]benzoyl]-6-hydroxy-1-benzothiophen-2-yl]phenyl]boronic acid	O=C1CCC(N2CC3=CC(C4CCN(CCN5CCC(COC6=CC=C(C(=O)C7=C(C8=CC=C(B(O)O)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C47H49BN4O8S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-TD54R5	SCHEMBL26625144	[4-[3-[4-[[1-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]ethyl]piperidin-4-yl]methoxy]phenoxy]-6-hydroxy-1-benzothiophen-2-yl]phenyl]boronic acid	O=C1CCC(N2CC3=CC(C4CCN(CCN5CCC(COC6=CC=C(OC7=C(C8=CC=C(B(O)O)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C46H49BN4O8S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-IT1JD0	SCHEMBL26625040	[3-[4-[[1-[2-[4-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-1-yl]ethyl]piperidin-4-yl]methoxy]benzoyl]-2-(4-fluorophenyl)-1-benzothiophen-6-yl]boronic acid	O=C1CCC(N2C(=O)C3=CC=C(C4CCN(CCN5CCC(COC6=CC=C(C(=O)C7=C(C8=CC=C(F)C=C8)SC8=CC(B(O)O)=CC=C87)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C47H46BFN4O8S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-GX7RLX	SCHEMBL26625274	[3-[4-[[1-[2-[4-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-1-yl]ethyl]piperidin-4-yl]methoxy]phenoxy]-2-(4-fluorophenyl)-1-benzothiophen-6-yl]boronic acid	O=C1CCC(N2C(=O)C3=CC=C(C4CCN(CCN5CCC(COC6=CC=C(OC7=C(C8=CC=C(F)C=C8)SC8=CC(B(O)O)=CC=C87)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C46H46BFN4O8S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-IEC8SD	SCHEMBL26625316	[3-[4-[[1-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]ethyl]piperidin-4-yl]methoxy]benzoyl]-2-(4-fluorophenyl)-1-benzothiophen-6-yl]boronic acid	O=C1CCC(N2CC3=CC(C4CCN(CCN5CCC(COC6=CC=C(C(=O)C7=C(C8=CC=C(F)C=C8)SC8=CC(B(O)O)=CC=C87)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C47H48BFN4O7S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-6AFRR4	SCHEMBL26625285	[3-[4-[[1-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]ethyl]piperidin-4-yl]methoxy]phenoxy]-2-(4-fluorophenyl)-1-benzothiophen-6-yl]boronic acid	O=C1CCC(N2CC3=CC(C4CCN(CCN5CCC(COC6=CC=C(OC7=C(C8=CC=C(F)C=C8)SC8=CC(B(O)O)=CC=C87)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C46H48BFN4O7S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-30VVED	SCHEMBL26625297	2-(2,6-Dioxopiperidin-3-yl)-5-[1-[2-[4-[[4-[6-hydroxy-2-(4-hydroxyphenyl)-1-benzothiophene-3-carbonyl]phenoxy]methyl]piperidin-1-yl]ethyl]piperidin-4-yl]isoindole-1,3-dione; SCHEMBL30619801	O=C1CCC(N2C(=O)C3=CC=C(C4CCN(CCN5CCC(COC6=CC=C(C(=O)C7=C(C8=CC=C(O)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C47H46N4O8S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-IU2J6E	SCHEMBL26625336	2-(2,6-Dioxopiperidin-3-yl)-5-[1-[2-[4-[[4-[[6-hydroxy-2-(4-hydroxyphenyl)-1-benzothiophen-3-yl]oxy]phenoxy]methyl]piperidin-1-yl]ethyl]piperidin-4-yl]isoindole-1,3-dione; SCHEMBL30619800	O=C1CCC(N2C(=O)C3=CC=C(C4CCN(CCN5CCC(COC6=CC=C(OC7=C(C8=CC=C(O)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C46H46N4O8S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-Y3FFKE	SCHEMBL26625061	3-[6-[1-[2-[4-[[4-[6-hydroxy-2-(4-hydroxyphenyl)-1-benzothiophene-3-carbonyl]phenoxy]methyl]piperidin-1-yl]ethyl]piperidin-4-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(C4CCN(CCN5CCC(COC6=CC=C(C(=O)C7=C(C8=CC=C(O)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C47H48N4O7S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-2CIYEK	SCHEMBL26625190	3-[6-[1-[2-[4-[[4-[[6-hydroxy-2-(4-hydroxyphenyl)-1-benzothiophen-3-yl]oxy]phenoxy]methyl]piperidin-1-yl]ethyl]piperidin-4-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(C4CCN(CCN5CCC(COC6=CC=C(OC7=C(C8=CC=C(O)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C46H48N4O7S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-4AK0M8	SCHEMBL26625098	2-(2,6-Dioxopiperidin-3-yl)-5-[1-[3-[4-[[4-[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophene-3-carbonyl]phenoxy]methyl]piperidin-1-yl]propyl]piperidin-4-yl]isoindole-1,3-dione; SCHEMBL30619812	O=C1CCC(N2C(=O)C3=CC=C(C4CCN(CCCN5CCC(COC6=CC=C(C(=O)C7=C(C8=CC=C(F)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C48H47FN4O7S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-3Q1P9N	SCHEMBL26625132	2-(2,6-Dioxopiperidin-3-yl)-5-[1-[3-[4-[[4-[[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]methyl]piperidin-1-yl]propyl]piperidin-4-yl]isoindole-1,3-dione; SCHEMBL30619708	O=C1CCC(N2C(=O)C3=CC=C(C4CCN(CCCN5CCC(COC6=CC=C(OC7=C(C8=CC=C(F)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C47H47FN4O7S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-J147ED	WO2023212599A9_147	.	O=C1CCC(N2CC3=CC(C4CCN(CCCN5CCC(COC6=CC=C(C(=O)C7=C(C8=CC=C(F)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C48H49FN4O6S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-HR6M5N	SCHEMBL26625104	3-[6-[1-[3-[4-[[4-[[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]phenoxy]methyl]piperidin-1-yl]propyl]piperidin-4-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30619726	O=C1CCC(N2CC3=CC(C4CCN(CCCN5CCC(COC6=CC=C(OC7=C(C8=CC=C(F)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C47H49FN4O6S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-6LVE1J	SCHEMBL26625121	[4-[3-[4-[[1-[3-[4-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-1-yl]propyl]piperidin-4-yl]methoxy]benzoyl]-6-hydroxy-1-benzothiophen-2-yl]phenyl]boronic acid	O=C1CCC(N2C(=O)C3=CC=C(C4CCN(CCCN5CCC(COC6=CC=C(C(=O)C7=C(C8=CC=C(B(O)O)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C48H49BN4O9S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-6NT5HP	SCHEMBL26625369	[4-[3-[4-[[1-[3-[4-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-1-yl]propyl]piperidin-4-yl]methoxy]phenoxy]-6-hydroxy-1-benzothiophen-2-yl]phenyl]boronic acid	O=C1CCC(N2C(=O)C3=CC=C(C4CCN(CCCN5CCC(COC6=CC=C(OC7=C(C8=CC=C(B(O)O)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C47H49BN4O9S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-N6FL6L	SCHEMBL26625309	[4-[3-[4-[[1-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]propyl]piperidin-4-yl]methoxy]benzoyl]-6-hydroxy-1-benzothiophen-2-yl]phenyl]boronic acid	O=C1CCC(N2CC3=CC(C4CCN(CCCN5CCC(COC6=CC=C(C(=O)C7=C(C8=CC=C(B(O)O)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C48H51BN4O8S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-QF5QEG	SCHEMBL26625216	[4-[3-[4-[[1-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]propyl]piperidin-4-yl]methoxy]phenoxy]-6-hydroxy-1-benzothiophen-2-yl]phenyl]boronic acid	O=C1CCC(N2CC3=CC(C4CCN(CCCN5CCC(COC6=CC=C(OC7=C(C8=CC=C(B(O)O)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C47H51BN4O8S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-4LN5QK	WO2023212599A9_153	.	O=C1CCC(N2C(=O)C3=CC=C(C4CCN(CCCN5CCC(COC6=CC=C(C(=O)C7=C(C8=CC=C(F)C=C8)SC8=CC(B(O)O)=CC=C87)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C48H48BFN4O8S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-OV572U	WO2023212599A9_154	[3-[4-[[1-[3-[4-[2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-1-yl]propyl]piperidin-4-yl]methoxy]phenoxy]-2-(4-fluorophenyl)-1-benzothiophen-6-yl]boronic acid	O=C1CCC(N2C(=O)C3=CC=C(C4CCN(CCCN5CCC(COC6=CC=C(OC7=C(C8=CC=C(F)C=C8)SC8=CC(B(O)O)=CC=C87)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C47H48BFN4O8S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-PWZ7TJ	SCHEMBL26625179	[3-[4-[[1-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]propyl]piperidin-4-yl]methoxy]benzoyl]-2-(4-fluorophenyl)-1-benzothiophen-6-yl]boronic acid	O=C1CCC(N2CC3=CC(C4CCN(CCCN5CCC(COC6=CC=C(C(=O)C7=C(C8=CC=C(F)C=C8)SC8=CC(B(O)O)=CC=C87)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C48H50BFN4O7S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-RSTHXY	SCHEMBL26625227	[3-[4-[[1-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]propyl]piperidin-4-yl]methoxy]phenoxy]-2-(4-fluorophenyl)-1-benzothiophen-6-yl]boronic acid	O=C1CCC(N2CC3=CC(C4CCN(CCCN5CCC(COC6=CC=C(OC7=C(C8=CC=C(F)C=C8)SC8=CC(B(O)O)=CC=C87)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C47H50BFN4O7S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-QSLP0V	SCHEMBL26625372	2-(2,6-Dioxopiperidin-3-yl)-5-[1-[3-[4-[[4-[6-hydroxy-2-(4-hydroxyphenyl)-1-benzothiophene-3-carbonyl]phenoxy]methyl]piperidin-1-yl]propyl]piperidin-4-yl]isoindole-1,3-dione; SCHEMBL30619704	O=C1CCC(N2C(=O)C3=CC=C(C4CCN(CCCN5CCC(COC6=CC=C(C(=O)C7=C(C8=CC=C(O)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C48H48N4O8S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-KJJ6X9	SCHEMBL26625136	2-(2,6-Dioxopiperidin-3-yl)-5-[1-[3-[4-[[4-[[6-hydroxy-2-(4-hydroxyphenyl)-1-benzothiophen-3-yl]oxy]phenoxy]methyl]piperidin-1-yl]propyl]piperidin-4-yl]isoindole-1,3-dione; SCHEMBL30619787	O=C1CCC(N2C(=O)C3=CC=C(C4CCN(CCCN5CCC(COC6=CC=C(OC7=C(C8=CC=C(O)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C47H48N4O8S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-217NZY	SCHEMBL26625394	3-[6-[1-[3-[4-[[4-[6-hydroxy-2-(4-hydroxyphenyl)-1-benzothiophene-3-carbonyl]phenoxy]methyl]piperidin-1-yl]propyl]piperidin-4-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(C4CCN(CCCN5CCC(COC6=CC=C(C(=O)C7=C(C8=CC=C(O)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C48H50N4O7S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-9XSJGR	SCHEMBL26625188	3-[6-[1-[3-[4-[[4-[[6-hydroxy-2-(4-hydroxyphenyl)-1-benzothiophen-3-yl]oxy]phenoxy]methyl]piperidin-1-yl]propyl]piperidin-4-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(C4CCN(CCCN5CCC(COC6=CC=C(OC7=C(C8=CC=C(O)C=C8)SC8=CC(O)=CC=C87)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C47H50N4O7S	ERα	P03372	CRBN	WO-2023212599-A9
TPD-9O6O0M	SCHEMBL26625064	3-[6-[4-[4-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperazine-1-carbonyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(N4CCN(C(=O)N5CCN(C6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C44H46N6O5	ERα	P03372	CRBN	WO-2023212599-A9
TPD-M341KS	SCHEMBL26625231	N-(2,6-dioxopiperidin-3-yl)-4-[4-[4-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperazine-1-carbonyl]piperazin-1-yl]benzamide	O=C1CCC(NC(=O)C2=CC=C(N3CCN(C(=O)N4CCN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)CC3)C=C2)C(=O)N1	C43H46N6O5	ERα	P03372	CRBN	WO-2023212599-A9
TPD-TCDO8I	WO2023212599A9_163	.	O=C1CCN(C2=CC=C(N3CCN(C(=O)N4CCN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)CC3)C=C2)C(=O)N1	C41H44N6O4	ERα	P03372	CRBN	WO-2023212599-A9
TPD-X0W368	SCHEMBL26625152	3-[6-[4-[1-[4-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperazine-1-carbonyl]piperidin-4-yl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(N4CCN(C5CCN(C(=O)N6CCN(C7=CC=C([C@@H]8C9=CC=C(O)C=C9CC[C@@H]8C8=CC=CC=C8)C=C7)CC6)CC5)CC4)=C3)C2=O)C(=O)N1	C49H55N7O5	ERα	P03372	CRBN	WO-2023212599-A9
TPD-XLV24R	SCHEMBL26625243	N-(2,6-dioxopiperidin-3-yl)-4-[4-[1-[4-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperazine-1-carbonyl]piperidin-4-yl]piperazin-1-yl]benzamide; SCHEMBL30619790	O=C1CCC(NC(=O)C2=CC=C(N3CCN(C4CCN(C(=O)N5CCN(C6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)CC3)C=C2)C(=O)N1	C48H55N7O5	ERα	P03372	CRBN	WO-2023212599-A9
TPD-018BAC	SCHEMBL26625067	1-[4-[4-[1-[4-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperazine-1-carbonyl]piperidin-4-yl]piperazin-1-yl]phenyl]-1,3-diazinane-2,4-dione	O=C1CCN(C2=CC=C(N3CCN(C4CCN(C(=O)N5CCN(C6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)CC3)C=C2)C(=O)N1	C46H53N7O4	ERα	P03372	CRBN	WO-2023212599-A9
TPD-FUP8NO	SCHEMBL26625259	3-[6-[4-[[1-[4-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperazine-1-carbonyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(N4CCN(CC5CCN(C(=O)N6CCN(C7=CC=C([C@@H]8C9=CC=C(O)C=C9CC[C@@H]8C8=CC=CC=C8)C=C7)CC6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C50H57N7O5	ERα	P03372	CRBN	WO-2023212599-A9
TPD-4ERTB3	SCHEMBL26625100	N-(2,6-dioxopiperidin-3-yl)-4-[4-[[1-[4-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperazine-1-carbonyl]piperidin-4-yl]methyl]piperazin-1-yl]benzamide; SCHEMBL30619715	O=C1CCC(NC(=O)C2=CC=C(N3CCN(CC4CCN(C(=O)N5CCN(C6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)CC3)C=C2)C(=O)N1	C49H57N7O5	ERα	P03372	CRBN	WO-2023212599-A9
TPD-H2NT3E	SCHEMBL26624957	1-[4-[4-[[1-[4-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperazine-1-carbonyl]piperidin-4-yl]methyl]piperazin-1-yl]phenyl]-1,3-diazinane-2,4-dione	O=C1CCN(C2=CC=C(N3CCN(CC4CCN(C(=O)N5CCN(C6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)CC3)C=C2)C(=O)N1	C47H55N7O4	ERα	P03372	CRBN	WO-2023212599-A9
TPD-BFF8NM	SCHEMBL26625222	3-[6-[4-[4-[[4-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperazin-1-yl]methyl]piperidine-1-carbonyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(N4CCN(C(=O)N5CCC(CN6CCN(C7=CC=C([C@@H]8C9=CC=C(O)C=C9CC[C@@H]8C8=CC=CC=C8)C=C7)CC6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C50H57N7O5	ERα	P03372	CRBN	WO-2023212599-A9
TPD-MU9FVC	SCHEMBL26625147	N-(2,6-dioxopiperidin-3-yl)-4-[4-[4-[[4-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperazin-1-yl]methyl]piperidine-1-carbonyl]piperazin-1-yl]benzamide; SCHEMBL30619749	O=C1CCC(NC(=O)C2=CC=C(N3CCN(C(=O)N4CCC(CN5CCN(C6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)CC3)C=C2)C(=O)N1	C49H57N7O5	ERα	P03372	CRBN	WO-2023212599-A9
TPD-J3KJF1	WO2023212599A9_172	.	O=C1CCN(C2=CC=C(N3CCN(C(=O)N4CCC(CN5CCN(C6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)CC3)C=C2)C(=O)N1	C47H55N7O4	ERα	P03372	CRBN	WO-2023212599-A9
TPD-MQQXZ1	SCHEMBL26625268	4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-N-[2-[4-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperazin-1-yl]ethyl]piperazine-1-carboxamide; SCHEMBL30619808	O=C1CCC(N2CC3=C(C=CC(N4CCN(C(=O)NCCN5CCN(C6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C46H51N7O5	ERα	P03372	CRBN	WO-2023212599-A9
TPD-METUDW	SCHEMBL26625239	4-[4-[(2,6-dioxopiperidin-3-yl)carbamoyl]phenyl]-N-[2-[4-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperazin-1-yl]ethyl]piperazine-1-carboxamide; SCHEMBL30619743	O=C1CCC(NC(=O)C2=CC=C(N3CCN(C(=O)NCCN4CCN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)CC3)C=C2)C(=O)N1	C45H51N7O5	ERα	P03372	CRBN	WO-2023212599-A9
TPD-ZT8ESJ	SCHEMBL26625076	4-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]-N-[2-[4-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperazin-1-yl]ethyl]piperazine-1-carboxamide	O=C1CCN(C2=CC=C(N3CCN(C(=O)NCCN4CCN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)CC3)C=C2)C(=O)N1	C43H49N7O4	ERα	P03372	CRBN	WO-2023212599-A9
TPD-ESREXD	SCHEMBL26625279	3-[6-[4-[4-[2-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]ethyl]piperazine-1-carbonyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(N4CCN(C(=O)N5CCN(CCOC6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C46H50N6O6	ERα	P03372	CRBN	WO-2023212599-A9
TPD-0C2S51	SCHEMBL26625280	N-(2,6-dioxopiperidin-3-yl)-4-[4-[4-[2-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]ethyl]piperazine-1-carbonyl]piperazin-1-yl]benzamide; SCHEMBL30619710	O=C1CCC(NC(=O)C2=CC=C(N3CCN(C(=O)N4CCN(CCOC5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)CC3)C=C2)C(=O)N1	C45H50N6O6	ERα	P03372	CRBN	WO-2023212599-A9
TPD-FI0ZZU	SCHEMBL30619825	1-[4-[4-[4-[2-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]ethyl]piperazine-1-carbonyl]piperazin-1-yl]phenyl]-1,3-diazinane-2,4-dione	O=C1CCN(C2=CC=C(N3CCN(C(=O)N4CCN(CCOC5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)CC3)C=C2)C(=O)N1	C43H48N6O5	ERα	P03372	CRBN	WO-2023212599-A9
TPD-IOFY0J	WO2023212599A9_179	.	O=C1CCC(N2CC3=CC(C4CCN(C(=O)N5CCC(CCOC6=CC=C(C7C8=C(C=C(O)C=C8)CCC7C7=CC=CC=C7)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C48H52N4O6	ERα	P03372	CRBN	WO-2023212599-A9
TPD-1MD5A2	WO2023212599A9_180	.	O=C1CCC(NC(=O)C2=CC=C(C3CCN(C(=O)N4CCC(CCOC5=CC=C(C6C7=C(C=C(O)C=C7)CCC6C6=CC=CC=C6)C=C5)CC4)CC3)C=C2)C(=O)N1	C47H52N4O6	ERα	P03372	CRBN	WO-2023212599-A9
TPD-WNDWST	WO2023212599A9_181	.	O=C1CCN(C2=CC=C(C3CCN(C(=O)N4CCC(CCOC5=CC=C(C6C7=C(C=C(O)C=C7)CCC6C6=CC=CC=C6)C=C5)CC4)CC3)C=C2)C(=O)N1	C45H50N4O5	ERα	P03372	CRBN	WO-2023212599-A9
TPD-CILLGM	WO2023212599A9_182	.	O=C1CCC(N2CC3=CC(N4CCN(C(=O)NCC5CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C46H50N6O5	ERα	P03372	CRBN	WO-2023212599-A9
TPD-LOC8SD	SCHEMBL26625324	4-[4-[(2,6-dioxopiperidin-3-yl)carbamoyl]phenyl]-N-[[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperazine-1-carboxamide; SCHEMBL30619745	O=C1CCC(NC(=O)C2=CC=C(N3CCN(C(=O)NCC4CCN(C5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)CC3)C=C2)C(=O)N1	C45H50N6O5	ERα	P03372	CRBN	WO-2023212599-A9
TPD-LGA0A7	SCHEMBL26625277	4-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]-N-[[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperazine-1-carboxamide	O=C1CCN(C2=CC=C(N3CCN(C(=O)NCC4CCN(C5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)CC3)C=C2)C(=O)N1	C43H48N6O4	ERα	P03372	CRBN	WO-2023212599-A9
TPD-O0Y75F	SCHEMBL26625385	1-[4-[4-[[4-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]-1,3-diazinane-2,4-dione	O=C1CCN(C2=CC=C(N3CCC(CN4CCN(C5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)CC3)C=C2)C(=O)N1	C42H47N5O3	ERα	P03372	CRBN	WO-2023212599-A9
TPD-T5HWIX	WO2023212599A9_186	.	O=C1CCN(NC(=O)C2=CC=C(N3CCC(CN4CCN(C5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)CC3)C=C2)C(=O)N1	C43H48N6O4	ERα	P03372	CRBN	WO-2023212599-A9
TPD-A5O91X	SCHEMBL26625212	3-[6-[4-[4-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperazine-1-carbonyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(N4CCC(C(=O)N5CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C45H47N5O5	ERα	P03372	CRBN	WO-2023212599-A9
TPD-H3F6I9	SCHEMBL26625256	N-(2,6-dioxopiperidin-3-yl)-4-[4-[4-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperazine-1-carbonyl]piperidin-1-yl]benzamide; SCHEMBL30619785	O=C1CCC(NC(=O)C2=CC=C(N3CCC(C(=O)N4CCN(C5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)CC3)C=C2)C(=O)N1	C44H47N5O5	ERα	P03372	CRBN	WO-2023212599-A9
TPD-4G7BTK	SCHEMBL26625125	3-[4-[4-[4-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperazine-1-carbonyl]piperidin-1-yl]anilino]piperidine-2,6-dione; SCHEMBL30619693	O=C1CCC(NC2=CC=C(N3CCC(C(=O)N4CCN(C5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)CC3)C=C2)C(=O)N1	C43H47N5O4	ERα	P03372	CRBN	WO-2023212599-A9
TPD-Z9IAEZ	WO2023212599A9_190	.	O=C1CCN(C2=CC=C(N3CCC(C(=O)N4CCN(C5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)CC3)C=C2)C(=O)N1	C42H45N5O4	ERα	P03372	CRBN	WO-2023212599-A9
TPD-M5USCD	SCHEMBL26625173	1-[4-[4-[2-[4-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperazin-1-yl]-2-oxoethyl]piperidin-1-yl]phenyl]-1,3-diazinane-2,4-dione	O=C1CCN(C2=CC=C(N3CCC(CC(=O)N4CCN(C5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)CC3)C=C2)C(=O)N1	C43H47N5O4	ERα	P03372	CRBN	WO-2023212599-A9
TPD-6ZDXST	SCHEMBL26625010	1-[4-[4-[2-[4-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperazin-1-yl]ethyl]piperazin-1-yl]phenyl]-1,3-diazinane-2,4-dione	O=C1CCN(C2=CC=C(N3CCN(CCN4CCN(C5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)CC3)C=C2)C(=O)N1	C42H48N6O3	ERα	P03372	CRBN	WO-2023212599-A9
TPD-P8LTKS	WO2023212599A9_193	.	O=C1CCC(N2CC3=C(C=CC(N4CCC(N5CCC(C(=O)N6CCN(C7=CC=C([C@@H]8C9=C(C=C(O)C=C9)CC[C@@H]8C8=CC=CC=C8)C=C7)CC6)CC5)CC4)=C3)C2=O)C(=O)N1	C50H56N6O5	ERα	P03372	CRBN	WO-2023212599-A9
TPD-AD5MR0	WO2023212599A9_194	.	O=C1CCC(NC(=O)C2=CC=C(N3CCC(N4CCC(CN5CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)CC3)C=C2)C(=O)N1	C49H58N6O4	ERα	P03372	CRBN	WO-2023212599-A9
TPD-VIW08E	WO2023212599A9_195	.	O=C1CCC(NC2=CC=C(N3CCC(N4CCC(CN5CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)CC3)C=C2)C(=O)N1	C48H58N6O3	ERα	P03372	CRBN	WO-2023212599-A9
TPD-6O1UKH	WO2023212599A9_196	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=C1C=C(N1CCC(N3CCC(CN4CCN(C5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)CC3)CC1)C=C2	C50H59N7O4	ERα	P03372	CRBN	WO-2023212599-A9
TPD-SAJEH4	WO2023212599A9_197	.	O=C1CCC(NC(=O)C2=CC=C(N3CCC(N4CCC(C(=O)N5CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)CC3)C=C2)C(=O)N1	C49H56N6O5	ERα	P03372	CRBN	WO-2023212599-A9
TPD-2U6LD0	SCHEMBL26625043	1-[4-[4-[1-[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidine-4-carbonyl]piperidin-4-yl]piperazin-1-yl]phenyl]-1,3-diazinane-2,4-dione	O=C1CCN(C2=CC=C(N3CCN(C4CCN(C(=O)C5CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)CC3)C=C2)C(=O)N1	C47H54N6O4	ERα	P03372	CRBN	WO-2023212599-A9
TPD-11DHEG	SCHEMBL26625201	3-[6-[4-[[1-[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidine-4-carbonyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC5CCN(C(=O)C6CCN(C7=CC=C([C@@H]8C9=CC=C(O)C=C9CC[C@@H]8C8=CC=CC=C8)C=C7)CC6)CC5)CC4)=C3)C2=O)C(=O)N1	C51H58N6O5	ERα	P03372	CRBN	WO-2023212599-A9
TPD-9H0CMR	SCHEMBL26625195	N-(2,6-dioxopiperidin-3-yl)-4-[4-[[1-[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidine-4-carbonyl]piperidin-4-yl]methyl]piperazin-1-yl]benzamide; SCHEMBL30619734	O=C1CCC(NC(=O)C2=CC=C(N3CCN(CC4CCN(C(=O)C5CCN(C6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)CC3)C=C2)C(=O)N1	C50H58N6O5	ERα	P03372	CRBN	WO-2023212599-A9
TPD-K59VT2	SCHEMBL26625052	N-(2,6-dioxopiperidin-3-yl)-4-[4-[[1-[[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]benzamide; SCHEMBL30619692	O=C1CCC(NC(=O)C2=CC=C(N3CCN(CC4CCN(CC5CCN(C6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)CC3)C=C2)C(=O)N1	C50H60N6O4	ERα	P03372	CRBN	WO-2023212599-A9
TPD-937LRU	SCHEMBL26625070	3-[4-[4-[[1-[[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]anilino]piperidine-2,6-dione	O=C1CCC(NC2=CC=C(N3CCN(CC4CCN(CC5CCN(C6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)CC3)C=C2)C(=O)N1	C49H60N6O3	ERα	P03372	CRBN	WO-2023212599-A9
TPD-PVNUD9	SCHEMBL26625063	1-[4-[4-[[1-[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidine-4-carbonyl]piperidin-4-yl]methyl]piperazin-1-yl]phenyl]-1,3-diazinane-2,4-dione	O=C1CCN(C2=CC=C(N3CCN(CC4CCN(C(=O)C5CCN(C6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)CC3)C=C2)C(=O)N1	C48H56N6O4	ERα	P03372	CRBN	WO-2023212599-A9
TPD-NZYK8E	SCHEMBL26625422	1-[4-[4-[[1-[[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]phenyl]-1,3-diazinane-2,4-dione	O=C1CCN(C2=CC=C(N3CCN(CC4CCN(CC5CCN(C6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)CC3)C=C2)C(=O)N1	C48H58N6O3	ERα	P03372	CRBN	WO-2023212599-A9
TPD-2TDISQ	SCHEMBL26625060	3-[6-[4-[4-[[4-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperazin-1-yl]methyl]piperidine-1-carbonyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(N4CCC(C(=O)N5CCC(CN6CCN(C7=CC=C([C@@H]8C9=CC=C(O)C=C9CC[C@@H]8C8=CC=CC=C8)C=C7)CC6)CC5)CC4)=C3)C2=O)C(=O)N1	C51H58N6O5	ERα	P03372	CRBN	WO-2023212599-A9
TPD-6NYVAE	SCHEMBL26625380	N-(2,6-dioxopiperidin-3-yl)-4-[4-[4-[[4-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperazin-1-yl]methyl]piperidine-1-carbonyl]piperidin-1-yl]benzamide; SCHEMBL30619725	O=C1CCC(NC(=O)C2=CC=C(N3CCC(C(=O)N4CCC(CN5CCN(C6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)CC3)C=C2)C(=O)N1	C50H58N6O5	ERα	P03372	CRBN	WO-2023212599-A9
TPD-39EX3A	SCHEMBL26625399	1-[4-[4-[4-[[4-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperazin-1-yl]methyl]piperidine-1-carbonyl]piperidin-1-yl]phenyl]-1,3-diazinane-2,4-dione	O=C1CCN(C2=CC=C(N3CCC(C(=O)N4CCC(CN5CCN(C6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)CC3)C=C2)C(=O)N1	C48H56N6O4	ERα	P03372	CRBN	WO-2023212599-A9
TPD-6LSDYP	SCHEMBL26625162	1-[4-[4-[[4-[[4-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperazin-1-yl]methyl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-1,3-diazinane-2,4-dione	O=C1CCN(C2=CC=C(N3CCC(CN4CCC(CN5CCN(C6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)CC3)C=C2)C(=O)N1	C48H58N6O3	ERα	P03372	CRBN	WO-2023212599-A9
TPD-WLMEGK	SCHEMBL26625007	1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-N-[2-[4-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperazin-1-yl]ethyl]piperidine-4-carboxamide	O=C1CCC(N2CC3=C(C=CC(N4CCC(C(=O)NCCN5CCN(C6=CC=C([C@@H]7C8=CC=C(O)C=C8CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C47H52N6O5	ERα	P03372	CRBN	WO-2023212599-A9
TPD-342Z3Y	SCHEMBL26625041	N-(2,6-dioxopiperidin-3-yl)-4-[4-[4-[4-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperazin-1-yl]butanoyl]piperazin-1-yl]benzamide; SCHEMBL30619737	O=C1CCC(NC(=O)C2=CC=C(N3CCN(C(=O)CCCN4CCN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)CC3)C=C2)C(=O)N1	C46H52N6O5	ERα	P03372	CRBN	WO-2023212599-A9
TPD-S9D1QZ	SCHEMBL26625305	1-[4-[4-[4-[4-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperazin-1-yl]butanoyl]piperazin-1-yl]phenyl]-1,3-diazinane-2,4-dione	O=C1CCN(C2=CC=C(N3CCN(C(=O)CCCN4CCN(C5=CC=C([C@@H]6C7=CC=C(O)C=C7CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)CC3)C=C2)C(=O)N1	C44H50N6O4	ERα	P03372	CRBN	WO-2023212599-A9
TPD-D8U707	SCHEMBL26624970	3-[6-[4-[1-[2-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]ethyl]piperidine-4-carbonyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(N4CCN(C(=O)C5CCN(CCOC6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C47H51N5O6	ERα	P03372	CRBN	WO-2023212599-A9
TPD-GCWNCS	SCHEMBL26625312	3-[6-[4-[4-[2-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]ethyl]piperazine-1-carbonyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(N4CCC(C(=O)N5CCN(CCOC6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C47H51N5O6	ERα	P03372	CRBN	WO-2023212599-A9
TPD-NPNCT7	SCHEMBL26625592	N-(2,6-dioxopiperidin-3-yl)-4-[4-[1-[2-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]ethyl]piperidine-4-carbonyl]piperazin-1-yl]benzamide; SCHEMBL30619802	O=C1CCC(NC(=O)C2=CC=C(N3CCN(C(=O)C4CCN(CCOC5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)CC3)C=C2)C(=O)N1	C46H51N5O6	ERα	P03372	CRBN	WO-2023212599-A9
TPD-ZP7E6N	SCHEMBL26625223	N-(2,6-dioxopiperidin-3-yl)-4-[4-[[1-[2-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]ethyl]piperidin-4-yl]methyl]piperazin-1-yl]benzamide; SCHEMBL30619807	O=C1CCC(NC(=O)C2=CC=C(N3CCN(CC4CCN(CCOC5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)CC3)C=C2)C(=O)N1	C46H53N5O5	ERα	P03372	CRBN	WO-2023212599-A9
TPD-PO7Q6X	SCHEMBL30619829	1-[4-[4-[1-[2-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]ethyl]piperidine-4-carbonyl]piperazin-1-yl]phenyl]-1,3-diazinane-2,4-dione	O=C1CCN(C2=CC=C(N3CCN(C(=O)C4CCN(CCOC5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)CC3)C=C2)C(=O)N1	C44H49N5O5	ERα	P03372	CRBN	WO-2023212599-A9
TPD-BQTL6I	SCHEMBL26625345	3-[6-[4-[4-[2-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]ethyl]piperidine-1-carbonyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(N4CCC(C(=O)N5CCC(CCOC6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C48H52N4O6	ERα	P03372	CRBN	WO-2023212599-A9
TPD-UAUUX6	SCHEMBL26625286	N-(2,6-dioxopiperidin-3-yl)-4-[4-[4-[2-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]ethyl]piperidine-1-carbonyl]piperidin-1-yl]benzamide; SCHEMBL30619774	O=C1CCC(NC(=O)C2=CC=C(N3CCC(C(=O)N4CCC(CCOC5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)CC3)C=C2)C(=O)N1	C47H52N4O6	ERα	P03372	CRBN	WO-2023212599-A9
TPD-1D3NQX	WO2023212599A9_220	.	O=C1CCN(C2=CC=C(N3CCN(CC4CCN(CCOC5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)CC3)C=C2)C(=O)N1	C44H51N5O4	ERα	P03372	CRBN	WO-2023212599-A9
TPD-NTUS9M	SCHEMBL26625296	3-[4-[4-[[1-[2-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]ethyl]piperidin-4-yl]methyl]piperazin-1-yl]anilino]piperidine-2,6-dione	O=C1CCC(NC2=CC=C(N3CCN(CC4CCN(CCOC5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)CC3)C=C2)C(=O)N1	C45H53N5O4	ERα	P03372	CRBN	WO-2023212599-A9
TPD-WC7NHK	SCHEMBL26625449	3-[5-[4-[[1-[2-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]ethyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(N3CCN(CC4CCN(CCOC5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)CC3)C=C21	C47H54N6O5	ERα	P03372	CRBN	WO-2023212599-A9
TPD-QX03RD	SCHEMBL26625160	3-[6-[4-[3-[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]propanoyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(N4CCN(C(=O)CCC5CCN(C6=CC=C([C@@H]7C8=C(C=C(O)C=C8)CC[C@@H]7C7=CC=CC=C7)C=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C47H51N5O5	ERα	P03372	CRBN	WO-2023212599-A9
TPD-3ULC83	SCHEMBL26625151	1-[4-[4-[3-[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]propanoyl]piperazin-1-yl]phenyl]-1,3-diazinane-2,4-dione	O=C1CCN(C2=CC=C(N3CCN(C(=O)CCC4CCN(C5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)CC3)C=C2)C(=O)N1	C44H49N5O4	ERα	P03372	CRBN	WO-2023212599-A9
TPD-OP74FR	SCHEMBL26625091	N-(2,6-dioxopiperidin-3-yl)-4-[4-[2-[4-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperazin-1-yl]ethyl]piperazin-1-yl]benzamide; SCHEMBL30619695	O=C1CCC(NC(=O)C2=CC=C(N3CCN(CCN4CCN(C5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)CC3)C=C2)C(=O)N1	C44H50N6O4	ERα	P03372	CRBN	WO-2023212599-A9
TPD-FC634U	SCHEMBL26624998	3-[4-[4-[2-[4-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperazin-1-yl]ethyl]piperazin-1-yl]anilino]piperidine-2,6-dione	O=C1CCC(NC2=CC=C(N3CCN(CCN4CCN(C5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)CC3)C=C2)C(=O)N1	C43H50N6O3	ERα	P03372	CRBN	WO-2023212599-A9
TPD-DL2X8T	SCHEMBL26625260	3-[5-[4-[2-[4-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperazin-1-yl]ethyl]piperazin-1-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	CN1C(=O)N(C2CCC(=O)NC2=O)C2=C1C=C(N1CCN(CCN3CCN(C4=CC=C([C@@H]5C6=C(C=C(O)C=C6)CC[C@@H]5C5=CC=CC=C5)C=C4)CC3)CC1)C=C2	C45H51N7O4	ERα	P03372	CRBN	WO-2023212599-A9
TPD-CUKASD	SCHEMBL26625226	N-(2,6-dioxopiperidin-3-yl)-4-[4-[3-[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]propanoyl]piperazin-1-yl]benzamide; SCHEMBL30619761	O=C1CCC(NC(=O)C2=CC=C(N3CCN(C(=O)CCC4CCN(C5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)CC3)C=C2)C(=O)N1	C46H51N5O5	ERα	P03372	CRBN	WO-2023212599-A9
TPD-OP77NC	SCHEMBL26625178	3-[4-[4-[3-[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]propyl]piperazin-1-yl]anilino]piperidine-2,6-dione	O=C1CCC(NC2=CC=C(N3CCN(CCCC4CCN(C5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)CC3)C=C2)C(=O)N1	C45H53N5O3	ERα	P03372	CRBN	WO-2023212599-A9
TPD-M3TK88	SCHEMBL26625058	3-[5-[4-[3-[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]propyl]piperazin-1-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	CN1C(=O)N(C2CCC(=O)NC2=O)C2=C1C=C(N1CCN(CCCC3CCN(C4=CC=C([C@@H]5C6=C(C=C(O)C=C6)CC[C@@H]5C5=CC=CC=C5)C=C4)CC3)CC1)C=C2	C47H54N6O4	ERα	P03372	CRBN	WO-2023212599-A9
TPD-3ADSJB	SCHEMBL26625117	1-[4-[4-[3-[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]propyl]piperazin-1-yl]phenyl]-1,3-diazinane-2,4-dione	O=C1CCN(C2=CC=C(N3CCN(CCCC4CCN(C5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)CC3)C=C2)C(=O)N1	C44H51N5O3	ERα	P03372	CRBN	WO-2023212599-A9
TPD-R8IJAG	WO2023212599A9_233	.	O=C1CCC(NC2=CC=C(N3CCC(CN4CCN(C5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)CC3)C=C2)C(=O)N1	C43H49N5O3	ERα	P03372	CRBN	WO-2023212599-A9
TPD-SSIP8H	SCHEMBL26625242	3-[5-[4-[[4-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperazin-1-yl]methyl]piperidin-1-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	CN1C(=O)N(C2CCC(=O)NC2=O)C2=C1C=C(N1CCC(CN3CCN(C4=CC=C([C@@H]5C6=C(C=C(O)C=C6)CC[C@@H]5C5=CC=CC=C5)C=C4)CC3)CC1)C=C2	C45H50N6O4	ERα	P03372	CRBN	WO-2023212599-A9
TPD-BO96DD	WO2023215906A1_4	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl N-[2-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-4-yl]ethyl]carbamate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)NCCC4=CC=CC6=C4N(C)C(=O)N6C4CCC(=O)NC4=O)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC(O)=C2	C50H50F2N10O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-VO6RUS	WO2023215906A1_5	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl N-[5-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]pentyl]carbamate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)NCCCCCC4=CC=C6C(=C4)N(C)C(=O)N6C4CCC(=O)NC4=O)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC(O)=C2	C53H56F2N10O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-6GP37O	WO2023215906A1_6	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)NCCCCC4=CC=C6C(=C4)N(C)C(=O)N6C4CCC(=O)NC4=O)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC(O)=C2	C52H54F2N10O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-H5M3XT	WO2023215906A1_7	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl N-[5-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-4-yl]pentyl]carbamate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)NCCCCCC4=C6C(=CC=C4)N(C4CCC(=O)NC4=O)C(=O)N6C)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC(O)=C2	C53H56F2N10O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-I2731S	WO2023215906A1_8	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)NCCCCC4=CC=CC6=C4N(C)C(=O)N6C4CCC(=O)NC4=O)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC(O)=C2	C52H54F2N10O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-XQWOQJ	WO2023215906A1_9	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl N-[11-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]undecyl]carbamate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)NCCCCCCCCCCCC4=CC=C6C(=C4)N(C)C(=O)N6C4CCC(=O)NC4=O)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC(O)=C2	C59H68F2N10O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-CUK0MZ	SCHEMBL26635105	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl N-[9-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]nonyl]carbamate	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=NC(OC[C@@]56CCCN5[C@H](COC(=O)NCCCCCCCCCC5=CC=C7C(=C5)N(C)C(=O)N7C5CCC(=O)NC5=O)CC6)=NC(N5CC6CCC(C5)N6)=C4C=N3)=C21	C57H64F2N10O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-U9MZ52	SCHEMBL26829615	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl N-[11-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-4-yl]undecyl]carbamate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)NCCCCCCCCCCCC4=CC=CC6=C4N(C)C(=O)N6C4CCC(=O)NC4=O)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC(O)=C2	C59H68F2N10O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-96GHDC	WO2023215906A1_12	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl N-[9-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-4-yl]nonyl]carbamate	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=NC(OC[C@@]56CCCN5[C@H](COC(=O)NCCCCCCCCCC5=CC=CC7=C5N(C)C(=O)N7C5CCC(=O)NC5=O)CC6)=NC(N5CC6CCC(C5)N6)=C4C=N3)=C21	C57H64F2N10O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-8AO727	WO2023215906A1_13	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)NCCCCCCCCCCC4=CC=C6C(=C4)N(C)C(=O)N6C4CCC(=O)NC4=O)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC(O)=C2	C58H66F2N10O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-E3BD32	WO2023215906A1_14	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl N-[10-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-4-yl]decyl]carbamate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)NCCCCCCCCCCC4=CC=CC6=C4N(C)C(=O)N6C4CCC(=O)NC4=O)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC(O)=C2	C58H66F2N10O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-K7CQ03	WO2023215906A1_15	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)NCCCCCCCCCCNC4=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC(O)=C2	C58H64F2N10O8	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-UM2KCS	WO2023215906A1_16	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)NCCCCCCCCCNC4=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=C(O)C=C2	C57H62F2N10O8	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-WIF0TF	WO2023215906A1_17	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4C(COC(=O)NCCCCCCNC4=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC(O)=C2	C54H56F2N10O8	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-7DU7FJ	SCHEMBL26829927	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl N-[8-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]octyl]carbamate	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=NC(OC[C@@]56CCCN5[C@H](COC(=O)NCCCCCCCCNC5=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C5)CC6)=NC(N5CC6CCC(C5)N6)=C4C=N3)=C21	C56H60F2N10O8	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-NGPDDJ	WO2023215906A1_19	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)NCCCCNC4=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC(O)=C2	C52H52F2N10O8	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-SVXW7P	WO2023215906A1_20	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl N-[3-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]propyl]carbamate	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=NC(OC[C@@]56CCCN5[C@H](COC(=O)NCCCNC5=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C5)CC6)=NC(N5CC6CCC(C5)N6)=C4C=N3)=C21	C51H50F2N10O8	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-2BGDTT	WO2023215906A1_21	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)NCCCCCCNC4=CC=CC6=C4C(=O)N(C4CCC(=O)NC4=O)C6=O)CC5)=NC(N4CC5CC(C4)N5)=C3C=N1)=CC(O)=C2	C53H54F2N10O8	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-ZIJFI5	WO2023215906A1_22	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@]45CCCN4[C@@H](COC(=O)NCCCCCCNC4=CC=CC6=C4C(=O)N(C4CCC(=O)NC4=O)C6=O)CC5)=NC(N4CC5CC(C4)N5)=C3C=N1)=CC(O)=C2	C53H54F2N10O8	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-62FGFI	WO2023215906A1_23	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OCC45CCCN4C(COC(=O)NCCCCCCCCCNC4=CC=CC6=C4C(=O)N(C4CCC(=O)NC4=O)C6=O)CC5)=NC(N4CC5CC(C4)N5)=C3C=N1)=CC(O)=C2	C56H60F2N10O8	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-X969JS	WO2023215906A1_24	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OCC45CCCN4C(COC(=O)NCCCCCCNC4=CC=CC6=C4C(=O)N(C4CCC(=O)NC4=O)C6=O)CC5)=NC(N4CC5CC(C4)N5)=C3C=N1)=CC(O)=C2	C53H54F2N10O8	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-0JQVR0	WO2023215906A1_25	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@]45CCCN4[C@@H](COC(=O)NCCOCCOCCNC4=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC(O)=C2	C54H56F2N10O10	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-BEPSUX	WO2023215906A1_26	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)NCCCCCCCCNC4=CC=CC6=C4C(=O)N(C4CCC(=O)NC4=O)C6=O)CC5)=NC(N4CC5CC(C4)N5)=C3C=N1)=CC(O)=C2	C55H58F2N10O8	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-Q9HQ0P	WO2023215906A1_27	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@]45CCCN4[C@@H](COC(=O)NCCOCCOCCOCCNC4=CC=CC6=C4C(=O)N(C4CCC(=O)NC4=O)C6=O)CC5)=NC(N4CC5CC(C4)N5)=C3C=N1)=CC(O)=C2	C55H58F2N10O11	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-7JEKZP	WO2023215906A1_28	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)NCCOCCOCCOCCNC4=CC=CC6=C4C(=O)N(C4CCC(=O)NC4=O)C6=O)CC5)=NC(N4CC5CC(C4)N5)=C3C=N1)=CC(O)=C2	C55H58F2N10O11	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-B5UDV8	WO2023215906A1_29	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)NCCCCCCCCC4=CC6=C(C=C4)N(C4CCC(=O)NC4=O)C(=O)N6C)CC5)=NC(N4CC5CC(C4)N5)=C3C=N1)=CC=C2	C55H60F2N10O6	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-2IR69E	SCHEMBL26635036	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 4-[3-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-4-yl]prop-2-ynoxy]piperidine-1-carboxylate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCC#CC6=CC=CC7=C6N(C)C(=O)N7C6CCC(=O)NC6=O)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C56H56F2N10O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-KRBVZB	SCHEMBL26635049	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 4-[3-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-4-yl]propoxy]piperidine-1-carboxylate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCCCC6=CC=CC7=C6N(C)C(=O)N7C6CCC(=O)NC6=O)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C56H60F2N10O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-ITSA97	WO2023215906A1_32	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCCCC6=CC=CC7=C6N(C)C(=O)N7C6CCC(=O)NC6=O)CC4)CC5)=NC(N4CC5CC(C4)N5)=C3C=N1)=CC(O)=C2	C55H58F2N10O8	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-LWYZO6	WO2023215906A1_33	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCC#CC6=CC=CC7=C6N(C)C(=O)N7C6CCC(=O)NC6=O)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC(O)=C2	C56H56F2N10O8	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-SYAW5T	WO2023215906A1_34	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCCCC6=C7C(=CC=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC4)CC5)=NC(N4CCCC5(CCO5)C4)=C3C=N1)=CC(O)=C2	C57H65F2N9O9	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-MMHC4I	WO2023215906A1_35	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCCCC6=C7C(=CC=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC4)CC5)=NC(N4CCCC5(CCO5)C4)=C3C=N1)=CC(O)=C2	C57H61F2N9O9	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-MGSMF2	WO2023215906A1_36	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCCCC6=C7C(=CC=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC4)CC5)=NC(N4CCCC5(CCO5)C4)=C3C=N1)=CC=C2	C57H61F2N9O8	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-6HPE1S	WO2023215906A1_37	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCC6=C7C(=CC=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C54H56F2N10O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-56II01	WO2023215906A1_38	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=C8C(=CC=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)CC6)CC4)CC5)=NC(N4CC5CC(C4)N5)=C3C=N1)=CC=C2	C58H63F2N11O6	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-W7FDZ2	WO2023215906A1_39	.	C#CC1=C(C2=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)NCCCC(=O)N4CCC(C6=CC=CC7=C6N(C)C(=O)N7C6CCC(=O)NC6=O)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N2)C=CC=C1C1=CC=CC2=C(F)C=CC=C12	C63H65F2N11O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-UMW7KB	WO2023215906A1_40	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC6(CC4)CN(CCCC4=CC=CC7=C4N(C)C(=O)N7C4CCC(=O)NC4=O)CCO6)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C59H65F2N11O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-6KIAI0	WO2023215906A1_41	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=C1C(CCCCC1CCN(C(=O)OC[C@@H]3CC[C@]4(COC5=NC(N6CC7CC(C6)N7)=C6C=NC(C7=CC=CC8=C7C(O)=C(F)C=C8)=C(F)C6=N5)CCCN34)CC1)=CC=C2	C54H60F2N10O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-TW4G7I	SCHEMBL30733865	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 3-[[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperazin-1-yl]methyl]azetidine-1-carboxylate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CC(CN6CCN(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)C4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C56H60F2N12O6	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-FK6064	WO2023215906A1_43	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CCCCC6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC4)CC5)=NC(N4CC5CC(C4)N5)=C3C=N1)=CC=C2	C56H60F2N10O6	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-CJIY3H	WO2023215906A1_44	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C59H65F2N11O6	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-4WMS2N	WO2023215906A1_45	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl N-[4-[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidin-1-yl]-4-oxobutyl]carbamate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)NCCCC(=O)N4CCC(C6=CC=C7C(=C6)N(C)C(=O)N7C6CCC(=O)NC6=O)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C57H61F2N11O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-GHNYEN	WO2023215906A1_46	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC6(CC4)CN(CC#CC4=CC=CC7=C4N(C)C(=O)N7C4CCC(=O)NC4=O)CCO6)CC5)=NC(N4CC5CC(C4)N5)=C3C=N1)=CC=C2	C58H59F2N11O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-R0CK0I	WO2023215906A1_47	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CC6CCN(CC7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C60H67F2N11O6	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-VM70G7	WO2023215906A1_48	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CC6CCN(C7=C8C(=CC=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C59H65F2N11O6	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-2JRPDR	WO2023215906A1_49	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CCC6CCN(CC7=CC=CC8=C7N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C61H69F2N11O6	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-3ILQ4O	WO2023215906A1_50	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 4-[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]but-3-ynoxy]piperidine-1-carboxylate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCCC#CC6=CC=C7C(=C6)N(C)C(=O)N7C6CCC(=O)NC6=O)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C57H58F2N10O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-46X2W3	WO2023215906A1_51	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(C6CCN(CC7=CC=CC8=C7N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C59H65F2N11O6	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-FZXU8L	WO2023215906A1_52	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OC6CCN(CC7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C59H65F2N11O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-QRQ472	WO2023215906A1_53	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(N6CCN(CC7=CC=CC8=C7N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C58H64F2N12O6	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-3EX1KW	WO2023215906A1_54	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 4-[1-[[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-4-yl]methyl]azetidin-3-yl]oxypiperidine-1-carboxylate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OC6CN(CC7=CC=CC8=C7N(C)C(=O)N8C7CCC(=O)NC7=O)C6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C57H61F2N11O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-U2MWRF	SCHEMBL26831452	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 4-[1-[[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]methyl]piperidin-4-yl]piperidine-1-carboxylate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(C6CCN(CC7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C59H65F2N11O6	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-UZBW4L	WO2023215906A1_56	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(N6CCN(CC7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C58H64F2N12O6	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-V6S9ZS	WO2023215906A1_57	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(NC6CCN(CC7=C8C(=CC=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)CC6)CC4)CC5)=NC(N4CC5CC(C4)N5)=C3C=N1)=CC=C2	C58H64F2N12O6	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-PT9TGE	WO2023215906A1_58	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCCCCCCC6=CC=CC7=C6N(C)C(=O)N7C6CCC(=O)NC6=O)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C59H66F2N10O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-71ZSRN	WO2023215906A1_59	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCCCCCCCC6=CC=CC7=C6N(C)C(=O)N7C6CCC(=O)NC6=O)CC4)CC5)=NC(N4CC5CC(C4)N5)=C3C=N1)=CC=C2	C59H66F2N10O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-6CJ95Z	WO2023215906A1_60	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC6(CCC(CCC7=CC=CC8=C7N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CC5CC(C4)N5)=C3C=N1)=CC=C2	C59H64F2N10O6	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-V4NTGU	WO2023215906A1_61	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 6-[2-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-4-yl]ethyl]-2-azaspiro[3.3]heptane-2-carboxylate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CC6(CC(CCC7=CC=CC8=C7N(C)C(=O)N8C7CCC(=O)NC7=O)C6)C4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C56H58F2N10O6	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-UTW4ZN	WO2023215906A1_62	.	C#CC1=C(F)C=CC=C1C1=C(F)C2=NC(OC[C@@]34CCCN3[C@H](COC(=O)N3CCC(OCC5CCN(CC6=CC=CC7=C6N(C)C(=O)N7C6CCC(=O)NC6=O)CC5)CC3)CC4)=NC(N3CC4CC(C3)N4)=C2C=N1	C55H63F2N11O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-LE0H43	WO2023215906A1_63	.	C#CC1=C(F)C=CC=C1C1=CC=CC2=C1C#CC=C2C1=C(F)C2=NC(OC[C@@]34CCCN3[C@H](COC(=O)N3CCC(COC5CN(CC6=CC=CC7=C6N(C)C(=O)N7C6CCC(=O)NC6=O)C5)CC3)CC4)=NC(N3CC4CCC(C3)N4)=C2C=N1	C64H65F2N11O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-BXC190	WO2023215906A1_64	.	C#CC1=C(F)C=CC=C1C1=C(F)C2=NC(OC[C@@]34CCCN3[C@H](COC(=O)N3CCN(C5CCN(CC6=C7C(=CC=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC5)CC3)CC4)=NC(N3CC4CCC(C3)N4)=C2C=N1	C54H62F2N12O6	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-UZDFRG	WO2023215906A1_65	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(N6CCC(CC7=CC=CC8=C7N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CC5CC(C4)N5)=C3C=N1)=CC=C2	C58H63F2N11O6	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-F2UC7X	WO2023215906A1_66	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(N6CCC(OC7=C8C(=CC=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)CC6)CC4)CC5)=NC(N4CC5CC(C4)N5)=C3C=N1)=CC=C2	C57H61F2N11O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-4LED6Q	WO2023215906A1_67	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 2-[2-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]ethyl]-7-azaspiro[3.5]nonane-7-carboxylate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC6(CC4)CC(CCC4=CC=C7C(=C4)N(C)C(=O)N7C4CCC(=O)NC4=O)C6)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C58H62F2N10O6	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-IBS4L8	WO2023215906A1_68	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(COC6CCN(CC7=CC8=C(C=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)CC6)CC4)CC5)=NC(N4CC5CC(C4)N5)=C3C=N1)=CC=C2	C59H65F2N11O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-GWMW4A	WO2023215906A1_69	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CCC6CCN(CC7=CC8=C(C=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)CC6)CC4)CC5)=NC(N4CC5CC(C4)N5)=C3C=N1)=CC=C2	C60H67F2N11O6	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-GBOB1R	SCHEMBL26832070	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 4-[1-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidin-4-yl]piperidine-1-carboxylate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(C6CCN(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C58H63F2N11O6	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-WRUCI3	WO2023215906A1_71	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 4-[[1-[[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]methyl]piperidin-4-yl]methoxy]piperidine-1-carboxylate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCC6CCN(CC7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C60H67F2N11O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-SQA71Q	WO2023215906A1_72	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 4-[1-[[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]methyl]piperidin-4-yl]piperazine-1-carboxylate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCN(C6CCN(CC7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C58H64F2N12O6	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-T41S36	WO2023215906A1_73	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 4-[[1-[[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]methyl]azetidin-3-yl]oxymethyl]piperidine-1-carboxylate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(COC6CN(CC7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)C6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C58H63F2N11O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-MAPIRP	WO2023215906A1_74	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 4-[1-[[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]methyl]azetidin-3-yl]oxypiperidine-1-carboxylate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OC6CN(CC7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)C6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C57H61F2N11O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-VX4EIR	WO2023215906A1_75	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 4-[4-[[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]methyl]piperidin-1-yl]piperidine-1-carboxylate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(N6CCC(CC7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C59H65F2N11O6	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-960N9N	WO2023215906A1_76	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@]45CCCN4[C@@H](COC(=O)N4CCC(CN6CCC(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C59H65F2N11O6	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-7X4C86	WO2023215906A1_77	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@]45CCCN4[C@@H](COC(=O)N4CCC(CC6CCN(CC7=CC=CC8=C7N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C60H67F2N11O6	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-E33LY8	WO2023215906A1_78	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CC(CN6CCC(OC7=C8C(=CC=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)CC6)C4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C57H61F2N11O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-RZ5A9D	SCHEMBL26832313	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 4-[[4-[3-methyl-1-(1-methyl-2,6-dioxopiperidin-3-yl)-2-oxobenzimidazol-4-yl]piperidin-1-yl]methyl]piperidine-1-carboxylate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=C8C(=CC=C7)N(C7CCC(=O)N(C)C7=O)C(=O)N8C)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C60H67F2N11O6	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-FB778C	WO2023215906A1_80	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl (3R)-3-[[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidin-1-yl]methyl]pyrrolidine-1-carboxylate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CC[C@H](CN6CCC(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)C4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C58H63F2N11O6	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-0SQBO8	SCHEMBL26832319	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl (3S)-3-[[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidin-1-yl]methyl]pyrrolidine-1-carboxylate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CC[C@@H](CN6CCC(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)C4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C58H63F2N11O6	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-JJXDOK	WO2023215906A1_82	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC(O)=C2	C59H65F2N11O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-6ZRS8V	WO2023215906A1_83	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CC(OC6CCN(CC7=C8C(=CC=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)CC6)C4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C57H61F2N11O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-71I2M8	WO2023215906A1_84	.	CN1C(=O)C(C2CCC(=O)NC2=O)C2=CC=CC(CN3CCN(CCC4CCN(C(=O)OC[C@@H]5CC[C@]6(COC7=NC(N8CC9CCC(C8)N9)=C8C=NC(C9=CC=CC%10=C9C(C#N)=C(F)C=C%10)=C(F)C8=N7)CCCN56)CC4)CC3)=C21	C60H68F2N12O6	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-X2GKHW	WO2023215906A1_85	.	C#CC1=C(F)C=CC=C1C1=C(F)C2=NC(OC[C@@]34CCCN3[C@H](COC(=O)N3CCN(CCC5CCN(CC6=C7C(=CC=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC5)CC3)CC4)=NC(N3CC4CCC(C3)N4)=C2C=N1	C56H66F2N12O6	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-T3MKC5	SCHEMBL26635006	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 4-[2-[4-[[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]methyl]piperazin-1-yl]ethyl]piperidine-1-carboxylate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CCN6CCN(CC7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C60H68F2N12O6	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-ENPFAS	WO2023215906A1_88	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCN(CCC6CCN(CC7=CC8=C(C=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)CC6)CC4)CC5)=NC(N4CC5CC(C4)N5)=C3C=N1)=CC=C2	C59H66F2N12O6	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-EYF348	SCHEMBL26635010	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 3-[1-[[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]methyl]piperidin-4-yl]oxyazetidine-1-carboxylate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CC(OC6CCN(CC7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)C4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C57H61F2N11O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-QFLFZ8	WO2023215906A1_90	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N(C)CCCCCN(CC)C/C=C/N(C)C(=O)N(/C=C/C)C4CCC(=O)NC4=O)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C56H69F2N11O6	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-STAIXF	WO2023215906A1_91	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)N(C)C7=O)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C60H67F2N11O6	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-LQI5QN	WO2023215906A1_92	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCC#CC#CC6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC4)CC5)=NC(N4CC5CC(C4)N5)=C3C=N1)=CC=C2	C57H54F2N10O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-4KG829	WO2023215906A1_93	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCC#CC#CC6=C7C(=CC=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C58H56F2N10O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-IOJ2CT	SCHEMBL26634950	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 4-[[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]triazol-1-yl]methyl]piperidine-1-carboxylate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6C=C(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)N=N6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C56H57F2N13O6	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-6SIXSE	WO2023215906A1_95	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CCN6C=C(C7=CC8=C(C=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)N=N6)CC4)CC5)=NC(N4CC5CC(C4)N5)=C3C=N1)=CC=C2	C56H57F2N13O6	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-SDLMDC	SCHEMBL26634896	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 4-[[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-4-yl]triazol-1-yl]methyl]piperidine-1-carboxylate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6C=C(C7=C8C(=CC=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)N=N6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C56H57F2N13O6	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-5YHYZV	WO2023215906A1_97	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=CC(C3=CN(CCC4CCN(C(=O)OC[C@@H]5CC[C@]6(COC7=NC(N8CC9CCC(C8)N9)=C8C=NC(C9=CC=CC%10=C9C(C#N)=C(F)C=C%10)=C(F)C8=N7)CCCN56)CC4)N=N3)=C21	C56H58F2N14O6	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-D7I5UG	WO2023215906A1_98	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OC6CCN(C7=CC8=C(C=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)CC6)CC4)CC5)=NC(N4CC5CC(C4)N5)=C3C=N1)=CC=C2	C57H61F2N11O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-KBUTJA	WO2023215906A1_99	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OC6CCN(C(C=C)[C@H]7CN(C)C(=O)N7C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C57H67F2N11O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-NMGG72	SCHEMBL26635003	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 4-[[3-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-4-yl]oxyazetidin-1-yl]methyl]piperidine-1-carboxylate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CC(OC7=C8C(=CC=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)C6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C57H61F2N11O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-CX0N8X	SCHEMBL26635274	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 3-[[1-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidin-4-yl]methoxy]azetidine-1-carboxylate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CC(OCC6CCN(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)C4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C57H61F2N11O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-CGQXDD	WO2023215906A1_102	.	C#CC1=C(F)C=CC=C1C1=C(F)C2=NC(OC[C@@]34CCCN3[C@H](COC(=O)N3CCC(COC5CN(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)C5)CC3)CC4)=NC(N3CC4CC(C3)N4)=C2C=N1	C52H57F2N11O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-JPELOY	WO2023215906A1_103	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CC6CC(CN7CCC(C8=CC=C9C(=C8)N(C)C(=O)N9C8CCC(=O)NC8=O)CC7)C6C4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C60H65F2N11O6	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-YY1GB7	WO2023215906A1_104	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(N3CCC(OCC4CN(C(=O)OC[C@@H]5CC[C@]6(COC7=NC(N8CC9CCC(C8)N9)=C8C=NC(C9=CC=CC%10=C9C(C#N)=C(F)C=C%10)=C(F)C8=N7)CCCN56)C4)CC3)C=C21	C56H60F2N12O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-70QJEH	WO2023215906A1_105	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(C#CCOCCC3CCN(C(=O)OC[C@@H]4CC[C@@]5(COC6=NC(N7CC8CC(C7)N8)=C7C=NC(C8=CC=CC9=C8C(O)=C(F)C=C9)=C(F)C7=N6)CCCN45)CC3)C=C21	C55H58F2N10O8	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-NLL2PD	WO2023215906A1_106	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(N3CCN(CC4CCN(C(=O)OC[C@@H]5CC[C@@]6(COC7=NC(N8CC9CC(C8)N9)=C8C=NC(C9=CC=CC%10=CC=C(F)C(O)=C%109)=C(F)C8=N7)CCCN56)CC4)CC3)C=C21	C55H62F2N12O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-KTY1FL	WO2023215906A1_107	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CCCC(C#CCCOC3CCN(C(=O)OC[C@@H]4CC[C@]5(COC6=NC(N7CC8CC(C7)N8)=C7C=NC(C8=CC=CC9=C8C(C#N)=CC=C9)=C(F)C7=N6)CCCN45)CC3)=C21	C55H58FN11O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-LU8TKV	WO2023215906A1_108	.	C#CC1=C(F)C=CC2=C1C(C1=NC=C3C(N4CC5CC(C4)N5)=NC(OC[C@@]45CCCN4[C@@H](COC(=O)N4CCC(CN(C)C6CCN(C7=C8C(=CC=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)CC6)CC4)CC5)=NC3=C1F)=CC=C2	C59H66F2N12O6	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-IS8L1E	WO2023215906A1_109	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=CC(N3CCC(N(C)CCCNC(=O)OC[C@@H]4CC[C@]5(COC6=NC(N7CC8CC(C7)N8)=C7C=NC(C8=CC=CC9=C8C(C#N)=C(F)C=C9)=C(F)C7=N6)CCCN45)CC3)=C21	C55H61F2N13O6	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-VC3CYE	WO2023215906A1_110	.	N#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCC[C@@H]4[C@H](COC(=O)NCCCC(=O)N4CCN(C6=C7NC(=O)N(C8CCC(=O)NC8=O)C7=CC=C6)CC4)CC5)=NC(N4CC5CC(C4)N5)=C3C=N1)=CC=C2	C54H56F2N12O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-8LHS7X	WO2023215906A1_111	.	C#CC1=C(F)C=CC2=C1C(C1N=CC3=C(N4CC5CCC(C4)N5)N=C(OC[C@@]45CCCN4[C@H](COC(=O)N4CCO[C@@H](CN6CCN(C7=C8C(=CC=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)CC6)C4)CC5)N=C3C1F)=CCC2	C57H66F2N12O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-5UUHB4	WO2023215906A1_112	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=CC(N3CCN(CC4CCN(C(=O)OC[C@@H]5CC[C@@]6(COC7=NC(N8CC9CC(C8)N9)=C8C=NC(C9=CCCC%10=C9C(C#N)=C(F)C=C%10)=C(F)C8=N7)CCCN56)CC4)CC3)=C21	C56H63F2N13O6	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-QWK4A6	WO2023215906A1_113	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=CC(N3CCN(CC4CN(C(=O)OC[C@@H]5CC[C@@H](COC6=NC(N7CC8CCC(C7)N8)=C7C=NC(C8=CC=CC9=C8C(N)C(F)C=C9)=C(F)C7=N6)N5CCC#N)C4)CC3)=C21	C54H62F2N14O6	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-KQIV8Z	WO2023215906A1_114	.	COC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCCCC#CC6=CC=C7C(=C6)N(C)C(=O)N7C6CCC(=O)NC6=O)CC4)CC5)=NC(N4CC5CC(C4)N5)=C3C=N1)=CC=C2	C56H60F2N10O8	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-RCZLKT	WO2023215906A1_115	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(C#CCOC3CCN(C(=O)OC[C@@H]4CC[C@@]5(COC6=NC(N7CC8CC(C7)N8)=C7C=NC(C8=CC=CC9=C8C(O)=C(F)C=C9)=C(F)C7=N6)CCCN45)CC3)C=C21	C53H54F2N10O8	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-JGM9NP	WO2023215906A1_116	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCC6=CC=C7C(=C6)N(C)C(=O)N7C6CCC(=O)NC6=O)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C54H56F2N10O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-4Z0V2V	WO2023215906A1_117	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCCCCC6=CC=CC7=C6N(C)C(=O)N7C6CCC(=O)NC6=O)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C57H62F2N10O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-LKX3KF	WO2023215906A1_118	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCCCCC6=CC=C7C(=C6)N(C)C(=O)N7C6CCC(=O)NC6=O)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C57H62F2N10O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-KIH156	WO2023215906A1_119	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCCCC#CC6=CC=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC4)CC5)=NC(N4CC5CC(C4)N5)=C3C=N1)=CC=C2	C57H55F2N9O8	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-C70LHZ	WO2023215906A1_120	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(CCCCCOC3CCN(C(=O)OC[C@@H]4CC[C@]5(COC6=NC(N7CC8CC(C7)N8)=C7C=NC(C8=CC=CC9=C8C(C#N)=C(F)C=C9)=C(F)C7=N6)CCCN45)CC3)C=C21	C56H61F2N11O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-ABUJXF	WO2023215906A1_121	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=CC(N3CCC4(CC3)CN(C(=O)OC[C@@H]3CC[C@]5(COC6=NC(N7CC8CC(C7)N8)=C7C=NC(C8=CCCC9=C8C(C#N)=C(F)C=C9)=C(F)C7=N6)CCCN35)C4)=C21	C53H56F2N12O6	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-76BD8Z	WO2023215906A1_122	.	C#CC1=C(F)C=CC=C1C1=C(F)C2=NC(OC[C@@]34CCCN3[C@H](COC(=O)N3CCC(OCCCCCC5=C6C(=CC=C5)N(C5CCC(=O)NC5=O)C(=O)N6C)CC3)CC4)=NC(N3CC4CCC(C3)N4)=C2C=N1	C54H62F2N10O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-OFV71K	WO2023215906A1_123	.	C#CC1=C(F)C=CC=C1C1=C(F)C2=NC(OCC34CCCN3[C@H](COC(=O)NCCOCCN3CCN(C5=C6C(=CC=C5)N(C5CCC(=O)NC5=O)C(=O)N6C)CC3)CC4)=NC(N3CC4CCC(C3)N4)=C2C=N1	C52H60F2N12O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-G7N2D0	WO2023215906A1_124	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=C1C(CCC1CC3(CCN(C(=O)OC[C@@H]4CC[C@]5(COC6=NC(N7CC8CC(C7)N8)=C7C=NC(C8=CC=CC9=C8C(C#N)=C(F)C=C9)=C(F)C7=N6)CCCN45)CC3)C1)=CC=C2	C56H59F2N11O6	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-FLI6SJ	WO2023215906A1_125	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=C1C(C#CCN1CCO[C@H](CNC(=O)OC[C@@H]3CC[C@]4(COC5=NC(N6CC7CC(C6)N7)=C6C=NC(C7=CC=CC8=C7C(C#N)=C(F)C=C8)=C(F)C6=N5)CCCN34)C1)=CC=C2	C54H54F2N12O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-QOWDWD	SCHEMBL26635292	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl N-[[(2R)-4-[3-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-4-yl]propyl]morpholin-2-yl]methyl]carbamate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)NC[C@@H]4CN(CCCC6=CC=CC7=C6N(C)C(=O)N7C6CCC(=O)NC6=O)CCO4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C56H61F2N11O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-KN9M7Q	WO2023215906A1_127	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=CC(N3CCC(C4CCN(C(=O)OC[C@@H]5CC[C@@]6(COC7=NC(N8CC9CC(C8)N9)=C8C=NC(C9=CC=CC%10=C9C(C#N)=C(F)C=C%10)=C(F)C8=N7)CCCN56)CC4)CC3)=C21	C56H60F2N12O6	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-2VHZJG	WO2023215906A1_128	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=C1C(CN1CCC(OCC3CCN(C(=O)OC[C@@H]4CC[C@@]5(COC6=NC(N7CC8CCC(C7)N8)=C7C=NC(C8=CC=CC9=CC(F)=C(F)C(O)=C98)C(F)C7=N6)CCCN45)CC3)CC1)=CC=C2	C58H68F3N11O8	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-F05B4K	WO2023215906A1_129	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=CC(N3CCC4(CCN(C(=O)OC[C@@H]5CC[C@@]6(COC7=NC(N8CC9CC(C8)N9)=C8C=NC(C9=CC=CC%10=C9C(O)=C(F)C=C%10)=C(F)C8=N7)CCCN56)CC4)CC3)=C21	C54H59F2N11O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-U36W5O	WO2023215906A1_130	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OC6CCN(CC7=CC=CC8=C7N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C59H65F2N11O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-TFON1T	WO2023215906A1_131	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=CC(N3CCN(C4CCN(C(=O)OC[C@@H]5CC[C@@]6(COC7=NC(N8CC9CC(C8)N9)=C8C=NC(C9=CC=CC%10=C9C(C#N)=C(F)C=C%10)=C(F)C8=N7)CCCN56)CC4)CC3)=C21	C55H59F2N13O6	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-E7JBXJ	WO2023215906A1_132	.	C#CC1=C(F)C=CC=C1C1=C(F)C2=NC(OC[C@@]34CCCN3[C@H](COC(=O)N3CCC(CC5CCN(CC6=C7C(=CC=C6)C(C6CCC(=O)NC6=O)C(=O)N7C)CC5)CC3)CC4)=NC(N3CC4CCC(C3)N4)=C2C=N1	C57H66F2N10O6	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-WM7QM8	SCHEMBL26635019	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 4-[2-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]ethoxy]piperidine-1-carboxylate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCCC6=CC=C7C(=C6)N(C)C(=O)N7C6CCC(=O)NC6=O)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C55H58F2N10O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-8U0BMW	WO2023215906A1_134	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N(C)CCC4CCN(CC6=C7C(=CC=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C57H63F2N11O6	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-Q8MORU	SCHEMBL26635146	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 4-[2-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-4-yl]ethoxy]piperidine-1-carboxylate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCCC6=CC=CC7=C6N(C)C(=O)N7C6CCC(=O)NC6=O)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C55H58F2N10O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-F2LUTR	WO2023215906A1_136	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OCC45CCCN4[C@H](COC(=O)N4CCC(OCCCC6C=C7C(=CC6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C56H62F2N10O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-K177RH	WO2023215906A1_138	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(CCCCCCCCNC(=O)OC[C@H]3CC[C@@]4(COC5=NC(N6CC7CCC(C6)N7)=C6C=NC(C7=CC(O)=CC8=C7C(C#N)=C(F)C=C8)=C(F)C6=N5)CCCN34)C=C21	C55H61F2N11O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-9CX3Z7	WO2023215906A1_139	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)NCCCCCCCC4=CC=C6C(=C4)N(C)C(=O)N6C4CCC(=O)NC4=O)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC(O)=C2	C55H60F2N10O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-G0T7SF	WO2023215906A1_140	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCC[C@@H]4[C@H](COC(=O)NCCCCCCCCC4=C6C(=CC=C4)N(C4CCC(=O)NC4=O)C(=O)N6C)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC(O)=C2	C57H63F2N9O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-ECQCJP	WO2023215906A1_141	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)NCCCCCCCC4=C6C(=CC=C4)N(C4CCC(=O)NC4=O)C(=O)N6C)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC(O)=C2	C55H60F2N10O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-VW43LT	WO2023215906A1_142	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)NCCCCCCC4=CC=C6C(=C4)N(C)C(=O)N6C4CCC(=O)NC4=O)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC(O)=C2	C54H58F2N10O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-HDDQ11	WO2023215906A1_143	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)NCCCCCCC4=CC=CC6=C4N(C)C(=O)N6C4CCC(=O)NC4=O)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC(O)=C2	C54H58F2N10O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-BH3VCU	WO2023215906A1_144	.	C#CC1=C(F)C=CC=C1C1=C(F)C2=NC(OC[C@@]34CCCN3[C@H](COC(=O)N3CCC(OCCCC5=C6C(=CC=C5)N(C5CCC(=O)N(C)C5=O)C(=O)N6C)CC3)CC4)=NC(N3CC4CCC(C3)N4)=C2C=N1	C53H60F2N10O7	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-EJSLDH	WO2023215906A1_145	.	C#CC1=C(F)C=CC=C1C1=C(F)C2=NC(OC[C@@]34CCCN3[C@H](COC(=O)N3CCC(CNC5CCN(CC6=CC=CC7=C6N(C)C(=O)N7C6CCC(=O)NC6=O)CC5)CC3)CC4)=NC(N3CC4CCC(C3)N4)=C2C=N1	C56H66F2N12O6	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-3WWLXV	WO2023215906A1_146	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)NCCCC(=O)N4CCN(C6=CC=C(N7CCC(=O)NC7=O)C=C6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C53H57F2N11O6	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-Y6WNTC	SCHEMBL26635012	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl N-[5-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperazin-1-yl]-5-oxopentyl]carbamate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)NCCCCC(=O)N4CCN(C6=CC=C(N7CCC(=O)NC7=O)C=C6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C54H59F2N11O6	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-L6W590	WO2023215906A1_148	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl N-[6-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperazin-1-yl]-6-oxohexyl]carbamate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)NCCCCCC(=O)N4CCN(C6=CC=C(N7CCC(=O)NC7=O)C=C6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C55H61F2N11O6	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-3XWF4E	WO2023215906A1_149	.	C#CC1=C(F)C=CC=C1C1=C(F)C2=NC(OC[C@@]34CCCN3[C@H](COC(=O)NCCCCCCC(=O)N3CCN(C5=CC=C(N6CCC(=O)NC6=O)C=C5)CC3)CC4)=NC(N3CC4CCC(C3)N4)=C2C=N1	C52H61F2N11O6	KRAS	P01116	CRBN	WO-2023215906-A1
TPD-FDQP7S	WO2023222012A1_100	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CC5CN(C[C@@H]6[C@H]7CN(c8ccc9c(c8)C(=O)N(C8CCC(=O)NC8=O)C9=O)C[C@@H]67)CC5C4)nn3)CC2)CC1Cl	C43H46ClN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-O6SL07	WO2023222012A1_101	.	CC1(C)[C@H](NC(=O)c2ccc(N3CCN(C[C@@H]4[C@H]5CN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)C[C@@H]45)CC3)nn2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C43H45ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-1RVDT6	WO2023222012A1_102	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCN(C[C@@H]5[C@H]6CN(c7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)C[C@@H]56)CC4)nn3)CC2)cc1Cl	C41H42ClN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-XHOM7M	WO2023222012A1_103	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(N5CC6(CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)C6)C5)CC4)nn3)CC2)cc1Cl	C42H43ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-HVCA33	WO2023222012A1_104	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCN(C[C@@H]5[C@H]6CN(c7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)C[C@@H]56)CC4)cn3)CC2)cc1Cl	C41H42ClN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-42WIJ3	WO2023222012A1_105	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3nnc(N4CC5(CCN(CC6CCN(c7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)C4)s3)CC2)cc1Cl	C42H46ClN9O6S	AR	P10275	CRBN	WO-2023222012-A1
TPD-5HRIOP	WO2023222012A1_106	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ncc(N4CC5(CCN(C6CCN(c7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)C4)cn3)CC2)cc1Cl	C43H46ClN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-VLVIWZ	WO2023222012A1_107	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3nnc(N4CC5(CCN(CC6CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)C4)s3)CC2)cc1Cl	C42H45ClFN9O6S	AR	P10275	CRBN	WO-2023222012-A1
TPD-INNGO5	WO2023222012A1_108	.	N#Cc1ccc(CN2CCC(NC(=O)c3ccc(N4CCC(CN5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)nn3)CC2)cc1Cl	C41H45ClN10O5	AR	P10275	CRBN	WO-2023222012-A1
TPD-19U6OK	WO2023222012A1_109	.	N#Cc1ccc(OC2CC3(CC(NC(=O)c4ccc(N5CCC(CN6CCN(c7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)nn4)C3)C2)cc1Cl	C42H44ClN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-503WXW	WO2023222012A1_110	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(O[C@H]5CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)nn3)CC2)cc1Cl	C40H40ClFN8O7	AR	P10275	CRBN	WO-2023222012-A1
TPD-N1C0E8	WO2023222012A1_111	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(O[C@@H]5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4)cc3)CC2)cc1Cl	C42H43ClN6O7	AR	P10275	CRBN	WO-2023222012-A1
TPD-OCRQVU	WO2023222012A1_112	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cn([C@H]4CC[C@H](CN5CCC6(CC5)CN(c5cc7c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)cn3)CC2)cc1Cl	C44H48ClFN8O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-P3UVSQ	WO2023222012A1_113	.	Cc1cc(O[C@H]2CC[C@H](NC(=O)c3cn([C@H]4CC[C@H](CN5CCC6(CC5)CN(c5cc7c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)cn3)CC2)ccc1C#N	C45H51FN8O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-50TX2E	WO2023222012A1_114	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cn([C@H]4CC[C@H](CN5CCC6(CC5)CN(c5ccc7c(c5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)nn3)CC2)cc1Cl	C43H48ClN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-SRA9XQ	WO2023222012A1_115	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cn([C@H]4CC[C@H](CN5CCC6(CC5)CN(c5cc7c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)nn3)CC2)cc1Cl	C43H47ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-OFZ5XF	WO2023222012A1_116	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnn([C@H]4CC[C@H](CN5CCC6(CC5)CN(c5ccc7c(c5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)n3)CC2)cc1Cl	C43H48ClN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-0F16IG	WO2023222012A1_117	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnn([C@H]4CC[C@H](CN5CCC6(CC5)CN(c5cc7c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)n3)CC2)cc1Cl	C43H47ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-KZPXSP	WO2023222012A1_118	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(NC5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)nn3)CC2)cc1Cl	C41H44ClN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-77RUUT	WO2023222012A1_119	.	CN(C1CCN(c2ccc(C(=O)N[C@H]3CC[C@H](Oc4ccc(C#N)c(Cl)c4)CC3)nn2)CC1)C1CCN(c2cc3c(cc2F)C(=O)N(C2CCC(=O)NC2=O)C3=O)CC1	C42H45ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-SD5APQ	WO2023222012A1_120	.	N#Cc1ccc(OC2CC3(C2)CN(C(=O)c2ccc(N4CCC(CN5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)nn2)C3)cc1Cl	C41H42ClN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-SG7IWA	WO2023222012A1_121	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CC6(C5)CN(c5ccc7c(c5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)nn3)CC2)cc1Cl	C42H44ClN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-P11F8U	WO2023222012A1_122	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CC6(C5)CN(c5cc7c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)nn3)CC2)cc1Cl	C42H43ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-8BFLKK	WO2023222012A1_123	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCC(CN5CC6(C5)CN(c5cc7c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)cn3)CC2)cc1Cl	C42H43ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-UEJVVA	WO2023222012A1_124	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CC5(CN(CC6CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)C5)C4)nn3)CC2)cc1Cl	C42H43ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-JWPNPF	WO2023222012A1_125	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CC5(CN(CC6CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)C5)C4)cn3)CC2)cc1Cl	C42H43ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-BX7ZO4	WO2023222012A1_126	.	N#Cc1ccc(O[C@H]2C=C[C@H](NC(=O)c3ccc(N4CCN(C[C@@H]5[C@H]6CN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)C[C@@H]56)CC4)nn3)CC2)cc1Br	C41H39BrFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-NM8ZR8	WO2023222012A1_127	.	N#Cc1ccc(O[C@H]2C=C[C@H](NC(=O)c3cnc(N4CCN(C[C@@H]5[C@H]6CN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)C[C@@H]56)CC4)cn3)CC2)cc1Br	C41H39BrFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-Q09PHO	WO2023222012A1_128	.	N#Cc1ccc(O[C@H]2C=C[C@H](NC(=O)c3cnc(N4CCN(C[C@@H]5[C@H]6CN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)C[C@@H]56)CC4)nc3)CC2)cc1Cl	C41H39ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-6C9ILL	WO2023222012A1_129	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CC5(CC(N6CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)C5)C4)nn3)CC2)cc1Cl	C41H41ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-Y39PJ2	WO2023222012A1_130	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CC5(CC(N6CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)C5)C4)cn3)CC2)cc1Cl	C41H41ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-8BAYKS	WO2023222012A1_131	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC6(CC5)CN(c5ccc7c(c5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)nn3)CC2)cc1	C44H49N9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-0ZVNCI	WO2023222012A1_132	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC6(CC5)CN(c5cc7c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)nn3)CC2)cc1	C44H48FN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-GWJ9VG	WO2023222012A1_133	.	CN(C(=O)c1ccc(N2CCC(CN3CCN(c4cc5c(cc4F)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)nn1)[C@H]1CC[C@H](Oc2ccc(C#N)c(Cl)c2)CC1	C42H45ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-UDJ5EW	WO2023222012A1_134	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCN(C5CC6(C5)CN(c5cc7c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)cn3)CC2)cc1Cl	C41H41ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-BI0D3E	WO2023222012A1_135	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)c3ncc(N4CCC(CN5CCC6(CC5)CN(c5ccc7c(c5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)cn3)CC2)CC1Cl	C44H50ClN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-MQL4Q8	WO2023222012A1_136	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC6(CC5)CN(c5ccc7c(c5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)nn3)CC2)CC1C(F)(F)F	C45H50F3N9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-1CSJEI	WO2023222012A1_137	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CC(CN5CC6CN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6C5)C4)nn3)CC2)cc1Cl	C41H41ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-ZQQX3Q	WO2023222012A1_138	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CC(CN5CC6CN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6C5)C4)cn3)CC2)cc1Cl	C41H41ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-M1JZK5	WO2023222012A1_139	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC(Nc6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)nn3)CC2)cc1Cl	C42H45ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-X0FR90	WO2023222012A1_140	.	C/C(=C\C=C(\C#N)CCl)O[C@H]1CC[C@H](NC(=O)c2cnc(N(C)CC(C)CN3CC4CN(c5cc6c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4C3)nc2)CC1	C42H49ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-QIEZ9M	WO2023222012A1_141	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCC(CN5CCC6(CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)C6)C5)CC4)cn3)CC2)cc1Cl	C44H47ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-XWUPQX	WO2023222012A1_142	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC6(CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)C6)C5)CC4)nn3)CC2)cc1Cl	C44H47ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-Z9JISY	WO2023222012A1_143	.	Cc1cc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC(Nc6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)nn3)CC2)ccc1C#N	C43H49N9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-D7RKL3	WO2023222012A1_145	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCC(CN5CCC(Nc6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cn3)CC2)cc1Cl	C42H45ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-V8TZGC	WO2023222012A1_146	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCC(CN5CCC(Nc6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cn3)CC2)cc1Cl	C42H46ClN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-KTAIJS	WO2023222012A1_147	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC(Oc6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)nn3)CC2)cc1Cl	C42H45ClN8O7	AR	P10275	CRBN	WO-2023222012-A1
TPD-ZV5SS4	WO2023222012A1_148	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ncc(N4CCC(CN5CCC6(CC5)CN(c5cc7c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)cn3)CC2)cc1Cl	C44H47ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-X8PQCX	WO2023222012A1_149	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ncc(N4CCC(CN5CCC6(CC5)CN(c5ccc7c(c5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)cn3)CC2)cc1Cl	C44H48ClN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-NSDHDE	WO2023222012A1_150	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ncc(N4CC5(CCN(CC6CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)C4)cn3)CC2)cc1Cl	C44H47ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-ET0PKS	WO2023222012A1_151	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC6(CC5)CN(c5ccc7c(c5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)nn3)CC2)cc1C(F)(F)F	C45H48F3N9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-LM6BKQ	WO2023222012A1_152	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC6(CC5)CN(c5cc7c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)nn3)CC2)cc1C(F)(F)F	C45H47F4N9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-KCR37K	WO2023222012A1_153	.	COc1cc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC6(CC5)CN(c5ccc7c(c5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)nn3)CC2)ccc1C#N	C45H51N9O7	AR	P10275	CRBN	WO-2023222012-A1
TPD-P3830C	WO2023222012A1_154	.	CCOc1cc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC6(CC5)CN(c5ccc7c(c5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)nn3)CC2)ccc1C#N	C46H53N9O7	AR	P10275	CRBN	WO-2023222012-A1
TPD-QJ7L8K	WO2023222012A1_155	.	COCCOc1cc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC6(CC5)CN(c5ccc7c(c5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)nn3)CC2)ccc1C#N	C47H55N9O8	AR	P10275	CRBN	WO-2023222012-A1
TPD-SRFD50	WO2023222012A1_156	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CC5CN(CC6CCN(c7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5C4)cn3)CC2)cc1Cl	C43H46ClN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-4GDGF1	WO2023222012A1_157	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CC5CN(CC6CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5C4)cn3)CC2)cc1Cl	C43H45ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-K7SFGO	WO2023222012A1_158	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCC(CN5CCC6(CC5)CN(c5cc7c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)nn3)CC2)cc1Cl	C43H46ClFN10O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-JCQQL9	WO2023222012A1_159	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CC5CN(CC6CN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)C6)CC5C4)cn3)CC2)cc1Cl	C41H41ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-TO321F	WO2023222012A1_160	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CC5CN(CC6CN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)C6)CC5C4)nn3)CC2)cc1Cl	C41H41ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-U9FP9N	WO2023222012A1_161	.	CC1(C)[C@H](NC(=O)c2ccc(N3CC4CN(CC5CN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)CC4C3)nn2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C43H45ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-ZQJSKE	WO2023222012A1_162	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC5(CCN(CC6CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)C5)C4)nn3)CC2)cc1Cl	C44H47ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-E7VUGW	WO2023222012A1_163	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCC5(CCN(CC6CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)C5)C4)cn3)CC2)cc1Cl	C44H47ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-WPKC3B	WO2023222012A1_164	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(N5CCC6(CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)C6)C5)CC4)nn3)CC2)cc1Cl	C43H45ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-OXG2HW	WO2023222012A1_165	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCC(N5CCC6(CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)C6)C5)CC4)cn3)CC2)cc1Cl	C43H45ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-KA149G	WO2023222012A1_166	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC5(CCN(C6CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)C5)C4)nn3)CC2)cc1Cl	C43H45ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-R9EZWF	WO2023222012A1_167	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCC5(CCN(C6CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)C5)C4)cn3)CC2)cc1Cl	C43H45ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-J8EGGR	WO2023222012A1_168	.	C[C@H]1CN(c2ccc(C(=O)N[C@H]3CC[C@H](Oc4ccc(C#N)c(Cl)c4)CC3)nn2)CCN1C[C@H]1[C@@H]2CN(c3cc4c(cc3F)C(=O)N(C3CCC(=O)NC3=O)C4=O)C[C@@H]21	C42H43ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-4WW8DJ	WO2023222012A1_169	.	C[C@H]1CN(c2cnc(C(=O)N[C@H]3CC[C@H](Oc4ccc(C#N)c(Cl)c4)CC3)cn2)CCN1C[C@H]1[C@@H]2CN(c3cc4c(cc3F)C(=O)N(C3CCC(=O)NC3=O)C4=O)C[C@@H]21	C42H43ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-EZBTZF	WO2023222012A1_170	.	C[C@H]1CN(C[C@@H]2[C@H]3CN(c4cc5c(cc4F)C(=O)N(C4CCC(=O)NC4=O)C5=O)C[C@@H]23)CCN1c1ccc(C(=O)N[C@H]2CC[C@H](Oc3ccc(C#N)c(Cl)c3)CC2)nn1	C42H43ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-2CWAA2	WO2023222012A1_171	.	C[C@H]1CN(C[C@@H]2[C@H]3CN(c4cc5c(cc4F)C(=O)N(C4CCC(=O)NC4=O)C5=O)C[C@@H]23)CCN1c1cnc(C(=O)N[C@H]2CC[C@H](Oc3ccc(C#N)c(Cl)c3)CC2)cn1	C42H43ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-JG06DF	WO2023222012A1_172	.	N#Cc1ccc(O[C@H]2CC[C@H](N3Cc4nc(NC5CCN(CC6CCN(c7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)ccc4C3=O)CC2)cc1Cl	C44H47ClN8O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-MW6S0X	WO2023222012A1_173	.	N#Cc1ccc(O[C@H]2CC[C@H](N3Cc4nc(N5CCC(CN6CCC(Nc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)ccc4C3=O)CC2)cc1Cl	C44H47ClN8O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-YKQD0F	WO2023222012A1_174	.	N#Cc1ccc(O[C@@H]2C[C@@H]3CN(C(=O)c4cnc(N5CCC(CN6CCN(c7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)cn4)C[C@@H]3C2)cc1Cl	C42H44ClN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-313L9V	WO2023222012A1_175	.	N#Cc1ccc(O[C@H]2C[C@@H]3CN(C(=O)c4ccc(N5CCC(CN6CCN(c7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)nn4)C[C@@H]3C2)cc1Cl	C42H44ClN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-X07FQN	WO2023222012A1_176	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4C[C@@H]5[C@@H](CN6CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)[C@@H]5C4)cn3)CC2)cc1Cl	C41H41ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-86WV1E	WO2023222012A1_177	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4C[C@@H]5[C@@H](CN6CCN(c7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)[C@@H]5C4)cn3)CC2)cc1Cl	C41H42ClN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-9C0CT5	WO2023222012A1_178	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4C[C@@H]5[C@@H](CN6CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)[C@@H]5C4)nn3)CC2)cc1Cl	C41H41ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-NUDYE0	WO2023222012A1_179	.	CN(CCN(C)c1ccc2c(c1)C(=O)N(C1CCC(=O)NC1=O)C2=O)C[C@@H]1[C@H]2CN(c3ccc(C(=O)N[C@H]4CC[C@H](Oc5ccc(C#N)c(Cl)c5)CC4)nn3)C[C@@H]12	C41H44ClN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-YF4UP8	WO2023222012A1_180	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CC6(CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)C6)C5)CC4)nn3)CC2)cc1Cl	C43H45ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-I6P5UF	WO2023222012A1_181	.	CC1(C)[C@H](NC(=O)c2ccc(N3C[C@@H]4[C@@H](CN5CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)[C@@H]4C3)nn2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C43H45ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-6AEXI1	WO2023222012A1_182	.	CC1(C)[C@H](NC(=O)c2cnc(N3C[C@@H]4[C@@H](CN5CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)[C@@H]4C3)cn2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C43H45ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-EWLHSL	WO2023222012A1_183	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC5(CN(CC6CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)C5)C4)nn3)CC2)cc1Cl	C43H45ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-5TW01X	WO2023222012A1_184	.	Cc1cc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC6(C5)CN(c5cc7c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)nn3)CC2)ccc1C#N	C44H48FN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-DOAJIQ	WO2023222012A1_185	.	Cc1cc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC6(C5)CN(c5ccc7c(c5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)nn3)CC2)ccc1C#N	C44H49N9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-AR6Z18	WO2023222012A1_186	.	Cc1cc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCC(CN5CCC6(C5)CN(c5cc7c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)cn3)CC2)ccc1C#N	C44H48FN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-67T50Q	WO2023222012A1_187	.	Cc1cc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCC(CN5CCC6(C5)CN(c5ccc7c(c5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)cn3)CC2)ccc1C#N	C44H49N9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-J9H7TR	WO2023222012A1_188	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCC(CN5CC6(CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)C6)C5)CC4)cn3)CC2)cc1Cl	C43H45ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-MBSF5Q	WO2023222012A1_189	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCC5(CN(CC6CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)C5)C4)cn3)CC2)CC1Cl	C43H47ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-SZLG2H	WO2023222012A1_190	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC5(CC4)CN(CC4CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC4)C5)nn3)CC2)cc1Cl	C44H48ClN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-QNXXPJ	WO2023222012A1_191	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC6(CC5)CN(c5cc7c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)cc3)CC2)cc1Cl	C46H49ClFN7O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-L7DTNY	WO2023222012A1_192	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC6(CC5)CN(c5ccc7c(c5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)cc3)CC2)cc1Cl	C46H50ClN7O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-C9WH5N	WO2023222012A1_193	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3nnc(N4CC5(CCN(C6CCN(c7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)C4)[nH]3)CC2)cc1Cl	C41H45ClN10O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-XGHMVT	WO2023222012A1_194	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CC5(CCN(CC6CCN(c7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)C4)cc3)CC2)cc1Cl	C46H50ClN7O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-Z259LJ	WO2023222012A1_195	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC6(CC5)CN(c5cc7c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C7)C6)CC4)nn3)CC2)cc1Cl	C44H49ClFN9O5	AR	P10275	CRBN	WO-2023222012-A1
TPD-PMXP4F	WO2023222012A1_196	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC6(CC5)CN(c5ccc7c(c5)CN(C5CCC(=O)NC5=O)C7=O)C6)CC4)nn3)CC2)cc1Cl	C44H50ClN9O5	AR	P10275	CRBN	WO-2023222012-A1
TPD-8N6QHF	WO2023222012A1_197	.	COc1cc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCC(CN5CCC6(CC5)CN(c5ccc7c(c5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)nn3)CC2)ccc1C#N	C44H50N10O7	AR	P10275	CRBN	WO-2023222012-A1
TPD-FAXRO7	WO2023222012A1_199	.	CC(C#Cc1ccc2c(c1)CN([C@H]1C(C)(C)[C@H](Oc3ccc(C#N)c(Cl)c3)C1(C)C)C2=O)N1CCN(c2cc3c(cc2F)C(=O)N(C2CCC(=O)NC2=O)C3=O)CC1	C44H42ClFN6O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-BFQ0OM	WO2023222012A1_200	.	N#Cc1ccc(O[C@H]2CC[C@H](N3Cc4nc(N5CCC(CN6CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)ccc4C3=O)CC2)cc1Cl	C43H44ClFN8O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-K6PJI5	WO2023222012A1_202	.	CC1(C)[C@H](Oc2ccc(C#N)c(Cl)c2)C(C)(C)[C@H]1N1Cc2nc(N3CCC(CN4CCN(c5cc6c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)ccc2C1=O	C45H48ClFN8O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-1Z53IC	WO2023222012A1_203	.	N#Cc1ccc(O[C@H]2CC[C@H](N3Cc4nc(N5CCC(CN6CCN(c7cc8c(cc7F)CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)ccc4C3=O)CC2)cc1Cl	C43H46ClFN8O5	AR	P10275	CRBN	WO-2023222012-A1
TPD-5ZJCZI	WO2023222012A1_204	.	N#Cc1ccc(O[C@H]2CC[C@H](N3Cc4nc(N5CCC(CN6CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8)CC6)CC5)ccc4C3=O)CC2)cc1Cl	C43H46ClFN8O5	AR	P10275	CRBN	WO-2023222012-A1
TPD-3SVBZQ	WO2023222012A1_205	.	CC1(C)[C@H](Oc2ccc(C#N)c(Cl)c2)C(C)(C)[C@H]1N1Cc2nc(N3CCC(CN4CCN(c5cc6c(cc5F)CN(C5CCC(=O)NC5=O)C6=O)CC4)CC3)ccc2C1=O	C45H50ClFN8O5	AR	P10275	CRBN	WO-2023222012-A1
TPD-BO7CBL	WO2023222012A1_206	.	CC1(C)[C@H](Oc2ccc(C#N)c(Cl)c2)C(C)(C)[C@H]1N1Cc2nc(N3CCC(CN4CCN(c5cc6c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C6)CC4)CC3)ccc2C1=O	C45H50ClFN8O5	AR	P10275	CRBN	WO-2023222012-A1
TPD-97AD59	WO2023222012A1_207	.	CC(C)OC(=O)OCN1C(=O)CCC(N2Cc3cc(N4CCN(CC5CCN(c6ccc7c(n6)CN(C6CCC(Oc8ccc(C#N)c(Cl)c8)CC6)C7=O)CC5)CC4)c(F)cc3C2=O)C1=O	C48H54ClFN8O8	AR	P10275	CRBN	WO-2023222012-A1
TPD-6RSV92	WO2023222012A1_208	.	N#Cc1ccc(O[C@H]2CC[C@H](N3Cc4nc(N5CC[C@@H](CN6CCN(c7cc8c(cc7F)CN(C7CCC(=O)NC7=O)C8=O)CC6)C5)ccc4C3=O)CC2)cc1Cl	C42H44ClFN8O5	AR	P10275	CRBN	WO-2023222012-A1
TPD-0ZDN0Q	WO2023222012A1_209	.	N#Cc1ccc(O[C@H]2CC[C@H](N3Cc4nc(N5CC[C@@H](CN6CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8)CC6)C5)ccc4C3=O)CC2)cc1Cl	C42H44ClFN8O5	AR	P10275	CRBN	WO-2023222012-A1
TPD-H5D0IK	WO2023222012A1_210	.	N#Cc1ccc(O[C@H]2CC[C@H](N3Cc4nc(N5CCN(CC6CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)ccc4C3=O)CC2)cc1Cl	C43H44ClFN8O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-VKJ69T	WO2023222012A1_211	.	N#Cc1ccc(O[C@H]2CC[C@H](N3Cc4nc(N5CCN(CC6CCN(c7cc8c(cc7F)CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)ccc4C3=O)CC2)cc1Cl	C43H46ClFN8O5	AR	P10275	CRBN	WO-2023222012-A1
TPD-LUX9WQ	WO2023222012A1_212	.	N#Cc1ccc(O[C@H]2CC[C@H](N3Cc4nc(N5CCN(CC6CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8)CC6)CC5)ccc4C3=O)CC2)cc1Cl	C43H46ClFN8O5	AR	P10275	CRBN	WO-2023222012-A1
TPD-2V79SF	WO2023222012A1_213	.	CC1(C)[C@H](NC(=O)c2ccc(N3CCC(CN4CCN(c5cc6c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C6)CC4)CC3)nc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C44H50ClFN8O5	AR	P10275	CRBN	WO-2023222012-A1
TPD-5H2Z0F	WO2023222012A1_214	.	CC1(C)[C@H](NC(=O)c2ccc(N3CCC(CN4CCN(c5cc6c(cc5F)CN(C5CCC(=O)NC5=O)C6=O)CC4)CC3)nc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C44H50ClFN8O5	AR	P10275	CRBN	WO-2023222012-A1
TPD-CSC7EY	WO2023222012A1_215	.	CC(C)(C)N(C(=O)c1ccc(N2CCC(CN3CCN(c4cc5c(cc4F)CN(C4CCC(=O)NC4=O)C5=O)CC3)CC2)nc1)[C@H]1C(C)(C)[C@H](Oc2ccc(C#N)c(Cl)c2)C1(C)C	C48H58ClFN8O5	AR	P10275	CRBN	WO-2023222012-A1
TPD-W8F3GW	WO2023222012A1_216	.	CC(C)(C)N(C(=O)c1ccc(N2CCC(CN3CCN(c4cc5c(cc4F)C(=O)N(C4CCC(=O)NC4=O)C5)CC3)CC2)nc1)[C@H]1C(C)(C)[C@H](Oc2ccc(C#N)c(Cl)c2)C1(C)C	C48H58ClFN8O5	AR	P10275	CRBN	WO-2023222012-A1
TPD-788YRI	WO2023222012A1_217	.	N#Cc1ccc(O[C@H]2CC[C@H](N3Cc4nc(N5CCC(CN6CCN(c7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)ccc4C3=O)CC2)cc1Cl	C43H45ClN8O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-DXPJEE	WO2023222012A1_218	.	N#Cc1ccc(O[C@@H]2C[C@@H]3CN(C(=O)c4ccc(N5CCC(CN6CCN(c7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)nn4)C[C@@H]3C2)cc1Cl	C42H44ClN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-3UW660	WO2023222012A1_219	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)C3=CCC(N4CCC(NC5CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)C=C3)CC2)cc1Cl	C43H47ClFN7O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-8DZTJ7	WO2023222012A1_220	.	N#Cc1ccc(O[C@H]2CC[C@@H](NC(=O)c3cnc(N4C[C@@H]5CN(C6CCN(c7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)C[C@@H]5C4)nc3)CC2)cc1Cl	C42H44ClN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-89LLPI	WO2023222012A1_221	.	CC1(C)[C@H](NC(=O)c2ccc(N3CCC(N4C[C@H]5CN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)C[C@H]5C4)CC3)nn2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C44H47ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-PV52K6	WO2023222012A1_222	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4C[C@H]5C[C@@H](CN6CC7CN(C8=CC9C(=O)N(C%10CCC(=O)NC%10=O)C(=O)C9C=C8F)CC7C6)C[C@H]5C4)nn3)CC2)cc1Cl	C45H49ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-E9QLSG	WO2023222012A1_223	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CC(N5CC6CN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6C5)C4)nn3)CC2)cc1Cl	C40H39ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-1ZSJO6	WO2023222012A1_224	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4C[C@H]5C[C@@H](CN6CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)C[C@H]5C4)nn3)CC2)cc1Cl	C43H45ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-JQWJTT	WO2023222012A1_225	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CC(N5CC6CN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6C5)C4)cn3)CC2)cc1Cl	C40H39ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-LK1MF3	WO2023222012A1_226	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCN(C[C@@H]5C[C@@H]6CN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)C[C@@H]6C5)CC4)nn3)CC2)cc1Cl	C43H45ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-QPPZWD	WO2023222012A1_227	.	N#Cc1ccc(Oc2ccc(NC(=O)c3ccc(N4CCC(CN5CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)nn3)cc2)cc1Cl	C41H37ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-WNG6TV	WO2023222012A1_228	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCC(N5CC6(CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)C5)CC4)cn3)CC2)cc1Cl	C43H45ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-0GK6P8	WO2023222012A1_229	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCC(N5CC6(CCN(c7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)C5)CC4)cn3)CC2)cc1Cl	C43H46ClN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-J8749V	WO2023222012A1_230	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC6(CC5)CN(c5ccc7c(c5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)nn3)CC2)cc1Cl	C44H48ClN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-K04XE7	WO2023222012A1_231	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC6(CC5)CN(c5cc7c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)nn3)CC2)cc1Cl	C44H47ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-1T6SX1	WO2023222012A1_232	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CC5(CCN(CC6CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)C4)nn3)CC2)cc1Cl	C44H47ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-2WV0JA	WO2023222012A1_233	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCC(CN5CCC6(CC5)CN(c5cc7c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)cn3)CC2)cc1Cl	C44H47ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-5O7R69	WO2023222012A1_234	.	Cc1cc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCC(CN5CC6(CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)C5)CC4)cn3)CC2)ccc1C#N	C45H50FN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-FVEH69	WO2023222012A1_235	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CC5(CCN(CC6CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)C4)cn3)CC2)cc1Cl	C44H47ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-V9QW6M	WO2023222012A1_236	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCC(N5CC6(CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)C5)CC4)cn3)CC2)cc1C(F)(F)F	C44H45F4N9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-AKW8TW	WO2023222012A1_237	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CC5CC4CN5C[C@H]4[C@@H]5CN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)C[C@@H]54)nn3)CC2)cc1Cl	C42H41ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-EF3S13	WO2023222012A1_238	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CC5CC4CN5C[C@H]4[C@@H]5CN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)C[C@@H]54)cn3)CC2)cc1Cl	C42H41ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-1F8KZI	WO2023222012A1_239	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4C[C@H]5CC[C@@H](C4)N5CC[C@H]4CCN(c5cc6c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)nn3)CC2)cc1Cl	C43H45ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-A26RJ9	WO2023222012A1_240	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4C[C@H]5CC[C@@H](C4)N5CC[C@H]4CCN(c5cc6c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)cn3)CC2)cc1Cl	C43H45ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-EX6TJE	WO2023222012A1_241	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCC(CN5CCC6(CC5)CN(C5=CC7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7C=C5)C6)CC4)cn3)CC2)cc1Cl	C44H50ClN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-8OF5G4	WO2023222012A1_242	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CC5(CCN(C6CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)C4)cn3)CC2)cc1Cl	C43H45ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-N97NVR	WO2023222012A1_243	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3nnc(N4CCC(CN5CCC6(CC5)CN(c5ccc7c(c5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)s3)CC2)cc1Cl	C42H46ClN9O6S	AR	P10275	CRBN	WO-2023222012-A1
TPD-2UD7WK	WO2023222012A1_244	.	Cc1cc2c(cc1N1CC3(CCN(CC4CCN(c5nnc(C(=O)N[C@H]6CC[C@H](Oc7ccc(C#N)c(Cl)c7)CC6)s5)CC4)CC3)C1)C(=O)N(C1CCC(=O)NC1=O)C2=O	C43H48ClN9O6S	AR	P10275	CRBN	WO-2023222012-A1
TPD-FDX0SL	WO2023222012A1_245	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnn([C@H]4CC[C@H](CN5CCC6(CC5)CN(c5ccc7c(c5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)c3)CC2)cc1Cl	C44H49ClN8O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-9I89OL	WO2023222012A1_246	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnn([C@H]4CC[C@H](CN5CCC6(CC5)CN(c5cc7c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)c3)CC2)cc1Cl	C44H48ClFN8O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-WIOH22	WO2023222012A1_247	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC6(CC5)CN(c5ccc7c(=O)n(C8CCC(=O)NC8=O)cnc7c5)C6)CC4)nn3)CC2)cc1Cl	C44H49ClN10O5	AR	P10275	CRBN	WO-2023222012-A1
TPD-WIQHC7	WO2023222012A1_248	.	CC1(C)[C@H](Oc2ccc(C#N)c(Cl)c2)C(C)(C)[C@H]1N1Cc2cc(N3CCC(CN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)CC3)ccc2C1=O	C46H52ClN7O5	AR	P10275	CRBN	WO-2023222012-A1
TPD-RI4WRC	WO2023222012A1_249	.	CC1(C)[C@H](Oc2ccc(C#N)c(Cl)c2)C(C)(C)[C@H]1N1Cc2cc(N3CCC(CN4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)ccc2C1=O	C46H50ClN7O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-ZMUAOT	WO2023222012A1_250	.	CC1(C)[C@H](Oc2ccc(C#N)c(Cl)c2)C(C)(C)[C@H]1N1Cc2cc(N3CCC(CN4CCN(c5cc6c(cc5F)CN(C5CCC(=O)NC5=O)C6=O)CC4)CC3)ccc2C1=O	C46H51ClFN7O5	AR	P10275	CRBN	WO-2023222012-A1
TPD-OEY4GR	WO2023222012A1_251	.	CC1(C)[C@H](Oc2ccc(C#N)c(Cl)c2)C(C)(C)[C@H]1N1Cc2cc(N3CCC(CN4CCN(c5cc6c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C6)CC4)CC3)ccc2C1=O	C46H51ClFN7O5	AR	P10275	CRBN	WO-2023222012-A1
TPD-W2R6QW	WO2023222012A1_252	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CC6CN(c7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6C5)CC4)nn3)CC2)cc1Cl	C43H46ClN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-9ZOPO8	WO2023222012A1_253	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CC6CN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6C5)CC4)nn3)CC2)cc1Cl	C43H45ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-Q1ET53	WO2023222012A1_254	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCC(CN5CC6CN(c7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6C5)CC4)cn3)CC2)cc1Cl	C43H46ClN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-5QD6I8	WO2023222012A1_255	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCC(CN5CC6CN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6C5)CC4)cn3)CC2)cc1Cl	C43H45ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-2F4LLC	WO2023222012A1_257	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCC(CN5CC6CN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6C5)CC4)nc3)CC2)cc1Cl	C43H45ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-5ORZ4M	WO2023222012A1_258	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCC(CN5CC6CN(c7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6C5)CC4)nc3)CC2)cc1Cl	C43H46ClN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-05GX7I	WO2023222012A1_259	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CC5CN(CC6CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5C4)nn3)CC2)cc1Cl	C43H45ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-TVRVQK	WO2023222012A1_260	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CC5CN(CC6CCN(c7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5C4)nn3)CC2)cc1Cl	C43H46ClN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-2451LE	WO2023222012A1_262	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)C3C=CC(N4CCC5(CCN(CC6CCN(c7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)CC4)N=N3)CC2)cc1Cl	C46H54ClN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-ULRWMN	WO2023222012A1_263	.	C[C@@H]1CN(C[C@@H]2[C@H]3CN(c4cc5c(cc4F)C(=O)N(C4CCC(=O)NC4=O)C5=O)C[C@@H]23)CCN1c1ccc(C(=O)N[C@H]2CC[C@H](Oc3ccc(C#N)c(Cl)c3)CC2)nn1	C42H43ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-DBR9MD	WO2023222012A1_264	.	C[C@@H]1CN(C[C@@H]2[C@H]3CN(c4cc5c(cc4F)C(=O)N(C4CCC(=O)NC4=O)C5=O)C[C@@H]23)CCN1c1cnc(C(=O)N[C@H]2CC[C@H](Oc3ccc(C#N)c(Cl)c3)CC2)cn1	C42H43ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-RPXP9U	WO2023222012A1_265	.	C[C@@H]1CN(c2ccc(C(=O)N[C@H]3CC[C@H](Oc4ccc(C#N)c(Cl)c4)CC3)nn2)CCN1C[C@H]1[C@@H]2CN(c3cc4c(cc3F)C(=O)N(C3CCC(=O)NC3=O)C4=O)C[C@@H]21	C42H43ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-J3GTS4	WO2023222012A1_266	.	C[C@@H]1CN(c2cnc(C(=O)N[C@H]3CC[C@H](Oc4ccc(C#N)c(Cl)c4)CC3)cn2)CCN1C[C@H]1[C@@H]2CN(c3cc4c(cc3F)C(=O)N(C3CCC(=O)NC3=O)C4=O)C[C@@H]21	C42H43ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-JV1VCA	WO2023222012A1_267	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCC(CN5CCC6(CC5)CN(c5ccc7c(c5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)nc3)CC2)cc1Cl	C44H48ClN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-041F7M	WO2023222012A1_268	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCC(CN5CCC6(CC5)CN(c5cc7c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)nc3)CC2)cc1Cl	C44H47ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-2QQS0U	WO2023222012A1_269	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC5(CC4)CC(N4CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC4)C5)nn3)CC2)cc1Cl	C43H45ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-RKUFZQ	WO2023222012A1_270	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCN(C5CC6(CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)C5)CC4)nn3)CC2)cc1Cl	C43H45ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-G8RQUC	WO2023222012A1_271	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCN(C5CC6(CCN(c7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)C5)CC4)nn3)CC2)cc1Cl	C43H46ClN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-IIKPKG	WO2023222012A1_272	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CC5CN(CC6CCN(C7C=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=CC7F)CC6)CC5C4)nc3)CC2)cc1Cl	C43H47ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-PW35EW	WO2023222012A1_273	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CC5(CCN(C6CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)C4)nc3)CC2)cc1Cl	C43H45ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-ZN8MVA	WO2023222012A1_274	.	C=Nc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC6(CC5)CN(c5ccc7c(c5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)nn3)CC2)cc1Br	C44H50BrN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-VZB31E	WO2023222012A1_275	.	C=Nc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC6(CC5)CN(c5ccc7c(c5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)nn3)CC2)cc1C	C45H53N9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-UKAEU2	WO2023222012A1_276	.	C=Nc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC6(CC5)CN(c5ccc7c(c5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)nn3)CC2)cc1OC	C45H53N9O7	AR	P10275	CRBN	WO-2023222012-A1
TPD-PVCFM5	WO2023222012A1_277	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCN(C5CC6(CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)C5)CC4)cn3)CC2)cc1Cl	C43H45ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-XM6BNO	WO2023222012A1_278	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCN(C5CC6(CCN(c7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)C5)CC4)cn3)CC2)cc1Cl	C43H46ClN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-NJDTCA	WO2023222012A1_280	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCC(N5CCC6(CC5)CN(c5ccc7c(c5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)cn3)CC2)cc1Cl	C43H46ClN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-7RI6OZ	WO2023222012A1_281	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(N5CCC6(CC5)CN(c5ccc7c(c5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)nn3)CC2)cc1Cl	C43H46ClN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-H5F9QZ	WO2023222012A1_282	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CC5(CCN(CC6CCN(c7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)C4)nn3)CC2)cc1Cl	C44H48ClN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-49Q2FX	WO2023222012A1_283	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CC5(CCN(CC6CCN(c7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)C4)cn3)CC2)cc1Cl	C44H48ClN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-OQ382N	WO2023222012A1_285	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCN(CC5CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)nn3)CC2)cc1C(F)(F)F	C42H43F4N9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-GXONXN	WO2023222012A1_286	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCN(C[C@@H]5[C@H]6CN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)C[C@@H]56)CC4)cn3)CC2)cc1Cl	C42H42ClFN8O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-1F3SIK	WO2023222012A1_287	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCC(N5CCC6(CC5)CN(c5cc7c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)cn3)CC2)cc1Cl	C43H45ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-ALAV0I	WO2023222012A1_289	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCC5(CC4)CN(C4CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC4)C5)cn3)CC2)cc1Cl	C43H45ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-GMOJV5	WO2023222012A1_290	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCN(C(=O)O[C@H]5C[C@@H]6CN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)C[C@@H]6C5)CC4)nn3)CC2)cc1Cl	C43H43ClFN9O8	AR	P10275	CRBN	WO-2023222012-A1
TPD-651NJ3	WO2023222012A1_291	.	CC1(C)[C@H](NC(=O)c2ccc(N3CCC(NC4CCN(c5cc6c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)nn2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C43H47ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-ZT098Q	WO2023222012A1_293	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4C[C@H]5C[C@@H](N6CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)C[C@H]5C4)nn3)CC2)cc1Cl	C42H43ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-15JPCR	WO2023222012A1_294	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4C[C@H]5C[C@@H](N6CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)C[C@H]5C4)nc3)CC2)cc1Cl	C42H43ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-JGGWZ8	WO2023222012A1_295	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCN([C@@H]5C[C@@H]6CN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)C[C@@H]6C5)CC4)cn3)CC2)cc1Cl	C42H43ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-XX3G2R	WO2023222012A1_296	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCN([C@@H]5C[C@@H]6CN(c7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)C[C@@H]6C5)CC4)cn3)CC2)cc1Cl	C42H44ClN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-JXB1RS	WO2023222012A1_297	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCN([C@@H]5C[C@@H]6CN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)C[C@@H]6C5)CC4)nn3)CC2)cc1Cl	C42H43ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-GSOD7G	WO2023222012A1_298	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCN([C@@H]5C[C@@H]6CN(c7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)C[C@@H]6C5)CC4)nn3)CC2)cc1Cl	C42H44ClN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-CH1T67	WO2023222012A1_299	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCN([C@@H]5C[C@@H]6CN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)C[C@@H]6C5)CC4)nc3)CC2)cc1Cl	C42H43ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-8D0JUV	WO2023222012A1_300	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCN([C@@H]5C[C@@H]6CN(c7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)C[C@@H]6C5)CC4)nc3)CC2)cc1Cl	C42H44ClN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-SX7SBS	WO2023222012A1_301	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCN(C(=O)O[C@H]5C[C@@H]6CN(c7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)C[C@@H]6C5)CC4)cn3)CC2)cc1Cl	C43H44ClN9O8	AR	P10275	CRBN	WO-2023222012-A1
TPD-LXKDST	WO2023222012A1_302	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(NC5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3)CC2)cc1Cl	C43H46ClN7O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-R4OTMO	WO2023222012A1_303	.	N#Cc1ccc(O[C@H]2C[C@H]3C[C@@H](NC(=O)c4cnc(N5CCC(CN6CCN(c7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)cn4)C[C@H]3C2)cc1Cl	C43H46ClN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-QR03EB	WO2023222012A1_304	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(OC5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3)CC2)cc1Cl	C43H45ClN6O7	AR	P10275	CRBN	WO-2023222012-A1
TPD-3WIG56	WO2023222012A1_305	.	CN(C(=O)c1ccc(N2CCC(CN3CCN(c4cc5c(cc4F)C(=O)N(C4CCC(=O)NC4=O)C5)CC3)CC2)nc1)[C@H]1CC[C@H](Oc2ccc(C#N)c(Cl)c2)CC1	C43H48ClFN8O5	AR	P10275	CRBN	WO-2023222012-A1
TPD-K2BYJQ	WO2023222012A1_306	.	CN(C(=O)c1ccc(N2CCC(CN3CCN(c4cc5c(cc4F)CN(C4CCC(=O)NC4=O)C5=O)CC3)CC2)nc1)[C@H]1CC[C@H](Oc2ccc(C#N)c(Cl)c2)CC1	C43H48ClFN8O5	AR	P10275	CRBN	WO-2023222012-A1
TPD-F0DTUY	WO2023222012A1_307	.	CN1C(=O)CCC(N2Cc3cc(F)c(N4CCN(CC5CCN(c6ccc7c(n6)CN([C@H]6CC[C@H](Oc8ccc(C#N)c(Cl)c8)CC6)C7=O)CC5)CC4)cc3C2=O)C1=O	C44H48ClFN8O5	AR	P10275	CRBN	WO-2023222012-A1
TPD-STE7RU	WO2023222012A1_308	.	COCCOCCOCCOCCOC(=O)OCN1C(=O)CCC(N2Cc3cc(N4CCN(CC5CCN(c6ccc7c(n6)CN([C@H]6CC[C@H](Oc8ccc(C#N)c(Cl)c8)CC6)C7=O)CC5)CC4)c(F)cc3C2=O)C1=O	C54H66ClFN8O12	AR	P10275	CRBN	WO-2023222012-A1
TPD-NXBTW6	WO2023222012A1_309	.	CC1=NC2C=C(N3CCN(CC4CCN(c5ccc6c(n5)CN([C@H]5CC[C@H](Oc7ccc(C#N)c(Cl)c7)CC5)C6=O)CC4)CC3)C=CC2C(=O)N1C1CCC(=O)NC1=O	C44H50ClN9O5	AR	P10275	CRBN	WO-2023222012-A1
TPD-3696YR	WO2023222012A1_310	.	CC1(C)[C@H](Oc2ccc(C#N)c(Cl)c2)C(C)(C)[C@H]1N1Cc2cc(C#Cc3cnn(C4CN(c5cc6c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)c3)ccc2C1=O	C44H37ClFN7O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-0BWOCJ	WO2023222012A1_311	.	N#Cc1ccc(O[C@H]2CC[C@H](N3Cc4cc(N5CCC(CN6CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)ncc4C3=O)CC2)cc1Cl	C43H44ClFN8O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-0OH31C	WO2023222012A1_312	.	N#Cc1ccc(O[C@H]2CC[C@H](N3Cc4cc(N5CCC(CN6CCN(c7ccc8c(c7)CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)ncc4C3=O)CC2)cc1Cl	C43H47ClN8O5	AR	P10275	CRBN	WO-2023222012-A1
TPD-RZHR9W	WO2023222012A1_313	.	N#Cc1ccc(O[C@H]2CC[C@H](N3Cc4cc(N5CCC(CN6CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8)CC6)CC5)ncc4C3=O)CC2)cc1Cl	C43H46ClFN8O5	AR	P10275	CRBN	WO-2023222012-A1
TPD-WLVPKN	WO2023222012A1_314	.	N#Cc1ccc(O[C@H]2CC[C@H](N3Cc4cc(N5CCC(CN6CCN(c7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)ncc4C3=O)CC2)cc1Cl	C43H45ClN8O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-Q3EI43	WO2023222012A1_315	.	CC1(C)[C@H](Oc2ccc(C#N)c(Cl)c2)C(C)(C)[C@H]1N1Cc2nc(C#CC3CCN(C4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)ccc2C1=O	C47H48ClN7O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-EGZPFV	WO2023222012A1_316	.	CC1(C)[C@H](Oc2ccc(C#N)c(Cl)c2)C(C)(C)[C@H]1N1Cc2nc(C#CC3CCN(C4CCN(c5cc6c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)ccc2C1=O	C47H47ClFN7O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-Y796RG	WO2023222012A1_317	.	CC1(C)[C@H](Oc2ccc(N=O)c(Cl)c2)C(C)(C)[C@H]1N1Cc2nc(C#CC3CCN(C4CN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)CC3)ccc2C1=O	C44H44ClN7O7	AR	P10275	CRBN	WO-2023222012-A1
TPD-TQDX25	WO2023222012A1_318	.	CC1(C)[C@H](Oc2ccc(N=O)c(Cl)c2)C(C)(C)[C@H]1N1Cc2nc(C#CC3CCN(C4CN(c5cc6c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)CC3)ccc2C1=O	C44H43ClFN7O7	AR	P10275	CRBN	WO-2023222012-A1
TPD-2MOQLP	WO2023222012A1_319	.	CC1(C)[C@H](Oc2ccc(C#N)c(Cl)c2)C(C)(C)[C@H]1N1Cc2nc(C#CC3CN(C4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C3)ccc2C1=O	C45H44ClN7O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-LQ9VO8	WO2023222012A1_320	.	CC1(C)[C@H](Oc2ccc(C#N)c(Cl)c2)C(C)(C)[C@H]1N1Cc2nc(C#CC3CN(C4CCN(c5cc6c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C3)ccc2C1=O	C45H43ClFN7O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-J52K8P	WO2023222012A1_322	.	CC1(C)[C@H](Oc2ccc(C#N)c(Cl)c2)C(C)(C)[C@H]1N1Cc2nc(C#CC3CN(C4CN(c5cc6c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)C3)ccc2C1=O	C43H39ClFN7O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-AE1NZK	WO2023222012A1_323	.	N#Cc1ccc(O[C@H]2CC[C@H](N3Cc4nc(C#CC5CCN(C6CCN(c7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)ccc4C3=O)CC2)cc1Cl	C45H44ClN7O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-GN0VCV	WO2023222012A1_324	.	N#Cc1ccc(O[C@H]2CC[C@H](N3Cc4nc(C#CC5CCN(C6CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)ccc4C3=O)CC2)cc1Cl	C45H43ClFN7O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-WXUZC4	WO2023222012A1_326	.	CC1(C)[C@H](Oc2ccc(C#N)c(Cl)c2)C(C)(C)[C@H]1N1Cc2nc(C#C[C@H]3CC[C@H](N4CCN(c5cc6c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)ccc2C1=O	C47H47ClFN7O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-8BUTBR	WO2023222012A1_328	.	CC1(C)[C@H](Oc2ccc(C#N)c(Cl)c2)C(C)(C)[C@H]1N1Cc2nc(C#CC3CC(NC4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C3)ccc2C1=O	C46H46ClN7O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-4DSWSN	WO2023222012A1_330	.	CC1(C)[C@H](Oc2ccc(C#N)c(Cl)c2)C(C)(C)[C@H]1N1Cc2nc(C#CC3CC(NC4CCN(c5cc6c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C3)ccc2C1=O	C46H45ClFN7O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-939VPQ	WO2023222012A1_331	.	CN(C1CCN(c2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)CC1)C1CC(C#Cc2ccc3c(n2)CN([C@H]2C(C)(C)[C@H](Oc4ccc(C#N)c(Cl)c4)C2(C)C)C3=O)C1	C47H48ClN7O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-421CTD	WO2023222012A1_332	.	CN(C1CCN(c2cc3c(cc2F)C(=O)N(C2CCC(=O)NC2=O)C3=O)CC1)C1CC(C#Cc2ccc3c(n2)CN([C@H]2C(C)(C)[C@H](Oc4ccc(C#N)c(Cl)c4)C2(C)C)C3=O)C1	C47H47ClFN7O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-HLM2EU	WO2023222012A1_333	.	CC1(C)[C@H](OC2=CCC(C#N)C(Cl)=C2)C(C)(C)[C@H]1N1Cc2nc(C#CC3CCN(CC4CCN(c5cc6c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)ccc2C1=O	C48H51ClFN7O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-ULCFJB	WO2023222012A1_334	.	CC1(C)[C@H](Oc2ccc(C#N)c(Cl)c2)C(C)(C)[C@H]1N1Cc2nc(C#CC3CCN(CC4CN(c5cc6c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)CC3)ccc2C1=O	C46H45ClFN7O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-O4504K	WO2023222012A1_335	.	Cc1cc(O[C@H]2C(C)(C)[C@H](N3Cc4nc(C#CC5CN(CC6CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)C5)ccc4C3=O)C2(C)C)ccc1C#N	C47H48FN7O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-BNU1LM	WO2023222012A1_336	.	CC(C)(C#Cc1ccc2c(n1)CN([C@H]1C(C)(C)[C@H](Oc3ccc(C#N)c(Cl)c3)C1(C)C)C2=O)N1CCN(c2cc3c(cc2F)C(=O)N(C2CCC(=O)NC2=O)C3=O)CC1	C44H43ClFN7O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-SVUTU7	WO2023222012A1_338	.	CC(C)(C#Cc1ccc2c(n1)CN([C@H]1C(C)(C)[C@H](Oc3ccc(C#N)c(Cl)c3)C1(C)C)C2=O)NC1CCN(c2cc3c(cc2F)C(=O)N(C2CCC(=O)NC2=O)C3=O)CC1	C45H45ClFN7O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-E3KKBN	WO2023222012A1_340	.	CC1(C)[C@H](Oc2ccc(C#N)c(Cl)c2)C(C)(C)[C@H]1N1Cc2nc(C#CC3CCC(N4CC5CN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5C4)CC3)ccc2C1=O	C49H49ClFN7O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-VEOJVP	WO2023222012A1_342	.	CC1(C)[C@H](Oc2ccc(C#N)c(Cl)c2)C(C)(C)[C@H]1N1Cc2nc(C#CC3CCC(N4CC5(CN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)C4)CC3)ccc2C1=O	C48H47ClFN7O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-YTDVJ1	WO2023222012A1_344	.	CC1(C)[C@H](Oc2ccc(C#N)c(Cl)c2)C(C)(C)[C@H]1N1Cc2nc(C#CC3CCC(N4CC5CC4CN5c4cc5c(cc4F)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)ccc2C1=O	C48H47ClFN7O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-WM0LKC	WO2023222012A1_345	.	CC1(C)[C@H](Oc2ccc(C#N)c(Cl)c2)C(C)(C)[C@H]1N1Cc2nc(C#CC3CCN(CC4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)ccc2C1=O	C48H50ClN7O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-6AKE9K	WO2023222012A1_346	.	CC1(C)[C@H](Oc2ccc(C#N)c(Cl)c2)C(C)(C)[C@H]1N1Cc2nc(C#CC3CCN(CC4CN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)CC3)ccc2C1=O	C46H46ClN7O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-X9Q2NB	WO2023222012A1_347	.	CC1(C)[C@H](Oc2ccc(C#N)c(Cl)c2)C(C)(C)[C@H]1N1Cc2nc(C#CC3CN(CC4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C3)ccc2C1=O	C46H46ClN7O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-B06P85	WO2023222012A1_349	.	CC1(C)[C@H](Oc2ccc(C#N)c(Cl)c2)C(C)(C)[C@H]1N1Cc2nc(C#CC3CCC(N4CC5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5C4)CC3)ccc2C1=O	C49H50ClN7O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-P8CZRQ	WO2023222012A1_351	.	CC1(C)[C@H](Oc2ccc(C#N)c(Cl)c2)C(C)(C)[C@H]1N1Cc2nc(C#CC3CCC(N4CC5(CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)C4)CC3)ccc2C1=O	C48H48ClN7O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-WAU8HH	WO2023222012A1_353	.	CC1(C)[C@H](Oc2ccc(C#N)c(Cl)c2)C(C)(C)[C@H]1N1Cc2nc(C#CC3CCC(N4CC5CC4CN5c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)ccc2C1=O	C48H48ClN7O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-13IK4R	WO2023222012A1_354	.	CC1(C)[C@H](Oc2ccc(C#N)c(Cl)c2)C(C)(C)[C@H]1N1Cc2nc(C#C[C@H]3C[C@@H](N4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C3)ccc2C1=O	C45H44ClN7O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-G11C9C	WO2023222012A1_355	.	CC1(C)[C@H](Oc2ccc(C#N)c(Cl)c2)C(C)(C)[C@H]1N1Cc2nc(C#C[C@H]3C[C@H](N4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C3)ccc2C1=O	C45H44ClN7O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-GVZCEV	WO2023222012A1_356	.	CC1(C)[C@H](Oc2ccc(C#N)c(Cl)c2)C(C)(C)[C@H]1N1Cc2nc(C#C[C@H]3C[C@@H](N4CCN(c5cc6c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C3)ccc2C1=O	C45H43ClFN7O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-A5GUOU	WO2023222012A1_357	.	CC1(C)[C@H](Oc2ccc(C#N)c(Cl)c2)C(C)(C)[C@H]1N1Cc2nc(C#C[C@H]3C[C@H](N4CCN(c5cc6c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C3)ccc2C1=O	C45H43ClFN7O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-GR3T24	WO2023222012A1_359	.	CC1(C)[C@H](Oc2ccc(C#N)c(Cl)c2)C(C)(C)[C@H]1N1Cc2nc(C#CC3CC(N4CC5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5C4)C3)ccc2C1=O	C47H46ClN7O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-K2RRT1	WO2023222012A1_361	.	CC1(C)[C@H](Oc2ccc(C#N)c(Cl)c2)C(C)(C)[C@H]1N1Cc2nc(C#CC3CC(N4CC5CN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5C4)C3)ccc2C1=O	C47H45ClFN7O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-P7J70C	WO2023222012A1_362	.	CC1(C)[C@H](Oc2ccc(C#N)c(Cl)c2)C(C)(C)[C@H]1N1Cc2nc(C#CC3CCC(N4CCC5(CC4)CN(c4ccc6c(c4)C(=O)N(C4CCC(=O)NC4=O)C6=O)C5)CC3)ccc2C1=O	C50H52ClN7O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-6JILI5	WO2023222012A1_363	.	CC1(C)[C@H](Oc2ccc(C#N)c(Cl)c2)C(C)(C)[C@H]1N1Cc2nc(C#CC3CCC(N4CCC5(CC4)CN(c4cc6c(cc4F)C(=O)N(C4CCC(=O)NC4=O)C6=O)C5)CC3)ccc2C1=O	C50H51ClFN7O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-7K3Q6U	WO2023222012A1_365	.	CC1(C)[C@H](Oc2ccc(C#N)c(Cl)c2)C(C)(C)[C@H]1N1Cc2nc(C#CC3CCC(N4CCC5(CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)C4)CC3)ccc2C1=O	C50H52ClN7O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-ELBE1Q	WO2023222012A1_367	.	CC1(C)[C@H](Oc2ccc(C#N)c(Cl)c2)C(C)(C)[C@H]1N1Cc2nc(C#CC3CCC(N4CCC5(CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)C4)CC3)ccc2C1=O	C50H51ClFN7O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-LO8BIP	WO2023222012A1_369	.	CC1(C)[C@H](Oc2ccc(C#N)c(Cl)c2)C(C)(C)[C@H]1N1Cc2nc(C#CC3CCC(N4CC5(CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)C4)CC3)ccc2C1=O	C49H50ClN7O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-HOW4KY	WO2023222012A1_371	.	CC1(C)[C@H](Oc2ccc(C#N)c(Cl)c2)C(C)(C)[C@H]1N1Cc2nc(C#CC3CCC(N4CC5(CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)C4)CC3)ccc2C1=O	C49H49ClFN7O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-RYAZXK	WO2023222012A1_373	.	CC1(C)[C@H](Oc2ccc(C#N)c(Cl)c2)C(C)(C)[C@H]1N1Cc2nc(C#CC3CCC(N4CCC5(CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)C4)CC3)ccc2C1=O	C49H50ClN7O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-TCT9XF	WO2023222012A1_375	.	CC1(C)[C@H](Oc2ccc(C#N)c(Cl)c2)C(C)(C)[C@H]1N1Cc2nc(C#CC3CCC(N4CCC5(CN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)C4)CC3)ccc2C1=O	C49H49ClFN7O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-T4PMDY	WO2023222012A1_377	.	CC1(C)C(Oc2ccc(C#N)c(Cl)c2)C(C)(C)C1N1Cc2nc(C#CC3CCC(N4CC5(CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)CC3)ccc2C1=O	C50H52ClN7O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-AFLPL6	WO2023222012A1_379	.	CC1(C)C(Oc2ccc(C#N)c(Cl)c2)C(C)(C)C1N1Cc2nc(C#CC3CCC(N4CC5(CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)CC3)ccc2C1=O	C50H51ClFN7O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-1SIH8Q	WO2023222012A1_380	.	CC1(C)[C@H](Oc2ccc(C#N)c(Cl)c2)C(C)(C)[C@H]1N1Cc2nc(C#C[C@H]3CC[C@H](N4CCN(c5cc6c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)cnc2C1=O	C46H46ClFN8O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-1IM09Z	WO2023222012A1_381	.	CC1(C)[C@H](Oc2ccc(C#N)c(Cl)c2)C(C)(C)[C@H]1N1Cc2nc(C#C[C@H]3CC[C@H](N4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)cnc2C1=O	C46H47ClN8O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-14ANO9	WO2023222012A1_382	.	CC1(C)[C@H](Oc2ccc(C#N)c(Cl)c2)C(C)(C)[C@H]1N1Cc2nc(N3CCC(CN4CCN(c5cc6c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)ncc2C1=O	C44H47ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-1GOEZI	WO2023222012A1_383	.	CC1(C)[C@H](Oc2ccc(C#N)c(Cl)c2)C(C)(C)[C@H]1N1Cc2nc(N3CCC(CN4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)ncc2C1=O	C44H48ClN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-WMULL3	WO2023222012A1_384	.	CC1(C)[C@H](Oc2ccc(C#N)c(Cl)c2)C(C)(C)[C@H]1N1Cc2nc(N3CCC(CN4CCN(c5cc6c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)cnc2C1=O	C44H47ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-P3PJ2K	WO2023222012A1_385	.	CC1(C)[C@H](Oc2ccc(C#N)c(Cl)c2)C(C)(C)[C@H]1N1Cc2nc(N3CCC(CN4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)cnc2C1=O	C44H48ClN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-NMNNM6	WO2023222012A1_387	.	CC1(C)[C@H](Oc2ccc(C#N)c(Cl)c2)C(C)(C)[C@H]1N1Cc2nc(C#CC3CCC(N4CC5CC4CN5c4cc5c(cc4F)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)cnc2C1=O	C47H46ClFN8O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-RV80FN	WO2023222012A1_389	.	CC1(C)[C@H](Oc2ccc(C#N)c(Cl)c2)C(C)(C)[C@H]1N1Cc2nc(C#CC3CCC(N4CC5CC4CN5c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)cnc2C1=O	C47H47ClN8O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-3FREBM	WO2023222012A1_390	.	CC(=O)c1cc(N2CCN([C@H]3C[C@H](C#Cc4cnc5c(n4)CN([C@H]4C(C)(C)[C@H](Oc6ccc(C#N)c(Cl)c6)C4(C)C)C5=O)C3)CC2)ccc1C(=O)NC1CCC(=O)NC1=O	C45H47ClN8O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-Q31BBZ	WO2023222012A1_391	.	CC(=O)c1cc(N2CCN([C@H]3C[C@H](C#Cc4cnc5c(n4)CN([C@H]4C(C)(C)[C@H](Oc6ccc(C#N)c(Cl)c6)C4(C)C)C5=O)C3)CC2)c(F)cc1C(=O)NC1CCC(=O)NC1=O	C45H46ClFN8O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-IO72HB	WO2023222012A1_392	.	COc1cc(O[C@H]2C(C)(C)[C@H](N3Cc4nc(C#C[C@H]5C[C@H](N6CCN(c7ccc(C(=O)NC8CCC(=O)NC8=O)c(C(C)=O)c7)CC6)C5)ccc4C3=O)C2(C)C)ccc1C#N	C47H51N7O7	AR	P10275	CRBN	WO-2023222012-A1
TPD-JA83P1	WO2023222012A1_393	.	COc1cc(O[C@H]2C(C)(C)[C@H](N3Cc4nc(C#C[C@H]5C[C@H](N6CCN(c7cc(C(C)=O)c(C(=O)NC8CCC(=O)NC8=O)cc7F)CC6)C5)ccc4C3=O)C2(C)C)ccc1C#N	C47H50FN7O7	AR	P10275	CRBN	WO-2023222012-A1
TPD-TOC85O	WO2023222012A1_394	.	CC1(C)[C@H](Oc2ccc(C#N)c(Cl)c2)C(C)(C)[C@H]1N1Cc2nc(C#C[C@H]3C[C@H](N4CCN(c5cnn(C6CCC(=O)NC6=O)c(=O)c5)CC4)C3)ccc2C1=O	C41H43ClN8O5	AR	P10275	CRBN	WO-2023222012-A1
TPD-DQGVIH	WO2023222012A1_395	.	CC1(C)[C@H](Oc2ccc(C#N)c(Cl)c2)C(C)(C)[C@H]1N1Cc2nc(C#C[C@H]3C[C@H](N4CCN(c5cc(=O)n(C6CCC(=O)NC6=O)cn5)CC4)C3)ccc2C1=O	C41H43ClN8O5	AR	P10275	CRBN	WO-2023222012-A1
TPD-XNWRHJ	WO2023222012A1_396	.	CC1(C)[C@H](Oc2ccc(C#N)c(Cl)c2)C(C)(C)[C@H]1N1Cc2nc(C#C[C@H]3C[C@H](N4CCN(c5ccc6c(=O)n(C7CCC(=O)NC7=O)cnc6c5)CC4)C3)ccc2C1=O	C45H45ClN8O5	AR	P10275	CRBN	WO-2023222012-A1
TPD-2M51CX	WO2023222012A1_397	.	CC1(C)[C@H](Oc2ccc(C#N)c(Br)c2)C(C)(C)[C@H]1N1Cc2nc(C#C[C@H]3CC[C@H](N4CCN(c5cc6c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)ccc2C1=O	C47H47BrFN7O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-WGURIY	WO2023222012A1_398	.	CC1(C)[C@H](Oc2ccc(C#N)c(Br)c2)C(C)(C)[C@H]1N1Cc2nc(C#C[C@H]3CC[C@H](N4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)ccc2C1=O	C47H48BrN7O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-6MUW5K	WO2023222012A1_399	.	COc1cc(O[C@H]2C(C)(C)[C@H](N3Cc4nc(C#C[C@H]5CC[C@H](N6CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)ccc4C3=O)C2(C)C)ccc1C#N	C48H50FN7O7	AR	P10275	CRBN	WO-2023222012-A1
TPD-XTCKWX	WO2023222012A1_400	.	COc1cc(O[C@H]2C(C)(C)[C@H](N3Cc4nc(C#C[C@H]5CC[C@H](N6CCN(c7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)ccc4C3=O)C2(C)C)ccc1C#N	C48H51N7O7	AR	P10275	CRBN	WO-2023222012-A1
TPD-G5FJ9B	WO2023222012A1_401	.	Cc1cc(O[C@H]2C(C)(C)[C@H](N3Cc4nc(C#C[C@H]5CC[C@H](N6CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)ccc4C3=O)C2(C)C)ccc1C#N	C48H50FN7O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-F8WPER	WO2023222012A1_402	.	Cc1cc(O[C@H]2C(C)(C)[C@H](N3Cc4nc(C#C[C@H]5CC[C@H](N6CCN(c7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)ccc4C3=O)C2(C)C)ccc1C#N	C48H51N7O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-1W24Z7	WO2023222012A1_413	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3nc(N4CCC(CN5CCC6(CC5)CN(c5ccc7c(c5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)no3)CC2)cc1Cl	C42H46ClN9O7	AR	P10275	CRBN	WO-2023222012-A1
TPD-SRX5M2	WO2023222012A1_414	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3nnc(N4CCC(CN5CCC6(CC5)CN(c5ccc7c(c5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)o3)CC2)cc1Cl	C42H46ClN9O7	AR	P10275	CRBN	WO-2023222012-A1
TPD-D8ASJY	WO2023222012A1_415	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3noc(N4CCC(CN5CCC6(CC5)CN(c5ccc7c(c5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)n3)CC2)cc1Cl	C42H46ClN9O7	AR	P10275	CRBN	WO-2023222012-A1
TPD-BFLJ4M	WO2023222012A1_416	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccn(C4CCC(CN5CCC6(CC5)CN(c5ccc7c(c5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)n3)CC2)cc1Cl	C44H49ClN8O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-C77BY1	WO2023222012A1_417	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCC(CN5CCC6(CC5)CN(c5cc7c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C7)C6)CC4)nn3)CC2)cc1Cl	C43H48ClFN10O5	AR	P10275	CRBN	WO-2023222012-A1
TPD-L4QIPM	WO2023222012A1_418	.	CC1(CN2CC3(CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)C2)CCN(c2ccc(C(=O)N[C@H]3CC[C@H](Oc4ccc(C#N)c(Cl)c4)CC3)nn2)CC1	C45H50ClN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-K8Q1N5	WO2023222012A1_419	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCC(CN5CCC6(CC5)CN(c5ccc7c(c5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)nn3)CC2)cc1Br	C43H47BrN10O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-1ZDBCD	WO2023222012A1_420	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCC(CN5CCC6(CC5)CN(c5ccc7c(c5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)nn3)CC2)cc1C(F)(F)F	C44H47F3N10O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-DF28NX	WO2023222012A1_421	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ncc(N4CCC(CN5CCC6(CC5)CN(c5ccc7c(c5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)nn3)CC2)cc1Cl	C43H47ClN10O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-ZVRPL9	WO2023222012A1_422	.	Cc1cc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(C)(CN5CCC6(CC5)CN(c5ccc7c(c5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)nn3)CC2)ccc1C#N	C46H53N9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-X2YA2L	WO2023222012A1_423	.	Cc1cc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(O)(CN5CCC6(CC5)CN(c5ccc7c(c5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)nn3)CC2)ccc1C#N	C45H51N9O7	AR	P10275	CRBN	WO-2023222012-A1
TPD-NH4VYV	WO2023222012A1_424	.	Cc1cc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(F)(CN5CCC6(CC5)CN(c5ccc7c(c5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)nn3)CC2)ccc1C#N	C45H50FN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-P2D6OA	WO2023222012A1_425	.	N#Cc1ccc(O[C@H]2CC[C@H](NCc3ccc(N4CCC(CN5CCC6(CC5)CN(c5ccc7c(c5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)nn3)CC2)cc1Cl	C44H50ClN9O5	AR	P10275	CRBN	WO-2023222012-A1
TPD-IIU184	WO2023222012A1_426	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCC(F)(CN5CCC6(CC5)CN(c5ccc7c(c5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)nn3)CC2)cc1Cl	C43H46ClFN10O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-Z0598E	WO2023222012A1_427	.	N#Cc1ncc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC6(CC5)CN(c5ccc7c(c5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)nn3)CC2)cc1Cl	C43H47ClN10O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-LGF1UP	WO2023222012A1_430	.	CCOc1cc(O[C@H]2C(C)(C)[C@H](N3Cc4nc(C#C[C@H]5CC[C@H](N6CCN(c7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)ccc4C3=O)C2(C)C)ccc1C#N	C49H53N7O7	AR	P10275	CRBN	WO-2023222012-A1
TPD-OWO0U3	WO2023222012A1_431	.	CC1(C)[C@H](Oc2ccc(C#N)c(Br)c2)C(C)(C)[C@H]1N1Cc2nc(C#C[C@H]3C[C@H](N4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C3)ccc2C1=O	C45H44BrN7O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-GJ63JU	WO2023222012A1_432	.	CC1(C)[C@H](Oc2ccc(C#N)c(Cl)c2)C(C)(C)[C@H]1N1Cc2nc(C#C[C@H]3CC[C@H](N4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)ccc2C1=O	C47H48ClN7O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-K3509N	WO2023222012A1_51	.	CC1(C)[C@H](Oc2ccc(C#N)c(Cl)c2)C(C)(C)[C@H]1N1Cc2cc(C#CC3CCN(C4CCN(c5cc6c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)ccc2C1=O	C48H48ClFN6O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-S0ICTU	WO2023222012A1_56	.	N#Cc1ccc(O[C@H]2CC[C@H](N3Cc4nc(N5CCC(CN6CCN(c7ccc8c(c7)CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)ccc4C3=O)CC2)cc1Cl	C43H47ClN8O5	AR	P10275	CRBN	WO-2023222012-A1
TPD-AKA7GI	WO2023222012A1_57	.	N#Cc1ccc(O[C@H]2CC[C@H](N3Cc4nc(N5CCC(CN6CCN(c7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)ccc4C3=O)CC2)cc1Cl	C43H45ClN8O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-MS3WI9	WO2023222012A1_58	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3)CC2)cc1Cl	C44H48ClN7O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-F0O6MQ	WO2023222012A1_59	.	N#Cc1ccc(O[C@H]2CC[C@H](N3Cc4nc(N5CCC(OC6CCN(c7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)ccc4C3=O)CC2)cc1Cl	C43H44ClN7O7	AR	P10275	CRBN	WO-2023222012-A1
TPD-XXGAKG	WO2023222012A1_60	.	N#Cc1ccc(O[C@H]2CC[C@H](N3Cc4nc(N5CCC(OC6CCN(c7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)ccc4C3=O)CC2)cc1Cl	C43H44ClN7O7	AR	P10275	CRBN	WO-2023222012-A1
TPD-L9ZVDG	WO2023222012A1_61	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(N5CC6(CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)C5)CC4)nn3)CC2)cc1Cl	C43H45ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-Y74JVP	WO2023222012A1_62	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(N5CC6CN(c7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6C5)CC4)nn3)CC2)cc1Cl	C42H44ClN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-CSL1MA	WO2023222012A1_63	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCC(N5CC6CN(c7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6C5)CC4)cn3)CC2)cc1Cl	C42H44ClN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-KX4WFC	WO2023222012A1_64	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCC(N5CC6CN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6C5)CC4)cn3)CC2)cc1Cl	C42H43ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-Y6FS5C	WO2023222012A1_65	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(N5CC6CN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6C5)CC4)nn3)CC2)cc1Cl	C42H43ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-K9AUO8	WO2023222012A1_67	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CC5CN(C6CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5C4)nn3)CC2)cc1Cl	C42H43ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-2MQZXJ	WO2023222012A1_68	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCC(N5CC6CN(c7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6C5)CC4)nc3)CC2)cc1Cl	C42H44ClN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-OI0292	WO2023222012A1_69	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CC5CN(C6CCN(c7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5C4)cn3)CC2)cc1Cl	C42H44ClN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-A2G3QJ	WO2023222012A1_70	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CC5CN(C6CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5C4)cn3)CC2)cc1Cl	C42H43ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-NAQBHQ	WO2023222012A1_71	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC5(CC4)CN(C4CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC4)C5)nn3)CC2)cc1Cl	C43H45ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-X3F1OW	WO2023222012A1_72	.	CC1(C)[C@H](NC(=O)c2ccc(N3CC4CN(C5CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4C3)nn2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C44H47ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-37V6GX	WO2023222012A1_73	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCC(NC5CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cn3)CC2)cc1Cl	C41H43ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-EQI9T0	WO2023222012A1_74	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC5(CC4)CN(C4CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC4)C5)nn3)CC2)cc1Cl	C43H46ClN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-4DQI35	WO2023222012A1_75	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC5(CC4)CN(CC4CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC4)C5)nn3)CC2)cc1Cl	C44H47ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-OKMQC9	WO2023222012A1_76	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCC5(CC4)CN(CC4CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC4)C5)cn3)CC2)cc1Cl	C44H47ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-GCXQ10	WO2023222012A1_77	.	N#CC1=CCC(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(N5CC6(CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)C5)CC4)nc3)CC2)C=C1Cl	C44H48ClFN8O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-6VPCC7	WO2023222012A1_78	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(N5CC6(CCN(c7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)C5)CC4)nn3)CC2)cc1Cl	C43H46ClN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-SHP684	WO2023222012A1_79	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(N5CC6(CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)C5)CC4)nn3)CC2)cc1C(F)(F)F	C44H45F4N9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-V4H93M	WO2023222012A1_80	.	CC1(C)[C@H](NC(=O)c2ccc(N3CCC(N4CC5(CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)CC3)nn2)C(C)(C)[C@@H]1Oc1ccc(C#N)c(Cl)c1	C45H49ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-ZLCH2T	WO2023222012A1_81	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CC5(CCN(C6CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)C5)C4)nn3)CC2)cc1Cl	C42H43ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-535N3X	WO2023222012A1_82	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CC5(CCN(C6CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)C5)C4)cn3)CC2)cc1Cl	C42H43ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-92QMGD	WO2023222012A1_83	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3nnc(N4CCC(N5CCC6(CC5)CN(c5cc7c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)s3)CC2)cc1Cl	C41H43ClFN9O6S	AR	P10275	CRBN	WO-2023222012-A1
TPD-NHATTH	WO2023222012A1_84	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ncn([C@H]4CC[C@H](CN5CCC6(CC5)CN(c5ccc7c(c5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)n3)CC2)cc1Cl	C43H48ClN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-DXDMVO	WO2023222012A1_85	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ncn([C@H]4CC[C@H](CN5CCC6(CC5)CN(c5cc7c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)n3)CC2)cc1Cl	C43H47ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-61O30A	WO2023222012A1_86	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ncnn3[C@H]3CC[C@H](CN4CCC5(CC4)CN(c4ccc6c(c4)C(=O)N(C4CCC(=O)NC4=O)C6=O)C5)CC3)CC2)cc1Cl	C43H48ClN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-1FZBET	WO2023222012A1_87	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ncnn3[C@H]3CC[C@H](CN4CCC5(CC4)CN(c4cc6c(cc4F)C(=O)N(C4CCC(=O)NC4=O)C6=O)C5)CC3)CC2)cc1Cl	C43H47ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-F2MT5K	WO2023222012A1_88	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CC5(CCN(C6CCN(c7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)C4)nn3)CC2)cc1Cl	C43H46ClN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-5J51S5	WO2023222012A1_89	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CC5(CCN(C6CCN(c7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)C4)cn3)CC2)cc1Cl	C43H46ClN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-33SUAA	WO2023222012A1_90	.	CC1(C)[C@H](Oc2ccc(C#N)c(Cl)c2)C(C)(C)[C@H]1N1Cc2nc(N3CCC(CN4CCC5(CC4)CN(c4cc6c(cc4F)C(=O)N(C4CCC(=O)NC4=O)C6=O)C5)CC3)ccc2C1=O	C48H52ClFN8O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-UJOT2T	WO2023222012A1_91	.	CN(C(=O)c1ccc(N2CCC3(CC2)CN(CC2CCN(c4cc5c(cc4F)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC2)C3)nn1)[C@H]1CC[C@H](OC2=CC=C(C#N)C(Cl)C2)CC1	C45H51ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-FXX4NG	WO2023222012A1_92	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CC5(CN(C[C@@H]6[C@H]7CN(c8cc9c(cc8F)C(=O)N(C8CCC(=O)NC8=O)C9=O)C[C@@H]67)C5)C4)nn3)CC2)cc1Cl	C42H41ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-2J43RK	WO2023222012A1_93	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCCN(C[C@@H]5[C@H]6CN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)C[C@@H]56)CC4)nn3)CC2)cc1Cl	C42H43ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-3A5JVW	WO2023222012A1_94	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCN(C[C@@H]5[C@H]6CN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)C[C@@H]56)CC4)cn3)CC2)cc1C(F)(F)F	C42H41F4N9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-T2O51D	WO2023222012A1_95	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCN(C[C@@H]5[C@H]6CN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)C[C@@H]56)CC4)nn3)CC2)cc1C(F)(F)F	C42H41F4N9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-WDX01P	WO2023222012A1_96	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CC5(CCN(CC6CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)C5)C4)cn3)CC2)cc1Cl	C43H45ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-8N6SGF	WO2023222012A1_97	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CC5(CCN(C6CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)C4)nn3)CC2)cc1Cl	C43H45ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-YPUG3I	WO2023222012A1_98	.	Cc1cc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CC5(CCN(CC6CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)C5)C4)nn3)CC2)ccc1C#N	C44H48FN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-BWYD7P	WO2023222012A1_99	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3cnc(N4CCN(C[C@@H]5[C@H]6CN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)C[C@@H]56)CC4)cn3)CC2)cc1Cl	C41H41ClFN9O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-MQ7LXR	WO2023222012A1_ARD2128	.	CC1(C)[C@H](NC(=O)c2ccc(N3CCN(CC4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)cc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C45H50ClN7O6	AR	P10275	CRBN	WO-2023222012-A1
TPD-2UN8ON	WO2023222762A1_1	.	CC1(C)CCN(Cc2cc(F)c(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCOCCOCCNc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)cc2F)CC1	C49H63F2N11O8	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-JSZTIH	WO2023222762A1_2	.	CC1(C)CCN(Cc2cc(F)c(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCOCCOCCOCCNc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)cc2F)CC1	C51H67F2N11O9	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-20Y89W	WO2023222762A1_3	.	CC1(C)CCN(Cc2cc(F)c(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCOCCOCCOCCOCCNc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)cc2F)CC1	C53H71F2N11O10	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-HD3V5H	WO2023222762A1_4	.	CC1(C)CCN(Cc2cc(F)c(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCOCCOCCOCCOCCOCCNc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)cc2F)CC1	C55H75F2N11O11	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-4CO30E	WO2023222762A1_5	.	CC1(C)CCN(Cc2cc(F)c(N3CC(=O)NC4(CCN(C5=NCNC(NCCCNC(=O)CCCCCCCCn6cc(CNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)=C5)CC4)C3)cc2F)CC1	C54H72F2N14O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-DETWNY	WO2023222762A1_6	.	CC1(C)CCN(Cc2cc(F)c(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCN6CC(CNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)N=N6)ncn5)CC4)C3)cc2F)CC1	C54H72F2N14O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-I4EQEY	SCHEMBL26656834	N-[3-[[6-[4-[4-[(4,4-dimethylpiperidin-1-yl)methyl]-2,5-difluorophenyl]-2-oxo-1,4,9-triazaspiro[5.5]undecan-9-yl]pyrimidin-4-yl]amino]propyl]-11-[4-[[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]methyl]triazol-1-yl]undecanamide; SCHEMBL30665458	CC1(C)CCN(Cc2cc(F)c(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCn6cc(CNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2F)CC1	C56H74F2N14O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-V03XHW	WO2023222762A1_8	.	CC1(C)CCN(Cc2cc(F)c(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCn6cc(CNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2F)CC1	C56H74F2N14O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-E9AMIG	WO2023222762A1_9	.	CC1(C)CCN(Cc2cc(F)c(N3CC(=O)NC4(CCN(c5cc(NCCCOC(=O)CCCCCCCCCCCCn6cc(CNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2F)CC1	C58H77F2N13O7	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-63B1DY	WO2023222762A1_10	.	CC1(C)CCN(Cc2cc(F)c(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCCn6cc(CNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2F)CC1	C58H78F2N14O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-OYPBPS	WO2023222762A1_11	.	CC1(C)CCN(Cc2cc(F)c(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCCCCn6cc(CNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2F)CC1	C60H82F2N14O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-E85TUH	WO2023222762A1_12	.	CC1(C)CCN(Cc2cc(F)c(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCCCCn6cc(CNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2F)CC1	C60H82F2N14O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-1VK11G	SCHEMBL26656826	N-[3-[[6-[4-[4-[(4,4-dimethylpiperidin-1-yl)methyl]-2,5-difluorophenyl]-2-oxo-1,4,9-triazaspiro[5.5]undecan-9-yl]pyrimidin-4-yl]amino]propyl]-9-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]nonanamide; SCHEMBL30665454	CC1(C)CCN(Cc2cc(F)c(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCNc6cccc7c6CN(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)cc2F)CC1	C51H69F2N11O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-WRND68	WO2023222762A1_14	.	CC1(C)CCN(Cc2cc(F)c(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCNc6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)cc2F)CC1	C51H69F2N11O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-13EWFE	SCHEMBL26656799	N-[3-[[6-[4-[4-[(4,4-dimethylpiperidin-1-yl)methyl]-2,5-difluorophenyl]-2-oxo-1,4,9-triazaspiro[5.5]undecan-9-yl]pyrimidin-4-yl]amino]propyl]-11-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]undecanamide; SCHEMBL30665569	CC1(C)CCN(Cc2cc(F)c(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCNc6cccc7c6CN(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)cc2F)CC1	C53H73F2N11O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-8KVWOQ	WO2023222762A1_16	.	CC1(C)CCN(Cc2cc(F)c(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCNc6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)cc2F)CC1	C53H73F2N11O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-BBT866	WO2023222762A1_17	.	CC1(C)CCN(Cc2cc(F)c(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCCNc6cccc7c6CN(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)cc2F)CC1	C55H77F2N11O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-5BK9T5	WO2023222762A1_18	.	CC1(C)CCN(Cc2cc(F)c(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCCNc6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)cc2F)CC1	C55H77F2N11O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-JPE35C	WO2023222762A1_19	.	CC1(C)CCN(Cc2cc(F)c(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCCCCNc6cccc7c6CN(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)cc2F)CC1	C57H81F2N11O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-7MVAA1	WO2023222762A1_20	.	CC1(C)CCN(Cc2cc(F)c(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCCCCNc6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)cc2F)CC1	C57H81F2N11O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-HM93V4	WO2023222762A1_21	.	CC1(C)CCN(Cc2cc(F)c(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCn6cc(CN7CCN(c8cccc9c8C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)nn6)ncn5)CC4)C3)cc2F)CC1	C55H71F2N15O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-8S56C9	WO2023222762A1_22	.	CC1(C)CCN(Cc2cc(F)c(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCn6cc(CN7CCN(c8ccc9c(c8)C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)nn6)ncn5)CC4)C3)cc2F)CC1	C55H71F2N15O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-R96QPG	WO2023222762A1_25	.	CC1(C)CCN(Cc2cc(F)c(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCn6cc(CN7CCN(c8cccc9c8C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)nn6)ncn5)CC4)C3)cc2F)CC1	C57H75F2N15O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-EA92ZY	WO2023222762A1_26	.	CC1(C)CCN(Cc2cc(F)c(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCn6cc(CN7CCN(c8ccc9c(c8)C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)nn6)ncn5)CC4)C3)cc2F)CC1	C57H75F2N15O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-2AXQ81	WO2023222762A1_27	.	CC1(C)CCN(Cc2cc(F)c(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCn6cc(CN7CCN(c8cccc9c8C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)nn6)ncn5)CC4)C3)cc2F)CC1	C61H83F2N15O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-JS3A3P	WO2023222762A1_28	.	CC1(C)CCN(Cc2cc(F)c(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCn6cc(CN7CCN(c8ccc9c(c8)C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)nn6)ncn5)CC4)C3)cc2F)CC1	C61H83F2N15O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-81Z2PH	WO2023222762A1_29	.	CC1(C)CCN(Cc2cc(F)c(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(CNC(=O)CCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2F)CC1	C56H69F2N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-DN5SJB	WO2023222762A1_30	.	CC1(C)CCN(Cc2cc(F)c(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(CNC(=O)CCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2F)CC1	C56H69F2N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-GGPWVX	WO2023222762A1_31	.	CC1(C)CCN(Cc2cc(F)c(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(CNC(=O)CCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2F)CC1	C58H73F2N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-72QNUH	WO2023222762A1_33	.	CC1(C)CCN(Cc2cc(F)c(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(CNC(=O)CCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2F)CC1	C60H77F2N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-DP7TMB	WO2023222762A1_34	.	CC1(C)CCN(Cc2cc(F)c(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(CNC(=O)CCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2F)CC1	C58H73F2N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-7AXXVB	WO2023222762A1_35	.	CC1(C)CCN(Cc2cc(F)c(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(CNC(=O)CCCCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2F)CC1	C62H81F2N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-BLYGJQ	WO2023222762A1_36	.	CC1(C)CCN(Cc2cc(F)c(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(CNC(=O)CCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2F)CC1	C60H77F2N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-MV5963	WO2023222762A1_37	.	CC1(C)CCN(Cc2cc(F)c(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(C(=O)NCCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2F)CC1	C59H75F2N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-4TIJTU	WO2023222762A1_38	.	CC1(C)CCN(Cc2cc(F)c(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(C(=O)NCCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2F)CC1	C59H75F2N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-OWED6C	WO2023222762A1_39	.	CC1(C)CCN(Cc2cc(F)c(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(C(=O)NCCCCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2F)CC1	C61H79F2N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-447Z8J	WO2023222762A1_40	.	CC1(C)CCN(Cc2cc(F)c(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(C(=O)NCCCCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2F)CC1	C61H79F2N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-BLJSLI	WO2023222762A1_41	.	CC1(C)CCN(Cc2cc(F)c(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(C(=O)NCCCCCCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2F)CC1	C63H83F2N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-ZK9FL0	WO2023222762A1_42	.	CC1(C)CCN(Cc2cc(F)c(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(C(=O)NCCCCCCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2F)CC1	C63H83F2N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-4YHXWN	WO2023222762A1_43	.	CC1(C)CCN(Cc2cc(F)c(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(C(=O)NCCCCCCCCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2F)CC1	C65H87F2N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-B3JJHE	WO2023222762A1_44	.	CC1(C)CCN(Cc2cc(F)c(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(C(=O)NCCCCCCCCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2F)CC1	C65H87F2N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-ZN09AF	WO2023222762A1_45	.	CC1(C)CCN(Cc2cc(F)c(N3CC(=O)NC4(CCN(c5cc(NCc6cn(CCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2F)CC1	C54H71F2N13O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-2JZ5UB	WO2023222762A1_46	.	CC1(C)CCN(Cc2cc(F)c(N3CC(=O)NC4(CCN(c5cc(NCC6=NC(CCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)N=N6)ncn5)CC4)C3)cc2F)CC1	C54H71F2N13O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-4JR6Y9	WO2023222762A1_47	.	CC1(C)CCN(Cc2cc(F)c(N3CC(=O)NC4(CCN(c5cc(NCc6cn(CCCCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2F)CC1	C56H75F2N13O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-FGVGWA	WO2023222762A1_48	.	CC1(C)CCN(Cc2cc(F)c(N3CC(=O)NC4(CCN(c5cc(NCC6=NC(CCCCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)N=N6)ncn5)CC4)C3)cc2F)CC1	C56H75F2N13O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-JQ02W4	WO2023222762A1_49	.	CC1(C)CCN(Cc2cc(F)c(N3CC(=O)NC4(CCN(c5cc(NCc6cn(CCCCCCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2F)CC1	C58H79F2N13O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-3XTJPR	WO2023222762A1_50	.	CC1(C)CCN(Cc2cc(F)c(N3CC(=O)NC4(CCN(c5cc(NCC6=NC(CCCCCCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)N=N6)ncn5)CC4)C3)cc2F)CC1	C58H79F2N13O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-HS1AB1	WO2023222762A1_51	.	CC1(C)CCN(Cc2cc(F)c(N3CC(=O)NC4(CCN(c5cc(NCc6cn(CCCCCCCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2F)CC1	C59H81F2N13O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-AWH3NH	WO2023222762A1_52	.	CC1(C)CCN(Cc2cc(F)c(N3CC(=O)NC4(CCN(c5cc(NCC6=NC(CCCCCCCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)N=N6)ncn5)CC4)C3)cc2F)CC1	C59H81F2N13O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-LMOTYP	WO2023222762A1_53	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCOCCOCCNc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)cc2C(F)(F)F)CC1	C50H64F3N11O8	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-0BCTHY	WO2023222762A1_54	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCOCCOCCOCCNc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)cc2C(F)(F)F)CC1	C52H68F3N11O9	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-9WZ7FY	WO2023222762A1_55	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCOCCOCCOCCOCCNc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)cc2C(F)(F)F)CC1	C54H72F3N11O10	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-YTCNVT	WO2023222762A1_56	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCOCCOCCOCCOCCOCCNc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)cc2C(F)(F)F)CC1	C56H76F3N11O11	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-0UC1Z8	WO2023222762A1_57	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCn6cc(CNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2C(F)(F)F)CC1	C55H71F3N14O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-2T3MGV	WO2023222762A1_58	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCn6cc(CNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8O)nn6)ncn5)CC4)C3)cc2C(F)(F)F)CC1	C55H73F3N14O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-D579WG	WO2023222762A1_59	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCn6cc(CNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2C(F)(F)F)CC1	C57H75F3N14O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-79YSS6	WO2023222762A1_60	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCn6cc(CNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8O)nn6)ncn5)CC4)C3)cc2C(F)(F)F)CC1	C57H77F3N14O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-E7OO8T	WO2023222762A1_61	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCCn6cc(CNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2C(F)(F)F)CC1	C59H79F3N14O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-JB7541	WO2023222762A1_62	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCCn6cc(CNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8O)nn6)ncn5)CC4)C3)cc2C(F)(F)F)CC1	C59H81F3N14O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-9IN0EJ	WO2023222762A1_63	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCCCCn6cc(CNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2C(F)(F)F)CC1	C61H83F3N14O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-E1CBYD	WO2023222762A1_64	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCCCCn6cc(CNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8O)nn6)ncn5)CC4)C3)cc2C(F)(F)F)CC1	C61H85F3N14O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-5IZ4DD	WO2023222762A1_65	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCNc6cccc7c6CN(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)cc2C(F)(F)F)CC1	C52H70F3N11O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-XAN6IW	WO2023222762A1_66	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCNc6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)cc2C(F)(F)F)CC1	C52H70F3N11O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-KEWMHM	WO2023222762A1_67	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCNc6cccc7c6CN(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)cc2C(F)(F)F)CC1	C54H74F3N11O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-GSOGHB	WO2023222762A1_68	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCNc6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)cc2C(F)(F)F)CC1	C54H74F3N11O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-DW93W8	WO2023222762A1_69	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCCNc6cccc7c6CN(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)cc2C(F)(F)F)CC1	C56H78F3N11O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-EZZHVH	WO2023222762A1_70	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCCNc6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)cc2C(F)(F)F)CC1	C56H78F3N11O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-3GS1KO	WO2023222762A1_71	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCCCCNc6cccc7c6CN(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)cc2C(F)(F)F)CC1	C58H82F3N11O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-PNFOT4	WO2023222762A1_72	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCCCCNc6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)cc2C(F)(F)F)CC1	C58H82F3N11O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-9UXE6U	WO2023222762A1_73	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCn6cc(CN7CCN(c8cccc9c8C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)nn6)ncn5)CC4)C3)cc2C(F)(F)F)CC1	C56H72F3N15O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-VSHARF	WO2023222762A1_74	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCn6cc(CN7CCN(c8ccc9c(c8)C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)nn6)ncn5)CC4)C3)cc2C(F)(F)F)CC1	C56H72F3N15O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-1N2H54	WO2023222762A1_77	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCn6cc(CN7CCN(c8cccc9c8C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)nn6)ncn5)CC4)C3)cc2C(F)(F)F)CC1	C58H76F3N15O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-JPR3HW	WO2023222762A1_78	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCn6cc(CN7CCN(c8ccc9c(c8)C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)nn6)ncn5)CC4)C3)cc2C(F)(F)F)CC1	C58H76F3N15O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-Z8WIB5	WO2023222762A1_79	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCn6cc(CN7CCN(c8cccc9c8C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)nn6)ncn5)CC4)C3)cc2C(F)(F)F)CC1	C62H84F3N15O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-C70M0O	WO2023222762A1_80	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCn6cc(CN7CCN(c8ccc9c(c8)C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)nn6)ncn5)CC4)C3)cc2C(F)(F)F)CC1	C62H84F3N15O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-7MLY5W	WO2023222762A1_81	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(CNC(=O)CCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2C(F)(F)F)CC1	C57H70F3N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-EUD1RL	WO2023222762A1_82	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(CNC(=O)CCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2C(F)(F)F)CC1	C57H70F3N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-WUVEP8	WO2023222762A1_83	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(CNC(=O)CCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2C(F)(F)F)CC1	C59H74F3N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-CRUOL6	WO2023222762A1_84	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(CNC(=O)CCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2C(F)(F)F)CC1	C59H74F3N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-M60KNB	WO2023222762A1_85	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(CNC(=O)CCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2C(F)(F)F)CC1	C61H78F3N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-2VK4M1	WO2023222762A1_86	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(CNC(=O)CCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2C(F)(F)F)CC1	C61H78F3N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-K3HGBN	WO2023222762A1_87	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(CNC(=O)CCCCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2C(F)(F)F)CC1	C63H82F3N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-4ZD1GU	WO2023222762A1_88	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(CNC(=O)CCCCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2C(F)(F)F)CC1	C63H82F3N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-LSR4RD	WO2023222762A1_89	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(C(=O)NCCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2C(F)(F)F)CC1	C60H76F3N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-I364JR	WO2023222762A1_90	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(C(=O)NCCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2C(F)(F)F)CC1	C60H76F3N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-KVIO5Q	WO2023222762A1_91	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(C(=O)NCCCCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2C(F)(F)F)CC1	C62H80F3N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-F4FP5F	WO2023222762A1_92	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(C(=O)NCCCCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2C(F)(F)F)CC1	C62H80F3N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-E9FJ2I	WO2023222762A1_93	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(C(=O)NCCCCCCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2C(F)(F)F)CC1	C64H84F3N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-GORUM7	WO2023222762A1_94	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(C(=O)NCCCCCCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2C(F)(F)F)CC1	C64H84F3N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-GYP5FN	WO2023222762A1_95	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(C(=O)NCCCCCCCCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2C(F)(F)F)CC1	C66H88F3N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-PDG6TI	WO2023222762A1_96	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(C(=O)NCCCCCCCCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2C(F)(F)F)CC1	C66H88F3N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-XQEAGU	WO2023222762A1_97	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cn(CCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2C(F)(F)F)CC1	C55H72F3N13O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-3MXWHI	WO2023222762A1_98	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cn(CCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2C(F)(F)F)CC1	C55H72F3N13O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-EPV8LX	WO2023222762A1_99	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cn(CCCCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2C(F)(F)F)CC1	C57H76F3N13O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-5SMZPB	WO2023222762A1_100	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cn(CCCCCCCCCCCCCCNc7ccc8c(c7)CN(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2C(F)(F)F)CC1	C57H78F3N13O4	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-U83MYG	WO2023222762A1_101	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cn(CCCCCCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2C(F)(F)F)CC1	C59H80F3N13O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-KLZN85	WO2023222762A1_102	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cn(CCCCCCCCCCCCCCCCNc7ccc8c(c7)CN(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2C(F)(F)F)CC1	C59H82F3N13O4	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-JASLCE	WO2023222762A1_103	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cn(CCCCCCCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2C(F)(F)F)CC1	C60H82F3N13O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-LWZRS8	WO2023222762A1_104	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cn(CCCCCCCCCCCCCCCCCNc7ccc8c(c7)CN(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2C(F)(F)F)CC1	C60H84F3N13O4	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-QM3550	WO2023222762A1_105	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCOCCOCCNc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)c(F)c2F)CC1	C49H63F2N11O8	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-HUT8YL	WO2023222762A1_106	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCOCCOCCOCCNc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)c(F)c2F)CC1	C51H67F2N11O9	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-EEAKU7	WO2023222762A1_107	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCOCCOCCOCCOCCNc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)c(F)c2F)CC1	C53H71F2N11O10	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-YW6DXE	WO2023222762A1_108	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCOCCOCCOCCOCCOCCNc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)c(F)c2F)CC1	C55H75F2N11O11	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-LW96FB	WO2023222762A1_109	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCn6cc(CNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)c(F)c2F)CC1	C54H70F2N14O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-4WDEPQ	WO2023222762A1_110	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCn6cc(CNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)c(F)c2F)CC1	C54H70F2N14O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-J63H30	WO2023222762A1_111	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCn6cc(CNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)c(F)c2F)CC1	C56H74F2N14O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-41O9RN	WO2023222762A1_112	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCn6cc(CNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)c(F)c2F)CC1	C56H74F2N14O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-JZ5BA3	WO2023222762A1_113	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCCn6cc(CNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)c(F)c2F)CC1	C58H78F2N14O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-W5G0I7	WO2023222762A1_114	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCCn6cc(CNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)c(F)c2F)CC1	C58H78F2N14O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-6PIKH7	WO2023222762A1_115	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCCCCn6cc(CNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)c(F)c2F)CC1	C60H82F2N14O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-PCADWS	WO2023222762A1_116	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCCCCn6cc(CNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)c(F)c2F)CC1	C60H82F2N14O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-BUSAYM	WO2023222762A1_117	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCNc6cccc7c6CN(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)c(F)c2F)CC1	C51H69F2N11O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-K5R7VQ	WO2023222762A1_118	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCNc6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)c(F)c2F)CC1	C51H69F2N11O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-PUBU0V	WO2023222762A1_119	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCNc6cccc7c6CN(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)c(F)c2F)CC1	C53H73F2N11O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-FIK959	WO2023222762A1_120	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCNc6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)c(F)c2F)CC1	C53H73F2N11O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-GPEUKD	WO2023222762A1_121	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCCNc6cccc7c6CN(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)c(F)c2F)CC1	C55H77F2N11O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-XLL8L8	WO2023222762A1_122	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCCNc6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)c(F)c2F)CC1	C55H77F2N11O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-P8NYLZ	WO2023222762A1_123	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCCCCNc6cccc7c6CN(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)c(F)c2F)CC1	C57H81F2N11O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-YE5UXL	WO2023222762A1_124	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCCCCNc6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)c(F)c2F)CC1	C57H81F2N11O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-E5ZNMW	WO2023222762A1_125	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCn6cc(CN7CCN(c8cccc9c8C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)nn6)ncn5)CC4)C3)c(F)c2F)CC1	C55H71F2N15O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-ZFBIMG	WO2023222762A1_126	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCn6cc(CN7CCN(c8ccc9c(c8)C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)nn6)ncn5)CC4)C3)c(F)c2F)CC1	C55H71F2N15O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-KPLIH7	WO2023222762A1_129	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCn6cc(CN7CCN(c8cccc9c8C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)nn6)ncn5)CC4)C3)c(F)c2F)CC1	C57H75F2N15O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-YQ10FY	WO2023222762A1_130	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCn6cc(CN7CCN(c8ccc9c(c8)C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)nn6)ncn5)CC4)C3)c(F)c2F)CC1	C57H75F2N15O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-6T8BYO	WO2023222762A1_131	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCn6cc(CN7CCN(c8cccc9c8C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)nn6)ncn5)CC4)C3)c(F)c2F)CC1	C61H83F2N15O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-XL4GQZ	WO2023222762A1_132	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCn6cc(CN7CCN(c8ccc9c(c8)C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)nn6)ncn5)CC4)C3)c(F)c2F)CC1	C61H83F2N15O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-YLSOFK	WO2023222762A1_133	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(CNC(=O)CCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)c(F)c2F)CC1	C56H69F2N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-LLF7P6	WO2023222762A1_134	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(CNC(=O)CCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)c(F)c2F)CC1	C56H69F2N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-0DPTKQ	WO2023222762A1_135	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(CNC(=O)CCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)c(F)c2F)CC1	C58H73F2N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-X8IBZ3	WO2023222762A1_136	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(CNC(=O)CCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)c(F)c2F)CC1	C58H73F2N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-K0ZIF1	WO2023222762A1_137	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(CNC(=O)CCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)c(F)c2F)CC1	C60H77F2N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-7S7PD0	WO2023222762A1_138	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(CNC(=O)CCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)c(F)c2F)CC1	C60H77F2N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-GS8UUS	WO2023222762A1_139	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(CNC(=O)CCCCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)c(F)c2F)CC1	C62H81F2N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-HC6AAO	WO2023222762A1_140	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(CNC(=O)CCCCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)c(F)c2F)CC1	C62H81F2N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-9ZQ66Z	WO2023222762A1_141	.	C=C1c2cccc(NCCCCCCCCCCCCNC(=O)c3cccc(CNc4cc(N5CCC6(CC5)CN(c5ccc(CN7CCC(C)(C)CC7)c(F)c5F)CC(=O)N6)ncn4)c3)c2C(=O)N1C1CCC(=O)NC1=O	C60H77F2N11O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-WXNOMR	WO2023222762A1_142	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(C(=O)NCCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)c(F)c2F)CC1	C59H75F2N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-XOU0W5	WO2023222762A1_143	.	C=C1c2cccc(NCCCCCCCCCCCCCCNC(=O)c3cccc(CNc4cc(N5CCC6(CC5)CN(c5ccc(CN7CCC(C)(C)CC7)c(F)c5F)CC(=O)N6)ncn4)c3)c2C(=O)N1C1CCC(=O)NC1=O	C62H81F2N11O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-6CKQW4	WO2023222762A1_144	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(C(=O)NCCCCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)c(F)c2F)CC1	C61H79F2N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-9297PI	WO2023222762A1_145	.	C=C1c2cccc(NCCCCCCCCCCCCCCCCNC(=O)c3cccc(CNc4cc(N5CCC6(CC5)CN(c5ccc(CN7CCC(C)(C)CC7)c(F)c5F)CC(=O)N6)ncn4)c3)c2C(=O)N1C1CCC(=O)NC1=O	C64H85F2N11O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-0PZLJZ	WO2023222762A1_146	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(C(=O)NCCCCCCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)c(F)c2F)CC1	C63H83F2N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-7KYQ4D	WO2023222762A1_147	.	C=C1c2cccc(NCCCCCCCCCCCCCCCCCCNC(=O)c3cccc(CNc4cc(N5CCC6(CC5)CN(c5ccc(CN7CCC(C)(C)CC7)c(F)c5F)CC(=O)N6)ncn4)c3)c2C(=O)N1C1CCC(=O)NC1=O	C66H89F2N11O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-91X3YA	WO2023222762A1_148	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(C(=O)NCCCCCCCCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)c(F)c2F)CC1	C65H87F2N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-AOGCWS	WO2023222762A1_149	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cn(CCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)c(F)c2F)CC1	C54H71F2N13O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-ZLMQAR	WO2023222762A1_150	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cn(CCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)c(F)c2F)CC1	C54H71F2N13O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-4BSD3T	WO2023222762A1_151	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cn(CCCCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)c(F)c2F)CC1	C56H75F2N13O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-5JISY2	WO2023222762A1_152	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cn(CCCCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)c(F)c2F)CC1	C56H75F2N13O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-RHTEFM	WO2023222762A1_153	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cn(CCCCCCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)c(F)c2F)CC1	C58H79F2N13O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-7AQ1ZC	WO2023222762A1_154	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cn(CCCCCCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)c(F)c2F)CC1	C58H79F2N13O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-VGTT9Y	WO2023222762A1_155	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cn(CCCCCCCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)c(F)c2F)CC1	C59H81F2N13O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-HPI68C	WO2023222762A1_156	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cn(CCCCCCCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)c(F)c2F)CC1	C59H81F2N13O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-LAHVPH	WO2023222762A1_157	.	CC1(C)CCN(Cc2c(F)cc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCOCCOCCNc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)cc2F)CC1	C49H63F2N11O8	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-PXNG3F	WO2023222762A1_158	.	CC1(C)CCN(Cc2c(F)cc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCOCCOCCOCCNc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)cc2F)CC1	C51H67F2N11O9	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-JW1DY0	WO2023222762A1_159	.	CC1(C)CCN(Cc2c(F)cc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCOCCOCCOCCOCCNc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)cc2F)CC1	C53H71F2N11O10	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-K5EC7Y	WO2023222762A1_160	.	CC1(C)CCN(Cc2c(F)cc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCOCCOCCOCCOCCOCCNc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)cc2F)CC1	C55H75F2N11O11	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-2Q3FNB	WO2023222762A1_161	.	CC1(C)CCN(Cc2c(F)cc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCn6cc(CNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2F)CC1	C54H70F2N14O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-4NO2UC	WO2023222762A1_162	.	CC1(C)CCN(Cc2c(F)cc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCn6cc(CNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2F)CC1	C54H70F2N14O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-N4OXAL	WO2023222762A1_163	.	CC1(C)CCN(Cc2c(F)cc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCn6cc(CNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2F)CC1	C56H74F2N14O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-U51SD4	WO2023222762A1_164	.	CC1(C)CCN(Cc2c(F)cc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCn6cc(CNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2F)CC1	C56H74F2N14O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-PN9ADK	WO2023222762A1_165	.	CC1(C)CCN(Cc2c(F)cc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCCn6cc(CNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2F)CC1	C58H78F2N14O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-NQJSQJ	WO2023222762A1_166	.	CC1(C)CCN(Cc2c(F)cc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCCn6cc(CNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2F)CC1	C58H78F2N14O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-WXIL7X	WO2023222762A1_167	.	CC1(C)CCN(Cc2c(F)cc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCCCCn6cc(CNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2F)CC1	C60H82F2N14O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-OJWCWR	WO2023222762A1_168	.	CC1(C)CCN(Cc2c(F)cc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCCCCn6cc(CNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2F)CC1	C60H82F2N14O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-KDWFOE	WO2023222762A1_169	.	CC1(C)CCN(Cc2c(F)cc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCNc6cccc7c6CN(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)cc2F)CC1	C51H69F2N11O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-VGM16C	WO2023222762A1_170	.	CC1(C)CCN(Cc2c(F)cc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCNc6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)cc2F)CC1	C51H69F2N11O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-XLSTA8	WO2023222762A1_171	.	CC1(C)CCN(Cc2c(F)cc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCNc6cccc7c6CN(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)cc2F)CC1	C53H73F2N11O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-OAL36Y	WO2023222762A1_172	.	CC1(C)CCN(Cc2c(F)cc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCNc6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)cc2F)CC1	C53H73F2N11O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-RCII5T	WO2023222762A1_173	.	CC1(C)CCN(Cc2c(F)cc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCCNc6cccc7c6CN(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)cc2F)CC1	C55H77F2N11O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-54UWF4	WO2023222762A1_174	.	CC1(C)CCN(Cc2c(F)cc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCCNc6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)cc2F)CC1	C55H77F2N11O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-IS9YOH	WO2023222762A1_175	.	CC1(C)CCN(Cc2c(F)cc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCCCCNc6cccc7c6CN(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)cc2F)CC1	C57H81F2N11O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-U19X1H	WO2023222762A1_176	.	CC1(C)CCN(Cc2c(F)cc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCCCCNc6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)cc2F)CC1	C57H81F2N11O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-QCQQCP	WO2023222762A1_177	.	CC1(C)CCN(Cc2c(F)cc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCn6cc(CN7CCN(c8cccc9c8C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)nn6)ncn5)CC4)C3)cc2F)CC1	C55H71F2N15O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-0A1HMJ	WO2023222762A1_178	.	CC1(C)CCN(Cc2c(F)cc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCn6cc(CN7CCN(c8ccc9c(c8)C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)nn6)ncn5)CC4)C3)cc2F)CC1	C55H71F2N15O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-SHSBQ7	WO2023222762A1_180	.	CC1(C)CCN(Cc2c(F)cc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCn6cc(CN7CCN(c8ccc9c(c8)C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)nn6)ncn5)CC4)C3)cc2F)CC1	C57H75F2N15O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-PXCU46	WO2023222762A1_181	.	CC1(C)CCN(Cc2c(F)cc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCn6cc(CN7CCN(c8cccc9c8C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)nn6)ncn5)CC4)C3)cc2F)CC1	C57H75F2N15O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-3QJIJU	WO2023222762A1_183	.	CC1(C)CCN(Cc2c(F)cc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCn6cc(CN7CCN(c8cccc9c8C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)nn6)ncn5)CC4)C3)cc2F)CC1	C61H83F2N15O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-7ROW0V	WO2023222762A1_184	.	CC1(C)CCN(Cc2c(F)cc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCn6cc(CN7CCN(c8ccc9c(c8)C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)nn6)ncn5)CC4)C3)cc2F)CC1	C61H83F2N15O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-NCU6YP	WO2023222762A1_185	.	CC1(C)CCN(Cc2c(F)cc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(CNC(=O)CCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2F)CC1	C56H69F2N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-2HVDH9	WO2023222762A1_186	.	CC1(C)CCN(Cc2c(F)cc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(CNC(=O)CCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2F)CC1	C56H69F2N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-Q1QA5I	WO2023222762A1_187	.	CC1(C)CCN(Cc2c(F)cc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(CNC(=O)CCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2F)CC1	C58H73F2N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-OW4ZWC	WO2023222762A1_188	.	CC1(C)CCN(Cc2c(F)cc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(CNC(=O)CCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2F)CC1	C58H73F2N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-TLKKRS	WO2023222762A1_189	.	CC1(C)CCN(Cc2c(F)cc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(CNC(=O)CCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2F)CC1	C60H77F2N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-QNDNXK	WO2023222762A1_190	.	CC1(C)CCN(Cc2c(F)cc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(CNC(=O)CCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2F)CC1	C60H77F2N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-KFADMC	WO2023222762A1_191	.	CC1(C)CCN(Cc2c(F)cc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(CNC(=O)CCCCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2F)CC1	C62H81F2N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-J88VG8	WO2023222762A1_192	.	CC1(C)CCN(Cc2c(F)cc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(CNC(=O)CCCCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2F)CC1	C62H81F2N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-YVZQ2Q	WO2023222762A1_193	.	CC1(C)CCN(Cc2c(F)cc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(C(=O)NCCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2F)CC1	C59H75F2N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-XEE1IA	WO2023222762A1_194	.	CC1(C)CCN(Cc2c(F)cc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(C(=O)NCCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2F)CC1	C59H75F2N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-4OBHWT	WO2023222762A1_195	.	CC1(C)CCN(Cc2c(F)cc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(C(=O)NCCCCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2F)CC1	C61H79F2N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-896IFA	WO2023222762A1_196	.	CC1(C)CCN(Cc2c(F)cc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(C(=O)NCCCCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2F)CC1	C61H79F2N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-W2CIPN	WO2023222762A1_197	.	CC1(C)CCN(Cc2c(F)cc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(C(=O)NCCCCCCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2F)CC1	C63H83F2N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-5PBUJU	WO2023222762A1_198	.	CC1(C)CCN(Cc2c(F)cc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(C(=O)NCCCCCCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2F)CC1	C63H83F2N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-WWW78Q	WO2023222762A1_199	.	CC1(C)CCN(Cc2c(F)cc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(C(=O)NCCCCCCCCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2F)CC1	C65H87F2N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-5LGCDE	WO2023222762A1_200	.	CC1(C)CCN(Cc2c(F)cc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(C(=O)NCCCCCCCCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2F)CC1	C65H87F2N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-T1R3UD	WO2023222762A1_201	.	CC1(C)CCN(Cc2c(F)cc(N3CC(=O)NC4(CCN(c5cc(NCc6cn(CCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2F)CC1	C54H71F2N13O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-IIMIVH	WO2023222762A1_202	.	CC1(C)CCN(Cc2c(F)cc(N3CC(=O)NC4(CCN(c5cc(NCc6cn(CCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2F)CC1	C54H71F2N13O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-2E0KYM	WO2023222762A1_203	.	CC1(C)CCN(Cc2c(F)cc(N3CC(=O)NC4(CCN(c5cc(NCc6cn(CCCCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2F)CC1	C56H75F2N13O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-XTDBPP	WO2023222762A1_204	.	CC1(C)CCN(Cc2c(F)cc(N3CC(=O)NC4(CCN(c5cc(NCc6cn(CCCCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2F)CC1	C56H75F2N13O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-C7CUB8	WO2023222762A1_205	.	CC1(C)CCN(Cc2c(F)cc(N3CC(=O)NC4(CCN(c5cc(NCc6cn(CCCCCCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2F)CC1	C58H79F2N13O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-6YF0IX	WO2023222762A1_206	.	CC1(C)CCN(Cc2c(F)cc(N3CC(=O)NC4(CCN(c5cc(NCc6cn(CCCCCCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2F)CC1	C58H79F2N13O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-GJ1J8Y	WO2023222762A1_207	.	CC1(C)CCN(Cc2c(F)cc(N3CC(=O)NC4(CCN(c5cc(NCc6cn(CCCCCCCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2F)CC1	C59H81F2N13O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-OVYFHP	WO2023222762A1_208	.	CC1(C)CCN(Cc2c(F)cc(N3CC(=O)NC4(CCN(c5cc(NCc6cn(CCCCCCCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2F)CC1	C59H81F2N13O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-IIWN93	WO2023222762A1_209	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCOCCOCCOCCNc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)c(Cl)c2)CC1	C51H68ClN11O9	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-R8RR4O	WO2023222762A1_211	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCOCCOCCOCCOCCNc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)c(Cl)c2)CC1	C53H72ClN11O10	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-VDGK2S	WO2023222762A1_212	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCOCCOCCOCCOCCOCCNC6=CC=CC7C(=O)N(C8CCC(=O)NC8=O)C(=O)C67)ncn5)CC4)C3)c(Cl)c2)CC1	C55H78ClN11O11	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-QQ9MHG	WO2023222762A1_213	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCn6cc(CNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)c(Cl)c2)CC1	C54H71ClN14O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-ACCLPR	WO2023222762A1_214	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCn6cc(CNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)c(Cl)c2)CC1	C54H71ClN14O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-P5VG6I	WO2023222762A1_215	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCn6cc(CNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)c(Cl)c2)CC1	C56H75ClN14O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-RHTAJV	WO2023222762A1_216	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCn6cc(CNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)c(Cl)c2)CC1	C56H75ClN14O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-5MPXM2	WO2023222762A1_217	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCCn6cc(CNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)c(Cl)c2)CC1	C58H79ClN14O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-M0MNAP	WO2023222762A1_218	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCCn6cc(CNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)c(Cl)c2)CC1	C58H79ClN14O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-23XZ7J	WO2023222762A1_219	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCCCCn6cc(CNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)c(Cl)c2)CC1	C60H83ClN14O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-JC2RGX	WO2023222762A1_220	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCCCCn6cc(CNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)c(Cl)c2)CC1	C60H83ClN14O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-5RSI5E	WO2023222762A1_221	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCNc6cccc7c6CN(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)c(Cl)c2)CC1	C51H70ClN11O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-8A4G8Q	WO2023222762A1_222	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCNc6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)c(Cl)c2)CC1	C51H70ClN11O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-JTMBXQ	WO2023222762A1_223	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCNc6cccc7c6CN(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)c(Cl)c2)CC1	C53H74ClN11O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-X2DPBL	WO2023222762A1_224	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCNc6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)c(Cl)c2)CC1	C53H74ClN11O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-EPO5RM	WO2023222762A1_225	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCCNc6cccc7c6CN(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)c(Cl)c2)CC1	C55H78ClN11O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-B095SC	WO2023222762A1_226	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCCNc6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)c(Cl)c2)CC1	C55H78ClN11O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-RTATIL	WO2023222762A1_227	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCCCCNc6cccc7c6CN(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)c(Cl)c2)CC1	C57H82ClN11O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-IQ4WUH	WO2023222762A1_228	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCCCCNc6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)c(Cl)c2)CC1	C57H82ClN11O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-DARNFT	WO2023222762A1_229	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCn6cc(CN7CCN(c8cccc9c8C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)nn6)ncn5)CC4)C3)c(Cl)c2)CC1	C55H72ClN15O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-EH2ZHU	WO2023222762A1_230	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCn6cc(CN7CCN(c8ccc9c(c8)C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)nn6)ncn5)CC4)C3)c(Cl)c2)CC1	C55H72ClN15O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-H87TS2	WO2023222762A1_233	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCn6cc(CN7CCN(c8cccc9c8C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)nn6)ncn5)CC4)C3)c(Cl)c2)CC1	C57H76ClN15O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-TOG6RQ	WO2023222762A1_234	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCn6cc(CN7CCN(c8ccc9c(c8)C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)nn6)ncn5)CC4)C3)c(Cl)c2)CC1	C57H76ClN15O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-NAXKQD	WO2023222762A1_235	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCn6cc(CN7CCN(c8cccc9c8C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)nn6)ncn5)CC4)C3)c(Cl)c2)CC1	C61H84ClN15O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-I2AEE8	WO2023222762A1_236	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCn6cc(CN7CCN(c8ccc9c(c8)C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)nn6)ncn5)CC4)C3)c(Cl)c2)CC1	C61H84ClN15O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-DRQ230	WO2023222762A1_237	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(CNC(=O)CCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)c(Cl)c2)CC1	C56H70ClN11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-UE5P10	WO2023222762A1_238	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(CNC(=O)CCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)c(Cl)c2)CC1	C56H70ClN11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-538XEU	WO2023222762A1_239	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(CNC(=O)CCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)c(Cl)c2)CC1	C58H74ClN11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-RMDKAN	WO2023222762A1_240	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(CNC(=O)CCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)c(Cl)c2)CC1	C58H74ClN11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-KELM66	WO2023222762A1_241	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(CNC(=O)CCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)c(Cl)c2)CC1	C60H78ClN11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-1G1XCF	WO2023222762A1_242	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(CNC(=O)CCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)c(Cl)c2)CC1	C60H78ClN11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-MX50NV	WO2023222762A1_243	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(CNC(=O)CCCCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)c(Cl)c2)CC1	C62H82ClN11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-DWJC8Z	WO2023222762A1_244	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(CNC(=O)CCCCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)c(Cl)c2)CC1	C62H82ClN11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-WQKYE0	WO2023222762A1_245	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(C(=O)CNCCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)c(Cl)c2)CC1	C60H78ClN11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-VPWFGN	WO2023222762A1_246	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(C(=O)NCCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)c(Cl)c2)CC1	C59H76ClN11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-1XQCJI	WO2023222762A1_247	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(C(=O)CNCCCCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)c(Cl)c2)CC1	C62H82ClN11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-SXFSN4	WO2023222762A1_248	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(C(=O)NCCCCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)c(Cl)c2)CC1	C61H80ClN11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-IA6B2M	WO2023222762A1_249	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(C(=O)CNCCCCCCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)c(Cl)c2)CC1	C64H86ClN11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-AA1MX4	WO2023222762A1_250	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(C(=O)NCCCCCCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)c(Cl)c2)CC1	C63H84ClN11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-E10Z46	WO2023222762A1_251	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(C(=O)CNCCCCCCCCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)c(Cl)c2)CC1	C66H90ClN11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-H611X8	WO2023222762A1_252	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(C(=O)NCCCCCCCCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)c(Cl)c2)CC1	C65H88ClN11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-CBT45V	WO2023222762A1_253	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cn(CCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)c(Cl)c2)CC1	C54H72ClN13O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-ERNENZ	WO2023222762A1_254	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cn(CCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)c(Cl)c2)CC1	C54H72ClN13O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-JZF8V2	WO2023222762A1_255	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cn(CCCCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)c(Cl)c2)CC1	C56H76ClN13O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-0XJRAR	WO2023222762A1_256	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cn(CCCCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)c(Cl)c2)CC1	C56H76ClN13O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-PGDY6E	WO2023222762A1_257	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cn(CCCCCCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)c(Cl)c2)CC1	C58H80ClN13O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-ZMTRWG	WO2023222762A1_258	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cn(CCCCCCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)c(Cl)c2)CC1	C58H80ClN13O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-3Z86PS	WO2023222762A1_259	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cn(CCCCCCCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)c(Cl)c2)CC1	C59H82ClN13O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-0ER7GP	WO2023222762A1_260	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cn(CCCCCCCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)c(Cl)c2)CC1	C59H82ClN13O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-MFJA3U	WO2023222762A1_261	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCOCCOCCNc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)cc2Cl)CC1	C49H64ClN11O8	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-QEG4AV	WO2023222762A1_262	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCOCCOCCOCCNc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)cc2Cl)CC1	C51H68ClN11O9	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-JP1L7E	WO2023222762A1_263	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCOCCOCCOCCOCCNc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)cc2Cl)CC1	C53H72ClN11O10	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-TXPTH0	WO2023222762A1_264	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCNCCOCCOCCOCCOCCNc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)cc2Cl)CC1	C55H77ClN12O10	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-MWUCZ5	WO2023222762A1_265	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCn6cc(CNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2Cl)CC1	C54H71ClN14O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-QJ3T9E	WO2023222762A1_266	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCn6cc(CNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2Cl)CC1	C54H71ClN14O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-0VMNA0	WO2023222762A1_267	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCn6cc(CNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2Cl)CC1	C56H75ClN14O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-HBR1MF	WO2023222762A1_268	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCn6cc(CNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2Cl)CC1	C56H75ClN14O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-6ZCHBW	WO2023222762A1_269	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCCn6cc(CNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2Cl)CC1	C58H79ClN14O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-YU52T0	WO2023222762A1_270	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCCn6cc(CNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2Cl)CC1	C58H79ClN14O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-WTHH9P	WO2023222762A1_271	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCCCCn6cc(CNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2Cl)CC1	C60H83ClN14O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-TWN4IR	WO2023222762A1_272	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCCCCn6cc(CNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2Cl)CC1	C60H83ClN14O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-QMOLQ6	WO2023222762A1_273	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCNc6cccc7c6CN(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)cc2Cl)CC1	C51H70ClN11O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-PV5JL6	WO2023222762A1_274	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCNc6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)cc2Cl)CC1	C51H70ClN11O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-CRK0RJ	WO2023222762A1_275	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCNc6cccc7c6CN(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)cc2Cl)CC1	C53H74ClN11O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-7G0DLG	WO2023222762A1_276	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCNc6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)cc2Cl)CC1	C53H74ClN11O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-9K6GXO	WO2023222762A1_277	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCCNc6cccc7c6CN(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)cc2Cl)CC1	C55H78ClN11O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-HK2NJT	WO2023222762A1_278	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCCNc6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)cc2Cl)CC1	C55H78ClN11O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-4I7CXD	WO2023222762A1_279	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCCCCNc6cccc7c6CN(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)cc2Cl)CC1	C57H82ClN11O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-X72S5M	WO2023222762A1_280	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCCCCNc6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)cc2Cl)CC1	C57H82ClN11O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-BD4LGS	WO2023222762A1_281	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCn6cc(CN7CCN(c8cccc9c8C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)nn6)ncn5)CC4)C3)cc2Cl)CC1	C55H72ClN15O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-SF4ERH	WO2023222762A1_282	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCn6cc(CN7CCN(c8ccc9c(c8)C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)nn6)ncn5)CC4)C3)cc2Cl)CC1	C55H72ClN15O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-S96ZN9	WO2023222762A1_285	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCn6cc(CN7CCN(c8cccc9c8C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)nn6)ncn5)CC4)C3)cc2Cl)CC1	C57H76ClN15O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-CBCX88	WO2023222762A1_286	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCn6cc(CN7CCN(c8ccc9c(c8)C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)nn6)ncn5)CC4)C3)cc2Cl)CC1	C57H76ClN15O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-DPI55H	WO2023222762A1_287	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCn6cc(CN7CCN(c8cccc9c8C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)nn6)ncn5)CC4)C3)cc2Cl)CC1	C61H84ClN15O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-S27H8M	WO2023222762A1_288	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCn6cc(CN7CCN(c8ccc9c(c8)C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)nn6)ncn5)CC4)C3)cc2Cl)CC1	C61H84ClN15O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-3C32DL	WO2023222762A1_289	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(CNC(=O)CCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2Cl)CC1	C56H70ClN11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-KD1WS3	WO2023222762A1_290	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(CNC(=O)CCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2Cl)CC1	C56H70ClN11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-1BDSJK	WO2023222762A1_291	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(CNC(=O)CCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2Cl)CC1	C58H74ClN11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-LX4KI5	WO2023222762A1_292	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(CNC(=O)CCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2Cl)CC1	C58H74ClN11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-S62P06	WO2023222762A1_293	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(CNC(=O)CCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2Cl)CC1	C60H78ClN11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-OZPCEI	WO2023222762A1_294	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(CNC(=O)CCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2Cl)CC1	C60H78ClN11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-6ZG7UJ	WO2023222762A1_295	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(CNC(=O)CCCCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2Cl)CC1	C62H82ClN11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-9MZEYY	WO2023222762A1_296	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(CNC(=O)CCCCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2Cl)CC1	C62H82ClN11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-P53POX	WO2023222762A1_297	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(C(=O)NCCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2Cl)CC1	C59H76ClN11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-26XNCP	WO2023222762A1_298	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(C(=O)NCCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2Cl)CC1	C59H76ClN11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-4BUST7	WO2023222762A1_299	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(C(=O)NCCCCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2Cl)CC1	C61H80ClN11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-VUUDAW	WO2023222762A1_300	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(C(=O)NCCCCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2Cl)CC1	C61H80ClN11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-YRZQVA	WO2023222762A1_301	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(C(=O)NCCCCCCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2Cl)CC1	C63H84ClN11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-HYV53W	WO2023222762A1_302	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(C(=O)NCCCCCCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2Cl)CC1	C63H84ClN11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-20IC0O	WO2023222762A1_303	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(C(=O)NCCCCCCCCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2Cl)CC1	C65H88ClN11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-KAJ0M6	WO2023222762A1_304	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(C(=O)NCCCCCCCCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2Cl)CC1	C65H88ClN11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-7HK0DZ	WO2023222762A1_305	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cn(CCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2Cl)CC1	C54H72ClN13O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-CXSM83	WO2023222762A1_306	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cn(CCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2Cl)CC1	C54H72ClN13O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-QS049J	WO2023222762A1_307	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cn(CCCCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2Cl)CC1	C56H76ClN13O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-RC2GCC	WO2023222762A1_308	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cn(CCCCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2Cl)CC1	C56H76ClN13O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-LUTLUK	WO2023222762A1_309	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cn(CCCCCCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2Cl)CC1	C58H80ClN13O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-PYIV01	WO2023222762A1_310	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cn(CCCCCCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2Cl)CC1	C58H80ClN13O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-CTBX26	WO2023222762A1_311	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cn(CCCCCCCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2Cl)CC1	C59H82ClN13O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-AI31A0	WO2023222762A1_312	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cn(CCCCCCCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2Cl)CC1	C59H82ClN13O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-ASVB5Q	WO2023222762A1_313	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCOCCOCCNc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)cc2)CC1	C49H65N11O8	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-9LN7EF	WO2023222762A1_314	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCOCCOCCOCCNc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)cc2)CC1	C51H69N11O9	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-QXVXQ9	SCHEMBL26656830	N-[3-[[6-[4-[4-[(4,4-dimethylpiperidin-1-yl)methyl]phenyl]-2-oxo-1,4,9-triazaspiro[5.5]undecan-9-yl]pyrimidin-4-yl]amino]propyl]-3-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethoxy]propanamide; SCHEMBL30665461	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCOCCOCCOCCOCCNc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)cc2)CC1	C53H73N11O10	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-CUHEB5	SCHEMBL26656843	N-[3-[[6-[4-[4-[(4,4-dimethylpiperidin-1-yl)methyl]phenyl]-2-oxo-1,4,9-triazaspiro[5.5]undecan-9-yl]pyrimidin-4-yl]amino]propyl]-3-[2-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]propanamide; SCHEMBL30665469	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCOCCOCCOCCOCCOCCNc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)cc2)CC1	C55H77N11O11	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-Y8954D	SCHEMBL26656814	N-[3-[[6-[4-[4-[(4,4-dimethylpiperidin-1-yl)methyl]phenyl]-2-oxo-1,4,9-triazaspiro[5.5]undecan-9-yl]pyrimidin-4-yl]amino]propyl]-9-[4-[[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]methyl]triazol-1-yl]nonanamide; SCHEMBL30665447	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCn6cc(CNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2)CC1	C54H72N14O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-TBTNFJ	WO2023222762A1_318	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCn6cc(CNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2)CC1	C54H72N14O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-0Z37DX	SCHEMBL30665452	N-[3-[[6-[4-[4-[(4,4-dimethylpiperidin-1-yl)methyl]phenyl]-2-oxo-1,4,9-triazaspiro[5.5]undecan-9-yl]pyrimidin-4-yl]amino]propyl]-11-[4-[[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]methyl]triazol-1-yl]undecanamide	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCn6cc(CNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2)CC1	C56H76N14O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-8VJJA8	WO2023222762A1_320	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCn6cc(CNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2)CC1	C56H76N14O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-2GI94N	WO2023222762A1_321	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCCn6cc(CNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2)CC1	C58H80N14O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-ZUS070	WO2023222762A1_322	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCCn6cc(CNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2)CC1	C58H80N14O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-FB8G3U	WO2023222762A1_323	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCCCCn6cc(CNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2)CC1	C60H84N14O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-3FSX1G	WO2023222762A1_324	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCCCCn6cc(CNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2)CC1	C60H84N14O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-8ZGA67	SCHEMBL26656837	N-[3-[[6-[4-[4-[(4,4-dimethylpiperidin-1-yl)methyl]phenyl]-2-oxo-1,4,9-triazaspiro[5.5]undecan-9-yl]pyrimidin-4-yl]amino]propyl]-9-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]nonanamide; SCHEMBL30665472	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCNc6cccc7c6CN(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)cc2)CC1	C51H71N11O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-755KKX	WO2023222762A1_326	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCNc6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)cc2)CC1	C51H71N11O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-C9WQEU	SCHEMBL30665450	N-[3-[[6-[4-[4-[(4,4-dimethylpiperidin-1-yl)methyl]phenyl]-2-oxo-1,4,9-triazaspiro[5.5]undecan-9-yl]pyrimidin-4-yl]amino]propyl]-11-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]undecanamide	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCNc6cccc7c6CN(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)cc2)CC1	C53H75N11O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-XC6OVX	WO2023222762A1_328	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCNc6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)cc2)CC1	C53H75N11O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-N5OIA4	WO2023222762A1_329	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCCNc6cccc7c6CN(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)cc2)CC1	C55H79N11O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-AK9FVA	WO2023222762A1_330	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCCNc6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)cc2)CC1	C55H79N11O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-D5CURZ	SCHEMBL26656798	N-[3-[[6-[4-[4-[(4,4-dimethylpiperidin-1-yl)methyl]phenyl]-2-oxo-1,4,9-triazaspiro[5.5]undecan-9-yl]pyrimidin-4-yl]amino]propyl]-15-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]pentadecanamide; SCHEMBL30665451	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCCCCNc6cccc7c6CN(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)cc2)CC1	C57H83N11O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-FI3EIM	WO2023222762A1_332	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCCCCNc6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)ncn5)CC4)C3)cc2)CC1	C57H83N11O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-E4XSY4	WO2023222762A1_333	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCn6cc(CN7CCN(c8cccc9c8C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)nn6)ncn5)CC4)C3)cc2)CC1	C55H73N15O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-IDPMOV	WO2023222762A1_334	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCn6cc(CN7CCN(c8ccc9c(c8)C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)nn6)ncn5)CC4)C3)cc2)CC1	C55H73N15O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-SYSXRZ	WO2023222762A1_337	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCn6cc(CN7CCN(c8cccc9c8C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)nn6)ncn5)CC4)C3)cc2)CC1	C57H77N15O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-8DG10S	WO2023222762A1_338	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCn6cc(CN7CCN(c8ccc9c(c8)C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)nn6)ncn5)CC4)C3)cc2)CC1	C57H77N15O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-GEZED1	WO2023222762A1_339	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCn6cc(CN7CCN(c8cccc9c8C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)nn6)ncn5)CC4)C3)cc2)CC1	C61H85N15O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-DR8CT5	WO2023222762A1_340	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCCCNC(=O)CCCCCCCCCCCn6cc(CN7CCN(c8ccc9c(c8)C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)nn6)ncn5)CC4)C3)cc2)CC1	C61H85N15O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-S3LGGC	WO2023222762A1_341	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(CNC(=O)CCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2)CC1	C56H71N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-JFDY2Y	WO2023222762A1_342	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(CNC(=O)CCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2)CC1	C56H71N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-EQVYWE	WO2023222762A1_343	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(CNC(=O)CCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2)CC1	C58H75N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-SZVHA3	WO2023222762A1_344	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(CNC(=O)CCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2)CC1	C58H75N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-ELPGI8	WO2023222762A1_345	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(CNC(=O)CCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2)CC1	C60H79N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-YHILYX	WO2023222762A1_346	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(CNC(=O)CCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2)CC1	C60H79N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-1XF95R	WO2023222762A1_347	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(CNC(=O)CCCCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2)CC1	C62H83N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-AIGST9	WO2023222762A1_348	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(CNC(=O)CCCCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2)CC1	C62H83N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-Y4RZDA	WO2023222762A1_349	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(C(=O)NCCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2)CC1	C59H77N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-P0Q062	WO2023222762A1_350	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(C(=O)NCCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2)CC1	C59H77N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-NB7V6T	WO2023222762A1_351	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(C(=O)NCCCCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2)CC1	C61H81N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-6UG2DN	WO2023222762A1_352	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(C(=O)NCCCCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2)CC1	C61H81N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-P2F2K5	WO2023222762A1_353	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(C(=O)NCCCCCCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2)CC1	C63H85N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-AD4599	WO2023222762A1_354	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(C(=O)NCCCCCCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2)CC1	C63H85N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-Z0TN9D	WO2023222762A1_355	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(C(=O)NCCCCCCCCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2)CC1	C65H89N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-GKJJM7	WO2023222762A1_356	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cccc(C(=O)NCCCCCCCCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)c6)ncn5)CC4)C3)cc2)CC1	C65H89N11O6	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-CZQRAI	WO2023222762A1_357	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cn(CCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2)CC1	C54H73N13O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-5HMD3C	WO2023222762A1_358	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cn(CCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2)CC1	C54H73N13O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-C5OJLM	WO2023222762A1_359	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cn(CCCCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2)CC1	C56H77N13O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-9WWODS	WO2023222762A1_360	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cn(CCCCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2)CC1	C56H77N13O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-S1G36V	WO2023222762A1_361	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cn(CCCCCCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2)CC1	C58H81N13O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-Z7TBKF	WO2023222762A1_362	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cn(CCCCCCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2)CC1	C58H81N13O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-9XTSKU	WO2023222762A1_363	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cn(CCCCCCCCCCCCCCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2)CC1	C59H83N13O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-56XYBX	WO2023222762A1_364	.	CC1(C)CCN(Cc2ccc(N3CC(=O)NC4(CCN(c5cc(NCc6cn(CCCCCCCCCCCCCCCCCNc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)nn6)ncn5)CC4)C3)cc2)CC1	C59H83N13O5	METTL14;METTL3	Q9HCE5/Q86U44	CRBN	WO-2023222762-A1
TPD-C8BJHO	WO2023227080A1_1	.	CN1CCN([C@@H]2CCCN(c3c(F)cc(C(N)=O)c4[nH]c(-c5ccc(C6CCN(CC7CCN(c8ccc(C(=O)N[C@H]9CCC(=O)NC9=O)nc8)CC7)CC6)cc5)cc34)C2)C1=O	C46H55FN10O5	BTK	Q06187	CRBN	WO-2023227080-A1
TPD-ZJR7L6	SCHEMBL26697126	2-[4-[1-[[1-[4-[(2,6-dioxopiperidin-3-yl)amino]phenyl]piperidin-4-yl]methyl]piperidin-4-yl]phenyl]-5-fluoro-4-[(3R)-3-(3-methyl-2-oxoimidazolidin-1-yl)piperidin-1-yl]-1H-indole-7-carboxamide	CN1CCN([C@@H]2CCCN(c3c(F)cc(C(N)=O)c4[nH]c(-c5ccc(C6CCN(CC7CCN(c8ccc(NC9CCC(=O)NC9=O)cc8)CC7)CC6)cc5)cc34)C2)C1=O	C46H56FN9O4	BTK	Q06187	CRBN	WO-2023227080-A1
TPD-QKLET1	SCHEMBL26697150	2-[4-[1-[[1-[4-(2,6-dioxopiperidin-3-yl)phenyl]piperidin-4-yl]methyl]piperidin-4-yl]phenyl]-5-fluoro-4-[(3R)-3-(3-methyl-2-oxoimidazolidin-1-yl)piperidin-1-yl]-1H-indole-7-carboxamide	CN1CCN([C@@H]2CCCN(c3c(F)cc(C(N)=O)c4[nH]c(-c5ccc(C6CCN(CC7CCN(c8ccc(C9CCC(=O)NC9=O)cc8)CC7)CC6)cc5)cc34)C2)C1=O	C46H55FN8O4	BTK	Q06187	CRBN	WO-2023227080-A1
TPD-K8QNT9	WO2023227080A1_4	2-[4-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperidin-4-yl]phenyl]-5-fluoro-4-[(3R)-3-(3-methyl-2-oxoimidazolidin-1-yl)piperidin-1-yl]-1H-indole-7-carboxamide	CN1CCN([C@@H]2CCCN(c3c(F)cc(C(N)=O)c4[nH]c(-c5ccc(C6CCN(CC7CCN(c8cc9c(cc8F)C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)CC6)cc5)cc34)C2)C1=O	C48H53F2N9O6	BTK	Q06187	CRBN	WO-2023227080-A1
TPD-WXT05P	WO2023227080A1_5	2-[4-[1-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]piperidin-4-yl]methyl]piperidin-4-yl]phenyl]-5-fluoro-4-[(3R)-3-(3-methyl-2-oxoimidazolidin-1-yl)piperidin-1-yl]-1H-indole-7-carboxamide	CN1CCN([C@@H]2CCCN(c3c(F)cc(C(N)=O)c4[nH]c(-c5ccc(C6CCN(CC7CCN(c8ccc(N9CCC(=O)NC9=O)cc8)CC7)CC6)cc5)cc34)C2)C1=O	C45H54FN9O4	BTK	Q06187	CRBN	WO-2023227080-A1
TPD-34WXS1	WO2023227080A1_6	.	NC(=O)c1cc(F)c(N2CCC[C@@H](N3CCOC3=O)C2)c2cc(-c3ccc(C4CCN(CC5CCN(c6ccc(C(=O)N[C@H]7CCC(=O)NC7=O)nc6)CC5)CC4)cc3)[nH]c12	C45H52FN9O6	BTK	Q06187	CRBN	WO-2023227080-A1
TPD-29AR17	WO2023227080A1_7	2-[4-[1-[1-[6-[[(3S)-2,6-dioxopiperidin-3-yl]carbamoyl]pyridin-3-yl]azetidin-3-yl]piperidin-4-yl]phenyl]-5-fluoro-4-[(3R)-3-(3-methyl-2-oxoimidazolidin-1-yl)piperidin-1-yl]-1H-indole-7-carboxamide	CN1CCN([C@@H]2CCCN(c3c(F)cc(C(N)=O)c4[nH]c(-c5ccc(C6CCN(C7CN(c8ccc(C(=O)N[C@H]9CCC(=O)NC9=O)nc8)C7)CC6)cc5)cc34)C2)C1=O	C43H49FN10O5	BTK	Q06187	CRBN	WO-2023227080-A1
TPD-UGPB3Q	WO2023227080A1_8	.	CN1CCN([C@@H]2CCCN(c3c(F)cc(C(N)=O)c4[nH]c(-c5ccc(C6CCN(C[C@@H]7CCN(c8ccc(C(=O)N[C@H]9CCC(=O)NC9=O)nc8)C7)CC6)cc5)cc34)C2)C1=O	C45H53FN10O5	BTK	Q06187	CRBN	WO-2023227080-A1
TPD-FHRSFA	WO2023227080A1_9	.	CN1CCN([C@@H]2CCCN(c3c(F)cc(C(N)=O)c4[nH]c(-c5ccc(C6CCN(C[C@@H]7CCN(c8ccc(N9CCC(=O)NC9=O)cc8)C7)CC6)cc5)cc34)C2)C1=O	C44H52FN9O4	BTK	Q06187	CRBN	WO-2023227080-A1
TPD-3BRPMN	WO2023227080A1_10	.	NC(=O)c1cc(F)c(N2CCCCC2)c2cc(-c3ccc(C4CCN(C[C@@H]5CCN(c6ccc(C(=O)N[C@H]7CCC(=O)NC7=O)nc6)C5)CC4)cc3)[nH]c12	C41H47FN8O4	BTK	Q06187	CRBN	WO-2023227080-A1
TPD-NXSE1E	WO2023227080A1_11	2-[4-[1-[[(3S)-1-[4-(2,4-dioxo-1,3-diazinan-1-yl)phenyl]pyrrolidin-3-yl]methyl]piperidin-4-yl]phenyl]-5-fluoro-4-piperidin-1-yl-1H-indole-7-carboxamide	NC(=O)c1cc(F)c(N2CCCCC2)c2cc(-c3ccc(C4CCN(C[C@@H]5CCN(c6ccc(N7CCC(=O)NC7=O)cc6)C5)CC4)cc3)[nH]c12	C40H46FN7O3	BTK	Q06187	CRBN	WO-2023227080-A1
TPD-01I4G0	WO2023227080A1_12	.	CN1CCN([C@@H]2CCCN(c3c(F)cc(C(N)=O)c4[nH]c(-c5ccc(C6CCN(CC7CCN(c8ncc(C(=O)N[C@H]9CCC(=O)NC9=O)s8)CC7)CC6)cc5)cc34)C2)C1=O	C44H53FN10O5S	BTK	Q06187	CRBN	WO-2023227080-A1
TPD-JXZLW9	WO2023227080A1_13	.	CN1CCN([C@@H]2CCCN(c3c(F)cc(C(N)=O)c4[nH]c(-c5ccc(C6CCN(CC7CCN(c8ncc(-c9ccc(=O)[nH]n9)cc8C(F)(F)F)CC7)CC6)cc5)cc34)C2)C1=O	C45H50F4N10O3	BTK	Q06187	CRBN	WO-2023227080-A1
TPD-2ERCSC	WO2023227080A1_14	.	CN1CCN([C@@H]2CCCN(c3c(F)cc(C(N)=O)c4[nH]c(-c5ccc(N6CCN(CC7CCN(c8ccc(C(=O)N[C@H]9CCC(=O)NC9=O)nc8)CC7)CC6)cc5)cc34)C2)C1=O	C45H54FN11O5	BTK	Q06187	CRBN	WO-2023227080-A1
TPD-693BH1	WO2023227080A1_15	.	CN1CCN([C@@H]2CCCN(c3c(F)cc(C(N)=O)c4[nH]c(-c5ccc(N6CCC(CN7CCN(c8ccc(N9CCC(=O)NC9=O)cc8)CC7)CC6)cc5)cc34)C2)C1=O	C44H53FN10O4	BTK	Q06187	CRBN	WO-2023227080-A1
TPD-P9VPCB	WO2023227080A1_16	2-[4-[4-[[1-[6-[[(3S)-2,6-dioxopiperidin-3-yl]carbamoyl]pyridin-3-yl]azetidin-3-yl]methyl]piperazin-1-yl]phenyl]-5-fluoro-4-[(3R)-3-(3-methyl-2-oxoimidazolidin-1-yl)piperidin-1-yl]-1H-indole-7-carboxamide	CN1CCN([C@@H]2CCCN(c3c(F)cc(C(N)=O)c4[nH]c(-c5ccc(N6CCN(CC7CN(c8ccc(C(=O)N[C@H]9CCC(=O)NC9=O)nc8)C7)CC6)cc5)cc34)C2)C1=O	C43H50FN11O5	BTK	Q06187	CRBN	WO-2023227080-A1
TPD-9MAQI1	SCHEMBL26697108	2-[4-[4-[[4-[6-[[(3S)-2,6-dioxopiperidin-3-yl]carbamoyl]pyridin-3-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]-5-fluoro-4-[(3R)-3-(3-methyl-2-oxoimidazolidin-1-yl)piperidin-1-yl]-1H-indole-7-carboxamide	CN1CCN([C@@H]2CCCN(c3c(F)cc(C(N)=O)c4[nH]c(-c5ccc(N6CCC(CN7CCN(c8ccc(C(=O)N[C@H]9CCC(=O)NC9=O)nc8)CC7)CC6)cc5)cc34)C2)C1=O	C45H54FN11O5	BTK	Q06187	CRBN	WO-2023227080-A1
TPD-SE44OS	WO2023227080A1_18	.	COc1cc(N2CCN(CC3CCN(c4ccc(-c5cc6c(N7CCC[C@@H](N8CCN(C)C8=O)C7)c(F)cc(C(N)=O)c6[nH]5)cc4)CC3)CC2)ccc1C(=O)N[C@H]1CCC(=O)NC1=O	C47H57FN10O6	BTK	Q06187	CRBN	WO-2023227080-A1
TPD-H2CNMG	WO2023227080A1_19	.	CN1CCN([C@@H]2CCCN(c3c(F)cc(C(N)=O)c4[nH]c(-c5ccc(C6CCN(CC7CCN(c8ccc(C(=O)N[C@H]9CCC(=O)NC9=O)nc8)CC7)CC6)cc5)c(Cl)c34)C2)C1=O	C46H54ClFN10O5	BTK	Q06187	CRBN	WO-2023227080-A1
TPD-OBJEHD	WO2023227080A1_20	.	CN1CCN([C@@H]2CCCN(c3c(F)cc(C(N)=O)c4[nH]c(-c5ccc(N6CCN(CC7CN(c8ccc(C9CCC(=O)NC9=O)cc8)C7)CC6)nc5)cc34)C2)C1=O	C42H49FN10O4	BTK	Q06187	CRBN	WO-2023227080-A1
TPD-04TC66	WO2023227080A1_21	.	CN1CCN([C@@H]2CCCN(c3c(F)cc(C(N)=O)c4[nH]c(-c5ccc(N6CCN(C7CN(c8ccc(C(=O)N[C@H]9CCC(=O)NC9=O)nc8)C7)CC6)nc5)cc34)C2)C1=O	C41H47FN12O5	BTK	Q06187	CRBN	WO-2023227080-A1
TPD-XVMGX2	WO2023227080A1_22	.	CN1CCN([C@@H]2CCCN(c3c(F)cc(C(N)=O)c4[nH]c(-c5ccc(C6CCN(CC7CCN(c8ccc(NC9CCC(=O)NC9=O)cc8F)CC7)CC6)cc5)cc34)C2)C1=O	C46H55F2N9O4	BTK	Q06187	CRBN	WO-2023227080-A1
TPD-1DH8ST	WO2023227080A1_23	.	CN1CCN([C@@H]2CCCN(c3c(F)cc(C(N)=O)c4[nH]c(-c5ccc(N6CCN(CC7CCN(c8ccc(NC9CCC(=O)NC9=O)cc8F)CC7)CC6)nc5)cc34)C2)C1=O	C44H53F2N11O4	BTK	Q06187	CRBN	WO-2023227080-A1
TPD-4PTMYJ	WO2023227080A1_24	2-[6-[4-[[1-[6-[[(3S)-2,6-dioxopiperidin-3-yl]carbamoyl]pyridin-3-yl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-3-yl]-5-fluoro-4-[(3R)-3-(3-methyl-2-oxoimidazolidin-1-yl)piperidin-1-yl]-1H-indole-7-carboxamide	CN1CCN([C@@H]2CCCN(c3c(F)cc(C(N)=O)c4[nH]c(-c5ccc(N6CCN(CC7CCN(c8ccc(C(=O)N[C@H]9CCC(=O)NC9=O)nc8)CC7)CC6)nc5)cc34)C2)C1=O	C44H53FN12O5	BTK	Q06187	CRBN	WO-2023227080-A1
TPD-WXHM88	WO2023227080A1_25	.	CN1CCN([C@@H]2CCCN(c3c(F)cc(C(N)=O)c4[nH]c(-c5ccc(N6CCN(CC7CN(c8ccc(C(=O)N[C@H]9CCC(=O)NC9=O)nc8)C7)CC6)nc5)cc34)C2)C1=O	C42H49FN12O5	BTK	Q06187	CRBN	WO-2023227080-A1
TPD-D9PQDK	WO2023233024A1_122	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3=CSC(C4=CC=C(C(=O)NC56CC7CC(CC(NCC(=O)N8CC9=CC=C(F)C=C9C8)(C7)C5)C6)C=C4)=C3)C(C)(C)C)C=C2)SC=N1	C54H60FN7O6S2	DPP9	Q86TI2	VHL	WO-2023233024-A1
TPD-XERRG8	SCHEMBL27358793	(2S,4R)-1-[(2S)-2-[[4-[4-[[3-[[2-(5-fluoro-1,3-dihydroisoindol-2-yl)-2-oxoethyl]amino]-1-adamantyl]carbamoyl]phenyl]benzoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3=CC=C(C4=CC=C(C(=O)NC56CC7CC(CC(NCC(=O)N8CC9=CC=C(F)C=C9C8)(C7)C5)C6)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C56H62FN7O6S	DPP9	Q86TI2	VHL	WO-2023233024-A1
TPD-BQA8T4	SCHEMBL30685227	(2S,4R)-1-[(2S)-2-[3-[2-[2-[3-[[3-[[2-(5-fluoro-1,3-dihydroisoindol-2-yl)-2-oxoethyl]amino]-1-adamantyl]amino]-3-oxopropoxy]ethoxy]ethoxy]propanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCOCCOCCOCCC(=O)NC34CC5CC(CC(NCC(=O)N6CC7=CC=C(F)C=C7C6)(C5)C3)C4)C(C)(C)C)C=C2)SC=N1	C52H70FN7O9S	DPP9	Q86TI2	VHL	WO-2023233024-A1
TPD-B794C9	WO2023233024A1_125	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCOCCOC3=CC=C(C4=CC=C(C(=O)NC56CC7CC(CC(NCC(=O)N8CC9=CC=C(F)C=C9C8)(C7)C5)C6)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C60H70FN7O8S	DPP9	Q86TI2	VHL	WO-2023233024-A1
TPD-8G0NZN	BDBM708314	US20240423977, Example I-1; BDBM708342; US20240423977, Example I-1; US20240423977, Example I-22	COC1=CC2=NN(C3CC4(CCN(C(=O)C5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C42H41F3N8O7	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-FWSKSI	BDBM708335	US20240423977, Example I-10; US20240423977, Example I-10	O=C1CCC(N2C(=O)C3=CC=C(N4CCC(C(=O)N5CCC6(CC5)CC(N5C=C7C=C(NC(=O)C8=CC=CC(C(F)(F)F)=N8)C(N8CC[C@@H](O)C8)=CC7=N5)C6)CC4)C=C3C2=O)C(=O)N1	C45H46F3N9O7	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-A3PBCX	WO2023241644A1_I-12F	.	CC(O)(C1=CC2=NN(C3CC4(CCN(C(=O)C5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1)C(F)(F)F	C44H42F6N8O7	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-ND0W2P	BDBM708319	US20240423977, Example I-13; US20240423977, Example I-13	COC1=CC2=NN(C3CC4(CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C42H43F3N8O6	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-48GVQP	BDBM708337	US20240423977, Example I-14; US20240423977, Example I-14	COC1=CC2=NN(C3CC4(C3)CN(C(=O)C3CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC3)C4)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C40H37F3N8O7	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-Y2DF95	BDBM708338	US20240423977, Example I-16; US20240423977, Example I-16	COC1=CC2=NN(C3CC4(CCC(NC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C42H43F3N8O6	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-G8ZC41	BDBM708339	US20240423977, Example I-17; US20240423977, Example I-17	COC1=CC2=NN(C3CC4(CCN(C(=O)C5CC6(C5)CN(C5=CC7=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)C3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C43H41F3N8O7	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-ETKOOU	BDBM708340	US20240423977, Example I-19; US20240423977, Example I-19	COC1=CC2=NN(C3CCC4(CC3)CN(C(=O)C3CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC3)C4)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C42H41F3N8O7	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-ZSIOAF	BDBM708315	US20240423977, Example I-2; US20240423977, Example I-2	COC1=CC2=NN(C3CC4(CCN(CC(=O)N5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C42H42F3N9O7	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-MMU82V	BDBM708341	US20240423977, Example I-20; US20240423977, Example I-20	COC1=CC2=NN(C3CC4(CCC(C(=O)N5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C42H41F3N8O7	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-JDL4C9	BDBM708332	US20240423977, Example I-5; US20240423977, Example I-5	CC(C)(O)C1=CC2=NN(C3CC4(CCN(C(=O)C5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C44H45F3N8O7	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-907B5D	BDBM708344	US20240423977, Example I-24; US20240423977, Example I-24	COC1=CC2=NN(C3CC4(CCN(C5CC6(CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)C5)CC4)C3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C44H45F3N8O6	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-QIHRYY	BDBM708345	US20240423977, Example I-25; US20240423977, Example I-25	COC1=CC2=NN(C3CC4(CCN(C(=O)C5CCN(C6=CC=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)C3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C42H41F3N8O7	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-UXMMPZ	BDBM708346	US20240423977, Example I-26; US20240423977, Example I-26	COC1=CC2=NN(C3CC4(CCN(C(=O)C5CCC6(CC5)CN(C5=CC7=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C6)CC4)C3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C45H45F3N8O7	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-CX4IK8	BDBM708347	US20240423977, Example I-27; US20240423977, Example I-27	COC1=CC2=NN(C3CCC4(CC3)CCN(C(=O)C3CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC3)CC4)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C44H45F3N8O7	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-J8WPWV	BDBM708348	US20240423977, Example I-28; US20240423977, Example I-28	COC1=CC2=NN([C@H]3C[C@@H]4CN(C(=O)C5CCN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C[C@@H]4C3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C41H39F3N8O7	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-0RK4YX	BDBM708349	US20240423977, Example I-29; US20240423977, Example I-29	COC1=CC2=NN(C3CC4(CCN(C(=O)[C@H]5CC[C@H](C(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)(C)C)CC5)CC4)C3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C54H64F3N9O7S	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-IIBCFL	BDBM708316	US20240423977, Example I-3; US20240423977, Example I-3	COC1=CC2=NN(C3CC4(CCN(C(=O)[C@H]5CC[C@H](CNC6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C44H45F3N8O7	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-66CMVH	BDBM708350	US20240423977, Example I-30; US20240423977, Example I-30	COC1=CC2=C(C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1)CN(C1CC3(CCN(C(=O)C4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)C1)C2=O	C43H42F3N7O8	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-O56OJB	BDBM708351	US20240423977, Example I-31; US20240423977, Example I-31	COC1=CC2=NN(C3CC4(CCN(C(=O)[C@H]5CC[C@H](OC6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C43H42F3N7O8	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-3F386C	WO2023241644A1_I-32	.	COC1=CC2=NN(C3CC4(CCN(C5=CN(C6CCN(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)C=C5)CC4)C3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C45H44F3N9O6	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-BAY5FQ	BDBM708353	US20240423977, Example I-33; US20240423977, Example I-33	COC1=CC2=NN(C3CC4(CCN(C(=O)C5(O)CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C42H41F3N8O8	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-RWX9XZ	BDBM708354	US20240423977, Example I-34; US20240423977, Example I-34	COC1=CC2=NN(C3CC4(CCN(C(=O)C5(F)CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C42H40F4N8O7	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-BLQMSV	BDBM708355	US20240423977, Example I-35; US20240423977, Example I-35	COC1=CC2=NN(C3CC4(CCN(C(=O)C5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5(F)F)CC4)C3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C42H39F5N8O7	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-1DIW1Y	BDBM708356	US20240423977, Example I-36; US20240423977, Example I-36	COC1=CC2=NN(C3CC4(CCN(C(=O)C5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C3)C=C2C=C1NC(=O)C1=COC(C2=CC=NC(C)=C2)=N1	C45H45N9O8	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-5UI842	BDBM708357	US20240423977, Example I-37; US20240423977, Example I-37	COC1=CC2=NN(C3CC4(CCN(C(=O)C5(C)CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C43H43F3N8O7	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-SKPZF9	BDBM708358	US20240423977, Example I-38; US20240423977, Example I-38	COC1=CC2=NN(C3CC4(CCN(C(=O)C5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C3)C=C2C=C1NC(=O)C1=CC=CC(C)=N1	C42H44N8O7	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-T2Z0GA	BDBM708317	US20240423977, Example I-4; US20240423977, Example I-4	COC1=CC2=NN(C3CC4(CCN(C(=O)[C@H]5CC[C@H](NC6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C43H43F3N8O7	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-4FGHOT	WO2023241644A1_I-41	.	COC1=CC2=NN(C3CC4(CCN(C(=O)C5CCN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)C3)C=C2C=C1NC(=O)C1=CC=CC(N2CCOCC2)=N1	C45H49N9O8	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-988EH4	BDBM708360	US20240423977, Example I-42; US20240423977, Example I-42	COC1=CC2=NN(C3CC4(CCN(C(=O)C5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C3)C=C2C=C1NC(=O)C1=CC=CC(C(F)F)=N1	C42H42F2N8O7	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-AEWO72	BDBM708361	US20240423977, Example I-43; US20240423977, Example I-43	COC1=CC2=NN(C3CC4(CCN(C(=O)C5CCN(C6=CC=C7C(=O)N(C8=NNC(=O)C=C8)C(=O)C7=C6)CC5)CC4)C3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C41H38F3N9O6	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-GMEBA5	BDBM708362	US20240423977, Example I-44; US20240423977, Example I-44	COC1=CC2=NN(C3CC4(CCN(C(=O)C5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C3)C=C2C=C1NC(=O)C1=C2N=C(N3C[C@H]4C[C@@H]3CO4)C=CN2N=C1	C47H49N11O8	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-EE7UXR	BDBM708363	US20240423977, Example I-45; US20240423977, Example I-45	O=C1CCC(N2C(=O)C3=CC=C(N4CCC(C(=O)N5CCC6(CC5)CN(C5=NC7=C(C=C(NC(=O)C8=CC=CC(C(F)(F)F)=N8)C(N8CC[C@@H](O)C8)=N7)O5)C6)CC4)C=C3C2=O)C(=O)N1	C43H43F3N10O8	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-6S3MVO	BDBM708364	US20240423977, Example I-46; US20240423977, Example I-46	COC1=CC2=NN(C3CC4(CCN(C(=O)C5CCN(C6=C(F)C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C3)C=C2C=C1NC(=O)C1=CC=CC(N2CCOCC2)=N1	C45H48FN9O8	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-MKARL5	BDBM708365	US20240423977, Example I-47; US20240423977, Example I-47	COC1=CC2=NN(C3CC4(CCN(C(=O)C5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C3)C=C2C=C1NC(=O)C1=NN(C(F)F)C=C1	C40H41F2N9O7	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-Z84OR6	BDBM708366	US20240423977, Example I-48; US20240423977, Example I-48	O=C1CCC(N2C(=O)C3=CC=C(N4CCC(C(=O)N5CCC6(CC5)CC(N5C=C7C=C(NC(=O)C8=CC=CC(C(F)(F)F)=N8)C(C(=O)O)=CC7=N5)C6)CC4)C=C3C2=O)C(=O)N1	C42H39F3N8O8	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-V8J3RN	BDBM708367	US20240423977, Example I-49; US20240423977, Example I-49	COC1=CC2=NN(C3CC4(CCN(C(=O)C5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C3)C=C2C=C1NC(=O)C1=C2N=C(N3CCN(C)CC3)C=CN2N=C1	C47H52N12O7	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-9OTH6W	BDBM708368	US20240423977, Example I-50; US20240423977, Example I-50	COC1=CC2=NN(C3CC4(CCN(C(=O)C5(F)CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C3)C=C2C=C1NC(=O)C1=CC=CC(N2CCOCC2)=N1	C45H48FN9O8	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-8CI1PN	BDBM708369	US20240423977, Example I-51; US20240423977, Example I-51	COC1=CC2=NN(C3CC4(CCN(C5CCN(C(=O)C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)C3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C42H41F3N8O7	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-9GXK66	BDBM708370	US20240423977, Example I-52; US20240423977, Example I-52	COC1=CC2=NN(C3CC4(CCN(C(=O)C5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C3)C=C2C=C1NC(=O)C1=CC=CC(N2CC3CC2CO3)=N1	C46H49N9O8	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-K61E4B	BDBM708371	US20240423977, Example I-53; US20240423977, Example I-53	O=C1CCC(N2C(=O)C3=CC=C(N4CCC(C(=O)N5CCC6(CC5)CC(N5C=C7C=C(NC(=O)C8=CC=CC(C(F)(F)F)=N8)C(F)=CC7=N5)C6)CC4)C=C3C2=O)C(=O)N1	C41H38F4N8O6	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-A6D11Y	BDBM708372	US20240423977, Example I-54; US20240423977, Example I-54	COC1=CC2=NN(C3CC4(CCN(C(=O)C5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C3)C=C2C=C1NC(=O)C1=COC(N2CCOCC2)=N1	C43H47N9O9	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-YM5BL6	BDBM708373	US20240423977, Example I-55; US20240423977, Example I-55	COC1=CC2=NN(C3CC4(CCN(C(=O)C5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5(F)F)CC4)C3)C=C2C=C1NC(=O)C1=CC=CC(N2CCOCC2)=N1	C45H47F2N9O8	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-ULUGZB	BDBM708374	US20240423977, Example I-56; US20240423977, Example I-56	COC1=CC2=C(C=NN2C2CC3(CCC(C(=O)N4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)C2)C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C42H41F3N8O7	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-XIIHCV	BDBM708375	US20240423977, Example I-57; BDBM708383; US20240423977, Example I-57; US20240423977, Example I-65	COC1=CC2=NN(C3CC4(CCN(C(=O)C5CCN(C6=CC=C7C(=O)N([C@H]8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C42H41F3N8O7	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-YDZ6E0	BDBM708376	US20240423977, Example I-58; BDBM708384; US20240423977, Example I-58; US20240423977, Example I-66	COC1=CC2=NN(C3CC4(CCN(C(=O)C5CCN(C6=CC=C7C(=O)N([C@@H]8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C42H41F3N8O7	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-C838T7	BDBM708377	US20240423977, Example I-59; US20240423977, Example I-59	COC1=CC2=NN(C3CC4(CCN(C(=O)[C@H]5CC[C@H](NC6=CC=C7C(=O)N([C@H]8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C43H43F3N8O7	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-NZXO2V	BDBM708378	US20240423977, Example I-60; US20240423977, Example I-60	COC1=CC2=NN(C3CC4(CCN(C(=O)[C@H]5CC[C@H](NC6=CC=C7C(=O)N([C@@H]8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C43H43F3N8O7	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-386PPX	BDBM708379	US20240423977, Example I-61; US20240423977, Example I-61	COC1=CC2=NN(C3CC4(CCN(C(=O)C5CCN(C6=C(F)C=C7C(=O)N([C@H]8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C42H40F4N8O7	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-97J7SI	BDBM708380	US20240423977, Example I-62; US20240423977, Example I-62	COC1=CC2=NN(C3CC4(CCN(C(=O)C5CCN(C6=C(F)C=C7C(=O)N([C@@H]8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C42H40F4N8O7	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-GRYCMW	BDBM708381	US20240423977, Example I-63; US20240423977, Example I-63	CC(C)(O)C1=CC2=NN(C3CC4(CCN(C(=O)C5CCN(C6=CC=C7C(=O)N([C@H]8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C44H45F3N8O7	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-YLINKF	WO2023241644A1_I-64	.	CC(C)(O)C1=CC2=NN(C3CC4(CCN(C(=O)C5CCN(C6=CC=C7C(=O)N([C@@H]8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C44H45F3N8O7	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-UWNFQ9	BDBM708333	US20240423977, Example I-7; US20240423977, Example I-7	COC1=CC2=NN(C3CC4(CCN(C(=O)C5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)CC5)CC4)C3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C42H43F3N8O6	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-51W0GW	BDBM708318	US20240423977, Example I-8; US20240423977, Example I-8	COC1=CC2=NN(C3CC4(CCN(C(=O)C5CCN(C6=C(F)C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C42H40F4N8O7	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-DGZSLH	WO2023241644A1_I-9	.	O=C1CCC(N2C(=O)C3=CC=C(N4CCC(C(=O)N5CCC6(CC5)CC(N5C=C7C=C(NC(=O)C8=CC=CC(C(F)(F)F)=N8)C(N8CCOCC8)=CC7=N5)C6)CC4)C=C3C2=O)C(=O)N1	C45H46F3N9O7	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-IQMFBY	WO2023241644A1_II-1	.	COC1=CC2=NN(C3CCN(CC(=O)N4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C39H38F3N9O7	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-REXWOT	BDBM708324	US20240423977, Example II-10; US20240423977, Example II-10	COC1=CC2=NN(C3CCN(C(C)C(=O)N4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C40H40F3N9O7	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-BD92SX	WO2023241644A1_II-12	.	COC1=CC2=NN(C3CCN(C4CC5(CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)C4)CC3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C41H41F3N8O6	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-44ZHUO	BDBM708326	US20240423977, Example II-13; US20240423977, Example II-13	COC1=CC2=NN(C3CC4CCC(C3)N4CC(=O)N3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C41H40F3N9O7	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-RVJXY2	BDBM708327	US20240423977, Example II-16; US20240423977, Example II-16	COC1=CC2=NN(C3CCN(C(=O)C4CCN(CC5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C40H39F3N8O7	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-LOP1D3	BDBM708328	US20240423977, Example II-17; US20240423977, Example II-17	COC1=CC2=NN(C3CCN(C4CCN(C(=O)C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C39H37F3N8O7	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-XZQROY	WO2023241644A1_II-2	.	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(C(=O)CN5CCC(N6C=C7C=C(NC(=O)C8=CC=CC(C(F)(F)F)=N8)C(OC(F)(F)F)=CC7=N6)CC5)CC4)C=C3C2=O)C(=O)N1	C39H35F6N9O7	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-D4KEJO	BDBM708331	US20240423977, Example II-20; US20240423977, Example II-20	COC1=CC2=NN(C3CCN(CC(=O)N4CCN(C5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)CC4)CC3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C39H38F3N9O7	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-K26VAB	WO2023241644A1_II-21	.	COC1=CC2=C(C=NN2C2CCN(C3CC4(CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)C3)CC2)C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C41H41F3N8O6	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-4Q0OWR	BDBM708321	US20240423977, Example II-4; US20240423977, Example II-4	COC1=CC2=NN(C3CCN(C(=O)CN4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C39H38F3N9O7	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-6MKE64	BDBM708322	US20240423977, Example II-5; US20240423977, Example II-5	COC1=CC2=NN(C3CCN(CC(=O)N4CCN(C5=C(F)C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C39H37F4N9O7	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-9NDL04	BDBM708323	US20240423977, Example II-6; US20240423977, Example II-6	CC(C)(O)C1=CC2=NN(C3CCN(CC(=O)N4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C41H42F3N9O7	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-DECEQF	BDBM708330	US20240423977, Example II-7; US20240423977, Example II-7	COC1=CC2=NN(C3CCN(CC(=O)N4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)CC6=C5)CC4)CC3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C39H40F3N9O6	IRAK4	Q9NWZ3	CRBN	WO-2023241644-A1
TPD-TK3PYN	WO2024002205A1_1	.	CN1C2=C(C=CC(N3CCN(CC4CN(C5=CC=C(C(=O)N[C@H]6CC[C@H](OC7=CC(Cl)=C(C#N)C=C7)CC6)N=N5)C4)CC3)=C2)C2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O	C42H43ClN10O6	AR	P10275	CRBN	WO-2024002205-A1
TPD-N1ITRX	WO2024002205A1_2	.	CN1C2=C(C=CC(C3CCN(CC4CN(C5=CC=C(C(=O)N[C@H]6CC[C@H](OC7=CC(Cl)=C(C#N)C=C7)CC6)N=N5)C4)CC3)=C2)C2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O	C43H44ClN9O6	AR	P10275	CRBN	WO-2024002205-A1
TPD-D57RWM	WO2024002205A1_3	.	CCN1C2=C(C=CC(N3CCN(CC4CN(C5=CC=C(C(=O)N[C@H]6CC[C@H](OC7=CC(Cl)=C(C#N)C=C7)CC6)N=N5)C4)CC3)=C2)C2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O	C43H45ClN10O6	AR	P10275	CRBN	WO-2024002205-A1
TPD-1T30R1	WO2024002205A1_4	.	CCN1C2=C(C=CC(N3CCN(CC4CCN(C5=CC=C(C(=O)N[C@H]6CC[C@H](OC7=CC(Cl)=C(C#N)C=C7)CC6)C=N5)CC4)CC3)=C2)C2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O	C46H50ClN9O6	AR	P10275	CRBN	WO-2024002205-A1
TPD-814GCQ	WO2024002205A1_5	.	CCN1C2=C(C=CC(N3CCN(CC4CCN(C5=CC=C(C(=O)N[C@H]6CC[C@@H](OC7=CC(Cl)=C(C#N)C=C7)CC6)C=N5)CC4)CC3)=C2)C2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O	C46H50ClN9O6	AR	P10275	CRBN	WO-2024002205-A1
TPD-QIS1IV	WO2024002205A1_6	.	CCN1C2=C(C=CC(N3CCN(CC4CCN(C5=CC=C(C(=O)N[C@H]6C(C)(C)[C@H](OC7=CC(Cl)=C(C#N)C=C7)C6(C)C)C=N5)CC4)CC3)=C2)C2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O	C48H54ClN9O6	AR	P10275	CRBN	WO-2024002205-A1
TPD-09F328	WO2024002205A1_7	.	CCN1C2=C(C=CC(N3CCN(CC4CCN(C5=CC=C(C(=O)N[C@H]6C(C)(C)[C@@H](OC7=CC(Cl)=C(C#N)C=C7)C6(C)C)C=N5)CC4)CC3)=C2)C2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O	C48H54ClN9O6	AR	P10275	CRBN	WO-2024002205-A1
TPD-EOCU32	WO2024002205A1_8	.	CCN1C2=C(C=CC(N3CCN(CC4CCN(C5=CC=C(C(=O)N[C@H]6C(C)(C)[C@H](OC7=CC(Cl)=C(C#N)C=C7)C6(C)C)N=N5)CC4)CC3)=C2)C2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O	C47H53ClN10O6	AR	P10275	CRBN	WO-2024002205-A1
TPD-M6JG3S	WO2024002205A1_9	.	CCN1C2=C(C=CC(N3CCN(CC4CCN(C5=CC=C(C(=O)N[C@H]6C(C)(C)[C@@H](OC7=CC(Cl)=C(C#N)C=C7)C6(C)C)N=N5)CC4)CC3)=C2)C2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O	C47H53ClN10O6	AR	P10275	CRBN	WO-2024002205-A1
TPD-180S5S	WO2024002205A1_10	.	CCN1C2=C(C=CC(C3CCN(CC4CN(C5=CC=C(C(=O)N[C@H]6CC[C@H](OC7=CC(Cl)=C(C#N)C=C7)CC6)N=N5)C4)CC3)=C2)C2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O	C44H46ClN9O6	AR	P10275	CRBN	WO-2024002205-A1
TPD-K4L81X	WO2024002205A1_11	.	CCN1C2=C(C=CC(C3CCN(CC4CCN(C5=CC=C(C(=O)N[C@H]6CC[C@H](OC7=CC(Cl)=C(C#N)C=C7)CC6)N=N5)CC4)CC3)=C2)C2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O	C46H50ClN9O6	AR	P10275	CRBN	WO-2024002205-A1
TPD-AYIU41	WO2024002205A1_12	.	CCN1C2=C(C=CC(C3CCN(CC4CCN(C5=CC=C(C(=O)N[C@H]6CC[C@@H](OC7=CC(Cl)=C(C#N)C=C7)CC6)N=N5)CC4)CC3)=C2)C2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O	C46H50ClN9O6	AR	P10275	CRBN	WO-2024002205-A1
TPD-N0A45F	WO2024002205A1_13	.	CN1C2=C(C=CC(N3CCC4(CC3)CC(CN3CCN(C5=CC=C(C(=O)N[C@H]6CC[C@H](OC7=CC(Cl)=C(C#N)C=C7)CC6)N=N5)CC3)C4)=C2)C2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O	C47H51ClN10O6	AR	P10275	CRBN	WO-2024002205-A1
TPD-6PZD1A	WO2024002205A1_14	.	CCN1C2=C(C=CC(N3CCC4(CC3)CC(CN3CCN(C5=CC=C(C(=O)N[C@H]6CC[C@H](OC7=CC(Cl)=C(C#N)C=C7)CC6)N=N5)CC3)C4)=C2)C2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O	C48H53ClN10O6	AR	P10275	CRBN	WO-2024002205-A1
TPD-WHRHSR	WO2024002205A1_15	.	CCN1C2=C(C=CC(N3CCN(CC4CCN(C5=CC=C(C(=O)N[C@H]6C(C)(C)[C@H](OC7=CC(Cl)=C(C#N)C=C7)C6(C)C)C=C5)CC4)CC3)=C2)C2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O	C49H55ClN8O6	AR	P10275	CRBN	WO-2024002205-A1
TPD-S2CRHU	WO2024002205A1_16	.	CCN1C2=C(C=CC(N3CCN(CC4CCN(C5=CC=C(C(=O)N[C@H]6C(C)(C)[C@@H](OC7=CC(Cl)=C(C#N)C=C7)C6(C)C)C=C5)CC4)CC3)=C2)C2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O	C49H55ClN8O6	AR	P10275	CRBN	WO-2024002205-A1
TPD-HYL4OU	WO2024002205A1_17	.	CCN1C2=C(C=CC(N3CCN(CC4CCN(C5=CC=C(C(=O)N[C@H]6CC[C@H](OC7=CC(Cl)=C(C#N)C=C7)CC6)N=N5)C4)CC3)=C2)C2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O	C44H47ClN10O6	AR	P10275	CRBN	WO-2024002205-A1
TPD-16ALZJ	WO2024002205A1_18	.	CCN1C2=C(C=CC(C3CCN(CC4CCN(C5=CC=C(C(=O)N[C@H]6CC[C@H](OC7=CC(Cl)=C(C#N)C=C7)CC6)N=N5)C4)CC3)=C2)C2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O	C45H48ClN9O6	AR	P10275	CRBN	WO-2024002205-A1
TPD-G2A9H0	WO2024002205A1_19	.	CN1C2=C(C=CC(N3CC4(CCN(CC5CCN(C6=CC=C(C(=O)N[C@H]7CC[C@H](OC8=CC(Cl)=C(C#N)C=C8)CC7)N=N6)CC5)CC4)C3)=C2)C2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O	C47H51ClN10O6	AR	P10275	CRBN	WO-2024002205-A1
TPD-FMW3Y1	WO2024002205A1_20	.	CCN1C2=C(C=CC(N3CC4(CCN(CC5CCN(C6=CC=C(C(=O)N[C@H]7CC[C@H](OC8=CC(Cl)=C(C#N)C=C8)CC7)N=N6)CC5)CC4)C3)=C2)C2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O	C48H53ClN10O6	AR	P10275	CRBN	WO-2024002205-A1
TPD-3JNK0X	WO2024002205A1_21	.	CN1C2=C(C=CC(N3CCN(CC4CCN(C5=CC=C(C(=O)N[C@H]6CC[C@H](OC7=CC(Cl)=C(C#N)C=C7)CC6)N=N5)CC4)CC3)=C2)C2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O	C44H47ClN10O6	AR	P10275	CRBN	WO-2024002205-A1
TPD-NLEKKX	WO2024002205A1_22	.	CN1C2=C(C=CC(N3CCN(CC4CCN(C5=CC=C(C(=O)N[C@H]6CC[C@@H](OC7=CC(Cl)=C(C#N)C=C7)CC6)N=N5)CC4)CC3)=C2)C2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O	C44H47ClN10O6	AR	P10275	CRBN	WO-2024002205-A1
TPD-2UBFJL	WO2024002205A1_23	.	CCN1C2=C(C=CC(N3CCN(CC4CCN(C5=CC=C(C(=O)N[C@H]6CC[C@H](OC7=CC(Cl)=C(C#N)C=C7)CC6)N=N5)CC4)CC3)=C2)C2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O	C45H49ClN10O6	AR	P10275	CRBN	WO-2024002205-A1
TPD-PASGCK	WO2024002205A1_24	.	CCN1C2=C(C=CC(C3CCN(CC4CCN(C5=CC=C(C(=O)N[C@H]6C(C)(C)[C@H](OC7=CC(Cl)=C(C#N)C=C7)C6(C)C)C=C5)CC4)CC3)=C2)C2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O	C50H56ClN7O6	AR	P10275	CRBN	WO-2024002205-A1
TPD-UDZP7H	WO2024002205A1_25	.	CCN1C2=C(C=CC(N3CCN(CC4CCN(C5=NC=C(C(=O)N[C@H]6CC[C@H](OC7=CC(Cl)=C(C#N)C=C7)CC6)C=N5)CC4)CC3)=C2)C2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O	C45H49ClN10O6	AR	P10275	CRBN	WO-2024002205-A1
TPD-1PNMNW	WO2024002205A1_26	.	CCN1C2=C(C=CC(N3CCN(CC4CCN(C5=NC=C(C(=O)N[C@H]6CC[C@@H](OC7=CC(Cl)=C(C#N)C=C7)CC6)C=N5)CC4)CC3)=C2)C2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O	C45H49ClN10O6	AR	P10275	CRBN	WO-2024002205-A1
TPD-AE6XJ7	WO2024002205A1_27	.	CN1C2=C(C=CC(N3CCN(CC4CCN(C5=CC=C(C(=O)N[C@H]6C(C)(C)[C@H](OC7=CC(Cl)=C(C#N)C=C7)C6(C)C)C=N5)CC4)CC3)=C2)C2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O	C47H52ClN9O6	AR	P10275	CRBN	WO-2024002205-A1
TPD-LQG0KN	WO2024002205A1_28	.	CN1C2=C(C=CC(N3CCN(CC4CCN(C5=CC=C(C(=O)N[C@H]6C(C)(C)[C@@H](OC7=CC(Cl)=C(C#N)C=C7)C6(C)C)C=N5)CC4)CC3)=C2)C2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O	C47H52ClN9O6	AR	P10275	CRBN	WO-2024002205-A1
TPD-QYM79M	WO2024002205A1_29	.	CN1C2=C(C=CC(C3CCN(CC4CCN(C5=CC=C(C(=O)N[C@H]6CC[C@H](OC7=CC(Cl)=C(C#N)C=C7)CC6)N=N5)CC4)CC3)=C2)C2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O	C45H48ClN9O6	AR	P10275	CRBN	WO-2024002205-A1
TPD-Q38KNG	WO2024002205A1_30	.	CN1C2=C(C=CC(C3CCN(CC4CCN(C5=CC=C(C(=O)N[C@H]6CC[C@@H](OC7=CC(Cl)=C(C#N)C=C7)CC6)N=N5)CC4)CC3)=C2)C2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O	C45H48ClN9O6	AR	P10275	CRBN	WO-2024002205-A1
TPD-ZS5PWD	WO2024002205A1_31	.	CN1C2=C(C=CC(N3CCN(CC4CC5(CCN(C6=CC=C(C(=O)N[C@H]7CC[C@H](OC8=CC(Cl)=C(C#N)C=C8)CC7)N=N6)CC5)C4)CC3)=C2)C2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O	C47H51ClN10O6	AR	P10275	CRBN	WO-2024002205-A1
TPD-SG2C63	WO2024002205A1_32	.	CCN1C2=C(C=CC(N3CCN(CC4CC5(CCN(C6=CC=C(C(=O)N[C@H]7CC[C@H](OC8=CC(Cl)=C(C#N)C=C8)CC7)N=N6)CC5)C4)CC3)=C2)C2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O	C48H53ClN10O6	AR	P10275	CRBN	WO-2024002205-A1
TPD-BWICZS	WO2024002205A1_33	.	CCN1C2=C(C=CC(N3CCN(CC4CCN(C5=CC=C(C(=O)N[C@H]6CC[C@@H](OC7=CC(Cl)=C(C#N)C=C7)CC6)N=N5)CC4)CC3)=C2)C2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O	C45H49ClN10O6	AR	P10275	CRBN	WO-2024002205-A1
TPD-583QIR	WO2024002205A1_35	.	CN1C2=C(C=CC(N3CCN(CC4CCN(C5=NC=C(C(=O)N[C@H]6CC[C@H](OC7=CC(Cl)=C(C#N)C=C7)CC6)C=N5)CC4)CC3)=C2)C2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O	C44H47ClN10O6	AR	P10275	CRBN	WO-2024002205-A1
TPD-27QSHP	WO2024002205A1_37	.	CN1C2=C(C=CC(N3CCC(CN4CC5(CCN(C6=CC=C(C(=O)N[C@H]7CC[C@H](OC8=CC(Cl)=C(C#N)C=C8)CC7)N=N6)CC5)C4)CC3)=C2)C2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O	C47H51ClN10O6	AR	P10275	CRBN	WO-2024002205-A1
TPD-SA8QVI	WO2024002205A1_38	.	CCN1C2=C(C=CC(N3CCC(CN4CC5(CCN(C6=CC=C(C(=O)N[C@H]7CC[C@H](OC8=CC(Cl)=C(C#N)C=C8)CC7)N=N6)CC5)C4)CC3)=C2)C2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O	C48H53ClN10O6	AR	P10275	CRBN	WO-2024002205-A1
TPD-WXM1KK	WO2024002205A1_39	.	CCN1C2=C(C=CC(N3CCN(CC4CCN(C5=CC=C(C(=O)N[C@H]6CC[C@@H](OC7=CC(Cl)=C(C#N)C=C7)CC6)N=N5)CC4)CC3)=C2)C2=C1C(=O)N([C@H]1CCC(=O)NC1=O)C2=O	C45H49ClN10O6	AR	P10275	CRBN	WO-2024002205-A1
TPD-2PPUTK	WO2024002205A1_40	.	CCN1C2=C(C=CC(N3CCC(CN4CCC(C5=CC=C(C(=O)N[C@H]6CC[C@H](OC7=CC(Cl)=C(C#N)C=C7)CC6)N=N5)CC4)CC3)=C2)C2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O	C46H50ClN9O6	AR	P10275	CRBN	WO-2024002205-A1
TPD-P4RIXX	WO2024002205A1_41	.	CN1C2=C(C=C(N3CCN(CC4CCN(C5=CC=C(C(=O)N[C@H]6CC[C@H](OC7=CC(Cl)=C(C#N)C=C7)CC6)N=N5)CC4)CC3)C=C2)C2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O	C44H47ClN10O6	AR	P10275	CRBN	WO-2024002205-A1
TPD-IJQ5GI	WO2024002205A1_42	.	CN1C2=C(C=C(N3CCN(CC4CCN(C5=CC=C(C(=O)N[C@H]6CC[C@@H](OC7=CC(Cl)=C(C#N)C=C7)CC6)N=N5)CC4)CC3)C=C2)C2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O	C44H47ClN10O6	AR	P10275	CRBN	WO-2024002205-A1
TPD-PM7UET	WO2024002205A1_43	.	CN1C2=C(C=CC(N3CCC(CN4CCC5(CC4)CN(C4=CC=C(C(=O)N[C@H]6CC[C@H](OC7=CC(Cl)=C(C#N)C=C7)CC6)N=N4)C5)CC3)=C2)C2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O	C47H51ClN10O6	AR	P10275	CRBN	WO-2024002205-A1
TPD-PGNIN4	WO2024002205A1_44	.	CCN1C2=C(C=CC(N3CCC(CN4CCC5(CC4)CN(C4=CC=C(C(=O)N[C@H]6CC[C@H](OC7=CC(Cl)=C(C#N)C=C7)CC6)N=N4)C5)CC3)=C2)C2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O	C48H53ClN10O6	AR	P10275	CRBN	WO-2024002205-A1
TPD-A7GDQN	WO2024002205A1_45	.	CCN1C2=C(C=CC(N3CCC(CN4CCN(C5=CC=C(C(=O)N[C@H]6CC[C@H](OC7=CC(Cl)=C(C#N)C=C7)CC6)N=N5)CC4)CC3)=C2)C2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O	C45H49ClN10O6	AR	P10275	CRBN	WO-2024002205-A1
TPD-E0P40P	WO2024002205A1_46	.	CN1C2=C(C=CC(N3CCC(CN4CCN(C5=CC=C(C(=O)N[C@H]6CC[C@H](OC7=CC(Cl)=C(C#N)C=C7)CC6)N=N5)CC4)CC3)=C2)C2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O	C44H47ClN10O6	AR	P10275	CRBN	WO-2024002205-A1
TPD-QJNXZU	WO2024002205A1_47	.	CN1C2=C(C=C(N3CCN(CC4CN(C5=CC=C(C(=O)N[C@H]6CC[C@H](OC7=CC(Cl)=C(C#N)C=C7)CC6)N=N5)C4)CC3)C=C2)C2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O	C42H43ClN10O6	AR	P10275	CRBN	WO-2024002205-A1
TPD-38Y2LV	WO2024002205A1_48	.	CCN1C2=C(C=CC(C3=CCN(CC4CCN(C5=CC=C(C(=O)N[C@H]6CC[C@H](OC7=CC(Cl)=C(C#N)C=C7)CC6)N=N5)CC4)CC3)=C2)C2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O	C46H48ClN9O6	AR	P10275	CRBN	WO-2024002205-A1
TPD-W5AX37	WO2024002205A1_49	.	CCN1C2=C(C=CC(C3=CCN(CC4CN(C5=CC=C(C(=O)N[C@H]6CC[C@H](OC7=CC(Cl)=C(C#N)C=C7)CC6)N=N5)C4)CC3)=C2)C2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O	C44H44ClN9O6	AR	P10275	CRBN	WO-2024002205-A1
TPD-BCRJZW	WO2024002205A1_50	.	CN1C2=C(C=CC(N3CCC4(CC3)CN(CC3CCN(C5=CC=C(C(=O)N[C@H]6CC[C@H](OC7=CC(Cl)=C(C#N)C=C7)CC6)N=N5)CC3)C4)=C2)C2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O	C47H51ClN10O6	AR	P10275	CRBN	WO-2024002205-A1
TPD-W014LK	WO2024002205A1_51	.	CCN1C2=C(C=CC(N3CCC4(CC3)CN(CC3CCN(C5=CC=C(C(=O)N[C@H]6CC[C@H](OC7=CC(Cl)=C(C#N)C=C7)CC6)N=N5)CC3)C4)=C2)C2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O	C48H53ClN10O6	AR	P10275	CRBN	WO-2024002205-A1
TPD-3UX8NK	SCHEMBL27027510	2-Chloro-4-[5-[6-[3-[[4-[2-(2,6-dioxopiperidin-3-yl)-4-methyl-1,3-dioxopyrrolo[3,4-b]indol-6-yl]piperazin-1-yl]methyl]azetidin-1-yl]-2-fluoropyridin-3-yl]-3,3-dimethyl-2-oxoindol-1-yl]benzonitrile	Cn1c2c(c3ccc(N4CCN(CC5CN(c6ccc(-c7ccc8c(c7)C(C)(C)C(=O)N8c7ccc(C#N)c(Cl)c7)c(F)n6)C5)CC4)cc31)C(=O)N(C1CCC(=O)NC1=O)C2=O	C46H41ClFN9O5	AR	P10275	CRBN	WO-2024002289-A1
TPD-AXLPOM	SCHEMBL27027513	2-Chloro-4-[5-[6-[3-[[4-[2-(2,6-dioxopiperidin-3-yl)-4-methyl-1,3-dioxopyrrolo[3,4-b]indol-6-yl]oxypiperidin-1-yl]methyl]azetidin-1-yl]-2-fluoropyridin-3-yl]-3,3-dimethyl-2-oxoindol-1-yl]benzonitrile	Cn1c2c(c3ccc(OC4CCN(CC5CN(c6ccc(-c7ccc8c(c7)C(C)(C)C(=O)N8c7ccc(C#N)c(Cl)c7)c(F)n6)C5)CC4)cc31)C(=O)N(C1CCC(=O)NC1=O)C2=O	C47H42ClFN8O6	AR	P10275	CRBN	WO-2024002289-A1
TPD-SLYXHB	SCHEMBL27027522	2-Chloro-4-[5-[6-[3-[[4-[2-(2,6-dioxopiperidin-3-yl)-4-ethyl-1,3-dioxopyrrolo[3,4-b]indol-6-yl]piperidin-1-yl]methyl]azetidin-1-yl]-2-fluoropyridin-3-yl]-3,3-dimethyl-2-oxoindol-1-yl]benzonitrile	CCn1c2c(c3ccc(C4CCN(CC5CN(c6ccc(-c7ccc8c(c7)C(C)(C)C(=O)N8c7ccc(C#N)c(Cl)c7)c(F)n6)C5)CC4)cc31)C(=O)N(C1CCC(=O)NC1=O)C2=O	C48H44ClFN8O5	AR	P10275	CRBN	WO-2024002289-A1
TPD-WJJ86Y	SCHEMBL27027532	2-Chloro-4-[5-[6-[4-[3-[2-(2,6-dioxopiperidin-3-yl)-4-ethyl-1,3-dioxopyrrolo[3,4-b]indol-6-yl]oxypropyl]piperazin-1-yl]-2-fluoropyridin-3-yl]-3,3-dimethyl-2-oxoindol-1-yl]benzonitrile	CCn1c2c(c3ccc(OCCCN4CCN(c5ccc(-c6ccc7c(c6)C(C)(C)C(=O)N7c6ccc(C#N)c(Cl)c6)c(F)n5)CC4)cc31)C(=O)N(C1CCC(=O)NC1=O)C2=O	C46H42ClFN8O6	AR	P10275	CRBN	WO-2024002289-A1
TPD-NK14H4	SCHEMBL27027567	2-Chloro-4-[5-[6-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-4-methyl-1,3-dioxopyrrolo[3,4-b]indol-6-yl]piperazin-1-yl]methyl]piperidin-1-yl]-2-fluoropyridin-3-yl]-3,3-dimethyl-2-oxoindol-1-yl]benzonitrile	Cn1c2c(c3ccc(N4CCN(CC5CCN(c6ccc(-c7ccc8c(c7)C(C)(C)C(=O)N8c7ccc(C#N)c(Cl)c7)c(F)n6)CC5)CC4)cc31)C(=O)N(C1CCC(=O)NC1=O)C2=O	C48H45ClFN9O5	AR	P10275	CRBN	WO-2024002289-A1
TPD-LFECEO	WO2024002289A1_6	.	CN1c2cc(N3CCN(CC4CN(c5ccc(-c6ccc7c(c6)C(C)(C)C(=O)N7c6ccc(C#N)c(C(F)(F)F)c6)c(F)n5)C4)CC3)ccc2C2C(=O)N(C3CCC(=O)NC3=O)C(=O)C21	C47H43F4N9O5	AR	P10275	CRBN	WO-2024002289-A1
TPD-HX31CB	SCHEMBL27027576	4-[5-[6-[3-[[7-[2-(2,6-Dioxopiperidin-3-yl)-4-methyl-1,3-dioxopyrrolo[3,4-b]indol-6-yl]-2,7-diazaspiro[3.5]nonan-2-yl]methyl]azetidin-1-yl]-2-fluoropyridin-3-yl]-3,3-dimethyl-2-oxoindol-1-yl]-2-(trifluoromethyl)benzonitrile	Cn1c2c(c3ccc(N4CCC5(CC4)CN(CC4CN(c6ccc(-c7ccc8c(c7)C(C)(C)C(=O)N8c7ccc(C#N)c(C(F)(F)F)c7)c(F)n6)C4)C5)cc31)C(=O)N(C1CCC(=O)NC1=O)C2=O	C50H45F4N9O5	AR	P10275	CRBN	WO-2024002289-A1
TPD-7XUDOW	SCHEMBL27027636	2-Chloro-4-[5-[6-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-4-methyl-1,3-dioxopyrrolo[3,4-b]indol-6-yl]piperidin-1-yl]methyl]piperidin-1-yl]-2-fluoropyridin-3-yl]-3,3-dimethyl-2-oxoindol-1-yl]benzonitrile	Cn1c2c(c3ccc(C4CCN(CC5CCN(c6ccc(-c7ccc8c(c7)C(C)(C)C(=O)N8c7ccc(C#N)c(Cl)c7)c(F)n6)CC5)CC4)cc31)C(=O)N(C1CCC(=O)NC1=O)C2=O	C49H46ClFN8O5	AR	P10275	CRBN	WO-2024002289-A1
TPD-S3BX57	SCHEMBL27027568	2-Chloro-4-[5-[6-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-4-ethyl-1,3-dioxopyrrolo[3,4-b]indol-6-yl]piperazin-1-yl]methyl]piperidin-1-yl]-2-fluoropyridin-3-yl]-3,3-dimethyl-2-oxoindol-1-yl]benzonitrile	CCn1c2c(c3ccc(N4CCN(CC5CCN(c6ccc(-c7ccc8c(c7)C(C)(C)C(=O)N8c7ccc(C#N)c(Cl)c7)c(F)n6)CC5)CC4)cc31)C(=O)N(C1CCC(=O)NC1=O)C2=O	C49H47ClFN9O5	AR	P10275	CRBN	WO-2024002289-A1
TPD-ILNAKN	SCHEMBL27027577	4-[5-[6-[3-[[7-[2-(2,6-Dioxopiperidin-3-yl)-4-ethyl-1,3-dioxopyrrolo[3,4-b]indol-6-yl]-2,7-diazaspiro[3.5]nonan-2-yl]methyl]azetidin-1-yl]-2-fluoropyridin-3-yl]-3,3-dimethyl-2-oxoindol-1-yl]-2-(trifluoromethyl)benzonitrile	CCn1c2c(c3ccc(N4CCC5(CC4)CN(CC4CN(c6ccc(-c7ccc8c(c7)C(C)(C)C(=O)N8c7ccc(C#N)c(C(F)(F)F)c7)c(F)n6)C4)C5)cc31)C(=O)N(C1CCC(=O)NC1=O)C2=O	C51H47F4N9O5	AR	P10275	CRBN	WO-2024002289-A1
TPD-KRVPXI	SCHEMBL27027570	2-Chloro-4-[5-[6-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-4-methyl-1,3-dioxopyrrolo[3,4-b]indol-6-yl]piperazin-1-yl]methyl]piperidin-1-yl]pyridazin-3-yl]-3,3-dimethyl-2-oxoindol-1-yl]benzonitrile	Cn1c2c(c3ccc(N4CCN(CC5CCN(c6ccc(-c7ccc8c(c7)C(C)(C)C(=O)N8c7ccc(C#N)c(Cl)c7)nn6)CC5)CC4)cc31)C(=O)N(C1CCC(=O)NC1=O)C2=O	C47H45ClN10O5	AR	P10275	CRBN	WO-2024002289-A1
TPD-3QUPX8	SCHEMBL27027578	4-[5-[6-[3-[[2-[2-(2,6-Dioxopiperidin-3-yl)-4-methyl-1,3-dioxopyrrolo[3,4-b]indol-6-yl]-2,7-diazaspiro[3.5]nonan-7-yl]methyl]azetidin-1-yl]-2-fluoropyridin-3-yl]-3,3-dimethyl-2-oxoindol-1-yl]-2-(trifluoromethyl)benzonitrile	Cn1c2c(c3ccc(N4CC5(CCN(CC6CN(c7ccc(-c8ccc9c(c8)C(C)(C)C(=O)N9c8ccc(C#N)c(C(F)(F)F)c8)c(F)n7)C6)CC5)C4)cc31)C(=O)N(C1CCC(=O)NC1=O)C2=O	C50H45F4N9O5	AR	P10275	CRBN	WO-2024002289-A1
TPD-TAN6JH	SCHEMBL27027580	4-[5-[6-[3-[[2-[2-(2,6-Dioxopiperidin-3-yl)-4-ethyl-1,3-dioxopyrrolo[3,4-b]indol-6-yl]-2,7-diazaspiro[3.5]nonan-7-yl]methyl]azetidin-1-yl]-2-fluoropyridin-3-yl]-3,3-dimethyl-2-oxoindol-1-yl]-2-(trifluoromethyl)benzonitrile	CCn1c2c(c3ccc(N4CC5(CCN(CC6CN(c7ccc(-c8ccc9c(c8)C(C)(C)C(=O)N9c8ccc(C#N)c(C(F)(F)F)c8)c(F)n7)C6)CC5)C4)cc31)C(=O)N(C1CCC(=O)NC1=O)C2=O	C51H47F4N9O5	AR	P10275	CRBN	WO-2024002289-A1
TPD-HVO7WH	SCHEMBL27027572	2-Chloro-4-[5-[6-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-4-ethyl-1,3-dioxopyrrolo[3,4-b]indol-6-yl]oxyethyl]piperazin-1-yl]-2-fluoropyridin-3-yl]-3,3-dimethyl-2-oxoindol-1-yl]benzonitrile	CCn1c2c(c3ccc(OCCN4CCN(c5ccc(-c6ccc7c(c6)C(C)(C)C(=O)N7c6ccc(C#N)c(Cl)c6)c(F)n5)CC4)cc31)C(=O)N(C1CCC(=O)NC1=O)C2=O	C45H40ClFN8O6	AR	P10275	CRBN	WO-2024002289-A1
TPD-60SFZW	SCHEMBL27027571	2-Chloro-4-[5-[6-[3-[[4-[2-(2,6-dioxopiperidin-3-yl)-4-ethyl-1,3-dioxopyrrolo[3,4-b]indol-6-yl]piperazin-1-yl]methyl]azetidin-1-yl]-2-fluoropyridin-3-yl]-3,3-dimethyl-2-oxoindol-1-yl]benzonitrile	CCn1c2c(c3ccc(N4CCN(CC5CN(c6ccc(-c7ccc8c(c7)C(C)(C)C(=O)N8c7ccc(C#N)c(Cl)c7)c(F)n6)C5)CC4)cc31)C(=O)N(C1CCC(=O)NC1=O)C2=O	C47H43ClFN9O5	AR	P10275	CRBN	WO-2024002289-A1
TPD-R1GH77	SCHEMBL27311664	4-[2-[4-[(3R,5R)-5-[(3-bromo-4-oxopyrido[1,2-a]pyrimidin-2-yl)amino]-1-methylpiperidin-3-yl]phenoxy]ethoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN1C[C@H](NC2=C(Br)C(=O)N3C=CC=CC3=N2)C[C@H](C2=CC=C(OCCOC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)C=C2)C1	C35H33BrN6O7	KAT2A;KAT2B	Q92830/Q92831	CRBN	WO-2024003533-A1
TPD-QI5TYA	SCHEMBL27311767	4-[2-[2-[4-[(3R,5R)-5-[(3-bromo-4-oxopyrido[1,2-a]pyrimidin-2-yl)amino]-1-methylpiperidin-3-yl]phenoxy]ethoxy]ethoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN1C[C@H](NC2=C(Br)C(=O)N3C=CC=CC3=N2)C[C@H](C2=CC=C(OCCOCCOC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)C=C2)C1	C37H37BrN6O8	KAT2A;KAT2B	Q92830/Q92831	CRBN	WO-2024003533-A1
TPD-4MGRSN	SCHEMBL27311769	5-[2-[2-[4-[(3R,5R)-5-[(3-bromo-4-oxopyrido[1,2-a]pyrimidin-2-yl)amino]-1-methylpiperidin-3-yl]phenoxy]ethoxy]ethoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN1C[C@H](NC2=C(Br)C(=O)N3C=CC=CC3=N2)C[C@H](C2=CC=C(OCCOCCOC3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C=C2)C1	C37H37BrN6O8	KAT2A;KAT2B	Q92830/Q92831	CRBN	WO-2024003533-A1
TPD-C1EGYJ	WO2024003533A1_4	.	O=C1CCC(N2C(=O)C3=CC=CC(OCCOCCOCCOC4=CC=C([C@@H]5CNC[C@H](NC6=C(Br)C(=O)N7C=CC=CC7=N6)C5)C=C4)=C3C2=O)C(=O)N1	C38H39BrN6O9	KAT2A;KAT2B	Q92830/Q92831	CRBN	WO-2024003533-A1
TPD-VYYLKJ	SCHEMBL27311773	4-[3-[4-[(3R,5R)-5-[(3-bromo-4-oxopyrido[1,2-a]pyrimidin-2-yl)amino]-1-methylpiperidin-3-yl]phenoxy]propoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN1C[C@H](NC2=C(Br)C(=O)N3C=CC=CC3=N2)C[C@H](C2=CC=C(OCCCOC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)C=C2)C1	C36H35BrN6O7	KAT2A;KAT2B	Q92830/Q92831	CRBN	WO-2024003533-A1
TPD-KMFET7	SCHEMBL27311775	4-[4-[4-[(3R,5R)-5-[(3-bromo-4-oxopyrido[1,2-a]pyrimidin-2-yl)amino]-1-methylpiperidin-3-yl]phenoxy]butoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN1C[C@H](NC2=C(Br)C(=O)N3C=CC=CC3=N2)C[C@H](C2=CC=C(OCCCCOC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)C=C2)C1	C37H37BrN6O7	KAT2A;KAT2B	Q92830/Q92831	CRBN	WO-2024003533-A1
TPD-S1IL49	SCHEMBL30746878	4-[5-[4-[(3R,5R)-5-[(3-bromo-4-oxopyrido[1,2-a]pyrimidin-2-yl)amino]-1-methylpiperidin-3-yl]phenoxy]pentoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN1C[C@H](NC2=C(Br)C(=O)N3C=CC=CC3=N2)C[C@H](C2=CC=C(OCCCCCOC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)C=C2)C1	C38H39BrN6O7	KAT2A;KAT2B	Q92830/Q92831	CRBN	WO-2024003533-A1
TPD-Q8B3LQ	SCHEMBL27311912	4-[2-[2-[2-[3-[(3R,5R)-5-[(3-bromo-4-oxopyrido[1,2-a]pyrimidin-2-yl)amino]-1-methylpiperidin-3-yl]phenoxy]ethoxy]ethoxy]ethoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN1C[C@H](NC2=C(Br)C(=O)N3C=CC=CC3=N2)C[C@H](C2=CC(OCCOCCOCCOC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)=CC=C2)C1	C39H41BrN6O9	KAT2A;KAT2B	Q92830/Q92831	CRBN	WO-2024003533-A1
TPD-V2AKND	SCHEMBL27311916	5-[2-[2-[2-[3-[(3R,5R)-5-[(3-bromo-4-oxopyrido[1,2-a]pyrimidin-2-yl)amino]-1-methylpiperidin-3-yl]phenoxy]ethoxy]ethoxy]ethoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN1C[C@H](NC2=C(Br)C(=O)N3C=CC=CC3=N2)C[C@H](C2=CC(OCCOCCOCCOC3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4=O)=CC=C2)C1	C39H41BrN6O9	KAT2A;KAT2B	Q92830/Q92831	CRBN	WO-2024003533-A1
TPD-IXW61J	SCHEMBL27311918	4-[2-[2-[4-[(3R,5R)-5-[(6-bromo-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)amino]-1-methylpiperidin-3-yl]phenoxy]ethoxy]ethoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN1C[C@H](NC2=C(Br)C(=O)N3C=CSC3=N2)C[C@H](C2=CC=C(OCCOCCOC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)C=C2)C1	C35H35BrN6O8S	KAT2A;KAT2B	Q92830/Q92831	CRBN	WO-2024003533-A1
TPD-B2ZQKE	SCHEMBL27312025	4-[2-[2-[2-[4-[(3R,5R)-5-[(6-bromo-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)amino]-1-methylpiperidin-3-yl]phenoxy]ethoxy]ethoxy]ethoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN1C[C@H](NC2=C(Br)C(=O)N3C=CSC3=N2)C[C@H](C2=CC=C(OCCOCCOCCOC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)C=C2)C1	C37H39BrN6O9S	KAT2A;KAT2B	Q92830/Q92831	CRBN	WO-2024003533-A1
TPD-I8PQD5	SCHEMBL27312027	4-[2-[2-[2-[3-[(3R,5R)-5-[(6-bromo-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)amino]-1-methylpiperidin-3-yl]phenoxy]ethoxy]ethoxy]ethoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN1C[C@H](NC2=C(Br)C(=O)N3C=CSC3=N2)C[C@H](C2=CC(OCCOCCOCCOC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)=CC=C2)C1	C37H39BrN6O9S	KAT2A;KAT2B	Q92830/Q92831	CRBN	WO-2024003533-A1
TPD-CR0WM3	SCHEMBL30746941	4-[4-[2-[4-[(3R,5R)-5-[(3-bromo-4-oxopyrido[1,2-a]pyrimidin-2-yl)amino]-1-methylpiperidin-3-yl]phenoxy]ethyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN1C[C@H](NC2=C(Br)C(=O)N3C=CC=CC3=N2)C[C@H](C2=CC=C(OCCN3CCN(C4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)C=C2)C1	C39H41BrN8O6	KAT2A;KAT2B	Q92830/Q92831	CRBN	WO-2024003533-A1
TPD-JIF1XD	SCHEMBL27312032	5-[4-[2-[4-[(3R,5R)-5-[(3-bromo-4-oxopyrido[1,2-a]pyrimidin-2-yl)amino]-1-methylpiperidin-3-yl]phenoxy]ethyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN1C[C@H](NC2=C(Br)C(=O)N3C=CC=CC3=N2)C[C@H](C2=CC=C(OCCN3CCN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)C=C2)C1	C39H41BrN8O6	KAT2A;KAT2B	Q92830/Q92831	CRBN	WO-2024003533-A1
TPD-JG9CSH	SCHEMBL27312159	4-[4-[2-[4-[(3R,5R)-5-[(3-bromo-4-oxopyrido[1,2-a]pyrimidin-2-yl)amino]-1-methylpiperidin-3-yl]phenoxy]ethyl]piperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN1C[C@H](NC2=C(Br)C(=O)N3C=CC=CC3=N2)C[C@H](C2=CC=C(OCCC3CCN(C4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)C=C2)C1	C40H42BrN7O6	KAT2A;KAT2B	Q92830/Q92831	CRBN	WO-2024003533-A1
TPD-8M4IP5	SCHEMBL27312160	4-[4-[[4-[(3R,5R)-5-[(3-bromo-4-oxopyrido[1,2-a]pyrimidin-2-yl)amino]-1-methylpiperidin-3-yl]phenoxy]methyl]piperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN1C[C@H](NC2=C(Br)C(=O)N3C=CC=CC3=N2)C[C@H](C2=CC=C(OCC3CCN(C4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)C=C2)C1	C39H40BrN7O6	KAT2A;KAT2B	Q92830/Q92831	CRBN	WO-2024003533-A1
TPD-SXKPUQ	SCHEMBL27312161	4-[2-[[4-[(3R,5R)-5-[(3-bromo-4-oxopyrido[1,2-a]pyrimidin-2-yl)amino]-1-methylpiperidin-3-yl]phenoxy]methyl]morpholin-4-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN1C[C@H](NC2=C(Br)C(=O)N3C=CC=CC3=N2)C[C@H](C2=CC=C(OCC3CN(C4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CCO3)C=C2)C1	C38H38BrN7O7	KAT2A;KAT2B	Q92830/Q92831	CRBN	WO-2024003533-A1
TPD-KTVPNP	SCHEMBL27312164	4-[3-[[4-[(3R,5R)-5-[(3-bromo-4-oxopyrido[1,2-a]pyrimidin-2-yl)amino]-1-methylpiperidin-3-yl]phenoxy]methyl]pyrrolidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN1C[C@H](NC2=C(Br)C(=O)N3C=CC=CC3=N2)C[C@H](C2=CC=C(OCC3CCN(C4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C3)C=C2)C1	C38H38BrN7O6	KAT2A;KAT2B	Q92830/Q92831	CRBN	WO-2024003533-A1
TPD-VTG3Q8	SCHEMBL30746928	4-[4-[2-[4-[(3R,5R)-5-[(6-bromo-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)amino]-1-methylpiperidin-3-yl]phenoxy]ethyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN1C[C@H](NC2=C(Br)C(=O)N3C=CSC3=N2)C[C@H](C2=CC=C(OCCN3CCN(C4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)C=C2)C1	C37H39BrN8O6S	KAT2A;KAT2B	Q92830/Q92831	CRBN	WO-2024003533-A1
TPD-WDTGCE	WO2024003533A1_20	.	O=C1CCC(N2C(=O)C3=CC=CC(OCC(=O)N4CCN(CCOC5=CC=C([C@@H]6CNC[C@H](NC7=C(Br)C(=O)N8C=CC=CC8=N7)C6)C=C5)CC4)=C3C2=O)C(=O)N1	C40H41BrN8O8	KAT2A;KAT2B	Q92830/Q92831	CRBN	WO-2024003533-A1
TPD-FVM5ZH	SCHEMBL27312284	4-[2-[4-[2-[4-[(3R,5R)-5-[(3-bromo-4-oxopyrido[1,2-a]pyrimidin-2-yl)amino]-1-methylpiperidin-3-yl]phenoxy]acetyl]piperazin-1-yl]ethoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN1C[C@H](NC2=C(Br)C(=O)N3C=CC=CC3=N2)C[C@H](C2=CC=C(OCC(=O)N3CCN(CCOC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)C=C2)C1	C41H43BrN8O8	KAT2A;KAT2B	Q92830/Q92831	CRBN	WO-2024003533-A1
TPD-H06MZ9	SCHEMBL30746970	2-[4-[(3R,5R)-5-[(3-bromo-4-oxopyrido[1,2-a]pyrimidin-2-yl)amino]-1-methylpiperidin-3-yl]phenoxy]-N-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyethyl]-N-methylacetamide	CN1C[C@H](NC2=C(Br)C(=O)N3C=CC=CC3=N2)C[C@H](C2=CC=C(OCC(=O)N(C)CCOC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)C=C2)C1	C38H38BrN7O8	KAT2A;KAT2B	Q92830/Q92831	CRBN	WO-2024003533-A1
TPD-HL860C	SCHEMBL27312446	4-[[1-[2-[4-[(3R,5R)-5-[(3-bromo-4-oxopyrido[1,2-a]pyrimidin-2-yl)amino]-1-methylpiperidin-3-yl]phenoxy]acetyl]azetidin-3-yl]methoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN1C[C@H](NC2=C(Br)C(=O)N3C=CC=CC3=N2)C[C@H](C2=CC=C(OCC(=O)N3CC(COC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C3)C=C2)C1	C39H38BrN7O8	KAT2A;KAT2B	Q92830/Q92831	CRBN	WO-2024003533-A1
TPD-0ICRYH	SCHEMBL27312448	4-[1-[2-[4-[(3R,5R)-5-[(3-bromo-4-oxopyrido[1,2-a]pyrimidin-2-yl)amino]-1-methylpiperidin-3-yl]phenoxy]acetyl]piperidin-4-yl]oxy-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN1C[C@H](NC2=C(Br)C(=O)N3C=CC=CC3=N2)C[C@H](C2=CC=C(OCC(=O)N3CCC(OC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)C=C2)C1	C40H40BrN7O8	KAT2A;KAT2B	Q92830/Q92831	CRBN	WO-2024003533-A1
TPD-YEJIZV	SCHEMBL27312451	4-[[1-[2-[4-[(3R,5R)-5-[(3-bromo-4-oxopyrido[1,2-a]pyrimidin-2-yl)amino]-1-methylpiperidin-3-yl]phenoxy]acetyl]piperidin-4-yl]methoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN1C[C@H](NC2=C(Br)C(=O)N3C=CC=CC3=N2)C[C@H](C2=CC=C(OCC(=O)N3CCC(COC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)C=C2)C1	C41H42BrN7O8	KAT2A;KAT2B	Q92830/Q92831	CRBN	WO-2024003533-A1
TPD-6M0QJ5	SCHEMBL27312454	4-[2-[1-[2-[4-[(3R,5R)-5-[(3-bromo-4-oxopyrido[1,2-a]pyrimidin-2-yl)amino]-1-methylpiperidin-3-yl]phenoxy]acetyl]piperidin-4-yl]ethoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN1C[C@H](NC2=C(Br)C(=O)N3C=CC=CC3=N2)C[C@H](C2=CC=C(OCC(=O)N3CCC(CCOC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)C=C2)C1	C42H44BrN7O8	KAT2A;KAT2B	Q92830/Q92831	CRBN	WO-2024003533-A1
TPD-ASDOOC	SCHEMBL27312456	4-[[1-[2-[4-[(3R,5R)-5-[(6-bromo-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)amino]-1-methylpiperidin-3-yl]phenoxy]ethyl]piperidin-4-yl]amino]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN1C[C@H](NC2=C(Br)C(=O)N3C=CSC3=N2)C[C@H](C2=CC=C(OCCN3CCC(NC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)C=C2)C1	C38H41BrN8O6S	KAT2A;KAT2B	Q92830/Q92831	CRBN	WO-2024003533-A1
TPD-CTXL8S	SCHEMBL27312596	4-[[1-[2-[4-[(3R,5R)-5-[(6-bromo-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)amino]-1-methylpiperidin-3-yl]phenoxy]acetyl]piperidin-4-yl]-methylamino]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN1C[C@H](NC2=C(Br)C(=O)N3C=CSC3=N2)C[C@H](C2=CC=C(OCC(=O)N3CCC(N(C)C4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)C=C2)C1	C39H41BrN8O7S	KAT2A;KAT2B	Q92830/Q92831	CRBN	WO-2024003533-A1
TPD-8Z052B	SCHEMBL27312599	4-[4-[2-[4-[(3R,5R)-5-[(6-bromo-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)amino]-1-methylpiperidin-3-yl]phenoxy]acetyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN1C[C@H](NC2=C(Br)C(=O)N3C=CSC3=N2)C[C@H](C2=CC=C(OCC(=O)N3CCN(C4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)C=C2)C1	C37H37BrN8O7S	KAT2A;KAT2B	Q92830/Q92831	CRBN	WO-2024003533-A1
TPD-HPFFV6	SCHEMBL27312603	4-[4-[2-[4-[(3R,5R)-5-[(6-bromo-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)amino]-1-methylpiperidin-3-yl]phenoxy]ethyl]piperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN1C[C@H](NC2=C(Br)C(=O)N3C=CSC3=N2)C[C@H](C2=CC=C(OCCC3CCN(C4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)C=C2)C1	C38H40BrN7O6S	KAT2A;KAT2B	Q92830/Q92831	CRBN	WO-2024003533-A1
TPD-476Z49	SCHEMBL27312755	4-[3-[2-[4-[(3R,5R)-5-[(6-bromo-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)amino]-1-methylpiperidin-3-yl]phenoxy]ethyl]pyrrolidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN1C[C@H](NC2=C(Br)C(=O)N3C=CSC3=N2)C[C@H](C2=CC=C(OCCC3CCN(C4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C3)C=C2)C1	C37H38BrN7O6S	KAT2A;KAT2B	Q92830/Q92831	CRBN	WO-2024003533-A1
TPD-J2CJZE	SCHEMBL27312760	4-[3-[2-[4-[(3R,5R)-5-[(6-bromo-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)amino]-1-methylpiperidin-3-yl]phenoxy]ethyl]azetidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN1C[C@H](NC2=C(Br)C(=O)N3C=CSC3=N2)C[C@H](C2=CC=C(OCCC3CN(C4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C3)C=C2)C1	C36H36BrN7O6S	KAT2A;KAT2B	Q92830/Q92831	CRBN	WO-2024003533-A1
TPD-68ETPX	SCHEMBL27312763	4-[7-[2-[4-[(3R,5R)-5-[(6-bromo-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)amino]-1-methylpiperidin-3-yl]phenoxy]ethyl]-2,7-diazaspiro[3.5]nonan-2-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN1C[C@H](NC2=C(Br)C(=O)N3C=CSC3=N2)C[C@H](C2=CC=C(OCCN3CCC4(CC3)CN(C3=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C3)C4)C=C2)C1	C40H43BrN8O6S	KAT2A;KAT2B	Q92830/Q92831	CRBN	WO-2024003533-A1
TPD-K7UMHF	SCHEMBL27312764	4-[2-[2-[4-[(3R,5R)-5-[(6-bromo-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)amino]-1-methylpiperidin-3-yl]phenoxy]ethyl]-2,7-diazaspiro[3.5]nonan-7-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN1C[C@H](NC2=C(Br)C(=O)N3C=CSC3=N2)C[C@H](C2=CC=C(OCCN3CC4(CCN(C5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)CC4)C3)C=C2)C1	C40H43BrN8O6S	KAT2A;KAT2B	Q92830/Q92831	CRBN	WO-2024003533-A1
TPD-3VXAGD	SCHEMBL27312902	4-[9-[2-[4-[(3R,5R)-5-[(6-bromo-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)amino]-1-methylpiperidin-3-yl]phenoxy]ethyl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN1C[C@H](NC2=C(Br)C(=O)N3C=CSC3=N2)C[C@H](C2=CC=C(OCCN3CCC4(CC3)CCN(C3=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C3)CC4)C=C2)C1	C42H47BrN8O6S	KAT2A;KAT2B	Q92830/Q92831	CRBN	WO-2024003533-A1
TPD-0DFZNS	SCHEMBL27312905	4-[4-[2-[4-[(3R,5R)-5-[(6-bromo-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)amino]-1-methylpiperidin-3-yl]phenoxy]ethoxy]piperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN1C[C@H](NC2=C(Br)C(=O)N3C=CSC3=N2)C[C@H](C2=CC=C(OCCOC3CCN(C4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)C=C2)C1	C38H40BrN7O7S	KAT2A;KAT2B	Q92830/Q92831	CRBN	WO-2024003533-A1
TPD-2T32YJ	SCHEMBL27312911	4-[[1-[2-[4-[(3R,5R)-5-[(6-bromo-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)amino]-1-methylpiperidin-3-yl]phenoxy]ethyl]piperidin-4-yl]-methylamino]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN1C[C@H](NC2=C(Br)C(=O)N3C=CSC3=N2)C[C@H](C2=CC=C(OCCN3CCC(N(C)C4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)C=C2)C1	C39H43BrN8O6S	KAT2A;KAT2B	Q92830/Q92831	CRBN	WO-2024003533-A1
TPD-NPX2DN	SCHEMBL27312914	4-[2-[2-[4-[(3R,5R)-5-[(6-bromo-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)amino]-1-methylpiperidin-3-yl]phenoxy]ethyl-methylamino]ethyl-methylamino]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN(CCOC1=CC=C([C@H]2C[C@@H](NC3=C(Br)C(=O)N4C=CSC4=N3)CN(C)C2)C=C1)CCN(C)C1=C2C(=O)N(C3CCC(=O)NC3=O)C(=O)C2=CC=C1	C37H41BrN8O6S	KAT2A;KAT2B	Q92830/Q92831	CRBN	WO-2024003533-A1
TPD-F4IJME	SCHEMBL27313065	4-[4-[4-[(3R,5R)-5-[(6-bromo-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)amino]-1-methylpiperidin-3-yl]phenoxy]butyl-methylamino]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN1C[C@H](NC2=C(Br)C(=O)N3C=CSC3=N2)C[C@H](C2=CC=C(OCCCCN(C)C3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)C=C2)C1	C36H38BrN7O6S	KAT2A;KAT2B	Q92830/Q92831	CRBN	WO-2024003533-A1
TPD-5IKGQK	SCHEMBL30746877	4-[3-[4-[(3R,5R)-5-[(6-bromo-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)amino]-1-methylpiperidin-3-yl]phenoxy]propyl-methylamino]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN1C[C@H](NC2=C(Br)C(=O)N3C=CSC3=N2)C[C@H](C2=CC=C(OCCCN(C)C3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)C=C2)C1	C35H36BrN7O6S	KAT2A;KAT2B	Q92830/Q92831	CRBN	WO-2024003533-A1
TPD-OQBKI6	SCHEMBL27313067	4-[4-[[4-[(3R,5R)-5-[(6-bromo-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)amino]-1-methylpiperidin-3-yl]phenoxy]methyl]piperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN1C[C@H](NC2=C(Br)C(=O)N3C=CSC3=N2)C[C@H](C2=CC=C(OCC3CCN(C4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)C=C2)C1	C37H38BrN7O6S	KAT2A;KAT2B	Q92830/Q92831	CRBN	WO-2024003533-A1
TPD-ZZP56Q	SCHEMBL30746876	4-[3-[[4-[(3R,5R)-5-[(6-bromo-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)amino]-1-methylpiperidin-3-yl]phenoxy]methyl]pyrrolidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN1C[C@H](NC2=C(Br)C(=O)N3C=CSC3=N2)C[C@H](C2=CC=C(OCC3CCN(C4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C3)C=C2)C1	C36H36BrN7O6S	KAT2A;KAT2B	Q92830/Q92831	CRBN	WO-2024003533-A1
TPD-CSOKNQ	SCHEMBL30746899	4-[5-[4-[(3R,5R)-5-[(6-bromo-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)amino]-1-methylpiperidin-3-yl]phenoxy]pentoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN1C[C@H](NC2=C(Br)C(=O)N3C=CSC3=N2)C[C@H](C2=CC=C(OCCCCCOC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)C=C2)C1	C36H37BrN6O7S	KAT2A;KAT2B	Q92830/Q92831	CRBN	WO-2024003533-A1
TPD-M83JFD	SCHEMBL27313181	4-[4-[4-[(3R,5R)-5-[(6-bromo-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)amino]-1-methylpiperidin-3-yl]phenoxy]butoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN1C[C@H](NC2=C(Br)C(=O)N3C=CSC3=N2)C[C@H](C2=CC=C(OCCCCOC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)C=C2)C1	C35H35BrN6O7S	KAT2A;KAT2B	Q92830/Q92831	CRBN	WO-2024003533-A1
TPD-LA9X60	SCHEMBL30746897	4-[[5-[[4-[(3R,5R)-5-[(6-bromo-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)amino]-1-methylpiperidin-3-yl]phenoxy]methyl]pyridin-2-yl]methoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione; SCHEMBL30746902	CN1C[C@H](NC2=C(Br)C(=O)N3C=CSC3=N2)C[C@H](C2=CC=C(OCC3=CC=C(COC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)N=C3)C=C2)C1	C38H34BrN7O7S	KAT2A;KAT2B	Q92830/Q92831	CRBN	WO-2024003533-A1
TPD-G25NHE	SCHEMBL27313185	4-[3-[2-[4-[(3R,5R)-5-[(6-bromo-5-oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)amino]-1-methylpiperidin-3-yl]phenoxy]ethoxy]piperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN1C[C@H](NC2=C(Br)C(=O)N3C=CSC3=N2)C[C@H](C2=CC=C(OCCOC3CCCN(C4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C3)C=C2)C1	C38H40BrN7O7S	KAT2A;KAT2B	Q92830/Q92831	CRBN	WO-2024003533-A1
TPD-7Q7847	CHEMBL4867584	N-[3-(3-chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl]-4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]benzamide; SCHEMBL20046414; SCHEMBL25059044; SCHEMBL25427977; SCHEMBL30622030; PD172150; PD172151	CC1(C)[C@H](NC(=O)c2ccc(N3CCC(CN4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)cc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C45H50ClN7O6	AR	P10275	CRBN	WO-2024006527-A1
TPD-HMJ1Q6	WO2024008097A1_7a	.	O=C1CCC(N2C(=O)c3cccc(NCCOCCN4CCN(c5ccc(Nc6ncc7ncc(=O)n(C8CCCC8)c7n6)cc5)CC4)c3C2=O)C(=O)N1	C38H42N10O6	CDK4;CDK6	P11802/Q00534	CRBN	WO-2024008097-A1
TPD-SBUZ0Q	WO2024008097A1_7b	.	O=C1CCC(N2C(=O)c3cccc(NCCOCCOCCN4CCN(c5ccc(Nc6ncc7ncc(=O)n(C8CCCC8)c7n6)cc5)CC4)c3C2=O)C(=O)N1	C40H46N10O7	CDK4;CDK6	P11802/Q00534	CRBN	WO-2024008097-A1
TPD-M1RH5P	WO2024008097A1_7c	6-[4-[4-[(8-cyclopentyl-7-oxopteridin-2-yl)amino]phenyl]piperazin-1-yl]-N-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]hexanamide	O=C1CCC(N2C(=O)c3cccc(NC(=O)CCCCCN4CCN(c5ccc(Nc6ncc7ncc(=O)n(C8CCCC8)c7n6)cc5)CC4)c3C2=O)C(=O)N1	C40H44N10O6	CDK4;CDK6	P11802/Q00534	CRBN	WO-2024008097-A1
TPD-D0DYAL	WO2024008097A1_7d	7-[4-[4-[(8-cyclopentyl-7-oxopteridin-2-yl)amino]phenyl]piperazin-1-yl]-N-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]heptanamide	O=C1CCC(N2C(=O)c3cccc(NC(=O)CCCCCCN4CCN(c5ccc(Nc6ncc7ncc(=O)n(C8CCCC8)c7n6)cc5)CC4)c3C2=O)C(=O)N1	C41H46N10O6	CDK4;CDK6	P11802/Q00534	CRBN	WO-2024008097-A1
TPD-LWVWC2	WO2024008097A1_7e	8-[4-[4-[(8-cyclopentyl-7-oxopteridin-2-yl)amino]phenyl]piperazin-1-yl]-N-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]-8-oxooctanamide	O=C1CCC(N2C(=O)c3cccc(NC(=O)CCCCCCC(=O)N4CCN(c5ccc(Nc6ncc7ncc(=O)n(C8CCCC8)c7n6)cc5)CC4)c3C2=O)C(=O)N1	C42H46N10O7	CDK4;CDK6	P11802/Q00534	CRBN	WO-2024008097-A1
TPD-LDBAOV	PROTAC CDK4/6 degrader 1	PROTAC CDK4/6 degrader 1; 3025082-14-5; orb2646121; EX-A13402; HY-163786	O=C(CCCCN1CCN(c2ccc(Nc3ncc4ncc(=O)n(C5CCCC5)c4n3)cc2)CC1)NCCNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O	C41H47N11O6	CDK4;CDK6	P11802/Q00534	CRBN	WO-2024008097-A1
TPD-RYEHEI	WO2024008097A1_7g	.	O=C(CCCCCN1CCN(c2ccc(Nc3ncc4ncc(=O)n(C5CCCC5)c4n3)cc2)CC1)NCCNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O	C42H49N11O6	CDK4;CDK6	P11802/Q00534	CRBN	WO-2024008097-A1
TPD-X7PM89	SCHEMBL29170288	2-[4-[4-[(8-cyclopentyl-7-oxopteridin-2-yl)amino]phenyl]piperazin-1-yl]-N-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]butyl]acetamide	O=C(CN1CCN(c2ccc(Nc3ncc4ncc(=O)n(C5CCCC5)c4n3)cc2)CC1)NCCCCNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O	C40H45N11O6	CDK4;CDK6	P11802/Q00534	CRBN	WO-2024008097-A1
TPD-UPSCH8	WO2024008097A1_7i	.	O=C1CCC(N2C(=O)c3cccc(NC(=O)CCCCCn4cc(CN5CCN(c6ccc(Nc7ncc8ncc(=O)n(C9CCCC9)c8n7)cc6)CC5)nn4)c3C2=O)C(=O)N1	C43H47N13O6	CDK4;CDK6	P11802/Q00534	CRBN	WO-2024008097-A1
TPD-1RACKE	WO2024008097A1_7j	.	O=C1CCC(N2C(=O)c3ccc(N4CCC(CN5CCN(c6ccc(Nc7ncc8ncc(=O)n(C9CCCC9)c8n7)cc6)CC5)CC4)cc3C2=O)C(=O)N1	C40H44N10O5	CDK4;CDK6	P11802/Q00534	CRBN	WO-2024008097-A1
TPD-4UYCRY	WO2024008097A1_7k	.	O=C1CCC(N2C(=O)c3ccc(N4CCN(CC5CCN(C(=O)CN6CCN(c7ccc(Nc8ncc9ncc(=O)n(C%10CCCC%10)c9n8)cc7)CC6)CC5)CC4)cc3C2=O)C(=O)N1	C46H54N12O6	CDK4;CDK6	P11802/Q00534	CRBN	WO-2024008097-A1
TPD-HT2W6R	WO2024008097A1_7l	.	O=C1CCC(N2C(=O)c3ccc(N4CCN(C(=O)CN5CCN(c6ccc(Nc7ncc8ncc(=O)n(C9CCCC9)c8n7)cc6)CC5)CC4)cc3C2=O)C(=O)N1	C40H43N11O6	CDK4;CDK6	P11802/Q00534	CRBN	WO-2024008097-A1
TPD-CU3295	WO2024010818A2_1	.	C[C@](O)(CNCCCCC(=O)Nc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O)C(=O)Nc1ccc(C#N)c(C(F)(F)F)c1	C30H29F3N6O7	AR	P10275	CRBN	WO-2024010818-A2
TPD-3DZ14B	WO2024010818A2_10	.	C[C@](O)(Cn1cc(F)cn1)C(=O)N(CC(=O)CCCCCCC(=O)Nc1ccc2c(c1)CN(C1CCC(=O)NC1=O)C2=O)c1ccc(C#N)c(C(F)(F)F)c1	C37H37F4N7O7	AR	P10275	CRBN	WO-2024010818-A2
TPD-3TBRC6	WO2024010818A2_11	.	C[C@](O)(Cn1cc(F)cn1)C(=O)N(CC(=O)CCCCCCC(=O)Nc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O)c1ccc(C#N)c(C(F)(F)F)c1	C37H35F4N7O8	AR	P10275	CRBN	WO-2024010818-A2
TPD-CLLBWJ	WO2024010818A2_12	.	C[C@](O)(Cn1cc(F)cn1)C(=O)N(CC(=O)CCCCCCC(=O)Nc1ccc2c(c1)C(=O)N(C1CCC(=O)NC1=O)C2=O)c1ccc(C#N)c(C(F)(F)F)c1	C37H35F4N7O8	AR	P10275	CRBN	WO-2024010818-A2
TPD-45AFZY	WO2024010818A2_13	.	CN(C(=O)[C@](C)(Cn1cc(F)cn1)OCc1ccc(N2CCN(C3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)cc1)c1ccc(C#N)c(C(F)(F)F)c1	C45H45F4N9O6	AR	P10275	CRBN	WO-2024010818-A2
TPD-MO0V59	WO2024010818A2_14	.	CN(C(=O)[C@](C)(Cn1cc(F)cn1)OCc1ccc(N2CCN(CC3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)cc1)c1ccc(C#N)c(C(F)(F)F)c1	C46H47F4N9O6	AR	P10275	CRBN	WO-2024010818-A2
TPD-50UL2A	WO2024010818A2_15	.	C=C(CO[C@@](C)(Cn1cc(F)cn1)C(=O)N(C)c1ccc(C#N)c(C(F)(F)F)c1)C(=O)N1CCN(C2CCN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)CC1	C42H43F4N9O7	AR	P10275	CRBN	WO-2024010818-A2
TPD-6V6OPN	WO2024010818A2_16	.	C=C(CO[C@@](C)(Cn1cc(F)cn1)C(=O)N(C)c1ccc(C#N)c(C(F)(F)F)c1)C(=O)N1CCN(CC2CCN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)CC1	C43H45F4N9O7	AR	P10275	CRBN	WO-2024010818-A2
TPD-4TNNGP	WO2024010818A2_17	.	C=C(CO[C@@](C)(Cn1cc(F)cn1)C(=O)Nc1ccc(C#N)c(C(F)(F)F)c1)C(=O)NCCCCC(=O)Nc1cccc2c1CN(C1CCC(=O)NC1=O)C2=O	C37H36F4N8O7	AR	P10275	CRBN	WO-2024010818-A2
TPD-WWT8U0	WO2024010818A2_18	.	C=C(CO[C@@](C)(Cn1cc(F)cn1)C(=O)Nc1ccc(C#N)c(C(F)(F)F)c1)C(=O)NCCCCC(=O)Nc1ccc2c(c1)CN(C1CCC(=O)NC1=O)C2=O	C37H36F4N8O7	AR	P10275	CRBN	WO-2024010818-A2
TPD-KNVPTB	WO2024010818A2_19	.	C=C(CO[C@@](C)(Cn1cc(F)cn1)C(=O)Nc1ccc(C#N)c(C(F)(F)F)c1)C(=O)NCCCCC(=O)Nc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O	C37H34F4N8O8	AR	P10275	CRBN	WO-2024010818-A2
TPD-POUP1L	WO2024010818A2_2	.	C[C@](O)(CNCCCCC(=O)Nc1cccc2c1CN(C1CCC(=O)NC1=O)C2=O)C(=O)Nc1ccc(C#N)c(C(F)(F)F)c1	C30H31F3N6O6	AR	P10275	CRBN	WO-2024010818-A2
TPD-ZA23K5	WO2024010818A2_20	.	C=C(CO[C@@](C)(Cn1cc(F)cn1)C(=O)Nc1ccc(C#N)c(C(F)(F)F)c1)C(=O)NCCCCC(=O)Nc1ccc2c(c1)C(=O)N(C1CCC(=O)NC1=O)C2=O	C37H34F4N8O8	AR	P10275	CRBN	WO-2024010818-A2
TPD-31KBDB	WO2024010818A2_21	.	C=C(CN(C(=O)[C@@](C)(O)Cn1cc(F)cn1)c1ccc(C#N)c(C(F)(F)F)c1)C(=O)NCCCCC(=O)Nc1cccc2c1CN(C1CCC(=O)NC1=O)C2=O	C37H36F4N8O7	AR	P10275	CRBN	WO-2024010818-A2
TPD-GU5D0I	WO2024010818A2_22	.	C=C(CN(C(=O)[C@@](C)(O)Cn1cc(F)cn1)c1ccc(C#N)c(C(F)(F)F)c1)C(=O)NCCCCC(=O)Nc1ccc2c(c1)CN(C1CCC(=O)NC1=O)C2=O	C37H36F4N8O7	AR	P10275	CRBN	WO-2024010818-A2
TPD-879IX1	WO2024010818A2_23	.	C=C(CN(C(=O)[C@@](C)(O)Cn1cc(F)cn1)c1ccc(C#N)c(C(F)(F)F)c1)C(=O)NCCCCC(=O)Nc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O	C37H34F4N8O8	AR	P10275	CRBN	WO-2024010818-A2
TPD-6NCPXY	WO2024010818A2_24	.	C=C(CN(C(=O)[C@@](C)(O)CN(/C=C/F)/N=C\C)c1ccc(C#N)c(C(F)(F)F)c1)C(=O)NCCCCC(=O)Nc1ccc2c(c1)C(=O)N(C1CCC(=O)NC1=O)C2=O	C38H38F4N8O8	AR	P10275	CRBN	WO-2024010818-A2
TPD-2XOL10	SCHEMBL25475790	N-[1-[(2S)-3-[4-cyano-3-(trifluoromethyl)anilino]-2-hydroxy-2-methyl-3-oxopropyl]pyrazol-4-yl]-5-[(4S)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]pentanamide; SCHEMBL30754444	C[C@](O)(Cn1cc(NC(=O)CCCC[C@@H]2SCC3NC(=O)NC32)cn1)C(=O)Nc1ccc(C#N)c(C(F)(F)F)c1	C25H28F3N7O4S	AR	P10275	CRBN	WO-2024010818-A2
TPD-6LC36D	WO2024010818A2_26	.	C[C@@](Cn1cc(F)cn1)(OC(=O)CCCC[C@@H]1SCC2NC(=O)NC21)C(=O)Nc1ccc(C#N)c(C(F)(F)F)c1	C25H26F4N6O4S	AR	P10275	CRBN	WO-2024010818-A2
TPD-VJOTZZ	WO2024010818A2_27	.	C[C@](O)(Cn1cc(F)cn1)C(=O)N(C(=O)CCCC[C@@H]1SCC2NC(=O)NC21)c1ccc(C#N)c(C(F)(F)F)c1	C25H26F4N6O4S	AR	P10275	CRBN	WO-2024010818-A2
TPD-2P6V7X	WO2024010818A2_28	.	CN(C)S(=O)(=O)c1ccc(NCCNC(=O)CO[C@@](C)(Cn2cc(F)cn2)C(=O)Nc2ccc(C#N)c(C(F)(F)F)c2)c2nonc12	C27H27F4N9O6S	AR	P10275	CRBN	WO-2024010818-A2
TPD-VNVDZX	WO2024010818A2_29	.	CN(C)S(=O)(=O)c1ccc(NCCNC(=O)CN(C(=O)[C@@H](O)Cn2cc(F)cn2)c2ccc(C#N)c(C(F)(F)F)c2)c2nonc12	C26H25F4N9O6S	AR	P10275	CRBN	WO-2024010818-A2
TPD-0DGD8E	WO2024010818A2_3	.	C[C@](O)(CNCCCCC(=O)Nc1ccc2c(c1)C(=O)N(C1CCC(=O)NC1=O)C2=O)C(=O)Nc1ccc(C#N)c(C(F)(F)F)c1	C30H29F3N6O7	AR	P10275	CRBN	WO-2024010818-A2
TPD-7ENMB5	WO2024010818A2_30	.	CN(C)S(=O)(=O)c1ccc(NCCNC(=O)c2cnn(C[C@](C)(O)C(=O)Nc3ccc(C#N)c(C(F)(F)F)c3)c2)c2nonc12	C26H26F3N9O6S	AR	P10275	CRBN	WO-2024010818-A2
TPD-US6ZO5	WO2024010818A2_4	.	C[C@](O)(CNCCCCC(=O)Nc1ccc2c(c1)C(=O)N(C1CCC(=O)NC1=O)C2)C(=O)Nc1ccc(C#N)c(C(F)(F)F)c1	C30H31F3N6O6	AR	P10275	CRBN	WO-2024010818-A2
TPD-DVEOC6	WO2024010818A2_5	.	C[C@@](Cn1cc(F)cn1)(OCC(=O)CCCCCCC(=O)Nc1cccc2c1CN(C1CCC(=O)NC1=O)C2=O)C(=O)Nc1ccc(C#N)c(C(F)(F)F)c1	C37H37F4N7O7	AR	P10275	CRBN	WO-2024010818-A2
TPD-COTY1I	WO2024010818A2_6	.	C[C@@](Cn1cc(F)cn1)(OCC(=O)CCCCCCC(=O)Nc1ccc2c(c1)CN(C1CCC(=O)NC1=O)C2=O)C(=O)Nc1ccc(C#N)c(C(F)(F)F)c1	C37H37F4N7O7	AR	P10275	CRBN	WO-2024010818-A2
TPD-WE9F46	WO2024010818A2_7	.	C[C@@](Cn1cc(F)cn1)(OCC(=O)CCCCCCC(=O)Nc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O)C(=O)Nc1ccc(C#N)c(C(F)(F)F)c1	C37H35F4N7O8	AR	P10275	CRBN	WO-2024010818-A2
TPD-DEZ3CV	WO2024010818A2_8	.	C[C@@](Cn1cc(F)cn1)(OCC(=O)CCCCCCC(=O)Nc1ccc2c(c1)C(=O)N(C1CCC(=O)NC1=O)C2=O)C(=O)Nc1ccc(C#N)c(C(F)(F)F)c1	C37H35F4N7O8	AR	P10275	CRBN	WO-2024010818-A2
TPD-GEIBMI	WO2024010818A2_9	.	C[C@](O)(Cn1cc(F)cn1)C(=O)N(CC(=O)CCCCCCC(=O)Nc1cccc2c1CN(C1CCC(=O)NC1=O)C2=O)c1ccc(C#N)c(C(F)(F)F)c1	C37H37F4N7O7	AR	P10275	CRBN	WO-2024010818-A2
TPD-OFUMN9	SCHEMBL26985752	(2S)-N-[4-cyano-3-(trifluoromethyl)phenyl]-3-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]-2-hydroxy-2-methylpropanamide	C[C@](O)(CN1CCN(CC2CCN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)CC1)C(=O)Nc1ccc(C#N)c(C(F)(F)F)c1	C35H38F3N7O6	AR	P10275	CRBN	WO-2024010818-A2
TPD-BYDN9P	SCHEMBL26985687	(2S)-N-[4-cyano-3-(trifluoromethyl)phenyl]-3-[4-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]pyrazol-1-yl]-2-hydroxy-2-methylpropanamide	C[C@](O)(Cn1cc(-c2ccc(N3CCC(CN4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)cc2)cn1)C(=O)Nc1ccc(C#N)c(C(F)(F)F)c1	C44H44F3N9O6	AR	P10275	CRBN	WO-2024010818-A2
TPD-M7ADE7	SCHEMBL26985846	(2S)-N-[4-cyano-3-(trifluoromethyl)phenyl]-3-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]pyrazol-1-yl]-2-hydroxy-2-methylpropanamide	C[C@](O)(Cn1cc(N2CCC(CN3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)cn1)C(=O)Nc1ccc(C#N)c(C(F)(F)F)c1	C38H40F3N9O6	AR	P10275	CRBN	WO-2024010818-A2
TPD-5924S6	SCHEMBL26985673	(2S)-N-[4-cyano-2-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]-5-(trifluoromethyl)phenyl]-3-(4-fluoropyrazol-1-yl)-2-hydroxy-2-methylpropanamide	C[C@](O)(Cn1cc(F)cn1)C(=O)Nc1cc(C(F)(F)F)c(C#N)cc1N1CCC(CN2CCN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)CC1	C38H39F4N9O6	AR	P10275	CRBN	WO-2024010818-A2
TPD-LP5NVO	WO2024012449A1_1	.	CC1(C)CCC(CN2CCN(c3ccc(C(=O)NS(=O)(=O)c4ccc(NCC5CCN(C6CCN(CCCSc7cccc8c7CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)c([N+](=O)[O-])c4)c(Oc4cnc5[nH]ccc5c4)c3)CC2)=C(c2ccc(C(F)(F)F)cc2)C1	C67H76F3N11O9S2	BCL2L1	Q07817	CRBN	WO-2024012449-A1
TPD-M0BNH8	WO2024012449A1_2	.	CC1(C)CCC(CN2CCN(c3ccc(C(=O)NS(=O)(=O)c4ccc(NCC5CCN(C6CCN(CCCCSc7cccc8c7CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)c([N+](=O)[O-])c4)c(Oc4cnc5[nH]ccc5c4)c3)CC2)=C(c2ccc(C(F)(F)F)cc2)C1	C68H78F3N11O9S2	BCL2L1	Q07817	CRBN	WO-2024012449-A1
TPD-Y9LFXU	WO2024012449A1_3	.	CC1(C)CCC(CN2CCN(c3ccc(C(=O)NS(=O)(=O)c4ccc(NCC5CCN(C6CCN(CCCCCSc7cccc8c7CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)c([N+](=O)[O-])c4)c(Oc4cnc5[nH]ccc5c4)c3)CC2)=C(c2ccc(C(F)F)cc2)C1	C69H81F2N11O9S2	BCL2L1	Q07817	CRBN	WO-2024012449-A1
TPD-53BA38	WO2024012449A1_4	.	CC1(C)CCC(CN2CCN(c3ccc(C(=O)NS(=O)(=O)c4ccc(NCC5CCN(C6CCN(CCCCOc7cccc8c7CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)c([N+](=O)[O-])c4)c(Oc4cnc5[nH]ccc5c4)c3)CC2)=C(c2ccc(C(F)(F)F)cc2)C1	C68H78F3N11O10S	BCL2L1	Q07817	CRBN	WO-2024012449-A1
TPD-N178OI	WO2024012449A1_5	.	CC1(C)CCC(CN2CCN(c3ccc(C(=O)NS(=O)(=O)c4ccc(NCC5CCN(C6CCN(CCCCCOc7cccc8c7CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)c([N+](=O)[O-])c4)c(Oc4cnc5[nH]ccc5c4)c3)CC2)=C(c2ccc(C(F)(F)F)cc2)C1	C69H80F3N11O10S	BCL2L1	Q07817	CRBN	WO-2024012449-A1
TPD-S1181W	WO2024012449A1_6	.	CN(CCCC#Cc1cccc2c1CN(C1CCC(=O)NC1=O)C2=O)CCN1CCC(CNc2ccc(S(=O)(=O)NC(=O)c3ccc(C4CCN(CC5=C(c6ccc(C(F)(F)F)cc6)CC(C)(C)CC5)CC4)cc3Oc3cnc4[nH]ccc4c3)cc2[N+](=O)[O-])CC1	C68H75F3N10O9S	BCL2L1	Q07817	CRBN	WO-2024012449-A1
TPD-G3WN9L	WO2024012449A1_7	.	CC1(C)CCC(CN2CCN(c3ccc(C(=O)NS(=O)(=O)c4ccc(NCC5CCN(C6CCN(CCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)c([N+](=O)[O-])c4)c(Oc4cnc5[nH]ccc5c4)c3)CC2)=C(c2ccc(C(F)(F)F)cc2)C1	C67H75F3N12O10S	BCL2L1	Q07817	CRBN	WO-2024012449-A1
TPD-A4ANBO	WO2024012449A1_8	.	CC1(C)CCC(CN2CCN(c3ccc(C(=O)NS(=O)(=O)c4ccc(NCC5CCN(C6CCN(CCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)c([N+](=O)[O-])c4)c(Oc4cnc5[nH]ccc5c4)c3)CC2)=C(c2ccc(C(F)(F)F)cc2)C1	C68H77F3N12O10S	BCL2L1	Q07817	CRBN	WO-2024012449-A1
TPD-S281OT	WO2024012449A1_9	.	CC1(C)CCC(CN2CCN(c3ccc(C(=O)NS(=O)(=O)c4ccc(NCC5CCN(C6CCN(CCCCCNc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)c([N+](=O)[O-])c4)c(Oc4cnc5[nH]ccc5c4)c3)CC2)=C(c2ccc(C(F)(F)F)cc2)C1	C69H79F3N12O10S	BCL2L1	Q07817	CRBN	WO-2024012449-A1
TPD-QWOU88	WO2024012449A1_10	.	CC1(C)CCC(CN2CCN(c3ccc(C(=O)NS(=O)(=O)c4ccc(NCC5CCN(CCCCCNc6cccc7c6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)c([N+](=O)[O-])c4)c(Oc4cnc5[nH]ccc5c4)c3)CC2)=C(c2ccc(C(F)(F)F)cc2)C1	C64H70F3N11O10S	BCL2L1	Q07817	CRBN	WO-2024012449-A1
TPD-P9P9XP	WO2024012449A1_11	.	CC1(C)CCC(CN2CCN(c3ccc(C(=O)NS(=O)(=O)c4ccc(NCC5CCN(C6CCN(CCCCNc7cccc8c7CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)c([N+](=O)[O-])c4)c(Oc4cnc5[nH]ccc5c4)c3)CC2)=C(c2ccc(CF)cc2)C1	C68H81FN12O9S	BCL2L1	Q07817	CRBN	WO-2024012449-A1
TPD-EUWLWO	WO2024012449A1_12	.	CC1(C)CCC(CN2CCN(c3ccc(C(=O)NS(=O)(=O)c4ccc(NCC5CCN(C6CCN(CCCCCCC#Cc7cccc8c7CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)c([N+](=O)[O-])c4)c(Oc4cnc5[nH]ccc5c4)c3)CC2)=C(c2ccc(C(F)(F)F)cc2)C1	C72H82F3N11O9S	BCL2L1	Q07817	CRBN	WO-2024012449-A1
TPD-PKZGAX	WO2024012449A1_13	.	CC1(C)CCC(CN2CCN(c3ccc(C(=O)NS(=O)(=O)c4ccc(NCC5CCN(C6CCN(CCCC#Cc7cccc8c7CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)c([N+](=O)[O-])c4)c(Oc4cnc5[nH]ccc5c4)c3)CC2)=C(c2ccc(C(F)(F)F)cc2)C1	C69H76F3N11O9S	BCL2L1	Q07817	CRBN	WO-2024012449-A1
TPD-VWGFAV	WO2024012449A1_14	.	CC1(C)CCC(CN2CCN(c3ccc(C(=O)NS(=O)(=O)c4ccc(NCC5CCN(C6CCN(CCCCCC#Cc7cccc8c7CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)c([N+](=O)[O-])c4)c(Oc4cnc5[nH]ccc5c4)c3)CC2)=C(c2ccc(C(F)(F)F)cc2)C1	C71H80F3N11O9S	BCL2L1	Q07817	CRBN	WO-2024012449-A1
TPD-QHTM8T	WO2024012449A1_16	.	CC1(C)CCC(CN2CCN(c3ccc(C(=O)NS(=O)(=O)c4ccc(NCC5CCN(C6CCN(CCCCCCCCC#Cc7cccc8c7CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)c([N+](=O)[O-])c4)c(Oc4cnc5[nH]ccc5c4)c3)CC2)=C(c2ccc(C(F)(F)F)cc2)C1	C74H86F3N11O9S	BCL2L1	Q07817	CRBN	WO-2024012449-A1
TPD-LCXHEO	WO2024012449A1_17	.	CC1(C)CCC(CN2CCN(c3ccc(C(=O)NS(=O)(=O)c4ccc(NCC5CCN(C6CCN(CCCCCCCCCC#Cc7cccc8c7CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)c([N+](=O)[O-])c4)c(Oc4cnc5[nH]ccc5c4)c3)CC2)=C(c2ccc(C(F)(F)F)cc2)C1	C75H88F3N11O9S	BCL2L1	Q07817	CRBN	WO-2024012449-A1
TPD-8JEEFT	WO2024012449A1_18	.	CC1(C)CCC(CN2CCN(c3ccc(C(=O)NS(=O)(=O)c4ccc(NCC5CCN(C6CCN(CCCCC#Cc7cccc8c7CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)c([N+](=O)[O-])c4)c(Oc4cnc5[nH]ccc5c4)c3)CC2)=C(c2ccc(C(F)(F)F)cc2)C1	C70H78F3N11O9S	BCL2L1	Q07817	CRBN	WO-2024012449-A1
TPD-6D244L	WO2024012449A1_19	.	CC1(C)CCC(CN2CCN(c3ccc(C(=O)NS(=O)(=O)c4ccc(NCC5CCN(C6CCN(CCCCCCOc7cccc8c7CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)c([N+](=O)[O-])c4)c(Oc4cnc5[nH]ccc5c4)c3)CC2)=C(c2ccc(C(F)(F)F)cc2)C1	C70H82F3N11O10S	BCL2L1	Q07817	CRBN	WO-2024012449-A1
TPD-UQCJ6D	WO2024012449A1_20	.	CC1(C)CCC(CN2CCN(c3ccc(C(=O)NS(=O)(=O)c4ccc(NCC5CCN(C6CCN(CCCCCCCOc7cccc8c7CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)c([N+](=O)[O-])c4)c(Oc4cnc5[nH]ccc5c4)c3)CC2)=C(c2ccc(C(F)(F)F)cc2)C1	C71H84F3N11O10S	BCL2L1	Q07817	CRBN	WO-2024012449-A1
TPD-C4YO8K	WO2024012449A1_21	.	CC1(C)CCC(CN2CCN(c3ccc(C(=O)NS(=O)(=O)c4ccc(NCC5CCN(C6CCN(CCCCCCCCOc7cccc8c7CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)c([N+](=O)[O-])c4)c(Oc4cnc5[nH]ccc5c4)c3)CC2)=C(c2ccc(C(F)(F)F)cc2)C1	C72H86F3N11O10S	BCL2L1	Q07817	CRBN	WO-2024012449-A1
TPD-YCPABZ	WO2024012449A1_22	.	CC1(C)CCC(CN2CCN(c3ccc(C(=O)NS(=O)(=O)c4ccc(NCC5CCN(C6CCN(CCCCCCCCCOc7cccc8c7CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)c([N+](=O)[O-])c4)c(Oc4cnc5[nH]ccc5c4)c3)CC2)=C(c2ccc(C(F)(F)F)cc2)C1	C73H88F3N11O10S	BCL2L1	Q07817	CRBN	WO-2024012449-A1
TPD-9285A4	WO2024012449A1_23	.	CC1(C)CCC(CN2CCN(c3ccc(C(=O)NS(=O)(=O)c4ccc(NCC5CCN(C6CCN(CCCCCCCCCCOc7cccc8c7CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)c([N+](=O)[O-])c4)c(Oc4cnc5[nH]ccc5c4)c3)CC2)=C(c2ccc(C(F)(F)F)cc2)C1	C74H90F3N11O10S	BCL2L1	Q07817	CRBN	WO-2024012449-A1
TPD-T4Y5FL	WO2024012449A1_24	.	CC1(C)CCC(CN2CCN(c3ccc(C(=O)NS(=O)(=O)c4ccc(NCC5CCN(C6CCN(CCCOc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)c([N+](=O)[O-])c4)c(Oc4cnc5[nH]ccc5c4)c3)CC2)=C(c2ccc(C(F)(F)F)cc2)C1	C67H74F3N11O11S	BCL2L1	Q07817	CRBN	WO-2024012449-A1
TPD-CN9WDI	WO2024012449A1_25	.	CC1(C)CCC(CN2CCN(c3ccc(C(=O)NS(=O)(=O)c4ccc(NCC5CCN(C6CCN(CCCCOc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)c([N+](=O)[O-])c4)c(Oc4ccc5[nH]ccc5c4)c3)CC2)=C(c2ccc(C(F)(F)F)cc2)C1	C69H77F3N10O11S	BCL2L1	Q07817	CRBN	WO-2024012449-A1
TPD-3S7V78	WO2024012449A1_26	.	CC1(C)CCC(CN2CCN(c3ccc(C(=O)NS(=O)(=O)c4ccc(NCC5CCN(C6CCN(CCCCCCOc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)c([N+](=O)[O-])c4)c(Oc4cnc5[nH]ccc5c4)c3)CC2)=C(c2ccc(C(F)(F)F)cc2)C1	C70H80F3N11O11S	BCL2L1	Q07817	CRBN	WO-2024012449-A1
TPD-90LKYC	WO2024012449A1_27	.	CC1(C)CCC(CN2CCN(c3ccc(C(=O)NS(=O)(=O)c4ccc(NCC5CCN(C6CCN(CCCCCCCOc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)c([N+](=O)[O-])c4)c(Oc4cnc5[nH]ccc5c4)c3)CC2)=C(c2ccc(C(F)(F)F)cc2)C1	C71H82F3N11O11S	BCL2L1	Q07817	CRBN	WO-2024012449-A1
TPD-5EUFY4	WO2024012449A1_28	.	CC1(C)CCC(CN2CCN(c3ccc(C(=O)NS(=O)(=O)c4ccc(NCC5CCN(C6CCN(CCCCCOc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)c([N+](=O)[O-])c4)c(Oc4cnc5[nH]ccc5c4)c3)CC2)=C(c2ccc(C(F)(F)F)cc2)C1	C69H78F3N11O11S	BCL2L1	Q07817	CRBN	WO-2024012449-A1
TPD-5HI5NO	WO2024012449A1_29	.	CC1(C)CCC(CN2CCN(c3ccc(C(=O)NS(=O)(=O)c4ccc(NCC5CCN(C6CCN(CCCCCCSc7cccc8c7CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)c([N+](=O)[O-])c4)c(Oc4cnc5[nH]ccc5c4)c3)CC2)=C(c2ccc(C(F)(F)F)cc2)C1	C70H82F3N11O9S2	BCL2L1	Q07817	CRBN	WO-2024012449-A1
TPD-3E5HDO	WO2024012449A1_30	.	CC1(C)CCC(CN2CCN(c3ccc(C(=O)NS(=O)(=O)c4ccc(NCC5CCN(C6CCN(CCCCCCCSc7cccc8c7CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)c([N+](=O)[O-])c4)c(Oc4cnc5[nH]ccc5c4)c3)CC2)=C(c2ccc(C(F)(F)F)cc2)C1	C71H84F3N11O9S2	BCL2L1	Q07817	CRBN	WO-2024012449-A1
TPD-OJZXKL	WO2024012449A1_31	.	CC1(C)CCC(CN2CCN(c3ccc(C(=O)NS(=O)(=O)c4ccc(NCC5CCN(C6CCN(CCCCCCCCSc7cccc8c7CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)c([N+](=O)[O-])c4)c(Oc4cnc5[nH]ccc5c4)c3)CC2)=C(c2ccc(C(F)(F)F)cc2)C1	C72H86F3N11O9S2	BCL2L1	Q07817	CRBN	WO-2024012449-A1
TPD-QLWPFO	WO2024012449A1_32	.	CC1(C)CCC(CN2CCN(c3ccc(C(=O)NS(=O)(=O)c4ccc(NCC5CCN(C6CCN(CCCCCCCCCSc7cccc8c7CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)c([N+](=O)[O-])c4)c(Oc4cnc5[nH]ccc5c4)c3)CC2)=C(c2ccc(C(F)(F)F)cc2)C1	C73H88F3N11O9S2	BCL2L1	Q07817	CRBN	WO-2024012449-A1
TPD-R7EYIF	WO2024012449A1_33	.	CC1(C)CCC(CN2CCN(c3ccc(C(=O)NS(=O)(=O)c4ccc(NCC5CCN(C6CCN(CCCC#Cc7cccc8c7C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)c([N+](=O)[O-])c4)c(Oc4cnc5[nH]ccc5c4)c3)CC2)=C(c2ccc(C(F)(F)F)cc2)C1	C69H74F3N11O10S	BCL2L1	Q07817	CRBN	WO-2024012449-A1
TPD-1K7NCS	WO2024012449A1_34	.	CC1(C)CCC(CN2CCN(c3ccc(C(=O)NS(=O)(=O)c4ccc(NCC5CCN(C6CCN(Cc7ccc(COc8cccc9c8CN(C8CCC(=O)NC8=O)C9=O)cc7)CC6)CC5)c([N+](=O)[O-])c4)c(Oc4cnc5[nH]ccc5c4)c3)CC2)=C(c2ccc(C(F)(F)F)cc2)C1	C72H78F3N11O10S	BCL2L1	Q07817	CRBN	WO-2024012449-A1
TPD-LS3ERQ	WO2024015340A1_CHR-106	(3R)-3-[(7S)-5-[[1-[2-fluoro-4-[(3S,4S)-7-hydroxy-3-phenyl-3,4-dihydro-2H-chromen-4-yl]-5-methoxyphenyl]piperidin-4-yl]methyl]-14-oxo-9-oxa-2,5,13-triazatetracyclo[8.7.0.02,7.011,15]heptadeca-1(10),11(15),16-trien-13-yl]piperidine-2,6-dione	[H][C@]12COC3=C(C=CC4=C3CN([C@@H]3CCC(=O)NC3=O)C4=O)N1CCN(CC1CCN(C3=CC(OC)=C([C@@H]4C5=C(C=C(O)C=C5)OC[C@@H]4C4=CC=CC=C4)C=C3F)CC1)C2	C46H48FN5O7	ERα	P03372	CRBN	WO-2024015340-A1
TPD-K204FS	SCHEMBL30719818	(3R)-3-[(7R)-5-[[2-[4-[(3R,4S)-7-hydroxy-3-phenyl-3,4-dihydro-2H-chromen-4-yl]phenyl]-2-azaspiro[3.5]nonan-7-yl]methyl]-13-oxo-9-oxa-2,5,14-triazatetracyclo[8.7.0.02,7.012,16]heptadeca-1(10),11,16-trien-14-yl]piperidine-2,6-dione	[H][C@@]12COC3=CC4=C(C=C3N1CCN(CC1CCC3(CC1)CN(C1=CC=C([C@H]5C6=C(C=C(O)C=C6)OC[C@H]5C5=CC=CC=C5)C=C1)C3)C2)CN([C@@H]1CCC(=O)NC1=O)C4=O	C48H51N5O6	ERα	P03372	CRBN	WO-2024015340-A1
TPD-5O85EG	WO2024015340A1_CHR-A59	.	[H][C@]12COC3=CC4=C(C=C3N1CCN(CC1CC3(CCN(C5=CC=C(C6C7=C(C=C(O)C=C7)OC[C@@H]6C6=CC=CC=C6)C=C5)CC3)C1)C2)CN([C@H]1CCC(=O)NC1=O)C4=O	C48H51N5O6	ERα	P03372	CRBN	WO-2024015340-A1
TPD-K2A4NX	SCHEMBL30719835	(3R)-3-[(7R)-5-[[7-[4-[(3S,4R)-7-hydroxy-3-phenyl-3,4-dihydro-2H-chromen-4-yl]phenyl]-7-azaspiro[3.5]nonan-2-yl]methyl]-14-oxo-9-oxa-2,5,13-triazatetracyclo[8.7.0.02,7.011,15]heptadeca-1(10),11(15),16-trien-13-yl]piperidine-2,6-dione	[H][C@@]12COC3=C(C=CC4=C3CN([C@@H]3CCC(=O)NC3=O)C4=O)N1CCN(CC1CC3(CCN(C4=CC=C([C@@H]5C6=C(C=C(O)C=C6)OC[C@@H]5C5=CC=CC=C5)C=C4)CC3)C1)C2	C48H51N5O6	ERα	P03372	CRBN	WO-2024015340-A1
TPD-XZN82P	SCHEMBL30719860	(3R)-3-[(7S)-5-[[7-[6-[(6S,8R)-7-[(1-fluorocyclopropyl)methyl]-8-methyl-3,6,8,9-tetrahydropyrazolo[4,3-f]isoquinolin-6-yl]pyridin-3-yl]-7-azaspiro[3.5]nonan-2-yl]methyl]-13-oxo-9-oxa-2,5,14-triazatetracyclo[8.7.0.02,7.012,16]heptadeca-1(10),11,16-trien-14-yl]piperidine-2,6-dione	C[C@@H]1CC2=C(C=CC3=C2C=NN3)[C@@H](C2=NC=C(N3CCC4(CC3)CC(CN3CCN5C6=CC7=C(C=C6OC[C@@H]5C3)C(=O)N([C@@H]3CCC(=O)NC3=O)C7)C4)C=C2)N1CC1(F)CC1	C47H54FN9O4	ERα	P03372	CRBN	WO-2024015340-A1
TPD-E5KWUB	WO2024015340A1_IDZ-A16	3-[(7R)-5-[[2-[6-[(6S,8R)-7-[(1-fluorocyclopropyl)methyl]-8-methyl-3,6,8,9-tetrahydropyrazolo[4,3-f]isoquinolin-6-yl]pyridin-3-yl]-2-azaspiro[3.5]nonan-7-yl]methyl]-14-oxo-9-oxa-2,5,13-triazatetracyclo[8.7.0.02,7.011,15]heptadeca-1(10),11(15),16-trien-13-yl]piperidine-2,6-dione	C[C@@H]1CC2=C(C=CC3=C2C=NN3)[C@@H](C2=NC=C(N3CC4(CCC(CN5CCN6C7=C(OC[C@H]6C5)C5=C(C=C7)C(=O)N(C6CCC(=O)NC6=O)C5)CC4)C3)C=C2)N1CC1(F)CC1	C47H54FN9O4	ERα	P03372	CRBN	WO-2024015340-A1
TPD-4D25E3	SCHEMBL30719816	(3S)-3-[(7R)-5-[[2-[5-[(6S,8R)-8-methyl-7-(2,2,2-trifluoroethyl)-3,6,8,9-tetrahydropyrazolo[4,3-f]isoquinolin-6-yl]pyridin-2-yl]-2-azaspiro[3.5]nonan-7-yl]methyl]-14-oxo-9-oxa-2,5,13-triazatetracyclo[8.7.0.02,7.011,15]heptadeca-1(10),11(15),16-trien-13-yl]piperidine-2,6-dione	C[C@@H]1CC2=C(C=CC3=C2C=NN3)[C@@H](C2=CC=C(N3CC4(CCC(CN5CCN6C7=C(OC[C@H]6C5)C5=C(C=C7)C(=O)N([C@H]6CCC(=O)NC6=O)C5)CC4)C3)N=C2)N1CC(F)(F)F	C45H50F3N9O4	ERα	P03372	CRBN	WO-2024015340-A1
TPD-VH8RMK	SCHEMBL30719770	(3S)-3-[(7R)-5-[[1-[5-[(6R,8R)-8-methyl-7-(2,2,2-trifluoroethyl)-3,6,8,9-tetrahydropyrazolo[4,3-f]isoquinolin-6-yl]pyridin-2-yl]piperidin-4-yl]methyl]-14-oxo-9-oxa-2,5,13-triazatetracyclo[8.7.0.02,7.011,15]heptadeca-1(10),11(15),16-trien-13-yl]piperidine-2,6-dione	C[C@@H]1CC2=C(C=CC3=C2C=NN3)[C@H](C2=CC=C(N3CCC(CN4CCN5C6=C(OC[C@H]5C4)C4=C(C=C6)C(=O)N([C@H]5CCC(=O)NC5=O)C4)CC3)N=C2)N1CC(F)(F)F	C42H46F3N9O4	ERα	P03372	CRBN	WO-2024015340-A1
TPD-4YAFR4	WO2024015340A1_IDZ-A21	(3S)-3-[(7R)-5-[[8-[5-[(6R,8R)-8-methyl-7-(2,2,2-trifluoroethyl)-3,6,8,9-tetrahydropyrazolo[4,3-f]isoquinolin-6-yl]pyridin-2-yl]-1-oxa-8-azaspiro[4.5]decan-3-yl]methyl]-14-oxo-9-oxa-2,5,13-triazatetracyclo[8.7.0.02,7.011,15]heptadeca-1(10),11(15),16-trien-13-yl]piperidine-2,6-dione	C[C@@H]1CC2=C(C=CC3=C2C=NN3)[C@H](C2=CC=C(N3CCC4(CC3)CC(CN3CCN5C6=C(OC[C@H]5C3)C3=C(C=C6)C(=O)N([C@H]5CCC(=O)NC5=O)C3)CO4)N=C2)N1CC(F)(F)F	C45H50F3N9O5	ERα	P03372	CRBN	WO-2024015340-A1
TPD-LGMDNP	SCHEMBL30719850	(3S)-3-[(7S)-5-[[1-[5-[(6S,8R)-8-methyl-7-(2,2,2-trifluoroethyl)-3,6,8,9-tetrahydropyrazolo[4,3-f]isoquinolin-6-yl]pyridin-2-yl]piperidin-4-yl]methyl]-13-oxo-9-oxa-2,5,14-triazatetracyclo[8.7.0.02,7.012,16]heptadeca-1(10),11,16-trien-14-yl]piperidine-2,6-dione	C[C@@H]1CC2=C(C=CC3=C2C=NN3)[C@@H](C2=CC=C(N3CCC(CN4CCN5C6=CC7=C(C=C6OC[C@@H]5C4)C(=O)N([C@H]4CCC(=O)NC4=O)C7)CC3)N=C2)N1CC(F)(F)F	C42H46F3N9O4	ERα	P03372	CRBN	WO-2024015340-A1
TPD-R25259	SCHEMBL30719862	(3S)-3-[(7R)-5-[[7-[5-[(6R,8R)-8-methyl-7-(2,2,2-trifluoroethyl)-3,6,8,9-tetrahydropyrazolo[4,3-f]isoquinolin-6-yl]pyridin-2-yl]-7-azaspiro[3.5]nonan-2-yl]methyl]-14-oxo-9-oxa-2,5,13-triazatetracyclo[8.7.0.02,7.011,15]heptadeca-1(10),11(15),16-trien-13-yl]piperidine-2,6-dione	C[C@@H]1CC2=C(C=CC3=C2C=NN3)[C@H](C2=CC=C(N3CCC4(CC3)CC(CN3CCN5C6=C(OC[C@H]5C3)C3=C(C=C6)C(=O)N([C@H]5CCC(=O)NC5=O)C3)C4)N=C2)N1CC(F)(F)F	C45H50F3N9O4	ERα	P03372	CRBN	WO-2024015340-A1
TPD-QAUVCU	SCHEMBL30719769	(3S)-3-[(7R)-5-[[7-[5-[(6S,8R)-8-methyl-7-(2,2,2-trifluoroethyl)-3,6,8,9-tetrahydropyrazolo[4,3-f]isoquinolin-6-yl]pyridin-2-yl]-7-azaspiro[3.5]nonan-2-yl]methyl]-14-oxo-9-oxa-2,5,13-triazatetracyclo[8.7.0.02,7.011,15]heptadeca-1(10),11(15),16-trien-13-yl]piperidine-2,6-dione	C[C@@H]1CC2=C(C=CC3=C2C=NN3)[C@@H](C2=CC=C(N3CCC4(CC3)CC(CN3CCN5C6=C(OC[C@H]5C3)C3=C(C=C6)C(=O)N([C@H]5CCC(=O)NC5=O)C3)C4)N=C2)N1CC(F)(F)F	C45H50F3N9O4	ERα	P03372	CRBN	WO-2024015340-A1
TPD-A6NCVD	WO2024015340A1_IND-A48	.	[H][C@@]12COC3=CC4=C(C=C3N1CCN(CC1CCN(C3=CC=C(C5C6=C(C[C@@H](C)N5CC(F)F)C5=C(C=CC=C5)N6)C(OC)=C3)CC1)C2)CN([C@@H]1CCC(=O)NC1=O)C4=O	C45H51F2N7O5	ERα	P03372	CRBN	WO-2024015340-A1
TPD-YU77OK	SCHEMBL30719806	(3S)-3-[(7R)-5-[[1-[4-[(1R,3R)-2-(2-fluoro-2-methylpropyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3-methoxyphenyl]piperidin-4-yl]methyl]-14-oxo-9-oxa-2,5,13-triazatetracyclo[8.7.0.02,7.011,15]heptadeca-1(10),11(15),16-trien-13-yl]piperidine-2,6-dione	COC1=CC(N2CCC(CN3CCN4C5=C(OC[C@H]4C3)C3=C(C=C5)C(=O)N([C@H]4CCC(=O)NC4=O)C3)CC2)=CC=C1[C@@H]1C2=C(C[C@@H](C)N1CC(C)(C)F)C1=CC=CC=C1N2	C47H56FN7O5	ERα	P03372	CRBN	WO-2024015340-A1
TPD-FO8E4W	SCHEMBL30719776	(10R)-12-[[1-[4-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3-methoxyphenyl]piperidin-4-yl]methyl]-N-(2,6-dioxopiperidin-3-yl)-8-oxa-1,6,12-triazatricyclo[8.4.0.02,7]tetradeca-2(7),3,5-triene-5-carboxamide	[H][C@@]12COC3=NC(C(=O)NC4CCC(=O)NC4=O)=CC=C3N1CCN(CC1CCN(C3=CC=C([C@@H]4C5=C(C[C@@H](C)N4CC(F)F)C4=C(C=CC=C4)N5)C(OC)=C3)CC1)C2	C43H50F2N8O5	ERα	P03372	CRBN	WO-2024015340-A1
TPD-6PK3X5	SCHEMBL30719819	(10R)-12-[[1-[4-[(1S,3S)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]-3-methoxyphenyl]piperidin-4-yl]methyl]-N-(2,6-dioxopiperidin-3-yl)-8-oxa-1,6,12-triazatricyclo[8.4.0.02,7]tetradeca-2(7),3,5-triene-5-carboxamide	[H][C@@]12COC3=NC(C(=O)NC4CCC(=O)NC4=O)=CC=C3N1CCN(CC1CCN(C3=CC=C([C@H]4C5=C(C[C@H](C)N4CC(F)F)C4=C(C=CC=C4)N5)C(OC)=C3)CC1)C2	C43H50F2N8O5	ERα	P03372	CRBN	WO-2024015340-A1
TPD-6DU4G9	WO2024015340A1_IND-A59	(3R)-3-[(7S)-5-[[(3S)-8-[5-[(1S,3S)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyrimidin-2-yl]-1-oxa-8-azaspiro[4.5]decan-3-yl]methyl]-14-oxo-9-oxa-2,5,13-triazatetracyclo[8.7.0.02,7.011,15]heptadeca-1(10),11(15),16-trien-13-yl]piperidine-2,6-dione	[H][C@]12COC3=C(C=CC4=C3CN([C@@H]3CCC(=O)NC3=O)C4=O)N1CCN(C[C@H]1COC3(CCN(C4=NC=C([C@H]5C6=C(C[C@H](C)N5CC(F)F)C5=C(C=CC=C5)N6)C=N4)CC3)C1)C2	C45H51F2N9O5	ERα	P03372	CRBN	WO-2024015340-A1
TPD-HW0WI7	SCHEMBL30719851	(3R)-3-[(7R)-5-[[(3S)-8-[5-[(1S,3S)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyrimidin-2-yl]-1-oxa-8-azaspiro[4.5]decan-3-yl]methyl]-13-oxo-9-oxa-2,5,14-triazatetracyclo[8.7.0.02,7.012,16]heptadeca-1(10),11,16-trien-14-yl]piperidine-2,6-dione	[H][C@@]12COC3=CC4=C(C=C3N1CCN(C[C@H]1COC3(CCN(C5=NC=C([C@H]6C7=C(C[C@H](C)N6CC(F)F)C6=C(C=CC=C6)N7)C=N5)CC3)C1)C2)CN([C@@H]1CCC(=O)NC1=O)C4=O	C45H51F2N9O5	ERα	P03372	CRBN	WO-2024015340-A1
TPD-R8UKX8	SCHEMBL30719830	(10R)-12-[[8-[5-[(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyrimidin-2-yl]-1-oxa-8-azaspiro[4.5]decan-3-yl]methyl]-N-[(3S)-2,6-dioxopiperidin-3-yl]-8-oxa-1,6,12-triazatricyclo[8.4.0.02,7]tetradeca-2(7),3,5-triene-5-carboxamide	[H][C@@]12COC3=NC(C(=O)N[C@H]4CCC(=O)NC4=O)=CC=C3N1CCN(CC1COC3(CCN(C4=NC=C([C@@H]5C6=C(C[C@@H](C)N5CC(F)F)C5=C(C=CC=C5)N6)C=N4)CC3)C1)C2	C43H50F2N10O5	ERα	P03372	CRBN	WO-2024015340-A1
TPD-KKZ2VC	SCHEMBL30719847	(3R)-3-[(7S)-5-[[(3S)-8-[5-[(1S,3S)-2-(2,2-difluoroethyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyrimidin-2-yl]-1-oxa-8-azaspiro[4.5]decan-3-yl]methyl]-13-oxo-9-oxa-2,5,14-triazatetracyclo[8.7.0.02,7.012,16]heptadeca-1(10),11,16-trien-14-yl]piperidine-2,6-dione	[H][C@]12COC3=CC4=C(C=C3N1CCN(C[C@H]1COC3(CCN(C5=NC=C([C@H]6C7=C(C[C@H](C)N6CC(F)F)C6=C(C=CC=C6)N7)C=N5)CC3)C1)C2)CN([C@@H]1CCC(=O)NC1=O)C4=O	C45H51F2N9O5	ERα	P03372	CRBN	WO-2024015340-A1
TPD-ZT2W98	SCHEMBL30719866	(3S)-3-[(7S)-5-[[1-[4-[(1R,2R)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]-3-methoxyphenyl]piperidin-4-yl]methyl]-13-oxo-9-oxa-2,5,14-triazatetracyclo[8.7.0.02,7.012,16]heptadeca-1(10),11,16-trien-14-yl]piperidine-2,6-dione	COC1=CC(N2CCC(CN3CCN4C5=C(C=C6C(=O)N([C@H]7CCC(=O)NC7=O)CC6=C5)OC[C@@H]4C3)CC2)=CC=C1[C@H]1C2=C(C=C(O)C=C2)CC[C@H]1C1=CC=CC=C1	C47H51N5O6	ERα	P03372	CRBN	WO-2024015340-A1
TPD-1OWYPK	WO2024015340A1_THP-A34	.	COC1=CC(N2CCC(CN3CCN4C5=C(C=C6C(=O)N([C@H]7CCC(=O)NC7=O)CC6=C5)OC[C@@H]4C3)CC2)=CC=C1[C@@H]1C2=C(C=C(O)C=C2)CC[C@@H]1C1=CC=CC=C1	C47H51N5O6	ERα	P03372	CRBN	WO-2024015340-A1
TPD-J7L5RY	SCHEMBL27263376	(3S)-3-[(7R)-5-[[1-[2-fluoro-4-[(1S,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]-5-methoxyphenyl]piperidin-4-yl]methyl]-14-oxo-9-oxa-2,5,13-triazatetracyclo[8.7.0.02,7.011,15]heptadeca-1(10),11(15),16-trien-13-yl]piperidine-2,6-dione; SCHEMBL30746300	COC1=CC(N2CCC(CN3CCN4C5=CC=C6C(=O)N([C@H]7CCC(=O)NC7=O)CC6=C5OC[C@H]4C3)CC2)=C(F)C=C1[C@@H]1C2=C(C=C(O)C=C2)CC[C@@H]1C1=CC=CC=C1	C47H50FN5O6	ERα	P03372	CRBN	WO-2024015340-A1
TPD-Z08Z6J	SCHEMBL27263406	(3S)-3-[(7R)-5-[[8-[4-[(1R,2R)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]-3-methoxyphenyl]-1-oxa-8-azaspiro[4.5]decan-3-yl]methyl]-14-oxo-9-oxa-2,5,13-triazatetracyclo[8.7.0.02,7.011,15]heptadeca-1(10),11(15),16-trien-13-yl]piperidine-2,6-dione; SCHEMBL30719803	COC1=CC(N2CCC3(CC2)CC(CN2CCN4C5=C(OC[C@H]4C2)C2=C(C=C5)C(=O)N([C@H]4CCC(=O)NC4=O)C2)CO3)=CC=C1[C@H]1C2=C(C=C(O)C=C2)CC[C@H]1C1=CC=CC=C1	C50H55N5O7	ERα	P03372	CRBN	WO-2024015340-A1
TPD-JL4664	SCHEMBL27263475	(3S)-3-[(7S)-5-[[8-[4-[(1R,2R)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]-3-methoxyphenyl]-1-oxa-8-azaspiro[4.5]decan-3-yl]methyl]-13-oxo-9-oxa-2,5,14-triazatetracyclo[8.7.0.02,7.012,16]heptadeca-1(10),11,16-trien-14-yl]piperidine-2,6-dione; SCHEMBL30746084	COC1=CC(N2CCC3(CC2)CC(CN2CCN4C5=CC6=C(C=C5OC[C@@H]4C2)C(=O)N([C@H]2CCC(=O)NC2=O)C6)CO3)=CC=C1[C@H]1C2=C(C=C(O)C=C2)CC[C@H]1C1=CC=CC=C1	C50H55N5O7	ERα	P03372	CRBN	WO-2024015340-A1
TPD-FZO633	SCHEMBL27263208	(3S)-3-[(7S)-5-[[2-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]-5-oxa-2-azaspiro[3.4]octan-7-yl]methyl]-13-oxo-9-oxa-2,5,14-triazatetracyclo[8.7.0.02,7.012,16]heptadeca-1(10),11,16-trien-14-yl]piperidine-2,6-dione	O=C1CC[C@H](N2CC3=C(C=C4OC[C@@H]5CN(CC6COC7(C6)CN(C6=CC=C([C@@H]8C9=C(C=C(O)C=C9)CC[C@@H]8C8=CC=CC=C8)C=C6)C7)CCN5C4=C3)C2=O)C(=O)N1	C47H49N5O6	ERα	P03372	CRBN	WO-2024015340-A1
TPD-QZRL3Y	WO2024017251A1_1	.	COc1cc(N2CCN(C(=O)CN3CCC(c4ccc(NC5CCC(=O)NC5=O)cc4)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCC2	C46H57BrN10O7S	EGFR	P00533	CRBN	WO-2024017251-A1
TPD-0WT7WY	WO2024017251A1_2	.	COc1cc(N2CCN(C(=O)CN3CCC(c4ccc5c(N6CCC(=O)NC6=O)nn(C)c5c4)C(F)(F)C3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCC2	C47H55BrF2N12O7S	EGFR	P00533	CRBN	WO-2024017251-A1
TPD-S3H9JB	WO2024017251A1_3	.	C=Cc1cnc2nc1Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCCc1cc(c(OC)cc1N1CCN(C(=O)CN3CCC(c4ccc(NC5CCC(=O)NC5=O)cc4)CC3)CC1)N2	C48H60N10O7S	EGFR	P00533	CRBN	WO-2024017251-A1
TPD-9OYPZ7	WO2024017251A1_4	.	C=Cc1cnc2nc1Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCCc1cc(c(OC)cc1N1CCN(C(=O)CN3CCC(c4ccc5c(N6CCC(=O)NC6=O)nn(C)c5c4)C(F)(F)C3)CC1)N2	C49H58F2N12O7S	EGFR	P00533	CRBN	WO-2024017251-A1
TPD-72HDS1	WO2024017251A1_5	.	COc1cc(N2CCC(CN3CCN(C(=O)[C@H](C)Nc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCC2	C50H60BrN11O9S	EGFR	P00533	CRBN	WO-2024017251-A1
TPD-I2KTW5	WO2024017251A1_6	.	CN(c1cc2ccc1Nc1nc(ncc1Br)Nc1cc(F)c(N3CCN(C(=O)CN4CCC(c5ccc6c(N7CCC(=O)NC7=O)nn(C)c6c5)C(F)(F)C4)CC3)c(c1)CCCCCO2)S(C)(=O)=O	C46H52BrF3N12O6S	EGFR	P00533	CRBN	WO-2024017251-A1
TPD-7J59RC	WO2024017251A1_7	.	COc1cc(N2CCN(C(=O)CN3CCC(c4ccc5c(C6CCC(=O)NC6=O)nn(C)c5c4)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCC2	C48H58BrN11O7S	EGFR	P00533	CRBN	WO-2024017251-A1
TPD-QLH6NC	WO2024017251A1_8	.	CN(c1cc2ccc1Nc1nc(ncc1Br)Nc1cc(F)c(N3CCN(C(=O)CN4CCC(c5ccc6c(C7CCC(=O)NC7=O)nn(C)c6c5)CC4)CC3)c(c1)CCCCCO2)S(C)(=O)=O	C47H55BrFN11O6S	EGFR	P00533	CRBN	WO-2024017251-A1
TPD-8H0HII	WO2024017251A1_9	.	COc1cc(N2CCN(C(=O)CN3CCN(c4ccc5c(C6CCC(=O)NC6=O)nn(C)c5c4)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCC2	C47H57BrN12O7S	EGFR	P00533	CRBN	WO-2024017251-A1
TPD-BQ98CE	WO2024017251A1_10	.	COc1cc(N2CCN(C(=O)CN3CCC(c4ccc5c(C6CCC(=O)NC6=O)nn(C)c5c4)C(F)(F)C3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCC2	C48H56BrF2N11O7S	EGFR	P00533	CRBN	WO-2024017251-A1
TPD-32RR3J	WO2024017251A1_11	.	CN(c1cc2ccc1Nc1nc(ncc1Br)Nc1cc(F)c(N3CCN(C(=O)CN4CCC(c5ccc6c(C7CCC(=O)NC7=O)nn(C)c6c5)C(F)(F)C4)CC3)c(c1)CCCCCO2)S(C)(=O)=O	C47H53BrF3N11O6S	EGFR	P00533	CRBN	WO-2024017251-A1
TPD-E67QCO	WO2024017251A1_12	.	COc1cc(N2CCN(C(=O)CN3CCC(c4ccc5c(N6CCC(=O)NC6=O)nn(C)c5c4)C(F)(F)C3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCOC2=O	C47H53BrF2N12O9S	EGFR	P00533	CRBN	WO-2024017251-A1
TPD-7C0QVJ	WO2024017251A1_13	.	COc1cc(N2CCN(C(=O)CN3CCC(c4ccc5c(C6CCC(=O)NC6=O)nn(C)c5c4)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCOC2=O	C48H56BrN11O9S	EGFR	P00533	CRBN	WO-2024017251-A1
TPD-M7SCZQ	WO2024017251A1_14	.	COc1cc(N2CCN(C(=O)CN3CCC(c4ccc(NC5CCC(=O)NC5=O)cc4)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCOC2=O	C46H55BrN10O9S	EGFR	P00533	CRBN	WO-2024017251-A1
TPD-Q48SVK	WO2024017251A1_15	.	COc1cc(N2CCC(N3CCN(CC4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCOC2=O	C52H62BrN11O10S	EGFR	P00533	CRBN	WO-2024017251-A1
TPD-CRWR2N	WO2024017251A1_16	.	COc1cc(N2CCC(N3CCN(CC4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)CC2)c2cc1Nc1ncc(Cl)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCOC2=O	C52H62ClN11O10S	EGFR	P00533	CRBN	WO-2024017251-A1
TPD-A7E4RH	WO2024017251A1_17	.	COc1cc(N2CCC(N3CCN(CC4CCN(c5cc6c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCOC2=O	C52H61BrFN11O10S	EGFR	P00533	CRBN	WO-2024017251-A1
TPD-2RFBS5	WO2024017251A1_18	.	COc1cc(N2CCC(N3CCN(CC4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C1CC1)S(C)(=O)=O)OCCCCOC2=O	C54H64BrN11O10S	EGFR	P00533	CRBN	WO-2024017251-A1
TPD-KO0ORH	WO2024017251A1_19	.	COc1cc(N2CCC(N3CCN(C(=O)[C@H](C)Nc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCOC2=O	C49H56BrN11O11S	EGFR	P00533	CRBN	WO-2024017251-A1
TPD-OB4GF2	WO2024017251A1_20	.	COc1cc(N2CCN(CC3CCN(C(=O)[C@H](C)Nc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCOC2=O	C50H58BrN11O11S	EGFR	P00533	CRBN	WO-2024017251-A1
TPD-OS9L2U	WO2024017251A1_21	.	COc1cc(N2CCC(CN3CCC4(CC3)CCN(c3ccc5c(c3)C(=O)N(C3CCC(=O)NC3=O)C5=O)CC4)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCOC2=O	C52H61BrN10O10S	EGFR	P00533	CRBN	WO-2024017251-A1
TPD-24S1WM	WO2024017251A1_22	.	COc1cc(N2CCC(CN3CCC(C4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCOC2=O	C53H63BrN10O10S	EGFR	P00533	CRBN	WO-2024017251-A1
TPD-LOF4BI	WO2024017251A1_23	.	COc1cc(N2CCC3(CC2)CN(CC2CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC2)C3)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCOC2=O	C50H57BrN10O10S	EGFR	P00533	CRBN	WO-2024017251-A1
TPD-2YWAUX	WO2024017251A1_24	.	COc1cc(N2CCN(C(=O)CC3(O)CCN(c4ccc(NC5CCC(=O)NC5=O)cc4F)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCOC2=O	C46H54BrFN10O10S	EGFR	P00533	CRBN	WO-2024017251-A1
TPD-ITT1LA	WO2024017251A1_25	.	COc1cc(N2CCC3(CCN(CC4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCOC2=O	C52H61BrN10O10S	EGFR	P00533	CRBN	WO-2024017251-A1
TPD-LR2JN9	WO2024017251A1_26	.	COc1cc(N2CCC(N3CCN(CC4CN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCOC2=O	C50H58BrN11O10S	EGFR	P00533	CRBN	WO-2024017251-A1
TPD-XZ03TH	WO2024017251A1_27	.	COc1cc(N2CCC(N3CCN(C[C@@H]4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCOC2=O	C51H60BrN11O10S	EGFR	P00533	CRBN	WO-2024017251-A1
TPD-PNVAYV	WO2024017251A1_28	.	COc1cc(N2CCC(N3CCN(C[C@H]4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCOC2=O	C51H60BrN11O10S	EGFR	P00533	CRBN	WO-2024017251-A1
TPD-D1OUUL	WO2024017251A1_29	.	COc1cc(N2CCC(CN3CCN(C4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCOC2=O	C52H62BrN11O10S	EGFR	P00533	CRBN	WO-2024017251-A1
TPD-Q0W8OR	WO2024017251A1_30	.	COc1cc(N2CCC(N3CCN(CC4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCOC2=O	C52H64BrN11O9S	EGFR	P00533	CRBN	WO-2024017251-A1
TPD-CJU0JE	WO2024017251A1_31	.	COc1cc(N2CCC(N3CCN(CC4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1P(C)(C)=O)OCCCCOC2=O	C52H62BrN10O9P	EGFR	P00533	CRBN	WO-2024017251-A1
TPD-M562JE	WO2024017251A1_32	.	COc1cc(N2CCC(N3CCN(CCc4cc(F)c(C5CCC(=O)NC5=O)c(F)c4)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCOC2=O	C46H54BrF2N9O8S	EGFR	P00533	CRBN	WO-2024017251-A1
TPD-B4LONE	WO2024017251A1_33	.	COc1cc(N2CCC(CN3CCN(c4ccc5c(C6CCC(=O)NC6=O)nn(C)c5c4)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCOC2=O	C47H56BrN11O8S	EGFR	P00533	CRBN	WO-2024017251-A1
TPD-MFAGPC	SCHEMBL27036807	(6Z)-N-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperazin-1-yl]ethyl]-6-(5-fluoro-2-oxo-1H-indol-3-ylidene)-2-methyl-4,5-dihydro-1H-cyclopenta[b]pyrrole-3-carboxamide; SCHEMBL30741775	Cc1[nH]c2c(c1C(=O)NCCN1CCN(c3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC1)CC/C2=C1/C(=O)Nc2ccc(F)cc21	C36H34FN7O6	HPK1	Q92918	CRBN	WO-2024017372-A1
TPD-0R1IVY	SCHEMBL30741721	(6Z)-N-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]ethyl]-6-(5-fluoro-2-oxo-1H-indol-3-ylidene)-2-methyl-4,5-dihydro-1H-cyclopenta[b]pyrrole-3-carboxamide	Cc1[nH]c2c(c1C(=O)NCCN1CCN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC1)CC/C2=C1/C(=O)Nc2ccc(F)cc21	C36H34FN7O6	HPK1	Q92918	CRBN	WO-2024017372-A1
TPD-BOSI2H	SCHEMBL27036846	(6Z)-N-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]ethyl]-6-(5-fluoro-2-oxo-1H-indol-3-ylidene)-2-methyl-4,5-dihydro-1H-cyclopenta[b]pyrrole-3-carboxamide	Cc1[nH]c2c(c1C(=O)NCCN1CCN(c3cc4c(cc3F)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC1)CC/C2=C1/C(=O)Nc2ccc(F)cc21	C36H33F2N7O6	HPK1	Q92918	CRBN	WO-2024017372-A1
TPD-QJQ2G0	SCHEMBL27036943	(6Z)-N-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]ethyl]-6-(5-fluoro-2-oxo-1H-indol-3-ylidene)-2-methyl-4,5-dihydro-1H-cyclopenta[b]pyrrole-3-carboxamide; SCHEMBL30741703	Cc1[nH]c2c(c1C(=O)NCCN1CCN(c3ccc4c(c3)CN(C3CCC(=O)NC3=O)C4=O)CC1)CC/C2=C1/C(=O)Nc2ccc(F)cc21	C36H36FN7O5	HPK1	Q92918	CRBN	WO-2024017372-A1
TPD-JYZDBY	SCHEMBL27036883	(6Z)-N-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperazin-1-yl]propyl]-6-(5-fluoro-2-oxo-1H-indol-3-ylidene)-2-methyl-4,5-dihydro-1H-cyclopenta[b]pyrrole-3-carboxamide; SCHEMBL30741707	Cc1[nH]c2c(c1C(=O)NCCCN1CCN(c3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC1)CC/C2=C1/C(=O)Nc2ccc(F)cc21	C37H36FN7O6	HPK1	Q92918	CRBN	WO-2024017372-A1
TPD-EMZ7K3	SCHEMBL27036809	(6Z)-N-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]propyl]-6-(5-fluoro-2-oxo-1H-indol-3-ylidene)-2-methyl-4,5-dihydro-1H-cyclopenta[b]pyrrole-3-carboxamide	Cc1[nH]c2c(c1C(=O)NCCCN1CCN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC1)CC/C2=C1/C(=O)Nc2ccc(F)cc21	C37H36FN7O6	HPK1	Q92918	CRBN	WO-2024017372-A1
TPD-RMC9KJ	SCHEMBL27036764	(6Z)-N-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]propyl]-6-(5-fluoro-2-oxo-1H-indol-3-ylidene)-2-methyl-4,5-dihydro-1H-cyclopenta[b]pyrrole-3-carboxamide	Cc1[nH]c2c(c1C(=O)NCCCN1CCN(c3cc4c(cc3F)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC1)CC/C2=C1/C(=O)Nc2ccc(F)cc21	C37H35F2N7O6	HPK1	Q92918	CRBN	WO-2024017372-A1
TPD-AHDIS0	SCHEMBL27036797	(6Z)-N-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]propyl]-6-(5-fluoro-2-oxo-1H-indol-3-ylidene)-2-methyl-4,5-dihydro-1H-cyclopenta[b]pyrrole-3-carboxamide	Cc1[nH]c2c(c1C(=O)NCCCN1CCN(c3ccc4c(c3)CN(C3CCC(=O)NC3=O)C4=O)CC1)CC/C2=C1/C(=O)Nc2ccc(F)cc21	C37H38FN7O5	HPK1	Q92918	CRBN	WO-2024017372-A1
TPD-XY6KTW	SCHEMBL27036878	2-(2,6-dioxopiperidin-3-yl)-5-[5-[(6Z)-6-(5-fluoro-2-oxo-1H-indol-3-ylidene)-2-methyl-4,5-dihydro-1H-cyclopenta[b]pyrrole-3-carbonyl]-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-2-yl]isoindole-1,3-dione; SCHEMBL30741766	Cc1[nH]c2c(c1C(=O)N1CC3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3C1)CC/C2=C1/C(=O)Nc2ccc(F)cc21	C36H31FN6O6	HPK1	Q92918	CRBN	WO-2024017372-A1
TPD-GE083W	SCHEMBL30741752	2-(2,6-dioxopiperidin-3-yl)-5-[3-[1-[(6Z)-6-(5-fluoro-2-oxo-1H-indol-3-ylidene)-2-methyl-4,5-dihydro-1H-cyclopenta[b]pyrrole-3-carbonyl]azetidin-3-yl]azetidin-1-yl]isoindole-1,3-dione	Cc1[nH]c2c(c1C(=O)N1CC(C3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)C1)CC/C2=C1/C(=O)Nc2ccc(F)cc21	C36H31FN6O6	HPK1	Q92918	CRBN	WO-2024017372-A1
TPD-9TQ628	SCHEMBL27036891	2-(2,6-dioxopiperidin-3-yl)-5-[4-[(6Z)-6-(5-fluoro-2-oxo-1H-indol-3-ylidene)-2-methyl-4,5-dihydro-1H-cyclopenta[b]pyrrole-3-carbonyl]-1-oxa-4,9-diazaspiro[5.5]undecan-9-yl]isoindole-1,3-dione; SCHEMBL30741710	Cc1[nH]c2c(c1C(=O)N1CCOC3(CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)C1)CC/C2=C1/C(=O)Nc2ccc(F)cc21	C38H35FN6O7	HPK1	Q92918	CRBN	WO-2024017372-A1
TPD-YNUR0H	SCHEMBL30741877	2-(2,6-dioxopiperidin-3-yl)-5-[3-[4-[(6Z)-6-(5-fluoro-2-oxo-1H-indol-3-ylidene)-2-methyl-4,5-dihydro-1H-cyclopenta[b]pyrrole-3-carbonyl]piperazin-1-yl]prop-1-ynyl]isoindole-1,3-dione	Cc1[nH]c2c(c1C(=O)N1CCN(CC#Cc3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC1)CC/C2=C1/C(=O)Nc2ccc(F)cc21	C37H31FN6O6	HPK1	Q92918	CRBN	WO-2024017372-A1
TPD-09PVL7	SCHEMBL30741873	2-(2,6-dioxopiperidin-3-yl)-5-[2-[1-[(6Z)-6-(5-fluoro-2-oxo-1H-indol-3-ylidene)-2-methyl-4,5-dihydro-1H-cyclopenta[b]pyrrole-3-carbonyl]piperidin-4-yl]ethynyl]isoindole-1,3-dione	Cc1[nH]c2c(c1C(=O)N1CCC(C#Cc3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC1)CC/C2=C1/C(=O)Nc2ccc(F)cc21	C37H30FN5O6	HPK1	Q92918	CRBN	WO-2024017372-A1
TPD-PMW9QT	SCHEMBL30741875	2-(2,6-dioxopiperidin-3-yl)-5-[4-[3-[[(6Z)-6-(5-fluoro-2-oxo-1H-indol-3-ylidene)-2-methyl-4,5-dihydro-1H-cyclopenta[b]pyrrol-3-yl]amino]propyl]piperazin-1-yl]isoindole-1,3-dione	Cc1[nH]c2c(c1NCCCN1CCN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC1)CC/C2=C1/C(=O)Nc2ccc(F)cc21	C36H36FN7O5	HPK1	Q92918	CRBN	WO-2024017372-A1
TPD-3LF8DV	SCHEMBL27036798	(6Z)-N-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]ethyl]-6-(5-fluoro-2-oxo-1H-indol-3-ylidene)-2-methyl-4,5-dihydro-1H-cyclopenta[b]pyrrole-3-carboxamide; SCHEMBL30741756	Cc1[nH]c2c(c1C(=O)NCCC1CCN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC1)CC/C2=C1/C(=O)Nc2ccc(F)cc21	C37H35FN6O6	HPK1	Q92918	CRBN	WO-2024017372-A1
TPD-4J3KYT	SCHEMBL27036808	2-(2,6-dioxopiperidin-3-yl)-5-[4-[(6Z)-6-(5-fluoro-2-oxo-1H-indol-3-ylidene)-2-methyl-4,5-dihydro-1H-cyclopenta[b]pyrrole-3-carbonyl]piperazin-1-yl]isoindole-1,3-dione; SCHEMBL30741746	Cc1[nH]c2c(c1C(=O)N1CCN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC1)CC/C2=C1/C(=O)Nc2ccc(F)cc21	C34H29FN6O6	HPK1	Q92918	CRBN	WO-2024017372-A1
TPD-4OAWXB	SCHEMBL30741878	2-(2,6-dioxopiperidin-3-yl)-5-[4-[1-[(6Z)-6-(5-fluoro-2-oxo-1H-indol-3-ylidene)-2-methyl-4,5-dihydro-1H-cyclopenta[b]pyrrole-3-carbonyl]azetidin-3-yl]piperazin-1-yl]isoindole-1,3-dione	Cc1[nH]c2c(c1C(=O)N1CC(N3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)C1)CC/C2=C1/C(=O)Nc2ccc(F)cc21	C37H34FN7O6	HPK1	Q92918	CRBN	WO-2024017372-A1
TPD-B7MHIS	SCHEMBL30741864	2-(2,6-dioxopiperidin-3-yl)-5-[3-[4-[(6Z)-6-(5-fluoro-2-oxo-1H-indol-3-ylidene)-2-methyl-4,5-dihydro-1H-cyclopenta[b]pyrrole-3-carbonyl]piperazin-1-yl]azetidin-1-yl]isoindole-1,3-dione	Cc1[nH]c2c(c1C(=O)N1CCN(C3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)CC1)CC/C2=C1/C(=O)Nc2ccc(F)cc21	C37H34FN7O6	HPK1	Q92918	CRBN	WO-2024017372-A1
TPD-XHF28F	SCHEMBL27036795	2-(2,6-dioxopiperidin-3-yl)-5-[7-[(6Z)-6-(5-fluoro-2-oxo-1H-indol-3-ylidene)-2-methyl-4,5-dihydro-1H-cyclopenta[b]pyrrole-3-carbonyl]-2,7-diazaspiro[3.5]nonan-2-yl]isoindole-1,3-dione; SCHEMBL30741702	Cc1[nH]c2c(c1C(=O)N1CCC3(CC1)CN(c1ccc4c(c1)C(=O)N(C1CCC(=O)NC1=O)C4=O)C3)CC/C2=C1/C(=O)Nc2ccc(F)cc21	C37H33FN6O6	HPK1	Q92918	CRBN	WO-2024017372-A1
TPD-SWDH16	SCHEMBL27036791	2-(2,6-dioxopiperidin-3-yl)-5-[3-[(6Z)-6-(5-fluoro-2-oxo-1H-indol-3-ylidene)-2-methyl-4,5-dihydro-1H-cyclopenta[b]pyrrole-3-carbonyl]-3,9-diazaspiro[5.5]undecan-9-yl]isoindole-1,3-dione; SCHEMBL30741732	Cc1[nH]c2c(c1C(=O)N1CCC3(CC1)CCN(c1ccc4c(c1)C(=O)N(C1CCC(=O)NC1=O)C4=O)CC3)CC/C2=C1/C(=O)Nc2ccc(F)cc21	C39H37FN6O6	HPK1	Q92918	CRBN	WO-2024017372-A1
TPD-FMWOME	SCHEMBL27036950	2-(2,6-dioxopiperidin-3-yl)-5-[9-[(6Z)-6-(5-fluoro-2-oxo-1H-indol-3-ylidene)-2-methyl-4,5-dihydro-1H-cyclopenta[b]pyrrole-3-carbonyl]-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl]isoindole-1,3-dione; SCHEMBL30741739	Cc1[nH]c2c(c1C(=O)N1CCC3(CC1)CN(c1ccc4c(c1)C(=O)N(C1CCC(=O)NC1=O)C4=O)CCO3)CC/C2=C1/C(=O)Nc2ccc(F)cc21	C38H35FN6O7	HPK1	Q92918	CRBN	WO-2024017372-A1
TPD-5NGJVB	SCHEMBL27036847	2-(2,6-dioxopiperidin-3-yl)-5-[8-[(6Z)-6-(5-fluoro-2-oxo-1H-indol-3-ylidene)-2-methyl-4,5-dihydro-1H-cyclopenta[b]pyrrole-3-carbonyl]-2,8-diazaspiro[4.5]decan-2-yl]isoindole-1,3-dione; SCHEMBL30741706	Cc1[nH]c2c(c1C(=O)N1CCC3(CC1)CCN(c1ccc4c(c1)C(=O)N(C1CCC(=O)NC1=O)C4=O)C3)CC/C2=C1/C(=O)Nc2ccc(F)cc21	C38H35FN6O6	HPK1	Q92918	CRBN	WO-2024017372-A1
TPD-TAEP9K	SCHEMBL30741871	2-(2,6-dioxopiperidin-3-yl)-5-[4-[1-[(6Z)-6-(5-fluoro-2-oxo-1H-indol-3-ylidene)-2-methyl-4,5-dihydro-1H-cyclopenta[b]pyrrole-3-carbonyl]azetidin-3-yl]piperidin-1-yl]isoindole-1,3-dione	Cc1[nH]c2c(c1C(=O)N1CC(C3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)C1)CC/C2=C1/C(=O)Nc2ccc(F)cc21	C38H35FN6O6	HPK1	Q92918	CRBN	WO-2024017372-A1
TPD-RKNXP0	SCHEMBL30741870	2-(2,6-dioxopiperidin-3-yl)-5-[3-[1-[(6Z)-6-(5-fluoro-2-oxo-1H-indol-3-ylidene)-2-methyl-4,5-dihydro-1H-cyclopenta[b]pyrrole-3-carbonyl]azetidin-3-yl]prop-1-ynyl]isoindole-1,3-dione	Cc1[nH]c2c(c1C(=O)N1CC(CC#Cc3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C1)CC/C2=C1/C(=O)Nc2ccc(F)cc21	C36H28FN5O6	HPK1	Q92918	CRBN	WO-2024017372-A1
TPD-CLTMMJ	SCHEMBL30741867	3-[6-[3-[1-[(6Z)-6-(5-fluoro-2-oxo-1H-indol-3-ylidene)-2-methyl-4,5-dihydro-1H-cyclopenta[b]pyrrole-3-carbonyl]azetidin-3-yl]prop-1-ynyl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	Cc1[nH]c2c(c1C(=O)N1CC(CC#Cc3ccc4c(c3)CN(C3CCC(=O)NC3=O)C4=O)C1)CC/C2=C1/C(=O)Nc2ccc(F)cc21	C36H30FN5O5	HPK1	Q92918	CRBN	WO-2024017372-A1
TPD-82LPGC	SCHEMBL27036864	(6Z)-N-[(2R)-1-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]propan-2-yl]-6-(5-fluoro-2-oxo-1H-indol-3-ylidene)-2-methyl-4,5-dihydro-1H-cyclopenta[b]pyrrole-3-carboxamide; SCHEMBL30741729	Cc1[nH]c2c(c1C(=O)N[C@H](C)CN1CCN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC1)CC/C2=C1/C(=O)Nc2ccc(F)cc21	C37H36FN7O6	HPK1	Q92918	CRBN	WO-2024017372-A1
TPD-OP27EL	SCHEMBL27036701	(6Z)-N-[(2S)-1-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]propan-2-yl]-6-(5-fluoro-2-oxo-1H-indol-3-ylidene)-2-methyl-4,5-dihydro-1H-cyclopenta[b]pyrrole-3-carboxamide; SCHEMBL30741718	Cc1[nH]c2c(c1C(=O)N[C@@H](C)CN1CCN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC1)CC/C2=C1/C(=O)Nc2ccc(F)cc21	C37H36FN7O6	HPK1	Q92918	CRBN	WO-2024017372-A1
TPD-URDSIY	SCHEMBL30741866	2-(2,6-dioxopiperidin-3-yl)-5-[4-[[1-[(6Z)-6-(5-fluoro-2-oxo-1H-indol-3-ylidene)-2-methyl-4,5-dihydro-1H-cyclopenta[b]pyrrole-3-carbonyl]piperidin-4-yl]methyl]piperazin-1-yl]isoindole-1,3-dione	Cc1[nH]c2c(c1C(=O)N1CCC(CN3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC1)CC/C2=C1/C(=O)Nc2ccc(F)cc21	C40H40FN7O6	HPK1	Q92918	CRBN	WO-2024017372-A1
TPD-ZRRL94	SCHEMBL30741874	2-(2,6-dioxopiperidin-3-yl)-5-[4-[[1-[(6Z)-6-(5-fluoro-2-oxo-1H-indol-3-ylidene)-2-methyl-4,5-dihydro-1H-cyclopenta[b]pyrrole-3-carbonyl]piperidin-4-yl]methyl]piperidin-1-yl]isoindole-1,3-dione	Cc1[nH]c2c(c1C(=O)N1CCC(CC3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC1)CC/C2=C1/C(=O)Nc2ccc(F)cc21	C41H41FN6O6	HPK1	Q92918	CRBN	WO-2024017372-A1
TPD-2PFLMK	SCHEMBL27036858	(6Z)-N-[3-[4-[4-(2,6-dioxopiperidin-3-yl)oxyphenyl]piperazin-1-yl]propyl]-6-(5-fluoro-2-oxo-1H-indol-3-ylidene)-2-methyl-4,5-dihydro-1H-cyclopenta[b]pyrrole-3-carboxamide	Cc1[nH]c2c(c1C(=O)NCCCN1CCN(c3ccc(OC4CCC(=O)NC4=O)cc3)CC1)CC/C2=C1/C(=O)Nc2ccc(F)cc21	C35H37FN6O5	HPK1	Q92918	CRBN	WO-2024017372-A1
TPD-O1CJUO	SCHEMBL27036868	(6Z)-N-[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]propyl]-6-(5-fluoro-2-oxo-1H-indol-3-ylidene)-2-methyl-4,5-dihydro-1H-cyclopenta[b]pyrrole-3-carboxamide; SCHEMBL30741725	Cc1[nH]c2c(c1C(=O)NCCCN1Cc3cc4c(cc3C1)C(=O)N(C1CCC(=O)NC1=O)C4=O)CC/C2=C1/C(=O)Nc2ccc(F)cc21	C35H31FN6O6	HPK1	Q92918	CRBN	WO-2024017372-A1
TPD-LQ2HR2	SCHEMBL27036983	(6Z)-N-[3-[4-[4-[(2,6-dioxopiperidin-3-yl)amino]-2-fluorophenyl]piperazin-1-yl]propyl]-6-(5-fluoro-2-oxo-1H-indol-3-ylidene)-2-methyl-4,5-dihydro-1H-cyclopenta[b]pyrrole-3-carboxamide	Cc1[nH]c2c(c1C(=O)NCCCN1CCN(c3ccc(NC4CCC(=O)NC4=O)cc3F)CC1)CC/C2=C1/C(=O)Nc2ccc(F)cc21	C35H37F2N7O4	HPK1	Q92918	CRBN	WO-2024017372-A1
TPD-RO8DWE	SCHEMBL27036900	(6Z)-N-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]butan-2-yl]-6-(5-fluoro-2-oxo-1H-indol-3-ylidene)-2-methyl-4,5-dihydro-1H-cyclopenta[b]pyrrole-3-carboxamide; SCHEMBL30741771	Cc1[nH]c2c(c1C(=O)NC(C)CCN1CCN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC1)CC/C2=C1/C(=O)Nc2ccc(F)cc21	C38H38FN7O6	HPK1	Q92918	CRBN	WO-2024017372-A1
TPD-JLINV1	SCHEMBL27036815	(6Z)-N-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]-2-methylpropyl]-6-(5-fluoro-2-oxo-1H-indol-3-ylidene)-2-methyl-4,5-dihydro-1H-cyclopenta[b]pyrrole-3-carboxamide; SCHEMBL30741719	Cc1[nH]c2c(c1C(=O)NCC(C)CN1CCN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC1)CC/C2=C1/C(=O)Nc2ccc(F)cc21	C38H38FN7O6	HPK1	Q92918	CRBN	WO-2024017372-A1
TPD-8V873U	SCHEMBL27036835	(6Z)-N-[[1-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]cyclopropyl]methyl]-6-(5-fluoro-2-oxo-1H-indol-3-ylidene)-2-methyl-4,5-dihydro-1H-cyclopenta[b]pyrrole-3-carboxamide; SCHEMBL30741755	Cc1[nH]c2c(c1C(=O)NCC1(CN3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC1)CC/C2=C1/C(=O)Nc2ccc(F)cc21	C39H38FN7O6	HPK1	Q92918	CRBN	WO-2024017372-A1
TPD-CRCKBX	WO2024017372A1_39	.	Cc1[nH]c2c(c1C(=O)NCCCN1CCN(c3ccc(OC4CCC(=O)NC4=O)cn3)CC1)CC/C2=C1/C(=O)Nc2ccc(F)cc21	C34H36FN7O5	HPK1	Q92918	CRBN	WO-2024017372-A1
TPD-LB4JCU	WO2024017372A1_40	.	O=C1CCC(N2C(=O)c3ccc(N4CCN(CCCNC(=O)c5c[nH]c6c5CC/C6=C5/C(=O)Nc6ccc(F)cc65)CC4)cc3C2=O)C(=O)N1	C36H34FN7O6	HPK1	Q92918	CRBN	WO-2024017372-A1
TPD-299HH1	SCHEMBL27036754	(6Z)-N-[3-[4-[5-(2,6-dioxopiperidin-3-yl)oxypyrimidin-2-yl]piperazin-1-yl]propyl]-6-(5-fluoro-2-oxo-1H-indol-3-ylidene)-2-methyl-4,5-dihydro-1H-cyclopenta[b]pyrrole-3-carboxamide	Cc1[nH]c2c(c1C(=O)NCCCN1CCN(c3ncc(OC4CCC(=O)NC4=O)cn3)CC1)CC/C2=C1/C(=O)Nc2ccc(F)cc21	C33H35FN8O5	HPK1	Q92918	CRBN	WO-2024017372-A1
TPD-7EBUF7	SCHEMBL27036870	(6Z)-N-[3-[4-[4-(2,6-dioxopiperidin-3-yl)oxy-2-fluorophenyl]piperazin-1-yl]propyl]-6-(5-fluoro-2-oxo-1H-indol-3-ylidene)-2-methyl-4,5-dihydro-1H-cyclopenta[b]pyrrole-3-carboxamide	Cc1[nH]c2c(c1C(=O)NCCCN1CCN(c3ccc(OC4CCC(=O)NC4=O)cc3F)CC1)CC/C2=C1/C(=O)Nc2ccc(F)cc21	C35H36F2N6O5	HPK1	Q92918	CRBN	WO-2024017372-A1
TPD-54P1MD	WO2024017372A1_45	.	Cc1[nH]c2c(c1C(=O)NCCCN1CCN(c3ccc(NC4CCC(=O)NC4=O)nc3)CC1)CC/C2=C1/C(=O)Nc2ccc(F)cc21	C34H37FN8O4	HPK1	Q92918	CRBN	WO-2024017372-A1
TPD-PFYZBM	WO2024017392A1_50'	.	CCc1cccc2cc(O)cc(-c3c(F)cc4c(N5CC6CCC(C5)N6)nc(OC[C@@H]5CCCN5CCCOCCC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)c5ccc(-c6scnc6C)cc5)C(C)(C)C)nc4c3F)c12	C60H73F2N9O7S	KRAS	P01116	VHL	WO-2024017392-A1
TPD-564HZT	WO2024017392A1_51	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCOCC[C@@H]2CN3C[C@H](F)C[C@]3(COc3nc(N4CC5CCC(C4)N5)c4cnc(-c5cc(O)cc6cccc(C7CC7)c56)c(F)c4n3)C2)C(C)(C)C)cc1	C62H74F2N10O7S	KRAS	P01116	VHL	WO-2024017392-A1
TPD-CF2D88	WO2024017392A1_52'	.	CCc1c(F)ccc2cc(O)cc(-c3c(F)cc4c(N5CC6CCC(C5)N6)nc(OC[C@]56C[C@@H](F)CN5C[C@@H](COCC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)c5ccc(-c7scnc7C)cc5)C(C)(C)C)C6)nc4c3F)c12	C60H69F4N9O7S	KRAS	P01116	VHL	WO-2024017392-A1
TPD-S00CJZ	WO2024017392A1_53'	.	CCc1c(F)ccc2cc(O)cc(-c3c(F)cc4c(N5CC6CCC(C5)N6)nc(OC[C@]56C[C@@H](F)CN5C[C@@H](CCN5CCC[C@@H](C(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8scnc8C)cc7)C(C)(C)C)C5)C6)nc4c3F)c12	C65H78F4N10O6S	KRAS	P01116	VHL	WO-2024017392-A1
TPD-5XVAPG	WO2024017392A1_54'	.	CCc1c(F)ccc2cc(O)cc(-c3c(F)cc4c(N5CC6CCC(C5)N6)nc(OC[C@]56C[C@@H](F)CN5C[C@@H](CCN5CCC[C@H](C(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8scnc8C)cc7)C(C)(C)C)C5)C6)nc4c3F)c12	C65H78F4N10O6S	KRAS	P01116	VHL	WO-2024017392-A1
TPD-C5NLRT	WO2024017392A1_55'	.	CCc1c(F)ccc2cc(O)cc(-c3c(F)cc4c(N5CC6CCC(C5)N6)nc(OC[C@]56C[C@@H](F)CN5C[C@@H](CN5CCN(c7ccc(NC8CCC(=O)NC8=O)cc7F)CC5)C6)nc4c3F)c12	C50H54F5N9O4	KRAS	P01116	CRBN	WO-2024017392-A1
TPD-JP5KJI	WO2024017392A1_56''	.	CCc1c(F)ccc2cc(O)cc(-c3c(F)cc4c(N5CC6CCC(C5)N6)nc(OC[C@]56C[C@@H](F)CN5C[C@@H](CN5CCC(CN7CCN(c8ccc9c(c8)CN([C@H]8CCC(=O)NC8=O)C9=O)CC7)CC5)C6)nc4c3F)c12	C58H66F4N10O5	KRAS	P01116	CRBN	WO-2024017392-A1
TPD-6BHB2P	WO2024017392A1_56'	.	CCc1c(F)ccc2cc(O)cc(-c3c(F)cc4c(N5CC6CCC(C5)N6)nc(OC[C@]56C[C@@H](F)CN5C[C@@H](CN5CCC(CN7CCN(c8ccc9c(c8)CN([C@@H]8CCC(=O)NC8=O)C9=O)CC7)CC5)C6)nc4c3F)c12	C58H66F4N10O5	KRAS	P01116	CRBN	WO-2024017392-A1
TPD-Q1TIIG	WO2024017392A1_56a'	.	CCc1c(F)ccc2cc(O)cc(-c3c(F)cc4c(N5CC6CCC(C5)N6)nc(OC[C@]56C[C@@H](F)CN5C[C@@H](CN5CCC(CN7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC5)C6)nc4c3F)c12	C58H66F4N10O5	KRAS	P01116	CRBN	WO-2024017392-A1
TPD-CTFY3T	WO2024017392A1_57'	.	CCc1c(F)ccc2cc(O)cc(-c3c(F)cc4c(N5CC6CCC(C5)N6)nc(OC[C@@]56CC(COCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8scnc8C)cc7)C(C)(C)C)CN5C[C@H](F)C6)nc4c3F)c12	C61H71F4N9O7S	KRAS	P01116	VHL	WO-2024017392-A1
TPD-J4A4R9	WO2024017392A1_58'	.	CCc1cccc2cc(O)cc(-c3c(F)cc4c(N5CC6CCC(C5)N6)nc(OC[C@@]56CC[C@H](CCOCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8scnc8C)cc7)C(C)(C)C)N5C[C@H](F)C6)nc4c3F)c12	C62H74F3N9O7S	KRAS	P01116	VHL	WO-2024017392-A1
TPD-AZIOF6	WO2024017392A1_59''	.	CCc1c(F)ccc2cc(O)cc(-c3c(F)cc4c(N5CC6CCC(C5)N6)nc(OC[C@@]56CC(OCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8scnc8C)cc7)C(C)(C)C)CN5C[C@H](F)C6)nc4c3F)c12	C59H67F4N9O7S	KRAS	P01116	VHL	WO-2024017392-A1
TPD-VIJC8T	WO2024017392A1_59'	.	CCc1cccc2cc(O)cc(-c3c(F)cc4c(N5CC6CCC(C5)N6)nc(OC[C@]56C[C@@H](F)CN5C[C@@H](OCC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)c5ccc(-c7scnc7C)cc5)C(C)(C)C)C6)nc4c3F)c12	C59H68F3N9O7S	KRAS	P01116	VHL	WO-2024017392-A1
TPD-8WJVTJ	WO2024017392A1_59	.	CCc1c(F)ccc2cc(O)cc(-c3c(F)cc4c(N5CC6CCC(C5)N6)nc(OC[C@]56C[C@@H](F)CN5C[C@@H](OCC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)c5ccc(-c7scnc7C)cc5)C(C)(C)C)C6)nc4c3F)c12	C59H67F4N9O7S	KRAS	P01116	VHL	WO-2024017392-A1
TPD-WBUEKO	WO2024017392A1_60'	.	CCc1cccc2cc(O)cc(-c3c(F)c4c5c(nc(OC[C@]67C[C@@H](F)CN6C[C@@H](CN6CCC(CN8CCN(c9ccc%10c(c9)CN(C9CCC(=O)NC9=O)C%10=O)CC8)CC6)C7)nc5c3F)N3CC5CCC(N5)C3CO4)c12	C59H67F3N10O6	KRAS	P01116	CRBN	WO-2024017392-A1
TPD-KBVUYL	WO2024017392A1_61'	.	CCc1cccc2cc(O)cc(-c3c(F)c4c5c(nc(OC[C@]67C[C@@H](F)CN6C[C@@H](CN6CCC(CN8CCN(c9ccc%10c(c9)CN(C9CCC(=O)NC9=O)C%10=O)CC8)CC6)C7)nc5c3F)N3CC5CCC(N5)C3CCO4)c12	C60H69F3N10O6	KRAS	P01116	CRBN	WO-2024017392-A1
TPD-WTEDA8	WO2024017392A1_62''	.	Cc1cc(N)cc(-c2c(F)c3c4c(nc(OC[C@]56C[C@@H](F)CN5C[C@@H](CN5CCC(CN7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC5)C6)nc4c2F)N2CC4CCC(N4)C2CO3)c1C(F)(F)F	C55H63F6N11O5	KRAS	P01116	CRBN	WO-2024017392-A1
TPD-MOIO0S	WO2024017392A1_63'	.	CCc1c(F)ccc2cc(O)cc(-c3c(F)cc4c(N5CC6CCC(C5)N6)nc(OC[C@]56C[C@@H](F)CN5C[C@@H](CCN5CCC(CN7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC5)C6)nc4c3F)c12	C59H68F4N10O5	KRAS	P01116	CRBN	WO-2024017392-A1
TPD-SS16H9	WO2024017392A1_64'	.	CCc1c(F)ccc2cc(O)cc(-c3c(F)cc4c(N5CC6CCC(C5)N6)nc(OC[C@@H]5CCCN5CCCN5CCC[C@H](C(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)c6ccc(-c7scnc7C)cc6)C(C)(C)C)C5)nc4c3F)c12	C63H77F3N10O6S	KRAS	P01116	VHL	WO-2024017392-A1
TPD-37SF74	WO2024017392A1_65'	.	Cc1cc(N)cc(-c2c(F)c3c4c(nc(OC[C@]56C[C@@H](F)CN5C[C@@H](CN5CCN(c7ccc(NC8CCC(=O)NC8=O)cc7F)CC5)C6)nc4c2F)N2CC4CCC(N4)C2CO3)c1C(F)(F)F	C47H51F7N10O4	KRAS	P01116	CRBN	WO-2024017392-A1
TPD-KGL628	WO2024017392A1_65a	.	Cc1cc(N)nc(-c2c(F)c3c4c(nc(OC[C@]56C[C@@H](F)CN5C[C@@H](CN5CCN(c7ccc(NC8CCC(=O)NC8=O)cc7F)CC5)C6)nc4c2F)N2CC4CCC(N4)C2CO3)c1C(F)(F)F	C46H50F7N11O4	KRAS	P01116	CRBN	WO-2024017392-A1
TPD-0ZNJE4	WO2024017392A1_66'	.	CCNC(=O)c1nnc(-c2cc(C(C)C)c(O)cc2O)n1-c1ccc(CN2CCN(CC3CCN(C[C@@H]4CN5C[C@H](F)C[C@]5(COc5nc(N6CC7CCC(C6)N7)c6cc(F)c(-c7cc(O)cc8ccc(F)c(CC)c78)c(F)c6n5)C4)CC3)CC2)cc1	C66H78F4N12O5	KRAS	P01116	VHL	WO-2024017392-A1
TPD-Y42VU5	WO2024017392A1_67	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC[C@]56C[C@@H](F)CN5C[C@@H](CN5CCC(CN7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC5)C6)nc4c3F)c12	C57H62F3N11O5	KRAS	P01116	CRBN	WO-2024017392-A1
TPD-E73MX4	WO2024017392A1_68'	.	CCc1c(F)ccc2cc(O)cc(-c3c(F)cc4c(N5CC6CCC(C5)N6)nc(OC[C@]56C[C@@H](F)CN5C[C@@H](CCN5CCC(CN7CCN(c8cc9c(cc8F)C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)CC5)C6)nc4c3F)c12	C59H65F5N10O6	KRAS	P01116	CRBN	WO-2024017392-A1
TPD-WLIJJ7	WO2024017392A1_69'	.	CCc1c(F)ccc2cc(O)cc(-c3c(F)cc4c(N5CC6CCC(C5)N6)nc(OC[C@]56C[C@@H](F)CN5C[C@@H](CCN5CCC(CN7CCN(c8ccc(C9CCC(=O)NC9=O)cc8)CC7)CC5)C6)nc4c3F)c12	C57H67F4N9O4	KRAS	P01116	CRBN	WO-2024017392-A1
TPD-WEXC4G	WO2024017392A1_70'	.	CCc1c(F)ccc2cc(O)cc(-c3c(F)cc4c(N5CC6CCC(C5)N6)nc(OC[C@]56C[C@@H](F)CN5C[C@@H](CN5CCC(CN7CCN(c8ccc(C9CCC(=O)NC9=O)cc8)CC7)CC5)C6)nc4c3F)c12	C56H65F4N9O4	KRAS	P01116	CRBN	WO-2024017392-A1
TPD-AOEKT5	WO2024017392A1_71'	.	CCc1c(F)ccc2cc(O)cc(-c3c(F)cc4c(N5CC6CCC(C5)N6)nc(OC[C@]56C[C@@H](F)CN5C[C@@H](CN5CCC(CN7CCN(c8cc9c(cc8F)C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)CC5)C6)nc4c3F)c12	C58H63F5N10O6	KRAS	P01116	CRBN	WO-2024017392-A1
TPD-KXXBUC	WO2024017392A1_72'	.	CCc1c(F)ccc2cc(O)cc(-c3c(F)cc4c(N5CC6CCC(C5)N6)nc(OC[C@]56C[C@@H](F)CN5C[C@@H](CCN5CCC(CN7CCN(c8ccc(C(=O)N[C@H]9CCC(=O)NC9=O)c(F)c8)CC7)CC5)C6)nc4c3F)c12	C58H67F5N10O5	KRAS	P01116	CRBN	WO-2024017392-A1
TPD-7D14HI	WO2024017392A1_73'	.	CCc1c(F)ccc2cc(O)cc(-c3c(F)cc4c(N5CC6CCC(C5)N6)nc(OC[C@]56C[C@@H](F)CN5C[C@@H](CN5CCC(CN7CCN(c8ccc(C(=O)N[C@H]9CCC(=O)NC9=O)c(F)c8)CC7)CC5)C6)nc4c3F)c12	C57H65F5N10O5	KRAS	P01116	CRBN	WO-2024017392-A1
TPD-23LHQQ	WO2024017392A1_74	.	CCc1c(F)ccc2cc(O)cc(-c3c(F)cc4c(N5CC6CCC(C5)N6)nc(OC[C@]56C[C@@H](F)CN5C[C@@H](CCN5CCC(CN7CCN(c8ccc(N9CCC(=O)NC9=O)cc8)CC7)CC5)C6)nc4c3F)c12	C56H66F4N10O4	KRAS	P01116	CRBN	WO-2024017392-A1
TPD-42GJXZ	SCHEMBL27064448	6-[3-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperidin-1-yl]propanoylamino]-4-[2-methoxy-3-(1-methyl-1,2,4-triazol-3-yl)anilino]-N-methylpyridazine-3-carboxamide; SCHEMBL30683381	CNC(=O)c1nnc(NC(=O)CCN2CCC(C3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)CC2)cc1Nc1cccc(-c2ncn(C)n2)c1OC	C40H44N12O7	TYK2	P29597	CRBN	WO-2024020221-A1
TPD-ZJ6XYJ	SCHEMBL30683395	6-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]propanoylamino]-4-[2-methoxy-3-(1-methyl-1,2,4-triazol-3-yl)anilino]-N-methylpyridazine-3-carboxamide	CNC(=O)c1nnc(NC(=O)CCN2CCN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)cc1Nc1cccc(-c2ncn(C)n2)c1OC	C36H38N12O7	TYK2	P29597	CRBN	WO-2024020221-A1
TPD-9LDMCN	SCHEMBL30683400	6-[3-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]methyl]piperidin-1-yl]propanoylamino]-4-[2-methoxy-3-(1-methyl-1,2,4-triazol-3-yl)anilino]-N-methylpyridazine-3-carboxamide	CNC(=O)c1nnc(NC(=O)CCN2CCC(CC3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)CC2)cc1Nc1cccc(-c2ncn(C)n2)c1OC	C41H46N12O7	TYK2	P29597	CRBN	WO-2024020221-A1
TPD-O0FFGD	SCHEMBL27064485	6-[3-[4-[6-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]pyrimidin-4-yl]piperazin-1-yl]propanoylamino]-4-[2-methoxy-3-(1-methyl-1,2,4-triazol-3-yl)anilino]-N-methylpyridazine-3-carboxamide; SCHEMBL30683402	CNC(=O)c1nnc(NC(=O)CCN2CCN(c3cc(N4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)ncn3)CC2)cc1Nc1cccc(-c2ncn(C)n2)c1OC	C44H48N16O7	TYK2	P29597	CRBN	WO-2024020221-A1
TPD-7EIGT6	SCHEMBL27064500	6-[3-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methoxymethyl]piperidin-1-yl]propanoylamino]-4-[2-methoxy-3-(1-methyl-1,2,4-triazol-3-yl)anilino]-N-methylpyridazine-3-carboxamide; SCHEMBL30683389; SCHEMBL30683390	CNC(=O)c1nnc(NC(=O)CCN2CCC(COCC3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)cc1Nc1cccc(-c2ncn(C)n2)c1OC	C44H52N12O8	TYK2	P29597	CRBN	WO-2024020221-A1
TPD-56GSMA	SCHEMBL27064530	6-[3-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methylamino]propanoylamino]-4-[2-methoxy-3-(1-methyl-1,2,4-triazol-3-yl)anilino]-N-methylpyridazine-3-carboxamide; SCHEMBL30683396	CNC(=O)c1nnc(NC(=O)CCNCC2CCN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)cc1Nc1cccc(-c2ncn(C)n2)c1OC	C38H42N12O7	TYK2	P29597	CRBN	WO-2024020221-A1
TPD-N8GVTR	SCHEMBL30683387	6-[3-[3-[[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperazin-1-yl]methyl]azetidin-1-yl]propanoylamino]-4-[2-methoxy-3-(1-methyl-1,2,4-triazol-3-yl)anilino]-N-methylpyridazine-3-carboxamide	CNC(=O)c1nnc(NC(=O)CCN2CC(CN3CCN(C4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)C2)cc1Nc1cccc(-c2ncn(C)n2)c1OC	C45H54N14O7	TYK2	P29597	CRBN	WO-2024020221-A1
TPD-0K6JBU	SCHEMBL27064553	6-[3-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]propyl]piperidin-1-yl]propanoylamino]-4-[2-methoxy-3-(1-methyl-1,2,4-triazol-3-yl)anilino]-N-methylpyridazine-3-carboxamide; SCHEMBL30683385	CNC(=O)c1nnc(NC(=O)CCN2CCC(CCCN3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)cc1Nc1cccc(-c2ncn(C)n2)c1OC	C44H53N13O7	TYK2	P29597	CRBN	WO-2024020221-A1
TPD-R9YNZF	SCHEMBL30683397	6-[3-[4-[2-[1-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxyphenyl]piperidin-4-yl]ethyl]piperidin-1-yl]propanoylamino]-4-[2-methoxy-3-(1-methyl-1,2,4-triazol-3-yl)anilino]-N-methylpyridazine-3-carboxamide	CNC(=O)c1nnc(NC(=O)CCN2CCC(CCC3CCN(c4ccc(Oc5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)cc4)CC3)CC2)cc1Nc1cccc(-c2ncn(C)n2)c1OC	C50H56N12O8	TYK2	P29597	CRBN	WO-2024020221-A1
TPD-N5IGS5	SCHEMBL27064579	6-[3-[4-[[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]amino]methyl]piperidin-1-yl]propanoylamino]-4-[2-methoxy-3-(1-methyl-1,2,4-triazol-3-yl)anilino]-N-methylpyridazine-3-carboxamide; SCHEMBL30683394	CNC(=O)c1nnc(NC(=O)CCN2CCC(CNc3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)cc1Nc1cccc(-c2ncn(C)n2)c1OC	C38H42N12O7	TYK2	P29597	CRBN	WO-2024020221-A1
TPD-KZH7UI	SCHEMBL27439044	4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]-N-[4-[4-[3-[3-[[3-(4-hydroxycyclohexyl)-4-imino-5,6-diphenylpyrrolo[2,3-d]pyrimidin-7-yl]methyl]phenyl]prop-2-ynyl]piperazin-1-yl]-4-oxobutyl]butanamide	N=c1c2c(-c3ccccc3)c(-c3ccccc3)n(Cc3cccc(C#CCN4CCN(C(=O)CCCNC(=O)CCCNc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)c3)c2ncn1[C@H]1CC[C@H](O)CC1	C59H62N10O7	eEF1A2	Q05639	CRBN	WO-2024026064-A1
TPD-HR1FSL	SCHEMBL27439046	3-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]-N-[4-[4-[3-[3-[[3-(4-hydroxycyclohexyl)-4-imino-5,6-diphenylpyrrolo[2,3-d]pyrimidin-7-yl]methyl]phenyl]prop-2-ynyl]piperazin-1-yl]-4-oxobutyl]propanamide	N=c1c2c(-c3ccccc3)c(-c3ccccc3)n(Cc3cccc(C#CCN4CCN(C(=O)CCCNC(=O)CCOCCOCCOCCNc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)c3)c2ncn1[C@H]1CC[C@H](O)CC1	C64H72N10O10	eEF1A2	Q05639	CRBN	WO-2024026064-A1
TPD-T39YI9	WO2024026064A1_3	.	N=c1c2c(-c3ccccc3)c(-c3ccccc3)n(Cc3cccc(C#CCCC(=O)NCCCNC(=O)CCCNc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)c3)c2ncn1[C@H]1CC[C@H](O)CC1	C56H57N9O7	eEF1A2	Q05639	CRBN	WO-2024026064-A1
TPD-R9ZXZM	WO2024026064A1_4	.	N=c1c2c(-c3ccccc3)c(-c3ccccc3)n(Cc3cccc(C#CCCC(=O)NCCCNC(=O)CCCCCNc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)c3)c2ncn1[C@H]1CC[C@H](O)CC1	C58H61N9O7	eEF1A2	Q05639	CRBN	WO-2024026064-A1
TPD-3LNULQ	WO2024026064A1_5	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCC(=O)NCCCNC(=O)CCC#Cc2cccc(Cn3c(-c4ccccc4)c(-c4ccccc4)c4c(=N)n([C@H]5CC[C@H](O)CC5)cnc43)c2)C(C)(C)C)cc1	C69H82N10O7S	eEF1A2	Q05639	VHL	WO-2024026064-A1
TPD-01FXO9	SCHEMBL29960929	6-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]-N-[6-[3-[[3-(4-hydroxycyclohexyl)-4-imino-5,6-diphenylpyrrolo[2,3-d]pyrimidin-7-yl]methyl]phenyl]hex-5-ynyl]hexanamide	N=c1c2c(-c3ccccc3)c(-c3ccccc3)n(Cc3cccc(C#CCCCCNC(=O)CCCCCNc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)c3)c2ncn1[C@H]1CC[C@H](O)CC1	C56H58N8O6	eEF1A2	Q05639	CRBN	WO-2024026064-A1
TPD-91Q6RU	WO2024026064A1_7	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](C)NC(=O)CCCC(=O)NCCCCC#Cc2cccc(Cn3c(-c4ccccc4)c(-c4ccccc4)c4c(=N)n([C@H]5CC[C@H](O)CC5)cnc43)c2)cc1	C61H67N9O6S	eEF1A2	Q05639	VHL	WO-2024026064-A1
TPD-JZ1CDY	WO2024026064A1_8	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](C)NC(=O)CCC(=O)NCCCCC#Cc2cccc(Cn3c(-c4ccccc4)c(-c4ccccc4)c4c(=N)n([C@H]5CC[C@@H](On6nnc7ccccc76)CC5)cnc43)c2)cc1	C66H68N12O6S	eEF1A2	Q05639	VHL	WO-2024026064-A1
TPD-JIK2FU	WO2024026064A1_9	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](C)NC(=O)CCC(=O)NCCCCC#Cc2cccc(Cn3c(-c4ccccc4)c(-c4ccccc4)c4c(=N)n([C@H]5CC[C@H](O)CC5)cnc43)c2)cc1	C60H65N9O6S	eEF1A2	Q05639	VHL	WO-2024026064-A1
TPD-C9QUGQ	SCHEMBL29960946	3-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]-N-[6-[3-[[3-(4-hydroxycyclohexyl)-4-imino-5,6-diphenylpyrrolo[2,3-d]pyrimidin-7-yl]methyl]phenyl]hex-5-ynyl]propanamide	N=c1c2c(-c3ccccc3)c(-c3ccccc3)n(Cc3cccc(C#CCCCCNC(=O)CCOCCOCCOCCNc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)c3)c2ncn1[C@H]1CC[C@H](O)CC1	C59H64N8O9	eEF1A2	Q05639	CRBN	WO-2024026064-A1
TPD-H8PQFN	WO2024026064A1_11	.	Cc1ncsc1-c1ccc(CNC(=O)C2C[C@@H](O)CN2C(=O)[C@H](C)NC(=O)CCCC(=O)NCCCCC#Cc2cccc(Cn3c(-c4ccccc4)c(-c4ccccc4)c4c(N[C@H]5CC[C@H](O)CC5)ncnc43)c2)cc1	C61H67N9O6S	eEF1A2	Q05639	VHL	WO-2024026064-A1
TPD-JCVSQG	WO2024026064A1_12	.	Cc1ncsc1-c1ccc(CNC(=O)C2C[C@H](O)CN2C(=O)[C@H](C)NC(=O)CCCC(=O)NCCCCC#Cc2cccc(Cn3c(-c4ccccc4)c(-c4ccccc4)c4c(=N)n([C@H]5CC[C@H](O)CC5)cnc43)c2)cc1	C61H67N9O6S	eEF1A2	Q05639	VHL	WO-2024026064-A1
TPD-3FWHCA	WO2024026064A1_13	.	CN[C@@H](C)C(=O)N[C@H](C(=O)N1C[C@@H](NC(=O)CCCC(=O)NCCCCC#Cc2cccc(Cn3c(-c4ccccc4)c(-c4ccccc4)c4c(=N)n([C@H]5CC[C@H](O)CC5)cnc43)c2)CC1C(=O)N[C@@H]1CCCc2ccccc21)C1CCCCC1	C69H84N10O6	eEF1A2	Q05639	VHL	WO-2024026064-A1
TPD-Q0C3CP	WO2024026064A1_14	.	N=c1c2c(-c3ccccc3)c(-c3ccccc3)n(Cc3cccc(C#CCCCCNC(=O)CCCC(=O)NCCOCCOCCOCCOCCNc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)c3)c2ncn1[C@H]1CC[C@H](O)CC1	C65H75N9O11	eEF1A2	Q05639	CRBN	WO-2024026064-A1
TPD-EN3QA7	WO2024026064A1_15	.	N=c1c2c(-c3ccccc3)c(-c3ccccc3)n(Cc3cccc(C#CCCCCNC(=O)CCCC(=O)NCCOCCOCCNc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)c3)c2ncn1[C@H]1CC[C@H](O)CC1	C61H67N9O9	eEF1A2	Q05639	CRBN	WO-2024026064-A1
TPD-6LN8SQ	WO2024026064A1_16	.	N=c1c2c(-c3ccccc3)c(-c3ccccc3)n(Cc3cccc(C#CCN4CCN(C(=O)CCCCCNc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)c3)c2ncn1[C@H]1CC[C@H](O)CC1	C57H59N9O6	eEF1A2	Q05639	CRBN	WO-2024026064-A1
TPD-F5KRXM	WO2024026064A1_17	.	C[C@@H](C(=O)N[C@H](C(=O)N1C[C@@H](NC(=O)CCCC#Cc2cccc(Cn3c(-c4ccccc4)c(-c4ccccc4)c4c(=N)n(C5CCC(O)CC5)cnc43)c2)CC1C(=O)N[C@@H]1CCCc2ccccc21)C1CCCCC1)N(C)C(=O)OC(C)(C)C	C69H83N9O7	eEF1A2	Q05639	VHL	WO-2024026064-A1
TPD-GWT7YV	WO2024026064A1_18	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)C(NC(=O)CCCCC(=O)NCCCNC(=O)CCC#Cc2cccc(Cn3c(-c4ccccc4)c(-c4ccccc4)c4c(=N)n([C@H]5CC[C@H](O)CC5)cnc43)c2)C(C)(C)C)cc1	C67H78N10O7S	eEF1A2	Q05639	VHL	WO-2024026064-A1
TPD-TGHCF3	WO2024026064A1_19	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCC(=O)NCCCNC(=O)CCC#Cc2cccc(Cn3c(-c4ccccc4)c(-c4ccccc4)c4c(=N)n([C@H]5CC[C@H](O)CC5)cnc43)c2)C(C)(C)C)cc1	C65H74N10O7S	eEF1A2	Q05639	VHL	WO-2024026064-A1
TPD-C82KK0	WO2024026064A1_20	.	N=c1c2c(-c3ccccc3)c(-c3ccccc3)n(Cc3cccc(C#CCCC(=O)NCCCNC(=O)CCOCCOCCNc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)c3)c2ncn1[C@H]1CC[C@H](O)CC1	C59H63N9O9	eEF1A2	Q05639	CRBN	WO-2024026064-A1
TPD-RF9852	WO2024026064A1_21	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCC(=O)NCCCC(=O)N2CCN(CC#Cc3cccc(Cn4c(-c5ccccc5)c(-c5ccccc5)c5c(=N)n([C@H]6CC[C@H](O)CC6)cnc54)c3)CC2)C(C)(C)C)cc1	C68H79N11O7S	eEF1A2	Q05639	VHL	WO-2024026064-A1
TPD-EWC4QY	WO2024026064A1_22	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCC(=O)NCCCC(=O)N2CCN(CC#Cc3cccc(Cn4c(-c5ccccc5)c(-c5ccccc5)c5c(=N)n([C@H]6CC[C@H](O)CC6)cnc54)c3)CC2)C(C)(C)C)cc1	C70H83N11O7S	eEF1A2	Q05639	VHL	WO-2024026064-A1
TPD-98OM8S	WO2024026064A1_23	.	N=c1c2c(-c3ccccc3)c(-c3ccccc3)n(Cc3cccc(C#CCN4CCN(C(=O)CCCNC(=O)CCOCCOCCNc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)c3)c2ncn1[C@H]1CC[C@H](O)CC1	C62H68N10O9	eEF1A2	Q05639	CRBN	WO-2024026064-A1
TPD-8CJCY6	WO2024026064A1_24	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)C(NC(=O)CCCCCCC(=O)NCCCC(=O)N2CCN(CC#Cc3cccc(Cn4c(-c5ccccc5)c(-c5ccccc5)c5c(=N)n([C@H]6CC[C@H](O)CC6)cnc54)c3)CC2)C(C)(C)C)cc1	C72H87N11O7S	eEF1A2	Q05639	VHL	WO-2024026064-A1
TPD-LBWC0D	WO2024026064A1_25	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCOCCOCCOCCC(=O)NCCCC(=O)N2CCN(CC#Cc3cccc(Cn4c(-c5ccccc5)c(-c5ccccc5)c5c(=N)n([C@H]6CC[C@H](O)CC6)cnc54)c3)CC2)C(C)(C)C)cc1	C74H91N11O10S	eEF1A2	Q05639	VHL	WO-2024026064-A1
TPD-Z4V7IJ	WO2024026064A1_26	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCOCCC(=O)NCCCC(=O)N2CCN(CC#Cc3cccc(Cn4c(-c5ccccc5)c(-c5ccccc5)c5c(=N)n([C@H]6CC[C@H](O)CC6)cnc54)c3)CC2)C(C)(C)C)cc1	C70H83N11O8S	eEF1A2	Q05639	VHL	WO-2024026064-A1
TPD-879A3R	WO2024026064A1_27	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCOCCOCCOCCC(=O)NCCCNC(=O)CCC#Cc2cccc(Cn3c(-c4ccccc4)c(-c4ccccc4)c4c(=N)n([C@H]5CC[C@H](O)CC5)cnc43)c2)C(C)(C)C)cc1	C71H86N10O10S	eEF1A2	Q05639	VHL	WO-2024026064-A1
TPD-JOFHNV	WO2024026064A1_28	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCOCCC(=O)NCCCNC(=O)CCC#Cc2cccc(Cn3c(-c4ccccc4)c(-c4ccccc4)c4c(=N)n([C@H]5CC[C@H](O)CC5)cnc43)c2)C(C)(C)C)cc1	C67H78N10O8S	eEF1A2	Q05639	VHL	WO-2024026064-A1
TPD-LC4NJ9	WO2024026064A1_29	.	N=c1c2c(-c3ccccc3)c(-c3ccccc3)n(Cc3cccc(C#CCCC(=O)NCCCNC(=O)CCOCCNc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)c3)c2ncn1[C@H]1CC[C@H](O)CC1	C57H59N9O8	eEF1A2	Q05639	CRBN	WO-2024026064-A1
TPD-6MKR0Y	WO2024026064A1_30	.	N=c1c2c(-c3ccccc3)c(-c3ccccc3)n(Cc3cccc(C#CCCC(=O)NCCCNC(=O)CCOCCOCCOCCNc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)c3)c2ncn1[C@H]1CC[C@H](O)CC1	C61H67N9O10	eEF1A2	Q05639	CRBN	WO-2024026064-A1
TPD-UYPBUO	WO2024026064A1_31	.	N=c1c2c(-c3ccccc3)c(-c3ccccc3)n(Cc3cccc(C#CCN4CCN(C(=O)CCCNC(=O)CCCCCNc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)c3)c2ncn1[C@H]1CC[C@H](O)CC1	C61H66N10O7	eEF1A2	Q05639	CRBN	WO-2024026064-A1
TPD-E2FPRQ	SCHEMBL27440079	3-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]-N-[[4-[[3-(4-hydroxycyclohexyl)-4-imino-5,6-diphenylpyrrolo[2,3-d]pyrimidin-7-yl]methyl]phenyl]methyl]propanamide	N=c1c2c(-c3ccccc3)c(-c3ccccc3)n(Cc3ccc(CNC(=O)CCOCCNc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)cc3)c2ncn1[C@H]1CC[C@H](O)CC1	C50H50N8O7	eEF1A2	Q05639	CRBN	WO-2024026064-A1
TPD-L5SXU1	SCHEMBL27440107	6-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]-N-[[4-[[3-(4-hydroxycyclohexyl)-4-imino-5,6-diphenylpyrrolo[2,3-d]pyrimidin-7-yl]methyl]phenyl]methyl]hexanamide; SCHEMBL30742516	N=c1c2c(-c3ccccc3)c(-c3ccccc3)n(Cc3ccc(CNC(=O)CCCCCNc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)cc3)c2ncn1[C@H]1CC[C@H](O)CC1	C51H52N8O6	eEF1A2	Q05639	CRBN	WO-2024026064-A1
TPD-5I5IBN	WO2024026064A1_34	.	Cc1c(-c2ccccc2)c2c(=N)n([C@H]3CC[C@H](O)CC3)cnc2n1Cc1ccc(CNC(=O)CCOCCOCCOCCNc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)cc1	C49H56N8O9	eEF1A2	Q05639	CRBN	WO-2024026064-A1
TPD-JLMNUU	SCHEMBL27440157	4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]-N-[[4-[[3-(4-hydroxycyclohexyl)-4-imino-5,6-diphenylpyrrolo[2,3-d]pyrimidin-7-yl]methyl]phenyl]methyl]butanamide	N=c1c2c(-c3ccccc3)c(-c3ccccc3)n(Cc3ccc(CNC(=O)CCCNc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)cc3)c2ncn1[C@H]1CC[C@H](O)CC1	C49H48N8O6	eEF1A2	Q05639	CRBN	WO-2024026064-A1
TPD-S0KRKX	SCHEMBL27440173	3-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]-N-[[4-[[3-(4-hydroxycyclohexyl)-4-imino-5,6-diphenylpyrrolo[2,3-d]pyrimidin-7-yl]methyl]phenyl]methyl]propanamide	N=c1c2c(-c3ccccc3)c(-c3ccccc3)n(Cc3ccc(CNC(=O)CCOCCOCCNc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)cc3)c2ncn1[C@H]1CC[C@H](O)CC1	C52H54N8O8	eEF1A2	Q05639	CRBN	WO-2024026064-A1
TPD-TCPDMQ	SCHEMBL27440330	3-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]-N-[[3-[[3-(4-hydroxycyclohexyl)-4-imino-5,6-diphenylpyrrolo[2,3-d]pyrimidin-7-yl]methyl]phenyl]methyl]propanamide	N=c1c2c(-c3ccccc3)c(-c3ccccc3)n(Cc3cccc(CNC(=O)CCOCCOCCOCCNc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)c3)c2ncn1C1CCC(O)CC1	C54H58N8O9	eEF1A2	Q05639	CRBN	WO-2024026064-A1
TPD-V55EWO	WO2024026064A1_38	4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]-N-[[3-[[3-(4-hydroxycyclohexyl)-4-imino-5,6-diphenylpyrrolo[2,3-d]pyrimidin-7-yl]methyl]phenyl]methyl]butanamide	N=c1c2c(-c3ccccc3)c(-c3ccccc3)n(Cc3cccc(CNC(=O)CCCNc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)c3)c2ncn1[C@H]1CC[C@H](O)CC1	C49H48N8O6	eEF1A2	Q05639	CRBN	WO-2024026064-A1
TPD-AHDYIL	SCHEMBL27440289	3-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]-N-[[3-[[3-(4-hydroxycyclohexyl)-4-imino-5,6-diphenylpyrrolo[2,3-d]pyrimidin-7-yl]methyl]phenyl]methyl]propanamide; SCHEMBL30742595	N=c1c2c(-c3ccccc3)c(-c3ccccc3)n(Cc3cccc(CNC(=O)CCOCCOCCNc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)c3)c2ncn1[C@H]1CC[C@H](O)CC1	C52H54N8O8	eEF1A2	Q05639	CRBN	WO-2024026064-A1
TPD-9U0ZWE	SCHEMBL27440396	N-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethyl]-4-[[3-(4-hydroxycyclohexyl)-4-imino-5,6-diphenylpyrrolo[2,3-d]pyrimidin-7-yl]methyl]benzamide	N=c1c2c(-c3ccccc3)c(-c3ccccc3)n(Cc3ccc(C(=O)NCCOCCNc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)cc3)c2ncn1[C@H]1CC[C@H](O)CC1	C49H48N8O7	eEF1A2	Q05639	CRBN	WO-2024026064-A1
TPD-WVYPVE	WO2024026064A1_41	.	N=c1c2c(-c3ccccc3)c(-c3ccccc3)n(Cc3ccc(C(=O)NCCOCCOCCNc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)cc3)c2ncn1[C@H]1CC[C@H](O)CC1	C51H52N8O8	eEF1A2	Q05639	CRBN	WO-2024026064-A1
TPD-QQEU6L	WO2024026064A1_42	.	C[C@@H](C(=O)N[C@H](C(=O)N1C[C@@H](NC(=O)c2ccc(Cn3c(-c4ccccc4)c(-c4ccccc4)c4c(=N)n([C@H]5CC[C@H](O)CC5)cnc43)cc2)C[C@H]1C(=O)N[C@@H]1CCCc2ccccc21)C1CCCCC1)N(C)C(=O)OC(C)(C)C	C64H77N9O7	eEF1A2	Q05639	VHL	WO-2024026064-A1
TPD-5J59K0	SCHEMBL27440445	N-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethyl]-4-[[3-(4-hydroxycyclohexyl)-4-imino-5,6-diphenylpyrrolo[2,3-d]pyrimidin-7-yl]methyl]benzamide	N=c1c2c(-c3ccccc3)c(-c3ccccc3)n(Cc3ccc(C(=O)NCCNc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)cc3)c2ncn1[C@H]1CC[C@H](O)CC1	C47H44N8O6	eEF1A2	Q05639	CRBN	WO-2024026064-A1
TPD-V6LUAM	SCHEMBL27440368	N-[5-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]pentyl]-4-[[3-(4-hydroxycyclohexyl)-4-imino-5,6-diphenylpyrrolo[2,3-d]pyrimidin-7-yl]methyl]benzamide	N=c1c2c(-c3ccccc3)c(-c3ccccc3)n(Cc3ccc(C(=O)NCCCCCNc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)cc3)c2ncn1[C@H]1CC[C@H](O)CC1	C50H50N8O6	eEF1A2	Q05639	CRBN	WO-2024026064-A1
TPD-R2YKAA	WO2024026064A1_45	.	O=C(CCCCCNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O)NCc1cccc(Cn2c(-c3ccccc3)c(-c3ccccc3)c3c(N[C@H]4CC[C@H](O)CC4)ncnc32)c1	C51H52N8O6	eEF1A2	Q05639	CRBN	WO-2024026064-A1
TPD-VHRW3U	SCHEMBL27438529	6-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]-N-[[3-[[3-(4-hydroxycyclohexyl)-4-imino-5,6-diphenylpyrrolo[2,3-d]pyrimidin-7-yl]methyl]phenyl]methyl]hexanamide; SCHEMBL27440254	N=c1c2c(-c3ccccc3)c(-c3ccccc3)n(Cc3cccc(CNC(=O)CCCCCNc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)c3)c2ncn1[C@H]1CC[C@H](O)CC1	C51H52N8O6	eEF1A2	Q05639	CRBN	WO-2024026064-A1
TPD-RH71WH	WO2024026064A1_47	.	O=C(CCOCCNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O)NCc1cccc(Cn2c(-c3ccccc3)c(-c3ccccc3)c3c(N[C@H]4CC[C@H](O)CC4)ncnc32)c1	C50H50N8O7	eEF1A2	Q05639	CRBN	WO-2024026064-A1
TPD-LZJKYN	SCHEMBL27440274	3-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]-N-[[3-[[3-(4-hydroxycyclohexyl)-4-imino-5,6-diphenylpyrrolo[2,3-d]pyrimidin-7-yl]methyl]phenyl]methyl]propanamide; SCHEMBL30742518	N=c1c2c(-c3ccccc3)c(-c3ccccc3)n(Cc3cccc(CNC(=O)CCOCCNc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)c3)c2ncn1[C@H]1CC[C@H](O)CC1	C50H50N8O7	eEF1A2	Q05639	CRBN	WO-2024026064-A1
TPD-EDLJ4B	WO2024026064A1_49	.	O=C1CCC(N2C(=O)c3cccc(NCCCCCNC(=O)c4ccc(Cn5c(-c6ccccc6)c(-c6ccccc6)c6c(NC7CCC(O)CC7)ncnc65)cc4)c3C2=O)C(=O)N1	C50H50N8O6	eEF1A2	Q05639	CRBN	WO-2024026064-A1
TPD-PY8R0L	SCHEMBL30742562	(2S,4S)-1-[(2S)-2-cyclohexyl-2-[[(2S)-2-(methylamino)propanoyl]amino]acetyl]-4-[[4-[[3-(4-hydroxycyclohexyl)-4-imino-5,6-diphenylpyrrolo[2,3-d]pyrimidin-7-yl]methyl]benzoyl]amino]-N-[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]pyrrolidine-2-carboxamide	CN[C@@H](C)C(=O)N[C@H](C(=O)N1C[C@@H](NC(=O)c2ccc(Cn3c(-c4ccccc4)c(-c4ccccc4)c4c(=N)n(C5CCC(O)CC5)cnc43)cc2)C[C@H]1C(=O)N[C@@H]1CCCc2ccccc21)C1CCCCC1	C59H69N9O5	eEF1A2	Q05639	VHL	WO-2024026064-A1
TPD-YPB02X	WO2024026064A1_51	.	CN[C@@H](C)C(=O)N[C@H](C(=O)N1C[C@@H](NC(=O)CCCC#Cc2cccc(Cn3c(-c4ccccc4)c(-c4ccccc4)c4c(=N)n([C@H]5CC[C@H](O)CC5)cnc43)c2)C[C@H]1C(=O)N[C@@H]1CCCc2ccccc21)C1CCCCC1	C64H75N9O5	eEF1A2	Q05639	CRBN	WO-2024026064-A1
TPD-DE4HJ0	WO2024026064A1_52	.	O=C1CCC(N2C(=O)c3cccc(NCCCCCNC(=O)c4ccc(Cn5cc(-c6ccccc6)c6c(NC7CCC(O)CC7)ncnc65)cc4)c3C2=O)C(=O)N1	C44H46N8O6	eEF1A2	Q05639	CRBN	WO-2024026064-A1
TPD-5YOOFB	WO2024026064A1_53	.	N=c1c2c(-c3ccccc3)c(-c3ccccc3)n(Cc3ccc(C(=O)NCCCCCNc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)cc3)c2ncn1C1CCOCC1	C49H48N8O6	eEF1A2	Q05639	CRBN	WO-2024026064-A1
TPD-7PCND3	WO2024026064A1_54	.	N=c1c2c(-c3ccccc3)c(-c3ccccc3)n(Cc3ccccc3)c2ncn1[C@H]1CC[C@H](OC(=O)CCCCCNc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)CC1	C50H49N7O6	eEF1A2	Q05639	CRBN	WO-2024026064-A1
TPD-7QS1EZ	SCHEMBL27438903	Methyl 5-amino-4-[4-[[4-[4-(7-benzyl-4-imino-5,6-diphenylpyrrolo[2,3-d]pyrimidin-3-yl)cyclohexyl]oxy-4-oxobutyl]amino]-1,3-dioxoisoindol-2-yl]-5-oxopentanoate	COC(=O)CCC(C(N)=O)N1C(=O)c2cccc(NCCCC(=O)O[C@H]3CC[C@H](n4cnc5c(c(-c6ccccc6)c(-c6ccccc6)n5Cc5ccccc5)c4=N)CC3)c2C1=O	C49H49N7O7	eEF1A2	Q05639	CRBN	WO-2024026064-A1
TPD-DIKB2R	SCHEMBL27438900	[4-(7-Benzyl-4-imino-5,6-diphenylpyrrolo[2,3-d]pyrimidin-3-yl)cyclohexyl] 4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]butanoate; SCHEMBL30742574	N=c1c2c(-c3ccccc3)c(-c3ccccc3)n(Cc3ccccc3)c2ncn1[C@H]1CC[C@H](OC(=O)CCCNc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)CC1	C48H45N7O6	eEF1A2	Q05639	CRBN	WO-2024026064-A1
TPD-XCCEK4	SCHEMBL27440538	[4-(7-Benzyl-4-imino-5,6-diphenylpyrrolo[2,3-d]pyrimidin-3-yl)cyclohexyl] 3-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]propanoate; SCHEMBL30742540	N=c1c2c(-c3ccccc3)c(-c3ccccc3)n(Cc3ccccc3)c2ncn1[C@H]1CC[C@H](OC(=O)CCOCCOCCOCCNc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)CC1	C53H55N7O9	eEF1A2	Q05639	CRBN	WO-2024026064-A1
TPD-JNVTLU	SCHEMBL27254022	2-(2,6-Dioxopiperidin-3-yl)-4-[2-[4-[4-[[5-(3-methylphenyl)imidazo[1,2-a]pyrazin-8-yl]amino]phenyl]piperazin-1-yl]-2-oxoethoxy]isoindole-1,3-dione	CC1=CC=CC(C2=CN=C(NC3=CC=C(N4CCN(C(=O)COC5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)CC4)C=C3)C3=NC=CN23)=C1	C38H34N8O6	IRAK3	Q9Y616	CRBN	WO-2024026256-A1
TPD-54M20M	SCHEMBL27254194	2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxy-N-[4-[4-[4-[[5-(3-methylphenyl)imidazo[1,2-a]pyrazin-8-yl]amino]phenyl]piperazin-1-yl]-4-oxobutyl]acetamide	CC1=CC=CC(C2=CN=C(NC3=CC=C(N4CCN(C(=O)CCCNC(=O)COC5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)CC4)C=C3)C3=NC=CN23)=C1	C42H41N9O7	IRAK3	Q9Y616	CRBN	WO-2024026256-A1
TPD-327GNU	SCHEMBL27254198	2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxy-N-[2-[3-[4-[4-[[5-(3-methylphenyl)imidazo[1,2-a]pyrazin-8-yl]amino]phenyl]piperazin-1-yl]-3-oxopropoxy]ethyl]acetamide	CC1=CC=CC(C2=CN=C(NC3=CC=C(N4CCN(C(=O)CCOCCNC(=O)COC5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)CC4)C=C3)C3=NC=CN23)=C1	C43H43N9O8	IRAK3	Q9Y616	CRBN	WO-2024026256-A1
TPD-1VZMVK	SCHEMBL27254023	2-(2,6-Dioxopiperidin-3-yl)-5-[2-[4-[4-[[5-(3-methylphenyl)imidazo[1,2-a]pyrazin-8-yl]amino]phenyl]piperazin-1-yl]-2-oxoethoxy]isoindole-1,3-dione	CC1=CC=CC(C2=CN=C(NC3=CC=C(N4CCN(C(=O)COC5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)C=C3)C3=NC=CN23)=C1	C38H34N8O6	IRAK3	Q9Y616	CRBN	WO-2024026256-A1
TPD-SGJ2K0	SCHEMBL27254037	2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxy-N-[4-[4-[4-[[5-(3-methylphenyl)imidazo[1,2-a]pyrazin-8-yl]amino]phenyl]piperazin-1-yl]-4-oxobutyl]acetamide	CC1=CC=CC(C2=CN=C(NC3=CC=C(N4CCN(C(=O)CCCNC(=O)COC5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)C=C3)C3=NC=CN23)=C1	C42H41N9O7	IRAK3	Q9Y616	CRBN	WO-2024026256-A1
TPD-1N6RL5	SCHEMBL27254038	2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxy-N-[2-[3-[4-[4-[[5-(3-methylphenyl)imidazo[1,2-a]pyrazin-8-yl]amino]phenyl]piperazin-1-yl]-3-oxopropoxy]ethyl]acetamide	CC1=CC=CC(C2=CN=C(NC3=CC=C(N4CCN(C(=O)CCOCCNC(=O)COC5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)C=C3)C3=NC=CN23)=C1	C43H43N9O8	IRAK3	Q9Y616	CRBN	WO-2024026256-A1
TPD-UQKTM0	SCHEMBL27254039	2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxy-N-[2-[4-[4-[[5-(3-methylphenyl)imidazo[1,2-a]pyrazin-8-yl]amino]phenyl]piperazin-1-yl]ethyl]acetamide	CC1=CC=CC(C2=CN=C(NC3=CC=C(N4CCN(CCNC(=O)COC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)C3=NC=CN23)=C1	C40H39N9O6	IRAK3	Q9Y616	CRBN	WO-2024026256-A1
TPD-JIJV4S	SCHEMBL27254040	2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxy-N-[2-[4-[4-[[5-(3-methylphenyl)imidazo[1,2-a]pyrazin-8-yl]amino]pyrazol-1-yl]piperidin-1-yl]ethyl]acetamide	CC1=CC=CC(C2=CN=C(NC3=CN(C4CCN(CCNC(=O)COC5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)N=C3)C3=NC=CN23)=C1	C38H38N10O6	IRAK3	Q9Y616	CRBN	WO-2024026256-A1
TPD-D73MB0	SCHEMBL27254042	2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxy-N-[2-[4-[3-[[5-(3-methylphenyl)imidazo[1,2-a]pyrazin-8-yl]amino]phenyl]piperidin-1-yl]ethyl]acetamide	CC1=CC=CC(C2=CN=C(NC3=CC=CC(C4CCN(CCNC(=O)COC5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)=C3)C3=NC=CN23)=C1	C41H40N8O6	IRAK3	Q9Y616	CRBN	WO-2024026256-A1
TPD-YM5872	SCHEMBL27254067	2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxy-N-[2-[4-[4-[[5-(3-methylphenyl)imidazo[1,2-a]pyrazin-8-yl]amino]phenyl]piperidin-1-yl]ethyl]acetamide	CC1=CC=CC(C2=CN=C(NC3=CC=C(C4CCN(CCNC(=O)COC5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)C=C3)C3=NC=CN23)=C1	C41H40N8O6	IRAK3	Q9Y616	CRBN	WO-2024026256-A1
TPD-6UD40S	SCHEMBL27254068	2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxy-N-[2-[4-[3-[[5-(3-methylphenyl)imidazo[1,2-a]pyrazin-8-yl]amino]phenyl]piperazin-1-yl]ethyl]acetamide	CC1=CC=CC(C2=CN=C(NC3=CC=CC(N4CCN(CCNC(=O)COC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)=C3)C3=NC=CN23)=C1	C40H39N9O6	IRAK3	Q9Y616	CRBN	WO-2024026256-A1
TPD-AXNFHR	SCHEMBL27254070	3-[6-[9-[4-[4-[[5-(3-methylphenyl)imidazo[1,2-a]pyrazin-8-yl]amino]pyrazol-1-yl]piperidin-1-yl]-3-azaspiro[5.5]undecane-3-carbonyl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CC1=CC=CC(C2=CN=C(NC3=CN(C4CCN(C5CCC6(CC5)CCN(C(=O)C5=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C5)CC6)CC4)N=C3)C3=NC=CN23)=C1	C45H50N10O4	IRAK3	Q9Y616	CRBN	WO-2024026256-A1
TPD-EFN6AM	WO2024027706A1_1	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC#CC3=CC=C(OCCCC4=C(C(=O)O)N=C(N5CCC6=CC=CC(C(=O)NC7=NC8=C(C=CC=C8)S7)=C6C5)S4)C=C3)C(C)(C)C)C=C2)SC=N1	C62H68N8O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-SGQDH1	WO2024027706A1_10	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCCC#CC3=CC=C(OCCCC4=C(C(=O)O)N=C(N5CCC6=CC=CC(C(=O)NC7=NC8=C(C=CC=C8)S7)=C6C5)S4)C=C3)C(C)(C)C)C=C2)SC=N1	C63H70N8O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-IFZW0X	WO2024027706A1_100	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC3=CN(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)N=C3)C(C)(C)C)C=C2)SC=N1	C64H72N10O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-XXFX97	WO2024027706A1_101	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCN3C=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)C=N3)C(C)(C)C)C=C2)SC=N1	C64H72N10O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-ZU8HU6	WO2024027706A1_102	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCC3=CN(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)N=C3)C(C)(C)C)C=C2)SC=N1	C63H70N10O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-LNOGP1	WO2024027706A1_103	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC3=CC4=C(C=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)N=C3)C(C)(C)C)C=C2)SC=N1	C64H71N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-ZSSF5V	WO2024027706A1_104	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC3=NC(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)=NO3)C(C)(C)C)C=C2)SC=N1	C63H70N10O9S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-RPZMPZ	WO2024027706A1_105	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC3=NC(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)=NS3)C(C)(C)C)C=C2)SC=N1	C63H70N10O8S4	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-Y29XCY	WO2024027706A1_106	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC3=CN=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)S3)C(C)(C)C)C=C2)SC=N1	C64H71N9O8S4	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-D20MTF	WO2024027706A1_107	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC3=NC=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)S3)C(C)(C)C)C=C2)SC=N1	C64H71N9O8S4	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-UC6SQC	WO2024027706A1_108	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC3=NN=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)S3)C(C)(C)C)C=C2)SC=N1	C63H70N10O8S4	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-VZRTCI	WO2024027706A1_109	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC3=NOC(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)=N3)C(C)(C)C)C=C2)SC=N1	C63H70N10O9S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-V3O4ZQ	WO2024027706A1_11	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCC#CC3=CC=C(OCCCC4=C(C(=O)O)N=C(N5CCC6=CC=CC(C(=O)NC7=NC8=C(C=CC=C8)S7)=C6C5)S4)C=C3)C(C)(C)C)C=C2)SC=N1	C60H64N8O10S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-FBAMGR	WO2024027706A1_110	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCN3CCN(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C65H78N10O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-PZ5PA9	WO2024027706A1_111	.	C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](NC(=O)CCCCCCCC#CC1=CC=C(OCCCC2=C(C(=O)O)N=C(N3CCC4=CC=CC(C(=O)NC5=NC6=C(C=CC=C6)S5)=C4C3)S2)C=C1)C(C)(C)C)C1=CC=CC=C1	C59H67N7O8S2	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-DKV8PZ	WO2024027706A1_112	.	C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](NC(=O)CCCCCCC#CC1=CC=C(OCCCC2=C(C(=O)O)N=C(N3CCC4=CC=CC(C(=O)NC5=NC6=C(C=CC=C6)S5)=C4C3)S2)C=C1)C(C)(C)C)C1=CC=CC=C1	C58H65N7O8S2	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-9CPFTS	WO2024027706A1_113	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC#CC3=CC=C(OCCCC4=C(C(=O)O)N=C(N5CCC6=CC=CC(C(=O)NC7=NC8=C(C=CC=C8)S7)=C6C5)S4)C=C3)C(C)(C)C)C=C2)OC=N1	C63H70N8O9S2	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-PH29DO	WO2024027706A1_114	.	CC1=C(C2=CC=C(C3(NC(=O)[C@@H]4C[C@@H](O)CN4C(=O)[C@@H](NC(=O)CCCCCCCC#CC4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)C(C)(C)C)CC3)C=C2)SC=N1	C64H70N8O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-LJWCJ9	WO2024027706A1_115	.	CC1=C(C2=CC=C(N(C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC#CC3=CC=C(OCCCC4=C(C(=O)O)N=C(N5CCC6=CC=CC(C(=O)NC7=NC8=C(C=CC=C8)S7)=C6C5)S4)C=C3)C(C)(C)C)C=C2)SC=N1	C62H69N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-TWDWOG	WO2024027706A1_116	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3[C@@H](F)[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC#CC3=CC=C(OCCCC4=C(C(=O)O)N=C(N5CCC6=CC=CC(C(=O)NC7=NC8=C(C=CC=C8)S7)=C6C5)S4)C=C3)C(C)(C)C)C=C2)SC=N1	C63H69FN8O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-152G8R	WO2024027706A1_117	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(O)[C@@H](NC(=O)CCOC3CCC(C#CC4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C64H72N8O9S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-L6UW4A	WO2024027706A1_118	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCC3CCC(C#CC4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C64H70N8O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-VEEBRN	WO2024027706A1_119	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCC3CCC(C#CC4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C65H72N8O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-ICHLEB	WO2024027706A1_12	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCC#CC3=CC=C(OCCCC4=C(C(=O)O)N=C(N5CCC6=CC=CC(C(=O)NC7=NC8=C(C=CC=C8)S7)=C6C5)S4)C=C3)C(C)(C)C)C=C2)SC=N1	C61H66N8O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-XZQFCA	WO2024027706A1_120	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCC3CCC(C#CC4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C64H70N8O9S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-QYCD89	WO2024027706A1_121	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CC3CCC(OCCCC#CC4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=CC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C67H75N7O9S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-B2OGSL	WO2024027706A1_122	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CC3CCC(OCCC#CC4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=CC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C66H73N7O9S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-1C03HO	WO2024027706A1_123	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)[C@H]3CC[C@H](OCCCC#CC4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C65H72N8O9S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-33Q9CF	WO2024027706A1_124	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCOC3CCC(CC#CC4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C65H72N8O9S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-X8CUGZ	WO2024027706A1_125	.	CC(C)=C(SC=N)C1=CC=C([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCCCCC#CC2=CC=C(OCCCC3=C(C(=O)O)N=C(N4CCC5=CC=CC(C(=O)NC6=NC7=C(C=CC=C7)S6)=C5C4)S3)C=C2)C(C)(C)C)C=C1	C63H72N8O9S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-4H2WL4	WO2024027706A1_126	.	CC(C)=C(SC=N)C1=CC=C([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCCCC#CC2=CC=C(OCCCC3=C(C(=O)O)N=C(N4CCC5=CC=CC(C(=O)NC6=NC7=C(C=CC=C7)S6)=C5C4)S3)C=C2)C(C)(C)C)C=C1	C65H76N8O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-PRKFP4	WO2024027706A1_127	.	CC(C)=C(SC=N)C1=CC=C([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCCCCC#CC2=CC=C(OCCCC3=C(C(=O)O)N=C(N4CCC5=CC=CC(C(=O)NC6=NC7=C(C=CC=C7)S6)=C5C4)S3)C=C2)C(C)(C)C)C=C1	C66H78N8O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-LDESPK	WO2024027706A1_128	.	CC(C)=C(SC=N)C1=CC=C([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCCCCCC#CC2=CC=C(OCCCC3=C(C(=O)O)N=C(N4CCC5=CC=CC(C(=O)NC6=NC7=C(C=CC=C7)S6)=C5C4)S3)C=C2)C(C)(C)C)C=C1	C64H74N8O9S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-V7I3B3	WO2024027706A1_129	.	CC(C)=C(SC=N)C1=CC=C([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCCC2CCC(C#CC3=CC=C(OCCCC4=C(C(=O)O)N=C(N5CCC6=CC=CC(C(=O)NC7=NC8=C(C=CC=C8)S7)=C6C5)S4)C=C3)CC2)C(C)(C)C)C=C1	C66H76N8O9S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-IBZNF1	WO2024027706A1_13	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CC3CCC4(CC3)CCN(CC#CC3=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C3)CC4)C(C)(C)C)C=C2)SC=N1	C67H75N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-S48U0O	WO2024027706A1_130	.	CC(C)=C(SC=N)C1=CC=C([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COC2CCC(CC#CC3=CC=C(OCCCC4=C(C(=O)O)N=C(N5CCC6=CC=CC(C(=O)NC7=NC8=C(C=CC=C8)S7)=C6C5)S4)C=C3)CC2)C(C)(C)C)C=C1	C65H74N8O9S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-5YBNFJ	WO2024027706A1_131	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCOC3CCC(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C66H78N8O9S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-TP4PH0	WO2024027706A1_132	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC3=NC=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)N3)C(C)(C)C)C=C2)SC=N1	C64H72N10O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-TJKVZE	WO2024027706A1_133	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCC([C@H]4C[C@@H](C#CC5=CC=C(OCCCC6=C(C(=O)O)N=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=C(C=CC=C%10)S9)=C8C7)S6)C=C5)C4)CC3)C(C)(C)C)C=C2)SC=N1	C66H73N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-1ASCJO	WO2024027706A1_134	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCC([C@H]4C[C@H](C#CC5=CC=C(OCCCC6=C(C(=O)O)N=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=C(C=CC=C%10)S9)=C8C7)S6)C=C5)C4)CC3)C(C)(C)C)C=C2)SC=N1	C66H73N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-T8KAES	WO2024027706A1_135	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3CCC4(CC3)CCN(CC#CC3=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C3)CC4)C(C)(C)C)C=C2)SC=N1	C67H75N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-M1EXAZ	WO2024027706A1_136	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CC3CCC4(CC3)CCN(C(C)C#CC3=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C3)CC4)C(C)(C)C)C=C2)SC=N1	C69H79N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-H65SEY	WO2024027706A1_137	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CC3CCC4(CC3)CCN(CC#CC3=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C3)CC4)C(C)(C)C)C=C2)SC=N1	C68H77N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-CLYLND	WO2024027706A1_138	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)[C@H]3CC[C@@H](C4CCN(CC#CC5=CC=C(OCCCC6=C(C(=O)O)N=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=C(C=CC=C%10)S9)=C8C7)S6)C=C5)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C68H77N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-A7DUCJ	WO2024027706A1_139	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)[C@H]3CC[C@H](C4CCN(CC#CC5=CC=C(OCCCC6=C(C(=O)O)N=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=C(C=CC=C%10)S9)=C8C7)S6)C=C5)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C68H77N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-1QAF5L	WO2024027706A1_14	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CC3CCC(N4CC(C#CC5=CC=C(OCCCC6=C(C(=O)O)N=C(NCCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7)S6)C=C5)C4)CC3)C(C)(C)C)C=C2)SC=N1	C64H71N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-Y3YWFA	WO2024027706A1_140	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)[C@H]3C[C@@H](C4CCN(CC#CC5=CC=C(OCCCC6=C(C(=O)O)N=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=C(C=CC=C%10)S9)=C8C7)S6)C=C5)CC4)C3)C(C)(C)C)C=C2)SC=N1	C66H73N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-XSSWVU	WO2024027706A1_141	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)[C@H]3C[C@H](C4CCN(CC#CC5=CC=C(OCCCC6=C(C(=O)O)N=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=C(C=CC=C%10)S9)=C8C7)S6)C=C5)CC4)C3)C(C)(C)C)C=C2)SC=N1	C66H73N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-D5V32O	WO2024027706A1_142	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)[C@H]3CC[C@@H](N4CCC(CC#CC5=CC=C(OCCCC6=C(C(=O)O)N=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=C(C=CC=C%10)S9)=C8C7)S6)C=C5)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C68H77N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-4034AZ	WO2024027706A1_143	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)[C@H]3CC[C@H](N4CCC(CC#CC5=CC=C(OCCCC6=C(C(=O)O)N=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=C(C=CC=C%10)S9)=C8C7)S6)C=C5)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C68H77N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-OOIITG	WO2024027706A1_144	.	C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](NC(=O)CC1CCC2(CC1)CCN(CC#CC1=CC=C(OCCCC3=C(C(=O)O)N=C(N4CCC5=CC=CC(C(=O)NC6=NC7=C(C=CC=C7)S6)=C5C4)S3)C=C1)CC2)C(C)(C)C)C1=CC=CC=C1	C64H74N8O8S2	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-U2O4HW	WO2024027706A1_145	.	CC1=C(C2=CC=C(C3(NC(=O)[C@@H]4C[C@@H](O)CN4C(=O)[C@@H](NC(=O)CC4CCC5(CC4)CCN(CC#CC4=CC=C(OCCCC6=C(C(=O)O)N=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=C(C=CC=C%10)S9)=C8C7)S6)C=C4)CC5)C(C)(C)C)CC3)C=C2)SC=N1	C69H77N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-DYVNJ3	WO2024027706A1_146	.	CC1=C(C2=CC=C(N(C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CC3CCC4(CC3)CCN(CC#CC3=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C3)CC4)C(C)(C)C)C=C2)SC=N1	C67H76N10O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-SDUPPF	WO2024027706A1_147	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCC3=CN=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)N=C3)C(C)(C)C)C=C2)SC=N1	C63H68N10O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-ZGGZQQ	WO2024027706A1_148	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCC4(CCC(C5C=NC(C6=CC=C(OCCCC7=C(C(=O)O)N=C(N8CCC9=CC=CC(C(=O)NC%10=NC%11=C(C=CC=C%11)S%10)=C9C8)S7)C=C6)=NC5)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C69H79N11O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-P0FB82	WO2024027706A1_149	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCC4(CC3)CCN(C3C=NC(C5=CC=C(OCCCC6=C(C(=O)O)N=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=C(C=CC=C%10)S9)=C8C7)S6)C=C5)=NC3)CC4)C(C)(C)C)C=C2)SC=N1	C68H78N12O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-FAFTSA	WO2024027706A1_15	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3CCN(C4CN(CC#CC5=CC=C(OCCCC6=C(C(=O)O)N=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=C(C=CC=C%10)S9)=C8C7)S6)C=C5)C4)CC3)C(C)(C)C)C=C2)SC=N1	C64H70N10O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-BN0D6W	WO2024027706A1_150	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CC3CCC4(CC3)CCN(CC3=CN=C(C5=CC=C(OCCCC6=C(C(=O)O)N=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=C(C=CC=C%10)S9)=C8C7)S6)C=C5)N=C3)CC4)C(C)(C)C)C=C2)SC=N1	C70H79N11O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-F80R0E	WO2024027706A1_151	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3CCC4(CC3)CCN(CC3=CN=C(C5=CC=C(OCCCC6=C(C(=O)O)N=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=C(C=CC=C%10)S9)=C8C7)S6)C=C5)N=C3)CC4)C(C)(C)C)C=C2)SC=N1	C69H77N11O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-M6VGB6	WO2024027706A1_152	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3CC4(CCN(CC5=CN=C(C6=CC=C(OCCCC7=C(C(=O)O)N=C(N8CCC9=CC=CC(C(=O)NC%10=NC%11=C(C=CC=C%11)S%10)=C9C8)S7)C=C6)N=C5)CC4)C3)C(C)(C)C)C=C2)SC=N1	C67H73N11O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-CXK9IA	WO2024027706A1_153	.	C=C/C(=C\C=C\C1=C(C)N=CS1)[C@H](C)NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](NC(=O)CCN1CCC(C2=CN=C(C3=CC=C(OCCCC4=C(C(=O)O)N=C(N5CCC6=CC=CC(C(=O)NC7=NC8=C(C=CC=C8)S7)=C6C5)S4)C=C3)N=C2)CC1)C(C)(C)C	C65H73N11O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-GRYECJ	WO2024027706A1_154	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCN3CCC(C4=CN=C(C5=CC=C(OCCCC6=C(C(=O)O)N=C(N7CCC8=CC=CC(C(=O)NC9NC%10=C(C=CC=C%10)S9)=C8C7)S6)C=C5)N=C4)CC3)C(C)(C)C)C=C2)SC=N1	C66H75N11O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-TZ43HO	WO2024027706A1_155	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCOC3CCN(C4=CN=C(C5=CC=C(OCCCC6=C(C(=O)O)N=C(N7CCC8=CC=CC(C(=O)NC9NC%10=C(C=CC=C%10)S9)=C8C7)S6)C=C5)N=C4)CC3)C(C)(C)C)C=C2)SC=N1	C66H75N11O9S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-XBU8EL	WO2024027706A1_156	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CC3CCN(C4=CN=C(C5=CC=C(OCCCC6=C(C(=O)O)N=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=C(C=CC=C%10)S9)=C8C7)S6)C=C5)N=C4)CC3)C(C)(C)C)C=C2)SC=N1	C64H69N11O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-8ES5R8	WO2024027706A1_157	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCC3CCN(C4=CN=C(C5=CC=C(OCCCC6=C(C(=O)O)N=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=C(C=CC=C%10)S9)=C8C7)S6)C=C5)N=C4)CC3)C(C)(C)C)C=C2)SC=N1	C65H71N11O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-9VS9JH	WO2024027706A1_158	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3CCN(CC4CN(C5=CN=C(C6=CC=C(OCCCC7=C(C(=O)O)N=C(N8CCC9=CC=CC(C(=O)NC%10=NC%11=C(C=CC=C%11)S%10)=C9C8)S7)C=C6)N=C5)C4)CC3)C(C)(C)C)C=C2)SC=N1	C67H74N12O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-6ZLKVT	WO2024027706A1_159	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3CCN(CC4CCN(C5=CN=C(C6=CC=C(OCCCC7=C(C(=O)O)N=C(N8CCC9=CC=CC(C(=O)NC%10=NC%11=C(C=CC=C%11)S%10)=C9C8)S7)C=C6)N=C5)C4)CC3)C(C)(C)C)C=C2)SC=N1	C68H76N12O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-XHWM6V	WO2024027706A1_16	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CC4(CCC(C#CC5=CC=C(OCCCC6=C(C(=O)O)N=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=C(C=CC=C%10)S9)=C8C7)S6)C=C5)CC4)C3)C(C)(C)C)C=C2)SC=N1	C64H69N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-9AOVCM	WO2024027706A1_160	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)[C@H]3CC[C@H](OCCCC4=CN=C(C5=CC=C(OCCCC6=C(C(=O)O)N=C(N7CCC8=CC=CC(C(O)NC9=NC%10=C(C=CC=C%10)S9)=C8C7)S6)C=C5)N=C4)CC3)C(C)(C)C)C=C2)SC=N1	C67H76N10O9S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-XZ68UX	WO2024027706A1_161	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)[C@H]3CC[C@@H](OCCCC4=CN=C(C5=CC=C(OCCCC6=C(C(=O)O)N=C(N7CCC8=CC=CC(C(O)NC9=NC%10=C(C=CC=C%10)S9)=C8C7)S6)C=C5)N=C4)CC3)C(C)(C)C)C=C2)SC=N1	C67H76N10O9S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-EYTTRE	WO2024027706A1_162	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCC([C@H]4CC[C@H](C#CC5=CC=C(OCCCC6=C(C(=O)O)N=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=C(C=CC=C%10)S9)=C8C7)S6)C=C5)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C68H77N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-RJ2A0F	WO2024027706A1_163	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCC([C@H]4CC[C@@H](C#CC5=CC=C(OCCCC6=C(C(=O)O)N=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=C(C=CC=C%10)S9)=C8C7)S6)C=C5)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C68H77N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-RC2YSV	WO2024027706A1_164	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CC3CCN([C@H]4CC[C@H](C#CC5=CC=C(OCCCC6=C(C(=O)O)N=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=C(C=CC=C%10)S9)=C8C7)S6)C=C5)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C68H77N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-3AMPQD	WO2024027706A1_165	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CC3CCN([C@H]4CC[C@@H](C#CC5=CC=C(OCCCC6=C(C(=O)O)N=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=C(C=CC=C%10)S9)=C8C7)S6)C=C5)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C68H77N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-OQH9F6	WO2024027706A1_166	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CC3CCN([C@H]4C[C@@H](C#CC5=CC=C(OCCCC6=C(C(=O)O)N=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=C(C=CC=C%10)S9)=C8C7)S6)C=C5)C4)CC3)C(C)(C)C)C=C2)SC=N1	C66H73N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-1GT5PO	WO2024027706A1_167	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CC3CCN([C@H]4C[C@H](C#CC5=CC=C(OCCCC6=C(C(=O)O)N=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=C(C=CC=C%10)S9)=C8C7)S6)C=C5)C4)CC3)C(C)(C)C)C=C2)SC=N1	C66H73N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-2J226O	WO2024027706A1_168	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCC4(CCC(C#CC5=CC=C(OCCCC6=C(C(=O)O)N=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=C(C=CC=C%10)S9)=C8C7)S6)C=C5)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C67H75N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-WRPJZ4	WO2024027706A1_169	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCC4(CCC(CC#CC5=CC=C(OCCCC6=C(C(=O)O)N=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=C(C=CC=C%10)S9)=C8C7)S6)C=C5)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C68H77N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-99NMNA	WO2024027706A1_17	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCN3CCC4(CC3)CC(C#CC3=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C3)C4)C(C)(C)C)C=C2)SC=N1	C65H71N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-TLTH0R	WO2024027706A1_170	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CC3CCC4(CC3)CCN(CC3=CC=C(C5=CC=C(OCCCC6=C(C(=O)O)N=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=C(C=CC=C%10)S9)=C8C7)S6)C=C5)C=C3)CC4)C(C)(C)C)C=C2)SC=N1	C72H81N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-8GRXJK	WO2024027706A1_171	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CC3CCC4(CC3)CCN(CC3CCC(C5=CC=C(OCCCC6=C(C(=O)O)N=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=C(C=CC=C%10)S9)=C8C7)S6)C=C5)CC3)CC4)C(C)(C)C)C=C2)SC=N1	C72H87N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-6CUD44	WO2024027706A1_172	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCC#CC3=CC=C(OCCCC4=C(C(=O)O)N=C(N5CCC6=CC=CC(C(=O)NC7=NC8=C(C=CC=C8)S7)=C6C5)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C64H70N8O8S2	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-APR68F	WO2024027706A1_173	.	CC1=CC(C2=NC=C(CCCCCCCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](C)C3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)C=N2)=CC=C1OCCCC1=C(C(=O)O)N=C(N2CCC3=CC=CC(C(=O)NC4=NC5=C(C=CC=C5)S4)=C3C2)C=C1	C68H76N10O8S2	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-YR21CR	WO2024027706A1_174	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC3=CN=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)C(Cl)=C3)C(C)(C)C)C=C2)SC=N1	C66H72ClN9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-SOKEO1	WO2024027706A1_175	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCC3CCN(C4=CN=C(C5=CC=C(OCCCC6=C(C(=O)O)N=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=C(C=CC=C%10)S9)=C8C7)S6)C=C5)N=C4)CC3)C(C)(C)C)C=C2)SC=N1	C66H73N11O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-2NSW1C	WO2024027706A1_176	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCC3CCN(C4=CN=C(C5=CC=C(OCCCC6=C(C(=O)O)N=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=C(C=CC=C%10)S9)=C8C7)S6)C=C5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C67H74N10O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-JHLHYD	WO2024027706A1_177	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC3=CN=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)C(C(F)(F)F)=C3)C(C)(C)C)C=C2)SC=N1	C67H72F3N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-CTZ1B6	WO2024027706A1_178	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC3=CC=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C(Cl)=C4)N=C3)C(C)(C)C)C=C2)SC=N1	C66H72ClN9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-LN1OLN	WO2024027706A1_179	.	CC1=CC(C2=CC=C(CCCCCCCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](C)C3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)C=N2)=CC=C1OCCCC1=C(C(=O)O)N=C(N2CCC3=CC=CC(C(=O)NC4=NC5=C(C=CC=C5)S4)=C3C2)S1	C67H75N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-OX8UPJ	WO2024027706A1_18	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3CC(CN4CCC(C#CC5=CC=C(OCCCC6=C(C(=O)O)N=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=C(C=CC=C%10)S9)=C8C7)S6)C=C5)CC4)C3)C(C)(C)C)C=C2)SC=N1	C65H71N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-3VTMGZ	WO2024027706A1_180	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC3=CC=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C(C(F)(F)F)=C4)N=C3)C(C)(C)C)C=C2)SC=N1	C67H72F3N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-UX8G69	WO2024027706A1_181	.	CC1=CC(OCCCC2=C(C(=O)O)N=C(N3CCC4=CC=CC(C(=O)NC5=NC6=C(C=CC=C6)S5)=C4C3)S2)=CC=C1C1=CC=C(CCCCCCCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)C=N1	C67H75N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-QRVQW8	WO2024027706A1_182	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC3=CC=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4Cl)N=C3)C(C)(C)C)C=C2)SC=N1	C66H72ClN9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-M1HX6I	WO2024027706A1_183	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC3=CC=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4C(F)(F)F)N=C3)C(C)(C)C)C=C2)SC=N1	C67H72F3N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-G7KBHH	WO2024027706A1_184	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC3=CN=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C(Cl)=C4)N=C3)C(C)(C)C)C=C2)SC=N1	C65H71ClN10O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-CZHIIH	WO2024027706A1_185	.	CC1=CC(C2=NC=C(CCCCCCCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](C)C3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)C=N2)=CC=C1OCCCC1=C(C(=O)O)N=C(N2CCC3=CC=CC(C(=O)NC4=NC5=C(C=CC=C5)S4)=C3C2)S1	C66H74N10O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-1MGTE7	WO2024027706A1_186	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC3=CN=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C(C(F)(F)F)=C4)N=C3)C(C)(C)C)C=C2)SC=N1	C66H71F3N10O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-B0ZH7T	WO2024027706A1_187	.	CC1=CC(OCCCC2=C(C(=O)O)N=C(N3CCC4=CC=CC(C(=O)NC5=NC6=C(C=CC=C6)S5)=C4C3)S2)=CC=C1C1=NC=C(CCCCCCCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)C=N1	C66H74N10O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-RYHW9E	WO2024027706A1_188	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC3=CN=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4Cl)N=C3)C(C)(C)C)C=C2)SC=N1	C65H71ClN10O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-PEN090	WO2024027706A1_189	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC3=CN=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4C(F)(F)F)N=C3)C(C)(C)C)C=C2)SC=N1	C66H71F3N10O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-73BXUX	WO2024027706A1_19	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCC(C4CC(C#CC5=CC=C(OCCCC6=C(C(=O)O)N=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=C(C=CC=C%10)S9)=C8C7)S6)C=C5)C4)CC3)C(C)(C)C)C=C2)SC=N1	C65H71N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-5V3WVQ	WO2024027706A1_190	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC#CC3=CC=C(OCCCC4=C(C(=O)O)N=C(N5CCC6=CC=CC(C(=O)NC7=NC8=C(C=CC=C8)S7)=C6C5)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C65H72N8O8S2	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-YEC3J9	WO2024027706A1_191	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCCC#CC3=CC=C(OCCCC4=C(C(=O)O)N=C(N5CCC6=CC=CC(C(=O)NC7=NC8=C(C=CC=C8)S7)=C6C5)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C66H74N8O8S2	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-JJACQC	WO2024027706A1_192	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC3=CC=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)C=C5)C=C4)N=C3)C(C)(C)C)C=C2)SC=N1	C68H75N9O8S2	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-FC4ERG	WO2024027706A1_193	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCOC3=CC=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)C=C5)C=C4)N=C3)C(C)(C)C)C=C2)SC=N1	C67H73N9O9S2	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-0ZH0M8	WO2024027706A1_194	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC3=NN=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)C=C5)C=C4)S3)C(C)(C)C)C=C2)SC=N1	C65H72N10O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-6LN5EN	WO2024027706A1_195	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC3=NC=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)C=C5)C=C4)N=C3)C(C)(C)C)C=C2)SC=N1	C67H74N10O8S2	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-QMYRSY	WO2024027706A1_196	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC3=CC=C(C4=NC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)C=C5)C=C4)N=C3)C(C)(C)C)C=C2)SC=N1	C67H74N10O8S2	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-2RPSKT	WO2024027706A1_197	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC3=CC=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)C=C5)C=C4)N=N3)C(C)(C)C)C=C2)SC=N1	C67H74N10O8S2	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-BM4506	WO2024027706A1_198	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC3=CC(F)=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)C=C5)C=C4)N=C3)C(C)(C)C)C=C2)SC=N1	C68H74FN9O8S2	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-T91UGM	WO2024027706A1_199	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC3=CC(Cl)=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)C=C5)C=C4)N=C3)C(C)(C)C)C=C2)SC=N1	C68H74ClN9O8S2	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-Z8TDDS	WO2024027706A1_2	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCOCC#CC3=CC=C(OCCCC4=C(C(=O)O)N=C(N5CCC6=CC=CC(C(=O)NC7=NC8=C(C=CC=C8)S7)=C6C5)S4)C=C3)C(C)(C)C)C=C2)SC=N1	C60H64N8O10S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-QGCA74	WO2024027706A1_20	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3CC(N4CCC(CC#CC5=CC=C(OCCCC6=C(C(=O)O)N=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=C(C=CC=C%10)S9)=C8C7)S6)C=C5)CC4)C3)C(C)(C)C)C=C2)SC=N1	C65H71N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-N1HXDJ	WO2024027706A1_200	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC3=CC(C(F)(F)F)=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)C=C5)C=C4)N=C3)C(C)(C)C)C=C2)SC=N1	C69H74F3N9O8S2	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-JAR56H	WO2024027706A1_201	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCCC3=CN=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)C=C5)C=C4)N=C3)C(C)(C)C)C=C2)SC=N1	C68H76N10O8S2	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-8NF7HX	WO2024027706A1_202	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCCC3=CC=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)C=C5)C=C4)N=C3)C(C)(C)C)C=C2)SC=N1	C69H77N9O8S2	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-T8UKPJ	WO2024027706A1_203	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC3=CC=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)C=C5)C=C4)N=C3F)C(C)(C)C)C=C2)SC=N1	C68H74FN9O8S2	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-D0OO0H	WO2024027706A1_204	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC3=CC=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)C=C5)C=C4)N=C3Cl)C(C)(C)C)C=C2)SC=N1	C68H74ClN9O8S2	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-QMHPPX	WO2024027706A1_205	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC3=CN=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)C=C5)C(Cl)=C4)N=C3)C(C)(C)C)C=C2)SC=N1	C67H73ClN10O8S2	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-O9Z73D	WO2024027706A1_207	.	CCC1=CC(C2=NC=C(CCCCCCCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](C)C3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)C=N2)=CC=C1OCCCC1=C(C(=O)O)N=C(N2CCC3=CC=CC(C(=O)NC4=NC5=C(C=CC=C5)S4)=C3C2)C=C1	C69H78N10O8S2	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-U2AHXC	WO2024027706A1_208	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC3=CN=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)C=C5)C(C(F)(F)F)=C4)N=C3)C(C)(C)C)C=C2)SC=N1	C68H73F3N10O8S2	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-L5KGJE	WO2024027706A1_209	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC3=CC(F)=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)C=C5)C(Cl)=C4)N=C3)C(C)(C)C)C=C2)SC=N1	C68H73ClFN9O8S2	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-3XY5ST	WO2024027706A1_21	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3CCC4(CC3)CCN(CC#CC3=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C3)CC4)C(C)(C)C)C=C2)SC=N1	C66H73N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-EDWVD2	WO2024027706A1_210	.	CC1=CC(C2=C(F)C=C(CCCCCCCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](C)C3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)C=N2)=CC=C1OCCCC1=C(C(=O)O)N=C(N2CCC3=CC=CC(C(=O)NC4=NC5=C(C=CC=C5)S4)=C3C2)C=C1	C69H76FN9O8S2	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-CGBBIZ	WO2024027706A1_211	.	CCC1=CC(C2=C(F)C=C(CCCCCCCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](C)C3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)C=N2)=CC=C1OCCCC1=C(C(=O)O)N=C(N2CCC3=CC=CC(C(=O)NC4=NC5=C(C=CC=C5)S4)=C3C2)C=C1	C70H78FN9O8S2	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-94QIOJ	WO2024027706A1_212	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC3=CC(F)=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)C=C5)C(C(F)(F)F)=C4)N=C3)C(C)(C)C)C=C2)SC=N1	C69H73F4N9O8S2	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-1LMT8R	WO2024027706A1_213	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC3=CC(Cl)=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)C=C5)C(Cl)=C4)N=C3)C(C)(C)C)C=C2)SC=N1	C68H73Cl2N9O8S2	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-RQI0PE	WO2024027706A1_214	.	CC1=CC(C2=C(Cl)C=C(CCCCCCCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](C)C3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)C=N2)=CC=C1OCCCC1=C(C(=O)O)N=C(N2CCC3=CC=CC(C(=O)NC4=NC5=C(C=CC=C5)S4)=C3C2)C=C1	C69H76ClN9O8S2	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-FXA0SH	WO2024027706A1_215	.	CCC1=CC(C2=C(Cl)C=C(CCCCCCCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](C)C3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)C=N2)=CC=C1OCCCC1=C(C(=O)O)N=C(N2CCC3=CC=CC(C(=O)NC4=NC5=C(C=CC=C5)S4)=C3C2)C=C1	C70H78ClN9O8S2	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-ZYYRNF	WO2024027706A1_216	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC3=CC(Cl)=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)C=C5)C(C(F)(F)F)=C4)N=C3)C(C)(C)C)C=C2)SC=N1	C69H73ClF3N9O8S2	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-HAFQGI	WO2024027706A1_217	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC3=CN=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)C=C5)C=C4Cl)N=C3)C(C)(C)C)C=C2)SC=N1	C67H73ClN10O8S2	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-VULJIJ	WO2024027706A1_218	.	CC1=CC(OCCCC2=C(C(=O)O)N=C(N3CCC4=CC=CC(C(=O)NC5=NC6=C(C=CC=C6)S5)=C4C3)C=C2)=CC=C1C1=NC=C(CCCCCCCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)C=N1	C68H76N10O8S2	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-1EU74V	WO2024027706A1_219	.	CCC1=CC(OCCCC2=C(C(=O)O)N=C(N3CCC4=CC=CC(C(=O)NC5=NC6=C(C=CC=C6)S5)=C4C3)C=C2)=CC=C1C1=NC=C(CCCCCCCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)C=N1	C69H78N10O8S2	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-P4A66B	WO2024027706A1_22	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCC4(CC3)CC(CC#CC3=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C3)C4)C(C)(C)C)C=C2)SC=N1	C65H71N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-FJS7GG	WO2024027706A1_220	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC3=CN=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)C=C5)C=C4C(F)(F)F)N=C3)C(C)(C)C)C=C2)SC=N1	C68H73F3N10O8S2	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-APAJKV	WO2024027706A1_221	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC3=CC(F)=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)C=C5)C=C4Cl)N=C3)C(C)(C)C)C=C2)SC=N1	C68H73ClFN9O8S2	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-OPMNPR	WO2024027706A1_222	.	CC1=CC(OCCCC2=C(C(=O)O)N=C(N3CCC4=CC=CC(C(=O)NC5=NC6=C(C=CC=C6)S5)=C4C3)C=C2)=CC=C1C1=C(F)C=C(CCCCCCCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)C=N1	C69H76FN9O8S2	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-4WOHT6	WO2024027706A1_223	.	CCC1=CC(OCCCC2=C(C(=O)O)N=C(N3CCC4=CC=CC(C(=O)NC5=NC6=C(C=CC=C6)S5)=C4C3)C=C2)=CC=C1C1=C(F)C=C(CCCCCCCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)C=N1	C70H78FN9O8S2	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-XGJ25M	WO2024027706A1_224	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC3=CC(F)=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)C=C5)C=C4C(F)(F)F)N=C3)C(C)(C)C)C=C2)SC=N1	C69H73F4N9O8S2	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-6F8B9D	WO2024027706A1_225	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC3=CC(Cl)=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)C=C5)C=C4Cl)N=C3)C(C)(C)C)C=C2)SC=N1	C68H73Cl2N9O8S2	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-3LW68T	WO2024027706A1_226	.	CC1=CC(OCCCC2=C(C(=O)O)N=C(N3CCC4=CC=CC(C(=O)NC5=NC6=C(C=CC=C6)S5)=C4C3)C=C2)=CC=C1C1=C(Cl)C=C(CCCCCCCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)C=N1	C69H76ClN9O8S2	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-X1P84I	WO2024027706A1_227	.	CCC1=CC(OCCCC2=C(C(=O)O)N=C(N3CCC4=CC=CC(C(=O)NC5=NC6=C(C=CC=C6)S5)=C4C3)C=C2)=CC=C1C1=C(Cl)C=C(CCCCCCCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)C=N1	C70H78ClN9O8S2	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-5HD899	WO2024027706A1_228	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC3=CC(Cl)=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)C=C5)C=C4C(F)(F)F)N=C3)C(C)(C)C)C=C2)SC=N1	C69H73ClF3N9O8S2	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-AL359A	WO2024027706A1_229	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC3=CN=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)C=C5)C=C4)N=C3)C(C)(C)C)C=C2)SC=N1	C67H74N10O8S2	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-2ABPE8	WO2024027706A1_23	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CC3CC4(CCN(CC#CC5=CC=C(OCCCC6=C(C(=O)O)N=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=C(C=CC=C%10)S9)=C8C7)S6)C=C5)CC4)C3)C(C)(C)C)C=C2)SC=N1	C65H71N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-94154U	WO2024027706A1_231	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CC3CCC4(CC3)CCN(CC#CC3=CC(Cl)=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C3)CC4)C(C)(C)C)C=C2)SC=N1	C68H76ClN9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-8QYT5B	WO2024027706A1_232	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCC(C)C3=CN=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)C(F)=C3)C(C)(C)C)C=C2)SC=N1	C66H72FN9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-IGAI5N	WO2024027706A1_233	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC3=CC(F)=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C(Cl)=C4)N=C3)C(C)(C)C)C=C2)SC=N1	C66H71ClFN9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-6LDI7F	WO2024027706A1_234	.	CC1=C(C2=C(F)C=C(CCCCCCCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](C)C3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)C=N2)C=CC(OCCCC2=C(C(=O)O)N=C(N3CCC4=CC=CC(C(=O)NC5=NC6=C(C=CC=C6)S5)=C4C3)S2)=C1	C67H74FN9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-89YHBN	WO2024027706A1_235	.	CC1=CC(OCCCC2=C(C(=O)O)N=C(N3CCC4=CC=CC(C(=O)NC5=NC6=C(C=CC=C6)S5)=C4C3)S2)=CC=C1C1=C(Cl)C=C(CCCCCCCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)C=N1	C67H74ClN9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-ZOH2L9	WO2024027706A1_236	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC3=CC(F)=C(C4=C(Cl)C=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)N=C3)C(C)(C)C)C=C2)SC=N1	C66H71ClFN9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-URJI7Z	WO2024027706A1_237	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC3=CN=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)C(F)=C3)C(C)(C)C)C=C2)SC=N1	C66H72FN9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-HQGKOY	WO2024027706A1_238	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC3=CC(Cl)=C(C4=C(Cl)C=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)N=C3)C(C)(C)C)C=C2)SC=N1	C66H71Cl2N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-ZS6IJA	WO2024027706A1_239	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCC(C)C3=CC=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)N=C3)C(C)(C)C)C=C2)SC=N1	C67H75N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-GSWTOG	WO2024027706A1_24	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3CC(CN4CC(C#CC5=CC=C(OCCCC6=C(C(=O)O)N=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=C(C=CC=C%10)S9)=C8C7)S6)C=C5)C4)C3)C(C)(C)C)C=C2)SC=N1	C63H67N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-GMEE3V	WO2024027706A1_240	.	CC1=CC(C2=NC=C(CCCCCCCCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](C)C3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)C=N2)=CC=C1OCCCC1=C(C(=O)O)N=C(N2CCC3=CC=CC(C(=O)NC4=NC5=C(C=CC=C5)S4)=C3C2)S1	C67H76N10O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-EMPC8G	WO2024027706A1_241	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCCC3=CN=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C(Cl)=C4)N=C3)C(C)(C)C)C=C2)SC=N1	C66H73ClN10O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-3PNGCJ	WO2024027706A1_242	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCCC3=CC=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)N=C3)C(C)(C)C)C=C2)SC=N1	C67H75N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-15W2YD	WO2024027706A1_243	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCCC3=CN=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)C(F)=C3)C(C)(C)C)C=C2)SC=N1	C67H74FN9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-IXD1RC	WO2024027706A1_244	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC3=CN=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C65H71N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-1JR2JU	WO2024027706A1_245	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC3=CN=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)C(F)=C3)C(C)(C)C)C=C2)SC=N1	C65H70FN9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-474TH1	WO2024027706A1_246	.	CC1=CC(C2=NC=C(CCCCCCCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCC3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)C=N2)=CC=C1OCCCC1=C(C(=O)O)N=C(N2CCC3=CC=CC(C(=O)NC4=NC5=C(C=CC=C5)S4)=C3C2)S1	C65H72N10O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-U6FVD7	WO2024027706A1_247	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC3=CN=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C(Cl)=C4)N=C3)C(C)(C)C)C=C2)SC=N1	C64H69ClN10O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-T58IQU	WO2024027706A1_248	.	CC1=CC(C2=NC=C(CCCCCCCCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCC3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)C=N2)=CC=C1OCCCC1=C(C(=O)O)N=C(N2CCC3=CC=CC(C(=O)NC4=NC5=C(C=CC=C5)S4)=C3C2)S1	C66H74N10O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-I843AR	WO2024027706A1_249	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCCC3=CN=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C(Cl)=C4)N=C3)C(C)(C)C)C=C2)SC=N1	C65H71ClN10O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-Q435TX	WO2024027706A1_25	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CC(CN4CC(C#CC5=CC=C(OCCCC6=C(C(=O)O)N=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=C(C=CC=C%10)S9)=C8C7)S6)C=C5)C4)C3)C(C)(C)C)C=C2)SC=N1	C63H68N10O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-05LD96	WO2024027706A1_250	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCCC3=CC=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)N=C3)C(C)(C)C)C=C2)SC=N1	C66H73N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-XIQ0IN	WO2024027706A1_251	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCCC3=CN=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)C(F)=C3)C(C)(C)C)C=C2)SC=N1	C66H72FN9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-W52F4J	WO2024027706A1_26	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CC3CC(N4CC(C#CC5=CC=C(OCCCC6=C(C(=O)O)N=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=C(C=CC=C%10)S9)=C8C7)S6)C=C5)C4)C3)C(C)(C)C)C=C2)SC=N1	C63H67N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-494N05	WO2024027706A1_27	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CC4(CCC(CC#CC5=CC=C(OCCCC6=C(C(=O)O)N=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=C(C=CC=C%10)S9)=C8C7)S6)C=C5)CC4)C3)C(C)(C)C)C=C2)SC=N1	C65H71N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-S3GZIN	WO2024027706A1_28	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC#CC3=CC=C(OCCCC4=C(C(=O)O)N=C(N5CCC6=CC=CC(C(=O)NC7=NC8=C(C=CC=C8)S7)=C6C5)S4)C=C3)C(C)(C)C)C=C2)SC=N1	C63H70N8O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-SJCZH2	WO2024027706A1_29	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3CCC(C4CCN(CC#CC5=CC=C(OCCCC6=C(C(=O)O)N=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=CC=CC=C%10S9)=C8C7)S6)C=C5)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C67H75N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-T7463Y	WO2024027706A1_3	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCOCC#CC3=CC=C(OCCCC4=C(C(=O)O)N=C(N5CCC6=CC=CC(C(=O)NC7=NC8=C(C=CC=C8)S7)=C6C5)S4)C=C3)C(C)(C)C)C=C2)SC=N1	C59H62N8O9S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-FRCWQD	WO2024027706A1_30	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCC4(CCC(C=CC5=CC=C(OCCCC6=C(C(=O)O)N=C(N7CCC8=C(C7)C(C(=O)NC7=NC9=CC=CC=C9S7)=CC=C8)S6)C=C5)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C66H75N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-W5NLVB	WO2024027706A1_31-A	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)[C@H]3CC[C@H](OCC#CC4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C63H68N8O9S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-12DA4P	WO2024027706A1_31-B	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)[C@H]3CC[C@@H](OCC#CC4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C63H68N8O9S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-SLNA6R	WO2024027706A1_31	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3CCC(OCC#CC4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C63H68N8O9S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-PZ083E	WO2024027706A1_33	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CC3CCC4(CC3)CN(CC#CC3=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C3)C4)C(C)(C)C)C=C2)SC=N1	C65H71N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-U5G8NQ	WO2024027706A1_34	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCOC3CCN(CC#CC4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C64H71N9O9S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-5NQTR6	WO2024027706A1_36	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCC#CC3=CC=C(OCCCC4=C(C(=O)O)N=C(N5CCC6=CC=CC(C(=O)NC7=NC8=C(C=CC=C8)S7)=C6C5)S4)C=C3)C(C)(C)C)C=C2)SC=N1	C62H68N8O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-1DWCZY	WO2024027706A1_37	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3CC(CC4CN(CC#CC5=CC=C(OCCCC6=C(C(=O)O)N=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=CC=CC=C%10S9)=C8C7)S6)C=C5)C4)C3)C(C)(C)C)C=C2)SC=N1	C64H69N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-VLNG4C	WO2024027706A1_38	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCC#CC3C=C(F)C(OCCCC4=C(C(=O)O)N=C(N5CCC6=CC=CC(C(=O)NC7=NC8=C(C=CC=C8)S7)=C6C5)S4)=CC3)C(C)(C)C)C=C2)SC=N1	C61H67FN8O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-8OYVI4	WO2024027706A1_39	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCC#CC3C=C(F)C(OCCCC4=C(C(=O)O)N=C(N5CCC6=CC=CC(C(=O)NC7=NC8=C(C=CC=C8)S7)=C6C5)S4)=CC3)C(C)(C)C)C=C2)SC=N1	C62H69FN8O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-W0WAW1	WO2024027706A1_4	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCOCC#CC3=CC=C(OCCCC4=C(C(=O)O)N=C(N5CCC6=CC=CC(C(=O)NC7=NC8=C(C=CC=C8)S7)=C6C5)S4)C=C3)C(C)(C)C)C=C2)SC=N1	C61H66N8O10S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-GL5XWQ	WO2024027706A1_40	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CC(N4CC(CC#CC5=CC=C(OCCCC6=C(C(=O)O)N=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=CC=CC=C%10S9)=C8C7)S6)C=C5)C4)C3)C(C)(C)C)C=C2)SC=N1	C63H68N10O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-XBU4JP	WO2024027706A1_41	.	CS/C(=N\C(=C\CCCOC1=CC=C(C#CCN2CCC(COCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](C)C3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)CC2)C=C1)C(=O)O)N1CCC2=CC=CC(C(=O)NC3=NC=CS3)=C2C1	C61H73N9O9S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-ZVEZHA	WO2024027706A1_42	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3CC4(CCN(CC#CC5=CC=C(OCCCC6=C(C(=O)O)N=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=C(C=CC=C%10)S9)=C8C7)S6)C=C5)CC4)C3)C(C)(C)C)C=C2)SC=N1	C65H71N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-QT9JGU	WO2024027706A1_43	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3CC4(CCN(CC#CC5=CC=C(OCCCC6=C(C(=O)O)N=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=C(C=CC=C%10)S9)=C8C7)S6)C=C5)CC4)C3)C(C)(C)C)C=C2)SC=N1	C64H69N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-4O9H1N	WO2024027706A1_44	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CC3CCC4(CC3)CCN(CC#CC3=CC(F)=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C3)CC4)C(C)(C)C)C=C2)SC=N1	C67H74FN9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-ZEK31F	WO2024027706A1_45	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CC3CCC4(CC3)CCN(CC#CC3=CC(F)=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C3)CC4)C(C)(C)C)C=C2)SC=N1	C68H76FN9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-PHOZEP	WO2024027706A1_46	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCC3=CN=C(C4=CC=C(OCCCC5=C(C(=O)O)NC(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)N=C3)C(C)(C)C)C=C2)SC=N1	C64H72N10O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-S2DNAO	WO2024027706A1_47	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3CCC4(CC3)CN(CC#CC3=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C3)C4)C(C)(C)C)C=C2)SC=N1	C65H71N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-CNP9K9	WO2024027706A1_48	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCC#CC3=CC=C(OCCCC4=C(C(=O)O)N=C(N5CCC6=CC=CC(C(=O)NC7=NC8=C(C=CC=C8)S7)=C6C5)S4)C=C3F)C(C)(C)C)C=C2)SC=N1	C61H65FN8O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-9V9IVK	WO2024027706A1_49	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCC#CC3=CC=C(OCCCC4=C(C(=O)O)N=C(N5CCC6=CC=CC(C(=O)NC7=NC8=C(C=CC=C8)S7)=C6C5)S4)C=C3F)C(C)(C)C)C=C2)SC=N1	C62H67FN8O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-XOJY8A	WO2024027706A1_5	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCCC#CC3=CC=C(OCCCC4=C(C(=O)O)N=C(N5CCC6=CC=CC(C(=O)NC7=NC8=C(C=CC=C8)S7)=C6C5)S4)C=C3)C(C)(C)C)C=C2)SC=N1	C61H66N8O9S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-AA7LBE	WO2024027706A1_50	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CC3CCC4(CC3)CCN(CC#CC3=CC(Cl)=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C3)CC4)C(C)(C)C)C=C2)SC=N1	C67H74ClN9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-QH1J7A	WO2024027706A1_51-A	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)[C@H]3CC[C@@H](OCCC#CC4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C64H70N8O9S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-OJ1LI6	WO2024027706A1_51-B	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)[C@H]3CC[C@H](OCCC#CC4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C64H70N8O9S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-QQ0G4V	WO2024027706A1_51	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3CCC(OCCC#CC4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C64H70N8O9S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-BDHPAI	WO2024027706A1_53	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3CCN(C4CCC(C#CC5=CC=C(OCCCC6=C(C(=O)O)N=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=C(C=CC=C%10)S9)=C8C7)S6)C=C5)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C66H73N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-JSS38D	WO2024027706A1_54	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CC(C4CC(C#CC5=CC=C(OCCCC6=C(C(=O)O)N=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=C(C=CC=C%10)S9)=C8C7)S6)C=C5)C4)C3)C(C)(C)C)C=C2)SC=N1	C63H67N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-EFF0MS	WO2024027706A1_55	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3CCN(C4CC(CC#CC5=CC=C(OCCCC6=C(C(=O)O)N=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=C(C=CC=C%10)S9)=C8C7)S6)C=C5)C4)CC3)C(C)(C)C)C=C2)SC=N1	C65H71N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-ZGOM8T	WO2024027706A1_56	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3CN(C4CCC(CC#CC5=CC=C(OCCCC6=C(C(=O)O)N=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=C(C=CC=C%10)S9)=C8C7)S6)C=C5)CC4)C3)C(C)(C)C)C=C2)SC=N1	C65H71N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-EJ88W1	WO2024027706A1_57	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CC3CN(C4CN(CC#CC5=CC=C(OCCCC6=C(C(=O)O)C=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=CC=CC=C%10S9)=C8C7)S6)C=C5)C4)C3)C(C)(C)C)C=C2)SC=N1	C64H69N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-4K1UEW	WO2024027706A1_58	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCC#CC3=CC=C(OCCCC4=C(C(=O)O)N=C(N5CCC6=CC=CC(C(=O)NC7=NC8=C(C=CC=C8)S7)=C6C5)S4)C=C3)C(C)(C)C)C=C2)SC=N1	C61H66N8O9S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-YH3K8P	WO2024027706A1_59	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCC#CC3=CC=C(OCCCC4=C(C(=O)O)N=C(N5CCC6=CC=CC(C(=O)NC7=NC8=C(C=CC=C8)S7)=C6C5)S4)C(Cl)=C3)C(C)(C)C)C=C2)SC=N1	C61H65ClN8O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-8DCH6B	WO2024027706A1_6	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCOCCOCC#CC3=CC=C(OCCCC4=C(C(=O)O)N=C(N5CCC6=CC=CC(C(=O)NC7=NC8=C(C=CC=C8)S7)=C6C5)S4)C=C3)C(C)(C)C)C=C2)SC=N1	C61H66N8O10S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-FT401L	WO2024027706A1_60	.	CC1=CC(C#CCCCCCCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)=CC=C1OCCCC1=C(C(=O)O)N=C(N2CCC3=CC=CC(C(=O)NC4=NC5=C(C=CC=C5)S4)=C3C2)S1	C62H68N8O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-Q3GLIM	WO2024027706A1_61	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCC#CC3=CC=C(OCCCC4=C(C(=O)O)N=C(N5CCC6=CC=CC(C(=O)NC7=NC8=C(C=CC=C8)S7)=C6C5)S4)C(C(F)(F)F)=C3)C(C)(C)C)C=C2)SC=N1	C62H65F3N8O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-QMD4O7	WO2024027706A1_62	.	CC1=C(OCCCC2=C(C(=O)O)N=C(N3CCC4=CC=CC(C(=O)NC5=NC6=C(C=CC=C6)S5)=C4C3)S2)C=CC(C#CCN2CCC3(CCC(CC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)NCC4=CC=C(C5=C(C)N=CS5)C=C4)C(C)(C)C)CC3)CC2)=C1	C68H77N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-5R1PYU	WO2024027706A1_63	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CC3CCC4(CC3)CCN(CC#CC3=CC(C(F)(F)F)=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C3)CC4)C(C)(C)C)C=C2)SC=N1	C68H74F3N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-IXVK7X	WO2024027706A1_64	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCN3C=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)N=N3)C(C)(C)C)C=C2)SC=N1	C61H67N11O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-AEACPG	WO2024027706A1_65	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCN3C=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)N=N3)C(C)(C)C)C=C2)SC=N1	C62H69N11O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-T5ICXV	WO2024027706A1_66	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCN3C=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)N=N3)C(C)(C)C)C=C2)SC=N1	C63H71N11O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-MFHRK5	WO2024027706A1_67	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCCN3C=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)N=N3)C(C)(C)C)C=C2)SC=N1	C64H73N11O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-KP0TQG	WO2024027706A1_68	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCON3C=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)N=N3)C(C)(C)C)C=C2)SC=N1	C62H69N11O9S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-RYJPUZ	WO2024027706A1_69	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCC3=CN(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)N=N3)C(C)(C)C)C=C2)SC=N1	C61H67N11O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-TDDBA0	WO2024027706A1_7	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCOCC#CC3=CC=C(OCCCC4=C(C(=O)O)N=C(N5CCC6=CC=CC(C(=O)NC7=NC8=C(C=CC=C8)S7)=C6C5)S4)C=C3)C(C)(C)C)C=C2)SC=N1	C61H66N8O9S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-NTIWFZ	WO2024027706A1_70	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCC3=CN(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)N=N3)C(C)(C)C)C=C2)SC=N1	C62H69N11O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-QQ0R6P	WO2024027706A1_71	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC3=CN(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)N=N3)C(C)(C)C)C=C2)SC=N1	C63H71N11O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-94Y3YS	WO2024027706A1_72	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCCC3=CN(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)N=N3)C(C)(C)C)C=C2)SC=N1	C64H73N11O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-49W3JZ	WO2024027706A1_73	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCC3=CC=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)N=C3)C(C)(C)C)C=C2)SC=N1	C65H71N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-DQ7X7T	WO2024027706A1_74	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC3=CC=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)N=C3)C(C)(C)C)C=C2)SC=N1	C66H73N9O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-0UNDSF	WO2024027706A1_75	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC3=CN=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)N=C3)C(C)(C)C)C=C2)SC=N1	C65H72N10O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-UZWQMH	WO2024027706A1_76	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCC(=O)N3CCN(CC#CC4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C64H70N10O9S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-P8I1TT	WO2024027706A1_77	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC#CC3=CC=C(OCCCC4=C(C(=O)O)N=C(N5CCC6=CC=CC(C(=O)NC7=NC8=C(C=CC=C8)S7)=C6C5)S4)C(F)=C3)C(C)(C)C)C=C2)SC=N1	C62H67FN8O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-4DBUPG	WO2024027706A1_78	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC#CC3=CC=C(OCCCC4=C(C(=O)O)N=C(N5CCC6=CC=CC(C(=O)NC7=NC8=C(C=CC=C8)S7)=C6C5)S4)C(F)=C3)C(C)(C)C)C=C2)SC=N1	C63H69FN8O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-LRT1Z6	WO2024027706A1_79	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC#CC3=CC=C(OCCCC4=C(C(=O)O)N=C(N5CCC6=CC=CC(C(=O)NC7=NC8=C(C=CC=C8)S7)=C6C5)S4)C=C3F)C(C)(C)C)C=C2)SC=N1	C63H69FN8O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-OFTA5Z	WO2024027706A1_8	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCOCCC#CC3=CC=C(OCCCC4=C(C(=O)O)N=C(N5CCC6=CC=CC(C(=O)NC7=NC8=C(C=CC=C8)S7)=C6C5)S4)C=C3)C(C)(C)C)C=C2)SC=N1	C61H66N8O9S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-UQC1LR	WO2024027706A1_80	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC#CC3=CC=C(OCCCC4=C(C(=O)O)N=C(N5CCC6=CC=CC(C(=O)NC7=NC8=C(C=CC=C8)S7)=C6C5)S4)C=C3F)C(C)(C)C)C=C2)SC=N1	C62H67FN8O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-M3E0PM	WO2024027706A1_81	.	CC1=C(C2=CC=C([C@H](CC(=O)NCCCCC#CC3=CC=C(OCCCC4=C(C(=O)O)N=C(N5CCC6=CC=CC(C(=O)NC7=NC8=C(C=CC=C8)S7)=C6C5)S4)C=C3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3(C#N)CC3)C(C)(C)C)C=C2)SC=N1	C65H68N10O9S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-9AT33V	WO2024027706A1_82	.	CC1=C(C2=CC=C([C@H](CC(=O)NCCCCC#CC3=CC=C(OCCCC4=C(C(=O)O)N=C(N5CCC6=CC=CC(C(=O)NC7=NC8=C(C=CC=C8)S7)=C6C5)S4)C=C3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3(F)CC3)C(C)(C)C)C=C2)SC=N1	C64H68FN9O9S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-QAPKRJ	WO2024027706A1_83	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCOC3=CN=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)N=C3)C(C)(C)C)C=C2)SC=N1	C62H66N10O10S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-HZXH3R	WO2024027706A1_84	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCOC3=CN=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C63H67N9O10S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-KUH1UK	WO2024027706A1_85	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCOC3=CN(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)N=C3)C(C)(C)C)C=C2)SC=N1	C60H64N10O10S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-SOMSYA	WO2024027706A1_86	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCN3C=C(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)C=N3)C(C)(C)C)C=C2)SC=N1	C61H66N10O9S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-OCULYF	WO2024027706A1_87	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCN3CCN(C4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C61H70N10O9S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-ZRWGLB	WO2024027706A1_88	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCN3CCN(C4=CC(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)=CC=C4)CC3)C(C)(C)C)C=C2)SC=N1	C62H72N10O9S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-8CVA3H	WO2024027706A1_89	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCN3CCOC(CCC#CC4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)C3)C(C)(C)C)C=C2)SC=N1	C63H69N9O9S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-0TGYUC	WO2024027706A1_9	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCCC#CC3=CC=C(OCCCC4=C(C(=O)O)N=C(C5CCC6=CC=CC(C(=O)NC7=NC8=C(C=CC=C8)S7)=C6C5)S4)C=C3)C(C)(C)C)C=C2)SC=N1	C61H65N7O9S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-MDT30J	WO2024027706A1_90	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCOC(CCC#CC4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)C3)C(C)(C)C)C=C2)SC=N1	C62H67N9O9S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-D40XF3	WO2024027706A1_91	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCOC(CCCC#CC4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)C3)C(C)(C)C)C=C2)SC=N1	C63H69N9O9S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-AX1S6O	WO2024027706A1_92	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCN3CCOC(CCCC#CC4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)C3)C(C)(C)C)C=C2)SC=N1	C64H71N9O9S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-30SOH1	WO2024027706A1_93	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCN(CCC#CC4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C62H68N10O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-Z6HMRW	WO2024027706A1_94	.	CC1=C(C2=CC=C(CNC(=O)C3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCN3CCN(CCC#CC4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C63H70N10O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-WBR2D3	WO2024027706A1_95	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCN3CC(N4CC(C#CC5=CC=C(OCCCC6=C(C(=O)O)N=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=C(C=CC=C%10)S9)=C8C7)S6)C=C5)C4)C3)C(C)(C)C)C=C2)SC=N1	C63H68N10O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-RV2L19	WO2024027706A1_96	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(CCCCCC#CC4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)=NO3)C(C)(C)C)C=C2)SC=N1	C63H66N8O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-WFB8CX	WO2024027706A1_97	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(CCCCC#CC4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)=NO3)C(C)(C)C)C=C2)SC=N1	C62H64N8O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-2MGXWM	WO2024027706A1_98	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(CCCCCC#CC4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)=NO3)C(C)C)C=C2)SC=N1	C62H64N8O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-5G8UIW	WO2024027706A1_99	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(CCCCC#CC4=CC=C(OCCCC5=C(C(=O)O)N=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)S5)C=C4)=NO3)C(C)C)C=C2)SC=N1	C61H62N8O8S3	BCL2L1	Q07817	VHL	WO-2024027706-A1
TPD-971IWP	WO2024027755A1_C001	.	Cc1cc(-c2cc3c(-c4cnn(C5CCN(C)CC5)c4)c[nH]c3nn2)cc(C)c1N1CCN(CCOCCOCCOCCOc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)CC1	C48H58N10O8	HPK1	Q92918	CRBN	WO-2024027755-A1
TPD-DY530J	WO2024027755A1_C002	.	Cc1cc(-c2cc3c(-c4cnn(C5CCN(C)CC5)c4)c[nH]c3nn2)cc(C)c1N1CCN(CCOCCOCCOCCOc2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)CC1	C48H58N10O8	HPK1	Q92918	CRBN	WO-2024027755-A1
TPD-8MR7DT	WO2024027755A1_C003	.	Cc1cc(-c2cc3c(-c4cnn(C5CCN(C)CC5)c4)c[nH]c3nn2)cc(C)c1N1CCN(C2CC3(CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)C2)CC1	C48H55N11O4	HPK1	Q92918	CRBN	WO-2024027755-A1
TPD-1J3OZW	WO2024027755A1_C004	.	Cc1cc(-c2cc3c(-c4cnn(C5CCN(C)CC5)c4)c[nH]c3nn2)cc(C)c1N1CCN(CC2CCN(C3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)CC2)CC1	C49H58N12O4	HPK1	Q92918	CRBN	WO-2024027755-A1
TPD-BVAKFO	WO2024027755A1_C005	.	Cc1cc(-c2cc3c(-c4cnn(C5CCN(C)CC5)c4)c[nH]c3nn2)cc(C)c1N1CCN(CC2CN(C3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)C2)CC1	C49H58N12O4	HPK1	Q92918	CRBN	WO-2024027755-A1
TPD-R9MMTH	WO2024027755A1_C006	.	Cc1cc(-c2cc3c(-c4cnn(C5CCN(C)CC5)c4)c[nH]c3nn2)cc(C)c1N1CCN(CCN2CCN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)CC1	C46H54N12O4	HPK1	Q92918	CRBN	WO-2024027755-A1
TPD-OKTH94	WO2024027755A1_C007	.	Cc1cc(-c2cc3c(-c4cnn(C5CCN(C)CC5)c4)c[nH]c3nn2)cc(C)c1N1CCN(CC2CN(C3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)C2)CC1	C47H54N12O4	HPK1	Q92918	CRBN	WO-2024027755-A1
TPD-0WJN2I	WO2024027755A1_C008	.	Cc1cc(-c2cc3c(-c4cnn(C5CCN(C)CC5)c4)c[nH]c3nn2)cc(C)c1N1CCN(CC2CN(C3CN(C4CN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)C3)C2)CC1	C50H59N13O4	HPK1	Q92918	CRBN	WO-2024027755-A1
TPD-SJF6QU	WO2024027755A1_C009	.	Cc1cc(-c2cc3c(-c4cnn(C5CCN(C)CC5)c4)c[nH]c3nn2)cc(C)c1N1CCN(CC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)CC1	C44H49N11O4	HPK1	Q92918	CRBN	WO-2024027755-A1
TPD-4P18FK	WO2024027755A1_C010	.	Cc1cc(-c2cc3c(-c4cnn(C5CCN(C)CC5)c4)c[nH]c3nn2)cc(C)c1N1CCN(CC2CCN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)CC1	C46H53N11O4	HPK1	Q92918	CRBN	WO-2024027755-A1
TPD-7RDFCS	WO2024027755A1_C011	.	Cc1cc(-c2cc3c(-c4cnn(C5CCN(C)CC5)c4)c[nH]c3nn2)cc(C)c1N1CCN(C2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)CC1	C43H47N11O4	HPK1	Q92918	CRBN	WO-2024027755-A1
TPD-FBBV2X	WO2024027755A1_C012	.	Cc1cc(-c2cc3c(-c4cnn(C5CCN(C)CC5)c4)c[nH]c3nn2)cc(C)c1N1CCN(CC2CCN(c3cc4c(cc3F)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)CC1	C46H52FN11O4	HPK1	Q92918	CRBN	WO-2024027755-A1
TPD-VFBRI1	WO2024027755A1_C013	.	COc1ccc(C(=O)N2CCC(CN3CCN(c4c(C)cc(-c5cc6c(-c7cnn(C8CCN(C)CC8)c7)c[nH]c6nn5)cc4C)CC3)CC2)cc1N1CCC(=O)NC1=O	C45H55N11O4	HPK1	Q92918	CRBN	WO-2024027755-A1
TPD-J9HHQA	WO2024027755A1_C014	.	Cc1cc(-c2cc3c(-c4cnn(C5CCN(C)CC5)c4)c[nH]c3nn2)cc(C)c1N1CCN(CCOc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)CC1	C42H46N10O5	HPK1	Q92918	CRBN	WO-2024027755-A1
TPD-LPMSM6	WO2024027755A1_C015	.	Cc1cc(C2=CC3C(c4cnn(C5CCN(C)CC5)c4)=CNC3N=N2)cc(C)c1N1CCN(C2CC3(C2)CN(c2ccc4c(c2)C(=O)N(C2CCC(=O)NC2=O)C4=O)C3)CC1	C46H53N11O4	HPK1	Q92918	CRBN	WO-2024027755-A1
TPD-16DWO3	WO2024027755A1_C016	.	Cc1cc(-c2cc3c(-c4cnn(C5CCN(C)CC5)c4)c[nH]c3nn2)cc(C)c1N1CCN(CC2CCN(C(=O)c3ccc(N4CCC(=O)NC4=O)cc3)CC2)CC1	C44H53N11O3	HPK1	Q92918	CRBN	WO-2024027755-A1
TPD-11CH3I	WO2024027755A1_C017	.	Cc1cc(-c2cc3c(-c4cnn(C5CCN(C)CC5)c4)c[nH]c3nn2)cc(C)c1N1CCN(CCCOc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)CC1	C43H48N10O5	HPK1	Q92918	CRBN	WO-2024027755-A1
TPD-TNAPZX	WO2024027755A1_C018	.	Cc1cc(-c2cc3c(-c4cnn(C5CCN(C)CC5)c4)c[nH]c3nn2)cc(C)c1N1CCN(CCOCCOc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)CC1	C44H50N10O6	HPK1	Q92918	CRBN	WO-2024027755-A1
TPD-B81J59	WO2024027755A1_C019	.	Cc1cc(-c2cc3c(-c4cnn(C5CCN(C)CC5)c4)c[nH]c3nn2)cc(C)c1N1CCN(CCOCCOCCOc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)CC1	C46H54N10O7	HPK1	Q92918	CRBN	WO-2024027755-A1
TPD-KQET2A	WO2024027755A1_C020	.	Cc1cc(-c2cc3c(-c4cnn(C5CCN(C)CC5)c4)c[nH]c3nn2)cc(C)c1N1CCN(CCOCCOCCOCCNc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)CC1	C48H59N11O7	HPK1	Q92918	CRBN	WO-2024027755-A1
TPD-BP1EL0	WO2024027755A1_C021	.	Cc1cc(-c2cc3c(-c4cnn(C5CCN(C)CC5)c4)c[nH]c3nn2)cc(C)c1N1CCN(C2CC3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3C2)CC1	C47H53N11O4	HPK1	Q92918	CRBN	WO-2024027755-A1
TPD-WKTYO3	WO2024027755A1_C022	.	Cc1cc(-c2cc3c(-c4cnn(C5CCN(C)CC5)c4)c[nH]c3nn2)cc(C)c1N1CCN(CC2CCN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)CC1	C45H51N11O4	HPK1	Q92918	CRBN	WO-2024027755-A1
TPD-G8ZN2X	WO2024027755A1_C023	.	Cc1cc(-c2cc3c(-c4cnn(C5CCN(C)CC5)c4)c[nH]c3nn2)cc(C)c1N1CCN(C2CCC(Nc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)CC1	C46H53N11O4	HPK1	Q92918	CRBN	WO-2024027755-A1
TPD-P4RRID	WO2024027755A1_C024	.	Cc1cc(-c2cc3c(-c4cnn(C5CCN(C)CC5)c4)c[nH]c3nn2)cc(C)c1N1CCN(CCCNc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)CC1	C43H49N11O4	HPK1	Q92918	CRBN	WO-2024027755-A1
TPD-MS3LJ7	WO2024027755A1_C025	.	Cc1cc(-c2cc3c(-c4cnn(C5CCN(C)CC5)c4)c[nH]c3nn2)cc(C)c1N1CCN(CCCCNc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)CC1	C44H51N11O4	HPK1	Q92918	CRBN	WO-2024027755-A1
TPD-IA2H70	WO2024027755A1_C026	.	Cc1cc(-c2cc3c(-c4cnn(C5CCN(C)CC5)c4)c[nH]c3nn2)cc(C)c1N1CCN(CC2CCN(C(=O)c3ccc(F)c(N4CCC(=O)NC4=O)c3)CC2)CC1	C44H52FN11O3	HPK1	Q92918	CRBN	WO-2024027755-A1
TPD-ZGZFOK	WO2024027755A1_C027	.	Cc1cc(F)c(C(=O)N2CCC(CN3CCN(c4c(C)cc(-c5cc6c(-c7cnn(C8CCN(C)CC8)c7)c[nH]c6nn5)cc4C)CC3)CC2)cc1N1CCC(=O)NC1=O	C45H54FN11O3	HPK1	Q92918	CRBN	WO-2024027755-A1
TPD-IFUDIP	WO2024027755A1_C028	.	Cc1cc(C2=CC3C(c4cnn(C5CCN(C)CC5)c4)=CNC3N=N2)cc(C)c1N1CCN(CC2CCN(C(=O)c3ccc(Cl)c(N4CCC(=O)NC4=O)c3)CC2)CC1	C44H54ClN11O3	HPK1	Q92918	CRBN	WO-2024027755-A1
TPD-OS2YRI	WO2024027755A1_C029	.	Cc1cc(-c2cc3c(-c4cnn(C5CCN(C)CC5)c4)c[nH]c3nn2)cc(C)c1N1CCN(CC2CCN(C(=O)c3cccc(N4CCC(=O)NC4=O)c3)CC2)CC1	C44H53N11O3	HPK1	Q92918	CRBN	WO-2024027755-A1
TPD-YI3XYL	WO2024027755A1_C030	.	Cc1cc(-c2cc3c(-c4cnn(C5CCN(C)CC5)c4)c[nH]c3nn2)cc(C)c1N1CCN(C(=O)c2ccc(N3CCC(=O)NC3=O)cc2)CC1	C38H42N10O3	HPK1	Q92918	CRBN	WO-2024027755-A1
TPD-XA6NLW	WO2024027755A1_C031	.	Cc1cc(-c2cc3c(-c4cnn(C5CCN(C)CC5)c4)c[nH]c3nn2)cc(C)c1N1CCN(C2CC(Oc3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)CC1	C44H48N10O5	HPK1	Q92918	CRBN	WO-2024027755-A1
TPD-QA6CVW	WO2024027755A1_C032	.	COc1ccc(C(=O)N2CCN(c3c(C)cc(-c4cc5c(-c6cnn(C7CCN(C)CC7)c6)c[nH]c5nn4)cc3C)CC2)cc1N1CCC(=O)NC1=O	C39H44N10O4	HPK1	Q92918	CRBN	WO-2024027755-A1
TPD-TXQ62Q	WO2024027755A1_C035	.	Cc1cc(-c2cc3c(-c4cnn(C5CCN(C)CC5)c4)c[nH]c3nn2)cc(C)c1N1CCN(C2CCC(Oc3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)CC1	C46H52N10O5	HPK1	Q92918	CRBN	WO-2024027755-A1
TPD-5JKQX3	WO2024027755A1_C036	.	Cc1cc(-c2cc3c(-c4cnn(C5CCN(C)CC5)c4)c[nH]c3nn2)cc(C)c1N1CCN(C2CC(Nc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)CC1	C44H49N11O4	HPK1	Q92918	CRBN	WO-2024027755-A1
TPD-TY5Z3G	WO2024027755A1_C037	.	COc1ccc(C(=O)N2CCC(N3CC(CN4CCN(c5c(C)cc(-c6cc7c(-c8cnn(C9CCN(C)CC9)c8)c[nH]c7nn6)cc5C)CC4)C3)CC2)cc1N1CCC(=O)NC1=O	C48H60N12O4	HPK1	Q92918	CRBN	WO-2024027755-A1
TPD-2PTTTW	WO2024027755A1_C038	.	Cc1cc(-c2cc3c(-c4cnn(C5CCN(C)CC5)c4)c[nH]c3nn2)cc(C)c1N1CCN(CC2CCN(C(=O)c3cc(N4CCC(=O)NC4=O)ccc3F)CC2)CC1	C44H52FN11O3	HPK1	Q92918	CRBN	WO-2024027755-A1
TPD-BZS97J	WO2024027755A1_C039	.	Cc1cc(-c2cc3c(-c4cnn(C5CCN(C)CC5)c4)c[nH]c3nn2)cc(C)c1N1CCN(C2CC(NC(=O)c3ccc(N4CCC(=O)NC4=O)cc3)C2)CC1	C42H49N11O3	HPK1	Q92918	CRBN	WO-2024027755-A1
TPD-BTSCA6	WO2024027755A1_C040	.	Cc1cc(-c2cc3c(-c4cnn(C5CCN(C)CC5)c4)c[nH]c3nn2)cc(C)c1N1CCN(C2CCC(=O)NC2=O)CC1	C32H39N9O2	HPK1	Q92918	CRBN	WO-2024027755-A1
TPD-EVUFW7	WO2024027755A1_C041	.	Cc1cc(-c2cc3c(-c4cnn(C5CCN(C)CC5)c4)c[nH]c3nn2)cc(C)c1N1CCN(CC2CN(C3CCN(C(=O)c4ccc(N5CCC(=O)NC5=O)cc4)CC3)C2)CC1	C47H58N12O3	HPK1	Q92918	CRBN	WO-2024027755-A1
TPD-A8YKRR	WO2024027755A1_C042	.	Cc1cc(-c2cc3c(-c4cnn(C5CCN(C)CC5)c4)c[nH]c3nn2)cc(C)c1N1CCN(c2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)CC1	C40H42N10O4	HPK1	Q92918	CRBN	WO-2024027755-A1
TPD-4MZPK5	WO2024027755A1_C043	.	Cc1cc(-c2cc3c(-c4cnn(C5CCN(C)CC5)c4)c[nH]c3nn2)cc(C)c1N1CCN(c2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)CC1	C40H42N10O4	HPK1	Q92918	CRBN	WO-2024027755-A1
TPD-NHE4WZ	WO2024027755A1_C044	.	Cc1cc(-c2cc3c(-c4cnn(C5CCN(C)CC5)c4)c[nH]c3nn2)cc(C)c1N1CCN(CCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCc2ccc(-c3scnc3C)cc2)C(C)(C)C)CC1	C52H66N12O4S	HPK1	Q92918	VHL	WO-2024027755-A1
TPD-ZP2VGA	WO2024027755A1_C045	.	Cc1cc(-c2cc3c(-c4cnn(C5CCN(C)CC5)c4)c[nH]c3nn2)cc(C)c1N1CCN(CCCCCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCc2ccc(-c3scnc3C)cc2)C(C)(C)C)CC1	C55H72N12O4S	HPK1	Q92918	VHL	WO-2024027755-A1
TPD-7ARIXJ	WO2024027755A1_C046	.	Cc1cc(-c2cc3c(-c4cnn(C5CCN(C)CC5)c4)c[nH]c3nn2)cc(C)c1N1CCN(CC2CN(C(=O)c3cccc(N4CCC(=O)NC4=O)c3)C2)CC1	C42H49N11O3	HPK1	Q92918	CRBN	WO-2024027755-A1
TPD-JV59W1	WO2024027755A1_C047	.	Cc1cc(-c2cc3c(-c4cnn(C5CCN(C)CC5)c4)c[nH]c3nn2)cc(C)c1N1CCN(C2CC(NC(=O)c3cccc(N4CCC(=O)NC4=O)c3)C2)CC1	C42H49N11O3	HPK1	Q92918	CRBN	WO-2024027755-A1
TPD-VVEM8B	WO2024027755A1_C048	.	Cc1cc(-c2cc3c(-c4cnn(C5CCN(C)CC5)c4)c[nH]c3nn2)cc(C)c1N1CCN(C(=O)c2cc(Cl)cc(N3CCC(=O)NC3=O)c2)CC1	C38H41ClN10O3	HPK1	Q92918	CRBN	WO-2024027755-A1
TPD-WWTSAV	WO2024027755A1_C049	.	Cc1cc(-c2cc3c(-c4cnn(C5CCN(C)CC5)c4)c[nH]c3nn2)cc(C)c1N1CCN(C2CC3(CCN(c4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)C2)CC1	C48H55N11O4	HPK1	Q92918	CRBN	WO-2024027755-A1
TPD-83EB49	WO2024027755A1_C050	.	Cc1cc(-c2cc3c(-c4cnn(C5CCN(C)CC5)c4)c[nH]c3nn2)cc(C)c1N1CCN(C2CC(NC(=O)c3cc(N4CCC(=O)NC4=O)ccc3Cl)C2)CC1	C42H48ClN11O3	HPK1	Q92918	CRBN	WO-2024027755-A1
TPD-8YH8IC	WO2024027755A1_C051	.	COc1cc(C(=O)N2CCN(c3c(C)cc(-c4cc5c(-c6cnn(C7CCN(C)CC7)c6)c[nH]c5nn4)cc3C)CC2)cc(N2CCC(=O)NC2=O)c1	C39H44N10O4	HPK1	Q92918	CRBN	WO-2024027755-A1
TPD-T5GEQ0	WO2024032529A1_1	.	O=C(CCCCCCCCCCCCCCc1nc2ccc(N3CCN(C(=O)c4cc(Cc5n[nH]c(=O)c6ccccc56)ccc4F)CC3)nc2[nH]1)NCCNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O	C56H64FN11O7	PARP1	P09874	CRBN	WO-2024032529-A1
TPD-9EKMBR	WO2024032529A1_2	.	O=C(CCCCCCCCCCCCCc1nc2ccc(N3CCN(C(=O)c4cc(Cc5n[nH]c(=O)c6ccccc56)ccc4F)CC3)nc2[nH]1)NCCNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O	C55H62FN11O7	PARP1	P09874	CRBN	WO-2024032529-A1
TPD-G4PQAS	WO2024032529A1_3	.	O=C(CCCCCCCCCCCCc1nc2ccc(N3CCN(C(=O)c4cc(Cc5n[nH]c(=O)c6ccccc56)ccc4F)CC3)nc2[nH]1)NCCNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O	C54H60FN11O7	PARP1	P09874	CRBN	WO-2024032529-A1
TPD-L55472	WO2024032529A1_4	.	O=C(CCCCCCCCCCCc1nc2ccc(N3CCN(C(=O)c4cc(Cc5n[nH]c(=O)c6ccccc56)ccc4F)CC3)nc2[nH]1)NCCNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O	C53H58FN11O7	PARP1	P09874	CRBN	WO-2024032529-A1
TPD-INIARF	WO2024032529A1_5	.	O=C(CCCCCCCCCCc1nc2ccc(N3CCN(C(=O)c4cc(Cc5n[nH]c(=O)c6ccccc56)ccc4F)CC3)nc2[nH]1)NCCNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O	C52H56FN11O7	PARP1	P09874	CRBN	WO-2024032529-A1
TPD-5G6AE3	WO2024032529A1_6	.	O=C(CCCCCCCCCc1nc2ccc(N3CCN(C(=O)c4cc(Cc5n[nH]c(=O)c6ccccc56)ccc4F)CC3)nc2[nH]1)NCCNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O	C51H54FN11O7	PARP1	P09874	CRBN	WO-2024032529-A1
TPD-XKP2BH	WO2024032529A1_7	.	O=C(CCCCCCCCc1nc2ccc(N3CCN(C(=O)c4cc(Cc5n[nH]c(=O)c6ccccc56)ccc4F)CC3)nc2[nH]1)NCCNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O	C50H52FN11O7	PARP1	P09874	CRBN	WO-2024032529-A1
TPD-A9P1X2	WO2024032529A1_8	.	O=C(CCCCCCCCCCCc1nc2ccc(N3CCN(C(=O)c4cc(Cc5n[nH]c(=O)c6ccccc56)ccc4F)CC3)nc2[nH]1)NCCOc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O	C53H57FN10O8	PARP1	P09874	CRBN	WO-2024032529-A1
TPD-48D0MW	WO2024032529A1_9	.	O=C1CCC(N2C(=O)c3cccc(N4CCN(C(=O)CCCCCCCCCCCc5nc6ccc(N7CCN(C(=O)c8cc(Cc9n[nH]c(=O)c%10ccccc9%10)ccc8F)CC7)nc6[nH]5)CC4)c3C2=O)C(=O)N1	C55H60FN11O7	PARP1	P09874	CRBN	WO-2024032529-A1
TPD-ECN4PG	WO2024032529A1_10	.	O=C(CN1CC2CN(CCCCCCc3nc4ccc(N5CCN(C(=O)c6cc(Cc7n[nH]c(=O)c8ccccc78)ccc6F)CC5)nc4[nH]3)CC2C1)NCCNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O	C55H60FN13O7	PARP1	P09874	CRBN	WO-2024032529-A1
TPD-9UIYUG	WO2024032529A1_11	.	O=C(CN1CCN(CCCCCCCc2nc3ccc(N4CCN(C(=O)c5cc(Cc6n[nH]c(=O)c7ccccc67)ccc5F)CC4)nc3[nH]2)CC1)NCCNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O	C54H60FN13O7	PARP1	P09874	CRBN	WO-2024032529-A1
TPD-AO8K5M	WO2024032529A1_12	.	O=C1CCC(N2C(=O)c3cccc(NCCOCCN4CCN(C(=O)C5CCN(CCCc6nc7ccc(N8CCN(C(=O)c9cc(Cc%10n[nH]c(=O)c%11ccccc%10%11)ccc9F)CC8)nc7[nH]6)CC5)CC4)c3C2=O)C(=O)N1	C56H62FN13O8	PARP1	P09874	CRBN	WO-2024032529-A1
TPD-0U3R9R	WO2024032529A1_13	.	O=C1CCC(N2C(=O)c3cccc(NCCC(=O)N4CCC(Cc5ccc(CNCCc6nc7ccc(N8CCN(C(=O)c9cc(Cc%10n[nH]c(=O)c%11ccccc%10%11)ccc9F)CC8)nc7[nH]6)cc5)CC4)c3C2=O)C(=O)N1	C57H57FN12O7	PARP1	P09874	CRBN	WO-2024032529-A1
TPD-HWXGHY	WO2024032529A1_14	.	O=C1CCC(N2C(=O)c3cccc(NCCNC(=O)c4cnc(N5CCC6(CCN(Cc7nc8ccc(N9CCN(C(=O)c%10cc(Cc%11n[nH]c(=O)c%12ccccc%11%12)ccc%10F)CC9)nc8[nH]7)CC6)CC5)nc4)c3C2=O)C(=O)N1	C56H56FN15O7	PARP1	P09874	CRBN	WO-2024032529-A1
TPD-PT1KNC	WO2024032529A1_15	.	O=C(CCCCCCCCCCCCOc1cc(N2CCN(C(=O)c3cc(Cc4n[nH]c(=O)c5ccccc45)ccc3F)CC2)nc2[nH]cnc12)NCCNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O	C54H60FN11O8	PARP1	P09874	CRBN	WO-2024032529-A1
TPD-0WLC0D	WO2024032600A1_1	.	COc1cc(N2CCC(CN3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)c(-c2cnn(C)c2)cc1Nc1ncc(Br)c(Nc2ccc(C(F)(F)F)cc2P(C)(C)=O)n1	C47H50BrF3N11O6P	EGFR	P00533	CRBN	WO-2024032600-A1
TPD-H9PXTS	WO2024032600A1_2	.	COc1cc(N2CCC(CN3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)c(-c2cnn(C)c2)cc1Nc1ncc(Cl)c(Nc2ccc(C(F)(F)F)cc2P(C)(C)=O)n1	C47H50ClF3N11O6P	EGFR	P00533	CRBN	WO-2024032600-A1
TPD-A98MZC	WO2024032600A1_3	.	COc1cc(N2CCC(CN3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)c(-c2cnn(C)c2)cc1Nc1ncc(Br)c(Nc2ccc(C3CC(F)(F)C3)cc2P(C)(C)=O)n1	C50H55BrF2N11O6P	EGFR	P00533	CRBN	WO-2024032600-A1
TPD-CQ7Y7V	WO2024032600A1_4	.	COc1cc(N2CCC(CN3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)c(-c2cnn(C)c2)cc1Nc1ncc(Cl)c(Nc2ccc(C3CC(F)(F)C3)cc2P(C)(C)=O)n1	C50H55ClF2N11O6P	EGFR	P00533	CRBN	WO-2024032600-A1
TPD-ZSFSZN	WO2024032600A1_5	.	Cn1cc(-c2cc(Nc3ncc(Br)c(Nc4ccc(C5CC5)cc4P(C)(C)=O)n3)c(OC(F)F)cc2N2CCC(CN3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)cn1	C49H53BrF2N11O6P	EGFR	P00533	CRBN	WO-2024032600-A1
TPD-QEW3C7	WO2024032600A1_6	.	CCn1cc(-c2cc(Nc3ncc(Cl)c(Nc4ccc(C5CC5)cc4P(C)(C)=O)n3)c(OC(F)F)cc2N2CCC(CN3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)cn1	C50H55ClF2N11O6P	EGFR	P00533	CRBN	WO-2024032600-A1
TPD-607IVX	WO2024032600A1_7	.	COc1cc(N2CCC(F)(CN3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)c(-c2cnn(C)c2)cc1Nc1ncc(Cl)c(Nc2ccc(C3CC3)cc2P(C)(C)=O)n1	C49H54ClFN11O6P	EGFR	P00533	CRBN	WO-2024032600-A1
TPD-6JQSZM	WO2024032600A1_8	.	COc1cc(N2CCC(F)(CN3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)c(-c2cnn(C)c2)cc1Nc1ncc(Br)c(Nc2ccc(F)cc2P(C)(C)=O)n1	C46H49BrF2N11O6P	EGFR	P00533	CRBN	WO-2024032600-A1
TPD-71IP1W	WO2024032600A1_9	.	COc1cc(N2CCC(F)(CN3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)c(-c2cnn(C)c2)cc1Nc1ncc(Cl)c(Nc2ccc(F)cc2P(C)(C)=O)n1	C46H49ClF2N11O6P	EGFR	P00533	CRBN	WO-2024032600-A1
TPD-7662BG	WO2024034593A1_1	.	CO[C@@H](C)COC1=NC2=C(OCC3=CC=C(C(=O)N4CCN(CC5=CC=C6C(=C5)N(C)C(=O)N6C5CCC(=O)NC5=O)C[C@@H]4C)C=C3)C(C3=C(C)C(F)=CC4=C3C=NN4)=C(C3CC3)C=C2C(OC2CN(C(=O)NCCN(C)C)C2)=N1	C58H67FN12O9	KRAS	P01116	CRBN	WO-2024034593-A1
TPD-GIRHV3	SCHEMBL30774981	1-[6-cyclopropyl-8-[[4-[(2S)-4-[[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]methyl]-2-methylpiperazine-1-carbonyl]phenyl]methoxy]-7-(6-fluoro-5-methyl-1H-indazol-4-yl)-2-[(2S)-2-methoxypropoxy]quinazolin-4-yl]azetidine-3-carbonitrile	CO[C@@H](C)COC1=NC2=C(OCC3=CC=C(C(=O)N4CCN(CC5=CC=C6C(=C5)N(C)C(=O)N6C5CCC(=O)NC5=O)C[C@@H]4C)C=C3)C(C3=C(C)C(F)=CC4=C3C=NN4)=C(C3CC3)C=C2C(N2CC(C#N)C2)=N1	C54H56FN11O7	KRAS	P01116	CRBN	WO-2024034593-A1
TPD-V7CM1G	SCHEMBL30774955	3-[5-[[(3S)-4-[4-[[4-[(3S,4R)-4-amino-3-fluoropiperidin-1-yl]-6-cyclopropyl-7-(6-fluoro-5-methyl-1H-indazol-4-yl)-2-[(2S)-2-methoxypropoxy]quinazolin-8-yl]oxymethyl]benzoyl]-3-methylpiperazin-1-yl]methyl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	CO[C@@H](C)COC1=NC2=C(OCC3=CC=C(C(=O)N4CCN(CC5=CC=C6C(=C5)N(C)C(=O)N6C5CCC(=O)NC5=O)C[C@@H]4C)C=C3)C(C3=C(C)C(F)=CC4=C3C=NN4)=C(C3CC3)C=C2C(N2CC[C@@H](N)[C@@H](F)C2)=N1	C55H61F2N11O7	KRAS	P01116	CRBN	WO-2024034593-A1
TPD-AKRE9J	WO2024034593A1_4	.	CO[C@@H](C)COC1=NC2=C(OCC3=CC=C(C(=O)N4CCN(CC5=CC=C6C(=C5)N(C)C(=O)N6C5CCC(=O)NC5=O)C[C@@H]4C)C=C3)C(C3=C(C)C(F)=CC4=C3C=NN4)=C(C3CC3)C=C2C(NCC2=CN=CC=C2)=N1	C56H58FN11O7	KRAS	P01116	CRBN	WO-2024034593-A1
TPD-WZ602Z	SCHEMBL31622461	(2S)-1-[6-cyclopropyl-8-[[4-[(2S)-4-[[3-(2,4-dioxo-1,3-diazinan-1-yl)-1-methylindazol-6-yl]methyl]-2-methylpiperazine-1-carbonyl]phenyl]methoxy]-7-(6-fluoro-5-methyl-1H-indazol-4-yl)-2-[(2S)-2-methoxypropoxy]quinazolin-4-yl]azetidine-2-carboxamide	CO[C@@H](C)COC1=NC2=C(C=C(C3CC3)C(C3=C(C)C(F)=CC4=C3C=NN4)=C2OCC2=CC=C(C(=O)N3CCN(CC4=CC5=C(C=C4)C(N4CCC(=O)NC4=O)=NN5C)C[C@@H]3C)C=C2)C(N2CC[C@H]2C(N)=O)=N1	C53H57FN12O7	KRAS	P01116	CRBN	WO-2024034593-A1
TPD-QM0YY7	WO2024034593A1_6	.	CC1=C(C2=C(C3CC3)C=C3C(N4CC[C@H]4C(N)=O)=NC(OCC(C)(C)CN(C)C)=NC3=C2OCC2=CC=C(C(=O)N3CCN(CC4=CC=C5C(=C4)N(C)C(=O)N5C4CCC(=O)NC4=O)C[C@@H]3C)C=C2)C2=C(C=C1F)NN=C2	C57H65FN12O7	KRAS	P01116	CRBN	WO-2024034593-A1
TPD-RH5RU7	WO2024034593A1_7	.	CC1=C(C2=C(C3CC3)C=C3C(N4CC[C@H]4C(N)=O)=NC(OC[C@@H]4CCN(C)C4)=NC3=C2OCC2=CC=C(C(=O)N3CCN(CC4=CC=C5C(=C4)N(C)N=C5N4CCC(=O)NC4=O)C[C@@H]3C)C=C2)C2=C(C=C1F)NN=C2	C55H60FN13O6	KRAS	P01116	CRBN	WO-2024034593-A1
TPD-FJRQU1	WO2024034593A1_8	.	CC1=C(C2=C(C3CC3)C=C3C(NC4CN(C5=NC=CC=N5)C4)=NC(OCC(C)(C)CN(C)C)=NC3=C2OCC2=CC=C(C(=O)N3CCN(CC4=CC=C5C(=C4)N(C)C(=O)N5C4CCC(=O)NC4=O)C[C@@H]3C)C=C2)C2=C(C=C1F)NN=C2	C60H67FN14O6	KRAS	P01116	CRBN	WO-2024034593-A1
TPD-KLUID1	WO2024034593A1_9	.	CC1=C(C2=C(C3CC3)C=C3C(N4CCOCC4)=NC(OCC(C)(C)CN(C)C)=NC3=C2OCC2=CC=C(C(=O)N3CCN(CC4=CC=C5C(=C4)N(C)C(=O)N5C4CCC(=O)NC4=O)C[C@@H]3C)C=C2)C2=C(C=C1F)NN=C2	C57H66FN11O7	KRAS	P01116	CRBN	WO-2024034593-A1
TPD-9VTWWV	WO2024034593A1_10	.	CC1=C(C2=C(C3CC3)C=C3C(N4CC(C#N)C4)=NC(OCC(C)(C)CN(C)C)=NC3=C2OCC2=CC=C(C(=O)N3CCN(CC4=CC=C5C(=C4)N(C)C(=O)N5C4CCC(=O)NC4=O)C[C@@H]3C)C=C2)C2=C(C=C1F)NN=C2	C57H63FN12O6	KRAS	P01116	CRBN	WO-2024034593-A1
TPD-VFPYPP	WO2024034593A1_11	.	CC1=C(C2=C(C3CC3)C=C3C(N4CC(C#N)C4)=NC(OCC(C)(C)CN(C)C)=NC3=C2OCC2=CC=C(C(=O)N3CCN(CC4=CC=C5C(=C4)N(C)N=C5N4CCC(=O)NC4=O)C[C@@H]3C)C=C2)C2=C(C=C1F)NN=C2	C56H62FN13O5	KRAS	P01116	CRBN	WO-2024034593-A1
TPD-9WV5LZ	WO2024034593A1_12	.	CO[C@@H](C)COC1=NC2=C(OCC3=CC=C(C(=O)N4CCN(CC5=CC=C6C(=C5)N(C)N=C6N5CCC(=O)NC5=O)CC4)C=C3)C(C3=C(C)C(F)=CC4=C3C=NN4)=C(C3CC3)C=C2C(N2CC(C#N)C2)=N1	C52H53FN12O6	KRAS	P01116	CRBN	WO-2024034593-A1
TPD-MPW2ZF	WO2024034593A1_13	.	CO[C@@H](C)COC1=NC2=C(OCC3=CC=C(C(=O)N4CCC5(CN(CC6=CC7=C(C=C6)C(N6CCC(=O)NC6=O)=NN7C)C5)C4)C=C3)C(C3=C(C)C(F)=CC4=C3C=NN4)=C(C3CC3)C=C2C(N2CC(C#N)C2)=N1	C54H55FN12O6	KRAS	P01116	CRBN	WO-2024034593-A1
TPD-LJM95Z	WO2024034593A1_14	.	CO[C@@H](C)COC1=NC2=C(OCC3=CC=C(C(=O)N4CCN(CC5=CC=C6C(=C5)N(C)N=C6N5CCC(=O)NC5=O)C[C@@H]4C)C=C3)C(C3=C(C)C(F)=CC4=C3C=NN4)=C(C3CC3)C=C2C(N2CC(C#N)C2)=N1	C53H55FN12O6	KRAS	P01116	CRBN	WO-2024034593-A1
TPD-0224RB	WO2024034593A1_15	.	CO[C@@H](C)COC1=NC2=C(OCC3=CC=C(C(=O)N4CC[C@H](CN(C)CC5=CC6=C(C=C5)C(N5CCC(=O)NC5=O)=NN6C)C4)C=C3)C(C3=C(C)C(F)=CC4=C3C=NN4)=C(C3CC3)C=C2C(N2CC(C#N)C2)=N1	C54H57FN12O6	KRAS	P01116	CRBN	WO-2024034593-A1
TPD-0I99U6	WO2024034593A1_16	.	CO[C@@H](C)COC1=NC2=C(C=C(C3CC3)C(C3=C(C)C(F)=CC4=C3C=NN4)=C2OCC2=CC=C(C(=O)N3CC4(CN(CC5=CC6=C(C=C5)C(N5CCC(=O)NC5=O)=NN6C)C4)C3)C=C2)C(N2CC(C#N)C2)=N1	C53H53FN12O6	KRAS	P01116	CRBN	WO-2024034593-A1
TPD-9LQZ1L	WO2024034593A1_17	.	CO[C@@H](C)COC1=NC2=C(OCC3=CC=C(C(=O)N4CCN(CC5=CC=C6C(=C5)N(C)C(=O)N6C5CCC(=O)NC5=O)C[C@@H]4C)C=C3)C(C3=C(C)C(F)=CC4=C3C=NN4)=C(C3CC3)C=C2C(OC2CN(C(=O)NCCN(C)C)C2)=C1	C59H68FN11O9	KRAS	P01116	CRBN	WO-2024034593-A1
TPD-AZ4GCP	WO2024034593A1_18	.	CO[C@@H](C)COC1=NC2=C(OCC3=CC=C(C(=O)N4CCN(CC5=CC=C6C(=C5)N(C)N=C6N5CCC(=O)NC5=O)C[C@@H]4C)C=C3)C(C3=C(C)C(F)=CC4=C3C=NN4)=C(C3CC3)C=C2C(OC2CN(C(=O)NCCN(C)C)C2)=C1	C58H67FN12O8	KRAS	P01116	CRBN	WO-2024034593-A1
TPD-ZXOYEB	WO2024034593A1_19	.	CO[C@@H](C)COC1=NC(N2CC[C@H]2C(N)=O)=C2C=C(C3CC3)C(C3=C(C)C(F)=CC4=C3C=NN4)=C(OCC3=CC=C(CN4CCN(CC5=CC=C6C(=C5)N(C)N=C6N5CCC(=O)NC5=O)C[C@@H]4C)C=C3)C2=N1	C53H59FN12O6	KRAS	P01116	CRBN	WO-2024034593-A1
TPD-PHQ5A2	WO2024034593A1_20	.	CO[C@@H](C)COC1=NC(N2CC[C@H]2C(N)=O)=C2C=C(C3CC3)C(C3=C(C)C(F)=CC4=C3C=NN4)=C(OCC3=CC=C(CN4CCN(CC5=CC=C6C(=C5)N(C)N=C6N5CCC(=O)NC5=O)CC4=O)C=C3)C2=N1	C52H55FN12O7	KRAS	P01116	CRBN	WO-2024034593-A1
TPD-39Q6M4	WO2024034593A1_21	.	CC1=C(C2=C(C3CC3)C=C3C(N4CC(C#N)C4)=NC(OC4CCOCC4)=NC3=C2OCC2=CC=C(C(=O)N3CCN(CC4=CC=C5C(=C4)N(C)N=C5N4CCC(=O)NC4=O)C[C@@H]3C)C=C2)C2=C(C=C1F)NN=C2	C54H55FN12O6	KRAS	P01116	CRBN	WO-2024034593-A1
TPD-SM5KZJ	WO2024034593A1_22	.	CO[C@@H](C)COC1=NC2=C(OCC3=CC=C(C(=O)N4CCC5(CCN(CCOC6=CC(N7CCC(=O)NC7=O)=CC=C6)CC5)CC4)C=C3)C(C3=C(C)C(F)=CC4=C3C=NN4)=C(C3CC3)C=C2C(N2CC(C#N)C2)=N1	C56H61FN10O7	KRAS	P01116	CRBN	WO-2024034593-A1
TPD-HMKUKR	SCHEMBL27064548	N-[4-(3-chloro-4-cyanophenoxy)cyclohexyl]-6-[4-[[4-[1-[(3R)-2,6-dioxopiperidin-3-yl]benzo[e][1]benzofuran-6-yl]piperazin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCN(c6cccc7c6ccc6occ([C@H]8CCC(=O)NC8=O)c67)CC5)CC4)nn3)CC2)cc1Cl	C45H47ClN8O5	AR	P10275	CRBN	WO-2024055994-A1
TPD-P8IH1S	SCHEMBL30836844	6-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]-N-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-imidazo[1,5-a]indol-7-yl]methyl]hexanamide	Cc1sc2c(c1C)C(c1ccc(Cl)cc1)=N[C@@H](CC(=O)NCCCCCC(=O)NCc1ccc3cc4n(c3c1)C(=O)N(C1CCC(=O)NC1=O)C4)c1nnc(C)n1-2	C41H42ClN9O5S	BRD4	O60885	CRBN	WO-2024067793-A1
TPD-R37M1O	SCHEMBL30836875	6-[[2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetyl]amino]-N-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-imidazo[1,5-a]indol-6-yl]methyl]hexanamide	Cc1sc2c(c1C)C(c1ccc(Cl)cc1)=N[C@@H](CC(=O)NCCCCCC(=O)NCc1ccc3c(c1)cc1n3C(=O)N(C3CCC(=O)NC3=O)C1)c1nnc(C)n1-2	C41H42ClN9O5S	BRD4	O60885	CRBN	WO-2024067793-A1
TPD-BCKJ44	SCHEMBL30857666	(2S,4R)-1-[(2S)-2-[3-[5-[4-[(3R)-3-[4-[[4-[4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]benzoyl]sulfamoyl]-2-(trifluoromethylsulfonyl)anilino]-4-phenylsulfanylbutyl]piperazin-1-yl]-5-oxopentoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](c2cc(OCCCCC(=O)N3CCN(CC[C@H](CSc4ccccc4)Nc4ccc(S(=O)(=O)NC(=O)c5ccc(N6CCN(CC7=C(c8ccc(Cl)cc8)CCC(C)(C)C7)CC6)cc5)cc4S(=O)(=O)C(F)(F)F)CC3)no2)C(C)C)cc1	C77H92ClF3N10O11S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-70FYGF	SCHEMBL30857590	(2S,4R)-1-[(2R)-2-[3-[5-[4-[(3R)-3-[4-[[4-[4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]benzoyl]sulfamoyl]-2-(trifluoromethylsulfonyl)anilino]-4-phenylsulfanylbutyl]piperazin-1-yl]-5-oxopentoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](c2cc(OCCCCC(=O)N3CCN(CC[C@H](CSc4ccccc4)Nc4ccc(S(=O)(=O)NC(=O)c5ccc(N6CCN(CC7=C(c8ccc(Cl)cc8)CCC(C)(C)C7)CC6)cc5)cc4S(=O)(=O)C(F)(F)F)CC3)no2)C(C)C)cc1	C77H92ClF3N10O11S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-714NHX	WO2024067818A1_1	(2S,4R)-1-[2-[3-[5-[4-[(3R)-3-[4-[[4-[4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]benzoyl]sulfamoyl]-2-(trifluoromethylsulfonyl)anilino]-4-phenylsulfanylbutyl]piperazin-1-yl]-5-oxopentoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)C(c2cc(OCCCCC(=O)N3CCN(CC[C@H](CSc4ccccc4)Nc4ccc(S(=O)(=O)NC(=O)c5ccc(N6CCN(CC7=C(c8ccc(Cl)cc8)CCC(C)(C)C7)CC6)cc5)cc4S(=O)(=O)C(F)(F)F)CC3)no2)C(C)C)cc1	C77H92ClF3N10O11S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-XXJNZH	WO2024067818A1_10	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCC(=O)N2CCN(CC[C@H](CSc3ccccc3)Nc3ccc(S(=O)(=O)NC(=O)c4ccc5c(c4)OC[C@@H]4CN(CC6=C(c7ccc(Cl)cc7)CCC(C)(C)C6)CCN54)cc3S(=O)(=O)C(F)(F)F)CC2)C(C)(C)C)cc1	C79H98ClF3N10O11S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-3T37SM	WO2024067818A1_11	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCC(=O)N2CCN(CC[C@H](CSc3ccccc3)Nc3ccc(S(=O)(=O)NC(=O)c4ccc5c(c4)OC[C@H]4CN(CC6=C(c7ccc(Cl)cc7)CCC(C)(C)C6)CCN54)cc3S(=O)(=O)C(F)(F)F)CC2)C(C)(C)C)cc1	C79H98ClF3N10O11S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-1FCU05	WO2024067818A1_12-1	.	C[C@@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](NC(=O)CCCCCC(=O)N1CCN(CC[C@H](CSc2ccccc2)Nc2ccc(S(=O)(=O)NC(=O)c3ccc4c(c3)OC[C@@H]3CN(CC5=C(c6ccc(Cl)cc6)CCC(C)(C)C5)CCN43)cc2S(=O)(=O)C(F)(F)F)CC1)C(C)(C)C)c1ccc2c(c1)OCc1ncsc1-2	C78H94ClF3N10O12S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-QX56Z7	WO2024067818A1_12-2	.	C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](NC(=O)CCCCCC(=O)N1CCN(CC[C@H](CSc2ccccc2)Nc2ccc(S(=O)(=O)NC(=O)c3ccc4c(c3)OC[C@@H]3CN(CC5=C(c6ccc(Cl)cc6)CCC(C)(C)C5)CCN43)cc2S(=O)(=O)C(F)(F)F)CC1)C(C)(C)C)c1ccc2c(c1)OCc1ncsc1-2	C78H94ClF3N10O12S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-4JI1R4	WO2024067818A1_13-1	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](c2cc(OCCCCC(=O)N3CCN(CC[C@H](CSc4ccccc4)Nc4ccc(S(=O)(=O)NC(=O)c5ccc6c(c5)OC[C@@H]5CN(CC7=C(c8ccc(Cl)cc8)CCC(C)(C)C7)CCN65)cc4S(=O)(=O)C(F)(F)F)CC3)no2)C(C)C)cc1	C78H92ClF3N10O12S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-XB49X9	WO2024067818A1_13-2	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](c2cc(OCCCCC(=O)N3CCN(CC[C@H](CSc4ccccc4)Nc4ccc(S(=O)(=O)NC(=O)c5ccc6c(c5)OC[C@@H]5CN(CC7=C(c8ccc(Cl)cc8)CCC(C)(C)C7)CCN65)cc4S(=O)(=O)C(F)(F)F)CC3)no2)C(C)C)cc1	C78H92ClF3N10O12S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-SD9TC3	WO2024067818A1_14	.	CC1(C)CCC(c2ccc(Cl)cc2)=C(CN2CCN3c4ccc(C(=O)NS(=O)(=O)c5ccc(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)NCc7ccc8c(c7)OCc7ncsc7-8)C(C)(C)C)CC6)CSc6ccccc6)c(S(=O)(=O)C(F)(F)F)c5)cc4OC[C@@H]3C2)C1	C77H92ClF3N10O12S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-6WDUI3	PROTAC BcI-2/BcI-xI Degrader-1	PROTAC BcI-2/BcI-xI Degrader-1; 3034200-49-9; orb2564493; EX-A9768; HY-158551; CS-1057371	CC1(C)CCC(c2ccc(Cl)cc2)=C(CN2CCN3c4ccc(C(=O)NS(=O)(=O)c5ccc(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)NCc7ccc8c(c7)OCCc7ncsc7-8)C(C)(C)C)CC6)CSc6ccccc6)c(S(=O)(=O)C(F)(F)F)c5)cc4OC[C@@H]3C2)C1	C78H94ClF3N10O12S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-P310LW	WO2024067818A1_16-1	.	C[C@@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](NC(=O)CCCCCCC(=O)N1CCN(CC[C@H](CSc2ccccc2)Nc2ccc(S(=O)(=O)NC(=O)c3ccc4c(c3)OC[C@@H]3CN(CC5=C(c6ccc(Cl)cc6)CCC(C)(C)C5)CCN43)cc2S(=O)(=O)C(F)(F)F)CC1)C(C)(C)C)c1ccc2c(c1)OCc1ncsc1-2	C79H96ClF3N10O12S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-G6D9UH	WO2024067818A1_16-2	.	C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](NC(=O)CCCCCCC(=O)N1CCN(CC[C@H](CSc2ccccc2)Nc2ccc(S(=O)(=O)NC(=O)c3ccc4c(c3)OC[C@@H]3CN(CC5=C(c6ccc(Cl)cc6)CCC(C)(C)C5)CCN43)cc2S(=O)(=O)C(F)(F)F)CC1)C(C)(C)C)c1ccc2c(c1)OCc1ncsc1-2	C79H96ClF3N10O12S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-JEVKI1	WO2024067818A1_17-1	.	CC(C)[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc2c(c1)OCc1ncsc1-2)c1cc(OCCCCC(=O)N2CCN(CC[C@H](CSc3ccccc3)Nc3ccc(S(=O)(=O)NC(=O)c4ccc5c(c4)OC[C@@H]4CN(CC6=C(c7ccc(Cl)cc7)CCC(C)(C)C6)CCN54)cc3S(=O)(=O)C(F)(F)F)CC2)no1	C77H88ClF3N10O13S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-7REL3O	WO2024067818A1_17-2	.	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc2c(c1)OCc1ncsc1-2)c1cc(OCCCCC(=O)N2CCN(CC[C@H](CSc3ccccc3)Nc3ccc(S(=O)(=O)NC(=O)c4ccc5c(c4)OC[C@@H]4CN(CC6=C(c7ccc(Cl)cc7)CCC(C)(C)C6)CCN54)cc3S(=O)(=O)C(F)(F)F)CC2)no1	C77H88ClF3N10O13S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-5CPCIX	SCHEMBL30857752	(2S,4R)-1-[(2S)-2-[3-[5-[4-[(3R)-3-[4-[[4-[(2S)-4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]-2-(hydroxymethyl)piperazin-1-yl]benzoyl]sulfamoyl]-2-(trifluoromethylsulfonyl)anilino]-4-phenylsulfanylbutyl]piperazin-1-yl]-5-oxopentoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-N-(4H-chromeno[3,4-d][1,3]thiazol-7-ylmethyl)-4-hydroxypyrrolidine-2-carboxamide	CC(C)[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc2c(c1)OCc1ncsc1-2)c1cc(OCCCCC(=O)N2CCN(CC[C@H](CSc3ccccc3)Nc3ccc(S(=O)(=O)NC(=O)c4ccc(N5CCN(CC6=C(c7ccc(Cl)cc7)CCC(C)(C)C6)C[C@H]5CO)cc4)cc3S(=O)(=O)C(F)(F)F)CC2)no1	C77H90ClF3N10O13S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-2LU2WW	SCHEMBL30857667	(2S,4R)-1-[(2R)-2-[3-[5-[4-[(3R)-3-[4-[[4-[(2S)-4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]-2-(hydroxymethyl)piperazin-1-yl]benzoyl]sulfamoyl]-2-(trifluoromethylsulfonyl)anilino]-4-phenylsulfanylbutyl]piperazin-1-yl]-5-oxopentoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-N-(4H-chromeno[3,4-d][1,3]thiazol-7-ylmethyl)-4-hydroxypyrrolidine-2-carboxamide	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc2c(c1)OCc1ncsc1-2)c1cc(OCCCCC(=O)N2CCN(CC[C@H](CSc3ccccc3)Nc3ccc(S(=O)(=O)NC(=O)c4ccc(N5CCN(CC6=C(c7ccc(Cl)cc7)CCC(C)(C)C6)C[C@H]5CO)cc4)cc3S(=O)(=O)C(F)(F)F)CC2)no1	C77H90ClF3N10O13S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-ZK1CN4	SCHEMBL30857650	(2S,4R)-1-[(2S)-2-[3-[5-[4-[(3R)-3-[4-[[4-[4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]benzoyl]sulfamoyl]-2-(trifluoromethylsulfonyl)anilino]-4-phenylsulfanylbutyl]piperazin-1-yl]-5-oxopentoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-N-(4H-chromeno[3,4-d][1,3]thiazol-7-ylmethyl)-4-hydroxypyrrolidine-2-carboxamide	CC(C)[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc2c(c1)OCc1ncsc1-2)c1cc(OCCCCC(=O)N2CCN(CC[C@H](CSc3ccccc3)Nc3ccc(S(=O)(=O)NC(=O)c4ccc(N5CCN(CC6=C(c7ccc(Cl)cc7)CCC(C)(C)C6)CC5)cc4)cc3S(=O)(=O)C(F)(F)F)CC2)no1	C76H88ClF3N10O12S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-5GZGRS	WO2024067818A1_19-2	.	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc2c(c1)OCc1ncsc1-2)c1cc(OCCCCC(=O)N2CCN(CC[C@H](CSc3ccccc3)Nc3ccc(S(=O)(=O)NC(=O)c4ccc(N5CCN(CC6=C(c7ccc(Cl)cc7)CCC(C)(C)C6)CC5)cc4)cc3S(=O)(=O)C(F)(F)F)CC2)no1	C76H88ClF3N10O12S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-6GDQIG	SCHEMBL30857616	(2S,4R)-1-[(2S)-2-[[7-[2-[(3R)-3-[4-[[4-[4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]benzoyl]sulfamoyl]-2-(trifluoromethylsulfonyl)anilino]-4-phenylsulfanylbutyl]-4,6-dihydropyrrolo[3,4-c]pyrazol-5-yl]-7-oxoheptanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCC(=O)N2Cc3cn(CC[C@H](CSc4ccccc4)Nc4ccc(S(=O)(=O)NC(=O)c5ccc(N6CCN(CC7=C(c8ccc(Cl)cc8)CCC(C)(C)C7)CC6)cc5)cc4S(=O)(=O)C(F)(F)F)nc3C2)C(C)(C)C)cc1	C78H93ClF3N11O10S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-2P1LL3	WO2024067818A1_2-2	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCC(=O)N2Cc3cnn(CC[C@H](CSc4ccccc4)Nc4ccc(S(=O)(=O)NC(=O)c5ccc(N6CCN(CC7=C(c8ccc(Cl)cc8)CCC(C)(C)C7)CC6)cc5)cc4S(=O)(=O)C(F)(F)F)c3C2)C(C)(C)C)cc1	C78H93ClF3N11O10S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-GLSBU4	WO2024067818A1_20-1	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](c2cc(OCCCCCC(=O)N3CCN(CC[C@H](CSc4ccccc4)Nc4ccc(S(=O)(=O)NC(=O)c5ccc6c(c5)OC[C@@H]5CN(CC7=C(c8ccc(Cl)cc8)CCC(C)(C)C7)CCN65)cc4S(=O)(=O)C(F)(F)F)CC3)no2)C(C)C)cc1	C79H94ClF3N10O12S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-CPM9PN	WO2024067818A1_20-2	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](c2cc(OCCCCCC(=O)N3CCN(CC[C@H](CSc4ccccc4)Nc4ccc(S(=O)(=O)NC(=O)c5ccc6c(c5)OC[C@@H]5CN(CC7=C(c8ccc(Cl)cc8)CCC(C)(C)C7)CCN65)cc4S(=O)(=O)C(F)(F)F)CC3)no2)C(C)C)cc1	C79H94ClF3N10O12S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-R2YMHG	WO2024067818A1_21	.	CC1(C)CCC(c2ccc(Cl)cc2)=C(CN2CCN3c4ccc(C(=O)NS(=O)(=O)c5ccc(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)NCc7ccc8c(c7)OCc7ncsc7-8)C(C)(C)C)CC6)CSc6ccccc6)c(S(=O)(=O)C(F)(F)F)c5)cc4NC(=O)[C@@H]3C2)C1	C77H91ClF3N11O12S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-7DGT8W	WO2024067818A1_22	.	CC1(C)CCC(c2ccc(Cl)cc2)=C(CN2CCN3c4ccc(C(=O)NS(=O)(=O)c5ccc(N[C@H](CCN6CCN(C(=O)CCCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)NCc7ccc8c(c7)OCc7ncsc7-8)C(C)(C)C)CC6)CSc6ccccc6)c(SOOC(F)(F)F)c5)cc4OC[C@@H]3C2)C1	C78H94ClF3N10O12S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-PRIJBJ	WO2024067818A1_23	(2S,4R)-1-[(2S)-2-[[7-[4-[(3R)-3-[4-[[4-[4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]benzoyl]sulfamoyl]-2-(trifluoromethylsulfonyl)anilino]-4-phenylsulfanylbutyl]piperazin-1-yl]-7-oxoheptanoyl]amino]-3,3-dimethylbutanoyl]-N-(4H-chromeno[3,4-d][1,3]thiazol-7-ylmethyl)-4-hydroxypyrrolidine-2-carboxamide	CC1(C)CCC(c2ccc(Cl)cc2)=C(CN2CCN(c3ccc(C(=O)NS(=O)(=O)c4ccc(N[C@H](CCN5CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)NCc6ccc7c(c6)OCc6ncsc6-7)C(C)(C)C)CC5)CSc5ccccc5)c(S(=O)(=O)C(F)(F)F)c4)cc3)CC2)C1	C76H92ClF3N10O11S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-MIB1YX	WO2024067818A1_24	.	Cc1noc2c1-c1ccc(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCC(=O)N3CCN(CC[C@H](CSc4ccccc4)Nc4ccc(S(=O)(=O)NC(=O)c5ccc(N6CCN(CC7=C(c8ccc(Cl)cc8)CCC(C)(C)C7)CC6)cc5)cc4S(=O)(=O)C(F)(F)F)CC3)C(C)(C)C)cc1OC2	C77H94ClF3N10O12S3	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-RZP9DD	WO2024067818A1_25	.	CC1(C)CCC(c2ccc(Cl)cc2)=C(CN2CCN3c4ccc(C(=O)NS(=O)(=O)c5ccc(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)NCc7ccc8c(c7)OCc7ncncc7-8)C(C)(C)C)CC6)CSc6ccccc6)c(SOOC(F)(F)F)c5)cc4OC[C@@H]3C2)C1	C78H93ClF3N11O12S3	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-GEZK4J	WO2024067818A1_26	.	CC(C)(C)[C@H](NC(=O)CCCCCC(=O)N1CCN(CC[C@H](CSc2ccccc2)Nc2ccc(S(=O)(=O)NC(=O)c3ccc(N4CCN(CC5=C(c6ccc(Cl)cc6)CC[C@@](C)(CO)C5)CC4)cc3)cc2S(=O)(=O)C(F)(F)F)CC1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc2c(c1)OCc1ncsc1-2	C76H92ClF3N10O12S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-KQLYQ9	WO2024067818A1_27	.	CC(C)(C)C(NC(=O)CCCCCC(=O)N1CCN(CCC(CSc2ccccc2)Nc2ccc(S(=O)(=O)NC(=O)c3ccc4c(c3)OC[C@@H]3CN(CC5=C(c6ccc(Cl)cc6)CCC6(CC6)C5)CCN43)cc2SOOC(F)(F)F)CC1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc2c(c1)OCc1ncsc1-2	C77H90ClF3N10O12S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-ATGCGX	WO2024067818A1_28-1	.	CC1(C)CCC(c2ccc(Cl)cc2)=C(CN2CCN3c4ccc(C(=O)NS(=O)(=O)c5ccc(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)NC(CO)c7ccc8c(c7)OCc7ncsc7-8)C(C)(C)C)CC6)CSc6ccccc6)c(S(=O)(=O)C(F)(F)F)c5)cc4OC[C@@H]3C2)C1	C78H94ClF3N10O13S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-YTUWF5	WO2024067818A1_28-2	.	CC1(C)CCC(c2ccc(Cl)cc2)=C(CN2CCN3c4ccc(C(=O)NS(=O)(=O)c5ccc(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](CO)c7ccc8c(c7)OCc7ncsc7-8)C(C)(C)C)CC6)CSc6ccccc6)c(S(=O)(=O)C(F)(F)F)c5)cc4OC[C@@H]3C2)C1	C78H94ClF3N10O13S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-U91T6E	WO2024067818A1_28	.	CC1(C)CCC(c2ccc(Cl)cc2)=C(CN2CCN3c4ccc(C(=O)NS(=O)(=O)c5ccc(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)NC(CO)c7ccc8c(c7)OCc7ncsc7-8)C(C)(C)C)CC6)CSc6ccccc6)c(S(=O)(=O)C(F)(F)F)c5)cc4NC(=O)[C@@H]3C2)C1	C78H93ClF3N11O13S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-FA1TSL	SCHEMBL30857663	(2S,4R)-1-[(2S)-2-[3-[5-[4-[(3R)-3-[4-[[4-[(2R)-4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]-2-(hydroxymethyl)piperazin-1-yl]benzoyl]sulfamoyl]-2-(trifluoromethylsulfonyl)anilino]-4-phenylsulfanylbutyl]piperazin-1-yl]-5-oxopentoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-N-(4H-chromeno[3,4-d][1,3]thiazol-7-ylmethyl)-4-hydroxypyrrolidine-2-carboxamide	CC(C)[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc2c(c1)OCc1ncsc1-2)c1cc(OCCCCC(=O)N2CCN(CC[C@H](CSc3ccccc3)Nc3ccc(S(=O)(=O)NC(=O)c4ccc(N5CCN(CC6=C(c7ccc(Cl)cc7)CCC(C)(C)C6)C[C@@H]5CO)cc4)cc3S(=O)(=O)C(F)(F)F)CC2)no1	C77H90ClF3N10O13S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-BRHZF7	SCHEMBL30857673	(2S,4R)-1-[(2R)-2-[3-[5-[4-[(3R)-3-[4-[[4-[(2R)-4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]-2-(hydroxymethyl)piperazin-1-yl]benzoyl]sulfamoyl]-2-(trifluoromethylsulfonyl)anilino]-4-phenylsulfanylbutyl]piperazin-1-yl]-5-oxopentoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-N-(4H-chromeno[3,4-d][1,3]thiazol-7-ylmethyl)-4-hydroxypyrrolidine-2-carboxamide	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc2c(c1)OCc1ncsc1-2)c1cc(OCCCCC(=O)N2CCN(CC[C@H](CSc3ccccc3)Nc3ccc(S(=O)(=O)NC(=O)c4ccc(N5CCN(CC6=C(c7ccc(Cl)cc7)CCC(C)(C)C6)C[C@@H]5CO)cc4)cc3S(=O)(=O)C(F)(F)F)CC2)no1	C77H90ClF3N10O13S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-BJL3PF	SCHEMBL30857552	(2S,4R)-1-[(2S)-2-[3-[5-[4-[(3R)-3-[4-[[4-[(2S)-4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]-2-(hydroxymethyl)piperazin-1-yl]benzoyl]sulfamoyl]-2-(trifluoromethylsulfonyl)anilino]-4-phenylsulfanylbutyl]piperazin-1-yl]-5-oxopentoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-N-(4H-chromeno[3,4-d][1,3]thiazol-7-ylmethyl)-4-hydroxypyrrolidine-2-carboxamide	CC(C)[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc2c(c1)OCc1ncsc1-2)c1cc(OCCCCC(=O)N2CCN(CC[C@H](CSc3ccccc3)Nc3ccc(S(=O)(=O)NC(=O)c4ccc(N5CCN(CC6=C(c7ccc(Cl)cc7)CC(C)(C)CC6)C[C@H]5CO)cc4)cc3S(=O)(=O)C(F)(F)F)CC2)no1	C77H90ClF3N10O13S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-6JBHJ9	SCHEMBL30857656	(2S,4R)-1-[(2R)-2-[3-[5-[4-[(3R)-3-[4-[[4-[(2S)-4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]-2-(hydroxymethyl)piperazin-1-yl]benzoyl]sulfamoyl]-2-(trifluoromethylsulfonyl)anilino]-4-phenylsulfanylbutyl]piperazin-1-yl]-5-oxopentoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-N-(4H-chromeno[3,4-d][1,3]thiazol-7-ylmethyl)-4-hydroxypyrrolidine-2-carboxamide	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc2c(c1)OCc1ncsc1-2)c1cc(OCCCCC(=O)N2CCN(CC[C@H](CSc3ccccc3)Nc3ccc(S(=O)(=O)NC(=O)c4ccc(N5CCN(CC6=C(c7ccc(Cl)cc7)CC(C)(C)CC6)C[C@H]5CO)cc4)cc3S(=O)(=O)C(F)(F)F)CC2)no1	C77H90ClF3N10O13S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-SVG845	WO2024067818A1_31	.	CC1(C)CCC(CN2CCN3c4ccc(C(=O)NS(=O)(=O)c5ccc(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)NCc7ccc8c(c7)OCc7ncsc7-8)C(C)(C)C)CC6)CSc6ccccc6)c(S(=O)(=O)C(F)(F)F)c5)cc4OC[C@@H]3C2)=C(c2ccc(Cl)cc2)C1	C77H92ClF3N10O12S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-H60OPY	WO2024067818A1_32	.	CC1(C)CCC(c2ccc(F)cc2)=C(CN2CCN3c4ccc(C(=O)NS(=O)(=O)c5ccc(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)NCc7ccc8c(c7)OCc7ncsc7-8)C(C)(C)C)CC6)CSc6ccccc6)c(S(=O)(=O)C(F)(F)F)c5)cc4OC[C@@H]3C2)C1	C77H92F4N10O12S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-TY8KXT	WO2024067818A1_33-1	.	CC1(C)CCC(CN2CCN3c4ccc(C(=O)NS(=O)(=O)c5ccc(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@H](CO)c7ccc8c(c7)OCc7ncsc7-8)C(C)(C)C)CC6)CSc6ccccc6)c(S(=O)(=O)C(F)(F)F)c5)cc4OC[C@@H]3C2)=C(c2ccc(Cl)cc2)C1	C78H94ClF3N10O13S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-GP8YEK	WO2024067818A1_33-2	.	CC1(C)CCC(CN2CCN3c4ccc(C(=O)NS(=O)(=O)c5ccc(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](CO)c7ccc8c(c7)OCc7ncsc7-8)C(C)(C)C)CC6)CSc6ccccc6)c(S(=O)(=O)C(F)(F)F)c5)cc4OC[C@@H]3C2)=C(c2ccc(Cl)cc2)C1	C78H94ClF3N10O13S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-GV22QZ	WO2024067818A1_33	.	CC1(C)CCC(CN2CCN3c4ccc(C(=O)NS(=O)(=O)c5ccc(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)NC(CO)c7ccc8c(c7)OCc7ncsc7-8)C(C)(C)C)CC6)CSc6ccccc6)c(S(=O)(=O)C(F)(F)F)c5)cc4OC[C@@H]3C2)=C(c2ccc(Cl)cc2)C1	C78H94ClF3N10O13S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-F5O3TM	WO2024067818A1_34	.	CC1(C)CCC(CN2CCN3c4ccc(C(=O)NS(=O)(=O)c5ccc(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)NCc7ccc8c(c7)OCc7ncsc7-8)C(C)(C)C)[C@H](CO)C6)CSc6ccccc6)c(S(=O)(=O)C(F)(F)F)c5)cc4OC[C@@H]3C2)=C(c2ccc(Cl)cc2)C1	C78H94ClF3N10O13S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-PXBN3Y	WO2024067818A1_37	.	CC1(C)CCC(c2ccc(Cl)cc2)=C(CN2CCN3c4ccc(C(=O)NS(=O)(=O)c5ccc(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)NCc7ccc8c(c7)OCc7ncsc7-8)C(C)(C)C)[C@H](CO)C6)CSc6ccccc6)c(S(=O)(=O)C(F)(F)F)c5)cc4OC[C@@H]3C2)C1	C78H94ClF3N10O13S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-CM0C0T	WO2024067818A1_38	.	CC1(C)CCC(c2ccc(Cl)cc2)=C(CN2CCN3c4ccc(C(=O)NS(=O)(=O)c5ccc(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)NCc7ccc8c(c7)OCc7ncsc7-8)C(C)(C)C)C[C@H]6CO)CSc6ccccc6)c(S(=O)(=O)C(F)(F)F)c5)cc4OC[C@@H]3C2)C1	C78H94ClF3N10O13S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-8P7JJR	WO2024067818A1_39	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)C(c2cc(=O)n(CCCCC(=O)N3CCN(CC[C@H](CSc4ccccc4)Nc4ccc(S(=O)(=O)NC(=O)c5ccc6c(c5)OC[C@@H]5CN(CC7=C(c8ccc(Cl)cc8)CCC(C)(C)C7)CCN65)cc4S(=O)(=O)C(F)(F)F)CC3)o2)C(C)C)cc1	C78H92ClF3N10O12S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-PMF9CG	WO2024067818A1_4	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCC(=O)N2CCN(CC[C@H](CSc3ccccc3)Nc3ccc(S(=O)(=O)NC(=O)c4ccc5c(c4)OC[C@H]4CN(CC6=C(c7ccc(Cl)cc7)CCC(C)(C)C6)CCN54)cc3S(=O)(=O)C(F)(F)F)CC2)C(C)(C)C)cc1	C78H96ClF3N10O11S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-O1W6LH	WO2024067818A1_40	.	CC1(C)CCC(c2ccc(Cl)cc2)=C(CC2(CO)CCN(c3ccc(C(=O)NS(=O)(=O)c4ccc(N[C@H](CCN5CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)NCc6ccc7c(c6)OCc6ncsc6-7)C(C)(C)C)CC5)CSc5ccccc5)c(S(=O)(=O)C(F)(F)F)c4)cc3)CC2)C1	C78H95ClF3N9O12S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-KXS8NO	WO2024067818A1_41	.	CC1(C)CCC(c2ccc(Cl)cc2)=C(CN2CCN3c4ccc(C(=O)NS(=O)(=O)c5ccc(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)NCc7ccc8c(c7)OCc7ncsc7-8)C(C)(C)C)CC6)CSc6ccccc6)c(S(=O)(=O)C(F)(F)F)c5)cc4N(CCO)C[C@@H]3C2)C1	C79H97ClF3N11O12S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-LMNQN4	SCHEMBL30857536	(2S,4R)-1-[(2S)-2-[3-[5-[4-[(3R)-3-[4-[[4-[(2S)-4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]-2-(2-hydroxyethyl)piperazin-1-yl]benzoyl]sulfamoyl]-2-(trifluoromethylsulfonyl)anilino]-4-phenylsulfanylbutyl]piperazin-1-yl]-5-oxopentoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-N-(4H-chromeno[3,4-d][1,3]thiazol-7-ylmethyl)-4-hydroxypyrrolidine-2-carboxamide	CC(C)[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc2c(c1)OCc1ncsc1-2)c1cc(OCCCCC(=O)N2CCN(CC[C@H](CSc3ccccc3)Nc3ccc(S(=O)(=O)NC(=O)c4ccc(N5CCN(CC6=C(c7ccc(Cl)cc7)CCC(C)(C)C6)C[C@@H]5CCO)cc4)cc3S(=O)(=O)C(F)(F)F)CC2)no1	C78H92ClF3N10O13S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-5VFW85	SCHEMBL30857539	(2S,4R)-1-[(2R)-2-[3-[5-[4-[(3R)-3-[4-[[4-[(2S)-4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]-2-(2-hydroxyethyl)piperazin-1-yl]benzoyl]sulfamoyl]-2-(trifluoromethylsulfonyl)anilino]-4-phenylsulfanylbutyl]piperazin-1-yl]-5-oxopentoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-N-(4H-chromeno[3,4-d][1,3]thiazol-7-ylmethyl)-4-hydroxypyrrolidine-2-carboxamide	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc2c(c1)OCc1ncsc1-2)c1cc(OCCCCC(=O)N2CCN(CC[C@H](CSc3ccccc3)Nc3ccc(S(=O)(=O)NC(=O)c4ccc(N5CCN(CC6=C(c7ccc(Cl)cc7)CCC(C)(C)C6)C[C@@H]5CCO)cc4)cc3S(=O)(=O)C(F)(F)F)CC2)no1	C78H92ClF3N10O13S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-XIB0KO	WO2024067818A1_43	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)C(C(C)C)n2cc(COCCCC(=O)N3CCN(CC[C@H](CSc4ccccc4)Nc4ccc(S(=O)(=O)NC(=O)c5ccc6c(c5)OCC5CN(CC7=C(c8ccc(Cl)cc8)CCC(C)(C)C7)CCN65)cc4S(=O)(=O)C(F)(F)F)CC3)nn2)cc1	C77H92ClF3N12O11S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-3RVP1K	WO2024067818A1_44	.	CC1(C)CCC(c2ccc(Cl)cc2)=C(CN2CCN3c4ccc(C(=O)NS(=O)(=O)c5ccc(N[C@H](CCN6C[C@H]7C[C@@H]6CN7C(=O)CCCCCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)NCc6ccc7c(c6)OCc6ncsc6-7)C(C)(C)C)CSc6ccccc6)c(S(=O)(=O)C(F)(F)F)c5)cc4OC[C@@H]3C2)C1	C78H92ClF3N10O12S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-WJ7YFJ	WO2024067818A1_45	.	CC1(C)CCC(c2ccc(Cl)cc2)=C(CN2CCN3c4ccc(C(=O)NS(=O)(=O)c5ccc(N[C@H](CCN6CC7CN(C(=O)CCCCCC(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)NCc8ccc9c(c8)OCc8ncsc8-9)C(C)(C)C)CC7C6)CSc6ccccc6)c(S(=O)(=O)C(F)(F)F)c5)cc4OC[C@@H]3C2)C1	C79H94ClF3N10O12S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-0DOSBE	WO2024067818A1_46	.	Cc1ncsc1-c1ccc2c(c1)OCCC2NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](NC(=O)CCCCCC(=O)N1CCN(CC[C@H](CSc2ccccc2)Nc2ccc(S(=O)(=O)NC(=O)c3ccc4c(c3)OC[C@@H]3CN(CC5=C(c6ccc(Cl)cc6)CCC(C)(C)C5)CCN43)cc2S(=O)(=O)C(F)(F)F)CC1)C(C)(C)C	C79H96ClF3N10O12S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-HFDQ6U	WO2024067818A1_47	.	CC1(C)CCC(c2ccc(Cl)cc2)=C(CN2CCN3c4ccc(C(=O)NS(=O)(=O)c5ccc(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)NCc7ccc8c(c7)OCc7ncoc7-8)C(C)(C)C)CC6)CSc6ccccc6)c(S(=O)(=O)C(F)(F)F)c5)cc4OC[C@@H]3C2)C1	C77H92ClF3N10O13S3	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-Y7JGZ2	WO2024067818A1_48	(2S,4R)-1-[(2S)-2-[[7-[4-[(3R)-3-[4-[[4-[4-[[2-(4-chlorophenyl)cyclohepten-1-yl]methyl]piperazin-1-yl]benzoyl]sulfamoyl]-2-(trifluoromethylsulfonyl)anilino]-4-phenylsulfanylbutyl]piperazin-1-yl]-7-oxoheptanoyl]amino]-3,3-dimethylbutanoyl]-N-(4H-chromeno[3,4-d][1,3]thiazol-7-ylmethyl)-4-hydroxypyrrolidine-2-carboxamide	CC(C)(C)[C@H](NC(=O)CCCCCC(=O)N1CCN(CC[C@H](CSc2ccccc2)Nc2ccc(S(=O)(=O)NC(=O)c3ccc(N4CCN(CC5=C(c6ccc(Cl)cc6)CCCCC5)CC4)cc3)cc2S(=O)(=O)C(F)(F)F)CC1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc2c(c1)OCc1ncsc1-2	C75H90ClF3N10O11S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-T31S4K	WO2024067818A1_49	N-(1,3-benzothiazol-2-yl)-2-[6-[[6-[[(2S)-1-[(2S,4R)-2-(4H-chromeno[3,4-d][1,3]thiazol-7-ylmethylcarbamoyl)-4-hydroxypyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-6-oxohexyl]sulfonylcarbamoyl]-5-[1-(cyclohexylmethyl)-5-methylpyrazol-4-yl]pyridin-2-yl]-3,4-dihydro-1H-isoquinoline-8-carboxamide	Cc1c(-c2ccc(N3CCc4cccc(C(=O)Nc5nc6ccccc6s5)c4C3)nc2C(=O)NS(=O)(=O)CCCCCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCc2ccc3c(c2)OCc2ncsc2-3)C(C)(C)C)cnn1CC1CCCCC1	C62H71N11O9S3	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-X4YPZI	WO2024067818A1_5	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCC(=O)N2CCN(CC[C@H](CSc3ccccc3)Nc3ccc(S(=O)(=O)NC(=O)c4ccc5c(c4)OC[C@@H]4CN(CC6=C(c7ccc(Cl)cc7)CCC(C)(C)C6)CCN54)cc3S(=O)(=O)C(F)(F)F)CC2)C(C)(C)C)cc1	C78H96ClF3N10O11S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-UV8599	WO2024067818A1_50	.	CC1(C)CCC(c2ccc(Cl)cc2)=C(CN2CCN3c4ccc(C(=O)NS(=O)(=O)c5ccc(N[C@H](CCN6C7CCC6CN(C(=O)CCCCCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)NCc6ccc8c(c6)OCc6ncsc6-8)C(C)(C)C)C7)CSc6ccccc6)c(S(=O)(=O)C(F)(F)F)c5)cc4OC[C@@H]3C2)C1	C79H94ClF3N10O12S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-9C1CH2	WO2024067818A1_51	.	CC1(C)CCC(c2ccc(Cl)cc2)=C(CN2CCN3c4ccc(C(=O)NS(=O)(=O)c5ccc(N[C@H](CCN6CC7(CCN(C(=O)CCCCCC(=O)NC(C(=O)N8C[C@H](O)C[C@H]8C(=O)NCc8ccc9c(c8)OCc8ncsc8-9)C(C)(C)C)CC7)C6)CSc6ccccc6)c(S(=O)(=O)C(F)(F)F)c5)cc4OC[C@@H]3C2)C1	C80H96ClF3N10O12S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-NDVJ5P	WO2024067818A1_52-1	.	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc2c(c1)OCc1ncsc1-2)c1cc(OCCCCC(=O)N2C[C@H]3C[C@@H]2CN3CC[C@H](CSc2ccccc2)Nc2ccc(S(=O)(=O)NC(=O)c3ccc4c(c3)OC[C@@H]3CN(CC5=C(c6ccc(Cl)cc6)CCC(C)(C)C5)CCN43)cc2S(=O)(=O)C(F)(F)F)no1	C78H88ClF3N10O13S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-7OE2OQ	WO2024067818A1_52-2	.	CC(C)[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc2c(c1)OCc1ncsc1-2)c1cc(OCCCCC(=O)N2C[C@H]3C[C@@H]2CN3CC[C@H](CSc2ccccc2)Nc2ccc(S(=O)(=O)NC(=O)c3ccc4c(c3)OC[C@@H]3CN(CC5=C(c6ccc(Cl)cc6)CCC(C)(C)C5)CCN43)cc2S(=O)(=O)C(F)(F)F)no1	C78H88ClF3N10O13S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-3T05RQ	SCHEMBL30857531	(2S,4R)-1-[(2R)-2-[3-[5-[(1R,4R)-5-[(3R)-3-[4-[[4-[4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]benzoyl]sulfamoyl]-2-(trifluoromethylsulfonyl)anilino]-4-phenylsulfanylbutyl]-2,5-diazabicyclo[2.2.1]heptan-2-yl]-5-oxopentoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-N-(4H-chromeno[3,4-d][1,3]thiazol-7-ylmethyl)-4-hydroxypyrrolidine-2-carboxamide	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc2c(c1)OCc1ncsc1-2)c1cc(OCCCCC(=O)N2C[C@H]3C[C@@H]2CN3CC[C@H](CSc2ccccc2)Nc2ccc(S(=O)(=O)NC(=O)c3ccc(N4CCN(CC5=C(c6ccc(Cl)cc6)CCC(C)(C)C5)CC4)cc3)cc2S(=O)(=O)C(F)(F)F)no1	C77H88ClF3N10O12S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-1TIYF1	SCHEMBL30857765	(2S,4R)-1-[(2S)-2-[3-[5-[(1R,4R)-5-[(3R)-3-[4-[[4-[4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]benzoyl]sulfamoyl]-2-(trifluoromethylsulfonyl)anilino]-4-phenylsulfanylbutyl]-2,5-diazabicyclo[2.2.1]heptan-2-yl]-5-oxopentoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-N-(4H-chromeno[3,4-d][1,3]thiazol-7-ylmethyl)-4-hydroxypyrrolidine-2-carboxamide	CC(C)[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc2c(c1)OCc1ncsc1-2)c1cc(OCCCCC(=O)N2C[C@H]3C[C@@H]2CN3CC[C@H](CSc2ccccc2)Nc2ccc(S(=O)(=O)NC(=O)c3ccc(N4CCN(CC5=C(c6ccc(Cl)cc6)CCC(C)(C)C5)CC4)cc3)cc2S(=O)(=O)C(F)(F)F)no1	C77H88ClF3N10O12S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-W19QYD	WO2024067818A1_54	(4aS)-3-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]-N-[4-[[(2R)-4-[(1S,4S)-5-[7-[[(2S)-1-[(2S,4R)-2-(4H-chromeno[3,4-d][1,3]thiazol-7-ylmethylcarbamoyl)-4-hydroxypyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-7-oxoheptanoyl]-2,5-diazabicyclo[2.2.1]heptan-2-yl]-1-phenylsulfanylbutan-2-yl]amino]-3-(trifluoromethylsulfonyl)phenyl]sulfonyl-2,4,4a,5-tetrahydro-1H-pyrazino[2,1-c][1,4]benzoxazine-8-carboxamide	CC1(C)CCC(c2ccc(Cl)cc2)=C(CN2CCN3c4ccc(C(=O)NS(=O)(=O)c5ccc(N[C@H](CCN6C[C@@H]7C[C@H]6CN7C(=O)CCCCCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)NCc6ccc7c(c6)OCc6ncsc6-7)C(C)(C)C)CSc6ccccc6)c(S(=O)(=O)C(F)(F)F)c5)cc4OC[C@@H]3C2)C1	C78H92ClF3N10O12S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-HIK455	WO2024067818A1_6	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCC(=O)N2CCN(CC[C@H](CSc3ccccc3)Nc3ccc(S(=O)(=O)NC(=O)c4ccc5c(c4)COCC4CN(CC6=C(c7ccc(Cl)cc7)CCC(C)(C)C6)CCN54)cc3S(=O)(=O)C(F)(F)F)CC2)C(C)(C)C)cc1	C79H98ClF3N10O11S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-G3E9QX	WO2024067818A1_7	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCC(=O)N2CCN(CC[C@H](CSc3ccccc3)Nc3ccc(S(=O)(=O)NC(=O)c4ccc5c(c4)OCCC4CN(CC6=C(c7ccc(Cl)cc7)CCC(C)(C)C6)CCN54)cc3S(=O)(=O)C(F)(F)F)CC2)C(C)(C)C)cc1	C79H98ClF3N10O11S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-QYZF73	WO2024067818A1_8	(2S,4R)-1-[(2S)-2-[[7-[4-[(3R)-3-[4-[[4-[4-[[7-(4-chlorophenyl)-2-methyl-2-azaspiro[3.5]non-6-en-6-yl]methyl]piperazin-1-yl]benzoyl]sulfamoyl]-2-(trifluoromethylsulfonyl)anilino]-4-phenylsulfanylbutyl]piperazin-1-yl]-7-oxoheptanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCC(=O)N2CCN(CC[C@H](CSc3ccccc3)Nc3ccc(S(=O)(=O)NC(=O)c4ccc(N5CCN(CC6=C(c7ccc(Cl)cc7)CCC7(C6)CN(C)C7)CC5)cc4)cc3S(=O)(=O)C(F)(F)F)CC2)C(C)(C)C)cc1	C78H97ClF3N11O10S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-D9J8R9	WO2024067818A1_9	(2S,4R)-1-[(2S)-2-[[7-[4-[(3R)-3-[4-[[4-[4-[[2-(4-chlorophenyl)phenyl]-hydroxymethyl]piperidin-1-yl]benzoyl]sulfamoyl]-2-(trifluoromethylsulfonyl)anilino]-4-phenylsulfanylbutyl]piperazin-1-yl]-7-oxoheptanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCC(=O)N2CCN(CC[C@H](CSc3ccccc3)Nc3ccc(S(=O)(=O)NC(=O)c4ccc(N5CCC(C(O)c6ccccc6-c6ccc(Cl)cc6)CC5)cc4)cc3S(=O)(=O)C(F)(F)F)CC2)C(C)(C)C)cc1	C76H89ClF3N9O11S4	BCL-2	P10415	VHL	WO-2024067818-A1
TPD-W5TG5Y	WO2024074848A1_BT150	.	O=C1CCC(N2C(=O)c3cccc(OCCCCCCC(=O)Nc4cccn([C@@H](CC5CC5)C(=O)N[C@@H](C[C@@H]5CCNC5=O)C(=O)C(=O)NCc5ccccc5)c4=O)c3C2=O)C(=O)N1	C46H51N7O11	3CL_pro	P0DTD1	CRBN	WO-2024074848-A1
TPD-DBWJT2	WO2024074848A1_BT152	.	O=C1CCC(N2C(=O)c3cccc(OCCCCCCCC(=O)Nc4cccn([C@@H](CC5CC5)C(=O)N[C@@H](C[C@@H]5CCNC5=O)C(=O)C(=O)NCc5ccccc5)c4=O)c3C2=O)C(=O)N1	C47H53N7O11	3CL_pro	P0DTD1	CRBN	WO-2024074848-A1
TPD-ESAAYG	WO2024074848A1_BT153	N-[1-[(2S)-1-[[(2S)-4-(benzylamino)-3,4-dioxo-1-[(3S)-2-oxopyrrolidin-3-yl]butan-2-yl]amino]-3-cyclopropyl-1-oxopropan-2-yl]-2-oxopyridin-3-yl]-9-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxynonanamide	O=C1CCC(N2C(=O)c3cccc(OCCCCCCCCC(=O)Nc4cccn([C@@H](CC5CC5)C(=O)N[C@@H](C[C@@H]5CCNC5=O)C(=O)C(=O)NCc5ccccc5)c4=O)c3C2=O)C(=O)N1	C48H55N7O11	3CL_pro	P0DTD1	CRBN	WO-2024074848-A1
TPD-9USBDU	SCHEMBL30800250	4-[2-(2-chlorophenyl)-6,8-dioxo-5,7-diazaspiro[3.4]octan-7-yl]-N-[6-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyhexyl]isoquinoline-6-carboxamide	O=C1CCC(N2C(=O)c3cccc(OCCCCCCNC(=O)c4ccc5cncc(N6C(=O)NC7(CC(c8ccccc8Cl)C7)C6=O)c5c4)c3C2=O)C(=O)N1	C41H37ClN6O8	3CL_pro	P0DTD1	CRBN	WO-2024074848-A1
TPD-Q3G8WN	SCHEMBL30800254	4-[2-(2-chlorophenyl)-6,8-dioxo-5,7-diazaspiro[3.4]octan-7-yl]-N-[6-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyhexyl]isoquinoline-7-carboxamide	O=C1CCC(N2C(=O)c3cccc(OCCCCCCNC(=O)c4ccc5c(N6C(=O)NC7(CC(c8ccccc8Cl)C7)C6=O)cncc5c4)c3C2=O)C(=O)N1	C41H37ClN6O8	3CL_pro	P0DTD1	CRBN	WO-2024074848-A1
TPD-XC4B90	SCHEMBL30800246	4-[2-(2-chlorophenyl)-6,8-dioxo-5,7-diazaspiro[3.4]octan-7-yl]-N-[8-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyoctyl]isoquinoline-6-carboxamide	O=C1CCC(N2C(=O)c3cccc(OCCCCCCCCNC(=O)c4ccc5cncc(N6C(=O)NC7(CC(c8ccccc8Cl)C7)C6=O)c5c4)c3C2=O)C(=O)N1	C43H41ClN6O8	3CL_pro	P0DTD1	CRBN	WO-2024074848-A1
TPD-CJHXDJ	WO2024074848A1_C10778O	.	O=C1CCC(N2C(=O)c3cccc(OCCCCNC(=O)c4ccc5cncc(N6C(=O)NC7(CC(c8ccccc8Cl)C7)C6=O)c5c4)c3C2=O)C(=O)N1	C39H33ClN6O8	3CL_pro	P0DTD1	CRBN	WO-2024074848-A1
TPD-IA6BVV	SCHEMBL30800279	4-[2-(2-chlorophenyl)-6,8-dioxo-5,7-diazaspiro[3.4]octan-7-yl]-N-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyethyl]isoquinoline-6-carboxamide	O=C1CCC(N2C(=O)c3cccc(OCCNC(=O)c4ccc5cncc(N6C(=O)NC7(CC(c8ccccc8Cl)C7)C6=O)c5c4)c3C2=O)C(=O)N1	C37H29ClN6O8	3CL_pro	P0DTD1	CRBN	WO-2024074848-A1
TPD-ZH69ZJ	SCHEMBL30800258	4-[2-(2-chlorophenyl)-6,8-dioxo-5,7-diazaspiro[3.4]octan-7-yl]-N-[6-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]amino]hexyl]isoquinoline-6-carboxamide	O=C1CCC(N2C(=O)c3ccc(NCCCCCCNC(=O)c4ccc5cncc(N6C(=O)NC7(CC(c8ccccc8Cl)C7)C6=O)c5c4)cc3C2=O)C(=O)N1	C41H38ClN7O7	3CL_pro	P0DTD1	CRBN	WO-2024074848-A1
TPD-D90JC6	WO2024074848A1_C10778R	4-[2-(2-chlorophenyl)-6,8-dioxo-5,7-diazaspiro[3.4]octan-7-yl]-N-[5-[[2-[4-(2,6-dioxopiperidin-3-yl)phenoxy]acetyl]amino]pentyl]isoquinoline-6-carboxamide	O=C(COc1ccc(C2CCC(=O)NC2=O)cc1)NCCCCCNC(=O)c1ccc2cncc(N3C(=O)NC4(CC(c5ccccc5Cl)C4)C3=O)c2c1	C40H39ClN6O7	3CL_pro	P0DTD1	CRBN	WO-2024074848-A1
TPD-HA9L8G	SCHEMBL30800261	4-[2-(2-chlorophenyl)-6,8-dioxo-5,7-diazaspiro[3.4]octan-7-yl]-N-[2-[2-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyethoxy]ethoxy]ethoxy]ethyl]isoquinoline-6-carboxamide	O=C1CCC(N2C(=O)c3cccc(OCCOCCOCCOCCNC(=O)c4ccc5cncc(N6C(=O)NC7(CC(c8ccccc8Cl)C7)C6=O)c5c4)c3C2=O)C(=O)N1	C43H41ClN6O11	3CL_pro	P0DTD1	CRBN	WO-2024074848-A1
TPD-81SFB8	WO2024074848A1_C10778T	4-[2-(2-chlorophenyl)-6,8-dioxo-5,7-diazaspiro[3.4]octan-7-yl]-N-[8-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyoctyl]isoquinoline-7-carboxamide	O=C1CCC(N2C(=O)c3cccc(OCCCCCCCCNC(=O)c4ccc5c(N6C(=O)NC7(CC(c8ccccc8Cl)C7)C6=O)cncc5c4)c3C2=O)C(=O)N1	C43H41ClN6O8	3CL_pro	P0DTD1	CRBN	WO-2024074848-A1
TPD-690SGD	SCHEMBL30800266	4-[2-(2-chlorophenyl)-6,8-dioxo-5,7-diazaspiro[3.4]octan-7-yl]-N-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxybutyl]isoquinoline-7-carboxamide	O=C1CCC(N2C(=O)c3cccc(OCCCCNC(=O)c4ccc5c(N6C(=O)NC7(CC(c8ccccc8Cl)C7)C6=O)cncc5c4)c3C2=O)C(=O)N1	C39H33ClN6O8	3CL_pro	P0DTD1	CRBN	WO-2024074848-A1
TPD-BT9SWI	SCHEMBL30800273	4-[2-(2-chlorophenyl)-6,8-dioxo-5,7-diazaspiro[3.4]octan-7-yl]-N-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyethyl]isoquinoline-7-carboxamide	O=C1CCC(N2C(=O)c3cccc(OCCNC(=O)c4ccc5c(N6C(=O)NC7(CC(c8ccccc8Cl)C7)C6=O)cncc5c4)c3C2=O)C(=O)N1	C37H29ClN6O8	3CL_pro	P0DTD1	CRBN	WO-2024074848-A1
TPD-WBPCR7	SCHEMBL30800277	4-[2-(2-chlorophenyl)-6,8-dioxo-5,7-diazaspiro[3.4]octan-7-yl]-N-[6-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]amino]hexyl]isoquinoline-7-carboxamide	O=C1CCC(N2C(=O)c3ccc(NCCCCCCNC(=O)c4ccc5c(N6C(=O)NC7(CC(c8ccccc8Cl)C7)C6=O)cncc5c4)cc3C2=O)C(=O)N1	C41H38ClN7O7	3CL_pro	P0DTD1	CRBN	WO-2024074848-A1
TPD-OMIXMT	WO2024074848A1_C10778X	4-[2-(2-chlorophenyl)-6,8-dioxo-5,7-diazaspiro[3.4]octan-7-yl]-N-[5-[[2-[4-(2,6-dioxopiperidin-3-yl)phenoxy]acetyl]amino]pentyl]isoquinoline-7-carboxamide	O=C(COc1ccc(C2CCC(=O)NC2=O)cc1)NCCCCCNC(=O)c1ccc2c(N3C(=O)NC4(CC(c5ccccc5Cl)C4)C3=O)cncc2c1	C40H39ClN6O7	3CL_pro	P0DTD1	CRBN	WO-2024074848-A1
TPD-VQNL74	SCHEMBL30800256	4-[2-(2-chlorophenyl)-6,8-dioxo-5,7-diazaspiro[3.4]octan-7-yl]-N-[2-[2-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyethoxy]ethoxy]ethoxy]ethyl]isoquinoline-7-carboxamide	O=C1CCC(N2C(=O)c3cccc(OCCOCCOCCOCCNC(=O)c4ccc5c(N6C(=O)NC7(CC(c8ccccc8Cl)C7)C6=O)cncc5c4)c3C2=O)C(=O)N1	C43H41ClN6O11	3CL_pro	P0DTD1	CRBN	WO-2024074848-A1
TPD-MNI58A	WO2024074848A1_TF355F1	N-[2-[[(1S)-1-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxybutoxy]phenyl]ethyl]amino]-2-oxo-1-pyridin-3-ylethyl]-N-(4-phenylphenyl)furan-2-carboxamide	C[C@H](NC(=O)C(c1cccnc1)N(C(=O)c1ccco1)c1ccc(-c2ccccc2)cc1)c1ccccc1OCCCCOc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O	C49H43N5O9	3CL_pro	P0DTD1	CRBN	WO-2024074848-A1
TPD-6HEO89	WO2024074848A1_TS284F2	N-dibenzofuran-3-yl-N-[2-[[(1S)-2-[3-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]propylamino]-2-oxo-1-phenylethyl]amino]-2-oxo-1-pyridin-3-ylethyl]furan-2-carboxamide	O=C1CCC(N2C(=O)c3cccc(NCCCNC(=O)[C@@H](NC(=O)C(c4cccnc4)N(C(=O)c4ccco4)c4ccc5c(c4)oc4ccccc45)c4ccccc4)c3C2=O)C(=O)N1	C48H39N7O9	3CL_pro	P0DTD1	CRBN	WO-2024074848-A1
TPD-FDXQ1N	WO2024074848A1_TS296	N-dibenzofuran-3-yl-N-[2-[[(1S)-2-[6-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]hexylamino]-2-oxo-1-phenylethyl]amino]-2-oxo-1-pyridin-3-ylethyl]furan-2-carboxamide	O=C1CCC(N2C(=O)c3cccc(NCCCCCCNC(=O)[C@@H](NC(=O)C(c4cccnc4)N(C(=O)c4ccco4)c4ccc5c(c4)oc4ccccc45)c4ccccc4)c3C2=O)C(=O)N1	C51H45N7O9	3CL_pro	P0DTD1	CRBN	WO-2024074848-A1
TPD-7ZUK5T	WO2024074848A1_TS297F1	N-dibenzofuran-3-yl-N-[2-[[(1S)-2-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethylamino]-2-oxo-1-phenylethyl]amino]-2-oxo-1-pyridin-3-ylethyl]furan-2-carboxamide	O=C1CCC(N2C(=O)c3cccc(NCCOCCOCCOCCNC(=O)[C@@H](NC(=O)C(c4cccnc4)N(C(=O)c4ccco4)c4ccc5c(c4)oc4ccccc45)c4ccccc4)c3C2=O)C(=O)N1	C53H49N7O12	3CL_pro	P0DTD1	CRBN	WO-2024074848-A1
TPD-Z5FTCQ	WO2024074848A1_TS301F1	N-dibenzofuran-3-yl-N-[2-[[(1S)-2-[5-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]pentylamino]-2-oxo-1-phenylethyl]amino]-2-oxo-1-pyridin-3-ylethyl]furan-2-carboxamide	O=C1CCC(N2C(=O)c3cccc(NCCCCCNC(=O)[C@@H](NC(=O)C(c4cccnc4)N(C(=O)c4ccco4)c4ccc5c(c4)oc4ccccc45)c4ccccc4)c3C2=O)C(=O)N1	C50H43N7O9	3CL_pro	P0DTD1	CRBN	WO-2024074848-A1
TPD-MHC84A	WO2024074848A1_TS302F1	N-dibenzofuran-3-yl-N-[2-[[(1S)-2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethylamino]-2-oxo-1-phenylethyl]amino]-2-oxo-1-pyridin-3-ylethyl]furan-2-carboxamide	O=C1CCC(N2C(=O)c3cccc(NCCOCCOCCNC(=O)[C@@H](NC(=O)C(c4cccnc4)N(C(=O)c4ccco4)c4ccc5c(c4)oc4ccccc45)c4ccccc4)c3C2=O)C(=O)N1	C51H45N7O11	3CL_pro	P0DTD1	CRBN	WO-2024074848-A1
TPD-QRAZSC	WO2024074848A1_TS303F1	N-dibenzofuran-3-yl-N-[2-[[(1S)-2-[2-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethylamino]-2-oxo-1-phenylethyl]amino]-2-oxo-1-pyridin-3-ylethyl]furan-2-carboxamide	O=C1CCC(N2C(=O)c3cccc(NCCOCCOCCOCCOCCNC(=O)[C@@H](NC(=O)C(c4cccnc4)N(C(=O)c4ccco4)c4ccc5c(c4)oc4ccccc45)c4ccccc4)c3C2=O)C(=O)N1	C55H53N7O13	3CL_pro	P0DTD1	CRBN	WO-2024074848-A1
TPD-RHURQG	WO2024074848A1_TS312F1	N-dibenzofuran-3-yl-N-[2-[[(1S)-2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethylamino]-2-oxo-1-phenylethyl]amino]-2-oxo-1-pyridin-3-ylethyl]furan-2-carboxamide	O=C1CCC(N2C(=O)c3cccc(NCCOCCNC(=O)[C@@H](NC(=O)C(c4cccnc4)N(C(=O)c4ccco4)c4ccc5c(c4)oc4ccccc45)c4ccccc4)c3C2=O)C(=O)N1	C49H41N7O10	3CL_pro	P0DTD1	CRBN	WO-2024074848-A1
TPD-MN10NS	WO2024074848A1_TS313F1	.	O=C1CCC(N2C(=O)c3cccc(NCCCCNC(=O)[C@@H](NC(=O)C(c4cccnc4)N(C(=O)c4ccco4)c4ccc5c(c4)oc4ccccc45)c4ccccc4)c3C2=O)C(=O)N1	C49H41N7O9	3CL_pro	P0DTD1	CRBN	WO-2024074848-A1
TPD-KUZAET	WO2024074848A1_TS325F2	N-[2-[[(1R)-1-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxybutoxy]phenyl]ethyl]amino]-2-oxo-1-pyridin-3-ylethyl]-N-(4-phenylphenyl)furan-2-carboxamide	C[C@@H](NC(=O)C(c1cccnc1)N(C(=O)c1ccco1)c1ccc(-c2ccccc2)cc1)c1cccc(OCCCCOc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)c1	C49H43N5O9	3CL_pro	P0DTD1	CRBN	WO-2024074848-A1
TPD-WO8K8U	WO2024074848A1_TS338F1	N-[(1S)-2-[[(1R)-1-[3-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyethoxy]phenyl]ethyl]amino]-2-oxo-1-pyridin-3-ylethyl]-N-(4-phenylphenyl)furan-2-carboxamide	C[C@@H](NC(=O)[C@H](c1cccnc1)N(C(=O)c1ccco1)c1ccc(-c2ccccc2)cc1)c1cccc(OCCOc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)c1	C47H39N5O9	3CL_pro	P0DTD1	CRBN	WO-2024074848-A1
TPD-I1YEYM	WO2024074848A1_TS339F2	N-[2-[[(1R)-1-[3-[8-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyoctoxy]phenyl]ethyl]amino]-2-oxo-1-pyridin-3-ylethyl]-N-(4-phenylphenyl)furan-2-carboxamide	C[C@@H](NC(=O)C(c1cccnc1)N(C(=O)c1ccco1)c1ccc(-c2ccccc2)cc1)c1cccc(OCCCCCCCCOc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)c1	C53H51N5O9	3CL_pro	P0DTD1	CRBN	WO-2024074848-A1
TPD-PZQNZW	WO2024074848A1_TS347F1	.	Cc1ncsc1-c1ccc(CNC(=O)C2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)C)c(OCCNC(=O)[C@@H](NC(=O)C(c2cccnc2)N(C(=O)c2ccco2)c2ccc3c(c2)oc2ccccc23)c2ccccc2)c1	C60H59FN8O10S	3CL_pro	P0DTD1	VHL	WO-2024074848-A1
TPD-L3XALY	WO2024074848A1_TS349F1	(2S,4R)-N-[[2-[6-[[(2S)-2-[[2-[dibenzofuran-3-yl(furan-2-carbonyl)amino]-2-pyridin-3-ylacetyl]amino]-2-phenylacetyl]amino]hexoxy]-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-1-[(2S)-2-[(1-fluorocyclopropanecarbonyl)amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)C)c(OCCCCCCNC(=O)[C@@H](NC(=O)C(c2cccnc2)N(C(=O)c2ccco2)c2ccc3c(c2)oc2ccccc23)c2ccccc2)c1	C64H67FN8O10S	3CL_pro	P0DTD1	VHL	WO-2024074848-A1
TPD-DL9TPV	WO2024074848A1_TS365F1	N-dibenzofuran-3-yl-N-[(1R)-2-[[(1S)-2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethylamino]-2-oxo-1-phenylethyl]amino]-2-oxo-1-pyridin-3-ylethyl]furan-2-carboxamide	O=C1CCC(N2C(=O)c3cccc(NCCNC(=O)[C@@H](NC(=O)[C@@H](c4cccnc4)N(C(=O)c4ccco4)c4ccc5c(c4)oc4ccccc45)c4ccccc4)c3C2=O)C(=O)N1	C47H37N7O9	3CL_pro	P0DTD1	CRBN	WO-2024074848-A1
TPD-BRB1GE	WO2024074848A1_TS369F1	N-dibenzofuran-3-yl-N-[(1R)-2-[[(1S)-2-[8-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]octylamino]-2-oxo-1-phenylethyl]amino]-2-oxo-1-pyridin-3-ylethyl]furan-2-carboxamide	O=C1CCC(N2C(=O)c3cccc(NCCCCCCCCNC(=O)[C@@H](NC(=O)[C@@H](c4cccnc4)N(C(=O)c4ccco4)c4ccc5c(c4)oc4ccccc45)c4ccccc4)c3C2=O)C(=O)N1	C53H49N7O9	3CL_pro	P0DTD1	CRBN	WO-2024074848-A1
TPD-N2IZO8	WO2024074848A1_TS370F1	.	O=C1CCC(N2C(=O)c3cccc(NCCCCCCCCCCNC(=O)[C@@H](NC(=O)[C@@H](c4cccnc4)N(C(=O)c4ccco4)c4ccc5c(c4)oc4ccccc45)c4ccccc4)c3C2=O)C(=O)N1	C55H53N7O9	3CL_pro	P0DTD1	CRBN	WO-2024074848-A1
TPD-3J0PG3	WO2024074848A1_TS449F1	N-[(1R)-2-[[(1S)-2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethylamino]-2-oxo-1-phenylethyl]amino]-2-oxo-1-pyridin-3-ylethyl]-N-(4-phenylphenyl)furan-2-carboxamide	O=C1CCC(N2C(=O)c3cccc(NCCNC(=O)[C@@H](NC(=O)[C@@H](c4cccnc4)N(C(=O)c4ccco4)c4ccc(-c5ccccc5)cc4)c4ccccc4)c3C2=O)C(=O)N1	C47H39N7O8	3CL_pro	P0DTD1	CRBN	WO-2024074848-A1
TPD-HNUZW1	WO2024074848A1_TS450F1	.	O=C1CCC(N2C(=O)c3cccc(NCCCNC(=O)[C@@H](NC(=O)C(c4cccnc4)N(C(=O)c4ccco4)c4ccc(-c5ccccc5)cc4)c4ccccc4)c3C2=O)C(=O)N1	C48H41N7O8	3CL_pro	P0DTD1	CRBN	WO-2024074848-A1
TPD-4ITIDT	WO2024074848A1_TS451F1	N-[(1R)-2-[[(1S)-2-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]butylamino]-2-oxo-1-phenylethyl]amino]-2-oxo-1-pyridin-3-ylethyl]-N-(4-phenylphenyl)furan-2-carboxamide	O=C1CCC(N2C(=O)c3cccc(NCCCCNC(=O)[C@@H](NC(=O)[C@@H](c4cccnc4)N(C(=O)c4ccco4)c4ccc(-c5ccccc5)cc4)c4ccccc4)c3C2=O)C(=O)N1	C49H43N7O8	3CL_pro	P0DTD1	CRBN	WO-2024074848-A1
TPD-I4OV9Z	WO2024074848A1_TS453F1b	.	O=C1CCC(N2C(=O)c3cccc(NCCOCCNC(=O)[C@@H](NC(=O)[C@@H](c4cccnc4)N(C(=O)c4ccco4)c4ccc(-c5ccccc5)cc4)c4ccccc4)c3C2=O)C(=O)N1	C49H43N7O9	3CL_pro	P0DTD1	CRBN	WO-2024074848-A1
TPD-DAA2ML	WO2024074848A1_TS454F1	N-[(1R)-2-[[(1R)-2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethylamino]-2-oxo-1-phenylethyl]amino]-2-oxo-1-pyridin-3-ylethyl]-N-(4-phenylphenyl)furan-2-carboxamide	O=C1CCC(N2C(=O)c3cccc(NCCOCCOCCNC(=O)[C@H](NC(=O)[C@@H](c4cccnc4)N(C(=O)c4ccco4)c4ccc(-c5ccccc5)cc4)c4ccccc4)c3C2=O)C(=O)N1	C51H47N7O10	3CL_pro	P0DTD1	CRBN	WO-2024074848-A1
TPD-O75ODO	WO2024074848A1_TS455F1	N-[(1R)-2-[[(1S)-2-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethylamino]-2-oxo-1-phenylethyl]amino]-2-oxo-1-pyridin-3-ylethyl]-N-(4-phenylphenyl)furan-2-carboxamide	O=C1CCC(N2C(=O)c3cccc(NCCOCCOCCOCCNC(=O)[C@@H](NC(=O)[C@@H](c4cccnc4)N(C(=O)c4ccco4)c4ccc(-c5ccccc5)cc4)c4ccccc4)c3C2=O)C(=O)N1	C53H51N7O11	3CL_pro	P0DTD1	CRBN	WO-2024074848-A1
TPD-CB48GD	WO2024074848A1_TS456F1	.	O=C1CCC(N2C(=O)c3cccc(NCCOCCOCCOCCOCCNC(=O)[C@@H](NC(=O)[C@@H](c4cccnc4)N(C(=O)c4ccco4)c4ccc(-c5ccccc5)cc4)c4ccccc4)c3C2=O)C(=O)N1	C55H55N7O12	3CL_pro	P0DTD1	CRBN	WO-2024074848-A1
TPD-2UPLEY	WO2024074848A1_TS457F1	N-[(1R)-2-[[(1S)-2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]-2-oxo-1-phenylethyl]amino]-2-oxo-1-pyridin-3-ylethyl]-N-(4-phenylphenyl)furan-2-carboxamide	O=C1CCC(N2Cc3c(NC(=O)[C@@H](NC(=O)[C@@H](c4cccnc4)N(C(=O)c4ccco4)c4ccc(-c5ccccc5)cc4)c4ccccc4)cccc3C2=O)C(=O)N1	C45H36N6O7	3CL_pro	P0DTD1	CRBN	WO-2024074848-A1
TPD-O8ER6A	WO2024074848A1_TS462	N-[(1R)-2-[[(1R)-2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]amino]ethoxy]ethylamino]-2-oxo-1-phenylethyl]amino]-2-oxo-1-pyridin-3-ylethyl]-N-(4-phenylphenyl)furan-2-carboxamide	O=C1CCC(N2C(=O)c3ccc(NCCOCCNC(=O)[C@H](NC(=O)[C@@H](c4cccnc4)N(C(=O)c4ccco4)c4ccc(-c5ccccc5)cc4)c4ccccc4)cc3C2=O)C(=O)N1	C49H43N7O9	3CL_pro	P0DTD1	CRBN	WO-2024074848-A1
TPD-BFLJOK	WO2024074848A1_TS464	N-[(1R)-2-[[(1R)-2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]amino]ethoxy]ethoxy]ethylamino]-2-oxo-1-phenylethyl]amino]-2-oxo-1-pyridin-3-ylethyl]-N-(4-phenylphenyl)furan-2-carboxamide	O=C1CCC(N2C(=O)c3ccc(NCCOCCOCCNC(=O)[C@H](NC(=O)[C@@H](c4cccnc4)N(C(=O)c4ccco4)c4ccc(-c5ccccc5)cc4)c4ccccc4)cc3C2=O)C(=O)N1	C51H47N7O10	3CL_pro	P0DTD1	CRBN	WO-2024074848-A1
TPD-QEQXAF	WO2024074848A1_TS465	N-[(1R)-2-[[(1R)-2-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]amino]ethoxy]ethoxy]ethoxy]ethylamino]-2-oxo-1-phenylethyl]amino]-2-oxo-1-pyridin-3-ylethyl]-N-(4-phenylphenyl)furan-2-carboxamide	O=C1CCC(N2C(=O)c3ccc(NCCOCCOCCOCCNC(=O)[C@H](NC(=O)[C@@H](c4cccnc4)N(C(=O)c4ccco4)c4ccc(-c5ccccc5)cc4)c4ccccc4)cc3C2=O)C(=O)N1	C53H51N7O11	3CL_pro	P0DTD1	CRBN	WO-2024074848-A1
TPD-DSTAD1	WO2024074848A1_TS466	N-[(1R)-2-[[(1R)-2-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]-2-oxo-1-phenylethyl]amino]-2-oxo-1-pyridin-3-ylethyl]-N-(4-phenylphenyl)furan-2-carboxamide	O=C1CCC(N2C(=O)c3ccc(N4CCN(C(=O)[C@H](NC(=O)[C@@H](c5cccnc5)N(C(=O)c5ccco5)c5ccc(-c6ccccc6)cc5)c5ccccc5)CC4)cc3C2=O)C(=O)N1	C49H41N7O8	3CL_pro	P0DTD1	CRBN	WO-2024074848-A1
TPD-EZB7D4	WO2024074848A1_TS467	N-[(1R)-2-[[(1R)-2-[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]-2-oxo-1-phenylethyl]amino]-2-oxo-1-pyridin-3-ylethyl]-N-(4-phenylphenyl)furan-2-carboxamide	O=C1CCC(N2C(=O)c3cc(F)c(N4CCN(C(=O)[C@H](NC(=O)[C@@H](c5cccnc5)N(C(=O)c5ccco5)c5ccc(-c6ccccc6)cc5)c5ccccc5)CC4)cc3C2=O)C(=O)N1	C49H40FN7O8	3CL_pro	P0DTD1	CRBN	WO-2024074848-A1
TPD-X2QP72	WO2024074848A1_TS470	N-[(1R)-2-[[(1R)-2-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]-2-oxo-1-phenylethyl]amino]-2-oxo-1-pyridin-3-ylethyl]-N-(4-phenylphenyl)furan-2-carboxamide	O=C1CCC(N2C(=O)c3ccc(N4CCN(CC5CCN(C(=O)[C@H](NC(=O)[C@@H](c6cccnc6)N(C(=O)c6ccco6)c6ccc(-c7ccccc7)cc6)c6ccccc6)CC5)CC4)cc3C2=O)C(=O)N1	C55H52N8O8	3CL_pro	P0DTD1	CRBN	WO-2024074848-A1
TPD-FFOJK9	WO2024074848A1_TS471	N-[(1R)-2-[[(1R)-2-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]-2-oxo-1-phenylethyl]amino]-2-oxo-1-pyridin-3-ylethyl]-N-(4-phenylphenyl)furan-2-carboxamide	O=C1CCC(N2C(=O)c3cc(F)c(N4CCN(CC5CCN(C(=O)[C@H](NC(=O)[C@@H](c6cccnc6)N(C(=O)c6ccco6)c6ccc(-c7ccccc7)cc6)c6ccccc6)CC5)CC4)cc3C2=O)C(=O)N1	C55H51FN8O8	3CL_pro	P0DTD1	CRBN	WO-2024074848-A1
TPD-UD8MPP	WO2024074848A1_TS476	N-[(1R)-2-[[(1R)-2-[2-[[2-[4-(2,6-dioxopiperidin-3-yl)phenoxy]acetyl]amino]ethylamino]-2-oxo-1-phenylethyl]amino]-2-oxo-1-pyridin-3-ylethyl]-N-(4-phenylphenyl)furan-2-carboxamide	O=C(COc1ccc(C2CCC(=O)NC2=O)cc1)NCCNC(=O)[C@H](NC(=O)[C@@H](c1cccnc1)N(C(=O)c1ccco1)c1ccc(-c2ccccc2)cc1)c1ccccc1	C47H42N6O8	3CL_pro	P0DTD1	CRBN	WO-2024074848-A1
TPD-I038SV	WO2024074848A1_TS477	N-[(1R)-2-[[(1R)-2-[4-[[2-[4-(2,6-dioxopiperidin-3-yl)phenoxy]acetyl]amino]butylamino]-2-oxo-1-phenylethyl]amino]-2-oxo-1-pyridin-3-ylethyl]-N-(4-phenylphenyl)furan-2-carboxamide	O=C(COc1ccc(C2CCC(=O)NC2=O)cc1)NCCCCNC(=O)[C@H](NC(=O)[C@@H](c1cccnc1)N(C(=O)c1ccco1)c1ccc(-c2ccccc2)cc1)c1ccccc1	C49H46N6O8	3CL_pro	P0DTD1	CRBN	WO-2024074848-A1
TPD-21GYX2	SMARCA2 degrader-17	PRT3789; 2755761-78-3; SMARCA2 degrader-17; orb2663586; SCHEMBL26957018; GTPL13837; PRT-3789; EX-A11407; compound 1 [WO2024076985A2]; HY-159607; (2S,4R)-4-hydroxy-1-[(2R)-2-[3-[(2S)-1-[(3R)-3-[(10S)-4-(2-hydroxyphenyl)-1,5,6,8,12-pentazatricyclo[8.4.0.02,7]tetradeca-2,4,6-trien-12-yl]pyrrolidin-1-yl]propan-2-yl]oxy-1,2-oxazol-5-yl]-3-methylbutanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(O[C@@H](C)CN4CC[C@@H](N5CCN6C7=C(N=NC(C8=C(O)C=CC=C8)=C7)NC[C@H]6C5)C4)=NO3)C(C)C)C=C2)SC=N1	C47H58N10O6S	SMARCA2	P51531	VHL	WO-2024076985-A2
TPD-LGBGDS	WO2024078581A1_P-001	.	O=C(CCCNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O)NCCN1CCC2(CC1)CC(CNc1ccc(S(=O)(=O)NC(=O)c3ccc(N4CCN([C@@H]5CCCCc6c(Cl)cccc65)CC4)cc3Oc3cnc4[nH]ccc4c3)cc1[N+](=O)[O-])C2	C63H69ClN12O11S	BCL2L1	Q07817	CRBN	WO-2024078581-A1
TPD-YDM27V	WO2024078581A1_P-002	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCC(=O)NCCN2CCC3(CC2)CC(CNc2ccc(S(=O)(=O)NC(=O)c4ccc(N5CCN([C@@H]6CCCCc7c(Cl)cccc76)CC5)cc4Oc4cnc5[nH]ccc5c4)cc2[N+](=O)[O-])C3)C(C)(C)C)cc1	C73H88ClN13O11S2	BCL2L1	Q07817	VHL	WO-2024078581-A1
TPD-Y0LRFF	WO2024078581A1_P-003	.	C=C(NS(=O)(=O)c1ccc(NCC2CC3(CCN(CCNC(=O)CCCCCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)NCc4ccc(-c5scnc5C)cc4)C(C)(C)C)CC3)C2)c([N+](=O)[O-])c1)c1ccc(N2CCN([C@@H]3CCCCc4c(Cl)cccc43)CC2)cc1Oc1cnc2[nH]ccc2c1	C76H94ClN13O10S2	BCL2L1	Q07817	VHL	WO-2024078581-A1
TPD-KL2EMN	WO2024078581A1_P-004	.	C=C(NS(=O)(=O)c1ccc(NCC2CC3(CCN(CCNC(=O)CCCCCCCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)NCc4ccc(-c5scnc5C)cc4)C(C)(C)C)CC3)C2)c([N+](=O)[O-])c1)c1ccc(N2CCN([C@@H]3CCCCc4c(Cl)cccc43)CC2)cc1Oc1cnc2[nH]ccc2c1	C78H98ClN13O10S2	BCL2L1	Q07817	VHL	WO-2024078581-A1
TPD-0DZN3S	WO2024078581A1_P-005	.	O=C(COCCOCCOc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O)NCCN1CCC2(CC1)CC(CNc1ccc(S(=O)(=O)NC(=O)c3ccc(N4CCN([C@@H]5CCCCc6c(Cl)cccc65)CC4)cc3Oc3cnc4[nH]ccc4c3)cc1[N+](=O)[O-])C2	C65H72ClN11O14S	BCL2L1	Q07817	CRBN	WO-2024078581-A1
TPD-YZW6HB	WO2024078581A1_P-006	.	O=C(COCCOCCOCCOCCOc1cccc2c1C(=O)N(C1CCCNC1=O)C2=O)NCCN1CCC2(CC1)CC(CNc1ccc(S(=O)(=O)NC(=O)c3ccc(N4CCN([C@@H]5CCCCc6c(Cl)cccc65)CC4)cc3Oc3cnc4[nH]ccc4c3)cc1[N+](=O)[O-])C2	C69H82ClN11O15S	BCL2L1	Q07817	CRBN	WO-2024078581-A1
TPD-GS2SH3	WO2024078581A1_P-007	.	O=C(CCCCCCNc1cccc2c1C(=O)C(N1CCC(=O)NC1=O)C2=O)NCCN1CCC2(CC1)CC(CNc1ccc(S(=O)(=O)NC(=O)c3ccc(N4CCN([C@@H]5CCCCc6c(Cl)cccc65)CC4)cc3Oc3cnc4[nH]ccc4c3)cc1[N+](=O)[O-])C2	C66H75ClN12O11S	BCL2L1	Q07817	CRBN	WO-2024078581-A1
TPD-ABH8KL	WO2024078581A1_P-008	.	O=C(CCCCCCCCCNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O)NCCN1CCC2(CC1)CC(CNc1ccc(S(=O)(=O)NC(=O)c3ccc(N4CCN([C@@H]5CCCCc6c(Cl)cccc65)CC4)cc3Oc3cnc4[nH]ccc4c3)cc1[N+](=O)[O-])C2	C69H81ClN12O11S	BCL2L1	Q07817	CRBN	WO-2024078581-A1
TPD-Y3SY9J	WO2024078581A1_P-009	.	C=C([C@@H](NC(=O)CCOCCOCCOCCOCCN(CCN1CCC2(CC1)CC(CNc1ccc(S(=O)(=O)NC(=O)c3ccc(N4CCC([C@@H]5CCCCc6c(Cl)cccc65)CC4)cc3Oc3cnc4[nH]ccc4c3)cc1[N+](=O)[O-])C2)C(=O)OC(C)(C)C)C(C)(C)C)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(-c2scnc2C)cc1	C86H113ClN12O15S2	BCL2L1	Q07817	VHL	WO-2024078581-A1
TPD-330QL1	WO2024078581A1_P-010	.	C=C([C@@H](NC(=O)CCOCCOCCOCCOCCNCCN1CCC2(CC1)CC(CNc1ccc(S(=O)(=O)NC(=O)c3ccc(N4CCC([C@@H]5CCCCc6c(Cl)cccc65)CC4)cc3Oc3cnc4[nH]ccc4c3)cc1[N+](=O)[O-])C2)C(C)(C)C)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(-c2scnc2C)cc1	C81H105ClN12O13S2	BCL2L1	Q07817	VHL	WO-2024078581-A1
TPD-PO7PVY	WO2024078581A1_P-011	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCOCCOCCN2CCC3(CC2)CC(CNc2ccc(S(=O)(=O)NC(=O)c4ccc(N5CCN([C@@H]6CCCCc7c(Cl)cccc76)CC5)cc4Oc4cnc5[nH]ccc5c4)cc2[N+](=O)[O-])C3)C(C)(C)C)cc1	C73H89ClN12O12S2	BCL2L1	Q07817	VHL	WO-2024078581-A1
TPD-JD2M8C	WO2024078581A1_P-012	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCOCCOCCOCCOCCN2CCC3(CC2)CC(CNc2ccc(S(=O)(=O)NC(=O)c4ccc(N5CCN([C@@H]6CCCCc7c(Cl)cccc76)CC5)cc4Oc4cnc5[nH]ccc5c4)cc2[N+](=O)[O-])C3)C(C)(C)C)cc1	C77H97ClN12O14S2	BCL2L1	Q07817	VHL	WO-2024078581-A1
TPD-Z2MFB4	WO2024078581A1_P-013	.	O=C(CCNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O)NCCN1CCC2(CC1)CC(CNc1ccc(S(=O)(=O)NC(=O)c3ccc(N4CCN([C@@H]5CCCCc6c(Cl)cccc65)CC4)cc3Oc3cnc4[nH]ccc4c3)cc1[N+](=O)[O-])C2	C62H67ClN12O11S	BCL2L1	Q07817	CRBN	WO-2024078581-A1
TPD-8NHJBM	WO2024078581A1_P-014	.	O=C(CNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O)NCCN1CCC2(CC1)CC(CNc1ccc(S(=O)(=O)NC(=O)c3ccc(N4CCN([C@@H]5CCCCc6c(Cl)cccc65)CC4)cc3Oc3cnc4[nH]ccc4c3)cc1[N+](=O)[O-])C2	C61H65ClN12O11S	BCL2L1	Q07817	CRBN	WO-2024078581-A1
TPD-OY32XJ	WO2024078581A1_P-015	.	O=C(CCCCNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O)NCCN1CCC2(CC1)CC(CNc1ccc(S(=O)(=O)NC(=O)c3ccc(N4CCN([C@@H]5CCCCc6c(Cl)cccc65)CC4)cc3Oc3cnc4[nH]ccc4c3)cc1[N+](=O)[O-])C2	C64H71ClN12O11S	BCL2L1	Q07817	CRBN	WO-2024078581-A1
TPD-W3X7WV	WO2024078581A1_P-016	.	O=C1CCC(N2C(=O)c3cccc(OC[C@H]4CC[C@H](CN5CCC6(CC5)CC(CNc5ccc(S(=O)(=O)NC(=O)c7ccc(N8CCN([C@@H]9CCCCc%10c(Cl)cccc%109)CC8)cc7Oc7cnc8[nH]ccc8c7)cc5[N+](=O)[O-])C6)CC4)c3C2=O)C(=O)N1	C65H71ClN10O11S	BCL2L1	Q07817	CRBN	WO-2024078581-A1
TPD-G5EK8K	WO2024078581A1_P-017	.	O=C1CCC(N2C(=O)c3cccc(NCCCCN4CCC5(CC4)CC(CNc4ccc(S(=O)(=O)NC(=O)c6ccc(N7CCN([C@@H]8CCCCc9c(Cl)cccc98)CC7)cc6Oc6cnc7[nH]ccc7c6)cc4[N+](=O)[O-])C5)c3C2=O)C(=O)N1	C61H66ClN11O10S	BCL2L1	Q07817	CRBN	WO-2024078581-A1
TPD-W9XPF7	WO2024078581A1_P-018	.	O=C1CCC(N2C(=O)c3cccc(OC[C@H]4CC[C@@H](CN5CCC6(CC5)CC(CNc5ccc(S(=O)(=O)NC(=O)c7ccc(N8CCN([C@@H]9CCCCc%10c(Cl)cccc%109)CC8)cc7Oc7cnc8[nH]ccc8c7)cc5[N+](=O)[O-])C6)CC4)c3C2=O)C(=O)N1	C65H71ClN10O11S	BCL2L1	Q07817	CRBN	WO-2024078581-A1
TPD-ATB2S3	WO2024078581A1_P-019	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCOCCOCCNCCN2CCC3(CC2)CC(CNc2ccc(S(=O)(=O)NC(=O)c4ccc(N5CCN([C@@H]6CCCCc7c(Cl)cccc76)CC5)cc4Oc4cnc5[nH]ccc5c4)cc2[N+](=O)[O-])C3)C(C)(C)C)cc1	C75H94ClN13O12S2	BCL2L1	Q07817	VHL	WO-2024078581-A1
TPD-19CVTV	WO2024078581A1_P-020	.	O=C1CCC(N2C(=O)c3cccc(OCc4cccc(CN5CCC6(CC5)CC(CNc5ccc(S(=O)(=O)NC(=O)c7ccc(N8CCN([C@@H]9CCCCc%10c(Cl)cccc%109)CC8)cc7Oc7cnc8[nH]ccc8c7)cc5[N+](=O)[O-])C6)c4)c3C2=O)C(=O)N1	C65H65ClN10O11S	BCL2L1	Q07817	CRBN	WO-2024078581-A1
TPD-OWG095	WO2024078581A1_P-021	.	O=C1CCC(N2C(=O)c3cccc(OCc4ccc(CN5CCC6(CC5)CC(CNc5ccc(S(=O)(=O)NC(=O)c7ccc(N8CCN([C@@H]9CCCCc%10c(Cl)cccc%109)CC8)cc7Oc7cnc8[nH]ccc8c7)cc5[N+](=O)[O-])C6)cc4)c3C2=O)C(=O)N1	C65H65ClN10O11S	BCL2L1	Q07817	CRBN	WO-2024078581-A1
TPD-D8Q070	WO2024078581A1_P-022	.	O=C1CCC(N2C(=O)c3cccc(OC[C@H]4CC[C@@H](CN5CCC6(CC5)CC(CNc5ccc(S(=O)(=O)NC(=O)c7ccc(N8CCN([C@@H]9CCCCc%10c(Cl)cccc%109)CC8)cc7Oc7cnc8[nH]ccc8c7)cc5[N+](=O)[O-])C6)C4)c3C2=O)C(=O)N1	C64H69ClN10O11S	BCL2L1	Q07817	CRBN	WO-2024078581-A1
TPD-PWXUAE	WO2024078581A1_P-023	.	O=C1CCC(N2C(=O)c3cccc(N[C@H]4CC[C@H](C(=O)N5CCC6(CC5)CC(CNc5ccc(S(=O)(=O)NC(=O)c7ccc(N8CCN([C@@H]9CCCCc%10c(Cl)cccc%109)CC8)cc7Oc7cnc8[nH]ccc8c7)cc5[N+](=O)[O-])C6)CC4)c3C2=O)C(=O)N1	C64H68ClN11O11S	BCL2L1	Q07817	CRBN	WO-2024078581-A1
TPD-15VB78	WO2024078581A1_P-024	.	O=C1CCC(C2C(=O)c3cccc(NC[C@H]4CC[C@H](C(=O)N5CCC6(CC5)CC(CNc5ccc(S(=O)(=O)NC(=O)C7=C(Oc8cnc9[nH]ccc9c8)CC(N8CCN([C@@H]9CCCCc%10c(Cl)cccc%109)CC8)C=C7)cc5[N+](=O)[O-])C6)CC4)c3C2=O)C(=O)N1	C66H73ClN10O11S	BCL2L1	Q07817	CRBN	WO-2024078581-A1
TPD-P051R5	WO2024078581A1_P-025	.	O=C1CCC(N2C(=O)c3cccc(OCC4CC(CN5CCC6(CC5)CC(CNc5ccc(S(=O)(=O)NC(=O)c7ccc(N8CCN([C@@H]9CCCCc%10c(Cl)cccc%109)CC8)cc7Oc7cnc8[nH]ccc8c7)cc5[N+](=O)[O-])C6)C4)c3C2=O)C(=O)N1	C63H67ClN10O11S	BCL2L1	Q07817	CRBN	WO-2024078581-A1
TPD-7QR5L8	WO2024078581A1_P-026	.	O=C1CCC(N2C(=O)c3cccc(OCC4CCC(C(=O)N5CCC6(CC5)CC(CNc5ccc(S(=O)(=O)NC(=O)c7ccc(N8CCN([C@@H]9CCCCc%10c(Cl)cccc%109)CC8)cc7Oc7cnc8[nH]ccc8c7)cc5[N+](=O)[O-])C6)CC4)c3C2=O)C(=O)N1	C65H69ClN10O12S	BCL2L1	Q07817	CRBN	WO-2024078581-A1
TPD-ELL513	WO2024078581A1_P-027	.	O=C1CCC(N2C(=O)c3cccc(N[C@H]4CC[C@@H](C(=O)N5CCC6(CC5)CC(CNc5ccc(S(=O)(=O)NC(=O)c7ccc(N8CCN([C@@H]9CCCCc%10c(Cl)cccc%109)CC8)cc7Oc7cnc8[nH]ccc8c7)cc5[N+](=O)[O-])C6)CC4)c3C2=O)C(=O)N1	C64H68ClN11O11S	BCL2L1	Q07817	CRBN	WO-2024078581-A1
TPD-9BIYV5	WO2024078581A1_P-028	.	O=C1CCC(C2C(=O)c3cccc(NC[C@H]4CC[C@@H](C(=O)N5CCC6(CC5)CC(CNc5ccc(S(=O)(=O)NC(=O)c7ccc(N8CCN([C@@H]9CCCCc%10c(Cl)cccc%109)CC8)cc7Oc7cnc8[nH]ccc8c7)cc5[N+](=O)[O-])C6)CC4)c3C2=O)C(=O)N1	C66H71ClN10O11S	BCL2L1	Q07817	CRBN	WO-2024078581-A1
TPD-ZAFHAL	WO2024078581A1_P-029	.	O=C1CCC(N2C(=O)c3cccc(OC[C@H]4CC[C@@H](C(=O)N5CCC6(CC5)CC(CNc5ccc(S(=O)(=O)NC(=O)c7ccc(N8CCN([C@@H]9CCCCc%10c(Cl)cccc%109)CC8)cc7Oc7cnc8[nH]ccc8c7)cc5[N+](=O)[O-])C6)CC4)c3C2=O)C(=O)N1	C65H69ClN10O12S	BCL2L1	Q07817	CRBN	WO-2024078581-A1
TPD-RAPIMF	WO2024078581A1_P-030	.	O=C1CCC(N2C(=O)c3cccc(OC[C@@H]4CCC[C@H](CN5CCC6(CC5)CC(CNc5ccc(S(=O)(=O)NC(=O)c7ccc(N8CCN([C@@H]9CCCCc%10c(Cl)cccc%109)CC8)cc7OC7=CNC8NC=CC8=C7)cc5[N+](=O)[O-])C6)C4)c3C2=O)C(=O)N1	C65H73ClN10O11S	BCL2L1	Q07817	CRBN	WO-2024078581-A1
TPD-C4TLY7	WO2024078581A1_P-031	.	CN1C(=O)CCC(N2C(=O)c3cccc(NCCCCN4CCC5(CC4)CC(CNc4ccc(S(=O)(=O)NC(=O)c6ccc(N7CCN([C@@H]8CCCCc9c(Cl)cccc98)CC7)cc6Oc6cnc7[nH]ccc7c6)cc4[N+](=O)[O-])C5)c3C2=O)C1=O	C62H68ClN11O10S	BCL2L1	Q07817	CRBN	WO-2024078581-A1
TPD-BE2PWF	WO2024078581A1_P-032	.	O=C1CCC(N2C(=O)c3ccc(NCCCCN4CCC5(CC4)CC(CNc4ccc(S(=O)(=O)NC(=O)c6ccc(N7CCN([C@@H]8CCCCc9c(Cl)cccc98)CC7)cc6Oc6cnc7[nH]ccc7c6)cc4[N+](=O)[O-])C5)cc3C2=O)C(=O)N1	C61H66ClN11O10S	BCL2L1	Q07817	CRBN	WO-2024078581-A1
TPD-KSV1OF	WO2024078581A1_P-033	.	O=C1CCC(N2C(=O)c3cccc(NCCC(F)CN4CCC5(CC4)CC(CNc4ccc(S(=O)(=O)NC(=O)c6ccc(N7CCN([C@@H]8CCCCc9c(Cl)cccc98)CC7)cc6Oc6cnc7[nH]ccc7c6)cc4[N+](=O)[O-])C5)c3C2=O)C(=O)N1	C61H65ClFN11O10S	BCL2L1	Q07817	CRBN	WO-2024078581-A1
TPD-6Y6OG1	WO2024078581A1_P-034	.	O=C1CCC(N2C(=O)c3ccc(N4CCC(CCN5CCC6(CC5)CC(CNc5ccc(S(=O)(=O)NC(=O)c7ccc(N8CCN([C@@H]9CCCCc%10c(Cl)cccc%109)CC8)cc7Oc7cnc8[nH]ccc8c7)cc5[N+](=O)[O-])C6)CC4)cc3C2=O)C(=O)N1	C64H70ClN11O10S	BCL2L1	Q07817	CRBN	WO-2024078581-A1
TPD-7T9WBI	WO2024078581A1_P-035	.	O=C1CCC(N2C(=O)c3ccc(N4CCN(CCN5CCC6(CC5)CC(CNc5ccc(S(=O)(=O)NC(=O)c7ccc(N8CCN([C@@H]9CCCCc%10c(Cl)cccc%109)CC8)cc7Oc7cnc8[nH]ccc8c7)cc5[N+](=O)[O-])C6)CC4)cc3C2=O)C(=O)N1	C63H69ClN12O10S	BCL2L1	Q07817	CRBN	WO-2024078581-A1
TPD-GVIYMY	WO2024078581A1_P-036	.	O=C1CCC(N2C(=O)c3ccc(N4CCC(CN5CCC6(CC5)CC(CNc5ccc(S(=O)(=O)NC(=O)c7ccc(N8CCN([C@@H]9CCCCc%10c(Cl)cccc%109)CC8)cc7Oc7cnc8[nH]ccc8c7)cc5[N+](=O)[O-])C6)CC4)cc3C2=O)C(=O)N1	C63H68ClN11O10S	BCL2L1	Q07817	CRBN	WO-2024078581-A1
TPD-NF5ZUV	WO2024078581A1_P-037	.	O=C1CCC(N2C(=O)c3ccc(OC[C@H]4CC[C@H](CN5CCC6(CC5)CC(CNc5ccc(S(=O)(=O)NC(=O)c7ccc(N8CCN([C@@H]9CCCCc%10c(Cl)cccc%109)CC8)cc7Oc7cnc8[nH]ccc8c7)cc5[N+](=O)[O-])C6)CC4)cc3C2=O)C(=O)N1	C65H71ClN10O11S	BCL2L1	Q07817	CRBN	WO-2024078581-A1
TPD-ENKFST	WO2024078581A1_P-038	.	O=C1CCC(N2C(=O)c3cccc(NCC(F)(F)CN4CCC5(CC4)CC(CNc4ccc(S(=O)(=O)NC(=O)c6ccc(N7CCN([C@@H]8CCCCc9c(Cl)cccc98)CC7)cc6Oc6cnc7[nH]ccc7c6)cc4[N+](=O)[O-])C5)c3C2=O)C(=O)N1	C60H62ClF2N11O10S	BCL2L1	Q07817	CRBN	WO-2024078581-A1
TPD-O547Q6	WO2024078581A1_P-039	.	O=C1CCC(N2C(=O)c3ccc(N4CCN(C(=O)CN5CCC6(CC5)CC(CNc5ccc(S(=O)(=O)NC(=O)c7ccc(N8CCN([C@@H]9CCCCc%10c(Cl)cccc%109)CC8)cc7Oc7cnc8[nH]ccc8c7)cc5[N+](=O)[O-])C6)CC4)cc3C2=O)C(=O)N1	C63H67ClN12O11S	BCL2L1	Q07817	CRBN	WO-2024078581-A1
TPD-HVMWFR	WO2024078581A1_P-040	.	CC(=O)N[C@@H](CCCCNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O)C(=O)NCCN1CCC2(CC1)CC(CNc1ccc(S(=O)(=O)NC(=O)c3ccc(N4CCN([C@@H]5CCCCc6c(Cl)cccc65)CC4)cc3Oc3cnc4[nH]ccc4c3)cc1[N+](=O)[O-])C2	C67H76ClN13O12S	BCL2L1	Q07817	CRBN	WO-2024078581-A1
TPD-Y4ST7Y	WO2024078581A1_P-041	.	O=C1CCC(N2C(=O)c3cccc(NCCC(F)(F)CC4CCC5(CC4)CC(CNc4ccc(S(=O)(=O)NC(=O)c6ccc(N7CCN([C@@H]8CCCCc9c(Cl)cccc98)CC7)cc6Oc6cnc7[nH]ccc7c6)cc4[N+](=O)[O-])C5)c3C2=O)C(=O)N1	C62H65ClF2N10O10S	BCL2L1	Q07817	CRBN	WO-2024078581-A1
TPD-A14S7A	WO2024078581A1_P-042	.	O=C1CCC(N2Cc3c(OC[C@H]4CC[C@H](CN5CCC6(CC5)CC(CNc5ccc(S(=O)(=O)NC(=O)c7ccc(N8CCN([C@@H]9CCCCc%10c(Cl)cccc%109)CC8)cc7Oc7cnc8[nH]ccc8c7)cc5[N+](=O)[O-])C6)CC4)cccc3C2=O)C(=O)N1	C65H73ClN10O10S	BCL2L1	Q07817	CRBN	WO-2024078581-A1
TPD-OACO94	WO2024078581A1_P-043	.	CC(=O)NCCCC[C@H](Nc1ccc2c(c1)C(=O)N(C1CCC(=O)NC1=O)C2=O)C(=O)NCCN1CCC2(CC1)CC(CNc1ccc(S(=O)(=O)NC(=O)c3ccc(N4CCN([C@@H]5CCCCc6c(Cl)cccc65)CC4)cc3Oc3cnc4[nH]ccc4c3)cc1[N+](=O)[O-])C2	C67H76ClN13O12S	BCL2L1	Q07817	CRBN	WO-2024078581-A1
TPD-QEID0G	WO2024078581A1_P-044	.	CN1C(=O)CCC(N2C(=O)c3cccc(OC[C@H]4CC[C@H](CN5CCC6(CC5)CC(CNc5ccc(S(=O)(=O)NC(=O)c7ccc(N8CCN([C@@H]9CCCCc%10c(Cl)cccc%109)CC8)cc7Oc7cnc8[nH]ccc8c7)cc5[N+](=O)[O-])C6)CC4)c3C2=O)C1=O	C66H73ClN10O11S	BCL2L1	Q07817	CRBN	WO-2024078581-A1
TPD-6JR710	WO2024078581A1_P-045	.	NCCCC[C@H](Nc1ccc2c(c1)CN(C1CCC(=O)NC1=O)C2=O)C(=O)NCCN1CCC2(CC1)CC(CNc1ccc(S(=O)(=O)NC(=O)c3ccc(N4CCN([C@@H]5CCCCc6c(Cl)cccc65)CC4)cc3Oc3cnc4[nH]ccc4c3)cc1[N+](=O)[O-])C2	C65H76ClN13O10S	BCL2L1	Q07817	CRBN	WO-2024078581-A1
TPD-1A7N6Y	WO2024078581A1_P-046	.	NC(CCCCNc1cccc2c1CN(C1CCC(=O)NC1=O)C2=O)C(=O)NCCN1CCC2(CC1)CC(CNc1ccc(S(=O)(=O)NC(=O)c3ccc(N4CCN([C@@H]5CCCCc6c(Cl)cccc65)CC4)cc3Oc3cnc4[nH]ccc4c3)cc1[N+](=O)[O-])C2	C65H76ClN13O10S	BCL2L1	Q07817	CRBN	WO-2024078581-A1
TPD-2JWVTO	WO2024078581A1_P-047	.	O=C1CCC(N2C(=O)c3cccc(OCCCNCCCN4CCC5(CC4)CC(CNc4ccc(S(=O)(=O)NC(=O)c6ccc(N7CCN([C@@H]8CCCCc9c(Cl)cccc98)CC7)cc6Oc6cnc7[nH]ccc7c6)cc4[N+](=O)[O-])C5)c3C2=O)C(=O)N1	C63H70ClN11O11S	BCL2L1	Q07817	CRBN	WO-2024078581-A1
TPD-PK4VAP	WO2024078581A1_P-048	.	C=C1NC(=O)CCC1N1C(=O)c2cccc(OCCC(N)CCN3CCC4(CC3)CC(CNc3ccc(S(=O)(=O)NC(=O)c5ccc(N6CCN([C@@H]7CCCCc8c(C)cccc87)CC6)cc5Oc5cnc6[nH]ccc6c5)cc3[N+](=O)[O-])C4)c2C1=O	C64H73N11O10S	BCL2L1	Q07817	CRBN	WO-2024078581-A1
TPD-NMO2XH	WO2024078581A1_P-049	.	O=C1CCC(N2C(=O)c3cccc(OCCCN(CCCO)CCCN4CCC5(CC4)CC(CNc4ccc(S(=O)(=O)NC(=O)c6ccc(N7CCN([C@@H]8CCCCc9c(Cl)cccc98)CC7)cc6Oc6cnc7[nH]ccc7c6)cc4[N+](=O)[O-])C5)c3C2=O)C(=O)N1	C66H76ClN11O12S	BCL2L1	Q07817	CRBN	WO-2024078581-A1
TPD-XXLNNL	WO2024078581A1_P-050	.	O=C1CCC(N2C(=O)c3cccc(N=NCCCC(F)(F)CN4CCC5(CC4)CC(CNc4ccc(S(=O)(=O)NC(=O)c6ccc(N7CCN([C@@H]8CCCCc9c(Cl)cccc98)CC7)cc6Oc6cnc7[nH]ccc7c6)cc4[N+](=O)[O-])C5)c3C2=O)C(=O)N1	C62H65ClF2N12O10S	BCL2L1	Q07817	CRBN	WO-2024078581-A1
TPD-5FHXZK	WO2024078581A1_P-051	.	O=C1CCC(N2C(=O)c3ccc(N4CCN(CCC5CCC6(CC5)CC(CNc5ccc(S(=O)(=O)NC(=O)c7ccc(N8CCN([C@@H]9CCCCc%10c(Cl)cccc%109)CC8)cc7Oc7cnc8[nH]ccc8c7)cc5[N+](=O)[O-])C6)CC4)cc3C2=O)C(=O)N1	C64H70ClN11O10S	BCL2L1	Q07817	CRBN	WO-2024078581-A1
TPD-22OLL3	WO2024078581A1_P-052	.	CC(C)(C)OC(=O)NC(CCN1CCC2(CC1)CC(CNc1ccc(S(=O)(=O)NC(=O)c3ccc(N4CCN([C@@H]5CCCCc6c(Cl)cccc65)CC4)cc3Oc3cnc4[nH]ccc4c3)cc1[N+](=O)[O-])C2)COc1ccc2c(c1)C(=O)N(C1CCC(=O)NC1=O)C2=O	C66H74ClN11O13S	BCL2L1	Q07817	CRBN	WO-2024078581-A1
TPD-H2C906	WO2024078581A1_P-053	.	NC(CCN1CCC2(CC1)CC(CNc1ccc(S(=O)(=O)NC(=O)c3ccc(N4CCN([C@@H]5CCCCc6c(Cl)cccc65)CC4)cc3Oc3cnc4[nH]ccc4c3)cc1[N+](=O)[O-])C2)COc1ccc2c(c1)C(=O)N(C1CCC(=O)NC1=O)C2=O	C61H66ClN11O11S	BCL2L1	Q07817	CRBN	WO-2024078581-A1
TPD-6V9H7V	WO2024078581A1_P-054	.	O=C1CCC(N2C(=O)c3ccc(N4CCN(CC5CCC6(CC5)CC(CNc5ccc(S(=O)(=O)NC(=O)c7ccc(N8CCN([C@@H]9CCCCc%10c(Cl)cccc%109)CC8)cc7Oc7cnc8[nH]ccc8c7)cc5[N+](=O)[O-])C6)CC4)cc3C2=O)C(=O)N1	C63H68ClN11O10S	BCL2L1	Q07817	CRBN	WO-2024078581-A1
TPD-S6ZZTH	WO2024078581A1_P-055	.	O=C1CCC(N2C(=O)c3cccc(OCCn4cc(CN5CCC6(CC5)CC(CNc5ccc(S(=O)(=O)NC(=O)c7ccc(N8CCN([C@@H]9CCCCc%10c(Cl)cccc%109)CC8)cc7Oc7cnc8[nH]ccc8c7)cc5[N+](=O)[O-])C6)nn4)c3C2=O)C(=O)N1	C62H64ClN13O11S	BCL2L1	Q07817	CRBN	WO-2024078581-A1
TPD-KEO9WX	WO2024078581A1_P-056	.	CC(=O)NC(CCN1CCC2(CC1)CC(CNc1ccc(S(=O)(=O)NC(=O)c3ccc(N4CCN([C@@H]5CCCCc6c(Cl)cccc65)CC4)cc3Oc3cnc4[nH]ccc4c3)cc1[N+](=O)[O-])C2)COc1ccc2c(c1)C(=O)N(C1CCC(=O)NC1=O)C2=O	C63H68ClN11O12S	BCL2L1	Q07817	CRBN	WO-2024078581-A1
TPD-IR9H21	WO2024078581A1_P-057	.	O=C1CCC(N2C(=O)c3ccc(N4CCC(N5CCC6(CC5)CC(CNc5ccc(S(=O)(=O)NC(=O)c7ccc(N8CCN([C@@H]9CCCCc%10c(Cl)cccc%109)CC8)cc7Oc7cnc8[nH]ccc8c7)cc5NOO)C6)CC4)cc3C2=O)C(=O)N1	C62H68ClN11O10S	BCL2L1	Q07817	CRBN	WO-2024078581-A1
TPD-NIPGWB	WO2024078581A1_P-058	.	O=C1CCC(N2C(=O)c3ccc(N4CC(N5CCC(N6CCC7(CC6)CC(CNc6ccc(S(=O)(=O)NC(=O)c8ccc(N9CCN([C@@H]%10CCCCc%11c(Cl)cccc%11%10)CC9)cc8Oc8cnc9[nH]ccc9c8)cc6NOO)C7)CC5)C4)cc3C2=O)C(=O)N1	C65H73ClN12O10S	BCL2L1	Q07817	CRBN	WO-2024078581-A1
TPD-IRCUF2	WO2024078581A1_P-059	.	O=C1CCC(N2Cc3c(OC[C@H]4CC[C@@H](CN5CCC6(CC5)CC(CNc5ccc(S(=O)(=O)NC(=O)c7ccc(N8CCN([C@@H]9CCCCc%10c(Cl)cccc%109)CC8)cc7Oc7cnc8[nH]ccc8c7)cc5NOO)C6)C4)cccc3C2=O)C(=O)N1	C64H73ClN10O10S	BCL2L1	Q07817	CRBN	WO-2024078581-A1
TPD-SZW04S	WO2024078581A1_P-060	.	O=C1CCC(N2Cc3c(NC[C@H]4CC[C@H](CN5CCC6(CC5)CC(CNc5ccc(S(=O)(=O)NC(=O)c7ccc(N8CCN([C@@H]9CCCCc%10c(Cl)cccc%109)CC8)cc7Oc7cnc8[nH]ccc8c7)cc5NOO)C6)CC4)cccc3C2=O)C(=O)N1	C65H76ClN11O9S	BCL2L1	Q07817	CRBN	WO-2024078581-A1
TPD-88TCWX	WO2024078581A1_P-061	.	O=C1CCC(N2C(=O)c3ccc(N4CC(N5CC(N6CCC7(CC6)CC(CNc6ccc(S(=O)(=O)NC(=O)c8ccc(N9CCN([C@@H]%10CCCCc%11c(Cl)cccc%11%10)CC9)cc8Oc8cnc9[nH]ccc9c8)cc6NOO)C7)C5)C4)cc3C2=O)C(=O)N1	C63H69ClN12O10S	BCL2L1	Q07817	CRBN	WO-2024078581-A1
TPD-OOMIUU	WO2024083255A1_2	.	COC1=CC2=NC(C)=NC(NCC3=CC(C4=C(CN)C=CC=C4)=CS3)=C2C=C1C1CCC(C(=O)N2CCC(CCOCC3CCN(C(=O)C4=CC=C(Cl)C(N5CCC(=O)NC5=O)=C4)CC3)CC2)CC1	C53H63ClN8O6S	SOS1	Q07889	CRBN	WO-2024083255-A1
TPD-BHFA5L	WO2024083255A1_4	.	CNCC1=C(C2=CSC([C@@H](C)NC3=C4C=C(C5CCC(C(=O)N6CCN(CC7CCC8(CC7)CCN(C(=O)C7=CC=C(C9CCC(=O)NC9=O)C=C7)CC8)CC6)CC5)C(OC)=CC4=NC(C)=N3)=C2)C=CC=C1	C58H72N8O5S	SOS1	Q07889	CRBN	WO-2024083255-A1
TPD-TL6U2B	WO2024083255A1_6	.	COC1=CC2=NC(C)=NC(N[C@H](C)C3=CC(C4=C(CN(C)C)C=CC=C4Cl)=CS3)=C2C=C1[C@H]1CC[C@H](C(=O)N2CCC(COCCN3CCN(C(=O)C4=CC=C(Cl)C(N5CCC(=O)NC5=O)=C4)CC3)CC2)CC1	C55H67Cl2N9O6S	SOS1	Q07889	CRBN	WO-2024083255-A1
TPD-9AY45I	WO2024083255A1_7	.	COC1=CC2=NC(C)=NC(N[C@H](C)C3=CC(N)=CC(C(F)(F)F)=C3)=C2C=C1C1CCC(C(=O)N2CCN(CCCC3CCN(C4=CC(N5CCC(=O)NC5=O)=C(Cl)C=C4)CC3)CC2)CC1	C48H59ClF3N9O4	SOS1	Q07889	CRBN	WO-2024083255-A1
TPD-HK1OWP	WO2024083255A1_8	.	COC1=CC2=NC(C)=NC(N[C@H](C)C3=CC(C4=C(CN(C)C)C=CC=C4Cl)=CS3)=C2C=C1C1CCC(C(=O)N2CCC(OCCCN3CCN(C(=O)C4=CC=C(Cl)C(N5CCC(=O)NC5=O)=C4)CC3)CC2)CC1	C55H67Cl2N9O6S	SOS1	Q07889	CRBN	WO-2024083255-A1
TPD-VGZDT9	WO2024083255A1_9	.	COC1=CC2=NC(C)=NC(N[C@H](C)C3=CC=CC(C#N)=C3C)=C2C=C1C1CCC(C(=O)N2CCN(CC3CCC4(CC3)CCN(C(=O)C3=CC(N5CCC(=O)NC5=O)=C(Cl)C=C3)CC4)CC2)CC1	C53H64ClN9O5	SOS1	Q07889	CRBN	WO-2024083255-A1
TPD-JF64R2	WO2024083255A1_10	.	CCCC(CCCC(=O)N1CCC(CCOC(C)(C)C2CCN(C(=O)C3=CC=C(Cl)C(N4CCC(=O)NC4=O)=C3)CC2)CC1)C1=CC2=C(N[C@H](C)C3=CC(C4=C(CN(C)C)C=CC=C4Cl)=CS3)N=C(C)N=C2C=C1OC	C59H76Cl2N8O6S	SOS1	Q07889	CRBN	WO-2024083255-A1
TPD-LLMB7G	WO2024083255A1_11	.	COC1=CC2=NC(C)=NC(N[C@H](C)C3=CC(N)=CC(C(F)(F)F)=C3)=C2C=C1C1CCC(C(=O)N2CCC(CCOC(C)(C)C3CCN(C(=O)C4=CC=C(Cl)C(N5CCC(=O)NC5=O)=C4)CC3)CC2)CC1	C52H64ClF3N8O6	SOS1	Q07889	CRBN	WO-2024083255-A1
TPD-3WN5F0	WO2024083255A1_13	.	CC1=NC(N[C@H](C)C2=CC(N)=CC(C(F)(F)F)=C2)=C2C=C(C3CCC(C(=O)N4CCN(CCCOC5CCN(C(=O)C6=CC=C(Cl)C(N7CCC(=O)NC7=O)=C6)CC5)CC4)CC3)C(O)=CC2=N1	C48H57ClF3N9O6	SOS1	Q07889	CRBN	WO-2024083255-A1
TPD-M2618D	PROTAC SOS1 degrader-8	PROTAC SOS1 degrader-8; orb2564655; HY-161634; CS-1054675; 3036155-11-7	Cc1c(C#N)cccc1[C@@H](C)Nc1nnc(C)c2cnc(N3CCN(C(=O)C4CCN(CC5CCC6(CC5)CCN(C(=O)c5ccc(Cl)c(N7CCC(=O)NC7=O)c5)CC6)CC4)CC3)cc12	C50H60ClN11O4	SOS1	Q07889	CRBN	WO-2024083257-A1
TPD-F3H2B8	PROTAC SOS1 degrader-9	PROTAC SOS1 degrader-9; orb2564535; HY-161636; CS-1054689; 3036155-21-9	Cc1ccc(C(=O)N2CCC3(CCC(CN4CCC(C(=O)N5CCN(c6cc7c(N[C@H](C)c8cccc(C#N)c8C)nnc(C)c7cn6)CC5)CC4)CC3)CC2)cc1N1CCC(=O)NC1=O	C51H63N11O4	SOS1	Q07889	CRBN	WO-2024083257-A1
TPD-L1YR8M	WO2024083257A1_11	.	COc1ccc(C(=O)N2CCC3(CCC(CN4CCC(C(=O)N5CCN(c6cc7c(N[C@H](C)c8cccc(C#N)c8C)nnc(C)c7cn6)CC5)CC4)CC3)CC2)cc1N1CCC(=O)NC1=O	C51H63N11O5	SOS1	Q07889	CRBN	WO-2024083257-A1
TPD-6FJ2CH	WO2024083257A1_12	.	Cc1c(C(F)F)cccc1[C@@H](C)Nc1nnc(C)c2cnc([C@H]3CC[C@H](C(=O)N4CCN(CC5CCC6(CC5)CCN(C(=O)c5ccc(Cl)c(N7CCC(=O)NC7=O)c5)CC6)CC4)CC3)cc12	C51H62ClF2N9O4	SOS1	Q07889	CRBN	WO-2024083257-A1
TPD-5AC673	WO2024083257A1_13	.	COc1ccc(C(=O)N2CCC3(CCC(CN4CCN(C(=O)[C@H]5CC[C@H](c6cc7c(N[C@H](C)c8cccc(C#N)c8C)nnc(C)c7cn6)CC5)CC4)CC3)CC2)cc1N1CCC(=O)NC1=O	C52H64N10O5	SOS1	Q07889	CRBN	WO-2024083257-A1
TPD-Y4ZBFR	WO2024083257A1_14	.	Cc1ccc(C(=O)N2CCC3(CCN(CC4CCN(C(=O)N5CCN(c6cc7c(N[C@H](C)c8cccc(C#N)c8C)nnc(C)c7cn6)CC5)CC4)CC3)CC2)cc1N1CCC(=O)NC1=O	C50H62N12O4	SOS1	Q07889	CRBN	WO-2024083257-A1
TPD-ADMWS5	PROTAC SOS1 degrader-7	PROTAC SOS1 degrader-7; orb2564451; HY-163582; CS-1054101; 3036155-26-4	Cc1ccc(C(=O)N2CCC3(CCC(CN4CCC(C(=O)N5CCN(c6cc7c(N[C@H](C)c8cccc(C(F)F)c8C)nnc(C)c7cn6)CC5)CC4)CC3)CC2)cc1N1CCC(=O)NC1=O	C51H64F2N10O4	SOS1	Q07889	CRBN	WO-2024083257-A1
TPD-JC5RRE	SCHEMBL30931904	1-[2-chloro-5-[9-[[4-[4-[1-[[(1R)-1-[3-(difluoromethyl)-2-methylphenyl]ethyl]amino]-4-methylpyrido[3,4-d]pyridazin-7-yl]piperazine-1-carbonyl]cyclohexyl]methyl]-3,9-diazaspiro[5.5]undecane-3-carbonyl]phenyl]-1,3-diazinane-2,4-dione	Cc1c(C(F)F)cccc1[C@@H](C)Nc1nnc(C)c2cnc(N3CCN(C(=O)[C@H]4CC[C@H](CN5CCC6(CC5)CCN(C(=O)c5ccc(Cl)c(N7CCC(=O)NC7=O)c5)CC6)CC4)CC3)cc12	C50H61ClF2N10O4	SOS1	Q07889	CRBN	WO-2024083257-A1
TPD-Y5PIFG	WO2024083257A1_17	.	Cc1c(C#N)cccc1[C@@H](C)Nc1nnc(C)c2cnc(N3CCN(C(=O)C4CCN(CC5CCC6(CC5)CCN(C(=O)c5ccc7c(c5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC6)CC4)CC3)cc12	C53H61N11O6	SOS1	Q07889	CRBN	WO-2024083257-A1
TPD-9JCXP6	WO2024083257A1_18	.	Cc1c(C#N)cccc1[C@@H](C)Nc1nnc(C)c2cnc(N3CCN(C(=O)N4CCC(CCOCC5CCN(C(=O)c6ccc(Cl)c(N7CCC(=O)NC7=O)c6)CC5)CC4)CC3)cc12	C47H56ClN11O5	SOS1	Q07889	CRBN	WO-2024083257-A1
TPD-S6V4QP	WO2024083257A1_19	.	Cc1c(C#N)cccc1[C@@H](C)Nc1nnc(C)c2cnc(C3CCN(C(=O)C4CCN(CCCCC5CCN(C(=O)c6ccc(Cl)c(N7CCC(=O)NC7=O)c6)CC5)CC4)CC3)cc12	C49H59ClN10O4	SOS1	Q07889	CRBN	WO-2024083257-A1
TPD-2XMXAX	WO2024083257A1_2	.	Cc1c(C#N)cccc1[C@@H](C)Nc1nnc(C)c2cnc(N3CCC(C(=O)N4CCC(CCOCC5CCN(C(=O)c6ccc(Cl)c(N7CCC(=O)NC7=O)c6)CC5)CC4)CC3)cc12	C48H57ClN10O5	SOS1	Q07889	CRBN	WO-2024083257-A1
TPD-D49XJN	WO2024083257A1_20	.	Cc1c(C#N)cccc1[C@@H](C)Nc1nnc(C)c2cnc(C3CCN(C(=O)C4CCN(CC5CCC6(CC5)CCN(C(=O)c5ccc(Cl)c(N7CCC(=O)NC7=O)c5)CC6)CC4)CC3)cc12	C51H61ClN10O4	SOS1	Q07889	CRBN	WO-2024083257-A1
TPD-342J7E	WO2024083257A1_21	.	Cc1ccc(C(=O)N2CCC3(CCC(CN4CCN(C(=O)[C@H]5CC[C@H](c6cc7c(N[C@H](C)c8cccc(C#N)c8C)nnc(C)c7cn6)CC5)CC4)CC3)CC2)cc1N1CCC(=O)NC1=O	C52H64N10O4	SOS1	Q07889	CRBN	WO-2024083257-A1
TPD-RGZ130	WO2024083257A1_22	.	Cc1c(C#N)cccc1[C@@H](C)Nc1nnc(C)c2cnc(N3CCN(C(=O)C4CCN(CC5CCC6(CC5)CCN(C(=O)c5ccc(F)c(N7CCC(=O)NC7=O)c5)CC6)CC4)CC3)cc12	C50H60FN11O4	SOS1	Q07889	CRBN	WO-2024083257-A1
TPD-45A76F	WO2024083257A1_23	1-[4-[9-[[4-[4-[1-[[(1R)-1-[3-(difluoromethyl)-2-methylphenyl]ethyl]amino]-4-methylpyrido[3,4-d]pyridazin-7-yl]piperazine-1-carbonyl]piperidin-1-yl]methyl]-3-azaspiro[5.5]undecane-3-carbonyl]phenyl]-1,3-diazinane-2,4-dione	Cc1c(C(F)F)cccc1[C@@H](C)Nc1nnc(C)c2cnc(N3CCN(C(=O)C4CCN(CC5CCC6(CC5)CCN(C(=O)c5ccc(N7CCC(=O)NC7=O)cc5)CC6)CC4)CC3)cc12	C50H62F2N10O4	SOS1	Q07889	CRBN	WO-2024083257-A1
TPD-7YRZY6	WO2024083257A1_24	.	Cc1c(C#N)cccc1[C@@H](C)Nc1nnc(C)c2cnc(N3CCN(C(=O)C4CCN(CC5CCC6(CC5)CCN(C(=O)c5ccc(C(F)(F)F)c(N7CCC(=O)NC7=O)c5)CC6)CC4)CC3)cc12	C51H60F3N11O4	SOS1	Q07889	CRBN	WO-2024083257-A1
TPD-4POGLN	WO2024083257A1_25	.	Cc1c(C#N)cccc1[C@@H](C)Nc1nnc(C)c2cnc(N3CCN(C(=O)C4CCN(CC5CCC6(CC5)CCN(C(=O)c5ccc(OC(F)(F)F)c(N7CCC(=O)NC7=O)c5)CC6)CC4)CC3)cc12	C51H60F3N11O5	SOS1	Q07889	CRBN	WO-2024083257-A1
TPD-UBGLUH	WO2024083257A1_26	.	Cc1c(C#N)cccc1[C@@H](C)Nc1nnc(C)c2cnc(N3CCC(C(=O)C4CCN(CCCCC5CCN(C(=O)c6ccc(Cl)c(N7CCC(=O)NC7=O)c6)CC5)CC4)CC3)cc12	C49H59ClN10O4	SOS1	Q07889	CRBN	WO-2024083257-A1
TPD-RPGJQN	WO2024083257A1_27	.	Cc1c(C#N)cccc1[C@@H](C)Nc1nnc(C)c2cnc(N3CCN(C(=O)C4CCN(CC5CCC6(CC5)CCN(C(=O)c5ccc(Br)c(N7CCC(=O)NC7=O)c5)CC6)CC4)CC3)cc12	C50H60BrN11O4	SOS1	Q07889	CRBN	WO-2024083257-A1
TPD-JGK8IB	WO2024083257A1_28	.	CCc1ccc(C(=O)N2CCC3(CCC(CN4CCC(C(=O)N5CCN(c6cc7c(N[C@H](C)c8cccc(C#N)c8C)nnc(C)c7cn6)CC5)CC4)CC3)CC2)cc1N1CCC(=O)NC1=O	C52H65N11O4	SOS1	Q07889	CRBN	WO-2024083257-A1
TPD-TW7GED	WO2024083257A1_29	.	Cc1c(C#N)cccc1[C@@H](C)Nc1nnc(C)c2cnc(N3CC4CCC(C3)N4C(=O)C3CCN(CC4CCC5(CC4)CCN(C(=O)c4ccc(Cl)c(N6CCC(=O)NC6=O)c4)CC5)CC3)cc12	C52H62ClN11O4	SOS1	Q07889	CRBN	WO-2024083257-A1
TPD-3A4UXW	WO2024083257A1_3	.	Cc1c(C#N)cccc1[C@@H](C)Nc1nnc(C)c2cnc(N3CCN(C(=O)C4CCN(CCCCN5CCN(C(=O)c6ccc(Cl)c(N7CCC(=O)NC7=O)c6)CC5)CC4)CC3)cc12	C47H57ClN12O4	SOS1	Q07889	CRBN	WO-2024083257-A1
TPD-ADRPD5	WO2024083257A1_30	.	Cc1c(C#N)cccc1[C@@H](C)Nc1nnc(C)c2cnc(N3CC4CC(C3)N4C(=O)C3CCN(CC4CCC5(CC4)CCN(C(=O)c4ccc(Cl)c(N6CCC(=O)NC6=O)c4)CC5)CC3)cc12	C51H60ClN11O4	SOS1	Q07889	CRBN	WO-2024083257-A1
TPD-WKWA6K	WO2024083257A1_31	.	Cc1ccc(C(=O)N2CCC3(CCC(CN4CCC(C(=O)N5CCN(c6cc7c(N[C@H](C)c8cccc9c8CCS9(=O)=O)nnc(C)c7cn6)CC5)CC4)CC3)CC2)cc1N1CCC(=O)NC1=O	C51H64N10O6S	SOS1	Q07889	CRBN	WO-2024083257-A1
TPD-PXYQMZ	WO2024083257A1_32	.	Cc1c(C#N)cccc1[C@@H](C)Nc1nnc(C)c2cnc(N3CCN(C(=O)C4CCN(CC5CCC6(CC5)CCN(C(=O)c5ccc7c(c5)C(=O)N(C5CCC(=O)NC5=O)C7)CC6)CC4)CC3)cc12	C53H63N11O5	SOS1	Q07889	CRBN	WO-2024083257-A1
TPD-JGZEJF	WO2024083257A1_33	.	Cc1nnc(N[C@H](C)c2cccc3c2CCS3(=O)=O)c2cc(N3CCN(C(=O)C4CCN(CC5CCC6(CC5)CCN(C(=O)c5ccc(Cl)c(N7CCC(=O)NC7=O)c5)CC6)CC4)CC3)ncc12	C50H61ClN10O6S	SOS1	Q07889	CRBN	WO-2024083257-A1
TPD-J4LU36	WO2024083257A1_34	1-[2-chloro-5-[9-[[4-[4-[4-methyl-1-[[(1R)-1-[2-methyl-3-(trifluoromethyl)phenyl]ethyl]amino]pyrido[3,4-d]pyridazin-7-yl]piperazine-1-carbonyl]piperidin-1-yl]methyl]-3-azaspiro[5.5]undecane-3-carbonyl]phenyl]-1,3-diazinane-2,4-dione	Cc1c([C@@H](C)Nc2nnc(C)c3cnc(N4CCN(C(=O)C5CCN(CC6CCC7(CC6)CCN(C(=O)c6ccc(Cl)c(N8CCC(=O)NC8=O)c6)CC7)CC5)CC4)cc23)cccc1C(F)(F)F	C50H60ClF3N10O4	SOS1	Q07889	CRBN	WO-2024083257-A1
TPD-2UWKAM	WO2024083257A1_35	.	Cc1c(C#N)cccc1[C@@H](C)Nc1nnc(C)c2cnc(N3CCC(C(=O)C4CCN(CC5CCC6(CC5)CCN(C(=O)c5ccc(Cl)c(N7CCC(=O)NC7=O)c5)CC6)CC4)CC3)cc12	C51H61ClN10O4	SOS1	Q07889	CRBN	WO-2024083257-A1
TPD-I8X4AY	WO2024083257A1_38	.	Cc1c(C#N)cccc1[C@@H](C)NC1=NNC(C)c2cnc(N3CCC(C(=O)C4CCN(CCCCC5CCN(C(=O)c6ccc(Cl)c(N7CCC(=O)NC7=O)c6)CC5)CC4)CC3)cc21	C49H61ClN10O4	SOS1	Q07889	CRBN	WO-2024083257-A1
TPD-780HCL	WO2024083257A1_4	.	Cc1ccc(C(=O)N2CCC3(CCC(CCN4CCC(C(=O)N5CCN(c6cc7c(N[C@H](C)c8cccc(C#N)c8C)nnc(C)c7cn6)CC5)CC4)CC3)CC2)cc1N1CCC(=O)NC1=O	C52H65N11O4	SOS1	Q07889	CRBN	WO-2024083257-A1
TPD-WFMEAL	WO2024083257A1_43	.	Cc1c(C#N)cccc1[C@@H](C)Nc1nnc(C)c2cnc(C3CCN(C(=O)C4CCN(CCOCC5CCN(C(=O)c6ccc(Cl)c(N7CCC(=O)NC7=O)c6)CC5)CC4)CC3)cc12	C48H57ClN10O5	SOS1	Q07889	CRBN	WO-2024083257-A1
TPD-O648GQ	WO2024083257A1_44	.	Cc1c(C#N)cccc1[C@@H](C)Nc1nnc(C)c2cnc(C3CCC(C(=O)N4CCN(CC5CCC6(CC5)CCN(C(=O)c5ccc(Br)c(N7CCC(=O)NC7=O)c5)CC6)CC4)CC3)cc12	C51H61BrN10O4	SOS1	Q07889	CRBN	WO-2024083257-A1
TPD-6ZK1K0	WO2024083257A1_45	1-[5-[9-[[4-[4-[1-[[(1R)-1-[3-amino-5-(trifluoromethyl)phenyl]ethyl]amino]-4-methylpyrido[3,4-d]pyridazin-7-yl]piperazine-1-carbonyl]piperidin-1-yl]methyl]-3-azaspiro[5.5]undecane-3-carbonyl]-2-methoxyphenyl]-1,3-diazinane-2,4-dione	COc1ccc(C(=O)N2CCC3(CCC(CN4CCC(C(=O)N5CCN(c6cc7c(N[C@H](C)c8cc(N)cc(C(F)(F)F)c8)nnc(C)c7cn6)CC5)CC4)CC3)CC2)cc1N1CCC(=O)NC1=O	C50H62F3N11O5	SOS1	Q07889	CRBN	WO-2024083257-A1
TPD-Q4VEM7	WO2024083257A1_46	.	Cc1c(C#N)cccc1[C@@H](C)Nc1nnc(C)c2cnc(N3CC4CC3CN4C(=O)C3CCN(CC4CCC5(CC4)CCN(C(=O)c4ccc(Cl)c(N6CCC(=O)NC6=O)c4)CC5)CC3)cc12	C51H60ClN11O4	SOS1	Q07889	CRBN	WO-2024083257-A1
TPD-V9HRTK	WO2024083257A1_47	.	Cc1ccc(C(=O)N2CCC3(CCC(CN4CCC(C(=O)C5CCN(c6cc7c(N[C@H](C)c8cccc9c8CCS9(=O)=O)nnc(C)c7cn6)CC5)CC4)CC3)CC2)cc1N1CCC(=O)NC1=O	C52H65N9O6S	SOS1	Q07889	CRBN	WO-2024083257-A1
TPD-4T2SEJ	WO2024083257A1_48	.	Cc1ccc(C(=O)N2CCC3(CCC(CN4CCN(C(=O)[C@H]5CC[C@H](c6cc7c(N[C@H](C)c8cccc9c8CCS9(=O)=O)nnc(C)c7cn6)CC5)CC4)CC3)CC2)cc1N1CCC(=O)NC1=O	C52H65N9O6S	SOS1	Q07889	CRBN	WO-2024083257-A1
TPD-S1TIRT	WO2024083257A1_49	.	Cc1c(C#N)cccc1[C@@H](C)Nc1nnc(C)c2cnc(OCC3(CN4CCN(CC5CCC6(CC5)CCN(C(=O)c5ccc(Cl)c(N7CCC(=O)NC7=O)c5)CC6)CC4)CC3)cc12	C49H59ClN10O4	SOS1	Q07889	CRBN	WO-2024083257-A1
TPD-EYJ6D9	WO2024083257A1_5-A	.	Cc1c(C#N)cccc1[C@@H](C)Nc1nnc(C)c2cnc([C@H]3CC[C@H](C(=O)N4CCC(CCOCC5CCN(C(=O)c6ccc(Cl)c(N7CCC(=O)NC7=O)c6)CC5)CC4)CC3)cc12	C49H58ClN9O5	SOS1	Q07889	CRBN	WO-2024083257-A1
TPD-VRLNY3	WO2024083257A1_5-B	.	Cc1c(C#N)cccc1[C@@H](C)Nc1nnc(C)c2cnc([C@H]3CC[C@@H](C(=O)N4CCC(CCOCC5CCN(C(=O)c6ccc(Cl)c(N7CCC(=O)NC7=O)c6)CC5)CC4)CC3)cc12	C49H58ClN9O5	SOS1	Q07889	CRBN	WO-2024083257-A1
TPD-BMG3K0	WO2024083257A1_50	.	Cc1c(C#N)cccc1[C@@H](C)Nc1nnc(C)c2cnc(OCC3(CN4CCN(CCC5CCC6(CC5)CCN(C(=O)c5ccc(Cl)c(N7CCC(=O)NC7=O)c5)CC6)CC4)CC3)cc12	C50H61ClN10O4	SOS1	Q07889	CRBN	WO-2024083257-A1
TPD-AZW1TD	WO2024083257A1_51	.	Cc1c(C#N)cccc1[C@@H](C)Nc1nnc(C)c2cnc(SCC3(CN4CCN(CCC5CCC6(CC5)CCN(C(=O)c5ccc(Cl)c(N7CCC(=O)NC7=O)c5)CC6)CC4)CC3)cc12	C50H61ClN10O3S	SOS1	Q07889	CRBN	WO-2024083257-A1
TPD-MASG9L	WO2024083257A1_52	.	Cc1c(C#N)cccc1[C@@H](C)Nc1nnc(C)c2cnc(NCC3(CN4CCN(CCC5CCC6(CC5)CCN(C(=O)c5ccc(Cl)c(N7CCC(=O)NC7=O)c5)CC6)CC4)CC3)cc12	C50H62ClN11O3	SOS1	Q07889	CRBN	WO-2024083257-A1
TPD-XESN2T	WO2024083257A1_53	.	Cc1c(C#N)cccc1[C@@H](C)Nc1nnc(C)c2cnc(OCC3(CN4CCN(CCCC5CCN(C(=O)c6ccc(Cl)c(N7CCC(=O)NC7=O)c6)CC5)CC4)CC3)cc12	C46H55ClN10O4	SOS1	Q07889	CRBN	WO-2024083257-A1
TPD-OV7BUJ	WO2024083257A1_54	.	Cc1c(C#N)cccc1[C@@H](C)Nc1nnc(C)c2cnc(OCC3(CN4CCN(CCCCC5CCN(C(=O)c6ccc(Cl)c(N7CCC(=O)NC7=O)c6)CC5)CC4)CC3)cc12	C47H57ClN10O4	SOS1	Q07889	CRBN	WO-2024083257-A1
TPD-ERBSX3	WO2024083257A1_55	.	Cc1c(C#N)cccc1[C@@H](C)Nc1nnc(C)c2cnc(OCC3(CN4CCN(CCCC5CCC6(CC5)CCN(C(=O)c5ccc(Cl)c(N7CCC(=O)NC7=O)c5)CC6)CC4)CC3)cc12	C51H63ClN10O4	SOS1	Q07889	CRBN	WO-2024083257-A1
TPD-Q9VMEO	WO2024083257A1_6	.	Cc1c(C#N)cccc1[C@@H](C)Nc1nnc(C)c2cnc(N3CCN(C(=O)C4CCN(CCCCC5CCN(C(=O)c6ccc(Cl)c(N7CCC(=O)NC7=O)c6)CC5)CC4)CC3)cc12	C48H58ClN11O4	SOS1	Q07889	CRBN	WO-2024083257-A1
TPD-5RMR2U	WO2024083257A1_7	.	Cc1c(C#N)cccc1[C@@H](C)Nc1nnc(C)c2cnc(N3CCN(C(=O)C4CCN(CCCC5CCN(C(=O)c6ccc(Cl)c(N7CCC(=O)NC7=O)c6)CC5)CC4)CC3)cc12	C47H56ClN11O4	SOS1	Q07889	CRBN	WO-2024083257-A1
TPD-ZOV2GX	WO2024083257A1_8	.	Cc1c(C#N)cccc1[C@@H](C)Nc1nnc(C)c2cnc(C3=CCC(C(=O)N4CCC(CCOCC5CCN(C(=O)c6ccc(Cl)c(N7CCC(=O)NC7=O)c6)CC5)CC4)CC3)cc12	C49H56ClN9O5	SOS1	Q07889	CRBN	WO-2024083257-A1
TPD-1U6VVJ	WO2024083257A1_9	.	Cc1nnc(N[C@H](C)c2cc(-c3c(Cl)cccc3CN(C)C)cs2)c2cc([C@H]3CC[C@H](C(=O)N4CCC(CCOCC5CCN(C(=O)c6ccc(Cl)c(N7CCC(=O)NC7=O)c6)CC5)CC4)CC3)ncc12	C54H65Cl2N9O5S	SOS1	Q07889	CRBN	WO-2024083257-A1
TPD-8HML69	WO2024094171A1_1	.	COc1cc(N2CCN(C(=O)CN3CCC(c4ccc(NC5CCC(=O)NC5=O)cc4)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCn1cc-2cn1	C48H57BrN12O7S	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-PDLAHQ	WO2024094171A1_10	.	COc1cc(N2CCC3(CC2)CN(CC2CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC2)C3)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCn1cc-2cn1	C52H59BrN12O8S	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-R8DAYV	WO2024094171A1_11	.	COc1cc(N2CCC(N3CCN(CC4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCn1cc-2cn1	C54H64BrN13O8S	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-6VIQN7	WO2024094171A1_12	.	COc1cc(N2CCC(N3CCN(C(=O)[C@H](C)Nc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCn1cc-2cn1	C51H58BrN13O9S	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-4N31QX	WO2024094171A1_13-1	.	COc1cc(N2CCC(CN3CCN(c4ccc5c(c4)C(=O)N([C@H]4CCC(=O)NC4=O)C5=O)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCn1cc-2cn1	C49H55BrN12O8S	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-8LG73Y	WO2024094171A1_13-2	.	COc1cc(N2CCC(CN3CCN(c4ccc5c(c4)C(=O)N([C@@H]4CCC(=O)NC4=O)C5=O)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCn1cc-2cn1	C49H55BrN12O8S	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-MO464E	WO2024094171A1_13	.	COc1cc(N2CCC(CN3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCn1cc-2cn1	C49H55BrN12O8S	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-RKOYRY	WO2024094171A1_14	.	COc1cc(N2CCC(CN3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C1CC1)S(C)(=O)=O)OCCCCn1cc-2cn1	C51H57BrN12O8S	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-C0KPWD	WO2024094171A1_15	.	COc1cc(N2CCN(CC3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C1CC1)S(C)(=O)=O)OCCCCn1cc-2cn1	C51H57BrN12O8S	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-BCB2LT	WO2024094171A1_16	.	COc1cc(N2CCN(CC3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)c2cc1Nc1ncc(Cl)c(n1)Nc1ccc(cc1N(C1CC1)S(C)(=O)=O)OCCCCn1cc-2cn1	C51H57ClN12O8S	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-TWQM33	WO2024094171A1_19-1	.	COc1cc(N2CCC(CN3CCN(c4ccc5c(c4)C(=O)N([C@H]4CCC(=O)NC4=O)C5=O)CC3)CC2)c2cc1Nc1ncc(Cl)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCn1cc-2cn1	C49H55ClN12O8S	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-Q39VMT	WO2024094171A1_19	.	COc1cc(N2CCC(CN3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)c2cc1Nc1ncc(Cl)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCn1cc-2cn1	C49H55ClN12O8S	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-GSV7O8	WO2024094171A1_2	.	COc1cc(N2CCN(C(=O)CN3CCC(c4ccc(NC5CCC(=O)NC5=O)cc4)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCn1cc-2cn1	C47H55BrN12O7S	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-8WYBH4	WO2024094171A1_20-1	.	COc1cc(N2CCC(CN3CCN(c4ccc5c(c4)C(=O)N([C@H]4CCC(=O)NC4=O)C5=O)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1P(C)(C)=O)OCCCCn1cc-2cn1	C49H55BrN11O7P	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-DL8WHK	WO2024094171A1_20	.	COc1cc(N2CCC(CN3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1P(C)(C)=O)OCCCCn1cc-2cn1	C49H55BrN11O7P	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-ABXOL7	WO2024094171A1_21	.	COc1cc(N2CCC(CN3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)c2cc1Nc1ncc(Cl)c(n1)Nc1ccc(cc1P(C)(C)=O)OCCCCn1cc-2cn1	C49H55ClN11O7P	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-TG89SX	WO2024094171A1_22	.	COc1cc(N2CCC(CN3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCCn1cc-2cn1	C50H57BrN12O8S	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-OPO64J	WO2024094171A1_23-1	.	COc1cc(N2CCC(CN3CCN(c4ccc5c(C6CCC(=O)NC6=O)nn(C)c5c4)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCn1cc-2cn1	C49H58BrN13O6S	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-HTN6SI	WO2024094171A1_23-2	.	COc1cc(N2CCC(CN3CCN(c4ccc5c([C@H]6CCC(=O)NC6=O)nn(C)c5c4)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCn1cc-2cn1	C49H58BrN13O6S	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-LF3346	WO2024094171A1_24-1	.	COc1cc(N2CCC(CN3CCN(c4cc5c(cc4F)c([C@@H]4CCC(=O)NC4=O)nn5C)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCn1cc-2cn1	C49H57BrFN13O6S	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-M5T0BF	WO2024094171A1_24-2	.	COc1cc(N2CCC(CN3CCN(c4cc5c(cc4F)c([C@H]4CCC(=O)NC4=O)nn5C)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCn1cc-2cn1	C49H57BrFN13O6S	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-0NZMOU	WO2024094171A1_24	.	COc1cc(N2CCC(CN3CCN(c4cc5c(cc4F)c(C4CCC(=O)NC4=O)nn5C)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCn1cc-2cn1	C49H57BrFN13O6S	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-UWJSLX	WO2024094171A1_25	.	COc1cc(N2CCC(CN3CCC(c4ccc5c(C6CCC(=O)NC6=O)nn(C)c5c4)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCn1cc-2cn1	C50H59BrN12O6S	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-6D1WN8	WO2024094171A1_26	.	COc1cc(N2CCC(CN3CCN(c4ccc5c(N6CCC(=O)NC6=O)nn(C)c5c4)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCn1cc-2cn1	C48H57BrN14O6S	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-1XWBPQ	WO2024094171A1_27	.	COc1cc(N2CCC(CN3CCC(c4ccc5c(N6CCC(=O)NC6=O)nn(C)c5c4)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCn1cc-2cn1	C49H58BrN13O6S	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-JS7B2T	WO2024094171A1_28	.	COc1cc(N2CCC(CN3CCC(c4ccc5c(N6CCC(=O)NC6=O)nn(C)c5c4)C(F)(F)C3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCn1cc-2cn1	C49H56BrF2N13O6S	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-U28I4A	WO2024094171A1_29	.	COc1cc(N2CCC(CN3CCN(c4ccc5c(c4)n(C)c(=O)n5C4CCC(=O)NC4=O)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCn1cc-2cn1	C49H58BrN13O7S	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-AXRTY0	WO2024094171A1_3	.	COc1cc(N2CCN(C(=O)CN3CCC(c4ccc(NC5CCC(=O)NC5=O)cc4)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCCn1cc-2cn1	C49H59BrN12O7S	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-CEC3TM	WO2024094171A1_30	.	COc1cc(N2CCC(CN3CCC(c4ccc5c(c4)n(C)c(=O)n5C4CCC(=O)NC4=O)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCn1cc-2cn1	C50H59BrN12O7S	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-5RFGNA	WO2024094171A1_31-1	.	COc1cc(N2CCC(CN3CC[C@@H](c4ccc5c(N6CCC(=O)NC6=O)nn(C)c5c4)C(F)(F)C3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1P(C)(C)=O)OCCCCn1cc-2cn1	C49H56BrF2N12O5P	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-2MMF0M	WO2024094171A1_31-2	.	COc1cc(N2CCC(CN3CC[C@H](c4ccc5c(N6CCC(=O)NC6=O)nn(C)c5c4)C(F)(F)C3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1P(C)(C)=O)OCCCCn1cc-2cn1	C49H56BrF2N12O5P	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-MA3RTR	WO2024094171A1_31	.	COc1cc(N2CCC(CN3CCC(c4ccc5c(N6CCC(=O)NC6=O)nn(C)c5c4)C(F)(F)C3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1P(C)(C)=O)OCCCCn1cc-2cn1	C49H56BrF2N12O5P	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-QXQ7SC	WO2024094171A1_32	.	COc1cc(N2CCC(CN3CCN(c4ccc5c(C6CCC(=O)NC6=O)nn(C)c5c4)[C@H](C)C3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCn1cc-2cn1	C50H60BrN13O6S	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-GTAVOU	WO2024094171A1_33	.	COc1cc(N2CCC(CN3CCN(c4ccc5c(C6CCC(=O)NC6=O)nn(C)c5c4)C4(CC4)C3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCn1cc-2cn1	C51H60BrN13O6S	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-66UH4E	WO2024094171A1_34	.	COc1cc(N2CCC(CN3C[C@H]4C[C@@H]3CN4c3ccc4c(C5CCC(=O)NC5=O)nn(C)c4c3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCn1cc-2cn1	C50H58BrN13O6S	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-GRWGBY	WO2024094171A1_35	.	COc1cc(N2CCC(CN3C[C@@H]4C[C@H]3CN4c3ccc4c(C5CCC(=O)NC5=O)nn(C)c4c3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCn1cc-2cn1	C50H58BrN13O6S	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-3I9GT2	WO2024094171A1_36	.	COc1cc(N2CCC(CN3CCCN(c4ccc5c(C6CCC(=O)NC6=O)nn(C)c5c4)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCn1cc-2cn1	C50H60BrN13O6S	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-IY8E7N	WO2024094171A1_37	.	COc1cc(N2CCC(CN3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1P(C)(C)=O)OCCCCCn1cc-2cn1	C50H57BrN11O7P	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-EM9VBJ	WO2024094171A1_38	.	COc1cc(N2CCC(CN3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1cc(F)c(cc1N(C)S(C)(=O)=O)OCCCCn1cc-2cn1	C49H54BrFN12O8S	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-5PUBB9	WO2024094171A1_39	.	COc1cc(N2CCC(CN3CCC(c4ccc5c(N6CCC(=O)NC6=O)nn(C)c5c4)C(F)(F)C3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1cc(F)c(cc1N(C)S(C)(=O)=O)OCCCCn1cc-2cn1	C49H55BrF3N13O6S	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-CCUH9T	WO2024094171A1_4	.	COc1cc(N2CCN(C(=O)CN3CCC(c4ccc5c(N6CCC(=O)NC6=O)nn(C)c5c4)C(F)(F)C3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCn1cc-2cn1	C49H55BrF2N14O7S	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-U7RLWU	WO2024094171A1_40	.	COc1cc(N2CCC(CN3CCC(c4ccc5c(N6CCC(=O)NC6=O)nn(C)c5c4)C(F)(F)C3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1cc(F)c(cc1P(C)(C)=O)OCCCCn1cc-2cn1	C49H55BrF3N12O5P	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-CHP8ZZ	WO2024094171A1_41	.	COc1cc(N2CCC(CN3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1cc(F)c(cc1P(C)(C)=O)OCCCCn1cc-2cn1	C49H54BrFN11O7P	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-G37YY7	WO2024094171A1_42	.	COc1cc(N2CCC(CN3CCN(c4ccc5c(C6CCC(=O)NC6=O)nn(C)c5c4)CC3)CC2)c2cc1Nc1ncc(Cl)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCn1cc-2cn1	C49H58ClN13O6S	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-VCYTJ5	WO2024094171A1_43	.	COc1cc(N2CCC(CN3CCN(c4ccc5c(C6CCC(=O)NC6=O)nn(C)c5c4F)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCn1cc-2cn1	C49H57BrFN13O6S	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-4N8Q27	WO2024094171A1_44	.	COc1cc(N2CCC(CN3CCN(c4ccc5c(C6CCC(=O)NC6=O)nn(C)c5c4)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCC[C@H](C)Cn1cc-2cn1	C50H60BrN13O6S	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-TJU54U	WO2024094171A1_45	.	COc1cc(N2CCC(CN3CCN(c4ccc5c(C6CCC(=O)NC6=O)nn(C)c5c4)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCC(C)(C)Cn1cc-2cn1	C51H62BrN13O6S	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-GBL2MV	WO2024094171A1_46	.	COc1cc(N2CCC(CN3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)c2cc1Nc1ncc(C(F)(F)F)c(n1)Nc1ccc(cc1P(C)(C)=O)OCCCCn1cc-2cn1	C50H55F3N11O7P	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-MEOIEU	WO2024094171A1_47	.	COc1cc(N2CCC(CN3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)c2cc1Nc1ncc(C(F)(F)F)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCn1cc-2cn1	C50H55F3N12O8S	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-99FFZT	WO2024094171A1_48	.	COc1cc(N2CCC(OC3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCn1cc-2cn1	C49H54BrN11O9S	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-VWLSLI	WO2024094171A1_49	.	COc1cc(N2CCC(N(C)C3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCn1cc-2cn1	C50H57BrN12O8S	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-JATOQO	WO2024094171A1_5	.	COc1cc(N2CCN(C(=O)CN3CCC(c4ccc5c(N6CCC(=O)NC6=O)nn(C)c5c4)C(F)(F)C3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCCn1cc-2cn1	C50H57BrF2N14O7S	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-HZVFHL	WO2024094171A1_50	.	COc1cc(N2CCC(N3CCN(CC4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)CC2)c2cc1Nc1ncc(Cl)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCn1cc-2cn1	C54H64ClN13O8S	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-01W85S	WO2024094171A1_51	.	COc1cc(N2CCC(CN3CCC(N4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCn1cc-2cn1	C54H64BrN13O8S	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-DGC0CO	WO2024094171A1_52	.	COc1cc(N2CCC(CN3CCN(C4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1NS(C)(=O)=O)OCCCCn1cc-2cn1	C53H62BrN13O8S	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-DY02DE	WO2024094171A1_54	.	COc1cc(N2CCC(CN3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)c2cc1Nc1ncc(Cl)c(n1)Nc1ccc(cc1P(C)(C)=O)OCCCCCn1cc-2cn1	C50H57ClN11O7P	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-K333VU	WO2024094171A1_55	.	COc1cc(N2CCC(CN3CCN(c4ccc(C(=O)NC5CCC(=O)NC5=O)c(F)c4)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCn1cc-2cn1	C48H56BrFN12O7S	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-L7J6C3	WO2024094171A1_56	.	COc1cc(N2CCC(N3CCN(CCc4ccc5c(C6CCC(=O)NC6=O)nn(C)c5c4)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCn1cc-2cn1	C50H60BrN13O6S	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-V64JN2	WO2024094171A1_57	.	COc1cc(N2CCC(N3CCN(CCc4cc(F)c(C5CCC(=O)NC5=O)c(F)c4)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCn1cc-2cn1	C48H56BrF2N11O6S	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-JVO9SK	WO2024094171A1_58	.	COc1cc(N2CCC(CCN3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCn1cc-2cn1	C50H57BrN12O8S	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-DRIJMQ	WO2024094171A1_59	.	COc1cc(N2CCC(O)(CN3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCn1cc-2cn1	C49H55BrN12O9S	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-A4DNQ9	WO2024094171A1_6	.	CN(c1cc2ccc1Nc1nc(ncc1Br)Nc1cc(F)c(N3CCN(C(=O)CN4CCC(c5ccc6c(N7CCC(=O)NC7=O)nn(C)c6c5)C(F)(F)C4)CC3)c(c1)-c1cnn(c1)CCCCO2)S(C)(=O)=O	C48H52BrF3N14O6S	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-ZVJJFU	WO2024094171A1_60	.	COc1cc(N2CCC(CN3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C[C@H]3CO)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCn1cc-2cn1	C50H57BrN12O9S	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-FKZ2JK	WO2024094171A1_61	.	COc1cc(N2CCC(CN3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C[C@@H]3CO)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCn1cc-2cn1	C50H57BrN12O9S	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-9WAK97	WO2024094171A1_7	.	CN(c1cc2ccc1Nc1nc(ncc1Br)Nc1cc(F)c(N3CCN(C(=O)CN4CCC(c5ccc6c(N7CCC(=O)NC7=O)nn(C)c6c5)C(F)(F)C4)CC3)c(c1)-c1cnn(c1)CCCCCO2)S(C)(=O)=O	C49H54BrF3N14O6S	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-JHP5VH	WO2024094171A1_8	.	CN(c1cc2ccc1Nc1nc(ncc1Br)Nc1cc(F)c(N3CCC(O)(CC(=O)N4CCC(c5ccc6c(N7CCC(=O)NC7=O)nn(C)c6c5)C(F)(F)C4)CC3)c(c1)-c1cnn(c1)CCCCO2)S(C)(=O)=O	C49H53BrF3N13O7S	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-VJIG58	WO2024094171A1_9	.	COc1cc(N2CCN(CC3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)c2cc1Nc1ncc(Br)c(n1)Nc1ccc(cc1N(C)S(C)(=O)=O)OCCCCn1cc-2cn1	C49H55BrN12O8S	EGFR	P00533	CRBN	WO-2024094171-A1
TPD-XE8DVI	WO2024098692A1_1	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=CC=CC(N7CCC(=O)NC7=O)=C6)CC5)CC4)C=C3)N=C2)N1C1=NC(C(C)(C)O)=CC=C1	C42H49N11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-YQMHH4	WO2024098692A1_2	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=CC=CC(N7CCC(=O)NC7=O)=C6)CC5)CC4)C=C3)N=C2)N1C1=NC2=C(C=C1)CC[C@]2(O)CC	C44H51N11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-UDOJ6J	WO2024098692A1_3	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=CN=CC(N7CCC(=O)NC7=O)=C6)CC5)CC4)C=C3)N=C2)N1C1=NC2=C(C=C1)CC[C@]2(O)CC	C43H50N12O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-NB688C	WO2024098692A1_5	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=CC=CC(N7CCC(=O)NC7=O)=C6Cl)CC5)CC4)C=C3)N=C2)N1C1=NC2=C(C=C1)CC[C@]2(O)CC	C44H50ClN11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-56GZZK	WO2024098692A1_6	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=CC=CC(N7CCC(=O)NC7=O)=C6C)CC5)CC4)C=C3)N=C2)N1C1=NC2=C(C=C1)CC[C@]2(O)CC	C45H53N11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-2AXVWP	WO2024098692A1_7	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=CN=CC(N7CCC(=O)NC7=O)=C6C)CC5)CC4)C=C3)N=C2)N1C1=CC=C2CC[C@](O)(CC)C2=N1	C44H52N12O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-L32OYB	WO2024098692A1_8	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=CN=CC(N7CCC(=O)NC7=O)=C6C)CC5)CC4)C=C3)N=C2)N1C1=NC(C(C)(C)O)=CC=C1	C42H50N12O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-2FW73Z	WO2024098692A1_9	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=CC=CC(N7CCC(=O)NC7=O)=C6F)CC5)CC4)C=C3)N=C2)N1C1=NC(C(C)(C)O)=CC=C1	C42H48FN11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-PVY6HU	WO2024098692A1_10	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=CC=CC(N7CCC(=O)NC7=O)=C6F)CC5)CC4)C=C3)N=C2)N1C1=NC2=C(C=C1)CC[C@]2(O)CC	C44H50FN11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-IFNSNA	WO2024098692A1_11	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=CC=CC(N7CCC(=O)NC7=O)=C6C)CC5)CC4)C=C3)N=C2)N1C1=NC(C(C)(C)O)=CC=C1	C43H51N11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-72EK28	WO2024098692A1_12	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=CC=CC(N7CCC(=O)NC7=O)=C6Cl)CC5)CC4)C=C3)N=C2)N1C1=NC(C(C)(C)O)=CC=C1	C42H48ClN11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-DDS6U7	WO2024098692A1_13	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=CC(Cl)=CC(N7CCC(=O)NC7=O)=C6)CC5)CC4)C=C3)N=C2)N1C1=NC(C(C)(C)O)=CC=C1	C42H48ClN11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-VU1Q85	WO2024098692A1_14	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=CC=CC(N7CCC(=O)NC7=O)=C6)CC5)CC4)C=C3)N=C2)N1C1=NN(C(C)C)C(=O)C=C1	C41H48N12O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-3CRB83	WO2024098692A1_15	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=CN=CC(N7CCC(=O)NC7=O)=C6)CC5)CC4)C=C3)N=C2)N1C1=NC(C(C)(C)O)=CC=C1	C41H48N12O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-40C3UI	WO2024098692A1_16	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCC(CN5CCN(C6=CC=CC(N7CCC(=O)NC7=O)=C6)CC5)CC4)C=C3)N=C2)N1C1=NC(C(C)(C)O)=CC=C1	C42H49N11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-M4YFQ5	WO2024098692A1_17	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(C5CCN(C6=CC=CC(N7CCC(=O)NC7=O)=C6)CC5)CC4)C=C3)N=C2)N1C1=NC(C(C)(C)O)=CC=C1	C41H47N11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-ZBYMGX	WO2024098692A1_18	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCC(CN5CCN(C6=CC=CC(N7CCC(=O)NC7=O)=C6)CC5)CC4)C=C3)N=C2)N1C1=NC2=C(C=C1)CC[C@]2(O)CC	C44H51N11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-910ANF	WO2024098692A1_21	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=CC=C(F)C(N7CCC(=O)NC7=O)=C6)CC5)CC4)C=C3)N=C2)N1C1=NC2=C(C=C1)CC[C@]2(O)CC	C44H50FN11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-NE392E	WO2024098692A1_22	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=CC=C(C)C(N7CCC(=O)NC7=O)=C6)CC5)CC4)C=C3)N=C2)N1C1=NC2=C(C=C1)CC[C@]2(O)CC	C45H53N11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-K5X68L	WO2024098692A1_23	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=CC=C(Cl)C(N7CCC(=O)NC7=O)=C6)CC5)CC4)C=C3)N=C2)N1C1=NC2=C(C=C1)CC[C@]2(O)CC	C44H50ClN11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-ROFUO9	WO2024098692A1_24	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=C(F)C=CC(N7CCC(=O)NC7=O)=C6)CC5)CC4)C=C3)N=C2)N1C1=NC2=C(C=C1)CC[C@]2(O)CC	C44H50FN11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-VW0SPM	WO2024098692A1_27	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=CC=C(C)C(N7CCC(=O)NC7=O)=C6)CC5)CC4)C=C3)N=C2)N1C1=NC(C(C)(C)O)=CC=C1	C43H51N11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-BH8JQ8	WO2024098692A1_28	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=C(F)C=C(C)C(N7CCC(=O)NC7=O)=C6)CC5)CC4)C=C3)N=C2)N1C1=NC(C(C)(C)O)=CC=C1	C43H50FN11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-XSTHPE	WO2024098692A1_29	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=C(F)C=CC(N7CCC(=O)NC7=O)=C6F)CC5)CC4)C=C3)N=C2)N1C1=NC(C(C)(C)O)=CC=C1	C42H47F2N11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-V6DDGX	WO2024098692A1_30	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=CC=C(F)C(N7CCC(=O)NC7=O)=C6)CC5)CC4)C=C3)N=C2)N1C1=NC(C(C)(C)O)=CC=C1	C42H48FN11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-T4YCPK	WO2024098692A1_31	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=C(C)C(N7CCC(=O)NC7=O)=CC=C6F)CC5)CC4)C=C3)N=C2)N1C1=NC(C(C)(C)O)=CC=C1	C43H50FN11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-B715Z4	WO2024098692A1_32	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=C(C)C(N7CCC(=O)NC7=O)=CC=C6F)CC5)CC4)C=C3)N=C2)N1C1=CC=C2CC[C@](O)(CC)C2=N1	C45H52FN11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-2N5QUL	WO2024098692A1_33	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=C(F)C=C(F)C(N7CCC(=O)NC7=O)=C6)CC5)CC4)C=C3)N=C2)N1C1=NC(C(C)(C)O)=CC=C1	C42H47F2N11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-RGNZU6	WO2024098692A1_34	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=CC=C(F)C(N7CCC(=O)NC7=O)=C6F)CC5)CC4)C=C3)N=C2)N1C1=NC(C(C)(C)O)=CC=C1	C42H47F2N11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-79F8J5	WO2024098692A1_35	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=CC=C(F)C(N7CCC(=O)NC7=O)=C6F)CC5)CC4)C=C3)N=C2)N1C1=NC2=C(C=C1)CC[C@]2(O)CC	C44H49F2N11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-H5J0EQ	WO2024098692A1_36	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=CC=CC(C7CCC(=O)NC7=O)=C6)CC5)CC4)C=C3)N=C2)N1C1=NC(C(C)(C)O)=CC=C1	C43H50N10O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-XZVELY	WO2024098692A1_37	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCC(CN5CCN(C6=CC=CC(C7CCC(=O)NC7=O)=C6)CC5)CC4)C=C3)N=C2)N1C1=NC(C(C)(C)O)=CC=C1	C43H50N10O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-Y80K8J	SCHEMBL25590491	1-[4-[4-[[4-[4-[[1-[6-(2-Hydroxypropan-2-yl)pyridin-2-yl]-3-oxo-2-prop-2-enylpyrazolo[3,4-d]pyrimidin-6-yl]amino]phenyl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]-1,3-diazinane-2,4-dione	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(C4CCN(CC5CCN(C6=CC=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)N=C2)N1C1=NC(C(C)(C)O)=CC=C1	C43H50N10O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-H1LXF8	WO2024098692A1_39	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=CC=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)N=C2)N1C1=NC(C(C)(C)O)=CC=C1	C42H49N11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-E5YLS5	WO2024098692A1_40	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(C4CCN(CC5CCN(C6=CC=CC(N7CCC(=O)NC7=O)=C6)CC5)CC4)C=C3)N=C2)N1C1=NC(C(C)(C)O)=CC=C1	C43H50N10O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-P12RAI	WO2024098692A1_43	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=CC(F)=CC(N7CCC(=O)NC7=O)=C6F)CC5)CC4)C=C3)N=C2)N1C1=NC2=C(C=C1)CC[C@]2(O)CC	C44H49F2N11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-GE92RT	WO2024098692A1_44	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=CC(C(F)F)=CC(N7CCC(=O)NC7=O)=C6)CC5)CC4)C=C3)N=C2)N1C1=NC(C(C)(C)O)=CC=C1	C43H49F2N11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-3F5V93	WO2024098692A1_45	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=CC=CC(N7CCC(=O)NC7=O)=C6F)CC5)[C@H](C)C4)C=C3)N=C2)N1C1=NC2=C(C=C1)CC[C@]2(O)CC	C45H52FN11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-NDM17B	WO2024098692A1_46	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CC6(C5)CN(C5=CC=CC(N7CCC(=O)NC7=O)=C5F)C6)CC4)C=C3)N=C2)N1C1=CC=C2CC[C@](O)(CC)C2=N1	C45H50FN11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-8KEXVI	WO2024098692A1_47	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=CC=CC(N7CCC(=O)NC7=O)=C6)CC5)[C@H](C)C4)C=C3)N=C2)N1C1=NC2=C(C=C1)CC[C@]2(O)CC	C45H53N11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-4VNGMC	WO2024098692A1_48	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=CC=CC(N7CCC(=O)NC7=O)=C6)CC5)[C@@H](C)C4)C=C3)N=C2)N1C1=NC2=C(C=C1)CC[C@]2(O)CC	C45H53N11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-K79PIM	WO2024098692A1_49	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4C[C@@H](C)N(CC5CCN(C6=CC=CC(N7CCC(=O)NC7=O)=C6F)CC5)[C@@H](C)C4)C=C3)N=C2)N1C1=NC2=C(C=C1)CC[C@]2(O)CC	C46H54FN11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-AYAXM5	WO2024098692A1_51	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(C5CC6(CCN(C7=C(Cl)C(N8CCC(=O)NC8=O)=CC=C7)C6)C5)CC4)C=C3)N=C2)N1C1=CC=C2CC[C@](O)(CC)C2=N1	C45H50ClN11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-BSKQ0V	WO2024098692A1_52	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CN(C6=CC=CC(N7CCC(=O)NC7=O)=C6F)C5)CC4)C=C3)N=C2)N1C1=NC2=C(C=C1)CC[C@]2(O)CC	C42H46FN11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-PPD01C	WO2024098692A1_53	.	C=CCN1C(=O)C2=C(N=C(NC3=CC(C)=C(N4CCN(CC5CCN(C6=CC=CC(N7CCC(=O)NC7=O)=C6F)CC5)CC4)C=C3)N=C2)N1C1=NC2=C(C=C1)CC[C@]2(O)CC	C45H52FN11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-VA49GG	WO2024098692A1_54	.	C=CCN1C(=O)C2=C(N=C(NC3=CC(C)=C(N4CCN(CC5CCN(C6=CC=CC(N7CCC(=O)NC7=O)=C6Cl)CC5)CC4)C=C3)N=C2)N1C1=NC2=C(C=C1)CC[C@]2(O)CC	C45H52ClN11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-UCPWWL	WO2024098692A1_55	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4C[C@@H](C)N(CC5CCN(C6=CC=CC(N7CCC(=O)NC7=O)=C6Cl)CC5)[C@@H](C)C4)C=C3)N=C2)N1C1=CC=C2CC[C@](O)(CC)C2=N1	C46H54ClN11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-8AVQ2M	WO2024098692A1_56	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(C5CC6(C5)CN(C5=C(Cl)C(N7CCC(=O)NC7=O)=CC=C5)C6)CC4)C=C3)N=C2)N1C1=NC2=C(C=C1)CC[C@]2(O)CC	C44H48ClN11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-NPUJDM	WO2024098692A1_58	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=CC=CC(N7CCC(=O)NC7=O)=C6Cl)CC5)[C@@H](C)C4)C=C3)N=C2)N1C1=NC2=C(C=C1)CC[C@]2(O)CC	C45H52ClN11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-ABQ6BY	WO2024098692A1_59	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=CC=CC(N7CCC(=O)NC7=O)=C6F)CC5)C[C@@H]4C)C=C3)N=C2)N1C1=NC2=C(C=C1)C1[CH]O[C@]2(CC)C1	C46H51FN11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-YNZ9H9	WO2024098692A1_61	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=CC=CC(N7CCC(=O)NC7=O)=C6F)CC5)[C@@H](C)C4)C=C3)N=C2)N1C1=NC2=C(C=C1)CC[C@]2(O)CC	C45H52FN11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-CB6BNX	WO2024098692A1_62	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCC6(CC5)CN(C5=CC=CC(N7CCC(=O)NC7=O)=C5Cl)C6)CC4)C=C3)N=C2)N1C1=CC=C2CC[C@](O)(CC)C2=N1	C47H54ClN11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-QUBQUB	WO2024098692A1_63	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=CC=CC(N7CCC(=O)NC7=O)=C6C#N)CC5)CC4)C=C3)N=C2)N1C1=CC=C2CC[C@](O)(CC)C2=N1	C45H50N12O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-NXH4RK	WO2024098692A1_64	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=CC=CC(N7CCC(=O)NC7=O)=C6C(F)(F)F)CC5)CC4)C=C3)N=C2)N1C1=CC=C2CC[C@](O)(CC)C2=N1	C45H50F3N11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-Y00ONR	WO2024098692A1_65	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=C(C(F)(F)F)C=CC(N7CCC(=O)NC7=O)=C6)CC5)CC4)C=C3)N=C2)N1C1=CC=C2CC[C@](O)(CC)C2=N1	C45H50F3N11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-EGY9L9	WO2024098692A1_66	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=CC=CC(N7CCC(=O)NC7=O)=C6C(=O)C(F)(F)F)CC5)CC4)C=C3)N=C2)N1C1=CC=C2CC[C@](O)(CC)C2=N1	C46H50F3N11O5	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-YSBDR6	WO2024098692A1_67	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=C(C)C=CC(N7CCC(=O)NC7=O)=C6)CC5)CC4)C=C3)N=C2)N1C1=NC2=C(C=C1)CC[C@]2(O)CC	C45H53N11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-UI5N55	WO2024098692A1_68	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=CC=CC(N7CCC(=O)NC7=O)=C6F)CC5)CC4)C=C3)N=C2)N1C1=NC2=C(C=C1)CC[C@@]2(C)O	C43H48FN11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-AE60JW	WO2024098692A1_70	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=C(Cl)C=CC(N7CCC(=O)NC7=O)=C6)CC5)CC4)C=C3)N=C2)N1C1=NC(C(C)(C)O)=CC=C1	C42H48ClN11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-2CA3R1	WO2024098692A1_74	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=C(C)C=CC(N7CCC(=O)NC7=O)=C6)CC5)CC4)C=C3)N=C2)N1C1=NC(C(C)(C)O)=CC=C1	C43H51N11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-5D0KYM	WO2024098692A1_75	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=CC=CC(N7CCC(=O)NC7=O)=C6OC)CC5)CC4)C=C3)N=C2)N1C1=CC=C2CC[C@](O)(CC)C2=N1	C45H53N11O5	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-T54R13	WO2024098692A1_76	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=CC=CC(N7CCC(=O)NC7=O)=C6Cl)CC5)CC4)C=C3)N=C2)N1C1=NN(C(C)C)C(=O)C=C1	C41H47ClN12O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-1PV88G	WO2024098692A1_77	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=CC=CC(N7CCC(=O)NC7=O)=C6Cl)CC5)CC4)C=C3)N=C2)N1C1=NC2=C(C=C1)CC[C@@]2(C)O	C43H48ClN11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-HTSCWY	WO2024098692A1_78	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=CC(F)=CC(N7CCC(=O)NC7=O)=C6Cl)CC5)CC4)C=C3)N=C2)N1C1=NC(C(C)(C)O)=CC=C1	C42H47ClFN11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-K4JWPV	WO2024098692A1_79	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=C(C)N=CC(N7CCC(=O)NC7=O)=C6)CC5)CC4)C=C3)N=C2)N1C1=NC(C(C)(C)O)=CC=C1	C42H50N12O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-K85LBD	WO2024098692A1_80	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=CC=C(F)C(N7CCC(=O)NC7=O)=C6C)CC5)CC4)C=C3)N=C2)N1C1=NC2=C(C=C1)CC[C@]2(O)CC	C45H52FN11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-UYFE2J	WO2024098692A1_81	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=CC=C(F)C(N7CCC(=O)NC7=O)=C6C)CC5)CC4)C=C3)N=C2)N1C1=NC(C(C)(C)O)=CC=C1	C43H50FN11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-R7YUEX	WO2024098692A1_82	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=C(F)C=CC(N7CCC(=O)NC7=O)=C6Cl)CC5)CC4)C=C3)N=C2)N1C1=NC(C(C)(C)O)=CC=C1	C42H47ClFN11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-5TQTW1	WO2024098692A1_83	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=C(Cl)C=C(F)C(N7CCC(=O)NC7=O)=C6)CC5)CC4)C=C3)N=C2)N1C1=NC(C(C)(C)O)=CC=C1	C42H47ClFN11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-D01DA3	WO2024098692A1_84	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=C(F)C=C(Cl)C(N7CCC(=O)NC7=O)=C6)CC5)CC4)C=C3)N=C2)N1C1=NC(C(C)(C)O)=CC=C1	C42H47ClFN11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-KKZY4E	WO2024098692A1_85	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=CC=C(F)C(N7CCC(=O)NC7=O)=C6Cl)CC5)CC4)C=C3)N=C2)N1C1=CC=C2CC[C@](O)(CC)C2=N1	C44H49ClFN11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-RQFULJ	WO2024098692A1_86	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=CC=C(F)C(C7CCC(=O)NC7=O)=C6)CC5)CC4)C=C3)N=C2)N1C1=NC2=C(C=C1)CC[C@]2(O)CC	C45H51FN10O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-CWJVNQ	WO2024098692A1_87	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=C(Cl)C(C7CCC(=O)NC7=O)=CC=C6)CC5)CC4)C=C3)N=C2)N1C1=NC2=C(C=C1)CC[C@]2(O)CC	C45H51ClN10O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-1M52UL	WO2024098692A1_88	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=CC=CC(C7CCC(=O)NC7=O)=C6F)CC5)CC4)C=C3)N=C2)N1C1=NC2=C(C=C1)CC[C@]2(O)CC	C45H51FN10O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-MSELR3	WO2024098692A1_89	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=CN=C(C)C(N7CCC(=O)NC7=O)=C6)CC5)CC4)C=C3)N=C2)N1C1=NC(C(C)(C)O)=CC=C1	C42H50N12O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-EYQG1W	WO2024098692A1_90	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=CN=C(C)C(N7CCC(=O)NC7=O)=C6)CC5)CC4)C=C3)N=C2)N1C1=NC2=C(C=C1)C1C[C@]2(CC)[C@@]1(C)O	C46H54N12O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-UO71X2	WO2024098692A1_91	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=CN=CC(N7CCC(=O)NC7=O)=C6Cl)CC5)CC4)C=C3)N=C2)N1C1=NC(C(C)(C)O)=CC=C1	C41H47ClN12O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-BST6RV	WO2024098692A1_92	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=CC(C#N)=CC(N7CCC(=O)NC7=O)=C6)CC5)CC4)C=C3)N=C2)N1C1=NC(C(C)(C)O)=CC=C1	C43H48N12O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-Y0IJ13	WO2024098692A1_93	.	CS(C)(=O)=NC1=NC(NC2=C(C#N)C=NC(NC3=CC=C(N4CCN(CC5CCN(C6=CC=CC(N7CCC(=O)NC7=O)=C6)CC5)CC4)C=C3)=N2)=CC=C1	C38H44N12O3S	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-K3PLEO	WO2024098692A1_94	.	C=CCN1C(=O)C2=C(N=C([N-]C3=CC=C(N4CCN([C@H]5CCN(C6=CC=CC(N7CCC(=O)[N-]C7=O)=C6Cl)C5)CC4)C=C3)N=C2)N1C1=NC2=C(C=C1)CC[C@]2(O)CC	C42H44ClN11O4-2	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-PEZB26	WO2024098692A1_97	.	C=CCN1C(=O)C2=C(N=C([N-]C3=CC=C(N4CCN(C[C@H]5CCN(C6=CC=CC(N7CCC(=O)[N-]C7=O)=C6Cl)C5)CC4)C=C3)N=C2)N1C1=NC2=C(C=C1)CC[C@]2(O)CC	C43H46ClN11O4-2	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-AJSMDE	WO2024098692A1_98	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCCN(C6=CC=CC(N7CCC(=O)NC7=O)=C6F)C5)CC4)C=C3)N=C2)N1C1=NC2=C(C=C1)CC[C@]2(O)CC	C44H50FN11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-OX6DTR	WO2024098692A1_100	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(C[C@@H]5CC6CC5CN6C5=CC=CC(N6CCC(=O)NC6=O)=C5F)CC4)C=C3)N=C2)N1C1=NC(C(C)(C)O)=CC=C1	C43H48FN11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-EPIPA6	WO2024098692A1_101	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN([C@H](C)C5CCN(C6=CC=CC(N7CCC(=O)NC7=O)=C6Cl)CC5)CC4)C=C3)N=C2)N1C1=NC2=C(C=C1)CC[C@]2(O)CC	C45H52ClN11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-M6C3QA	WO2024098692A1_103	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN([C@@H]5CCCN(C6=CC=CC(N7CCC(=O)NC7=O)=C6F)C5)CC4)C=C3)N=C2)N1C1=NC2=C(C=C1)CC[C@]2(O)CC	C43H48FN11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-TDAD7W	WO2024098692A1_104	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN([C@H]5C[C@H]6C[C@@]6(C6=CC=CC(N7CCC(=O)NC7=O)=C6F)C5)CC4)C=C3)N=C2)N1C1=NC2=C(C=C1)CC[C@]2(O)CC	C44H47FN10O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-KU4WLQ	WO2024098692A1_105	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCC(N6C=CC=C(N7CCC(=O)NC7=O)C6=O)CC5)CC4)C=C3)N=C2)N1C1=NC(C(C)(C)O)=CC=C1	C42H49N11O5	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-UXDFAF	WO2024098692A1_106	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=C(C)N=CC(N7CCC(=O)NC7=O)=C6C)CC5)CC4)C=C3)N=C2)N1C1=CC=C2CC[C@](O)(CC)C2=N1	C45H54N12O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-56GNBG	WO2024098692A1_107	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=CC=CC(N7CCC(=O)NC7=O)=C6Cl)[C@@H](C)C5)CC4)C=C3)N=C2)N1C1=NC2=C(C=C1)CC[C@]2(O)CC	C45H52ClN11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-SVDP6J	WO2024098692A1_108	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=CC=CC(N7CCC(=O)NC7=O)=C6Cl)[C@H](C)C5)CC4)C=C3)N=C2)N1C1=NC2=C(C=C1)CC[C@]2(O)CC	C45H52ClN11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-67WBZC	WO2024098692A1_109	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=CC=CC(N7CCC(=O)NC7=O)=C6Br)CC5)CC4)C=C3)N=C2)N1C1=NC2=C(C=C1)CC[C@]2(O)CC	C44H50BrN11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-PCC8CB	WO2024098692A1_110	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(C5CC6CN(C7=CC=CC(N8CCC(=O)NC8=O)=C7Cl)CC6C5)CC4)C=C3)N=C2)N1C1=NC2=C(C=C1)CC[C@]2(O)CC	C45H50ClN11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-Z55SKU	WO2024098692A1_111	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(C(C)(C)C5CCN(C6=CC=CC(N7CCC(=O)NC7=O)=C6Cl)CC5)CC4)C=C3)N=C2)N1C1=NC2=C(C=C1)CC[C@]2(O)CC	C46H54ClN11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-BDO75Q	WO2024098692A1_113	.	CC(C)(O)C1=NC(NC2=C(C#N)C=NC(NC3=CC=C(N4CCN(CC5CCN(C6=CC=CC(N7CCC(=O)NC7=O)=C6)CC5)CC4)C=C3)=N2)=CC=C1	C39H45N11O3	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-E56WDN	WO2024098692A1_114	.	C=CCN1C(=O)C2=C(N=C(NC3=CC=C(N4CCN(CC5CCN(C6=CC(C(F)F)=CC(N7CCC(=O)NC7=O)=C6)CC5)CC4)C=C3)N=C2)N1C1=NC2=C(C=C1)CC[C@]2(O)CC	C45H51F2N11O4	WEE1	P30291	CRBN	WO-2024098692-A1
TPD-GR2BW3	SCHEMBL27422257	(3S)-3-[6-[4-[[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027620	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC(CN5CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC5)CC4)CC1)=N3)=CC(O)=C2	C53H61F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-RUAH9S	SCHEMBL27422261	(3S)-3-[6-[4-[[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027484	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CC(CN4CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC4)C5)CC1)=N3)=CC(O)=C2	C56H65F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-ERHOYL	SCHEMBL27422268	(3S)-3-[6-[4-[[7-[[1-[[4-[[1-(dimethylamino)cyclobutyl]methylamino]-7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027548	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(NCC1(N(C)C)CCC1)=NC(OCC1(CN4CCC5(CC4)CC(CN4CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC4)C5)CC1)=N3)=CC(O)=C2	C57H68F2N10O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-G14E0Y	SCHEMBL27422278	(3S)-3-[6-[4-[[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-(2,3,6,7-tetrahydroazepin-1-yl)pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027528	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC=CCC1)=NC(OCC1(CN4CCC5(CC4)CC(CN4CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC4)C5)CC1)=N3)=CC(O)=C2	C56H63F2N9O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-YA70J0	SCHEMBL27422282	(3S)-3-[6-[4-[[7-[[1-[[7-[6-amino-4-methyl-3-(trifluoromethyl)pyridin-2-yl]-13-[1-(2-aminopyridin-3-yl)ethyl]-8-chloro-6-fluoro-10-oxa-2,4,13-triazatricyclo[7.4.1.05,14]tetradeca-1,3,5(14),6,8-pentaen-3-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CC1=C(C(F)(F)F)C(C2=C(Cl)C3=C4C(=NC(OCC5(CN6CCC7(CC6)CC(CN6CCN(C8=CC9=C(C=C8)C(=O)N([C@H]8CCC(=O)NC8=O)C9)CC6)C7)CC5)=NC4=C2F)N(C(C)C2=C(N)N=CC=C2)CCO3)=NC(N)=C1	C55H61ClF4N12O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-VTPRUE	SCHEMBL27422286	(3S)-3-[6-[4-[[1-[[1-[[7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027654	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC(CN5CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC5)CC4)CC1)=N3)=CC(O)=C2	C53H62FN9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-89LDO2	SCHEMBL27422290	(3S)-3-[6-[4-[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027615	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC(N5CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC5)CC4)CC1)=N3)=CC(O)=C2	C52H59F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-HL1H74	SCHEMBL27422295	(3S)-3-[6-[4-[[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-4-fluoropiperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027472	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC(F)(CN5CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC5)CC4)CC1)=N3)=CC(O)=C2	C53H60F3N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-YH8VNE	SCHEMBL27422301	(3R)-3-[6-[4-[[1-[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]azetidin-3-yl]azetidin-3-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027608	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CC(N5CC(CN6CCN(C7=CC8=C(C=C7)C(=O)N([C@@H]7CCC(=O)NC7=O)C8)CC6)C5)C4)CC1)=N3)=CC(O)=C2	C54H62F2N10O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-ZRAHP5	SCHEMBL27422305	(3S)-3-[6-[4-[[4-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperazin-1-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027575	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCN(CC5CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC5)CC4)CC1)=N3)=CC(O)=C2	C53H61F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-HSD4RG	SCHEMBL27422310	(3R)-3-[6-[4-[[2-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-2-azaspiro[3.3]heptan-6-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027631	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CC5(CC(CN6CCN(C7=CC8=C(C=C7)C(=O)N([C@@H]7CCC(=O)NC7=O)C8)CC6)C5)C4)CC1)=N3)=CC(O)=C2	C54H61F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-0RBGDP	SCHEMBL27422320	(3S)-3-[6-[4-[[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-4-hydroxypiperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027494	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC(O)(CN5CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC5)CC4)CC1)=N3)=CC(O)=C2	C53H61F2N9O7	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-GH6UYR	SCHEMBL27422326	3-[4-[4-[[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]phenyl]piperidine-2,6-dione; SCHEMBL31027642	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC(CN5CCN(C6=CC=C(C7CCC(=O)NC7=O)C=C6)CC5)CC4)CC1)=N3)=CC(O)=C2	C51H60F2N8O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-OYIDEO	SCHEMBL27422331	(3S)-3-[6-[4-[[1-[[1-[[4-[cyclopropyl(methyl)amino]-7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027556	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N(C)C1CC1)=NC(OCC1(CN4CCC(CN5CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC5)CC4)CC1)=N3)=CC(O)=C2	C51H58FN9O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-D3BAW4	SCHEMBL27422335	3-[6-[2-[[1-[[7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-2,7-diazaspiro[3.5]nonan-7-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027533	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CC5(CCN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)CC5)C4)CC1)=N3)=CC(O)=C2	C50H55FN8O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-I55PYG	SCHEMBL27422345	3-[6-[2-[[1-[[1-[[7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]azetidin-3-yl]methyl]-2,7-diazaspiro[3.5]nonan-7-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027486	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CC(CN5CC6(CCN(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8)CC6)C5)C4)CC1)=N3)=CC(O)=C2	C54H62FN9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-G186BO	SCHEMBL27422351	3-[6-[2-[[(3R)-1-[[1-[[7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]pyrrolidin-3-yl]methyl]-2,7-diazaspiro[3.5]nonan-7-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027730	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CC[C@@H](CN5CC6(CCN(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8)CC6)C5)C4)CC1)=N3)=CC(O)=C2	C55H64FN9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-23R6B6	SCHEMBL27422358	3-[6-[2-[[1-[[1-[[7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]methyl]-2,7-diazaspiro[3.5]nonan-7-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027557	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC(CN5CC6(CCN(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8)CC6)C5)CC4)CC1)=N3)=CC(O)=C2	C56H66FN9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-T8QRS2	SCHEMBL27422364	4-[[4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]-1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidine-4-carbonitrile; SCHEMBL31027666	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC(C#N)(CN5CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC5)CC4)CC1)=N3)=CC(O)=C2	C54H60F2N10O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-4HBOOA	SCHEMBL27422373	3-[4-[4-[[1-[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]azetidin-3-yl]methyl]piperazin-1-yl]phenyl]piperidine-2,6-dione; SCHEMBL31027584	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC(N5CC(CN6CCN(C7=CC=C(C8CCC(=O)NC8=O)C=C7)CC6)C5)CC4)CC1)=N3)=CC(O)=C2	C54H65F2N9O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-GLY2LJ	SCHEMBL27422380	3-[6-[2-[[(3S)-1-[[1-[[7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]pyrrolidin-3-yl]methyl]-2,7-diazaspiro[3.5]nonan-7-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027682	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CC[C@H](CN5CC6(CCN(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8)CC6)C5)C4)CC1)=N3)=CC(O)=C2	C55H64FN9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-PXHAZW	SCHEMBL27431644	(3S)-3-[6-[4-[[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-(1-oxa-8-azaspiro[3.5]nonan-8-yl)pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027562	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCCC4(CCO4)C1)=NC(OCC1(CN4CCC(CN5CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC5)CC4)CC1)=N3)=CC(O)=C2	C54H61F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-6JM77B	SCHEMBL27422386	3-[6-[4-[1-[[1-[[7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]oxypiperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027488	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC(OC5CCN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)CC5)CC4)CC1)=N3)=CC(O)=C2	C53H61FN8O7	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-D7370B	SCHEMBL27422395	(3S)-3-[6-[4-[[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-4-methoxypiperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027565	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC(CN5CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC5)(OC)CC4)CC1)=N3)=CC(O)=C2	C54H63F2N9O7	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-VKVQKV	SCHEMBL27422399	(3S)-3-[6-[4-[[7-[[1-[[7-[6-amino-2-methyl-3-(trifluoromethyl)pyridin-4-yl]-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027610	CC1=NC(N)=CC(C2=NC=C3C(N4CCC[C@@](C)(O)C4)=NC(OCC4(CN5CCC6(CC5)CC(CN5CCN(C7=CC=C8C(=O)N([C@H]9CCC(=O)NC9=O)CC8=C7)CC5)C6)CC4)=NC3=C2F)=C1C(F)(F)F	C51H61F4N11O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-MU7CNG	SCHEMBL27422412	(3S)-3-[6-[4-[[7-[[1-[[7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[[(1R,2R)-2-fluorocyclopropyl]-methylamino]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027606	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N(C)[C@@H]1C[C@H]1F)=NC(OCC1(CN4CCC5(CC4)CC(CN4CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC4)C5)CC1)=N3)=CC(O)=C2	C54H61F2N9O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-SISUK9	SCHEMBL27422416	3-[6-[2-[[1-[[1-[[7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-4-fluoropiperidin-4-yl]methyl]-2,7-diazaspiro[3.5]nonan-7-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027698	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC(F)(CN5CC6(CCN(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8)CC6)C5)CC4)CC1)=N3)=CC(O)=C2	C56H65F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-OFIZQT	SCHEMBL27422422	(3S)-3-[6-[4-[[1-[[1-[[7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[[(2R)-2-fluorocyclopropyl]-methylamino]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N(C)C1C[C@H]1F)=NC(OCC1(CN4CCC(CN5CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC5)CC4)CC1)=N3)=CC(O)=C2	C51H57F2N9O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-7LUWTX	SCHEMBL27422429	(3S)-3-[6-[2-[1-[[1-[[7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]-2,7-diazaspiro[3.5]nonan-7-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027585	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC(N5CC6(CCN(C7=CC8=C(C=C7)C(=O)N([C@H]7CCC(=O)NC7=O)C8)CC6)C5)CC4)CC1)=N3)=CC(O)=C2	C55H64FN9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-CZI6E9	SCHEMBL27422435	2-(2,6-dioxopiperidin-3-yl)-5-[4-[7-[[1-[[7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]piperazin-1-yl]isoindole-1,3-dione; SCHEMBL31027603	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CC(N4CCN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC4)C5)CC1)=N3)=CC(O)=C2	C55H62FN9O7	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-CA9NAR	SCHEMBL27422438	2-(2,6-dioxopiperidin-3-yl)-5-[4-[[7-[[1-[[7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]isoindole-1,3-dione; SCHEMBL31027521	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CC(CN4CCN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC4)C5)CC1)=N3)=CC(O)=C2	C56H64FN9O7	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-7390S0	SCHEMBL27422440	(3S)-3-[6-[4-[[1-[[1-[[7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-4-fluoropiperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027719	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC(F)(CN5CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC5)CC4)CC1)=N3)=CC(O)=C2	C53H61F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-FYY7RL	SCHEMBL27431830	3-[2-[[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]methyl]-1,3-dihydroisoindol-5-yl]piperidine-2,6-dione; SCHEMBL31027651	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CC(CN4CC6=CC=C(C7CCC(=O)NC7=O)C=C6C4)C5)CC1)=N3)=CC(O)=C2	C52H59F2N7O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-FCKVJ7	SCHEMBL27422446	(3S)-3-[6-[4-[3-[[1-[[7-(3-amino-7,8-difluoronaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-3-azaspiro[5.5]undecan-9-yl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027514	C[C@@]1(O)CCCN(C2=NC(OCC3(CN4CCC5(CCC(N6CCN(C7=CC8=C(C=C7)C(=O)N([C@H]7CCC(=O)NC7=O)C8)CC6)CC5)CC4)CC3)=NC3=C2C=NC(C2=CC(N)=CC4=C2C(F)=C(F)C=C4)=C3F)C1	C55H63F3N10O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-KFM8G9	SCHEMBL27422451	(3S)-3-[6-[4-[[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-methoxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027735	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(OC)C1)=NC(OCC1(CN4CCC5(CC4)CC(CN4CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC4)C5)CC1)=N3)=CC(O)=C2	C57H67F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-3BE5HP	SCHEMBL27422460	(3S)-3-[6-[4-[1-[[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-(1-oxa-8-azaspiro[3.5]nonan-8-yl)pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]methyl]azetidin-3-yl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027680	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCCC4(CCO4)C1)=NC(OCC1(CN4CCC(CN5CC(N6CCN(C7=CC8=C(C=C7)C(=O)N([C@H]7CCC(=O)NC7=O)C8)CC6)C5)CC4)CC1)=N3)=CC(O)=C2	C57H66F2N10O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-RB60PB	SCHEMBL27422470	(3S)-3-[6-[4-[1-[[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-(1-oxa-8-azaspiro[3.5]nonan-8-yl)pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]methyl]piperidin-4-yl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027635	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCCC4(CCO4)C1)=NC(OCC1(CN4CCC(CN5CCC(N6CCN(C7=CC8=C(C=C7)C(=O)N([C@H]7CCC(=O)NC7=O)C8)CC6)CC5)CC4)CC1)=N3)=CC(O)=C2	C59H70F2N10O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-PYS8FN	SCHEMBL27431882	3-[6-[4-[4-[[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-4-methylpiperidin-4-yl]methyl]piperazin-1-yl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027645	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC(C)(CN5CCN(C6CCN(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8)CC6)CC5)CC4)CC1)=N3)=CC(O)=C2	C59H72F2N10O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-X6NZ4Z	PROTAC K-Ras Degrader-3	3043670-68-1; PROTAC K-Ras Degrader-3; orb2665122; SCHEMBL27422476; SCHEMBL31027614; EX-A13388	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC(C)(CN5CC6(CCN(C7=CC8=C(C=C7)C(=O)N([C@H]7CCC(=O)NC7=O)C8)CC6)C5)CC4)CC1)=N3)=CC(O)=C2	C57H67F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-TUTWRI	SCHEMBL27422485	(3S)-3-[6-[4-[[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-(1-oxa-8-azaspiro[3.5]nonan-8-yl)pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-4-fluoropiperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027674	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCCC4(CCO4)C1)=NC(OCC1(CN4CCC(F)(CN5CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC5)CC4)CC1)=N3)=CC(O)=C2	C54H60F3N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-G891U8	SCHEMBL27431033	(3S)-3-[6-[4-[[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(4S)-1-oxa-8-azaspiro[3.5]nonan-8-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-2-fluoro-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027507	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@]4(CCO4)C1)=NC(OCC1(CN4CCC5(CC4)CC(F)(CN4CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC4)C5)CC1)=N3)=CC(O)=C2	C57H64F3N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-LP0LTC	WO2024118966A1_43	.	C=C1CCC(N2CC3=C(C=CC(N4CCC(N5CCC(OC6CCN(CC7(COC8=NC9=C(C=NC(C%10=CC(O)=CC%11=C%10C(CC)=C(F)C=C%11)=C9F)C(N9CCC[C@@](C)(O)C9)=N8)CC7)CC6)CC5)CC4)=C3)C2=O)C(=O)N1	C59H71F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-TZOZ67	SCHEMBL27423696	(3S)-3-[6-[4-[[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(4S)-1-oxa-8-azaspiro[3.5]nonan-8-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027588	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@]4(CCO4)C1)=NC(OCC1(CN4CCC(CN5CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC5)CC4)CC1)=N3)=CC(O)=C2	C54H61F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-PZPSKU	SCHEMBL27423715	(3S)-3-[6-[4-[[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(4R)-1-oxa-8-azaspiro[3.5]nonan-8-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027716	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@]4(CCO4)C1)=NC(OCC1(CN4CCC(CN5CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC5)CC4)CC1)=N3)=CC(O)=C2	C54H61F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-63ERXV	SCHEMBL27422509	3-[4-[4-[[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-2-fluoro-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione; SCHEMBL31027538	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CC(F)(CN4CCN(C6=CC(F)=C(C7CCC(=O)NC7=O)C(F)=C6)CC4)C5)CC1)=N3)=CC(O)=C2	C54H61F5N8O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-V57OEE	SCHEMBL27422516	3-[4-[4-[[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(4S)-1-oxa-8-azaspiro[3.5]nonan-8-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-2-fluoro-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione; SCHEMBL31027725	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@]4(CCO4)C1)=NC(OCC1(CN4CCC5(CC4)CC(F)(CN4CCN(C6=CC(F)=C(C7CCC(=O)NC7=O)C(F)=C6)CC4)C5)CC1)=N3)=CC(O)=C2	C55H61F5N8O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-4LEJ1T	PROTAC K-Ras Degrader-2	PROTAC K-Ras Degrader-2; orb2945179; SCHEMBL27422520; SCHEMBL31027637; HY-164365; 3043670-74-9	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC(C)(CN5CCN(C6=CC(F)=C(C7CCC(=O)NC7=O)C(F)=C6)CC5)CC4)CC1)=N3)=CC(O)=C2	C52H60F4N8O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-WWI61E	SCHEMBL27422526	3-[4-[4-[[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione; SCHEMBL31027684	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CC(CN4CCN(C6=CC(F)=C(C7CCC(=O)NC7=O)C(F)=C6)CC4)C5)CC1)=N3)=CC(O)=C2	C54H62F4N8O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-E2KJE6	SCHEMBL27422529	3-[4-[4-[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]piperazin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione; SCHEMBL31027611	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CC(N4CCN(C6=CC(F)=C(C7CCC(=O)NC7=O)C(F)=C6)CC4)C5)CC1)=N3)=CC(O)=C2	C53H60F4N8O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-1NMN8F	SCHEMBL27422533	3-[4-[4-[3-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-3-azaspiro[5.5]undecan-9-yl]piperazin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione; SCHEMBL31027550	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CCC(N6CCN(C7=CC(F)=C(C8CCC(=O)NC8=O)C(F)=C7)CC6)CC5)CC4)CC1)=N3)=CC(O)=C2	C55H64F4N8O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-ULP6C8	SCHEMBL27422540	(3S)-3-[6-[4-[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(4S)-1-oxa-8-azaspiro[3.5]nonan-8-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027746	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@]4(CCO4)C1)=NC(OCC1(CN4CCC5(CC4)CC(N4CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC4)C5)CC1)=N3)=CC(O)=C2	C56H63F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-W1O42U	SCHEMBL27422543	(3S)-3-[6-[4-[3-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(4S)-1-oxa-8-azaspiro[3.5]nonan-8-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-3-azaspiro[5.5]undecan-9-yl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027512	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@]4(CCO4)C1)=NC(OCC1(CN4CCC5(CCC(N6CCN(C7=CC8=C(C=C7)C(=O)N([C@H]7CCC(=O)NC7=O)C8)CC6)CC5)CC4)CC1)=N3)=CC(O)=C2	C58H67F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-8868YA	SCHEMBL27432136	(3S)-3-[6-[4-[[2-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(4S)-1-oxa-8-azaspiro[3.5]nonan-8-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-fluoro-2-azaspiro[3.5]nonan-7-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027529	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@]4(CCO4)C1)=NC(OCC1(CN4CC5(CCC(F)(CN6CCN(C7=CC8=C(C=C7)C(=O)N([C@H]7CCC(=O)NC7=O)C8)CC6)CC5)C4)CC1)=N3)=CC(O)=C2	C57H64F3N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-WD13Y3	SCHEMBL27422547	3-[4-[2-[3-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-3,9-diazaspiro[5.5]undecan-9-yl]ethyl]-2,6-difluorophenyl]piperidine-2,6-dione; SCHEMBL31027636	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CCN(CCC6=CC(F)=C(C7CCC(=O)NC7=O)C(F)=C6)CC5)CC4)CC1)=N3)=CC(O)=C2	C52H59F4N7O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-01NOZS	SCHEMBL27422552	3-[4-[2-[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]-2,7-diazaspiro[3.5]nonan-7-yl]-2,6-difluorophenyl]piperidine-2,6-dione; SCHEMBL31027587	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC(N5CC6(CCN(C7=CC(F)=C(C8CCC(=O)NC8=O)C(F)=C7)CC6)C5)CC4)CC1)=N3)=CC(O)=C2	C53H60F4N8O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-9PMAQ2	SCHEMBL27422556	3-[4-[2-[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]-2,7-diazaspiro[3.5]nonan-7-yl]-2,6-difluorophenyl]piperidine-2,6-dione; SCHEMBL31027659	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CC(N4CC6(CCN(C7=CC(F)=C(C8CCC(=O)NC8=O)C(F)=C7)CC6)C4)C5)CC1)=N3)=CC(O)=C2	C56H64F4N8O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-3RDERJ	SCHEMBL27422562	3-[4-[2-[2-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-2-azaspiro[3.5]nonan-7-yl]-2,7-diazaspiro[3.5]nonan-7-yl]-2,6-difluorophenyl]piperidine-2,6-dione; SCHEMBL31027509	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CC5(CCC(N6CC7(CCN(C8=CC(F)=C(C9CCC(=O)NC9=O)C(F)=C8)CC7)C6)CC5)C4)CC1)=N3)=CC(O)=C2	C56H64F4N8O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-VIYJZU	SCHEMBL27422566	3-[4-[4-[2-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-2-azaspiro[3.5]nonan-7-yl]piperazin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione; SCHEMBL31027657	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CC5(CCC(N6CCN(C7=CC(F)=C(C8CCC(=O)NC8=O)C(F)=C7)CC6)CC5)C4)CC1)=N3)=CC(O)=C2	C53H60F4N8O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-S7A687	SCHEMBL27422570	3-[4-[9-[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]-3,9-diazaspiro[5.5]undecan-3-yl]-2,6-difluorophenyl]piperidine-2,6-dione; SCHEMBL31027517	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC(N5CCC6(CCN(C7=CC(F)=C(C8CCC(=O)NC8=O)C(F)=C7)CC6)CC5)CC4)CC1)=N3)=CC(O)=C2	C55H64F4N8O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-10LYGC	SCHEMBL27422606	3-[4-[2-[4-[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-2,7-diazaspiro[3.5]nonan-2-yl]piperidin-1-yl]ethyl]-2,6-difluorophenyl]piperidine-2,6-dione; SCHEMBL31027704	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CN(C4CCN(CCC6=CC(F)=C(C7CCC(=O)NC7=O)C(F)=C6)CC4)C5)CC1)=N3)=CC(O)=C2	C55H64F4N8O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-9L9W1I	WO2024118966A1_63	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC(C)(CN5CCN(C6=CC7=C(C=C6)C(=O)N([C@@H]6CCC(=O)NC6=O)C7=O)CC5)CC4)CC1)=N3)=CC(O)=C2	C54H61F2N9O7	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-HGAMJH	SCHEMBL27422611	3-[5-[4-[[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-4-fluoropiperidin-4-yl]methyl]piperazin-1-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione; SCHEMBL31027630	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC(F)(CN5CCN(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC5)CC4)CC1)=N3)=CC(O)=C2	C53H61F3N10O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-XJAQ7M	SCHEMBL27432292	3-[4-[4-[[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-4-fluoropiperidin-4-yl]methyl]piperazin-1-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione; SCHEMBL31027699	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC(F)(CN5CCN(C6=CC=CC7=C6N(C)C(=O)N7C6CCC(=O)NC6=O)CC5)CC4)CC1)=N3)=CC(O)=C2	C53H61F3N10O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-9JCYWN	SCHEMBL27421916	3-[6-[4-[[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-4-fluoropiperidin-4-yl]methyl]piperazin-1-yl]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL31027506	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC(F)(CN5CCN(C6=CC7=C(C=C6)C(C6CCC(=O)NC6=O)=NN7C)CC5)CC4)CC1)=N3)=CC(O)=C2	C53H61F3N10O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-1OU388	SCHEMBL27432317	3-[7-[4-[[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-4-fluoropiperidin-4-yl]methyl]piperazin-1-yl]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL31027598	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC(F)(CN5CCN(C6=CC=CC7=C6N(C)N=C7C6CCC(=O)NC6=O)CC5)CC4)CC1)=N3)=CC(O)=C2	C53H61F3N10O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-U7UOGY	SCHEMBL27422615	(3S)-3-[6-[2-[[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-3-fluoroazetidin-3-yl]methyl]-2,7-diazaspiro[3.5]nonan-7-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027543	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CC(F)(CN5CC6(CCN(C7=CC8=C(C=C7)C(=O)N([C@H]7CCC(=O)NC7=O)C8)CC6)C5)C4)CC1)=N3)=CC(O)=C2	C54H60F3N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-01YRNX	SCHEMBL27422617	(3S)-3-[6-[4-[[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-3-fluoroazetidin-3-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027551	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CC(F)(CN5CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC5)C4)CC1)=N3)=CC(O)=C2	C51H56F3N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-NRZMPM	SCHEMBL27422618	3-[6-[3-[[4-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperazin-1-yl]methyl]-3-fluoroazetidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027561	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCN(CC5(F)CN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)C5)CC4)CC1)=N3)=CC(O)=C2	C51H56F3N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-VE1N2I	SCHEMBL27422620	3-[6-[4-[[4-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperazin-1-yl]methyl]-4-fluoropiperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027681	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCN(CC5(F)CCN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)CC5)CC4)CC1)=N3)=CC(O)=C2	C53H60F3N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-N0F07F	SCHEMBL27422625	(3S)-3-[6-[4-[1-[[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-4-fluoropiperidin-4-yl]methyl]piperidin-4-yl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027594	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC(F)(CN5CCC(N6CCN(C7=CC8=C(C=C7)C(=O)N([C@H]7CCC(=O)NC7=O)C8)CC6)CC5)CC4)CC1)=N3)=CC(O)=C2	C58H69F3N10O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-AN6SXZ	SCHEMBL27432439	3-[4-[4-[1-[[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-4-fluoropiperidin-4-yl]methyl]piperidin-4-yl]piperazin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione; SCHEMBL31027496	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC(F)(CN5CCC(N6CCN(C7=CC(F)=C(C8CCC(=O)NC8=O)C(F)=C7)CC6)CC5)CC4)CC1)=N3)=CC(O)=C2	C56H66F5N9O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-JMPQHS	SCHEMBL27432471	3-[4-[4-[[4-ethyl-1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione; SCHEMBL31027526	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC(CC)(CN5CCN(C6=CC(F)=C(C7CCC(=O)NC7=O)C(F)=C6)CC5)CC4)CC1)=N3)=CC(O)=C2	C53H62F4N8O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-K8645R	SCHEMBL31027527	3-[4-[4-[[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-4-propan-2-ylpiperidin-4-yl]methyl]piperazin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC(CN5CCN(C6=CC(F)=C(C7CCC(=O)NC7=O)C(F)=C6)CC5)(C(C)C)CC4)CC1)=N3)=CC(O)=C2	C54H64F4N8O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-XAAR48	SCHEMBL31027697	3-[4-[4-[1-[[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-4-methylpiperidin-4-yl]methyl]piperidin-4-yl]piperazin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC(C)(CN5CCC(N6CCN(C7=CC(F)=C(C8CCC(=O)NC8=O)C(F)=C7)CC6)CC5)CC4)CC1)=N3)=CC(O)=C2	C57H69F4N9O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-B1S6CS	SCHEMBL31027714	3-[4-[4-[1-[[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-4-methylpiperidin-4-yl]methyl]piperidin-4-yl]piperidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC(C)(CN5CCC(C6CCN(C7=CC(F)=C(C8CCC(=O)NC8=O)C(F)=C7)CC6)CC5)CC4)CC1)=N3)=CC(O)=C2	C58H70F4N8O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-NHIRZL	SCHEMBL31027505	(3S)-3-[6-[4-[4-[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]phenyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC(C5=CC=C(N6CCN(C7=CC8=C(C=C7)C(=O)N([C@H]7CCC(=O)NC7=O)C8)CC6)C=C5)CC4)CC1)=N3)=CC(O)=C2	C58H63F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-GW8LOK	SCHEMBL31027518	(3S)-3-[6-[4-[1-[[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-4-methylpiperidin-4-yl]methyl]piperidin-4-yl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC(C)(CN5CCC(C6CCN(C7=CC8=C(C=C7)C(=O)N([C@H]7CCC(=O)NC7=O)C8)CC6)CC5)CC4)CC1)=N3)=CC(O)=C2	C60H73F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-16VL16	SCHEMBL31027555	(3S)-3-[6-[4-[1-[[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-4-fluoropiperidin-4-yl]methyl]piperidin-4-yl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC(F)(CN5CCC(C6CCN(C7=CC8=C(C=C7)C(=O)N([C@H]7CCC(=O)NC7=O)C8)CC6)CC5)CC4)CC1)=N3)=CC(O)=C2	C59H70F3N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-ASDZGC	SCHEMBL27422645	3-[4-[4-[[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-4-fluoropiperidin-4-yl]methyl]piperazin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione; SCHEMBL31027473	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC(F)(CN5CCN(C6=CC(F)=C(C7CCC(=O)NC7=O)C(F)=C6)CC5)CC4)CC1)=N3)=CC(O)=C2	C51H57F5N8O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-01GZJY	SCHEMBL27422647	3-[4-[4-[[2-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-fluoro-2-azaspiro[3.5]nonan-7-yl]methyl]piperazin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione; SCHEMBL31027715	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CC5(CCC(F)(CN6CCN(C7=CC(F)=C(C8CCC(=O)NC8=O)C(F)=C7)CC6)CC5)C4)CC1)=N3)=CC(O)=C2	C54H61F5N8O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-KMC9I0	SCHEMBL27422650	3-[4-[4-[[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-4-fluoropiperidin-4-yl]methyl]piperazin-1-yl]-2-fluorophenyl]piperidine-2,6-dione; SCHEMBL31027683	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC(F)(CN5CCN(C6=CC(F)=C(C7CCC(=O)NC7=O)C=C6)CC5)CC4)CC1)=N3)=CC(O)=C2	C51H58F4N8O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-HFP3MW	SCHEMBL27422656	3-[4-[4-[2-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(4S)-1-oxa-8-azaspiro[3.5]nonan-8-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-2-azaspiro[3.5]nonan-7-yl]piperazin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione; SCHEMBL31027662	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@]4(CCO4)C1)=NC(OCC1(CN4CC5(CCC(N6CCN(C7=CC(F)=C(C8CCC(=O)NC8=O)C(F)=C7)CC6)CC5)C4)CC1)=N3)=CC(O)=C2	C54H60F4N8O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-MTDCZF	SCHEMBL27422660	(3S)-3-[6-[4-[[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(4S)-1-oxa-8-azaspiro[3.5]nonan-8-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-4-fluoropiperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027586	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@]4(CCO4)C1)=NC(OCC1(CN4CCC(F)(CN5CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC5)CC4)CC1)=N3)=CC(O)=C2	C54H60F3N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-3DXNQ4	SCHEMBL27422665	(3S)-3-[6-[4-[[7-[[1-[[7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027513	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CC(CN4CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC4)C5)CC1)=N3)=CC(O)=C2	C56H66FN9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-AEPZI2	SCHEMBL27422667	(3S)-3-[6-[4-[[7-[[1-[[7-(3-amino-8-ethyl-7-fluoronaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027695	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CC(CN4CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC4)C5)CC1)=N3)=CC(N)=C2	C56H66F2N10O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-NFLJJL	SCHEMBL27422670	(3S)-3-[6-[4-[[1-[[1-[[7-(3-amino-8-ethyl-7-fluoronaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027717	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC(CN5CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC5)CC4)CC1)=N3)=CC(N)=C2	C53H62F2N10O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-XBHDJU	SCHEMBL27422674	(3S)-3-[6-[4-[[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(1R,5R,6R)-6-hydroxy-3-azabicyclo[3.2.1]octan-3-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027671	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1C[C@@H]4C[C@H](C1)[C@H](O)C4)=NC(OCC1(CN4CCC5(CC4)CC(CN4CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC4)C5)CC1)=N3)=CC(O)=C2	C57H65F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-EMOYYL	SCHEMBL27422679	(3S)-3-[6-[4-[[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-(6-hydroxy-6-methyl-1,4-oxazepan-4-yl)pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027492	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCOCC(C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CC(CN4CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC4)C5)CC1)=N3)=CC(O)=C2	C56H65F2N9O7	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-OC5C4D	SCHEMBL27422682	(3S)-3-[6-[4-[[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-(6-hydroxy-6-methyl-1,4-oxazepan-4-yl)pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027706	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCOCC(C)(O)C1)=NC(OCC1(CN4CCC(CN5CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC5)CC4)CC1)=N3)=CC(O)=C2	C53H61F2N9O7	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-CHDJSH	SCHEMBL27422689	(3S)-3-[6-[4-[[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-(3-oxo-1,4-diazepan-1-yl)pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027678	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCCNC(=O)C1)=NC(OCC1(CN4CCC5(CC4)CC(CN4CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC4)C5)CC1)=N3)=CC(O)=C2	C55H62F2N10O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-WPVVWX	SCHEMBL27422697	3-chloro-5-[2-[[1-[[2-[[4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]-7-azaspiro[3.5]nonan-7-yl]methyl]cyclopropyl]methoxy]-7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-4-yl]-N,N-dimethyl-4,6,7,8-tetrahydropyrazolo[1,5-a][1,4]diazepine-2-carboxamide; SCHEMBL31027638	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCCN4N=C(C(=O)N(C)C)C(Cl)=C4C1)=NC(OCC1(CN4CCC5(CC4)CC(CN4CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC4)C5)CC1)=N3)=CC(O)=C2	C60H67ClF2N12O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-16RAKZ	SCHEMBL27422704	(3S)-3-[6-[4-[[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-(3-oxo-1,4-diazepan-1-yl)pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027559	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCCNC(=O)C1)=NC(OCC1(CN4CCC(CN5CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC5)CC4)CC1)=N3)=CC(O)=C2	C52H58F2N10O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-5QMCZN	SCHEMBL27422714	(3S)-3-[6-[4-[[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(1R,5R,6R)-6-hydroxy-3-azabicyclo[3.2.1]octan-3-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027658	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1C[C@@H]4C[C@H](C1)[C@H](O)C4)=NC(OCC1(CN4CCC(CN5CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC5)CC4)CC1)=N3)=CC(O)=C2	C54H61F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-Q7MMVY	WO2024118966A1_97	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCCC4(CC(O)C4)C1)=NC(OCC1(CN4CCC5(CC4)CC(CN4CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC4)C5)CC1)=N3)=CC(O)=C2	C58H67F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-WPNWGI	SCHEMBL27422730	(3S)-3-[6-[4-[[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-(2-hydroxy-6-azaspiro[3.5]nonan-6-yl)pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027503	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCCC4(CC(O)C4)C1)=NC(OCC1(CN4CCC(CN5CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC5)CC4)CC1)=N3)=CC(O)=C2	C55H63F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-DNO862	WO2024118966A1_99	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@]4(C1)C[C@H](O)C4)=NC(OCC1(CN4CCC5(CC4)CC(CN4CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC4)C5)CC1)=N3)=CC(O)=C2	C58H67F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-I3N42E	WO2024118966A1_100	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@]4(C1)C[C@@H](O)C4)=NC(OCC1(CN4CCC5(CC4)CC(CN4CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC4)C5)CC1)=N3)=CC(O)=C2	C58H67F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-VBFMMV	SCHEMBL27422750	(3S)-3-[6-[4-[[7-[[1-[[7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(1R,5R,6R)-6-hydroxy-3-azabicyclo[3.2.1]octan-3-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027474	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1C[C@@H]4C[C@H](C1)[C@H](O)C4)=NC(OCC1(CN4CCC5(CC4)CC(CN4CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC4)C5)CC1)=N3)=CC(O)=C2	C57H66FN9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-AO3QCR	SCHEMBL27422753	3-chloro-5-[2-[[1-[[2-[[4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]-7-azaspiro[3.5]nonan-7-yl]methyl]cyclopropyl]methoxy]-7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-4-yl]-N,N-dimethyl-4,6,7,8-tetrahydropyrazolo[1,5-a][1,4]diazepine-2-carboxamide; SCHEMBL31027577	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCCN4N=C(C(=O)N(C)C)C(Cl)=C4C1)=NC(OCC1(CN4CCC5(CC4)CC(CN4CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC4)C5)CC1)=N3)=CC(O)=C2	C60H68ClFN12O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-1MFXJZ	SCHEMBL27422754	(3S)-3-[6-[4-[[7-[[1-[[7-(7,8-difluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027490	C[C@@]1(O)CCCN(C2=NC(OCC3(CN4CCC5(CC4)CC(CN4CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC4)C5)CC3)=NC3=C2C=NC(C2=CC(O)=CC4=C2C(F)=C(F)C=C4)=C3F)C1	C54H60F3N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-TFWHNY	SCHEMBL27422758	(3S)-3-[6-[4-[[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(6S)-6-hydroxy-6-methyl-1,4-oxazepan-4-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027690	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCOC[C@@](C)(O)C1)=NC(OCC1(CN4CCC(CN5CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC5)CC4)CC1)=N3)=CC(O)=C2	C53H61F2N9O7	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-IOKZSZ	SCHEMBL27422761	(3S)-3-[6-[4-[[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(6S)-6-hydroxy-6-methyl-1,4-oxazepan-4-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027524	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCOC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CC(CN4CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC4)C5)CC1)=N3)=CC(O)=C2	C56H65F2N9O7	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-AAA3ND	SCHEMBL27422762	(3S)-3-[6-[4-[[7-[[1-[[7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(6S)-6-hydroxy-6-methyl-1,4-oxazepan-4-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027707	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCOC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CC(CN4CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC4)C5)CC1)=N3)=CC(O)=C2	C56H66FN9O7	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-7FIWIT	SCHEMBL27422764	(3S)-3-[6-[4-[[7-[[1-[[7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(6R)-6-hydroxy-6-methyl-1,4-oxazepan-4-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027471	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCOC[C@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CC(CN4CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC4)C5)CC1)=N3)=CC(O)=C2	C56H66FN9O7	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-444A25	SCHEMBL27422769	3-chloro-5-[2-[[1-[[4-[[4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]methyl]cyclopropyl]methoxy]-7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-4-yl]-N,N-dimethyl-4,6,7,8-tetrahydropyrazolo[1,5-a][1,4]diazepine-2-carboxamide; SCHEMBL31027549	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCCN4N=C(C(=O)N(C)C)C(Cl)=C4C1)=NC(OCC1(CN4CCC(CN5CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC5)CC4)CC1)=N3)=CC(O)=C2	C57H63ClF2N12O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-8VR9J6	SCHEMBL27422776	(3S)-3-[6-[4-[[7-[[1-[[7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoro-4-(1,4-oxazepan-4-yl)pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027532	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCCOCC1)=NC(OCC1(CN4CCC5(CC4)CC(CN4CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC4)C5)CC1)=N3)=CC(O)=C2	C55H64FN9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-EQQB3Y	SCHEMBL27422777	(3S)-3-[6-[4-[[1-[[1-[[7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoro-4-(1,4-oxazepan-4-yl)pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027542	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCCOCC1)=NC(OCC1(CN4CCC(CN5CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC5)CC4)CC1)=N3)=CC(O)=C2	C52H60FN9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-4W1N2P	SCHEMBL27422783	(3S)-3-[6-[4-[[1-[[1-[[7-(7,8-difluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027570	C[C@@]1(O)CCCN(C2=NC(OCC3(CN4CCC(CN5CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC5)CC4)CC3)=NC3=C2C=NC(C2=CC(O)=CC4=C2C(F)=C(F)C=C4)=C3F)C1	C51H56F3N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-A0EJAW	SCHEMBL27422786	(3S)-3-[6-[4-[[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(6R)-6-hydroxy-6-methyl-1,4-oxazepan-4-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027558	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCOC[C@](C)(O)C1)=NC(OCC1(CN4CCC(CN5CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC5)CC4)CC1)=N3)=CC(O)=C2	C53H61F2N9O7	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-XA4ENY	SCHEMBL27422791	(3S)-3-[6-[4-[[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(6R)-6-hydroxy-6-methyl-1,4-oxazepan-4-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027703	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCOC[C@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CC(CN4CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC4)C5)CC1)=N3)=CC(O)=C2	C56H65F2N9O7	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-NDORSN	SCHEMBL27422793	(3S)-3-[6-[4-[[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-(4-hydroxypiperidin-1-yl)pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027687	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC(O)CC1)=NC(OCC1(CN4CCC5(CC4)CC(CN4CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC4)C5)CC1)=N3)=CC(O)=C2	C55H63F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-PVMTFT	SCHEMBL27422796	(3S)-3-[6-[4-[[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-(4-hydroxypiperidin-1-yl)pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027579	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC(O)CC1)=NC(OCC1(CN4CCC(CN5CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC5)CC4)CC1)=N3)=CC(O)=C2	C52H59F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-OGINSV	SCHEMBL27422801	(3S)-3-[6-[4-[[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(4R)-4-hydroxyazepan-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027476	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@H](O)CC1)=NC(OCC1(CN4CCC5(CC4)CC(CN4CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC4)C5)CC1)=N3)=CC(O)=C2	C56H65F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-ABZ486	SCHEMBL27422803	(3S)-3-[6-[4-[[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(4R)-4-hydroxyazepan-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027576	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@H](O)CC1)=NC(OCC1(CN4CCC(CN5CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC5)CC4)CC1)=N3)=CC(O)=C2	C53H61F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-9O5PO3	SCHEMBL27422804	(3S)-3-[6-[4-[[1-[[1-[[7-(3-amino-8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027625	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC(CN5CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC5)CC4)CC1)=N3)=CC(N)=C2	C53H58F2N10O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-N6NZ3G	SCHEMBL27422805	(3S)-3-[6-[4-[[7-[[1-[[7-(3-amino-8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027612	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CC(CN4CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC4)C5)CC1)=N3)=CC(N)=C2	C56H62F2N10O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-ZVPYY4	SCHEMBL27422809	(3S)-3-[6-[4-[3-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-3-azaspiro[5.5]undecan-9-yl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027582	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CCC(N6CCN(C7=CC8=C(C=C7)C(=O)N([C@H]7CCC(=O)NC7=O)C8)CC6)CC5)CC4)CC1)=N3)=CC(O)=C2	C57H67F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-FA2EUQ	SCHEMBL27422810	(3S)-3-[6-[4-[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027732	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CC(N4CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC4)C5)CC1)=N3)=CC(O)=C2	C55H63F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-VB3ZQ0	SCHEMBL27422812	(3S)-3-[6-[4-[2-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-2-azaspiro[3.3]heptan-6-yl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027623	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CC5(CC(N6CCN(C7=CC8=C(C=C7)C(=O)N([C@H]7CCC(=O)NC7=O)C8)CC6)C5)C4)CC1)=N3)=CC(O)=C2	C53H59F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-5IOSWT	SCHEMBL27422814	(3S)-3-[6-[4-[[1-[[1-[[7-(8-chloro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027540	C[C@@]1(O)CCCN(C2=NC(OCC3(CN4CCC(CN5CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC5)CC4)CC3)=NC3=C2C=NC(C2=CC(O)=CC4=C2C(Cl)=CC=C4)=C3F)C1	C51H57ClFN9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-N9FBAC	SCHEMBL27422816	(3S)-3-[6-[4-[[7-[[1-[[4-(1,9-dioxa-6-azaspiro[3.6]decan-6-yl)-7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027593	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCOCC4(CCO4)C1)=NC(OCC1(CN4CCC5(CC4)CC(CN4CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC4)C5)CC1)=N3)=CC(O)=C2	C57H65F2N9O7	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-T4RIE8	SCHEMBL27422821	(3S)-3-[6-[4-[[1-[[1-[[4-(1,9-dioxa-6-azaspiro[3.6]decan-6-yl)-7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027491	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCOCC4(CCO4)C1)=NC(OCC1(CN4CCC(CN5CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC5)CC4)CC1)=N3)=CC(O)=C2	C54H61F2N9O7	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-CNGNH2	SCHEMBL27422826	(3S)-3-[6-[4-[[2-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-2-azaspiro[3.5]nonan-7-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027574	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CC5(CCC(CN6CCN(C7=CC8=C(C=C7)C(=O)N([C@H]7CCC(=O)NC7=O)C8)CC6)CC5)C4)CC1)=N3)=CC(O)=C2	C56H65F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-O7MOER	WO2024118966A1_127	.	C=C1NC(=O)CC[C@@H]1N1CC2=C(C=CC(N3CCN(CC4CCN(CC5(COC6=NC7=C(C=NC(C8=CC(O)=CC9=C8C(CC)=CC=C9)=C7F)C(N7CCNC(=O)CC7)=N6)CC5)CC4)CC3)=C2)C1=O	C53H61FN10O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-58IT12	SCHEMBL27422840	(3S)-3-[6-[4-[[7-[[1-[[7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoro-4-(5-oxo-1,4-diazepan-1-yl)pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027525	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCNC(=O)CC1)=NC(OCC1(CN4CCC5(CC4)CC(CN4CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC4)C5)CC1)=N3)=CC(O)=C2	C55H63FN10O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-C5YFVD	SCHEMBL27422849	(3S)-3-[6-[4-[[7-[[1-[[7-(8-chloro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027685	C[C@@]1(O)CCCN(C2=NC(OCC3(CN4CCC5(CC4)CC(CN4CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC4)C5)CC3)=NC3=C2C=NC(C2=CC(O)=CC4=C2C(Cl)=CC=C4)=C3F)C1	C54H61ClFN9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-FWJAE3	SCHEMBL27422851	(3S)-3-[6-[4-[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]azetidin-3-yl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027629	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CC(N5CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC5)C4)CC1)=N3)=CC(O)=C2	C50H55F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-C5D1EK	SCHEMBL27422855	(3S)-3-[6-[4-[[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-(3-fluoro-3-methylpiperidin-1-yl)pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027627	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCCC(C)(F)C1)=NC(OCC1(CN4CCC5(CC4)CC(CN4CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC4)C5)CC1)=N3)=CC(O)=C2	C56H64F3N9O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-JDG9MM	SCHEMBL27422864	3-[6-[3-[[4-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperazin-1-yl]methyl]azetidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027689	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCN(CC5CN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)C5)CC4)CC1)=N3)=CC(O)=C2	C51H57F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-QM115D	SCHEMBL27422872	(3S)-3-[6-[4-[[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-2-fluoro-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027621	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CC(F)(CN4CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC4)C5)CC1)=N3)=CC(O)=C2	C56H64F3N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-1HPEBX	SCHEMBL27422875	(3S)-3-[6-[4-[[7-[[1-[[7-[5-amino-3-chloro-2-(trifluoromethyl)phenyl]-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027567	C[C@@]1(O)CCCN(C2=NC(OCC3(CN4CCC5(CC4)CC(CN4CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC4)C5)CC3)=NC3=C2C=NC(C2=CC(N)=CC(Cl)=C2C(F)(F)F)=C3F)C1	C51H59ClF4N10O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-HBLGRK	SCHEMBL27422877	(3S)-3-[6-[4-[2-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-2-azaspiro[3.5]nonan-7-yl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027546	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CC5(CCC(N6CCN(C7=CC8=C(C=C7)C(=O)N([C@H]7CCC(=O)NC7=O)C8)CC6)CC5)C4)CC1)=N3)=CC(O)=C2	C55H63F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-Q7SAM2	SCHEMBL27422880	(3S)-3-[6-[4-[1-[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]azetidin-3-yl]azetidin-3-yl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027718	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CC(N5CC(N6CCN(C7=CC8=C(C=C7)C(=O)N([C@H]7CCC(=O)NC7=O)C8)CC6)C5)C4)CC1)=N3)=CC(O)=C2	C53H60F2N10O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-GNHMBV	SCHEMBL27422884	(3S)-3-[6-[4-[7-[[1-[[7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027477	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CC(N4CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC4)C5)CC1)=N3)=CC(O)=C2	C55H64FN9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-ABNWQU	WO2024118966A1_139	.	CCC1=C(F)C=CC2=CC(C)=CC(C3=C(F)C4=NC(OCC5(CN6CC(N7CCC(N8CCN(C9=CC%10=C(C=C9)C(=O)N([C@H]9CCC(=O)NC9=O)C%10)CC8)CC7)C6)CC5)=NC(N5CCC[C@@](C)(O)C5)=C4C=N3)=C21	C56H66F2N10O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-RHMXGL	SCHEMBL27422893	3-[6-[9-[[1-[[7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-3,9-diazaspiro[5.5]undecan-3-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027591	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CCN(C4=CC6=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C6)CC5)CC1)=N3)=CC(O)=C2	C52H59FN8O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-Q6LEZ6	SCHEMBL27422897	(3S)-3-[6-[4-[2-[[1-[[7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-2-azaspiro[3.5]nonan-7-yl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027520	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CC5(CCC(N6CCN(C7=CC8=C(C=C7)C(=O)N([C@H]7CCC(=O)NC7=O)C8)CC6)CC5)C4)CC1)=N3)=CC(O)=C2	C55H64FN9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-XETW0K	SCHEMBL27422905	3-[6-[2-[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]-2,7-diazaspiro[3.5]nonan-7-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027600	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC(N5CC6(CCN(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8)CC6)C5)CC4)CC1)=N3)=CC(O)=C2	C55H63F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-BF9EO8	SCHEMBL27422907	3-[6-[2-[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]azetidin-3-yl]-2,7-diazaspiro[3.5]nonan-7-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027618	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CC(N5CC6(CCN(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8)CC6)C5)C4)CC1)=N3)=CC(O)=C2	C53H59F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-I4L9NA	SCHEMBL27422910	3-[6-[9-[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]-3,9-diazaspiro[5.5]undecan-3-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027700	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC(N5CCC6(CCN(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8)CC6)CC5)CC4)CC1)=N3)=CC(O)=C2	C57H67F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-E9BESW	SCHEMBL27422911	(3S)-3-[6-[4-[1-[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]azetidin-3-yl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CCC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=NC(OCC5(CN6CCC(N7CC(N8CCN(C9=CC%10=C(C=C9)C(=O)N([C@H]9CCC(=O)NC9=O)C%10)CC8)C7)CC6)CC5)=NC(N5CCC[C@@](C)(O)C5)=C4C=N3)=C21	C55H64F2N10O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-AMNFTF	SCHEMBL27422916	(3S)-3-[6-[4-[1-[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]piperidin-4-yl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027478	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC(N5CCC(N6CCN(C7=CC8=C(C=C7)C(=O)N([C@H]7CCC(=O)NC7=O)C8)CC6)CC5)CC4)CC1)=N3)=CC(O)=C2	C57H68F2N10O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-VSB4VF	SCHEMBL27422917	(3S)-3-[6-[4-[1-[[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]methyl]piperidin-4-yl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027616	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC(CN5CCC(N6CCN(C7=CC8=C(C=C7)C(=O)N([C@H]7CCC(=O)NC7=O)C8)CC6)CC5)CC4)CC1)=N3)=CC(O)=C2	C58H70F2N10O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-KIIN77	SCHEMBL27422921	(3S)-3-[6-[4-[1-[[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]azetidin-3-yl]methyl]piperidin-4-yl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027723	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CC(CN5CCC(N6CCN(C7=CC8=C(C=C7)C(=O)N([C@H]7CCC(=O)NC7=O)C8)CC6)CC5)C4)CC1)=N3)=CC(O)=C2	C56H66F2N10O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-I3P1DZ	SCHEMBL27422924	(3S)-3-[6-[4-[[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-2-methyl-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027726	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CC(C)(CN4CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC4)C5)CC1)=N3)=CC(O)=C2	C57H67F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-H1T1IQ	SCHEMBL27422928	3-[6-[7-[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]-2,7-diazaspiro[3.5]nonan-2-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027510	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC(N5CCC6(CC5)CN(C5=CC7=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C7)C6)CC4)CC1)=N3)=CC(O)=C2	C55H63F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-7V29I5	SCHEMBL27422929	3-[6-[7-[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]azetidin-3-yl]-2,7-diazaspiro[3.5]nonan-2-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027749	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CC(N5CCC6(CC5)CN(C5=CC7=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C7)C6)C4)CC1)=N3)=CC(O)=C2	C53H59F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-BQ150D	SCHEMBL27422936	3-[6-[9-[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]azetidin-3-yl]-3,9-diazaspiro[5.5]undecan-3-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027655	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CC(N5CCC6(CCN(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8)CC6)CC5)C4)CC1)=N3)=CC(O)=C2	C55H63F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-9XSJ8Y	SCHEMBL27422944	3-[6-[6-[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]-2,6-diazaspiro[3.3]heptan-2-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027688	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC(N5CC6(CN(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8)C6)C5)CC4)CC1)=N3)=CC(O)=C2	C53H59F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-DLT0T4	SCHEMBL27422946	3-[6-[4-[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-2,7-diazaspiro[3.5]nonan-2-yl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027675	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CN(C4CCN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)CC4)C5)CC1)=N3)=CC(O)=C2	C55H63F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-R83R2R	SCHEMBL27422950	(3S)-3-[6-[4-[[1-[[1-[[7-(8-chloro-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027592	C[C@@]1(O)CCCN(C2=NC(OCC3(CN4CCC(CN5CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC5)CC4)CC3)=NC3=C2C=NC(C2=CC(O)=CC4=C2C(Cl)=C(F)C=C4)=C3F)C1	C51H56ClF2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-OGBO1S	SCHEMBL27422956	(3S)-3-[6-[4-[[7-[[1-[[7-(8-chloro-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027516	C[C@@]1(O)CCCN(C2=NC(OCC3(CN4CCC5(CC4)CC(CN4CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC4)C5)CC3)=NC3=C2C=NC(C2=CC(O)=CC4=C2C(Cl)=C(F)C=C4)=C3F)C1	C54H60ClF2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-G187XP	SCHEMBL27422958	3-[6-[6-[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]azetidin-3-yl]-2,6-diazaspiro[3.3]heptan-2-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027694	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CC(N5CC6(CN(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8)C6)C5)C4)CC1)=N3)=CC(O)=C2	C51H55F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-8U29S2	SCHEMBL27422963	3-[6-[4-[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-2-methyl-7-azaspiro[3.5]nonan-2-yl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027544	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CC(C)(N4CCN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)CC4)C5)CC1)=N3)=CC(O)=C2	C56H65F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-AEL6U8	SCHEMBL27422968	(3S)-3-[6-[4-[[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-(2-oxa-6-azabicyclo[5.1.0]octan-6-yl)pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027605	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCCOC4CC41)=NC(OCC1(CN4CCC(CN5CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC5)CC4)CC1)=N3)=CC(O)=C2	C53H59F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-6CN5HD	SCHEMBL27422972	3-[6-[6-[4-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperazin-1-yl]-2-azaspiro[3.3]heptan-2-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027547	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCN(C5CC6(C5)CN(C5=CC7=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C7)C6)CC4)CC1)=N3)=CC(O)=C2	C53H59F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-MF6BEJ	SCHEMBL27422974	3-[6-[2-[4-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperazin-1-yl]-7-azaspiro[3.5]nonan-7-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027519	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCN(C5CC6(CCN(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8)CC6)C5)CC4)CC1)=N3)=CC(O)=C2	C55H63F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-SL69LM	SCHEMBL27422979	3-[6-[3-[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-2,7-diazaspiro[3.5]nonan-2-yl]azetidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027639	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CN(C4CN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)C4)C5)CC1)=N3)=CC(O)=C2	C53H59F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-TIT6MP	SCHEMBL27422981	3-[6-[3-[9-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-3,9-diazaspiro[5.5]undecan-3-yl]azetidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027552	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CCN(C4CN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)C4)CC5)CC1)=N3)=CC(O)=C2	C55H63F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-4P8A8G	SCHEMBL27422985	(3S)-3-[6-[4-[[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-(2-oxa-6-azabicyclo[5.1.0]octan-6-yl)pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027495	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCCOC4CC41)=NC(OCC1(CN4CCC5(CC4)CC(CN4CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC4)C5)CC1)=N3)=CC(O)=C2	C56H63F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-SQ41HW	SCHEMBL27423019	3-[6-[3-[2-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-2,7-diazaspiro[3.5]nonan-7-yl]azetidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027677	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CC5(CCN(C6CN(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8)C6)CC5)C4)CC1)=N3)=CC(O)=C2	C53H59F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-K1YMW6	SCHEMBL27422997	3-[6-[4-[3-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3S)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-9-methyl-3-azaspiro[5.5]undecan-9-yl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027607	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CCC(C)(N4CCN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)CC4)CC5)CC1)=N3)=CC(O)=C2	C58H69F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-5JK9OV	SCHEMBL27423002	(3S)-3-[6-[4-[1-[1-[[1-[[7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]azetidin-3-yl]azetidin-3-yl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027667	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CC(N5CC(N6CCN(C7=CC8=C(C=C7)C(=O)N([C@H]7CCC(=O)NC7=O)C8)CC6)C5)C4)CC1)=N3)=CC(O)=C2	C53H61FN10O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-IQ9QFJ	SCHEMBL27423006	(3S)-3-[6-[4-[1-[1-[[1-[[7-(7,8-difluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]azetidin-3-yl]azetidin-3-yl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027641	C[C@@]1(O)CCCN(C2=NC(OCC3(CN4CC(N5CC(N6CCN(C7=CC8=C(C=C7)C(=O)N([C@H]7CCC(=O)NC7=O)C8)CC6)C5)C4)CC3)=NC3=C2C=NC(C2=CC(O)=CC4=C2C(F)=C(F)C=C4)=C3F)C1	C51H55F3N10O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-6TXT5H	SCHEMBL27423012	(3S)-3-[6-[4-[7-[[1-[[7-(7,8-difluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027691	C[C@@]1(O)CCCN(C2=NC(OCC3(CN4CCC5(CC4)CC(N4CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC4)C5)CC3)=NC3=C2C=NC(C2=CC(O)=CC4=C2C(F)=C(F)C=C4)=C3F)C1	C53H58F3N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-DBOTW7	SCHEMBL27423014	3-[6-[9-[4-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperazin-1-yl]-3-azaspiro[5.5]undecan-3-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027721	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCN(C5CCC6(CC5)CCN(C5=CC7=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C7)CC6)CC4)CC1)=N3)=CC(O)=C2	C57H67F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-45W0ZN	SCHEMBL27423022	(3S)-3-[6-[4-[[7-[[1-[[7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-2-fluoro-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027515	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CC(F)(CN4CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC4)C5)CC1)=N3)=CC(O)=C2	C56H65F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-BAOSIP	SCHEMBL27423025	(3S)-3-[6-[4-[[7-[[1-[[7-(7,8-difluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-2-fluoro-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027668	C[C@@]1(O)CCCN(C2=NC(OCC3(CN4CCC5(CC4)CC(F)(CN4CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC4)C5)CC3)=NC3=C2C=NC(C2=CC(O)=CC4=C2C(F)=C(F)C=C4)=C3F)C1	C54H59F4N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-XGNEWB	SCHEMBL27423029	(3S)-3-[6-[4-[[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(6S)-6-hydroxy-6-methyl-1,4-oxazepan-4-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-2-fluoro-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027696	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCOC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CC(F)(CN4CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC4)C5)CC1)=N3)=CC(O)=C2	C56H64F3N9O7	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-WT5HGI	SCHEMBL27423033	3-[6-[4-[[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]oxy]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027480	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CC(OC4CCN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)CC4)C5)CC1)=N3)=CC(O)=C2	C56H64F2N8O7	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-M9LBJB	SCHEMBL27423034	(3S)-3-[6-[4-[[2-[[1-[[7-(7,8-difluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-fluoro-2-azaspiro[3.5]nonan-7-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027590	C[C@@]1(O)CCCN(C2=NC(OCC3(CN4CC5(CCC(F)(CN6CCN(C7=CC8=C(C=C7)C(=O)N([C@H]7CCC(=O)NC7=O)C8)CC6)CC5)C4)CC3)=NC3=C2C=NC(C2=CC(O)=CC4=C2C(F)=C(F)C=C4)=C3F)C1	C54H59F4N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-RSNXU1	SCHEMBL27423036	(3S)-3-[6-[4-[[2-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-fluoro-2-azaspiro[3.5]nonan-7-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027652	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CC5(CCC(F)(CN6CCN(C7=CC8=C(C=C7)C(=O)N([C@H]7CCC(=O)NC7=O)C8)CC6)CC5)C4)CC1)=N3)=CC(O)=C2	C56H64F3N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-K6VVC7	SCHEMBL27423039	(3S)-3-[6-[4-[[2-[[1-[[7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-fluoro-2-azaspiro[3.5]nonan-7-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027504	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CC5(CCC(F)(CN6CCN(C7=CC8=C(C=C7)C(=O)N([C@H]7CCC(=O)NC7=O)C8)CC6)CC5)C4)CC1)=N3)=CC(O)=C2	C56H65F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-005PQR	SCHEMBL27423040	N-[(3S)-2,6-dioxopiperidin-3-yl]-4-[4-[[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-2-fluoro-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]-2-fluorobenzamide; SCHEMBL31027508	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CC(F)(CN4CCN(C6=CC=C(C(=O)N[C@H]7CCC(=O)NC7=O)C(F)=C6)CC4)C5)CC1)=N3)=CC(O)=C2	C55H63F4N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-TIB6JP	WO2024118966A1_181	.	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@](C)(O)C1)=NC(OCC1(CN4CCC(OC5CC6(CCN(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8)CC6)C5)CC4)CC1)=N3)=CC(O)=C2	C56H65FN8O7	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-OCUDME	WO2024118966A1_182	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@](C)(O)C1)=NC(OCC1(CN4CCC(OC5CC6(CCN(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8)CC6)C5)CC4)CC1)=N3)=CC(O)=C2	C56H64F2N8O7	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-GISOXX	SCHEMBL27423056	N-[(3S)-2,6-dioxopiperidin-3-yl]-4-[4-[[2-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-fluoro-2-azaspiro[3.5]nonan-7-yl]methyl]piperazin-1-yl]-2-fluorobenzamide; SCHEMBL31027626	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CC5(CCC(F)(CN6CCN(C7=CC=C(C(=O)N[C@H]8CCC(=O)NC8=O)C(F)=C7)CC6)CC5)C4)CC1)=N3)=CC(O)=C2	C55H63F4N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-V4V8YB	SCHEMBL27423061	3-[6-[7-[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]oxy-2-azaspiro[3.5]nonan-2-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027727	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC(OC5CCC6(CC5)CN(C5=CC7=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C7)C6)CC4)CC1)=N3)=CC(O)=C2	C56H64F2N8O7	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-TKWPHA	SCHEMBL27423062	3-[6-[4-[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-2-fluoro-7-azaspiro[3.5]nonan-2-yl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027609	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CC(F)(C4CCN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)CC4)C5)CC1)=N3)=CC(O)=C2	C56H63F3N8O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-M2ID1P	SCHEMBL27423067	3-[6-[4-[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027569	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CC(C4CCN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)CC4)C5)CC1)=N3)=CC(O)=C2	C56H64F2N8O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-DYNH6Q	SCHEMBL27423068	(3S)-3-[6-[4-[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-6,8-difluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]quinazolin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027554	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=C1F)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CC(N4CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC4)C5)CC1)=N3)=CC(O)=C2	C56H63F3N8O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-R8T1GN	WO2024118966A1_188	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=C1F)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CC(F)(N4CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC4)C5)CC1)=N3)=CC(O)=C2	C56H62F4N8O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-ZNBOSE	SCHEMBL27423079	3-[4-[2-[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]oxy-7-azaspiro[3.5]nonan-7-yl]-2,6-difluorophenyl]piperidine-2,6-dione; SCHEMBL31027568	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC(OC5CC6(CCN(C7=CC(F)=C(C8CCC(=O)NC8=O)C(F)=C7)CC6)C5)CC4)CC1)=N3)=CC(O)=C2	C54H61F4N7O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-XCXZ01	SCHEMBL27423083	3-[4-[9-[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]oxy-3-azaspiro[5.5]undecan-3-yl]-2,6-difluorophenyl]piperidine-2,6-dione; SCHEMBL31027632	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC(OC5CCC6(CC5)CCN(C5=CC(F)=C(C7CCC(=O)NC7=O)C(F)=C5)CC6)CC4)CC1)=N3)=CC(O)=C2	C56H65F4N7O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-UUR70F	SCHEMBL27423097	3-[4-[4-[[3-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-9-fluoro-3-azaspiro[5.5]undecan-9-yl]methyl]piperazin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione; SCHEMBL31027539	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CCC(F)(CN4CCN(C6=CC(F)=C(C7CCC(=O)NC7=O)C(F)=C6)CC4)CC5)CC1)=N3)=CC(O)=C2	C56H65F5N8O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-X1TE2F	SCHEMBL27423103	3-[4-[4-[[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-2-fluoro-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]-2,6-difluoroanilino]piperidine-2,6-dione; SCHEMBL31027485	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CC(F)(CN4CCN(C6=CC(F)=C(NC7CCC(=O)NC7=O)C(F)=C6)CC4)C5)CC1)=N3)=CC(O)=C2	C54H62F5N9O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-3XHOTA	SCHEMBL27423105	3-[4-[4-[[3-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-3-azaspiro[5.5]undecan-9-yl]oxy]piperidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione; SCHEMBL31027643	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CCC(OC6CCN(C7=CC(F)=C(C8CCC(=O)NC8=O)C(F)=C7)CC6)CC5)CC4)CC1)=N3)=CC(O)=C2	C56H65F4N7O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-SMLXBM	SCHEMBL27423108	3-[4-[3-[[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-2,7-diazaspiro[3.5]nonan-2-yl]methyl]-3-fluoroazetidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione; SCHEMBL31027487	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CN(CC4(F)CN(C6=CC(F)=C(C7CCC(=O)NC7=O)C(F)=C6)C4)C5)CC1)=N3)=CC(O)=C2	C52H57F5N8O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-YGCFYS	SCHEMBL27423111	3-[4-[4-[[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-2,7-diazaspiro[3.5]nonan-2-yl]methyl]-4-fluoropiperidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione; SCHEMBL31027649	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CN(CC4(F)CCN(C6=CC(F)=C(C7CCC(=O)NC7=O)C(F)=C6)CC4)C5)CC1)=N3)=CC(O)=C2	C54H61F5N8O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-ECBC8S	WO2024118966A1_197	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CCC(F)(CN4CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=S)C7)CC4)CC5)CC1)=N3)=CC(O)=C2	C58H68F3N9O5S	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-DV5IXB	SCHEMBL27423117	(3S)-3-[6-[4-[[3-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-3-azaspiro[5.5]undecan-9-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027553	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CCC(CN6CCN(C7=CC8=C(C=C7)C(=O)N([C@H]7CCC(=O)NC7=O)C8)CC6)CC5)CC4)CC1)=N3)=CC(O)=C2	C58H69F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-UGYSL7	SCHEMBL27423120	3-[6-[4-[[3-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-3-azaspiro[5.5]undecan-9-yl]oxy]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027686	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CCC(OC6CCN(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8)CC6)CC5)CC4)CC1)=N3)=CC(O)=C2	C58H68F2N8O7	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-BE6WAY	SCHEMBL27423122	3-[6-[9-[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]oxy-3-azaspiro[5.5]undecan-3-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027482	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC(OC5CCC6(CC5)CCN(C5=CC7=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C7)CC6)CC4)CC1)=N3)=CC(O)=C2	C58H68F2N8O7	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-20VY4K	SCHEMBL27423126	3-[4-[4-[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]piperazin-1-yl]-2,6-difluoroanilino]piperidine-2,6-dione; SCHEMBL31027583	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CC(N4CCN(C6=CC(F)=C(NC7CCC(=O)NC7=O)C(F)=C6)CC4)C5)CC1)=N3)=CC(O)=C2	C53H61F4N9O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-YLC0Z0	WO2024118966A1_202	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CC(F)(N4CCN(C6=CC=C(NC7CCC(=O)NC7=O)C(F)=C6)CC4)C5)CC1)=N3)=CC(O)=C2	C53H61F4N9O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-98TBS3	WO2024118966A1_203	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CC(F)(N4CCN(C6=CC(F)=C(NC7CCC(=O)NC7=O)C(F)=C6)CC4)C5)CC1)=N3)=CC(O)=C2	C53H60F5N9O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-9FRAFZ	SCHEMBL27423141	3-[4-[4-[[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]-2,6-difluoroanilino]piperidine-2,6-dione; SCHEMBL31027663	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CC(CN4CCN(C6=CC(F)=C(NC7CCC(=O)NC7=O)C(F)=C6)CC4)C5)CC1)=N3)=CC(O)=C2	C54H63F4N9O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-1HK9MM	SCHEMBL27423145	3-[4-[1-[[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]methyl]piperidin-4-yl]-2,6-difluoroanilino]piperidine-2,6-dione; SCHEMBL31027566	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CC(CN4CCC(C6=CC(F)=C(NC7CCC(=O)NC7=O)C(F)=C6)CC4)C5)CC1)=N3)=CC(O)=C2	C55H64F4N8O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-L195W3	SCHEMBL27423146	(3S)-3-[6-[4-[[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-6,8-difluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]quinazolin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027617	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=C1F)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CC(CN4CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC4)C5)CC1)=N3)=CC(O)=C2	C57H65F3N8O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-WTO9XA	WO2024118966A1_207	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=C1F)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CC(CN4CCN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)CC4)C5)CC1)=N3)=CC(O)=C2	C57H65F3N8O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-H78I9K	WO2024118966A1_208	.	[H]C12CN(CC3(COC4=NC5=C(C=NC(C6=CC(O)=CC7=C6C(CC)=C(F)C=C7)=C5F)C(N5CCC[C@@](C)(O)C5)=N4)CC3)C[C@@]1([H])[C@@H]2CN1CCN(C2=CC3=C(C=C2)C(=O)N([C@H]2CCC(=O)NC2=O)C3)CC1	C53H59F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-P4EAR3	WO2024118966A1_209	.	[H]C12CN(CC3(COC4=NC5=C(C=NC(C6=CC(O)=CC7=C6C(CC)=C(F)C=C7)=C5F)C(N5CCC[C@@](C)(O)C5)=N4)CC3)C[C@@]1([H])[C@H]2CN1CCN(C2=CC3=C(C=C2)C(=O)N([C@H]2CCC(=O)NC2=O)C3)CC1	C53H59F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-KB4LK9	SCHEMBL27423160	(3S)-3-[6-[4-[[7-[[1-[[7-(8-chloro-7-fluoro-3-hydroxynaphthalen-1-yl)-6,8-difluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]quinazolin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027536	C[C@@]1(O)CCCN(C2=NC(OCC3(CN4CCC5(CC4)CC(CN4CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC4)C5)CC3)=NC3=C2C=C(F)C(C2=CC(O)=CC4=C2C(Cl)=C(F)C=C4)=C3F)C1	C55H60ClF3N8O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-VBAVMA	SCHEMBL27423162	(3S)-3-[6-[4-[[1-[[1-[[7-(8-chloro-7-fluoro-3-hydroxynaphthalen-1-yl)-6,8-difluoro-4-[(3S)-3-hydroxy-3-methylpiperidin-1-yl]quinazolin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027541	C[C@]1(O)CCCN(C2=NC(OCC3(CN4CCC(CN5CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC5)CC4)CC3)=NC3=C2C=C(F)C(C2=CC(O)=CC4=C2C(Cl)=C(F)C=C4)=C3F)C1	C52H56ClF3N8O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-ZIX5JS	SCHEMBL27423168	(3S)-3-[6-[4-[[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-(3-hydroxy-3-methylpiperidin-1-yl)pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027580	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCCC(C)(O)C1)=NC(OCC1(CN4CCC(CN5CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC5)CC4)CC1)=N3)=CC(O)=C2	C53H61F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-4KRR41	SCHEMBL27423170	(3S)-3-[6-[4-[1-[[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-4-methylpiperidin-4-yl]methyl]piperidin-4-yl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027602	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC(C)(CN5CCC(N6CCN(C7=CC8=C(C=C7)C(=O)N([C@H]7CCC(=O)NC7=O)C8)CC6)CC5)CC4)CC1)=N3)=CC(O)=C2	C59H72F2N10O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-1K1U33	SCHEMBL27423173	3-[4-[4-[[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(4S)-1-oxa-8-azaspiro[3.5]nonan-8-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione; SCHEMBL31027534	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@]4(CCO4)C1)=NC(OCC1(CN4CCC(CN5CCN(C6=CC(F)=C(C7CCC(=O)NC7=O)C(F)=C6)CC5)CC4)CC1)=N3)=CC(O)=C2	C52H58F4N8O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-K83UI7	SCHEMBL27422536	(3S)-3-[6-[4-[[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(4S)-1-oxa-8-azaspiro[3.5]nonan-8-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-4-methylpiperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027640	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@]4(CCO4)C1)=NC(OCC1(CN4CCC(C)(CN5CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC5)CC4)CC1)=N3)=CC(O)=C2	C55H63F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-YI303K	SCHEMBL27423179	(3S)-3-[6-[4-[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-4-(trifluoromethyl)piperidin-4-yl]oxypiperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027650	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC(OC5CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC5)(C(F)(F)F)CC4)CC1)=N3)=CC(O)=C2	C54H59F5N8O7	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-TUX0T0	SCHEMBL27423182	(3S)-3-[6-[4-[[4-ethyl-1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL31027596	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC(CC)(CN5CCN(C6=CC7=C(C=C6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC5)CC4)CC1)=N3)=CC(O)=C2	C55H65F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-RN6JQW	SCHEMBL27423185	3-[4-[4-[[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(4S)-1-oxa-8-azaspiro[3.5]nonan-8-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-4-methylpiperidin-4-yl]methyl]piperazin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione; SCHEMBL31027483	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@]4(CCO4)C1)=NC(OCC1(CN4CCC(C)(CN5CCN(C6=CC(F)=C(C7CCC(=O)NC7=O)C(F)=C6)CC5)CC4)CC1)=N3)=CC(O)=C2	C53H60F4N8O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-45REGD	SCHEMBL27423188	3-[4-[4-[[(2R)-4-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(4S)-1-oxa-8-azaspiro[3.5]nonan-8-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]morpholin-2-yl]methyl]piperazin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione; SCHEMBL31027597	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@]4(CCO4)C1)=NC(OCC1(CN4CCO[C@H](CN5CCN(C6=CC(F)=C(C7CCC(=O)NC7=O)C(F)=C6)CC5)C4)CC1)=N3)=CC(O)=C2	C51H56F4N8O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-JV2ZBR	SCHEMBL27423191	3-[4-[4-[[(2S)-4-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(4S)-1-oxa-8-azaspiro[3.5]nonan-8-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]morpholin-2-yl]methyl]piperazin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione; SCHEMBL31027613	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@]4(CCO4)C1)=NC(OCC1(CN4CCO[C@@H](CN5CCN(C6=CC(F)=C(C7CCC(=O)NC7=O)C(F)=C6)CC5)C4)CC1)=N3)=CC(O)=C2	C51H56F4N8O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-TF449Y	SCHEMBL27423192	3-[6-[4-[7-[[1-[[7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]piperazin-1-yl]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL31027738	CCC1=CC=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CC(N4CCN(C6=CC7=C(C=C6)C(C6CCC(=O)NC6=O)=NN7C)CC4)C5)CC1)=N3)=CC(O)=C2	C55H65FN10O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-S1EFYB	SCHEMBL27423198	3-[6-[4-[[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL31027647	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CC(CN4CCN(C6=CC7=C(C=C6)C(C6CCC(=O)NC6=O)=NN7C)CC4)C5)CC1)=N3)=CC(O)=C2	C56H66F2N10O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-ESVR02	SCHEMBL27423204	3-[6-[4-[[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-2-fluoro-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL31027724	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CC(F)(CN4CCN(C6=CC7=C(C=C6)C(C6CCC(=O)NC6=O)=NN7C)CC4)C5)CC1)=N3)=CC(O)=C2	C56H65F3N10O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-YTZJMN	SCHEMBL27423207	3-[6-[4-[[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL31027628	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC(CN5CCN(C6=CC7=C(C=C6)C(C6CCC(=O)NC6=O)=NN7C)CC5)CC4)CC1)=N3)=CC(O)=C2	C53H62F2N10O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-0HBCSA	SCHEMBL27423213	3-[6-[4-[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(4S)-1-oxa-8-azaspiro[3.5]nonan-8-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]piperazin-1-yl]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL31027563	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@]4(CCO4)C1)=NC(OCC1(CN4CCC5(CC4)CC(N4CCN(C6=CC7=C(C=C6)C(C6CCC(=O)NC6=O)=NN7C)CC4)C5)CC1)=N3)=CC(O)=C2	C56H64F2N10O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-7GV28V	SCHEMBL27423220	3-[6-[4-[[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(4S)-1-oxa-8-azaspiro[3.5]nonan-8-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL31027733	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@]4(CCO4)C1)=NC(OCC1(CN4CCC5(CC4)CC(CN4CCN(C6=CC7=C(C=C6)C(C6CCC(=O)NC6=O)=NN7C)CC4)C5)CC1)=N3)=CC(O)=C2	C57H66F2N10O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-DVSYFQ	SCHEMBL27423229	3-[6-[4-[[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(4S)-1-oxa-8-azaspiro[3.5]nonan-8-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL31027475	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@]4(CCO4)C1)=NC(OCC1(CN4CCC(CN5CCN(C6=CC7=C(C=C6)C(C6CCC(=O)NC6=O)=NN7C)CC5)CC4)CC1)=N3)=CC(O)=C2	C54H62F2N10O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-M1L08G	SCHEMBL27423233	3-[6-[4-[[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(4S)-1-oxa-8-azaspiro[3.5]nonan-8-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-4-fluoropiperidin-4-yl]methyl]piperazin-1-yl]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL31027619	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@]4(CCO4)C1)=NC(OCC1(CN4CCC(F)(CN5CCN(C6=CC7=C(C=C6)C(C6CCC(=O)NC6=O)=NN7C)CC5)CC4)CC1)=N3)=CC(O)=C2	C54H61F3N10O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-JSTV9R	SCHEMBL27423238	3-[5-[4-[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]piperazin-1-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione; SCHEMBL31027523	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CC(N4CCN(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC4)C5)CC1)=N3)=CC(O)=C2	C55H64F2N10O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-V091X8	SCHEMBL27423242	3-[5-[4-[[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione; SCHEMBL31027705	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CC(CN4CCN(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC4)C5)CC1)=N3)=CC(O)=C2	C56H66F2N10O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-ADVAVQ	SCHEMBL27423246	3-[5-[4-[[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione; SCHEMBL31027500	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC(CN5CCN(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC5)CC4)CC1)=N3)=CC(O)=C2	C53H62F2N10O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-SHV33C	SCHEMBL27423249	3-[5-[4-[[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(4S)-1-oxa-8-azaspiro[3.5]nonan-8-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione; SCHEMBL31027501	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@]4(CCO4)C1)=NC(OCC1(CN4CCC5(CC4)CC(CN4CCN(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC4)C5)CC1)=N3)=CC(O)=C2	C57H66F2N10O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-B1WNNC	SCHEMBL27423251	3-[5-[4-[[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(4S)-1-oxa-8-azaspiro[3.5]nonan-8-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione; SCHEMBL31027481	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@]4(CCO4)C1)=NC(OCC1(CN4CCC(CN5CCN(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC5)CC4)CC1)=N3)=CC(O)=C2	C54H62F2N10O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-YQEMU9	SCHEMBL27423253	3-[5-[4-[[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(4S)-1-oxa-8-azaspiro[3.5]nonan-8-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-4-fluoropiperidin-4-yl]methyl]piperazin-1-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione; SCHEMBL31027711	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@]4(CCO4)C1)=NC(OCC1(CN4CCC(F)(CN5CCN(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC5)CC4)CC1)=N3)=CC(O)=C2	C54H61F3N10O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-D7F8U3	SCHEMBL27423254	3-[6-[4-[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]piperazin-1-yl]-2-oxo-1,3-benzoxazol-3-yl]piperidine-2,6-dione; SCHEMBL31027479	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CC(N4CCN(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)O7)CC4)C5)CC1)=N3)=CC(O)=C2	C54H61F2N9O7	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-L87K5X	SCHEMBL27423257	3-[6-[4-[[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]-2-oxo-1,3-benzoxazol-3-yl]piperidine-2,6-dione; SCHEMBL31027489	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CC(CN4CCN(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)O7)CC4)C5)CC1)=N3)=CC(O)=C2	C55H63F2N9O7	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-D3R75C	SCHEMBL27423262	3-[6-[4-[[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-2-fluoro-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]-2-oxo-1,3-benzoxazol-3-yl]piperidine-2,6-dione; SCHEMBL31027710	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CC(F)(CN4CCN(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)O7)CC4)C5)CC1)=N3)=CC(O)=C2	C55H62F3N9O7	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-1XTNLM	SCHEMBL27423267	3-[6-[4-[[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-oxo-1,3-benzoxazol-3-yl]piperidine-2,6-dione; SCHEMBL31027660	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC(CN5CCN(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)O7)CC5)CC4)CC1)=N3)=CC(O)=C2	C52H59F2N9O7	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-41WLS0	SCHEMBL27423275	3-[6-[4-[[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-4-fluoropiperidin-4-yl]methyl]piperazin-1-yl]-2-oxo-1,3-benzoxazol-3-yl]piperidine-2,6-dione; SCHEMBL31027502	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC(F)(CN5CCN(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)O7)CC5)CC4)CC1)=N3)=CC(O)=C2	C52H58F3N9O7	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-7HQPT2	SCHEMBL27423277	3-[6-[4-[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(4S)-1-oxa-8-azaspiro[3.5]nonan-8-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]piperazin-1-yl]-2-oxo-1,3-benzoxazol-3-yl]piperidine-2,6-dione; SCHEMBL31027545	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@]4(CCO4)C1)=NC(OCC1(CN4CCC5(CC4)CC(N4CCN(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)O7)CC4)C5)CC1)=N3)=CC(O)=C2	C55H61F2N9O7	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-8C1U2E	SCHEMBL27423281	3-[6-[4-[[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(4S)-1-oxa-8-azaspiro[3.5]nonan-8-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]-2-oxo-1,3-benzoxazol-3-yl]piperidine-2,6-dione; SCHEMBL31027564	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@]4(CCO4)C1)=NC(OCC1(CN4CCC5(CC4)CC(CN4CCN(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)O7)CC4)C5)CC1)=N3)=CC(O)=C2	C56H63F2N9O7	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-G6LWVG	SCHEMBL27423285	3-[6-[4-[[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(4S)-1-oxa-8-azaspiro[3.5]nonan-8-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-2-fluoro-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]-2-oxo-1,3-benzoxazol-3-yl]piperidine-2,6-dione; SCHEMBL31027720	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@]4(CCO4)C1)=NC(OCC1(CN4CCC5(CC4)CC(F)(CN4CCN(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)O7)CC4)C5)CC1)=N3)=CC(O)=C2	C56H62F3N9O7	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-V5O099	SCHEMBL27423288	3-[6-[4-[[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(4S)-1-oxa-8-azaspiro[3.5]nonan-8-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]-2-oxo-1,3-benzoxazol-3-yl]piperidine-2,6-dione; SCHEMBL31027535	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@]4(CCO4)C1)=NC(OCC1(CN4CCC(CN5CCN(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)O7)CC5)CC4)CC1)=N3)=CC(O)=C2	C53H59F2N9O7	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-YKZU4I	SCHEMBL27423292	3-[6-[4-[[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(4S)-1-oxa-8-azaspiro[3.5]nonan-8-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-4-fluoropiperidin-4-yl]methyl]piperazin-1-yl]-2-oxo-1,3-benzoxazol-3-yl]piperidine-2,6-dione; SCHEMBL31027595	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@]4(CCO4)C1)=NC(OCC1(CN4CCC(F)(CN5CCN(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)O7)CC5)CC4)CC1)=N3)=CC(O)=C2	C53H58F3N9O7	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-YUMIR3	SCHEMBL27423296	3-[5-[4-[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]piperazin-1-yl]indazol-1-yl]piperidine-2,6-dione; SCHEMBL31027537	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CC(N4CCN(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)N=C7)CC4)C5)CC1)=N3)=CC(O)=C2	C54H62F2N10O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-N4L0VT	SCHEMBL27423298	3-[5-[4-[[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]indazol-1-yl]piperidine-2,6-dione; SCHEMBL31027653	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CC(CN4CCN(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)N=C7)CC4)C5)CC1)=N3)=CC(O)=C2	C55H64F2N10O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-5C145Y	SCHEMBL27423305	3-[5-[4-[[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-2-fluoro-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]indazol-1-yl]piperidine-2,6-dione; SCHEMBL31027531	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CC(F)(CN4CCN(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)N=C7)CC4)C5)CC1)=N3)=CC(O)=C2	C55H63F3N10O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-O5IC2J	SCHEMBL27423306	3-[5-[4-[[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]indazol-1-yl]piperidine-2,6-dione; SCHEMBL31027644	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC(CN5CCN(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)N=C7)CC5)CC4)CC1)=N3)=CC(O)=C2	C52H60F2N10O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-X0SHKQ	SCHEMBL27423308	3-[5-[4-[[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-4-fluoropiperidin-4-yl]methyl]piperazin-1-yl]indazol-1-yl]piperidine-2,6-dione; SCHEMBL31027670	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC(F)(CN5CCN(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)N=C7)CC5)CC4)CC1)=N3)=CC(O)=C2	C52H59F3N10O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-BCGW06	SCHEMBL27423312	3-[5-[4-[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(4S)-1-oxa-8-azaspiro[3.5]nonan-8-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]piperazin-1-yl]indazol-1-yl]piperidine-2,6-dione; SCHEMBL31027601	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@]4(CCO4)C1)=NC(OCC1(CN4CCC5(CC4)CC(N4CCN(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)N=C7)CC4)C5)CC1)=N3)=CC(O)=C2	C55H62F2N10O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-3E5QB0	SCHEMBL27423316	3-[5-[4-[[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(4S)-1-oxa-8-azaspiro[3.5]nonan-8-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]indazol-1-yl]piperidine-2,6-dione; SCHEMBL31027673	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@]4(CCO4)C1)=NC(OCC1(CN4CCC5(CC4)CC(CN4CCN(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)N=C7)CC4)C5)CC1)=N3)=CC(O)=C2	C56H64F2N10O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-H12M37	SCHEMBL27423319	3-[5-[4-[[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(4S)-1-oxa-8-azaspiro[3.5]nonan-8-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-2-fluoro-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]indazol-1-yl]piperidine-2,6-dione; SCHEMBL31027578	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@]4(CCO4)C1)=NC(OCC1(CN4CCC5(CC4)CC(F)(CN4CCN(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)N=C7)CC4)C5)CC1)=N3)=CC(O)=C2	C56H63F3N10O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-LH8JMK	SCHEMBL27423323	3-[5-[4-[[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(4S)-1-oxa-8-azaspiro[3.5]nonan-8-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]indazol-1-yl]piperidine-2,6-dione; SCHEMBL31027497	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@]4(CCO4)C1)=NC(OCC1(CN4CCC(CN5CCN(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)N=C7)CC5)CC4)CC1)=N3)=CC(O)=C2	C53H60F2N10O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-DPWB9M	SCHEMBL27423328	3-[5-[4-[[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(4S)-1-oxa-8-azaspiro[3.5]nonan-8-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-4-fluoropiperidin-4-yl]methyl]piperazin-1-yl]indazol-1-yl]piperidine-2,6-dione; SCHEMBL31027661	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@]4(CCO4)C1)=NC(OCC1(CN4CCC(F)(CN5CCN(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)N=C7)CC5)CC4)CC1)=N3)=CC(O)=C2	C53H59F3N10O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-GO7RYS	SCHEMBL27423333	3-[5-[4-[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]piperazin-1-yl]-3,3-dimethyl-2-oxoindol-1-yl]piperidine-2,6-dione; SCHEMBL31027560	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CC(N4CCN(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)C7(C)C)CC4)C5)CC1)=N3)=CC(O)=C2	C57H67F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-O7XFRF	SCHEMBL27423340	3-[5-[4-[[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]-3,3-dimethyl-2-oxoindol-1-yl]piperidine-2,6-dione; SCHEMBL31027672	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CC(CN4CCN(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)C7(C)C)CC4)C5)CC1)=N3)=CC(O)=C2	C58H69F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-W3I2D8	SCHEMBL27423345	3-[5-[4-[[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-2-fluoro-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]-3,3-dimethyl-2-oxoindol-1-yl]piperidine-2,6-dione; SCHEMBL31027622	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CC(F)(CN4CCN(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)C7(C)C)CC4)C5)CC1)=N3)=CC(O)=C2	C58H68F3N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-UHFV1K	SCHEMBL27423348	3-[5-[4-[[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]methyl]piperazin-1-yl]-3,3-dimethyl-2-oxoindol-1-yl]piperidine-2,6-dione; SCHEMBL31027664	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC(CN5CCN(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)C7(C)C)CC5)CC4)CC1)=N3)=CC(O)=C2	C55H65F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-O6RUBX	SCHEMBL27423351	3-[5-[4-[[1-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-4-fluoropiperidin-4-yl]methyl]piperazin-1-yl]-3,3-dimethyl-2-oxoindol-1-yl]piperidine-2,6-dione; SCHEMBL31027692	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC(F)(CN5CCN(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)C7(C)C)CC5)CC4)CC1)=N3)=CC(O)=C2	C55H64F3N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-YNJFPN	SCHEMBL27423353	3-[5-[4-[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(4S)-1-oxa-8-azaspiro[3.5]nonan-8-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]piperazin-1-yl]-3,3-dimethyl-2-oxoindol-1-yl]piperidine-2,6-dione; SCHEMBL31027731	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@]4(CCO4)C1)=NC(OCC1(CN4CCC5(CC4)CC(N4CCN(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)C7(C)C)CC4)C5)CC1)=N3)=CC(O)=C2	C58H67F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-AMTV23	SCHEMBL27423355	3-[5-[4-[[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(4S)-1-oxa-8-azaspiro[3.5]nonan-8-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]-3,3-dimethyl-2-oxoindol-1-yl]piperidine-2,6-dione; SCHEMBL31027709	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@]4(CCO4)C1)=NC(OCC1(CN4CCC5(CC4)CC(CN4CCN(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)C7(C)C)CC4)C5)CC1)=N3)=CC(O)=C2	C59H69F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-0JQVE6	SCHEMBL27423360	3-[5-[4-[[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(4S)-1-oxa-8-azaspiro[3.5]nonan-8-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-2-fluoro-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]-3,3-dimethyl-2-oxoindol-1-yl]piperidine-2,6-dione; SCHEMBL31027470	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@]4(CCO4)C1)=NC(OCC1(CN4CCC5(CC4)CC(F)(CN4CCN(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)C7(C)C)CC4)C5)CC1)=N3)=CC(O)=C2	C59H68F3N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-LFKB0U	WO2024118966A1_268	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCCC4(CCO4)C1)=NC(OCC1(CN4CCC(CN5CCN(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)C7(C)C)CC5)CC4)CC1)=N3)=CC(O)=C2	C56H65F2N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-IQQF8Y	WO2024118966A1_269	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCCC4(CCO4)C1)=NC(OCC1(CN4CCC(F)(CN5CCN(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)C7(C)C)CC5)CC4)CC1)=N3)=CC(O)=C2	C56H64F3N9O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-NFSSYS	SCHEMBL27423382	3-[5-[4-[[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-2-fluoro-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione; SCHEMBL31027522	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CC(F)(CN4CCN(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC4)C5)CC1)=N3)=CC(O)=C2	C56H65F3N10O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-3JVBF8	SCHEMBL27423388	3-[5-[4-[[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(4S)-1-oxa-8-azaspiro[3.5]nonan-8-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-2-fluoro-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione; SCHEMBL31027646	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@]4(CCO4)C1)=NC(OCC1(CN4CCC5(CC4)CC(F)(CN4CCN(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC4)C5)CC1)=N3)=CC(O)=C2	C57H65F3N10O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-1IKC7N	SCHEMBL27431333	3-[5-[4-[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(4S)-1-oxa-8-azaspiro[3.5]nonan-8-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]piperazin-1-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione; SCHEMBL31027589	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@]4(CCO4)C1)=NC(OCC1(CN4CCC5(CC4)CC(N4CCN(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC4)C5)CC1)=N3)=CC(O)=C2	C56H64F2N10O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-LCR19R	SCHEMBL27423390	3-[6-[4-[[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(4S)-1-oxa-8-azaspiro[3.5]nonan-8-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-2-fluoro-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL31027634	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@]4(CCO4)C1)=NC(OCC1(CN4CCC5(CC4)CC(F)(CN4CCN(C6=CC7=C(C=C6)C(C6CCC(=O)NC6=O)=NN7C)CC4)C5)CC1)=N3)=CC(O)=C2	C57H65F3N10O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-4ED3PZ	SCHEMBL27430490	3-[6-[4-[7-[[1-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(3R)-3-hydroxy-3-methylpiperidin-1-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-7-azaspiro[3.5]nonan-2-yl]piperazin-1-yl]-1-methylindazol-3-yl]piperidine-2,6-dione; SCHEMBL31027669	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCC5(CC4)CC(N4CCN(C6=CC7=C(C=C6)C(C6CCC(=O)NC6=O)=NN7C)CC4)C5)CC1)=N3)=CC(O)=C2	C55H64F2N10O5	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-UREVXX	SCHEMBL31027571	N-[(3R)-1-[2-[[1-[[4-[[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperazin-1-yl]methyl]-4-fluoropiperidin-1-yl]methyl]cyclopropyl]methoxy]-7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-4-yl]piperidin-3-yl]acetamide	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@H](NC(C)=O)C1)=NC(OCC1(CN4CCC(F)(CN5CCN(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC5)CC4)CC1)=N3)=CC(O)=C2	C54H62F3N11O6	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-VXESMZ	SCHEMBL31027493	methyl N-[(3R)-1-[2-[[1-[[4-[[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperazin-1-yl]methyl]-4-fluoropiperidin-1-yl]methyl]cyclopropyl]methoxy]-7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-4-yl]piperidin-3-yl]carbamate	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=N1)C(N1CCC[C@@H](NC(=O)OC)C1)=NC(OCC1(CN4CCC(F)(CN5CCN(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC5)CC4)CC1)=N3)=CC(O)=C2	C54H62F3N11O7	KRAS	P01116	CRBN	WO-2024118966-A1
TPD-N5TALJ	WO2024120424A1_1	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCCC(C)(O)C5)nc(OCC5(CN6CCC(COc7ccc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)cc7)CC6)CC5)nc4c3F)c12	C66H77F2N9O8S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-9DSXA7	WO2024120424A1_2	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCCC(C)(O)C5)nc(OC[C@]56CCCN5[C@@H](COC(=O)N5CCC7(CC5)CC(C(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)c5ccc(-c8scnc8C)cc5)C(C)(C)C)C7)CC6)nc4c3F)c12	C67H82F2N10O9S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-E89U7F	WO2024120424A1_3	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCCC(C)(O)C5)nc(OCC5(CN6CCC(COc7ccc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)cc7)CC6)CC5)nc4c3F)c12	C66H73F2N9O8S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-4R5Y0Q	WO2024120424A1_4	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)c2ccc(OCC3CCN(CC4(COc5nc(N6CCCC(C)(O)C6)c6cnc(-c7cc(O)cc8ccc(F)c(F)c78)c(F)c6n5)CC4)CC3)cc2)C(C)(C)C)cc1	C64H72F3N9O8S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-D11NZE	WO2024120424A1_5	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCCC(C)(O)C5)nc(OCC5(CN6CCC7(CC6)CN(c6ccc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)cc6)C7)CC5)nc4c3F)c12	C67H74F2N10O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-EAC62O	WO2024120424A1_6	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCCC(C)(O)C5)nc(OCC5(CN6CCC7(CC6)CN(c6ccc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)cc6)C7)CC5)nc4c3F)c12	C67H78F2N10O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-UELX8R	WO2024120424A1_7	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCCC(C)(O)C5)nc(OCC5(CN6CCC7(CC6)CC(c6cn([C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)nn6)C7)CC5)nc4c3F)c12	C63H71F2N11O6S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-I05AFK	WO2024120424A1_8	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCCC(C)(O)C5)nc(OCC5(CN6CCC7(CC6)CC(c6cn([C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)nn6)C7)CC5)nc4c3F)c12	C63H75F2N11O6S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-PAED2O	WO2024120424A1_9	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCCC(C)(O)C5)nc(OC[C@]56CCCN5[C@@H](COC(=O)N5CCC7(CC5)CC(c5cn([C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)nn5)C7)CC6)nc4c3F)c12	C68H78F2N12O8S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-CLIAHT	WO2024120424A1_10	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCCC(C)(O)C5)nc(OC[C@]56CCCN5[C@@H](COC(=O)N5CCC7(CC5)CC(c5cn([C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)nn5)C7)CC6)nc4c3F)c12	C68H82F2N12O8S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-O8A78W	WO2024120424A1_11	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](n2cc(C3CC4(CCN(C(=O)OC[C@H]5CC[C@@]6(COc7nc(N8CCCC(C)(O)C8)c8cc(Cl)c(-c9cccc%10sc(N)c(C#N)c9%10)c(F)c8n7)CCCN56)CC4)C3)nn2)C(C)(C)C)cc1	C66H77ClFN13O7S2	KRAS	P01116	VHL	WO-2024120424-A1
TPD-TZYW8S	WO2024120424A1_12	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCCC(C)(O)C5)nc(OCC5(CN(C)CC6CC7(C6)CN(c6ccc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)cc6)C7)CC5)nc4c3F)c12	C68H76F2N10O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-9A79SY	WO2024120424A1_13	.	CCn1nccc1-c1ccc([C@H](CO)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](C(C)C)n2cc(C3CC4(CCN(C(=O)OC[C@H]5CC[C@@]6(COc7nc(N8CCCC(C)(O)C8)c8cc(Cl)c(-c9cccc%10sc(N)c(C#N)c9%10)c(F)c8n7)CCCN56)CC4)C3)nn2)cc1	C66H78ClFN14O8S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-7XF45R	WO2024120424A1_14	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCCC(C)(O)C5)nc(OCC5(CN6CCC7(CC6)CC(Oc6ccc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)cc6)C7)CC5)nc4c3F)c12	C68H75F2N9O8S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-8BOIMM	WO2024120424A1_15	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CC3(C2)CN(C(=O)OC[C@H]2CC[C@@]4(COc5nc(N6CCCC(C)(O)C6)c6cc(Cl)c(-c7cccc8sc(N)c(C#N)c78)c(F)c6n5)CCCN24)C3)C(C)(C)C)cc1	C63H73ClFN11O8S2	KRAS	P01116	VHL	WO-2024120424-A1
TPD-41EGYG	WO2024120424A1_16	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCCC(C)(O)C5)nc(OCC5(CN(C)C6CCC7(CC6)CN(c6ccc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)cc6)C7)CC5)nc4c3F)c12	C69H78F2N10O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-XQQPJ9	WO2024120424A1_17	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CC2C(=O)[C@@H](NC(=O)c2ccc(OCC3CCN(CC4(COc5nc(N6CCCC(C)(O)C6)c6cc(Cl)c(-c7cccc8sc(N)c(C#N)c78)c(F)c6n5)CC4)CC3)cc2)C(C)(C)C)cc1	C65H73ClFN9O7S2	KRAS	P01116	VHL	WO-2024120424-A1
TPD-YT942Y	WO2024120424A1_18	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCCC(C)(O)C5)nc(OCC5(CN6CCC7(CC6)CCN(c6ccc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)cc6)CC7)CC5)nc4c3F)c12	C69H78F2N10O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-TG1LGN	WO2024120424A1_19	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](n2cc(-c3ccc(OC[C@H]4CC[C@@]5(COc6nc(N7CCCC(C)(O)C7)c7cc(Cl)c(-c8cccc9sc(N)c(C#N)c89)c(F)c7n6)CCCN45)nc3)nn2)C(C)(C)C)cc1	C62H67ClFN13O6S2	KRAS	P01116	VHL	WO-2024120424-A1
TPD-FSO597	WO2024120424A1_20	.	CCc1c(F)ccc2cc(O)cc(-c3ccc4c(N5CCCC(C)(O)C5)nc(OC[C@]56CCCN5[C@@H](COC(=O)N5CCC7(CC5)CC(c5cn([C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)nn5)C7)CC6)nc4c3F)c12	C69H83F2N11O8S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-ZME4WU	WO2024120424A1_21	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](n2cc(-c3ccc(OC[C@H]4CC[C@@]5(COc6nc(N7CCCC(C)(O)C7)c7cc(Cl)c(-c8cccc9sc(N)c(C#N)c89)c(F)c7n6)CCCN45)cc3)nn2)C(C)(C)C)cc1	C63H68ClFN12O6S2	KRAS	P01116	VHL	WO-2024120424-A1
TPD-AFYSN8	WO2024120424A1_22	.	CCc1c(F)ccc2cc(O)cc(-c3c(F)cc4c(N5CCCC(C)(O)C5)nc(OC[C@]56CCCN5[C@@H](COC(=O)N5CCC7(CC5)CC(c5cn([C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)nn5)C7)CC6)nc4c3F)c12	C69H82F3N11O8S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-SUCKBR	WO2024120424A1_23	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](n2cc(C3CCN(C(=O)OC[C@H]4CC[C@@]5(COc6nc(N7CCCC(C)(O)C7)c7cc(Cl)c(-c8cccc9sc(N)c(C#N)c89)c(F)c7n6)CCCN45)CC3)nn2)C(C)(C)C)cc1	C63H73ClFN13O7S2	KRAS	P01116	VHL	WO-2024120424-A1
TPD-FK9AYI	WO2024120424A1_24	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](n2cc(C3CC4(CCN(C(=O)OC[C@H]5CC[C@@]6(COc7nc(N8CCCC(C)(O)C8)c8cc(F)c(-c9cc(O)cc%10ccc(F)c(F)c9%10)c(F)c8n7)CCCN56)CC4)C3)nn2)C(C)(C)C)cc1	C67H77F4N11O8S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-T15VAJ	WO2024120424A1_25	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](n2cc(-c3ccc(NC(=O)OC[C@H]4CC[C@@]5(COc6nc(N7CCCC(C)(O)C7)c7cc(Cl)c(-c8cccc9sc(N)c(C#N)c89)c(F)c7n6)CCCN45)cc3)nn2)C(C)(C)C)cc1	C64H69ClFN13O7S2	KRAS	P01116	VHL	WO-2024120424-A1
TPD-XTNNZN	WO2024120424A1_26	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](n2cc(C3CC4(CCN(C(=O)OC[C@H]5CC[C@@]6(COc7nc(N8CCCC(C)(O)C8)c8ccc(-c9cc(O)cc%10ccc(F)c(F)c9%10)c(F)c8n7)CCCN56)CC4)C3)nn2)C(C)(C)C)cc1	C67H78F3N11O8S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-3IMOYK	WO2024120424A1_27	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CC2CCN(C(=O)OC[C@H]3CC[C@@]4(COc5nc(N6CCCC(C)(O)C6)c6cc(Cl)c(-c7cccc8sc(N)c(C#N)c78)c(F)c6n5)CCCN34)CC2)C(C)(C)C)cc1	C63H75ClFN11O8S2	KRAS	P01116	VHL	WO-2024120424-A1
TPD-OFKILD	WO2024120424A1_28	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](n2cc(C3CC4(CCN(C(=O)OC[C@H]5CC[C@@]6(COc7nc(N8CCCC(C)(O)C8)c8cc(Cl)c(-c9ccc(F)c%10sc(N)c(C#N)c9%10)c(F)c8n7)CCCN56)CC4)C3)nn2)C(C)(C)C)cc1	C66H76ClF2N13O7S2	KRAS	P01116	VHL	WO-2024120424-A1
TPD-EF7WJ6	WO2024120424A1_29	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CC3(CCN(C(=O)OC[C@H]4CC[C@@]5(COc6nc(N7CCCC(C)(O)C7)c7cc(Cl)c(-c8cccc9sc(N)c(C#N)c89)c(F)c7n6)CCCN45)CC3)C2)C(C)(C)C)cc1	C65H77ClFN11O8S2	KRAS	P01116	VHL	WO-2024120424-A1
TPD-D36B2Q	WO2024120424A1_30	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](n2cc(C3CC4(CCN(C(=O)OC[C@H]5CC[C@@]6(COc7nc(N8CCCC(C)(O)C8)c8cc(Cl)c(-c9ccc(F)c%10sc(N)nc9%10)c(F)c8n7)CCCN56)CC4)C3)nn2)C(C)(C)C)cc1	C64H76ClF2N13O7S2	KRAS	P01116	VHL	WO-2024120424-A1
TPD-SKNBHW	WO2024120424A1_31	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCCC(C)(O)C5)nc(OCC5(CN(C)CC6CN(c7ccc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)NCc8ccc(-c9scnc9C)cc8)C(C)(C)C)cc7)C6)CC5)nc4c3F)c12	C64H70F2N10O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-GADCK0	WO2024120424A1_32	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCCC(C)(O)C5)nc(OCC5(CN6CCC(OCc7ccc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)NCc8ccc(-c9scnc9C)cc8)C(C)(C)C)cc7)CC6)CC5)nc4c3F)c12	C65H71F2N9O8S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-0XLE5U	WO2024120424A1_33	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCCC(C)(O)C5)nc(OCC5(CN6CCC(Oc7ccc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)NCc8ccc(-c9scnc9C)cc8)C(C)(C)C)cc7)CC6)CC5)nc4c3F)c12	C64H69F2N9O8S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-UPB3VK	WO2024120424A1_35	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCCC(C)(O)C5)nc(OCC5(CN(C)Cc6ccc(N7CCC(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)CC7)cc6)CC5)nc4c3F)c12	C67H76F2N10O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-2RMTMQ	WO2024120424A1_36	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCCC(C)(O)C5)nc(OCC5(CN6CC7(CCN(c8ccc(C(=O)N[C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)(C)C)cc8)CC7)C6)CC5)nc4c3F)c12	C67H74F2N10O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-TPRO2J	WO2024120424A1_37	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](n2cc(C3CC4(CCN(C(=O)OC[C@H]5CC[C@@]6(COc7nc(N8CCCn9nc(C(=O)N(C)C)cc9C8)c8cc(Cl)c(-c9cccc%10sc(N)c(C#N)c9%10)c(F)c8n7)CCCN56)CC4)C3)nn2)C(C)(C)C)cc1	C70H80ClFN16O7S2	KRAS	P01116	VHL	WO-2024120424-A1
TPD-11BUCJ	WO2024120424A1_38	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCCn6nc(C(=O)N(C)C)cc6C5)nc(OCC5(CN6CCC(OCc7ccc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)NCc8ccc(-c9scnc9C)cc8)C(C)(C)C)cc7)CC6)CC5)nc4c3F)c12	C69H74F2N12O8S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-FCVFJ1	WO2024120424A1_39	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](n2cc(-c3ccc(OC[C@H]4CC[C@@]5(COc6nc(N7CCCn8nc(C(=O)N(C)C)cc8C7)c7cc(Cl)c(-c8cccc9sc(N)c(C#N)c89)c(F)c7n6)CCCN45)cc3)nn2)C(C)(C)C)cc1	C67H71ClFN15O6S2	KRAS	P01116	VHL	WO-2024120424-A1
TPD-MUAJC5	WO2024120424A1_40	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCCn6nc(C(=O)N(C)C)cc6C5)nc(OCC5(CN6CCC(COc7ccc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)NCc8ccc(-c9scnc9C)cc8)C(C)(C)C)cc7)CC6)CC5)nc4c3F)c12	C69H74F2N12O8S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-4HI5F5	WO2024120424A1_42	.	CCc1c(F)ccc2cc(O)cc(-c3c(F)cc4c(N5CCCn6nc(C(=O)N(C)C)cc6C5)nc(OC[C@]56CCCN5[C@@H](COC(=O)N5CCC7(CC5)CC(c5cn([C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)nn5)C7)CC6)nc4c3F)c12	C73H85F3N14O8S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-FAUNPN	WO2024120424A1_43	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCCn6nc(C(=O)N(C)C)cc6C5)nc(OCC5(CN6CCC7(CC6)CN(c6ccc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)cc6)C7)CC5)nc4c3F)c12	C71H77F2N13O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-INT6W3	WO2024120424A1_44	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCCn6nc(C(=O)N(C)C)cc6C5)nc(OC[C@@]56CCCN5[C@H](COC(=O)N5CCC7(CC5)CC(C(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)c5ccc(-c8scnc8C)cc5)C(C)(C)C)C7)CC6)nc4c3F)c12	C71H85F2N13O9S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-U687PY	WO2024120424A1_45	.	CCc1c(F)ccc2cc(O)cc(-c3ccc4c(N5CCCn6nc(C(=O)N(C)C)cc6C5)nc(OC[C@]56CCCN5[C@@H](COC(=O)N5CCC7(CC5)CC(c5cn([C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)nn5)C7)CC6)nc4c3F)c12	C73H86F2N14O8S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-NRBM2E	WO2024120424A1_46	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)c2ccc(OCC3CCN(CC4(COc5nc(N6CCCn7nc(C(=O)N(C)C)cc7C6)c6cnc(-c7cc(O)cc8ccc(F)c(F)c78)c(F)c6n5)CC4)CC3)cc2)C(C)(C)C)cc1	C67H73F3N12O8S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-E47XO4	WO2024120424A1_47	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](n2cc(C3CC4(CCN(C(=O)OC[C@H]5CC[C@@]6(COc7nc(N8CCOCC(C)(O)C8)c8cc(Cl)c(-c9cccc%10sc(N)c(C#N)c9%10)c(F)c8n7)CCCN56)CC4)C3)nn2)C(C)(C)C)cc1	C66H77ClFN13O8S2	KRAS	P01116	VHL	WO-2024120424-A1
TPD-BGB87R	WO2024120424A1_48	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCOCC(C)(O)C5)nc(OCC5(CN6CCC(OCc7ccc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)NCc8ccc(-c9scnc9C)cc8)C(C)(C)C)cc7)CC6)CC5)nc4c3F)c12	C65H71F2N9O9S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-78QHQ5	WO2024120424A1_49	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](n2cc(-c3ccc(OC[C@H]4CC[C@@]5(COc6nc(N7CCOCC(C)(O)C7)c7cc(Cl)c(-c8cccc9sc(N)c(C#N)c89)c(F)c7n6)CCCN45)cc3)nn2)C(C)(C)C)cc1	C63H68ClFN12O7S2	KRAS	P01116	VHL	WO-2024120424-A1
TPD-WQSRZM	WO2024120424A1_50	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCOCC(C)(O)C5)nc(OCC5(CN6CCC(COc7ccc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)NCc8ccc(-c9scnc9C)cc8)C(C)(C)C)cc7)CC6)CC5)nc4c3F)c12	C65H71F2N9O9S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-UJZXIQ	WO2024120424A1_51	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCCC6(CC(O)C6)C5)nc(OC[C@]56CCCN5[C@@H](COC(=O)N5CCC7(CC5)CC(c5cn([C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)nn5)C7)CC6)nc4c3F)c12	C70H80F2N12O8S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-2WBU5N	WO2024120424A1_52	.	CCc1c(F)ccc2cc(O)cc(-c3c(F)cc4c(N5CCCC6(CC(O)C6)C5)nc(OC[C@]56CCCN5[C@@H](COC(=O)N5CCC7(CC5)CC(c5cn([C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)nn5)C7)CC6)nc4c3F)c12	C71H84F3N11O8S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-JJSRCD	WO2024120424A1_53	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCCC6(CC(O)C6)C5)nc(OCC5(CN6CCC7(CC6)CN(c6ccc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)cc6)C7)CC5)nc4c3F)c12	C69H76F2N10O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-SE4QLN	WO2024120424A1_54	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCCC6(CC(O)C6)C5)nc(OC[C@@]56CCCN5[C@H](COC(=O)N5CCC7(CC5)CC(C(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)c5ccc(-c8scnc8C)cc5)C(C)(C)C)C7)CC6)nc4c3F)c12	C69H84F2N10O9S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-DQHLZ9	WO2024120424A1_55	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCCC6(CNC(=O)N6)C5)nc(OC[C@]56CCCN5[C@@H](COC(=O)N5CCC7(CC5)CC(c5cn([C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)nn5)C7)CC6)nc4c3F)c12	C69H82F2N14O8S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-2UMGL5	WO2024120424A1_56	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)c2ccc(OCC3CCN(CC4(COc5nc(N6CCCC7(CNC(=O)N7)C6)c6cnc(-c7cc(O)cc8ccc(F)c(F)c78)c(F)c6n5)CC4)CC3)cc2)C(C)(C)C)cc1	C65H72F3N11O8S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-J5JAA2	WO2024120424A1_57	.	CCc1c(F)ccc2cc(O)cc(N3CCc4c(nc(OC[C@]56CCCN5[C@@H](COC(=O)N5CCC7(CC5)CC(c5cn([C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)nn5)C7)CC6)nc4N4CCCn5nc(C(=O)N(C)C)cc5C4)C3)c12	C72H90FN15O8S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-BL0NF7	WO2024120424A1_58	.	CCc1c(F)ccc2cc(O)cc(N3CCc4c(nc(OCC5(CN6CCC(OCc7ccc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)cc7)CC6)CC5)nc4N4CCCn5nc(C(=O)N(C)C)cc5C4)C3)c12	C70H85FN12O8S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-C8APKA	WO2024120424A1_59	.	CCc1c(F)ccc2cc(O)cc(N3CCc4c(nc(OC[C@]56CCCN5[C@@H](COc5ccc(-c7cn([C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)nn7)cc5)CC6)nc4N4CCCn5nc(C(=O)N(C)C)cc5C4)C3)c12	C69H81FN14O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-2ZGS0W	WO2024120424A1_60	.	CCc1c(F)ccc2cc(O)cc(N3CCc4c(nc(OCC5(CN6CCC(COc7ccc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)cc7)CC6)CC5)nc4N4CCCn5nc(C(=O)N(C)C)cc5C4)C3)c12	C70H85FN12O8S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-68N2DO	WO2024120424A1_61	.	CCc1c(F)ccc2cc(O)cc(N3CCc4c(nc(OCC5(CN6CCC7(CC6)CN(c6ccc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)cc6)C7)CC5)nc4N4CCCn5nc(C(=O)N(C)C)cc5C4)C3)c12	C71H86FN13O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-VYUASN	WO2024120424A1_62	.	CCc1c(F)ccc2cc(O)cc(N3CCc4c(nc(OC[C@@]56CCCN5[C@H](COC(=O)N5CCC7(CC5)CC(C(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)c5ccc(-c8scnc8C)cc5)C(C)(C)C)C7)CC6)nc4N4CCCn5nc(C(=O)N(C)C)cc5C4)C3F)c12	C71H89F2N13O9S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-HSL8NI	WO2024120424A1_63	.	CCc1c(F)ccc2cc(O)cc(N3CCc4c(nc(OC[C@]56CCCN5[C@@H](COC(=O)N5CCC7(CC5)CC(c5cn([C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)nn5)C7)CC6)nc4N4CCCn5nc(C(=O)N(C)C)c(Cl)c5C4)C3)c12	C72H89ClFN15O8S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-4KR2RZ	WO2024120424A1_64	.	CCc1c(F)ccc2cc(O)cc(N3CCc4c(nc(OCC5(CN6CCC(OCc7ccc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)cc7)CC6)CC5)nc4N4CCCn5nc(C(=O)N(C)C)c(Cl)c5C4)C3)c12	C70H84ClFN12O8S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-GSCRZ7	WO2024120424A1_65	.	CCc1c(F)ccc2cc(O)cc(N3CCc4c(nc(OC[C@]56CCCN5[C@@H](COc5ccc(-c7cn([C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)nn7)cc5)CC6)nc4N4CCCn5nc(C(=O)N(C)C)c(Cl)c5C4)C3)c12	C69H80ClFN14O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-WZM5CJ	WO2024120424A1_66	.	CCc1c(F)ccc2cc(O)cc(N3CCc4c(nc(OCC5(CN6CCC7(CC6)CN(c6ccc(C(=O)NC(C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)cc6)C7)CC5)nc4N4CCCn5nc(C(=O)N(C)C)c(Cl)c5C4)C3)c12	C71H85ClFN13O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-S5F3K5	WO2024120424A1_67	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCCN5CCC(COc6ccc(-c7cn([C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)C)nn7)cc6)CC5)nc4c3F)c12	C63H71F2N11O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-5IMRVN	WO2024120424A1_68	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCCN5CCC6(CC5)CC(Oc5cc([C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8scnc8C)cc7)C(C)C)on5)C6)nc4c3F)c12	C60H69F2N9O8S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-HEZ5J8	WO2024120424A1_69	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC(COc7ccc(-c8cn([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)nn8)cc7)CC6)CC5)nc4c3F)c12	C66H75F2N11O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-BIUPBL	WO2024120424A1_70	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCCN5CCC(CC6CN(c7cc([C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)C)on7)C6)CC5)nc4c3F)c12	C61H72F2N10O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-0KOO23	WO2024120424A1_71	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC7(CC6)CC(c6cn([C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)C)nn6)C7)CC5)nc4c3F)c12	C62H73F2N11O6S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-JWB56I	WO2024120424A1_72	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCCN5CCC(F)(COc6cc([C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8scnc8C)cc7)C(C)C)on6)CC5)nc4c3F)c12	C58H66F3N9O8S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-QM7QN8	WO2024120424A1_73	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC7(CC6)CC(Oc6ccc(-c8cn([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)nn8)cc6)C7)CC5)nc4c3F)c12	C68H77F2N11O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-5G8ABD	WO2024120424A1_74	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCCN5CCC(C)(COc6cc([C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8scnc8C)cc7)C(C)C)on6)CC5)nc4c3F)c12	C59H69F2N9O8S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-GMUPSD	WO2024120424A1_75	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC7(CC6)CN(c6ccc(-c8cn([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)nn8)cc6)C7)CC5)nc4c3F)c12	C67H76F2N12O6S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-IY2ZU1	WO2024120424A1_76	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCCN5CCC(C6CN(c7cc([C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)C)on7)C6)CC5)nc4c3F)c12	C60H70F2N10O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-DSKNAZ	WO2024120424A1_77	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OC[C@@H]5CC[C@H](COC(=O)N6CCN(c7cc([C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)C)on7)CC6)N5C)nc4c3F)c12	C62H73F2N11O9S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-PR024P	WO2024120424A1_78	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCCN5CCC(CC6(F)CN(c7cc([C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)C)on7)C6)CC5)nc4c3F)c12	C61H71F3N10O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-2T9UQ2	WO2024120424A1_79	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCCN5CCC(CCOc6cc([C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8scnc8C)cc7)C(C)C)on6)CC5)nc4c3F)c12	C59H69F2N9O8S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-2YDAQL	WO2024120424A1_80	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCCN5CCC(COc6cc([C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8scnc8C)cc7)C(C)C)on6)CC5)nc4c3F)c12	C58H67F2N9O8S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-EFO0FF	WO2024120424A1_82	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCCN5CCC6(CC5)CN(c5cc([C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8scnc8C)cc7)C(C)C)on5)C6)nc4c3F)c12	C59H68F2N10O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-K426OK	WO2024120424A1_83	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCCN5CCC(F)(CN6CCN(c7cc([C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)C)on7)CC6)CC5)nc4c3F)c12	C62H74F3N11O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-MQ68NQ	WO2024120424A1_84	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCCN5CCC(CN6CCN(c7cc([C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)C)on7)CC6)CC5)nc4c3F)c12	C62H75F2N11O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-YBIRXS	WO2024120424A1_85	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCCN5CCC(C(C)(C)N6CCN(c7cc([C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)C)on7)CC6)CC5)nc4c3F)c12	C64H79F2N11O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-UVEM6Y	WO2024120424A1_86	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OC[C@@H]5CC[C@@H](COC(=O)N6CCN(c7cc([C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)C)on7)CC6)N5C)nc4c3F)c12	C62H73F2N11O9S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-097A8Q	WO2024120424A1_87	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OC[C@]56CCCN5[C@H](COC(=O)N5CCC7(CC5)CC(C(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)c5ccc(-c8scnc8C)cc5)C(C)(C)C)C7)CC6)nc4c3F)c12	C67H82F2N10O9S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-7JM3MK	WO2024120424A1_88	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OC[C@]56CCCN5[C@@H](COC(=O)N5CCC7(CC5)CC(C(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)c5ccc(-c8scnc8C)cc5)C(C)(C)C)C7)CC6)nc4c3F)c12	C67H82F2N10O9S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-3VNEDZ	WO2024120424A1_89	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCCn6nc(C(=O)N(C)C)cc6C5)nc(OCC5(CN6CCC(COc7ccc(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)(C)C)cc7)CC6)CC5)nc4c3F)c12	C70H76F2N12O8S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-OXT1UO	WO2024120424A1_90	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCCOCC5)nc(OC[C@]56CCCN5[C@@H](COC(=O)N5CCC7(CC5)CC(C(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)c5ccc(-c8scnc8C)cc5)C(C)(C)C)C7)CC6)nc4c3F)c12	C66H76F2N10O9S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-KC2U7X	WO2024120424A1_91	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCCN5CCC(COc6ccc(-c7cc([C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)C)on7)cc6)CC5)nc4c3F)c12	C64H71F2N9O8S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-BWL0VA	WO2024120424A1_92	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC(CC7CN(c8cc([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)on8)C7)CC6)CC5)nc4c3F)c12	C64H76F2N10O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-ZEBP8P	WO2024120424A1_93	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC(OCc7ccc(-c8cn([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)nn8)cc7)CC6)CC5)nc4c3F)c12	C66H75F2N11O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-W3RYLO	WO2024120424A1_94	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC(C7CN(c8cc([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)on8)C7)CC6)CC5)nc4c3F)c12	C63H74F2N10O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-G9FKDJ	WO2024120424A1_95	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC(OCc7ccc(-c8cc([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)on8)cc7)CC6)CC5)nc4c3F)c12	C67H75F2N9O8S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-QOSYZL	WO2024120424A1_96	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC(COc7cc([C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)C)on7)CC6)CC5)nc4c3F)c12	C61H71F2N9O8S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-VY37SF	WO2024120424A1_97	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC(COc7ccc(-c8cc([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)on8)cc7)CC6)CC5)nc4c3F)c12	C67H75F2N9O8S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-0C9HFP	WO2024120424A1_98	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC(C)(COc7cc([C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)C)on7)CC6)CC5)nc4c3F)c12	C62H73F2N9O8S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-LK0LND	WO2024120424A1_99	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC7(CC6)CC(c6cc([C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)C)on6)C7)CC5)nc4c3F)c12	C63H73F2N9O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-R4A41F	WO2024120424A1_100	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC(F)(COc7cc([C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)C)on7)CC6)CC5)nc4c3F)c12	C61H70F3N9O8S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-DZ014S	WO2024120424A1_101	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC7(CC6)CC(Oc6ccc(-c8cc([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)on8)cc6)C7)CC5)nc4c3F)c12	C69H77F2N9O8S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-Z2KTDX	WO2024120424A1_102	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC(CCOc7cc([C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)C)on7)CC6)CC5)nc4c3F)c12	C62H73F2N9O8S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-TO14J3	WO2024120424A1_103	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC7(CC6)CN(c6ccc(-c8cc([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)on8)cc6)C7)CC5)nc4c3F)c12	C68H76F2N10O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-W3CL7S	WO2024120424A1_104	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC(CN7CCN(c8cc([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)on8)CC7)CC6)CC5)nc4c3F)c12	C65H79F2N11O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-S9OACA	WO2024120424A1_105	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC7(CC6)CN(c6cc([C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)C)on6)C7)CC5)nc4c3F)c12	C62H72F2N10O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-M9OFH8	WO2024120424A1_106	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC(COc7ccc(NC(=O)C[C@H](NC(=O)[C@@H]8C[C@@H](O)CN8C(=O)[C@@H](NC(=O)C8(C#N)CC8)C(C)(C)C)c8ccc(-c9scnc9C)cc8)cc7)CC6)CC5)nc4c3F)c12	C71H81F2N11O9S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-57NJGB	WO2024120424A1_107	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC(COc7ccc(NC(=O)C[C@H](NC(=O)[C@@H]8C[C@@H](O)CN8C(=O)[C@@H](c8cc(C)no8)C(C)C)c8ccc(-c9scnc9C)cc8)cc7)CC6)CC5)nc4c3F)c12	C69H78F2N10O9S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-JAWV55	WO2024120424A1_108	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(C#CC5(CN6CCC(c7ccc(-c8cn([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)nn8)cc7)CC6)CC5)nc4c3F)c12	C66H67F2N11O5S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-1PNYPC	WO2024120424A1_109	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(C#CC5(CN6CCC(c7ccc(-c8cn([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)nn8)cc7)CC6)CC5)nc4c3F)c12	C66H71F2N11O5S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-3JWH7K	WO2024120424A1_110	.	C=C1CN2[C@H](COC(=O)N3CCN(c4cc([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)c5ccc(-c6scnc6C)cc5)C(C)C)on4)CC3)CC[C@@]2(COc2nc(N3CCC[C@@](C)(O)C3)c3cnc(-c4cc(O)cc5ccc(F)c(CC)c45)cc3n2)C1	C65H76FN11O9S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-PWQ5B4	WO2024120424A1_111	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCN(CC7CCN(c8cc([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)on8)CC7)CC6)CC5)nc4c3F)c12	C65H79F2N11O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-E24FNK	WO2024120424A1_112	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCN(c7cc(C(C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)C)on7)CC6)CC5)nc4c3F)c12	C59H68F2N10O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-IC8S4E	WO2024120424A1_113	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6C[C@@H]7CN(c8cc([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)on8)C[C@@H]7C6)CC5)nc4c3F)c12	C61H70F2N10O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-B3S5DP	WO2024120424A1_114	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC(Oc7cc([C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)C)on7)CC6)CC5)nc4c3F)c12	C60H69F2N9O8S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-I2DXXV	WO2024120424A1_115	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC(N7CCN(c8cc([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)on8)CC7)CC6)CC5)nc4c3F)c12	C64H77F2N11O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-CB7MH2	WO2024120424A1_116	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CC(N7CCN(c8cc([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)on8)CC7)C6)CC5)nc4c3F)c12	C62H73F2N11O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-PNVLIV	WO2024120424A1_117	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC(Oc7ccc(-c8cn([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)nn8)nc7)CC6)CC5)nc4c3F)c12	C64H72F2N12O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-7Y1SXL	WO2024120424A1_118	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC7(CC6)CN(c6ccc(-c8cn([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)nn8)cn6)C7)CC5)nc4c3F)c12	C66H75F2N13O6S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-LLGHJ5	WO2024120424A1_119	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC(c7ccc(-c8cn([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)(C)C)nn8)cc7)CC6)CC5)nc4c3F)c12	C66H75F2N11O6S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-1S65YG	WO2024120424A1_120	.	C=C1CN2[C@H](COCc3cnnn3[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](C)c3ccc(-c4scnc4C)cc3)C(C)C)CC[C@@]2(COc2nc(N3CCC[C@@](C)(O)C3)c3cnc(-c4cc(O)cc5ccc(F)c(CC)c45)c(F)c3n2)C1	C60H69F2N11O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-NWZU4K	WO2024120424A1_121	.	C=C1CN2[C@H](COc3cc(-c4cn([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)c5ccc(-c6scnc6C)cc5)C(C)C)nn4)ccn3)CC[C@@]2(COc2nc(N3CCC[C@@](C)(O)C3)c3cnc(-c4cc(O)cc5ccc(F)c(CC)c45)c(F)c3n2)C1	C64H70F2N12O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-6XC8G1	WO2024120424A1_122	.	C=C1CN2[C@H](COCc3ccc(-c4cn([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)c5ccc(-c6scnc6C)cc5)C(C)C)nn4)cc3)CC[C@@]2(COc2nc(N3CCC[C@@](C)(O)C3)c3cnc(-c4cc(O)cc5ccc(F)c(CC)c45)cc3n2)C1	C66H74FN11O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-ZMU5K7	WO2024120424A1_123	.	C=C1CN2[C@H](CN3CCC(c4cn([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)c5ccc(-c6scnc6C)cc5)C(C)C)nn4)CC3)CC[C@@]2(COc2nc(N3CCC[C@@](C)(O)C3)c3cnc(-c4cc(O)cc5ccc(F)c(CC)c45)cc3n2)C1	C64H77FN12O6S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-N9RWAM	WO2024120424A1_124	.	C=C1CN2[C@H](COc3ccc(-c4cn([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)c5ccc(-c6scnc6C)cc5)C(C)C)nn4)cn3)CC[C@@]2(COc2nc(N3CCC[C@@](C)(O)C3)c3cnc(-c4cc(O)cc5ccc(F)c(CC)c45)c(F)c3n2)C1	C64H70F2N12O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-KWWGAG	WO2024120424A1_125	.	C=C1CN2[C@H](COC(=O)N3CCC(COc4cc([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)c5ccc(-c6scnc6C)cc5)C(C)C)on4)CC3)CC[C@@]2(COc2nc(N3CCC[C@@](C)(O)C3)c3cnc(-c4cc(O)cc5ccc(F)c(CC)c45)cc3n2)C1	C67H79FN10O10S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-QHWSEE	WO2024120424A1_126	.	C=C1CN2[C@H](COC(=O)NCC34CC(c5cn([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)c6ccc(-c7scnc7C)cc6)C(C)C)nn5)(C3)C4)CC[C@@]2(COc2nc(N3CCC[C@@](C)(O)C3)c3cnc(-c4cc(O)cc5ccc(F)c(CC)c45)cc3n2)C1	C66H77FN12O8S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-JE3RT2	WO2024120424A1_127	.	C=C1CN2[C@H](COC(=O)N3CCC4(CC3)CC(c3cn([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)c5ccc(-c6scnc6C)cc5)C(C)C)nn3)C4)CC[C@@]2(COc2nc(N3CCC[C@@](C)(O)C3)c3cnc(-c4cc(O)cc5ccc(F)c(CC)c45)cc3n2)C1	C68H81FN12O8S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-7GVDAN	WO2024120424A1_128	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC(N7CC(c8cn([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)nn8)C7)CC6)CC5)nc4c3F)c12	C62H74F2N12O6S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-LPKLXV	WO2024120424A1_129	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC(CN7CC(c8cn([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)nn8)C7)CC6)CC5)nc4c3F)c12	C63H76F2N12O6S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-UPWXZ4	WO2024120424A1_130	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC(CN7CCC(c8cn([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)nn8)CC7)CC6)CC5)nc4c3F)c12	C65H80F2N12O6S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-HEYK2Y	WO2024120424A1_131	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC(c7cn([C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)C)nn7)CC6)CC5)nc4c3F)c12	C59H69F2N11O6S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-ZRJG2B	WO2024120424A1_132	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCN(Cc7cn([C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)C)nn7)CC6)CC5)nc4c3F)c12	C59H70F2N12O6S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-HGRHAX	WO2024120424A1_133	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCN(c7ccc(-c8cn([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)nn8)cc7)CC6)CC5)nc4c3F)c12	C64H72F2N12O6S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-B926Y8	WO2024120424A1_134	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCN(c7cnc(-c8cn([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)nn8)cn7)CC6)CC5)nc4c3F)c12	C62H70F2N14O6S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-6T9M2D	WO2024120424A1_135	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC(Oc7ccc(-c8cn([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)nn8)cn7)CC6)CC5)nc4c3F)c12	C64H72F2N12O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-BAM6IS	WO2024120424A1_136	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC(Oc7cc(-c8cn([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)nn8)ccn7)CC6)CC5)nc4c3F)c12	C64H72F2N12O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-GB38VL	WO2024120424A1_137	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC(N7CCC(c8cn([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)nn8)CC7)CC6)CC5)nc4c3F)c12	C64H78F2N12O6S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-U8H5PK	WO2024120424A1_138	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC(n7cc(-c8cn([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)nn8)cn7)CC6)CC5)nc4c3F)c12	C62H71F2N13O6S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-DII5OI	WO2024120424A1_139	.	C=C1CN2[C@H](COC(=O)N3CCC4(CC3)CC(CNC(=O)C[C@H](NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(c3cc(C)no3)C(C)C)c3ccc(-c5scnc5C)cc3)C4)CC[C@@]2(COc2nc(N3CCC[C@@](C)(O)C3)c3cnc(-c4cc(O)cc5ccc(F)c(CC)c45)c(F)c3n2)C1	C72H85F2N11O10S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-4BXAM1	WO2024120424A1_140	.	C=C1CN2[C@H](COC(=O)N3CCC4(CC3)CC(C(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](C)c3ccc(-c5scnc5C)cc3)C(C)(C)C)C4)CC[C@@]2(COc2nc(N3CCC[C@@](C)(O)C3)c3cnc(-c4cc(O)cc5ccc(F)c(CC)c45)c(F)c3n2)C1	C68H82F2N10O9S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-BHA336	WO2024120424A1_141	.	C=C1CN2[C@H](COC(=O)N3CCC(Cc4cn([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)c5ccc(-c6scnc6C)cc5)C(C)C)nn4)CC3)CC[C@@]2(COc2nc(N3CCC[C@@](C)(O)C3)c3cnc(-c4cc(O)cc5ccc(F)c(CC)c45)c(F)c3n2)C1	C66H78F2N12O8S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-Q2EHQV	WO2024120424A1_142	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCN(c7ccc(-c8cn([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)nn8)cn7)CC6)CC5)nc4c3F)c12	C63H71F2N13O6S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-0XIA1L	PROTAC pan-KRAS degrader-1	PROTAC pan-KRAS degrader-1; EX-A13306; 3043908-63-7	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC(Oc7cnc(-c8cn([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)nn8)cn7)CC6)CC5)nc4c3F)c12	C63H71F2N13O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-GCYZ75	WO2024120424A1_145	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCN(Cc7nc(-c8cn([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)nn8)cs7)CC6)CC5)nc4c3F)c12	C62H71F2N13O6S2	KRAS	P01116	VHL	WO-2024120424-A1
TPD-2UWUDE	WO2024120424A1_146	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCN(Cc7ncc(-c8cn([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)nn8)s7)CC6)CC5)nc4c3F)c12	C62H71F2N13O6S2	KRAS	P01116	VHL	WO-2024120424-A1
TPD-OGKRW8	WO2024120424A1_147	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC(CC7CCN(c8cc([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)on8)CC7)CC6)CC5)nc4c3F)c12	C66H80F2N10O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-KBCI39	WO2024120424A1_148	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCN(CC78CC(c9cn([C@H](C(=O)N%10C[C@H](O)C[C@H]%10C(=O)N[C@@H](C)c%10ccc(-c%11scnc%11C)cc%10)C(C)C)nn9)(C7)C8)CC6)CC5)nc4c3F)c12	C64H76F2N12O6S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-B7PYK5	WO2024120424A1_149	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCN(C78CC(c9cn([C@H](C(=O)N%10C[C@H](O)C[C@H]%10C(=O)N[C@@H](C)c%10ccc(-c%11scnc%11C)cc%10)C(C)C)nn9)(C7)C8)CC6)CC5)nc4c3F)c12	C63H74F2N12O6S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-C9ZHQL	WO2024120424A1_150	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC7(CC6)CC(Oc6cc([C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)C)on6)C7)CC5)nc4c3F)c12	C63H73F2N9O8S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-Z9IX79	WO2024120424A1_151	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC(NC(=O)c7ccc(-c8cn([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)nn8)cc7)CC6)CC5)nc4c3F)c12	C66H74F2N12O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-RCUQFE	WO2024120424A1_152	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC(Nc7ccc(-c8cn([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)nn8)cn7)CC6)CC5)nc4c3F)c12	C64H73F2N13O6S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-EWMBMH	WO2024120424A1_153	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6C[C@@H]7C[C@H]6CN7c6cc([C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8scnc8C)cc7)C(C)C)on6)CC5)nc4c3F)c12	C60H68F2N10O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-ZHO8RU	WO2024120424A1_154	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC(N(C)c7ccc(-c8cn([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)nn8)cn7)CC6)CC5)nc4c3F)c12	C65H75F2N13O6S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-A4I0RW	WO2024120424A1_155	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC7(CC6)CCN(c6cc([C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)C)on6)CC7)CC5)nc4c3F)c12	C64H76F2N10O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-XH6Y00	WO2024120424A1_156	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCN(C7CN(c8cc([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)on8)C7)CC6)CC5)nc4c3F)c12	C62H73F2N11O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-C1VNCF	WO2024120424A1_157	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OC[C@]56CCCN5[C@@H](COc5ccc(-c7cn([C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)C)nn7)cn5)CC6)nc4c3F)c12	C63H70F2N12O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-L5JOOB	WO2024120424A1_158	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OC[C@]56CCCN5[C@@H](COc5ncc(-c7cn([C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)C)nn7)cn5)CC6)nc4c3F)c12	C62H69F2N13O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-ISPBDQ	WO2024120424A1_159	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OC[C@]56CCCN5[C@@H](COc5cnc(-c7cn([C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)C)nn7)cn5)CC6)nc4c3F)c12	C62H69F2N13O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-RHHPGM	WO2024120424A1_160	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC(Oc7ccc(-c8cn([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](CO)c9ccc(-c%10ccnn%10CC)cc9)C(C)C)nn8)cn7)CC6)CC5)nc4c3F)c12	C65H75F2N13O8	KRAS	P01116	VHL	WO-2024120424-A1
TPD-8N01H1	WO2024120424A1_161	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CC7(O)CN(c8cc([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)on8)CC7(O)C6)CC5)nc4c3F)c12	C61H70F2N10O9S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-DJIAUJ	WO2024120424A1_162	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC(O)(COc7cc([C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)C)on7)CC6)CC5)nc4c3F)c12	C61H71F2N9O9S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-7B97BR	WO2024120424A1_163	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC(N)(COc7cc([C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)C)on7)CC6)CC5)nc4c3F)c12	C61H72F2N10O8S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-AJOMZL	WO2024120424A1_164	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCN(C7CCN(c8cc([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)on8)CC7)CC6)CC5)nc4c3F)c12	C64H77F2N11O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-O7GMMO	WO2024120424A1_165	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCN(C7CC(c8cn([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)nn8)C7)CC6)CC5)nc4c3F)c12	C62H74F2N12O6S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-RPJTOK	WO2024120424A1_166	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCN(C7CCN(c8cc([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)on8)C7)CC6)CC5)nc4c3F)c12	C63H75F2N11O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-EP5D0A	WO2024120424A1_167	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC(Oc7ccc(-c8cn([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)nn8)nn7)CC6)CC5)nc4c3F)c12	C63H71F2N13O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-4OBPY1	WO2024120424A1_168	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC7(CC6)CN(c6cnc(-c8cn([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)nn8)cn6)C7)CC5)nc4c3F)c12	C65H74F2N14O6S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-GUEKZN	WO2024120424A1_169	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC(Oc7cnc(-c8cn([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)nn8)nc7)CC6)CC5)nc4c3F)c12	C63H71F2N13O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-22WAUW	WO2024120424A1_170	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC7(CC6)CN(c6cnc(-c8cn([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](CO)c9ccc(-c%10scnc%10C)cc9)C(C)C)nn8)cn6)C7)CC5)nc4c3F)c12	C65H74F2N14O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-7XSQT7	WO2024120424A1_171	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC(Oc7ccc(-c8cn([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](CO)c9ccc(-c%10scnc%10C)cc9)C(C)C)nn8)cn7)CC6)CC5)nc4c3F)c12	C64H72F2N12O8S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-QMK5C3	WO2024120424A1_172	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC(Oc7cnc(-c8cn([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](CO)c9ccc(-c%10c(C)cnn%10CC)cc9)C(C)C)nn8)cn7)CC6)CC5)nc4c3F)c12	C65H76F2N14O8	KRAS	P01116	VHL	WO-2024120424-A1
TPD-7PU7GS	WO2024120424A1_173	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCN(C(=O)c7cnc(-c8cn([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)nn8)cn7)CC6)CC5)nc4c3F)c12	C63H70F2N14O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-IRHHK5	WO2024120424A1_174	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCN(C(=O)Cc7cnc(-c8cn([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)nn8)cn7)CC6)CC5)nc4c3F)c12	C64H72F2N14O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-XYEPCO	WO2024120424A1_175	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCN(CCOc7cc([C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)C)on7)CC6)CC5)nc4c3F)c12	C61H72F2N10O8S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-YGEAKL	WO2024120424A1_176	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC(C)(Oc7ccc(-c8cn([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)nn8)cn7)CC6)CC5)nc4c3F)c12	C65H74F2N12O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-QJDVZ7	WO2024120424A1_177	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCN(Cc7cnc(-c8cn([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)nn8)cn7)CC6)CC5)nc4c3F)c12	C63H72F2N14O6S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-IS2FPE	WO2024120424A1_178	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC(Oc7cnc(-c8cn([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](CO)c9ccc(-c%10scnc%10C)cc9)C(C)C)nn8)cn7)CC6)CC5)nc4c3F)c12	C63H71F2N13O8S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-KXDNQ5	WO2024120424A1_179	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCN(Cc7ccc(-c8cn([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)nn8)cn7)CC6)CC5)nc4c3F)c12	C64H73F2N13O6S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-BJD73J	WO2024120424A1_180	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC(N(C)C78CC(c9cn([C@H](C(=O)N%10C[C@H](O)C[C@H]%10C(=O)N[C@@H](C)c%10ccc(-c%11scnc%11C)cc%10)C(C)C)nn9)(C7)C8)CC6)CC5)nc4c3F)c12	C65H78F2N12O6S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-5CH3M5	WO2024120424A1_181	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC(Oc7ncc(-c8cn([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)nn8)s7)CC6)CC5)nc4c3F)c12	C62H70F2N12O7S2	KRAS	P01116	VHL	WO-2024120424-A1
TPD-M8SMX8	WO2024120424A1_182	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC(Cn7cc(-c8cn([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)nn8)cn7)CC6)CC5)nc4c3F)c12	C63H73F2N13O6S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-K8CGLH	WO2024120424A1_183	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCN(C7CN(c8cnc(-c9cn([C@H](C(=O)N%10C[C@H](O)C[C@H]%10C(=O)N[C@@H](C)c%10ccc(-c%11scnc%11C)cc%10)C(C)C)nn9)cn8)C7)CC6)CC5)nc4c3F)c12	C65H75F2N15O6S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-P5FH0I	WO2024120424A1_184	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC(Oc7cnc(-c8cn([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@H](c9ccc(-c%10scnc%10C)cc9)[C@H](O)C(C)C)C(C)C)nn8)cn7)CC6)CC5)nc4c3F)c12	C66H77F2N13O8S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-5PL934	WO2024120424A1_185	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC(Oc7cnc(-c8cn([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9C)C(C)C)nn8)cn7)CC6)CC5)nc4c3F)c12	C64H73F2N13O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-UEPND2	WO2024120424A1_187	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCN(Cc7cnc(-c8cn([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)nn8)s7)CC6)CC5)nc4c3F)c12	C62H71F2N13O6S2	KRAS	P01116	VHL	WO-2024120424-A1
TPD-YX8UXD	WO2024120424A1_188	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OC[C@]56CCCN5[C@@H](COCc5cnc(-c7cn([C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)C)nn7)cn5)CC6)nc4c3F)c12	C63H71F2N13O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-Z82P8C	WO2024120424A1_189	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC7(CC6)CN(Cc6cnc(-c8cn([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)nn8)cn6)C7)CC5)nc4c3F)c12	C66H76F2N14O6S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-183QCO	WO2024120424A1_190	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC(Oc7cnc(-c8cn([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](CC(=O)NC)c9ccc(-c%10scnc%10C)cc9)C(C)C)nn8)cn7)CC6)CC5)nc4c3F)c12	C65H74F2N14O8S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-DFTQOY	WO2024120424A1_191	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCN(CCc7cnc(-c8cn([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)nn8)cn7)CC6)CC5)nc4c3F)c12	C64H74F2N14O6S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-SBG8CB	WO2024120424A1_192	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCN(C7CN(c8cnc(-c9cn([C@H](C(=O)N%10C[C@H](O)C[C@H]%10C(=O)N[C@@H](CO)c%10ccc(-c%11scnc%11C)cc%10)C(C)C)nn9)cn8)C7)CC6)CC5)nc4c3F)c12	C65H75F2N15O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-BNWB8J	WO2024120424A1_193	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC(Cc7cnc(-c8cn([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)nn8)cn7)CC6)CC5)nc4c3F)c12	C64H73F2N13O6S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-ZLEYU1	WO2024120424A1_194	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCN(C(C)c7cnc(-c8cn([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)nn8)cn7)CC6)CC5)nc4c3F)c12	C64H74F2N14O6S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-91E982	WO2024120424A1_195	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC(N7CCC(c8cnc(-c9cn([C@H](C(=O)N%10C[C@H](O)C[C@H]%10C(=O)N[C@@H](C)c%10ccc(-c%11scnc%11C)cc%10)C(C)C)nn9)cn8)CC7)CC6)CC5)nc4c3F)c12	C68H80F2N14O6S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-QSBV6E	WO2024120424A1_196	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC(N7CCN(c8cnc(-c9cn([C@H](C(=O)N%10C[C@H](O)C[C@H]%10C(=O)N[C@@H](C)c%10ccc(-c%11scnc%11C)cc%10)C(C)C)nn9)cn8)CC7)CC6)CC5)nc4c3F)c12	C67H79F2N15O6S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-N99M9A	WO2024120424A1_197	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCN(C7CCN(c8cnc(-c9cn([C@H](C(=O)N%10C[C@H](O)C[C@H]%10C(=O)N[C@@H](C)c%10ccc(-c%11scnc%11C)cc%10)C(C)C)nn9)cn8)CC7)CC6)CC5)nc4c3F)c12	C67H79F2N15O6S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-S02GRI	WO2024120424A1_198	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC(OCc7cnc(-c8cn([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)nn8)cn7)CC6)CC5)nc4c3F)c12	C64H73F2N13O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-6IBNFM	WO2024120424A1_199	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC(CNc7cnc(-c8cn([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)nn8)cn7)CC6)CC5)nc4c3F)c12	C64H74F2N14O6S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-QXSHWQ	WO2024120424A1_200	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC(CC7CN(c8cnc(-c9cn([C@H](C(=O)N%10C[C@H](O)C[C@H]%10C(=O)N[C@@H](C)c%10ccc(-c%11scnc%11C)cc%10)C(C)C)nn9)cn8)C7)CC6)CC5)nc4c3F)c12	C67H78F2N14O6S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-2MR0CZ	WO2024120424A1_202	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCN(Cc7cc(-c8cn([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)nn8)n(C)n7)CC6)CC5)nc4c3F)c12	C63H74F2N14O6S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-S55QZV	WO2024120424A1_203	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC(c7ccc(-c8cn([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)nn8)cn7)CC6)CC5)nc4c3F)c12	C64H72F2N12O6S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-0GF9AQ	WO2024120424A1_204	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCN(CCN(C)c7cc([C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)c8ccc(-c9scnc9C)cc8)C(C)C)on7)CC6)CC5)nc4c3F)c12	C62H75F2N11O7S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-3JWNUY	WO2024120424A1_205	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCN(Cc7cncc(-c8cn([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)nn8)n7)CC6)CC5)nc4c3F)c12	C63H72F2N14O6S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-UFQ5FT	WO2024120424A1_206	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCN(CC7CN(c8cnc(-c9cn([C@H](C(=O)N%10C[C@H](O)C[C@H]%10C(=O)N[C@@H](C)c%10ccc(-c%11scnc%11C)cc%10)C(C)C)nn9)cn8)C7)CC6)CC5)nc4c3F)c12	C66H77F2N15O6S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-S4ZQ6F	WO2024120424A1_207	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCC[C@@](C)(O)C5)nc(OCC5(CN6CCC(C#Cc7cnc(-c8cn([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)c9ccc(-c%10scnc%10C)cc9)C(C)C)nn8)cn7)CC6)CC5)nc4c3F)c12	C65H71F2N13O6S	KRAS	P01116	VHL	WO-2024120424-A1
TPD-T78VAO	WO2024126617A1_1	.	NC1=NC=C2/C=C/CN(C(=O)CCOCCOCCOCCNC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)CCCC(=O)N[C@@H]3CCC[C@H](C3)N3N=C(C4=CC=C(C(=O)NC5=NC=CC(C(F)(F)F)=C5)C=C4)C1=C23	C54H58F3N11O10	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-Y0EOY4	WO2024126617A1_2	.	NC1=NC=C2/C=C/CCN(C(=O)CCOCCOCCOCCNC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)CC(=O)N[C@@H]3CCC[C@H](C3)N3N=C(C4=CC=C(C(=O)NC5=NC=CC(C(F)(F)F)=C5)C=C4)C1=C23	C53H56F3N11O10	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-4K9FOI	WO2024126617A1_3	4-[(2R,6R,14E)-19-amino-11-[3-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]propanoyl]-8-oxo-1,7,11,18,22-pentazatetracyclo[14.6.1.12,6.020,23]tetracosa-14,16,18,20(23),21-pentaen-21-yl]-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide	NC1=NC=C2/C=C/CCN(C(=O)CCOCCOCCOCCNC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)CCC(=O)N[C@@H]3CCC[C@H](C3)N3N=C(C4=CC=C(C(=O)NC5=NC=CC(C(F)(F)F)=C5)C=C4)C1=C23	C54H58F3N11O10	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-2MRZD2	WO2024126617A1_4	4-[(2R,6R,14E)-19-amino-10-[3-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]propanoyl]-8-oxo-1,7,10,18,22-pentazatetracyclo[14.6.1.12,6.020,23]tetracosa-14,16,18,20(23),21-pentaen-21-yl]-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide	NC1=NC=C2/C=C/CCCN(C(=O)CCOCCOCCOCCNC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)CC(=O)N[C@@H]3CCC[C@H](C3)N3N=C(C4=CC=C(C(=O)NC5=NC=CC(C(F)(F)F)=C5)C=C4)C1=C23	C54H58F3N11O10	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-IA962T	WO2024126617A1_5	N-[2-[2-[2-[2-[3-[(2R,6R,13E)-18-amino-8-oxo-20-[4-[[4-(trifluoromethyl)pyridin-2-yl]carbamoyl]phenyl]-1,7,10,17,21-pentazatetracyclo[13.6.1.12,6.019,22]tricosa-13,15,17,19(22),20-pentaen-10-yl]-3-oxopropoxy]ethoxy]ethoxy]ethoxy]ethyl]-6-[3-(2,4-dioxo-1,3-diazinan-1-yl)azetidin-1-yl]pyridine-3-carboxamide	NC1=NC=C2/C=C/CCN(C(=O)CCOCCOCCOCCOCCNC(=O)C3=CN=C(N4CC(N5CCC(=O)NC5=O)C4)C=C3)CC(=O)N[C@@H]3CCC[C@H](C3)N3N=C(C4=CC=C(C(=O)NC5=NC=CC(C(F)(F)F)=C5)C=C4)C1=C23	C55H64F3N13O10	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-JVXONA	WO2024126617A1_6	N-[2-[2-[2-[3-[(2R,6R,13E)-18-amino-8-oxo-20-[4-[[4-(trifluoromethyl)pyridin-2-yl]carbamoyl]phenyl]-1,7,10,17,21-pentazatetracyclo[13.6.1.12,6.019,22]tricosa-13,15,17,19(22),20-pentaen-10-yl]-3-oxopropoxy]ethoxy]ethoxy]ethyl]-6-[3-(2,4-dioxo-1,3-diazinan-1-yl)azetidin-1-yl]pyridine-3-carboxamide	NC1=NC=C2/C=C/CCN(C(=O)CCOCCOCCOCCNC(=O)C3=CN=C(N4CC(N5CCC(=O)NC5=O)C4)C=C3)CC(=O)N[C@@H]3CCC[C@H](C3)N3N=C(C4=CC=C(C(=O)NC5=NC=CC(C(F)(F)F)=C5)C=C4)C1=C23	C53H60F3N13O9	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-KFZY6G	WO2024126617A1_7	N-[2-[2-[3-[(2R,6R,13E)-18-amino-8-oxo-20-[4-[[4-(trifluoromethyl)pyridin-2-yl]carbamoyl]phenyl]-1,7,10,17,21-pentazatetracyclo[13.6.1.12,6.019,22]tricosa-13,15,17,19(22),20-pentaen-10-yl]-3-oxopropoxy]ethoxy]ethyl]-6-[3-(2,4-dioxo-1,3-diazinan-1-yl)azetidin-1-yl]pyridine-3-carboxamide	NC1=NC=C2/C=C/CCN(C(=O)CCOCCOCCNC(=O)C3=CN=C(N4CC(N5CCC(=O)NC5=O)C4)C=C3)CC(=O)N[C@@H]3CCC[C@H](C3)N3N=C(C4=CC=C(C(=O)NC5=NC=CC(C(F)(F)F)=C5)C=C4)C1=C23	C51H56F3N13O8	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-I9J9Y4	WO2024126617A1_8	.	NC1=NC=C2/C=C/CCN(C(=O)CCOCCNC(=O)C3=CN=C(N4CC(N5CCC(=O)NC5=O)C4)C=C3)CC(=O)N[C@@H]3CCC[C@H](C3)N3N=C(C4=CC=C(C(=O)NC5=NC=CC(C(F)(F)F)=C5)C=C4)C1=C23	C49H52F3N13O7	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-FLZDB8	WO2024126617A1_9	N-[3-[(2R,6R,13E)-18-amino-8-oxo-20-[4-[[4-(trifluoromethyl)pyridin-2-yl]carbamoyl]phenyl]-1,7,10,17,21-pentazatetracyclo[13.6.1.12,6.019,22]tricosa-13,15,17,19(22),20-pentaen-10-yl]-3-oxopropyl]-6-[3-(2,4-dioxo-1,3-diazinan-1-yl)azetidin-1-yl]pyridine-3-carboxamide	NC1=NC=C2/C=C/CCN(C(=O)CCNC(=O)C3=CN=C(N4CC(N5CCC(=O)NC5=O)C4)C=C3)CC(=O)N[C@@H]3CCC[C@H](C3)N3N=C(C4=CC=C(C(=O)NC5=NC=CC(C(F)(F)F)=C5)C=C4)C1=C23	C47H48F3N13O6	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-BQK2UO	WO2024126617A1_10	N-[2-[2-[2-[2-[3-[(2R,6R,14E)-19-amino-8-oxo-21-[4-[[4-(trifluoromethyl)pyridin-2-yl]carbamoyl]phenyl]-1,7,10,18,22-pentazatetracyclo[14.6.1.12,6.020,23]tetracosa-14,16,18,20(23),21-pentaen-10-yl]-3-oxopropoxy]ethoxy]ethoxy]ethoxy]ethyl]-6-[3-(2,4-dioxo-1,3-diazinan-1-yl)azetidin-1-yl]pyridine-3-carboxamide	NC1=NC=C2/C=C/CCCN(C(=O)CCOCCOCCOCCOCCNC(=O)C3=CN=C(N4CC(N5CCC(=O)NC5=O)C4)C=C3)CC(=O)N[C@@H]3CCC[C@H](C3)N3N=C(C4=CC=C(C(=O)NC5=NC=CC(C(F)(F)F)=C5)C=C4)C1=C23	C56H66F3N13O10	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-9MLTB2	WO2024126617A1_11	N-[2-[2-[2-[3-[(2R,6R,14E)-19-amino-8-oxo-21-[4-[[4-(trifluoromethyl)pyridin-2-yl]carbamoyl]phenyl]-1,7,10,18,22-pentazatetracyclo[14.6.1.12,6.020,23]tetracosa-14,16,18,20(23),21-pentaen-10-yl]-3-oxopropoxy]ethoxy]ethoxy]ethyl]-6-[3-(2,4-dioxo-1,3-diazinan-1-yl)azetidin-1-yl]pyridine-3-carboxamide	NC1=NC=C2/C=C/CCCN(C(=O)CCOCCOCCOCCNC(=O)C3=CN=C(N4CC(N5CCC(=O)NC5=O)C4)C=C3)CC(=O)N[C@@H]3CCC[C@H](C3)N3N=C(C4=CC=C(C(=O)NC5=NC=CC(C(F)(F)F)=C5)C=C4)C1=C23	C54H62F3N13O9	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-6E2VVO	WO2024126617A1_12	.	NC1=NC=C2/C=C/CCCN(C(=O)CCOCCOCCNC(=O)C3=CN=C(N4CC(N5CCC(=O)NC5=O)C4)C=C3)CC(=O)N[C@@H]3CCC[C@H](C3)N3N=C(C4=CC=C(C(=O)NC5=NC=CC(C(F)(F)F)=C5)C=C4)C1=C23	C52H58F3N13O8	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-0JSQ69	WO2024126617A1_13	N-[2-[3-[(2R,6R,14E)-19-amino-8-oxo-21-[4-[[4-(trifluoromethyl)pyridin-2-yl]carbamoyl]phenyl]-1,7,10,18,22-pentazatetracyclo[14.6.1.12,6.020,23]tetracosa-14,16,18,20(23),21-pentaen-10-yl]-3-oxopropoxy]ethyl]-6-[3-(2,4-dioxo-1,3-diazinan-1-yl)azetidin-1-yl]pyridine-3-carboxamide	NC1=NC=C2/C=C/CCCN(C(=O)CCOCCNC(=O)C3=CN=C(N4CC(N5CCC(=O)NC5=O)C4)C=C3)CC(=O)N[C@@H]3CCC[C@H](C3)N3N=C(C4=CC=C(C(=O)NC5=NC=CC(C(F)(F)F)=C5)C=C4)C1=C23	C50H54F3N13O7	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-9IREMU	WO2024126617A1_14	N-[3-[(2R,6R,14E)-19-amino-8-oxo-21-[4-[[4-(trifluoromethyl)pyridin-2-yl]carbamoyl]phenyl]-1,7,10,18,22-pentazatetracyclo[14.6.1.12,6.020,23]tetracosa-14,16,18,20(23),21-pentaen-10-yl]-3-oxopropyl]-6-[3-(2,4-dioxo-1,3-diazinan-1-yl)azetidin-1-yl]pyridine-3-carboxamide	NC1=NC=C2/C=C/CCCN(C(=O)CCNC(=O)C3=CN=C(N4CC(N5CCC(=O)NC5=O)C4)C=C3)CC(=O)N[C@@H]3CCC[C@H](C3)N3N=C(C4=CC=C(C(=O)NC5=NC=CC(C(F)(F)F)=C5)C=C4)C1=C23	C48H50F3N13O6	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-VIVYSA	WO2024126617A1_15	4-[(2R,6R,13E)-18-amino-10-[6-[6-[3-(2,4-dioxo-1,3-diazinan-1-yl)azetidin-1-yl]pyridin-3-yl]hex-5-ynoyl]-8-oxo-1,7,10,17,21-pentazatetracyclo[13.6.1.12,6.019,22]tricosa-13,15,17,19(22),20-pentaen-20-yl]-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide	NC1=NC=C2/C=C/CCN(C(=O)CCCC#CC3=CC=C(N4CC(N5CCC(=O)NC5=O)C4)N=C3)CC(=O)N[C@@H]3CCC[C@H](C3)N3N=C(C4=CC=C(C(=O)NC5=NC=CC(C(F)(F)F)=C5)C=C4)C1=C23	C49H49F3N12O5	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-B0OFU4	WO2024126617A1_16	.	CC1=C(N2CCC(=O)NC2=O)C=C(C(=O)NCCOCCOCCC(=O)N2CCC/C=C/C3=CN=C(N)C4=C3N(N=C4C3=CC=C(C(=O)NC4=NC=CC(C(F)(F)F)=C4)C=C3)[C@@H]3CCC[C@H](C3)NC(=O)C2)C=C1	C51H56F3N11O8	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-CKDRJF	WO2024126617A1_17	N-[2-[2-[3-[(2R,6R,13E)-18-amino-8-oxo-20-[4-[[4-(trifluoromethyl)pyridin-2-yl]carbamoyl]phenyl]-1,7,10,17,21-pentazatetracyclo[13.6.1.12,6.019,22]tricosa-13,15,17,19(22),20-pentaen-10-yl]-3-oxopropoxy]ethoxy]ethyl]-3-(2,4-dioxo-1,3-diazinan-1-yl)-4-methylbenzamide	CC1=CC=C(C(=O)NCCOCCOCCC(=O)N2CC/C=C/C3=CN=C(N)C4=C3N(N=C4C3=CC=C(C(=O)NC4=CC(C(F)(F)F)=CC=N4)C=C3)[C@@H]3CCC[C@H](C3)NC(=O)C2)C=C1N1CCC(=O)NC1=O	C50H54F3N11O8	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-FTU75R	WO2024126617A1_18	4-[(2R,6R,14E)-19-amino-10-[7-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]hept-6-ynoyl]-8-oxo-1,7,10,18,22-pentazatetracyclo[14.6.1.12,6.020,23]tetracosa-14,16,18,20(23),21-pentaen-21-yl]-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide	NC1=NC=C2/C=C/CCCN(C(=O)CCCCC#CC3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4)CC(=O)N[C@@H]3CCC[C@H](C3)N3N=C(C4=CC=C(C(=O)NC5=NC=CC(C(F)(F)F)=C5)C=C4)C1=C23	C52H51F3N10O6	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-JMR026	WO2024126617A1_19	.	NC1=NC=C2/C=C/CCN(C(=O)CCCCC#CC3=CC=C4C(=O)N(C5CCC(=O)NC5=O)CC4=C3)CC(=O)N[C@@H]3CCC[C@H](C3)N3N=C(C4=CC=C(C(=O)NC5=CC(C(F)(F)F)=CC=N5)C=C4)C1=C23	C51H49F3N10O6	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-1ENR4H	WO2024126617A1_20	4-[(2R,6R,14E)-19-amino-10-[6-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]hex-5-ynoyl]-8-oxo-1,7,10,18,22-pentazatetracyclo[14.6.1.12,6.020,23]tetracosa-14,16,18,20(23),21-pentaen-21-yl]-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide	NC1=NC=C2/C=C/CCCN(C(=O)CCCC#CC3=CC=C4C(=O)N(C5CCC(=O)NC5=O)CC4=C3)CC(=O)N[C@@H]3CCC[C@H](C3)N3N=C(C4=CC=C(C(=O)NC5=NC=CC(C(F)(F)F)=C5)C=C4)C1=C23	C51H49F3N10O6	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-CG5C8F	WO2024126617A1_21	4-[(2R,6R,13E)-18-amino-10-[6-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]hex-5-ynoyl]-8-oxo-1,7,10,17,21-pentazatetracyclo[13.6.1.12,6.019,22]tricosa-13,15,17,19(22),20-pentaen-20-yl]-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide	NC1=NC=C2/C=C/CCN(C(=O)CCCC#CC3=CC=C4C(=O)N(C5CCC(=O)NC5=O)CC4=C3)CC(=O)N[C@@H]3CCC[C@H](C3)N3N=C(C4=CC=C(C(=O)NC5=CC(C(F)(F)F)=CC=N5)C=C4)C1=C23	C50H47F3N10O6	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-Y9I4FN	WO2024126617A1_22	.	NC1=NC=C2/C=C/CCCN(C(=O)CCN3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)C(=O)N[C@@H]3CCC[C@H](C3)N3N=C(C4=CC=C(C(=O)NC5=CC(C(F)(F)F)=CCN5)C=C4)C1=C23	C51H53F3N12O7	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-CAK7Y1	WO2024126617A1_23	.	NC1=NC=C2/C=C/CCN(C(=O)CCN3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC(=O)N[C@@H]3CCC[C@H](C3)N3N=C(C4=CC=C(C(=O)NC5=CC(C(F)(F)F)=CCN5)C=C4)C1=C23	C51H53F3N12O7	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-1R08AO	WO2024126617A1_24	.	C=C1CN(C(=O)CO[C@@H]2CCN(C3=CC=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)C2)CC/C=C/C2=CN=C(N)C3=C2N(N=C3C2=CC=C(C(=O)NC3=CC(C(F)(F)F)=CC=N3)C=C2)[C@@H]2CCC[C@H](C2)N1	C51H50F3N11O7	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-97H4E2	WO2024126617A1_26	N-[2-[3-[(2R,6R,14E)-19-amino-8-oxo-21-[4-[[4-(trifluoromethyl)pyridin-2-yl]carbamoyl]phenyl]-1,7,10,18,22-pentazatetracyclo[14.6.1.12,6.020,23]tetracosa-14,16,18,20(23),21-pentaen-10-yl]-3-oxopropoxy]ethyl]-3-(2,4-dioxo-1,3-diazinan-1-yl)-4-methylbenzamide	CC1=CC=C(C(=O)NCCOCCC(=O)N2CCC/C=C/C3=CN=C(N)C4=C3N(N=C4C3=CC=C(C(=O)NC4=NC=CC(C(F)(F)F)=C4)C=C3)[C@@H]3CCC[C@H](C3)NC(=O)C2)C=C1N1CCC(=O)NC1=O	C49H52F3N11O7	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-QS3LIL	WO2024126617A1_27	N-[2-[3-[(2R,6R,13E)-18-amino-8-oxo-20-[4-[[4-(trifluoromethyl)pyridin-2-yl]carbamoyl]phenyl]-1,7,10,17,21-pentazatetracyclo[13.6.1.12,6.019,22]tricosa-13,15,17,19(22),20-pentaen-10-yl]-3-oxopropoxy]ethyl]-3-(2,4-dioxo-1,3-diazinan-1-yl)-4-methylbenzamide	CC1=C(N2CCC(=O)NC2=O)C=C(C(=O)NCCOCCC(=O)N2CC/C=C/C3=CN=C(N)C4=C3N(N=C4C3=CC=C(C(=O)NC4=CC(C(F)(F)F)=CC=N4)C=C3)[C@@H]3CCC[C@H](C3)NC(=O)C2)C=C1	C48H50F3N11O7	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-6626PZ	WO2024126617A1_28	.	COC1=CC=C(C(=O)N2CCN(CCC(=O)N3CCC/C=C/C4=CN=C(N)C5=C4N(N=C5C4=CC=C(C(=O)NC5=NC=CC(C(F)(F)F)=C5)C=C4)[C@@H]4CCC[C@H](C4)NC(=O)C3)CC2)C=C1N1CCC(=O)NC1=O	C51H55F3N12O7	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-QYAHYA	WO2024126617A1_29	.	COC1=CC=C(C(=O)N2CCN(CCC(=O)N3CC/C=C/C4=CN=C(N)C5=C4N(N=C5C4=CC=C(C(=O)NC5=CC(C(F)(F)F)=CC=N5)C=C4)C4CCC[C@H](C4)NC(=O)C3)CC2)C=C1N1CCC(=O)NC1=O	C50H53F3N12O7	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-L2GY11	WO2024126617A1_30	N-[2-[2-[3-[(2R,6R,14E)-19-amino-8-oxo-21-[4-[[4-(trifluoromethyl)pyridin-2-yl]carbamoyl]phenyl]-1,7,10,18,22-pentazatetracyclo[14.6.1.12,6.020,23]tetracosa-14,16,18,20(23),21-pentaen-10-yl]-3-oxopropoxy]ethoxy]ethyl]-3-(2,4-dioxo-1,3-diazinan-1-yl)-4-methoxybenzamide	COC1=C(N2CCC(=O)NC2=O)C=C(C(=O)NCCOCCOCCC(=O)N2CCC/C=C/C3=CN=C(N)C4=C3N(N=C4C3=CC=C(C(=O)NC4=NC=CC(C(F)(F)F)=C4)C=C3)[C@@H]3CCC[C@H](C3)NC(=O)C2)C=C1	C51H56F3N11O9	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-FEBIRJ	WO2024126617A1_31	N-[2-[2-[3-[(2R,6R,13E)-18-amino-8-oxo-20-[4-[[4-(trifluoromethyl)pyridin-2-yl]carbamoyl]phenyl]-1,7,10,17,21-pentazatetracyclo[13.6.1.12,6.019,22]tricosa-13,15,17,19(22),20-pentaen-10-yl]-3-oxopropoxy]ethoxy]ethyl]-3-(2,4-dioxo-1,3-diazinan-1-yl)-4-methoxybenzamide	COC1=C(N2CCC(=O)NC2=O)C=C(C(=O)NCCOCCOCCC(=O)N2CC/C=C/C3=CN=C(N)C4=C3N(N=C4C3=CC=C(C(=O)NC4=CC(C(F)(F)F)=CC=N4)C=C3)[C@@H]3CCC[C@H](C3)NC(=O)C2)C=C1	C50H54F3N11O9	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-D32WV7	WO2024126617A1_32	.	COC1=CC=C(C(=O)NCCOCCC(=O)N2CCC/C=C/C3=CN=C(N)C4=C3N(N=C4C3=CC=C(C(=O)NC4=NC=CC(C(F)(F)F)=C4)C=C3)[C@@H]3CCC[C@H](C3)NC(=O)C2)C=C1N1CCC(=O)NC1=O	C49H52F3N11O8	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-92ULE7	WO2024126617A1_33	N-[2-[3-[(2R,6R,13E)-18-amino-8-oxo-20-[4-[[4-(trifluoromethyl)pyridin-2-yl]carbamoyl]phenyl]-1,7,10,17,21-pentazatetracyclo[13.6.1.12,6.019,22]tricosa-13,15,17,19(22),20-pentaen-10-yl]-3-oxopropoxy]ethyl]-3-(2,4-dioxo-1,3-diazinan-1-yl)-4-methoxybenzamide	COC1=C(N2CCC(=O)NC2=O)C=C(C(=O)NCCOCCC(=O)N2CC/C=C/C3=CN=C(N)C4=C3N(N=C4C3=CC=C(C(=O)NC4=CC(C(F)(F)F)=CC=N4)C=C3)[C@@H]3CCC[C@H](C3)NC(=O)C2)C=C1	C48H50F3N11O8	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-56VC57	WO2024126617A1_34	4-[(2R,6R,14E)-19-amino-10-[2-[(3R)-1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]pyrrolidin-3-yl]oxyacetyl]-8-oxo-1,7,10,18,22-pentazatetracyclo[14.6.1.12,6.020,23]tetracosa-14,16,18,20(23),21-pentaen-21-yl]-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide	NC1=NC=C2/C=C/CCCN(C(=O)CO[C@@H]3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)C3)CC(=O)N[C@@H]3CCC[C@H](C3)N3N=C(C4=CC=C(C(=O)NC5=NC=CC(C(F)(F)F)=C5)C=C4)C1=C23	C51H50F3N11O8	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-4LHB1J	WO2024126617A1_35	N-[2-[2-[3-[(2R,6R,14E)-19-amino-8-oxo-21-[4-[[4-(trifluoromethyl)pyridin-2-yl]carbamoyl]phenyl]-1,7,11,18,22-pentazatetracyclo[14.6.1.12,6.020,23]tetracosa-14,16,18,20(23),21-pentaen-11-yl]-3-oxopropoxy]ethoxy]ethyl]-3-(2,4-dioxo-1,3-diazinan-1-yl)-4-methylbenzamide	CC1=C(N2CCC(=O)NC2=O)C=C(C(=O)NCCOCCOCCC(=O)N2CC/C=C/C3=CN=C(N)C4=C3N(N=C4C3=CC=C(C(=O)NC4=CC(C(F)(F)F)=CC=N4)C=C3)[C@@H]3CCC[C@H](C3)NC(=O)CC2)C=C1	C51H56F3N11O8	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-Q1T21C	WO2024126617A1_36	4-[(2R,6R,14E)-19-amino-11-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]propanoyl]-8-oxo-1,7,11,18,22-pentazatetracyclo[14.6.1.12,6.020,23]tetracosa-14,16,18,20(23),21-pentaen-21-yl]-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide	NC1=NC=C2/C=C/CCN(C(=O)CCN3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CCC(=O)N[C@@H]3CCC[C@H](C3)N3N=C(C4=CC=C(C(=O)NC5=CC(C(F)(F)F)=CC=N5)C=C4)C1=C23	C52H53F3N12O7	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-EL6TWQ	WO2024126617A1_37	N-[2-[3-[(2R,6R,14E)-19-amino-8-oxo-21-[4-[[4-(trifluoromethyl)pyridin-2-yl]carbamoyl]phenyl]-1,7,11,18,22-pentazatetracyclo[14.6.1.12,6.020,23]tetracosa-14,16,18,20(23),21-pentaen-11-yl]-3-oxopropoxy]ethyl]-3-(2,4-dioxo-1,3-diazinan-1-yl)-4-methylbenzamide	CC1=C(N2CCC(=O)NC2=O)C=C(C(=O)NCCOCCC(=O)N2CC/C=C/C3=CN=C(N)C4=C3N(N=C4C3=CC=C(C(=O)NC4=CC(C(F)(F)F)=CC=N4)C=C3)[C@@H]3CCC[C@H](C3)NC(=O)CC2)C=C1	C49H52F3N11O7	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-7DI00M	WO2024126617A1_38	4-[(2R,6R,14E)-19-amino-11-[3-[4-[3-(2,4-dioxo-1,3-diazinan-1-yl)-4-methoxybenzoyl]piperazin-1-yl]propanoyl]-8-oxo-1,7,11,18,22-pentazatetracyclo[14.6.1.12,6.020,23]tetracosa-14,16,18,20(23),21-pentaen-21-yl]-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide	COC1=C(N2CCC(=O)NC2=O)C=C(C(=O)N2CCN(CCC(=O)N3CC/C=C/C4=CN=C(N)C5=C4N(N=C5C4=CC=C(C(=O)NC5=CC(C(F)(F)F)=CC=N5)C=C4)[C@@H]4CCC[C@H](C4)NC(=O)CC3)CC2)C=C1	C51H55F3N12O7	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-23N1IV	WO2024126617A1_39	N-[2-[2-[3-[(2R,6R,14E)-19-amino-8-oxo-21-[4-[[4-(trifluoromethyl)pyridin-2-yl]carbamoyl]phenyl]-1,7,11,18,22-pentazatetracyclo[14.6.1.12,6.020,23]tetracosa-14,16,18,20(23),21-pentaen-11-yl]-3-oxopropoxy]ethoxy]ethyl]-3-(2,4-dioxo-1,3-diazinan-1-yl)-4-methoxybenzamide	COC1=C(N2CCC(=O)NC2=O)C=C(C(=O)NCCOCCOCCC(=O)N2CC/C=C/C3=CN=C(N)C4=C3N(N=C4C3=CC=C(C(=O)NC4=CC(C(F)(F)F)=CC=N4)C=C3)[C@@H]3CCC[C@H](C3)NC(=O)CC2)C=C1	C51H56F3N11O9	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-DMQFPD	WO2024126617A1_40	N-[2-[3-[(2R,6R,14E)-19-amino-8-oxo-21-[4-[[4-(trifluoromethyl)pyridin-2-yl]carbamoyl]phenyl]-1,7,11,18,22-pentazatetracyclo[14.6.1.12,6.020,23]tetracosa-14,16,18,20(23),21-pentaen-11-yl]-3-oxopropoxy]ethyl]-3-(2,4-dioxo-1,3-diazinan-1-yl)-4-methoxybenzamide	COC1=C(N2CCC(=O)NC2=O)C=C(C(=O)NCCOCCC(=O)N2CC/C=C/C3=CN=C(N)C4=C3N(N=C4C3=CC=C(C(=O)NC4=CC(C(F)(F)F)=CC=N4)C=C3)[C@@H]3CCC[C@H](C3)NC(=O)CC2)C=C1	C49H52F3N11O8	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-89R3D9	WO2024126617A1_41	4-[(2R,6R,14E)-19-amino-11-[2-[(3R)-1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]pyrrolidin-3-yl]oxyacetyl]-8-oxo-1,7,11,18,22-pentazatetracyclo[14.6.1.12,6.020,23]tetracosa-14,16,18,20(23),21-pentaen-21-yl]-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide	NC1=NC=C2/C=C/CCN(C(=O)CO[C@@H]3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)C3)CCC(=O)N[C@@H]3CCC[C@H](C3)N3N=C(C4=CC=C(C(=O)NC5=CC(C(F)(F)F)=CC=N5)C=C4)C1=C23	C51H50F3N11O8	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-TKBXMH	WO2024126617A1_42	4-[(2R,6R,14E)-19-amino-10-[3-[1-[3-(2,4-dioxo-1,3-diazinan-1-yl)-4-methylbenzoyl]piperidin-4-yl]propanoyl]-8-oxo-1,7,10,18,22-pentazatetracyclo[14.6.1.12,6.020,23]tetracosa-14,16,18,20(23),21-pentaen-21-yl]-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide	CC1=CC=C(C(=O)N2CCC(CCC(=O)N3CCC/C=C/C4=CN=C(N)C5=C4N(N=C5C4=CC=C(C(=O)NC5=NC=CC(C(F)(F)F)=C5)C=C4)[C@@H]4CCC[C@H](C4)NC(=O)C3)CC2)C=C1N1CCC(=O)NC1=O	C52H56F3N11O6	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-R3AYM8	WO2024126617A1_43	4-[(2R,6R,14E)-19-amino-10-[3-[1-[3-(2,4-dioxo-1,3-diazinan-1-yl)-4-methoxybenzoyl]piperidin-4-yl]propanoyl]-8-oxo-1,7,10,18,22-pentazatetracyclo[14.6.1.12,6.020,23]tetracosa-14,16,18,20(23),21-pentaen-21-yl]-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide	COC1=CC=C(C(=O)N2CCC(CCC(=O)N3CCC/C=C/C4=CN=C(N)C5=C4N(N=C5C4=CC=C(C(=O)NC5=NC=CC(C(F)(F)F)=C5)C=C4)[C@@H]4CCC[C@H](C4)NC(=O)C3)CC2)C=C1N1CCC(=O)NC1=O	C52H56F3N11O7	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-BBP984	WO2024126617A1_44	.	NC1=NC=C2/C=C/CCCN(C(=O)CCC3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC(=O)N[C@@H]3CCC[C@H](C3)N3N=C(C4=CC=C(C(=O)NC5=NC=CC(C(F)(F)F)=C5)C=C4)C1=C23	C53H54F3N11O7	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-Z43UYJ	WO2024126617A1_45	4-[(2R,6R,14E)-19-amino-10-[[(3S)-1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]pyrrolidin-3-yl]methyl]-8-oxo-1,7,10,18,22-pentazatetracyclo[14.6.1.12,6.020,23]tetracosa-14,16,18,20(23),21-pentaen-21-yl]-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide	NC1=NC=C2/C=C/CCCN(C[C@@H]3CCN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)CC(=O)N[C@@H]3CCC[C@H](C3)N3N=C(C4=CC=C(C(=O)NC5=NC=CC(C(F)(F)F)=C5)C=C4)C1=C23	C50H50F3N11O6	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-DF7H8J	WO2024126617A1_46	.	CC1=C(N2CCC(=O)NC2=O)C=C(C(=O)N2CCC(CCC(=O)N3CC/C=C/C4=CN=C(N)C5=C4N(N=C5C4=CC=C(C(=O)NC5=CC(C(F)(F)F)=CC=N5)C=C4)[C@@H]4CCC[C@H](C4)NC(=O)CC3)CC2)C=C1	C52H56F3N11O6	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-BZB89P	WO2024126617A1_47	4-[(2R,6R,14E)-19-amino-11-[3-[1-[3-(2,4-dioxo-1,3-diazinan-1-yl)-4-methoxybenzoyl]piperidin-4-yl]propanoyl]-8-oxo-1,7,11,18,22-pentazatetracyclo[14.6.1.12,6.020,23]tetracosa-14,16,18,20(23),21-pentaen-21-yl]-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide	COC1=C(N2CCC(=O)NC2=O)C=C(C(=O)N2CCC(CCC(=O)N3CC/C=C/C4=CN=C(N)C5=C4N(N=C5C4=CC=C(C(=O)NC5=CC(C(F)(F)F)=CC=N5)C=C4)[C@@H]4CCC[C@H](C4)NC(=O)CC3)CC2)C=C1	C52H56F3N11O7	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-KU2P61	WO2024126617A1_48	4-[(2R,6R,14E)-19-amino-11-[3-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]propanoyl]-8-oxo-1,7,11,18,22-pentazatetracyclo[14.6.1.12,6.020,23]tetracosa-14,16,18,20(23),21-pentaen-21-yl]-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide	NC1=NC=C2/C=C/CCN(C(=O)CCC3CCN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CCC(=O)N[C@@H]3CCC[C@H](C3)N3N=C(C4=CC=C(C(=O)NC5=CC(C(F)(F)F)=CC=N5)C=C4)C1=C23	C53H54F3N11O7	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-FB0QKP	WO2024126617A1_49	(2S,4R)-1-[(2S)-2-[[4-[(2R,6R,14E)-19-amino-8-oxo-21-[4-[[4-(trifluoromethyl)pyridin-2-yl]carbamoyl]phenyl]-1,7,11,18,22-pentazatetracyclo[14.6.1.12,6.020,23]tetracosa-14,16,18,20(23),21-pentaen-11-yl]-4-oxobutanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCC(=O)N3CC/C=C/C4=CN=C(N)C5=C4N(N=C5C4=CC=C(C(=O)NC5=CC(C(F)(F)F)=CC=N5)C=C4)[C@@H]4CCC[C@H](C4)NC(=O)CC3)C(C)(C)C)C=C2)SC=N1	C58H65F3N12O7S	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-M9WGF6	WO2024126617A1_50	4-[(2R,6R,14E)-19-amino-11-[3-[4-[1-[3-(2,4-dioxo-1,3-diazinan-1-yl)-4-methylbenzoyl]piperidin-4-yl]oxypiperidin-1-yl]propanoyl]-8-oxo-1,7,11,18,22-pentazatetracyclo[14.6.1.12,6.020,23]tetracosa-14,16,18,20(23),21-pentaen-21-yl]-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide	CC1=C(N2CCC(=O)NC2=O)C=C(C(=O)N2CCC(OC3CCN(CCC(=O)N4CC/C=C/C5=CN=C(N)C6=C5N(N=C6C5=CC=C(C(=O)NC6=CC(C(F)(F)F)=CC=N6)C=C5)[C@@H]5CCC[C@H](C5)NC(=O)CC4)CC3)CC2)C=C1	C57H65F3N12O7	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-P3MG20	WO2024126617A1_51	4-[(2R,6R,14E)-19-amino-11-[3-[4-[1-[3-(2,4-dioxo-1,3-diazinan-1-yl)-4-methoxybenzoyl]piperidin-4-yl]oxypiperidin-1-yl]propanoyl]-8-oxo-1,7,11,18,22-pentazatetracyclo[14.6.1.12,6.020,23]tetracosa-14,16,18,20(23),21-pentaen-21-yl]-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide	COC1=C(N2CCC(=O)NC2=O)C=C(C(=O)N2CCC(OC3CCN(CCC(=O)N4CC/C=C/C5=CN=C(N)C6=C5N(N=C6C5=CC=C(C(=O)NC6=CC(C(F)(F)F)=CC=N6)C=C5)[C@@H]5CCC[C@H](C5)NC(=O)CC4)CC3)CC2)C=C1	C57H65F3N12O8	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-N7B5VC	WO2024126617A1_52	N-[2-[2-[3-[(2S,5R,13E)-18-amino-6-oxo-20-[4-[[4-(trifluoromethyl)pyridin-2-yl]carbamoyl]phenyl]-1,4,7,17,21-pentazatetracyclo[13.6.1.12,5.019,22]tricosa-13,15,17,19(22),20-pentaen-4-yl]-3-oxopropoxy]ethoxy]ethyl]-3-(2,4-dioxo-1,3-diazinan-1-yl)-4-methoxybenzamide	COC1=C(N2CCC(=O)NC2=O)C=C(C(=O)NCCOCCOCCC(=O)N2C[C@@H]3C[C@@H]2C(=O)NCCCCC/C=C/C2=CN=C(N)C4=C2N3N=C4C2=CC=C(C(=O)NC3=CC(C(F)(F)F)=CC=N3)C=C2)C=C1	C50H54F3N11O9	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-HBNXL0	WO2024126617A1_53	N-[2-[3-[(2S,5R,13E)-18-amino-6-oxo-20-[4-[[4-(trifluoromethyl)pyridin-2-yl]carbamoyl]phenyl]-1,4,7,17,21-pentazatetracyclo[13.6.1.12,5.019,22]tricosa-13,15,17,19(22),20-pentaen-4-yl]-3-oxopropoxy]ethyl]-3-(2,4-dioxo-1,3-diazinan-1-yl)-4-methoxybenzamide	COC1=C(N2CCC(=O)NC2=O)C=C(C(=O)NCCOCCC(=O)N2C[C@@H]3C[C@@H]2C(=O)NCCCCC/C=C/C2=CN=C(N)C4=C2N3N=C4C2=CC=C(C(=O)NC3=CC(C(F)(F)F)=CC=N3)C=C2)C=C1	C48H50F3N11O8	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-CU9MLQ	WO2024126617A1_54	.	COC1=C(N2CCC(=O)NC2=O)C=C(C(=O)NCCOCCOCCC(=O)N2CC/C=C/C3=CN=C(N)C4=C(C5=CC=C(C(=O)NC6=CC(C(F)(F)F)=CC=N6)C=C5)N=C(C5CC[C@H](C5)NC(=O)C2)N34)C=C1	C49H52F3N11O9	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-GLXTNU	WO2024126617A1_55	N-[2-[3-[(2R,5R,12E)-17-amino-7-oxo-19-[4-[[4-(trifluoromethyl)pyridin-2-yl]carbamoyl]phenyl]-6,9,16,20,21-pentazatetracyclo[12.6.1.12,5.018,21]docosa-1(20),12,14,16,18-pentaen-9-yl]-3-oxopropoxy]ethyl]-3-(2,4-dioxo-1,3-diazinan-1-yl)-4-methoxybenzamide	COC1=CC=C(C(=O)NCCOCCC(=O)N2CC/C=C/C3=CN=C(N)C4=C(C5=CC=C(C(=O)NC6=CC(C(F)(F)F)=CC=N6)C=C5)N=C([C@@H]5CC[C@H](C5)NC(=O)C2)N34)C=C1N1CCC(=O)NC1=O	C47H48F3N11O8	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-88NCG4	WO2024126617A1_56	N-[2-[2-[3-[(2R,5R,12E)-17-amino-19-[4-[[(5-fluoro-2-methoxybenzoyl)amino]methyl]phenyl]-7-oxo-6,9,16,20,21-pentazatetracyclo[12.6.1.12,5.018,21]docosa-1(20),12,14,16,18-pentaen-9-yl]-3-oxopropoxy]ethoxy]ethyl]-3-(2,4-dioxo-1,3-diazinan-1-yl)-4-methoxybenzamide	COC1=C(C(=O)NCC2=CC=C(C3=C4C(N)=NC=C5/C=C/CCN(C(=O)CCOCCOCCNC(=O)C6=CC(N7CCC(=O)NC7=O)=C(OC)C=C6)CC(=O)N[C@@H]6CC[C@H](C6)C(=N3)N54)C=C2)C=C(F)C=C1	C51H57FN10O10	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-KMI0F1	WO2024126617A1_57	N-[2-[3-[(2R,5R,12E)-17-amino-19-[4-[[(5-fluoro-2-methoxybenzoyl)amino]methyl]phenyl]-7-oxo-6,9,16,20,21-pentazatetracyclo[12.6.1.12,5.018,21]docosa-1(20),12,14,16,18-pentaen-9-yl]-3-oxopropoxy]ethyl]-3-(2,4-dioxo-1,3-diazinan-1-yl)-4-methoxybenzamide	COC1=CC=C(C(=O)NCCOCCC(=O)N2CC/C=C/C3=CN=C(N)C4=C(C5=CC=C(CNC(=O)C6=C(OC)C=CC(F)=C6)C=C5)N=C([C@@H]5CC[C@H](C5)NC(=O)C2)N34)C=C1N1CCC(=O)NC1=O	C49H53FN10O9	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-YKZPYT	WO2024126617A1_58	4-[(2R,6R,14E)-19-amino-10-[2-[1-[[6-[3-(2,4-dioxo-1,3-diazinan-1-yl)azetidin-1-yl]pyridin-3-yl]methyl]piperidin-4-yl]acetyl]-8-oxo-1,7,10,18,22-pentazatetracyclo[14.6.1.12,6.020,23]tetracosa-14,16,18,20(23),21-pentaen-21-yl]-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide	NC1=NC=C2/C=C/CCCN(C(=O)CC3CCN(CC4=CC=C(N5CC(N6CCC(=O)NC6=O)C5)N=C4)CC3)CC(=O)N[C@@H]3CCC[C@H](C3)N3N=C(C4=CC=C(C(=O)NC5=NC=CC(C(F)(F)F)=C5)C=C4)C1=C23	C52H58F3N13O5	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-YTRU9O	WO2024126617A1_59	4-[(2S,5R,13E)-18-amino-4-[2-[1-[[6-[3-(2,4-dioxo-1,3-diazinan-1-yl)azetidin-1-yl]pyridin-3-yl]methyl]piperidin-4-yl]acetyl]-6-oxo-1,4,7,17,21-pentazatetracyclo[13.6.1.12,5.019,22]tricosa-13,15,17,19(22),20-pentaen-20-yl]-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide	NC1=NC=C2/C=C/CCCCCNC(=O)[C@H]3C[C@@H](CN3C(=O)CC3CCN(CC4=CN=C(N5CC(N6CCC(=O)NC6=O)C5)C=C4)CC3)N3N=C(C4=CC=C(C(=O)NC5=CC(C(F)(F)F)=CC=N5)C=C4)C1=C23	C51H56F3N13O5	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-NSDZO7	WO2024126617A1_60	5-[4-[[4-[2-[(2S,5R,13E)-18-amino-6-oxo-20-[4-[[4-(trifluoromethyl)pyridin-2-yl]carbamoyl]phenyl]-1,4,7,17,21-pentazatetracyclo[13.6.1.12,5.019,22]tricosa-13,15,17,19(22),20-pentaen-4-yl]-2-oxoethyl]piperidin-1-yl]methyl]piperidin-1-yl]-N-(2,6-dioxopiperidin-3-yl)pyridine-2-carboxamide	NC1=NC=C2/C=C/CCCCCNC(=O)[C@H]3C[C@@H](CN3C(=O)CC3CCN(CC4CCN(C5=CN=C(C(=O)NC6CCC(=O)NC6=O)C=C5)CC4)CC3)N3N=C(C4=CC=C(C(=O)NC5=CC(C(F)(F)F)=CC=N5)C=C4)C1=C23	C55H62F3N13O6	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-9J77DO	WO2024126617A1_61	4-[(2R,6R,14E)-19-amino-11-[2-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperidin-4-yl]acetyl]-8-oxo-1,7,11,18,22-pentazatetracyclo[14.6.1.12,6.020,23]tetracosa-14,16,18,20(23),21-pentaen-21-yl]-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide	NC1=NC=C2/C=C/CCN(C(=O)CC3CCN(CC4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)CCC(=O)N[C@@H]3CCC[C@H](C3)N3N=C(C4=CC=C(C(=O)NC5=CC(C(F)(F)F)=CC=N5)C=C4)C1=C23	C58H63F3N12O7	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-51AC9Z	WO2024126617A1_62	4-[(2R,5R,12E)-17-amino-9-[3-[4-[3-(2,4-dioxo-1,3-diazinan-1-yl)-4-methylbenzoyl]piperazin-1-yl]propanoyl]-7-oxo-6,9,16,20,21-pentazatetracyclo[12.6.1.12,5.018,21]docosa-1(20),12,14,16,18-pentaen-19-yl]-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide	CC1=C(N2CCC(=O)NC2=O)C=C(C(=O)N2CCN(CCC(=O)N3CC/C=C/C4=CN=C(N)C5=C(C6=CC=C(C(=O)NC7=CC(C(F)(F)F)=CC=N7)C=C6)N=C([C@@H]6CC[C@H](C6)NC(=O)C3)N45)CC2)C=C1	C49H51F3N12O6	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-3KWDN9	WO2024126617A1_63	4-[(2R,5R,12E)-17-amino-9-[3-[4-[3-(2,4-dioxo-1,3-diazinan-1-yl)-4-methoxybenzoyl]piperazin-1-yl]propanoyl]-7-oxo-6,9,16,20,21-pentazatetracyclo[12.6.1.12,5.018,21]docosa-1(20),12,14,16,18-pentaen-19-yl]-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide	COC1=C(N2CCC(=O)NC2=O)C=C(C(=O)N2CCN(CCC(=O)N3CC/C=C/C4=CN=C(N)C5=C(C6=CC=C(C(=O)NC7=CC(C(F)(F)F)=CC=N7)C=C6)N=C([C@@H]6CC[C@H](C6)NC(=O)C3)N45)CC2)C=C1	C49H51F3N12O7	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-15NHIB	WO2024126617A1_64	N-[[4-[(2R,5R,12E)-17-amino-9-[3-[4-[3-(2,4-dioxo-1,3-diazinan-1-yl)-4-methylbenzoyl]piperazin-1-yl]propanoyl]-7-oxo-6,9,16,20,21-pentazatetracyclo[12.6.1.12,5.018,21]docosa-1(20),12,14,16,18-pentaen-19-yl]phenyl]methyl]-5-fluoro-2-methoxybenzamide	COC1=C(C(=O)NCC2=CC=C(C3=C4C(N)=NC=C5/C=C/CCN(C(=O)CCN6CCN(C(=O)C7=CC(N8CCC(=O)NC8=O)=C(C)C=C7)CC6)CC(=O)N[C@@H]6CC[C@H](C6)C(=N3)N54)C=C2)C=C(F)C=C1	C51H56FN11O7	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-1CSJHT	WO2024126617A1_65	N-[[4-[(2R,5R,12E)-17-amino-9-[3-[4-[3-(2,4-dioxo-1,3-diazinan-1-yl)-4-methoxybenzoyl]piperazin-1-yl]propanoyl]-7-oxo-6,9,16,20,21-pentazatetracyclo[12.6.1.12,5.018,21]docosa-1(20),12,14,16,18-pentaen-19-yl]phenyl]methyl]-5-fluoro-2-methoxybenzamide	COC1=C(C(=O)NCC2=CC=C(C3=C4C(N)=NC=C5/C=C/CCN(C(=O)CCN6CCN(C(=O)C7=CC(N8CCC(=O)NC8=O)=C(OC)C=C7)CC6)CC(=O)N[C@@H]6CC[C@H](C6)C(=N3)N54)C=C2)C=C(F)C=C1	C51H56FN11O8	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-WM7KP3	WO2024126617A1_66	4-[(2R,6R,14E)-19-amino-10-[2-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperidin-4-yl]acetyl]-8-oxo-1,7,10,18,22-pentazatetracyclo[14.6.1.12,6.020,23]tetracosa-14,16,18,20(23),21-pentaen-21-yl]-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide	NC1=NC=C2/C=C/CCCN(C(=O)CC3CCN(CC4CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)CC(=O)N[C@@H]3CCC[C@H](C3)N3N=C(C4=CC=C(C(=O)NC5=NC=CC(C(F)(F)F)=C5)C=C4)C1=C23	C58H63F3N12O7	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-GOGNN3	WO2024126617A1_67	4-[(2R,6R,13E)-18-amino-10-[2-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperidin-4-yl]acetyl]-8-oxo-1,7,10,17,21-pentazatetracyclo[13.6.1.12,6.019,22]tricosa-13,15,17,19(22),20-pentaen-20-yl]-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide	NC1=NC=C2/C=C/CCN(C(=O)CC3CCN(CC4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)CC(=O)N[C@@H]3CCC[C@H](C3)N3N=C(C4=CC=C(C(=O)NC5=CC(C(F)(F)F)=CC=N5)C=C4)C1=C23	C57H61F3N12O7	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-5FAJJ6	WO2024126617A1_68	.	NC1=NC=C2/C=C/CCCN(C(=O)CCC3CCN(CC4CCN(C5=CN=C(C(=O)NC6CCC(=O)NC6=O)C=C5)CC4)CC3)CC(=O)N[C@@H]3CCC[C@H](C3)N3N=C(C4=CC=C(C(=O)NC5=NC=CC(C(F)(F)F)=C5)C=C4)C1=C23	C57H66F3N13O6	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-WZW35U	WO2024126617A1_69	5-[4-[[4-[3-[(2S,5R,13E)-18-amino-6-oxo-20-[4-[[4-(trifluoromethyl)pyridin-2-yl]carbamoyl]phenyl]-1,4,7,17,21-pentazatetracyclo[13.6.1.12,5.019,22]tricosa-13,15,17,19(22),20-pentaen-4-yl]-3-oxopropyl]piperidin-1-yl]methyl]piperidin-1-yl]-N-(2,6-dioxopiperidin-3-yl)pyridine-2-carboxamide	NC1=NC=C2/C=C/CCCCCNC(=O)[C@H]3C[C@@H](CN3C(=O)CCC3CCN(CC4CCN(C5=CN=C(C(=O)NC6CCC(=O)NC6=O)C=C5)CC4)CC3)N3N=C(C4=CC=C(C(=O)NC5=CC(C(F)(F)F)=CC=N5)C=C4)C1=C23	C56H64F3N13O6	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-BX6PCZ	WO2024126617A1_70	.	CC1=C(N2CCC(=O)NC2=O)C=C(C(=O)N2CCC3(CCN(CC(=O)N4C[C@@H]5C[C@@H]4C(=O)NCCCCC/C=C/C4=CN=C(N)C6=C4N5N=C6C4=CC=C(C(=O)NC5=CC(C(F)(F)F)=CC=N5)C=C4)CC3)CC2)C=C1	C54H59F3N12O6	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-IG9773	WO2024126617A1_71	.	NC1=NC=C2/C=C/CCCN(C(=O)CN3CCC4(CC3)CCN(C(=O)C3=CC=CC(N5CCC(=O)NC5=O)=C3)CC4)CC(=O)N[C@@H]3CCC[C@H](C3)N3N=C(C4=CC=C(C(=O)NC5=NC=CC(C(F)(F)F)=C5)C=C4)C1=C23	C54H59F3N12O6	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-LGI7A6	WO2024126617A1_72	4-[(2S,5R,13E)-18-amino-4-[3-[3-[3-(2,4-dioxo-1,3-diazinan-1-yl)-4-methylbenzoyl]-3,9-diazaspiro[5.5]undecan-9-yl]propanoyl]-6-oxo-1,4,7,17,21-pentazatetracyclo[13.6.1.12,5.019,22]tricosa-13,15,17,19(22),20-pentaen-20-yl]-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide	CC1=C(N2CCC(=O)NC2=O)C=C(C(=O)N2CCC3(CCN(CCC(=O)N4C[C@@H]5C[C@@H]4C(=O)NCCCCC/C=C/C4=CN=C(N)C6=C4N5N=C6C4=CC=C(C(=O)NC5=CC(C(F)(F)F)=CC=N5)C=C4)CC3)CC2)C=C1	C55H61F3N12O6	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-W0C5J1	WO2024126617A1_73	.	CC1=CC=C(C(=O)N2CCC3(CCN(CCC(=O)N4CCC/C=C/C5=CN=C(N)C6=C5N(N=C6C5=CC=C(C(=O)NC6=NC=CC(C(F)(F)F)=C6)C=C5)[C@@H]5CCC[C@H](C5)NC(=O)C4)CC3)CC2)C=C1N1CCC(=O)NC1=O	C56H63F3N12O6	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-SWCMQW	WO2024126617A1_74	.	NC1=NC=C2/C=C/CCCCCNC(=O)[C@H]3C[C@@H](CN3C(=O)CCC3CCN(CC4=CN=C(N5CC(N6CCC(=O)NC6=O)C5)C=C4)CC3)N3N=C(C4=CC=C(C(=O)NC5=CC(C(F)(F)F)=CC=N5)C=C4)C1=C23	C52H58F3N13O5	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-FH5HOZ	WO2024126617A1_75	4-[(2R,5R,12E)-17-amino-9-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]propanoyl]-7-oxo-6,9,16,20,21-pentazatetracyclo[12.6.1.12,5.018,21]docosa-1(20),12,14,16,18-pentaen-19-yl]-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide	NC1=NC=C2/C=C/CCN(C(=O)CCN3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC(=O)N[C@@H]3CC[C@H](C3)C3=NC(C4=CC=C(C(=O)NC5=CC(C(F)(F)F)=CC=N5)C=C4)=C1N23	C50H49F3N12O7	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-LR4S0Q	WO2024126617A1_76	4-[(2R,5R,12E)-17-amino-9-[6-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]hex-5-ynoyl]-7-oxo-6,9,16,20,21-pentazatetracyclo[12.6.1.12,5.018,21]docosa-1(20),12,14,16,18-pentaen-19-yl]-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide	NC1=NC=C2/C=C/CCN(C(=O)CCCC#CC3=CC=C4C(=O)N(C5CCC(=O)NC5=O)CC4=C3)CC(=O)N[C@@H]3CC[C@H](C3)C3=NC(C4=CC=C(C(=O)NC5=CC(C(F)(F)F)=CC=N5)C=C4)=C1N23	C49H45F3N10O6	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-GON90A	WO2024126617A1_77	4-[(2R,6R,14E)-19-amino-11-[3-[1-[2-[4-(2,6-dioxopiperidin-3-yl)phenoxy]acetyl]piperidin-4-yl]propanoyl]-8-oxo-1,7,11,18,22-pentazatetracyclo[14.6.1.12,6.020,23]tetracosa-14,16,18,20(23),21-pentaen-21-yl]-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide	NC1=NC=C2/C=C/CCN(C(=O)CCC3CCN(C(=O)COC4=CC=C(C5CCC(=O)NC5=O)C=C4)CC3)CCC(=O)N[C@@H]3CCC[C@H](C3)N3N=C(C4=CC=C(C(=O)NC5=CC(C(F)(F)F)=CC=N5)C=C4)C1=C23	C53H57F3N10O7	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-I5XVGH	WO2024126617A1_78	4-[(2R,6R,14E)-19-amino-11-[2-[1-[[1-[3-(2,4-dioxo-1,3-diazinan-1-yl)-4-methylbenzoyl]piperidin-4-yl]methyl]piperidin-4-yl]acetyl]-8-oxo-1,7,11,18,22-pentazatetracyclo[14.6.1.12,6.020,23]tetracosa-14,16,18,20(23),21-pentaen-21-yl]-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide	CC1=CC=C(C(=O)N2CCC(CN3CCC(CC(=O)N4CC/C=C/C5=CN=C(N)C6=C5N(N=C6C5=CC=C(C(=O)NC6=CC(C(F)(F)F)=CC=N6)C=C5)[C@@H]5CCC[C@H](C5)NC(=O)CC4)CC3)CC2)C=C1N1CCC(=O)NC1=O	C57H65F3N12O6	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-XMW1IA	WO2024126617A1_79	4-[(2R,6R,14E)-19-amino-11-[3-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]oxypiperidin-1-yl]propanoyl]-8-oxo-1,7,11,18,22-pentazatetracyclo[14.6.1.12,6.020,23]tetracosa-14,16,18,20(23),21-pentaen-21-yl]-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide	NC1=NC=C2/C=C/CCN(C(=O)CCN3CCC(OC4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)CCC(=O)N[C@@H]3CCC[C@H](C3)N3N=C(C4=CC=C(C(=O)NC5=CC(C(F)(F)F)=CC=N5)C=C4)C1=C23	C58H63F3N12O8	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-1XSR4F	WO2024126617A1_80	.	CC1=CC=C(C(=O)N2CCC(CN3CCC(CC(=O)N4CCC/C=C/C5=CN=C(N)C6=C5N(N=C6C5=CC=C(C(=O)NC6=NC=CC(C(F)(F)F)=C6)C=C5)[C@@H]5CCC[C@H](C5)NC(=O)C4)CC3)CC2)C=C1N1CCC(=O)NC1=O	C57H65F3N12O6	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-BL3I3E	WO2024126617A1_81	4-[(2R,6R,13E)-18-amino-10-[2-[1-[[1-[3-(2,4-dioxo-1,3-diazinan-1-yl)-4-methylbenzoyl]piperidin-4-yl]methyl]piperidin-4-yl]acetyl]-8-oxo-1,7,10,17,21-pentazatetracyclo[13.6.1.12,6.019,22]tricosa-13,15,17,19(22),20-pentaen-20-yl]-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide	CC1=CC=C(C(=O)N2CCC(CN3CCC(CC(=O)N4CC/C=C/C5=CN=C(N)C6=C5N(N=C6C5=CC=C(C(=O)NC6=NC=CC(C(F)(F)F)=C6)C=C5)[C@@H]5CCC[C@H](C5)NC(=O)C4)CC3)CC2)C=C1N1CCC(=O)NC1=O	C56H63F3N12O6	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-ZXVFY7	WO2024126617A1_82	.	CC1=C(N2CCC(=O)NC2=O)C=C(C(=O)N2CCC(CN3CCC(CC(=O)N4C[C@@H]5C[C@@H]4C(=O)NCCCCC/C=C/C4=CN=C(N)C6=C4N5N=C6C4=CC=C(C(=O)NC5CC(C(F)(F)F)=CC=N5)C=C4)CC3)CC2)C=C1	C56H65F3N12O6	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-5J43PW	WO2024126617A1_83	N-[2-[2-[3-[(2R,5R,12E)-17-amino-7-oxo-19-[4-[[4-(trifluoromethyl)pyridin-2-yl]carbamoyl]phenyl]-6,9,16,20,21-pentazatetracyclo[12.6.1.12,5.018,21]docosa-1(20),12,14,16,18-pentaen-9-yl]-3-oxopropoxy]ethoxy]ethyl]-3-(2,4-dioxo-1,3-diazinan-1-yl)-4-methylbenzamide	CC1=C(N2CCC(=O)NC2=O)C=C(C(=O)NCCOCCOCCC(=O)N2CC/C=C/C3=CN=C(N)C4=C(C5=CC=C(C(=O)NC6=CC(C(F)(F)F)=CC=N6)C=C5)N=C([C@@H]5CC[C@H](C5)NC(=O)C2)N34)C=C1	C49H52F3N11O8	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-GSCZ4Z	WO2024126617A1_84	.	CC1=CC=C(C(=O)NCCOCCC(=O)N2CC/C=C/C3=CN=C(N)C4=C(C5=CC=C(C(=O)NC6=CC(C(F)(F)F)=CC=N6)C=C5)N=C([C@@H]5CC[C@H](C5)NC(=O)C2)N34)C=C1N1CCC(=O)NC1=O	C47H48F3N11O7	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-EUYZ72	WO2024126617A1_85	N-[2-[2-[3-[(2R,5R,12E)-17-amino-19-[4-[[(5-fluoro-2-methoxybenzoyl)amino]methyl]phenyl]-7-oxo-6,9,16,20,21-pentazatetracyclo[12.6.1.12,5.018,21]docosa-1(20),12,14,16,18-pentaen-9-yl]-3-oxopropoxy]ethoxy]ethyl]-3-(2,4-dioxo-1,3-diazinan-1-yl)-4-methylbenzamide	COC1=C(C(=O)NCC2=CC=C(C3=C4C(N)=NC=C5/C=C/CCN(C(=O)CCOCCOCCNC(=O)C6=CC(N7CCC(=O)NC7=O)=C(C)C=C6)CC(=O)N[C@@H]6CC[C@H](C6)C(=N3)N54)C=C2)C=C(F)C=C1	C51H57FN10O9	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-QONBJ5	WO2024126617A1_86	N-[2-[3-[(2R,5R,12E)-17-amino-19-[4-[[(5-fluoro-2-methoxybenzoyl)amino]methyl]phenyl]-7-oxo-6,9,16,20,21-pentazatetracyclo[12.6.1.12,5.018,21]docosa-1(20),12,14,16,18-pentaen-9-yl]-3-oxopropoxy]ethyl]-3-(2,4-dioxo-1,3-diazinan-1-yl)-4-methylbenzamide	COC1=C(C(=O)NCC2=CC=C(C3=C4C(N)=NC=C5/C=C/CCN(C(=O)CCOCCNC(=O)C6=CC=C(C)C(N7CCC(=O)NC7=O)=C6)CC(=O)N[C@@H]6CC[C@H](C6)C(=N3)N54)C=C2)C=C(F)C=C1	C49H53FN10O8	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-NRCMV1	WO2024126617A1_87	5-[4-[[4-[2-[(2R,6R,14E)-19-amino-8-oxo-21-[4-[[4-(trifluoromethyl)pyridin-2-yl]carbamoyl]phenyl]-1,7,10,18,22-pentazatetracyclo[14.6.1.12,6.020,23]tetracosa-14,16,18,20(23),21-pentaen-10-yl]-2-oxoethyl]piperidin-1-yl]methyl]piperidin-1-yl]-N-(2,6-dioxopiperidin-3-yl)pyridine-2-carboxamide	NC1=NC=C2/C=C/CCCN(C(=O)CC3CCN(CC4CCN(C5=CN=C(C(=O)NC6CCC(=O)NC6=O)C=C5)CC4)CC3)CC(=O)N[C@@H]3CCC[C@H](C3)N3N=C(C4=CC=C(C(=O)NC5=NC=CC(C(F)(F)F)=C5)C=C4)C1=C23	C56H64F3N13O6	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-7MB3BB	WO2024126617A1_88	4-[(2R,6R,14E)-19-amino-10-[3-[1-[[6-[3-(2,4-dioxo-1,3-diazinan-1-yl)azetidin-1-yl]pyridin-3-yl]methyl]piperidin-4-yl]propanoyl]-8-oxo-1,7,10,18,22-pentazatetracyclo[14.6.1.12,6.020,23]tetracosa-14,16,18,20(23),21-pentaen-21-yl]-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide	NC1=NC=C2/C=C/CCCN(C(=O)CCC3CCN(CC4=CN=C(N5CC(N6CCC(=O)NC6=O)C5)C=C4)CC3)CC(=O)N[C@@H]3CCC[C@H](C3)N3N=C(C4=CC=C(C(=O)NC5=NC=CC(C(F)(F)F)=C5)C=C4)C1=C23	C53H60F3N13O5	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-JMT19G	WO2024126617A1_89	4-[(2R,6R,14E)-19-amino-10-[4-[1-[3-(2,4-dioxo-1,3-diazinan-1-yl)-4-methylbenzoyl]piperidin-4-yl]butanoyl]-8-oxo-1,7,10,18,22-pentazatetracyclo[14.6.1.12,6.020,23]tetracosa-14,16,18,20(23),21-pentaen-21-yl]-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide	CC1=CC=C(C(=O)N2CCC(CCCC(=O)N3CCC/C=C/C4=CN=C(N)C5=C4N(N=C5C4=CC=C(C(=O)NC5=NC=CC(C(F)(F)F)=C5)C=C4)[C@@H]4CCC[C@H](C4)NC(=O)C3)CC2)C=C1N1CCC(=O)NC1=O	C53H58F3N11O6	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-7R4MV6	WO2024126617A1_90	.	COC1=CC=C(C(=O)N2CCC(CCCC(=O)N3CCC/C=C/C4=CN=C(N)C5=C4N(N=C5C4=CC=C(C(=O)NC5=NC=CC(C(F)(F)F)=C5)C=C4)[C@@H]4CCC[C@H](C4)NC(=O)C3)CC2)C=C1N1CCC(=O)NC1=O	C53H58F3N11O7	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-2P8H6R	WO2024126617A1_91	4-[(2S,5R,13E)-18-amino-4-[4-[1-[3-(2,4-dioxo-1,3-diazinan-1-yl)-4-methylbenzoyl]piperidin-4-yl]butanoyl]-6-oxo-1,4,7,17,21-pentazatetracyclo[13.6.1.12,5.019,22]tricosa-13,15,17,19(22),20-pentaen-20-yl]-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide	CC1=C(N2CCC(=O)NC2=O)C=C(C(=O)N2CCC(CCCC(=O)N3C[C@@H]4C[C@@H]3C(=O)NCCCCC/C=C/C3=CN=C(N)C5=C3N4N=C5C3=CC=C(C(=O)NC4=CC(C(F)(F)F)=CC=N4)C=C3)CC2)C=C1	C52H56F3N11O6	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-SB7MTE	WO2024126617A1_92	4-[(2S,5R,13E)-18-amino-4-[4-[1-[3-(2,4-dioxo-1,3-diazinan-1-yl)-4-methoxybenzoyl]piperidin-4-yl]butanoyl]-6-oxo-1,4,7,17,21-pentazatetracyclo[13.6.1.12,5.019,22]tricosa-13,15,17,19(22),20-pentaen-20-yl]-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide	COC1=C(N2CCC(=O)NC2=O)C=C(C(=O)N2CCC(CCCC(=O)N3C[C@@H]4C[C@@H]3C(=O)NCCCCC/C=C/C3=CN=C(N)C5=C3N4N=C5C3=CC=C(C(=O)NC4=CC(C(F)(F)F)=CC=N4)C=C3)CC2)C=C1	C52H56F3N11O7	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-AI4ANA	WO2024126617A1_93	.	NC1=NC=C2/C=C/CCCN(CCCCC3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC(=O)N[C@@H]3CCC[C@H](C3)N3N=C(C4=CC=C(C(=O)NC5=NC=CC(C(F)(F)F)=C5)C=C4)C1=C23	C54H58F3N11O6	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-5GUB3V	WO2024126617A1_94	.	NC1=CC=NC(NC(=O)C2=CC=C(C3=NN4C5=C3C(N)=NC=C5/C=C/CCCCCNC(=O)[C@H]3C[C@H]4CN3C(=O)CCCC3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)C=C2)=C1	C52H56N12O7	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-GWS61C	WO2024126617A1_95	.	NC1=NC=C2/C=C/CCCN(C(=O)CCC3CCN(C(=O)COC4=CC=C(C5CCC(=O)NC5=O)C=C4)CC3)CC(=O)N[C@@H]3CCC[C@H](C3)N3N=C(C4=CC=C(C(=O)NC5=NC=CC(C(F)(F)F)=C5)C=C4)C1=C23	C53H57F3N10O7	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-GTXBUT	WO2024126617A1_96	4-[(2R,6R,13E)-18-amino-10-[3-[1-[2-[4-(2,6-dioxopiperidin-3-yl)phenoxy]acetyl]piperidin-4-yl]propanoyl]-8-oxo-1,7,10,17,21-pentazatetracyclo[13.6.1.12,6.019,22]tricosa-13,15,17,19(22),20-pentaen-20-yl]-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide	NC1=NC=C2/C=C/CCN(C(=O)CCC3CCN(C(=O)COC4=CC=C(C5CCC(=O)NC5=O)C=C4)CC3)CC(=O)N[C@@H]3CCC[C@H](C3)N3N=C(C4=CC=C(C(=O)NC5=CC(C(F)(F)F)=CC=N5)C=C4)C1=C23	C52H55F3N10O7	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-WX2B81	WO2024126617A1_97	4-[(2R,6R,13E)-18-amino-10-[3-[1-[[6-[3-(2,6-dioxopiperidin-3-yl)azetidin-1-yl]pyridin-3-yl]methyl]piperidin-4-yl]propanoyl]-8-oxo-1,7,10,17,21-pentazatetracyclo[13.6.1.12,6.019,22]tricosa-13,15,17,19(22),20-pentaen-20-yl]-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide	NC1=NC=C2/C=C/CCN(C(=O)CCC3CCN(CC4=CN=C(N5CC(C6CCC(=O)NC6=O)C5)C=C4)CC3)CC(=O)N[C@@H]3CCC[C@H](C3)N3N=C(C4=CC=C(C(=O)NC5=CC(C(F)(F)F)=CC=N5)C=C4)C1=C23	C53H59F3N12O5	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-E0T6C4	WO2024126617A1_98	4-[(2R,6R,14E)-19-amino-11-[2-[4-[1-[3-(2,4-dioxo-1,3-diazinan-1-yl)-4-methylbenzoyl]piperidin-4-yl]oxypiperidin-1-yl]acetyl]-8-oxo-1,7,11,18,22-pentazatetracyclo[14.6.1.12,6.020,23]tetracosa-14,16,18,20(23),21-pentaen-21-yl]-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide	CC1=C(N2CCC(=O)NC2=O)C=C(C(=O)N2CCC(OC3CCN(CC(=O)N4CC/C=C/C5=CN=C(N)C6=C5N(N=C6C5=CC=C(C(=O)NC6=CC(C(F)(F)F)=CC=N6)C=C5)[C@@H]5CCC[C@H](C5)NC(=O)CC4)CC3)CC2)C=C1	C56H63F3N12O7	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-ESYIJM	WO2024126617A1_99	4-[(2R,6R,14E)-19-amino-11-[2-[4-[1-[3-(2,4-dioxo-1,3-diazinan-1-yl)-4-methoxybenzoyl]piperidin-4-yl]oxypiperidin-1-yl]acetyl]-8-oxo-1,7,11,18,22-pentazatetracyclo[14.6.1.12,6.020,23]tetracosa-14,16,18,20(23),21-pentaen-21-yl]-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide	COC1=C(N2CCC(=O)NC2=O)C=C(C(=O)N2CCC(OC3CCN(CC(=O)N4CC/C=C/C5=CN=C(N)C6=C5N(N=C6C5=CC=C(C(=O)NC6=CC(C(F)(F)F)=CC=N6)C=C5)[C@@H]5CCC[C@H](C5)NC(=O)CC4)CC3)CC2)C=C1	C56H63F3N12O8	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-S8E77F	WO2024126617A1_100	4-[(2R,6R,14E)-19-amino-11-[2-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]oxypiperidin-1-yl]acetyl]-8-oxo-1,7,11,18,22-pentazatetracyclo[14.6.1.12,6.020,23]tetracosa-14,16,18,20(23),21-pentaen-21-yl]-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide	NC1=NC=C2/C=C/CCN(C(=O)CN3CCC(OC4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)CCC(=O)N[C@@H]3CCC[C@H](C3)N3N=C(C4=CC=C(C(=O)NC5=CC(C(F)(F)F)=CC=N5)C=C4)C1=C23	C57H61F3N12O8	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-CIFICV	WO2024126617A1_101	N-[2-[3-[(2R,6R,13E)-18-amino-8-oxo-20-[4-[[4-(trifluoromethyl)pyridin-2-yl]carbamoyl]phenyl]-1,7,10,17,21-pentazatetracyclo[13.6.1.12,6.019,22]tricosa-13,15,17,19(22),20-pentaen-10-yl]-3-oxopropoxy]ethyl]-6-(2,4-dioxo-1,3,8-triazaspiro[4.5]decan-8-yl)pyridine-3-carboxamide	NC1=NC=C2/C=C/CCN(C(=O)CCOCCNC(=O)C3=CN=C(N4CCC5(CC4)NC(=O)NC5=O)C=C3)CC(=O)N[C@@H]3CCC[C@H](C3)N3N=C(C4=CC=C(C(=O)NC5=CC(C(F)(F)F)=CC=N5)C=C4)C1=C23	C49H52F3N13O7	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-DVYYV2	WO2024126617A1_102	4-[(2R,6R,13E)-18-amino-10-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]oxyacetyl]-8-oxo-1,7,10,17,21-pentazatetracyclo[13.6.1.12,6.019,22]tricosa-13,15,17,19(22),20-pentaen-20-yl]-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide	NC1=NC=C2/C=C/CCN(C(=O)COC3CN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)C3)CC(=O)N[C@@H]3CCC[C@H](C3)N3N=C(C4=CC=C(C(=O)NC5=CC(C(F)(F)F)=CC=N5)C=C4)C1=C23	C49H46F3N11O8	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-E8N24M	WO2024126617A1_103	.	C=C1NC(=O)NC12CCN(C1=CC=C(C(=O)N3CCN(CCC(=O)N4CC/C=C/C5=CN=C(N)C6=C5N(N=C6C5=CC=C(C(=O)NC6=CC(C(F)(F)F)=CC=N6)C=C5)[C@@H]5CCC[C@H](C5)NC(=O)C4)CC3)C=N1)CC2	C52H57F3N14O5	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-41YII2	WO2024126617A1_104	.	CN[C@@H](C)C(=O)N[C@H](C(=O)N1CC2=C(C=CC(OCCOCCOCC(=O)N3CC/C=C/C4=CN=C(N)C5=C4N(N=C5C4=CC=C(C(=O)NC5=CC(C(F)(F)F)=CC=N5)C=C4)[C@@H]4CCC[C@H](C4)NC(=O)C3)=C2)C[C@H]1C(=O)N[C@@H]1CCCC2=C1C=CC=C2)C(C)(C)C	C67H79F3N12O9	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-G3SFDS	WO2024126617A1_105	3-[4-[4-[[(2R,6R,14E)-19-amino-8-oxo-21-quinolin-3-yl-7,11,18,22,23-pentazatetracyclo[14.6.1.12,6.020,23]tetracosa-1(22),14,16,18,20-pentaen-11-yl]methyl]piperidin-1-yl]-3-fluorophenyl]piperidine-2,6-dione	NC1=NC=C2/C=C/CCN(CC3CCN(C4=CC=C(C5CCC(=O)NC5=O)C=C4F)CC3)CCC(=O)N[C@@H]3CCC[C@H](C3)C3=NC(C4=CN=C5C=CC=CC5=C4)=C1N23	C45H50FN9O3	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-NLRMQ2	WO2024126617A1_106	.	NC1=NC=C2/C=C/CCCCCNC(=O)[C@H]3C[C@@H](CN3CC3CCN(C4=CC=C(C5CCC(=O)NC5=O)C=C4F)CC3)N3N=C(C4=CC=C(C(=O)NC5=CC(C(F)(F)F)=CC=N5)C=C4)C1=C23	C48H50F4N10O4	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-TYZQFN	WO2024126617A1_107	4-[(2S,5R,13E)-18-amino-4-[3-[4-[4-(2,6-dioxopiperidin-3-yl)-2-fluorophenyl]piperazin-1-yl]propanoyl]-6-oxo-1,4,7,17,21-pentazatetracyclo[13.6.1.12,5.019,22]tricosa-13,15,17,19(22),20-pentaen-20-yl]-N-[4-(trifluoromethyl)pyridin-2-yl]benzamide	NC1=NC=C2/C=C/CCCCCNC(=O)[C@H]3C[C@@H](CN3C(=O)CCN3CCN(C4=CC=C(C5CCC(=O)NC5=O)C=C4F)CC3)N3N=C(C4=CC=C(C(=O)NC5=CC(C(F)(F)F)=CC=N5)C=C4)C1=C23	C49H51F4N11O5	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-8ZJ27C	WO2024126617A1_108	N-[2-[3-[(2R,6R,13E)-18-amino-20-[4-[2-[(5-tert-butyl-1,2-oxazol-3-yl)amino]-2-oxoethyl]phenyl]-8-oxo-7,10,17,21,22-pentazatetracyclo[13.6.1.12,6.019,22]tricosa-1(21),13,15,17,19-pentaen-10-yl]-3-oxopropoxy]ethyl]-3-(2,4-dioxo-1,3-diazinan-1-yl)-4-methoxybenzamide	COC1=C(N2CCC(=O)NC2=O)C=C(C(=O)NCCOCCC(=O)N2CC/C=C/C3=CN=C(N)C4=C(C5=CC=C(CC(=O)NC6=NOC(C(C)(C)C)=C6)C=C5)N=C([C@@H]5CCC[C@H](C5)NC(=O)C2)N34)C=C1	C50H59N11O9	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-08WSXE	WO2024126617A1_109	2-[4-[(2R,6R,13E)-18-amino-10-[3-[4-[3-(2,4-dioxo-1,3-diazinan-1-yl)-4-methoxybenzoyl]piperazin-1-yl]propanoyl]-8-oxo-7,10,17,21,22-pentazatetracyclo[13.6.1.12,6.019,22]tricosa-1(21),13,15,17,19-pentaen-20-yl]phenyl]-N-(5-tert-butyl-1,2-oxazol-3-yl)acetamide	COC1=C(N2CCC(=O)NC2=O)C=C(C(=O)N2CCN(CCC(=O)N3CC/C=C/C4=CN=C(N)C5=C(C6=CC=C(CC(=O)NC7=NOC(C(C)(C)C)=C7)C=C6)N=C([C@@H]6CCC[C@H](C6)NC(=O)C3)N45)CC2)C=C1	C52H62N12O8	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-022WI4	WO2024126617A1_110	2-[4-[(2R,6R,13E)-18-amino-10-[2-[1-[[6-[3-(2,4-dioxo-1,3-diazinan-1-yl)azetidin-1-yl]pyridin-3-yl]methyl]piperidin-4-yl]acetyl]-8-oxo-7,10,17,21,22-pentazatetracyclo[13.6.1.12,6.019,22]tricosa-1(21),13,15,17,19-pentaen-20-yl]phenyl]-N-(5-tert-butyl-1,2-oxazol-3-yl)acetamide	CC(C)(C)C1=CC(NC(=O)CC2=CC=C(C3=C4C(N)=NC=C5/C=C/CCN(C(=O)CC6CCN(CC7=CN=C(N8CC(N9CCC(=O)NC9=O)C8)C=C7)CC6)CC(=O)N[C@@H]6CCC[C@H](C6)C(=N3)N54)C=C2)=NO1	C53H65N13O6	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-RSHO7A	WO2024126617A1_111	2-[4-[(2R,6R,13E)-18-amino-10-[[1-[4-(2,6-dioxopiperidin-3-yl)-3-fluorophenyl]piperidin-4-yl]methyl]-8-oxo-7,10,17,21,22-pentazatetracyclo[13.6.1.12,6.019,22]tricosa-1(21),13,15,17,19-pentaen-20-yl]phenyl]-N-(5-tert-butyl-1,2-oxazol-3-yl)acetamide	CC(C)(C)C1=CC(NC(=O)CC2=CC=C(C3=C4C(N)=NC=C5/C=C/CCN(CC6CCN(C7=CC=C(C8CCC(=O)NC8=O)C(F)=C7)CC6)CC(=O)N[C@@H]6CCC[C@H](C6)C(=N3)N54)C=C2)=NO1	C50H59FN10O5	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-RL1SVY	WO2024126617A1_112	N-[2-[3-[(2R,6R,14E)-19-amino-21-[4-[2-[(5-tert-butyl-1,2-oxazol-3-yl)amino]-2-oxoethyl]phenyl]-8-oxo-7,10,18,22,23-pentazatetracyclo[14.6.1.12,6.020,23]tetracosa-1(22),14,16,18,20-pentaen-10-yl]-3-oxopropoxy]ethyl]-3-(2,4-dioxo-1,3-diazinan-1-yl)-4-methoxybenzamide	COC1=C(N2CCC(=O)NC2=O)C=C(C(=O)NCCOCCC(=O)N2CCC/C=C/C3=CN=C(N)C4=C(C5=CC=C(CC(=O)NC6=NOC(C(C)(C)C)=C6)C=C5)N=C([C@@H]5CCC[C@H](C5)NC(=O)C2)N34)C=C1	C51H61N11O9	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-J30B5O	WO2024126617A1_113	.	CC(C)C1=CC(NC(=O)CC2=CC=C(C3=C4C(N)=NC=C5/C=C/CCN(C[C@@H]6CCN(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8=O)C6)CCC(=O)N[C@@H]6CCC[C@H](C6)C(=N3)N54)C=C2)=NO1	C51H57N11O7	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-M0XWWQ	WO2024126617A1_114	2-[4-[(2R,6R,14E)-19-amino-11-[2-[4-(2,6-dioxopiperidin-3-yl)phenoxy]acetyl]-8-oxo-7,11,18,22,23-pentazatetracyclo[14.6.1.12,6.020,23]tetracosa-1(22),14,16,18,20-pentaen-21-yl]phenyl]-N-(5-tert-butyl-1,2-oxazol-3-yl)acetamide	CC(C)(C)C1=CC(NC(=O)CC2=CC=C(C3=C4C(N)=NC=C5/C=C/CCN(C(=O)COC6=CC=C(C7CCC(=O)NC7=O)C=C6)CCC(=O)N[C@@H]6CCC[C@H](C6)C(=N3)N54)C=C2)=NO1	C47H53N9O7	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-3PJV8L	WO2024126617A1_115	.	CC(C)C1=CC(NC(=O)CC2=CC=C(C3=C4C(N)=NC=C5/C=C/CCN(CC6CN(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8=O)C6)CCC(=O)N[C@@H]6CCC[C@H](C6)C(=N3)N54)C=C2)=NO1	C50H55N11O7	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-IPRPPR	WO2024126617A1_116	2-[4-[(2R,6R,14E)-19-amino-11-[[1-[4-(2,6-dioxopiperidin-3-yl)-2-fluorophenyl]piperidin-4-yl]methyl]-8-oxo-7,11,18,22,23-pentazatetracyclo[14.6.1.12,6.020,23]tetracosa-1(22),14,16,18,20-pentaen-21-yl]phenyl]-N-(5-tert-butyl-1,2-oxazol-3-yl)acetamide	CC(C)(C)C1=CC(NC(=O)CC2=CC=C(C3=C4C(N)=NC=C5/C=C/CCN(CC6CCN(C7=C(F)C=C(C8CCC(=O)NC8=O)C=C7)CC6)CCC(=O)N[C@@H]6CCC[C@H](C6)C(=N3)N54)C=C2)=NO1	C51H61FN10O5	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-NAWPAD	WO2024126617A1_117	2-[4-[(2R,6R,14E)-19-amino-11-[1-[4-(2,6-dioxopiperidin-3-yl)-2-fluorophenyl]piperidine-4-carbonyl]-8-oxo-7,11,18,22,23-pentazatetracyclo[14.6.1.12,6.020,23]tetracosa-1(22),14,16,18,20-pentaen-21-yl]phenyl]-N-(5-tert-butyl-1,2-oxazol-3-yl)acetamide	CC(C)(C)C1=CC(NC(=O)CC2=CC=C(C3=C4C(N)=NC=C5/C=C/CCN(C(=O)C6CCN(C7=C(F)C=C(C8CCC(=O)NC8=O)C=C7)CC6)CCC(=O)N[C@@H]6CCC[C@H](C6)C(=N3)N54)C=C2)=NO1	C51H59FN10O6	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-664FTI	WO2024126617A1_118	N-[2-[3-[(2R,6R,14E)-19-amino-21-[4-[2-[(5-tert-butyl-1,2-oxazol-3-yl)amino]-2-oxoethyl]phenyl]-8-oxo-7,11,18,22,23-pentazatetracyclo[14.6.1.12,6.020,23]tetracosa-1(22),14,16,18,20-pentaen-11-yl]-3-oxopropoxy]ethyl]-3-(2,4-dioxo-1,3-diazinan-1-yl)-4-methoxybenzamide	COC1=CC=C(C(=O)NCCOCCC(=O)N2CC/C=C/C3=CN=C(N)C4=C(C5=CC=C(CC(=O)NC6=NOC(C(C)(C)C)=C6)C=C5)N=C([C@@H]5CCC[C@H](C5)NC(=O)CC2)N34)C=C1N1CCC(=O)NC1=O	C51H61N11O9	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-VU3Z85	WO2024126617A1_119	2-[4-[(2R,6R,14E)-19-amino-11-[3-[4-[3-(2,4-dioxo-1,3-diazinan-1-yl)-4-methoxybenzoyl]piperazin-1-yl]propanoyl]-8-oxo-7,11,18,22,23-pentazatetracyclo[14.6.1.12,6.020,23]tetracosa-1(22),14,16,18,20-pentaen-21-yl]phenyl]-N-(5-tert-butyl-1,2-oxazol-3-yl)acetamide	COC1=C(N2CCC(=O)NC2=O)C=C(C(=O)N2CCN(CCC(=O)N3CC/C=C/C4=CN=C(N)C5=C(C6=CC=C(CC(=O)NC7=NOC(C(C)(C)C)=C7)C=C6)N=C([C@@H]6CCC[C@H](C6)NC(=O)CC3)N45)CC2)C=C1	C53H64N12O8	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-8Y5AOV	WO2024126617A1_120	2-[4-[(2R,6R,14E)-19-amino-10-[3-[4-[3-(2,4-dioxo-1,3-diazinan-1-yl)-4-methoxybenzoyl]piperazin-1-yl]propanoyl]-8-oxo-7,10,18,22,23-pentazatetracyclo[14.6.1.12,6.020,23]tetracosa-1(22),14,16,18,20-pentaen-21-yl]phenyl]-N-(5-tert-butyl-1,2-oxazol-3-yl)acetamide	COC1=C(N2CCC(=O)NC2=O)C=C(C(=O)N2CCN(CCC(=O)N3CCC/C=C/C4=CN=C(N)C5=C(C6=CC=C(CC(=O)NC7=NOC(C(C)(C)C)=C7)C=C6)N=C([C@@H]6CCC[C@H](C6)NC(=O)C3)N45)CC2)C=C1	C53H64N12O8	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-6XAO3G	WO2024126617A1_121	2-[4-[(2R,6R,13E)-18-amino-10-[[(3S)-1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]pyrrolidin-3-yl]methyl]-8-oxo-7,10,17,21,22-pentazatetracyclo[13.6.1.12,6.019,22]tricosa-1(21),13,15,17,19-pentaen-20-yl]phenyl]-N-(5-tert-butyl-1,2-oxazol-3-yl)acetamide	CC(C)(C)C1=CC(NC(=O)CC2=CC=C(C3=C4C(N)=NC=C5/C=C/CCN(C[C@@H]6CCN(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8=O)C6)CC(=O)N[C@@H]6CCC[C@H](C6)C(=N3)N54)C=C2)=NO1	C51H57N11O7	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-BJC1WT	WO2024126617A1_122	2-[4-[(2R,6R,14E)-19-amino-10-[[1-[4-(2,6-dioxopiperidin-3-yl)-2-fluorophenyl]piperidin-4-yl]methyl]-8-oxo-7,10,18,22,23-pentazatetracyclo[14.6.1.12,6.020,23]tetracosa-1(22),14,16,18,20-pentaen-21-yl]phenyl]-N-(5-tert-butyl-1,2-oxazol-3-yl)acetamide	CC(C)(C)C1=CC(NC(=O)CC2=CC=C(C3=C4C(N)=NC=C5/C=C/CCCN(CC6CCN(C7=C(F)C=C(C8CCC(=O)NC8=O)C=C7)CC6)CC(=O)N[C@@H]6CCC[C@H](C6)C(=N3)N54)C=C2)=NO1	C51H61FN10O5	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-A2HTSB	WO2024126617A1_123	2-[4-[(2R,6R,13E)-18-amino-10-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]methyl]-8-oxo-7,10,17,21,22-pentazatetracyclo[13.6.1.12,6.019,22]tricosa-1(21),13,15,17,19-pentaen-20-yl]phenyl]-N-(5-tert-butyl-1,2-oxazol-3-yl)acetamide	CC(C)(C)C1=CC(NC(=O)CC2=CC=C(C3=C4C(N)=NC=C5/C=C/CCN(CC6CN(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8=O)C6)CC(=O)N[C@@H]6CCC[C@H](C6)C(=N3)N54)C=C2)=NO1	C50H55N11O7	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-CH9BQX	WO2024126617A1_124	2-[4-[(2R,6R,14E)-19-amino-10-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]methyl]-8-oxo-7,10,18,22,23-pentazatetracyclo[14.6.1.12,6.020,23]tetracosa-1(22),14,16,18,20-pentaen-21-yl]phenyl]-N-(5-tert-butyl-1,2-oxazol-3-yl)acetamide	CC(C)(C)C1=CC(NC(=O)CC2=CC=C(C3=C4C(N)=NC=C5/C=C/CCCN(CC6CN(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8=O)C6)CC(=O)N[C@@H]6CCC[C@H](C6)C(=N3)N54)C=C2)=NO1	C51H57N11O7	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-S0DPLP	WO2024126617A1_125	.	CC(C)(C)C1=CC(NC(=O)CC2=CC=C(C3=C4C(N)=NC=C5/C=C/CCN(C(=O)CCC6CCN(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CCC(=O)N[C@@H]6CCC[C@H](C6)C(=N3)N54)C=C2)=NO1	C55H63N11O8	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-UJPS9J	WO2024126617A1_126	2-[4-[(2R,6R,13E)-18-amino-10-[3-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]propanoyl]-8-oxo-7,10,17,21,22-pentazatetracyclo[13.6.1.12,6.019,22]tricosa-1(21),13,15,17,19-pentaen-20-yl]phenyl]-N-(5-tert-butyl-1,2-oxazol-3-yl)acetamide	CC(C)(C)C1=CC(NC(=O)CC2=CC=C(C3=C4C(N)=NC=C5/C=C/CCN(C(=O)CCC6CCN(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC(=O)N[C@@H]6CCC[C@H](C6)C(=N3)N54)C=C2)=NO1	C54H61N11O8	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-MJKCGX	WO2024126617A1_127	2-[4-[(2R,6R,14E)-19-amino-10-[3-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]propanoyl]-8-oxo-7,10,18,22,23-pentazatetracyclo[14.6.1.12,6.020,23]tetracosa-1(22),14,16,18,20-pentaen-21-yl]phenyl]-N-(5-tert-butyl-1,2-oxazol-3-yl)acetamide	CC(C)(C)C1=CC(NC(=O)CC2=CC=C(C3=C4C(N)=NC=C5/C=C/CCCN(C(=O)CCC6CCN(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC(=O)N[C@@H]6CCC[C@H](C6)C(=N3)N54)C=C2)=NO1	C55H63N11O8	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-O698QZ	WO2024126617A1_128	2-[4-[(2R,6R,13E)-18-amino-10-[2-[4-(2,6-dioxopiperidin-3-yl)phenoxy]acetyl]-8-oxo-7,10,17,21,22-pentazatetracyclo[13.6.1.12,6.019,22]tricosa-1(21),13,15,17,19-pentaen-20-yl]phenyl]-N-(5-tert-butyl-1,2-oxazol-3-yl)acetamide	CC(C)(C)C1=CC(NC(=O)CC2=CC=C(C3=C4C(N)=NC=C5/C=C/CCN(C(=O)COC6=CC=C(C7CCC(=O)NC7=O)C=C6)CC(=O)N[C@@H]6CCC[C@H](C6)C(=N3)N54)C=C2)=NO1	C46H51N9O7	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-MF6FMD	WO2024126617A1_129	2-[4-[(2R,6R,14E)-19-amino-10-[2-[4-(2,6-dioxopiperidin-3-yl)phenoxy]acetyl]-8-oxo-7,10,18,22,23-pentazatetracyclo[14.6.1.12,6.020,23]tetracosa-1(22),14,16,18,20-pentaen-21-yl]phenyl]-N-(5-tert-butyl-1,2-oxazol-3-yl)acetamide	CC(C)(C)C1=CC(NC(=O)CC2=CC=C(C3=C4C(N)=NC=C5/C=C/CCCN(C(=O)COC6=CC=C(C7CCC(=O)NC7=O)C=C6)CC(=O)N[C@@H]6CCC[C@H](C6)C(=N3)N54)C=C2)=NO1	C47H53N9O7	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-28RDUO	WO2024126617A1_130	2-[4-[(2R,6R,14E)-19-amino-11-[[(3R)-1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]pyrrolidin-3-yl]methyl]-8-oxo-7,11,18,22,23-pentazatetracyclo[14.6.1.12,6.020,23]tetracosa-1(22),14,16,18,20-pentaen-21-yl]phenyl]-N-(5-tert-butyl-1,2-oxazol-3-yl)acetamide	CC(C)(C)C1=CC(NC(=O)CC2=CC=C(C3=C4C(N)=NC=C5/C=C/CCN(C[C@H]6CCN(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8=O)C6)CCC(=O)N[C@@H]6CCC[C@H](C6)C(=N3)N54)C=C2)=NO1	C52H59N11O7	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-P21ZWF	WO2024126617A1_131	2-[4-[(2R,6R,14E)-19-amino-10-[[(3S)-1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]pyrrolidin-3-yl]methyl]-8-oxo-7,10,18,22,23-pentazatetracyclo[14.6.1.12,6.020,23]tetracosa-1(22),14,16,18,20-pentaen-21-yl]phenyl]-N-(5-tert-butyl-1,2-oxazol-3-yl)acetamide	CC(C)(C)C1=CC(NC(=O)CC2=CC=C(C3=C4C(N)=NC=C5/C=C/CCCN(C[C@@H]6CCN(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8=O)C6)CC(=O)N[C@@H]6CCC[C@H](C6)C(=N3)N54)C=C2)=NO1	C52H59N11O7	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-TUFNEC	WO2024126617A1_132	2-[4-[(2R,6R,13E)-18-amino-10-[[(3R)-1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]pyrrolidin-3-yl]methyl]-8-oxo-7,10,17,21,22-pentazatetracyclo[13.6.1.12,6.019,22]tricosa-1(21),13,15,17,19-pentaen-20-yl]phenyl]-N-(5-tert-butyl-1,2-oxazol-3-yl)acetamide	CC(C)(C)C1=CC(NC(=O)CC2=CC=C(C3=C4C(N)=NC=C5/C=C/CCN(C[C@H]6CCN(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8=O)C6)CC(=O)N[C@@H]6CCC[C@H](C6)C(=N3)N54)C=C2)=NO1	C51H57N11O7	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-0ITCWV	WO2024126617A1_133	.	CC(C)(C)C1=CC(NC(=O)CC2=CC=C(C3=C4C(N)=NC=C5/C=C/CCCN(CC6CCN(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8=O)C6)CC(=O)N[C@@H]6CCC[C@H](C6)C(=N3)N54)C=C2)=NO1	C52H59N11O7	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-X0603H	WO2024126617A1_134	5-[4-[[(2R,6R,14E)-19-amino-21-[4-[2-[(5-tert-butyl-1,2-oxazol-3-yl)amino]-2-oxoethyl]phenyl]-8-oxo-7,11,18,22,23-pentazatetracyclo[14.6.1.12,6.020,23]tetracosa-1(22),14,16,18,20-pentaen-11-yl]methyl]piperidin-1-yl]-N-(2,6-dioxopiperidin-3-yl)pyridine-2-carboxamide	CC(C)(C)C1=CC(NC(=O)CC2=CC=C(C3=C4C(N)=NC=C5/C=C/CCN(CC6CCN(C7=CN=C(C(=O)NC8CCC(=O)NC8=O)C=C7)CC6)CCC(=O)N[C@@H]6CCC[C@H](C6)C(=N3)N54)C=C2)=NO1	C51H62N12O6	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-ZJBYTM	WO2024126617A1_135	5-[4-[[(2R,6R,13E)-18-amino-20-[4-[2-[(5-tert-butyl-1,2-oxazol-3-yl)amino]-2-oxoethyl]phenyl]-8-oxo-7,10,17,21,22-pentazatetracyclo[13.6.1.12,6.019,22]tricosa-1(21),13,15,17,19-pentaen-10-yl]methyl]piperidin-1-yl]-N-(2,6-dioxopiperidin-3-yl)pyridine-2-carboxamide	CC(C)(C)C1=CC(NC(=O)CC2=CC=C(C3=C4C(N)=NC=C5/C=C/CCN(CC6CCN(C7=CN=C(C(=O)NC8CCC(=O)NC8=O)C=C7)CC6)CC(=O)N[C@@H]6CCC[C@H](C6)C(=N3)N54)C=C2)=NO1	C50H60N12O6	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-NO6OYV	WO2024126617A1_136	5-[4-[[(2R,6R,14E)-19-amino-21-[4-[2-[(5-tert-butyl-1,2-oxazol-3-yl)amino]-2-oxoethyl]phenyl]-8-oxo-7,10,18,22,23-pentazatetracyclo[14.6.1.12,6.020,23]tetracosa-1(22),14,16,18,20-pentaen-10-yl]methyl]piperidin-1-yl]-N-(2,6-dioxopiperidin-3-yl)pyridine-2-carboxamide	CC(C)(C)C1=CC(NC(=O)CC2=CC=C(C3=C4C(N)=NC=C5/C=C/CCCN(CC6CCN(C7=CN=C(C(=O)NC8CCC(=O)NC8=O)C=C7)CC6)CC(=O)N[C@@H]6CCC[C@H](C6)C(=N3)N54)C=C2)=NO1	C51H62N12O6	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-ZIROW7	WO2024126617A1_137	5-[3-[[(2R,6R,13E)-18-amino-8-oxo-20-quinolin-3-yl-7,10,17,21,22-pentazatetracyclo[13.6.1.12,6.019,22]tricosa-1(21),13,15,17,19-pentaen-10-yl]methyl]azetidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	NC1=NC=C2/C=C/CCN(CC3CN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)CC(=O)N[C@@H]3CCC[C@H](C3)C3=NC(C4=CN=C5C=CC=CC5=C4)=C1N23	C44H44N10O5	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-162183	WO2024126617A1_138	5-[(3R)-3-[[(2R,6R,14E)-19-amino-8-oxo-21-quinolin-3-yl-7,11,18,22,23-pentazatetracyclo[14.6.1.12,6.020,23]tetracosa-1(22),14,16,18,20-pentaen-11-yl]methyl]pyrrolidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	NC1=NC=C2/C=C/CCN(C[C@H]3CCN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)CCC(=O)N[C@@H]3CCC[C@H](C3)C3=NC(C4=CN=C5C=CC=CC5=C4)=C1N23	C46H48N10O5	BTK	Q06187	CRBN	WO-2024126617-A1
TPD-EJIKS5	WO2024127022A1_056	.	CN1C(=O)C2=C(N=C(N3CCC(CCN4CCN(C5=CC6=C(C=C5F)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)N2CC2=NN=C(C3=CC=C(Cl)C(Cl)=C3)O2)N(C)C1=O	C40H40Cl2FN11O7	NUDT5	Q9UKK9	CRBN	WO-2024127022-A1
TPD-F7ACB6	WO2024127022A1_057	.	CN1C(=O)C2=C(N=C(N3CCN(C(=O)CCCCNC(=O)COC4=CC=CC5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)N2CC2=NN=C(C3=CC=C(Cl)C(Cl)=C3)O2)N(C)C1=O	C40H39Cl2N11O10	NUDT5	Q9UKK9	CRBN	WO-2024127022-A1
TPD-IQ5VVC	WO2024127022A1_063	.	CN1C(=O)C2=C(N=C(N3CCC(CN4CCN(C5=CC6=C(C=C5F)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)N2CC2=NN=C(C3=CC=C(Cl)C(Cl)=C3)O2)N(C)C1=O	C39H38Cl2FN11O7	NUDT5	Q9UKK9	CRBN	WO-2024127022-A1
TPD-53E9GC	SCHEMBL27466138	7-[[5-(3,4-Dichlorophenyl)-1,3,4-oxadiazol-2-yl]methyl]-8-[4-[3-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]propanoyl]piperazin-1-yl]-1,3-dimethylpurine-2,6-dione; SCHEMBL30962348	CN1C(=O)C2=C(N=C(N3CCN(C(=O)CCOCCOCCNC4=CC=CC5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)N2CC2=NN=C(C3=CC=C(Cl)C(Cl)=C3)O2)N(C)C1=O	C40H41Cl2N11O10	NUDT5	Q9UKK9	CRBN	WO-2024127022-A1
TPD-UXUDDH	SCHEMBL27466677	7-[[5-(3,4-Dichlorophenyl)-1,3,4-oxadiazol-2-yl]methyl]-8-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]-1,3-dimethylpurine-2,6-dione	CN1C(=O)C2=C(N=C(N3CCN(CC4CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)N2CC2=NN=C(C3=CC=C(Cl)C(Cl)=C3)O2)N(C)C1=O	C39H39Cl2N11O7	NUDT5	Q9UKK9	CRBN	WO-2024127022-A1
TPD-AWVQII	WO2024127022A1_071	.	CN1C(=O)C2=C(N=C(N3CCN(CC4CCN(C5=CC6=C(C=C5F)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)N2CC2=NN=C(C3=CC=C(Cl)C(Cl)=C3)O2)N(C)C1=O	C39H38Cl2FN11O7	NUDT5	Q9UKK9	CRBN	WO-2024127022-A1
TPD-0AZVQ6	WO2024127022A1_076	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCCCCCC(=O)N3CCN(C4=NC5=C(C(=O)N(C)C(=O)N5C)N4CC4=NN=C(C5=CC=C(Cl)C(Cl)=C5)O4)CC3)C(C)(C)C)C=C2)SC=N1	C53H66Cl2N12O10S	NUDT5	Q9UKK9	VHL	WO-2024127022-A1
TPD-79FDC4	WO2024127022A1_084	.	CN1C(=O)NC2=C(C1=O)N(CC1=NN=C(C3=CC=C(Cl)C(Cl)=C3)O1)C(N1CCN(OCCCCCCNC3=CC=CC4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC1)=N2	C38H39Cl2N11O8	NUDT5	Q9UKK9	CRBN	WO-2024127022-A1
TPD-ILAPM8	SCHEMBL27466646	7-[[5-(3,4-Dichlorophenyl)-1,3,4-oxadiazol-2-yl]methyl]-8-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]ethyl]piperazin-1-yl]-1,3-dimethylpurine-2,6-dione	CN1C(=O)C2=C(N=C(N3CCN(CCC4CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)N2CC2=NN=C(C3=CC=C(Cl)C(Cl)=C3)O2)N(C)C1=O	C40H41Cl2N11O7	NUDT5	Q9UKK9	CRBN	WO-2024127022-A1
TPD-4F30PR	WO2024127022A1_105	.	CN1C(=O)C2=C(N=C(N3CCN(CC4CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)CC3)N2CC2=NN=C(C3=CC=C(Cl)C(Cl)=C3)O2)N(C)C1=O	C38H37Cl2N11O7	NUDT5	Q9UKK9	CRBN	WO-2024127022-A1
TPD-YLX48B	WO2024127022A1_110	.	CN1C(=O)C2=C(N=C(N3CCN(CC4CCN(C5=CC=CC6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)N2CC2=NN=C(C3=CC=C(Cl)C(Cl)=C3)O2)N(C)C1=O	C39H39Cl2N11O7	NUDT5	Q9UKK9	CRBN	WO-2024127022-A1
TPD-94FVN1	WO2024127022A1_111	.	CN1C(=O)C2=C(N=C(N3CCN(C(=O)CCCNC4=CC=CC5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)N2CC2=NN=C(C3=CC=C(Cl)C(Cl)=C3)O2)N(C)C1=O	C37H35Cl2N11O8	NUDT5	Q9UKK9	CRBN	WO-2024127022-A1
TPD-JP8MDJ	WO2024127022A1_122	.	CN1C(=O)C2=C(N=C(N3CCN(C(=O)CCCCCNC4=CC=CC5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)N2CC2=NN=C(C3=CC=C(Cl)C(Cl)=C3)O2)N(C)C1=O	C39H39Cl2N11O8	NUDT5	Q9UKK9	CRBN	WO-2024127022-A1
TPD-XWBHYJ	WO2024127022A1_124	.	CN1C(=O)C2=C(N=C(N3CCN(C(=O)CCCCNC4=CC=CC5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)N2CC2=NN=C(C3=CC=C(Cl)C(Cl)=C3)O2)N(C)C1=O	C38H37Cl2N11O8	NUDT5	Q9UKK9	CRBN	WO-2024127022-A1
TPD-CQYQ3I	SCHEMBL27466129	7-[[5-(3,4-Dichlorophenyl)-1,3,4-oxadiazol-2-yl]methyl]-8-[4-[3-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]propanoyl]piperazin-1-yl]-1,3-dimethylpurine-2,6-dione; SCHEMBL30962344	CN1C(=O)C2=C(N=C(N3CCN(C(=O)CCOCCOCCOCCNC4=CC=CC5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)N2CC2=NN=C(C3=CC=C(Cl)C(Cl)=C3)O2)N(C)C1=O	C42H45Cl2N11O11	NUDT5	Q9UKK9	CRBN	WO-2024127022-A1
TPD-UATD3B	SCHEMBL27466626	7-[[5-(3,4-Dichlorophenyl)-1,3,4-oxadiazol-2-yl]methyl]-8-[4-[3-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethoxy]propanoyl]piperazin-1-yl]-1,3-dimethylpurine-2,6-dione; SCHEMBL30962349	CN1C(=O)C2=C(N=C(N3CCN(C(=O)CCOCCOCCOCCOCCNC4=CC=CC5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)N2CC2=NN=C(C3=CC=C(Cl)C(Cl)=C3)O2)N(C)C1=O	C44H49Cl2N11O12	NUDT5	Q9UKK9	CRBN	WO-2024127022-A1
TPD-W7KB66	WO2024127022A1_131	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)OCCOCCOCCC(=O)N3CCN(C4=NC5=C(C(=O)N(C)C(=O)N5C)N4CC4=NN=C(C5=CC=C(Cl)C(Cl)=C5)O4)CC3)C(C)(C)C)C=C2)SC=N1	C50H60Cl2N12O11S	NUDT5	Q9UKK9	VHL	WO-2024127022-A1
TPD-0UJOP7	WO2024127022A1_133	.	CN1C(=O)C2=C(N=C(N3CCN(C(=O)CCCCCCCCNC4=CC=CC5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)N2CC2=NN=C(C3=CC=C(Cl)C(Cl)=C3)O2)N(C)C1=O	C42H45Cl2N11O8	NUDT5	Q9UKK9	CRBN	WO-2024127022-A1
TPD-J4LCJS	WO2024127022A1_134	.	CN1C(=O)C2=C(N=C(N3CCN(C(=O)CCCCCCCNC4=CC=CC5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)N2CC2=NN=C(C3=CC=C(Cl)C(Cl)=C3)O2)N(C)C1=O	C41H43Cl2N11O8	NUDT5	Q9UKK9	CRBN	WO-2024127022-A1
TPD-OTQZX5	WO2024127022A1_135	.	CN1C(=O)C2=C(N=C(N3CCN(C(=O)CCCCCCCCOC4=CC=CC5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)N2CC2=NN=C(C3=CC=C(Cl)C(Cl)=C3)O2)N(C)C1=O	C42H44Cl2N10O9	NUDT5	Q9UKK9	CRBN	WO-2024127022-A1
TPD-2TB6XI	WO2024127022A1_136	.	CN1C(=O)C2=C(N=C(N3CCN(C(=O)CCCCCCOC4=CC=CC5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)N2CC2=NN=C(C3=CC=C(Cl)C(Cl)=C3)O2)N(C)C1=O	C40H40Cl2N10O9	NUDT5	Q9UKK9	CRBN	WO-2024127022-A1
TPD-CXQXMU	WO2024127022A1_137	.	CN1C(=O)C2=C(N=C(N3CCN(C(=O)CCOCCNC4=CC=CC5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)N2CC2=NN=C(C3=CC=C(Cl)C(Cl)=C3)O2)N(C)C1=O	C38H37Cl2N11O9	NUDT5	Q9UKK9	CRBN	WO-2024127022-A1
TPD-37G2A9	WO2024127022A1_159	.	CN1C(=O)C2=C(N=C(N3CCN(C(=O)NCCOCCOCCNC4=CC=CC5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)N2CC2=NN=C(C3=CC=C(Cl)C(Cl)=C3)O2)N(C)C1=O	C40H42Cl2N12O10	NUDT5	Q9UKK9	CRBN	WO-2024127022-A1
TPD-P78A74	SCHEMBL27466103	7-[[5-(3,4-Dichlorophenyl)-1,3,4-oxadiazol-2-yl]methyl]-8-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidine-1-carbonyl]piperazin-1-yl]-1,3-dimethylpurine-2,6-dione	CN1C(=O)C2=C(N=C(N3CCN(C(=O)N4CCC(CN5CCN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)CC3)N2CC2=NN=C(C3=CC=C(Cl)C(Cl)=C3)O2)N(C)C1=O	C44H47Cl2N13O8	NUDT5	Q9UKK9	CRBN	WO-2024127022-A1
TPD-VA5LO2	SCHEMBL27466528	7-[[5-(3,4-Dichlorophenyl)-1,3,4-oxadiazol-2-yl]methyl]-1,3-dimethyl-8-[4-[4-[[4-[2-(1-methyl-2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidine-1-carbonyl]piperazin-1-yl]purine-2,6-dione	CN1C(=O)CCC(N2C(=O)C3=C(C=C(N4CCN(CC5CCN(C(=O)N6CCN(C7=NC8=C(C(=O)N(C)C(=O)N8C)N7CC7=NN=C(C8=CC=C(Cl)C(Cl)=C8)O7)CC6)CC5)CC4)C=C3)C2=O)C1=O	C45H49Cl2N13O8	NUDT5	Q9UKK9	CRBN	WO-2024127022-A1
TPD-V9LOLF	PROTAC SMARCA2/4 degrader-37	orb2695173; SCHEMBL23773057; SCHEMBL31578728; PROTAC SMARCA2/4 degrader-37; HY-169861; 2688882-69-9	O=C1CCC(N2C(=O)c3cccc(NCCCCNC(=O)c4cccc(C#Cc5cc(NC(=O)Nc6ccnc(Cl)c6)ccn5)c4)c3C2=O)C(=O)N1	C37H31ClN8O6	SMARCA4	P51532	CRBN	WO-2024130027-A2
TPD-BBDXLW	SCHEMBL22845000	2-(2,6-dioxopiperidin-3-yl)-5-[8-[2-[3-[(1R,4R)-5-[(E)-3-(2-hydroxyphenyl)-3-oxoprop-1-enyl]-2,5-diazabicyclo[2.2.1]heptan-2-yl]phenyl]ethoxy]octylamino]isoindole-1,3-dione; SCHEMBL30207630	O=C1CCC(N2C(=O)c3ccc(NCCCCCCCCOCCc4cccc(N5C[C@H]6C[C@@H]5CN6/C=C/C(=O)c5ccccc5O)c4)cc3C2=O)C(=O)N1	C43H49N5O7	SMARCA4	P51532	CRBN	WO-2024130027-A2
TPD-A740Y6	WO2024131777A1_C001	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC(=CF)CN5CCC(CCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)NCc6ccc(-c7scnc7C)cc6)C(C)(C)C)CC5)nc4c3F)c12	C59H65F3N10O6S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-E65HMY	WO2024131777A1_C002	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC(=CF)CN5CCC(OCCC(=O)N[C@H](C(=O)N6C[C@H](O)CC6C(=O)NCc6ccc(-c7scnc7C)cc6)C(C)(C)C)CC5)nc4c3F)c12	C59H65F3N10O7S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-OEDP27	WO2024131777A1_C003A	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C/F)CN(C)CC5CCC(CC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)NCc6ccc(-c7scnc7C)cc6)C(C)(C)C)CC5)nc4c3F)c12	C61H69F3N10O6S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-HO8FPL	WO2024131777A1_C003B	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C\F)CN(C)CC5CCC(CC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)NCc6ccc(-c7scnc7C)cc6)C(C)(C)C)CC5)nc4c3F)c12	C61H69F3N10O6S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-UMWRT7	WO2024131777A1_C004	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC(=CF)CN(C)C5CCC(CC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)NCc6ccc(-c7scnc7C)cc6)C(C)(C)C)CC5)nc4c3F)c12	C60H67F3N10O6S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-K7DTX6	WO2024131777A1_C005	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC(=CF)CN5CCC(OCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)NCc6ccc(-c7scnc7C)cc6)C(C)(C)C)CC5)nc4c3F)c12	C58H63F3N10O7S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-YCNPMZ	WO2024131777A1_C006	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC(=CF)CN(C)CCCCCCC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)NCc5ccc(-c6scnc6C)cc5)C(C)(C)C)nc4c3F)c12	C59H67F3N10O6S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-F33XTB	WO2024131777A1_C007	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC(=CF)CN(C)Cc5ccc(CC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)NCc6ccc(-c7scnc7C)cc6)C(C)(C)C)cc5)nc4c3F)c12	C61H63F3N10O6S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-9ARPMC	WO2024131777A1_C008	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C/F)CN(C)C5CC6(CC(C(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)NCc7ccc(-c8scnc8C)cc7)C(C)(C)C)C6)C5)nc4c3F)c12	C60H65F3N10O6S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-ZG5FY8	WO2024131777A1_C010	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC(=CF)CN(C)CCc5ccccc5CC(=O)N[C@H](C(=O)N5C[C@@H](O)C[C@@H]5C(=O)NCc5ccc(-c6scnc6C)cc5)C(C)C)nc4c3F)c12	C61H63F3N10O6S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-UMCVBB	WO2024131777A1_C011	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC(=CF)CN5CCC(CCCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)NCc6ccc(-c7scnc7C)cc6)C(C)(C)C)CC5)nc4c3F)c12	C60H67F3N10O6S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-N7DGNM	WO2024131777A1_C011A	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C/F)CN(C)CCCCCC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)NCc5ccc(-c6scnc6C)cc5)C(C)(C)C)nc4c3F)c12	C58H65F3N10O6S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-DTTRY1	WO2024131777A1_C011B	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C\F)CN(C)CCCCCC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)NCc5ccc(-c6scnc6C)cc5)C(C)(C)C)nc4c3F)c12	C58H65F3N10O6S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-CAWQ2B	WO2024131777A1_C012A	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C/F)CN(C)CCCCCCCC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)NCc5ccc(-c6scnc6C)cc5)C(C)(C)C)nc4c3F)c12	C60H69F3N10O6S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-5G26HG	WO2024131777A1_C013	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC(=CF)CN(C)CC56CC(C(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)NCc7ccc(-c8scnc8C)cc7)C(C)(C)C)(C5)C6)nc4c3F)c12	C59H63F3N10O6S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-6C22UA	WO2024131777A1_C014A	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C/F)CN(C)CC56CC(CC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)NCc7ccc(-c8scnc8C)cc7)C(C)(C)C)(C5)C6)nc4c3F)c12	C60H65F3N10O6S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-6H2A3N	WO2024131777A1_C014B	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C\F)CN(C)CC56CC(CC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)NCc7ccc(-c8scnc8C)cc7)C(C)(C)C)(C5)C6)nc4c3F)c12	C60H65F3N10O6S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-PZ17HW	WO2024131777A1_C015A	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C/F)CN(C)CC56CCC(CC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)NCc7ccc(-c8scnc8C)cc7)C(C)(C)C)(CC5)CC6)nc4c3F)c12	C63H71F3N10O6S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-M0LLOS	WO2024131777A1_C015B	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C\F)CN(C)CC56CCC(CC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)NCc7ccc(-c8scnc8C)cc7)C(C)(C)C)(CC5)CC6)nc4c3F)c12	C63H71F3N10O6S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-T2KAUX	WO2024131777A1_C016A	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C/F)CN(C)CCC5CCC(CC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)NCc6ccc(-c7scnc7C)cc6)C(C)(C)C)CC5)nc4c3F)c12	C62H71F3N10O6S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-JJJABX	WO2024131777A1_C016B	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C\F)CN(C)CCC5CCC(CC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)NCc6ccc(-c7scnc7C)cc6)C(C)(C)C)CC5)nc4c3F)c12	C62H71F3N10O6S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-K8WS9E	WO2024131777A1_C017A	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C/F)CN(C)CCc5cccc(CC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)NCc6ccc(-c7scnc7C)cc6)C(C)(C)C)c5)nc4c3F)c12	C62H65F3N10O6S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-4D6YKR	WO2024131777A1_C017B	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C\F)CN(C)CCc5cccc(CC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)NCc6ccc(-c7scnc7C)cc6)C(C)(C)C)c5)nc4c3F)c12	C62H65F3N10O6S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-TY4YZ4	WO2024131777A1_C019	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC(=CF)CNCC56CCC(C(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)NCc7ccc(-c8scnc8C)cc7)C(C)(C)C)(CC5)CC6)nc4c3F)c12	C61H67F3N10O6S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-0263TX	WO2024131777A1_C020A	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C/F)CN(C)Cc5ccc(C(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)NCc6ccc(-c7scnc7C)cc6)C(C)(C)C)cc5)nc4c3F)c12	C60H61F3N10O6S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-8R0L4O	WO2024131777A1_C020B	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C\F)CN(C)Cc5ccc(C(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)NCc6ccc(-c7scnc7C)cc6)C(C)(C)C)cc5)nc4c3F)c12	C60H61F3N10O6S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-OUL2M2	WO2024131777A1_C021	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC(=CF)CN5CCC(CC6CCN(C(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)NCc7ccc(-c8scnc8C)cc7)C(C)(C)C)CC6)CC5)nc4c3F)c12	C63H72F3N11O6S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-KBWJ0S	WO2024131777A1_C022	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC(=CF)CN5CCC(OCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@H](CO)c6ccc(-c7scnc7C)cc6)C(C)(C)C)CC5)nc4c3F)c12	C59H65F3N10O8S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-9FSVK6	WO2024131777A1_C023A	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C/F)CN5CCC(OCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)c6ccc(-c7scnc7C)cc6)C(C)(C)C)CC5)nc4c3F)c12	C59H65F3N10O7S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-H0KZLV	WO2024131777A1_C023B	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C\F)CN5CCC(OCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)c6ccc(-c7scnc7C)cc6)C(C)(C)C)CC5)nc4c3F)c12	C59H65F3N10O7S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-SCOOKB	WO2024131777A1_D001	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC(=CF)CN(C)CCCCCCc5cn([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](CO)c6ccc(-c7scnc7C)cc6)C(C)C)nn5)nc4c3F)c12	C60H67F3N12O6S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-T60U7P	WO2024131777A1_D002-1	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC(=CF)CN(C)CCCCCc5cn([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](CO)c6ccc(-c7scnc7C)cc6)C(C)C)nn5)nc4c3F)c12	C59H65F3N12O6S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-CKGVQU	WO2024131777A1_D002-2	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C\F)CN5CCC(Oc6cc([C@@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)NCc7ccc(-c8scnc8C)cc7)C(C)C)on6)CC5)nc4c3F)c12	C58H59F3N10O7S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-YNIQFQ	WO2024131777A1_D003A	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C/F)CN(C)CCc5ccc(-c6cn([C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](CO)c7ccc(-c8scnc8C)cc7)C(C)C)nn6)cc5)nc4c3F)c12	C62H63F3N12O6S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-PYMO6A	WO2024131777A1_D003B	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C\F)CN(C)CCc5ccc(-c6cn([C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](CO)c7ccc(-c8scnc8C)cc7)C(C)C)nn6)cc5)nc4c3F)c12	C62H63F3N12O6S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-6IFMLO	WO2024131777A1_D004A	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C/F)CN5CCC(OCc6cn([C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](CO)c7ccc(-c8scnc8C)cc7)C(C)C)nn6)CC5)nc4c3F)c12	C59H63F3N12O7S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-MMPDZI	WO2024131777A1_D004B	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C\F)CN5CCC(OCc6cn([C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](CO)c7ccc(-c8scnc8C)cc7)C(C)C)nn6)CC5)nc4c3F)c12	C59H63F3N12O7S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-IZIPSF	WO2024131777A1_D005A	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C/F)CN(C)CCc5ccc(-c6cn([C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8scnc8C)cc7)C(C)C)nn6)cc5)nc4c3F)c12	C62H63F3N12O5S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-H0F1TY	WO2024131777A1_D005B	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C\F)CN(C)CCc5ccc(-c6cn([C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8scnc8C)cc7)C(C)C)nn6)cc5)nc4c3F)c12	C62H63F3N12O5S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-OZNQSY	WO2024131777A1_D006	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC(=CF)CN(C)CC(CC)CCCc5cn([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)NCc6ccc(-c7scnc7C)cc6)C(C)C)nn5)nc4c3F)c12	C60H67F3N12O5S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-3GUKW3	WO2024131777A1_D007	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC(=CF)CN(C)CCCc5ccc(-c6cn([C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)NC(CO)c7ccc(-c8scnc8C)cc7)C(C)C)nn6)cc5)nc4c3F)c12	C63H65F3N12O6S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-840EEQ	WO2024131777A1_D008	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC(=CF)CN(C)CCc5ccc(-c6cn([C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](CO)c7ccc(-c8scnc8C)cc7)C(C)C)nn6)c(F)c5)nc4c3F)c12	C62H62F4N12O6S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-9JAGWU	WO2024131777A1_D009A	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C/F)CN(C)CCCc5ccc(-c6cn([C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8scnc8C)cc7)C(C)C)nn6)cc5)nc4c3F)c12	C63H65F3N12O5S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-CJ74JQ	WO2024131777A1_D009B	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C\F)CN(C)CCCc5ccc(-c6cn([C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8scnc8C)cc7)C(C)C)nn6)cc5)nc4c3F)c12	C63H65F3N12O5S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-AJK7LM	WO2024131777A1_D010A	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C/F)CN(C)C[C@H](C)c5ccc(-c6cn([C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](CO)c7ccc(-c8scnc8C)cc7)C(C)C)nn6)cc5)nc4c3F)c12	C63H65F3N12O6S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-G1R9RN	WO2024131777A1_D010B	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C\F)CN(C)C[C@H](C)c5ccc(-c6cn([C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](CO)c7ccc(-c8scnc8C)cc7)C(C)C)nn6)cc5)nc4c3F)c12	C63H65F3N12O6S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-OVNYNJ	WO2024131777A1_D011A	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C/F)CN(C)CCc5ccc(-c6cn([C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8scnc8C)cc7)C(C)C)nn6)c(F)c5)nc4c3F)c12	C62H62F4N12O5S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-CYZOV2	WO2024131777A1_D011B	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C\F)CN(C)CCc5ccc(-c6cn([C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8scnc8C)cc7)C(C)C)nn6)c(F)c5)nc4c3F)c12	C62H62F4N12O5S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-W8VYNL	WO2024131777A1_D012A	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](C(C)C)n2cc(-c3ccc(CCN(C)C/C(=C\F)COc4nc(N5CC6CCC(C5)N6)c5cnc(-c6cc(O)cc7ccc(F)c(C)c67)c(F)c5n4)cn3)nn2)cc1	C60H64F3N13O5S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-NO5DUM	WO2024131777A1_D012B	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](C(C)C)n2cc(-c3ccc(CCN(C)C/C(=C/F)COc4nc(N5CC6CCC(C5)N6)c5cnc(-c6cc(O)cc7ccc(F)c(C)c67)c(F)c5n4)cn3)nn2)cc1	C60H64F3N13O5S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-C40JYT	WO2024131777A1_D013A	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C/F)CN(C)CCc5ccc(-c6cn([C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)NCc7ccc(-c8scnc8C)cc7)C(C)C)nn6)cc5Cl)nc4c3F)c12	C61H60ClF3N12O5S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-L7QJQT	WO2024131777A1_D013B	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C\F)CN(C)CCc5ccc(-c6cn([C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)NCc7ccc(-c8scnc8C)cc7)C(C)C)nn6)cc5Cl)nc4c3F)c12	C61H60ClF3N12O5S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-T62JT3	WO2024131777A1_D014A	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C/F)CN(C)Cc5ccc(OCc6cn([C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8scnc8C)cc7)C(C)C)nn6)c(F)c5)nc4c3F)c12	C62H62F4N12O6S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-IXZ62R	WO2024131777A1_D014B	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C\F)CN(C)Cc5ccc(OCc6cn([C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8scnc8C)cc7)C(C)C)nn6)c(F)c5)nc4c3F)c12	C62H62F4N12O6S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-6JFKEK	WO2024131777A1_D015	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC(=CF)CN(C)Cc5ccc(Cc6cn(C(C(=O)N7C[C@H](O)C[C@H]7C(=O)NCc7ccc(-c8scnc8C)cc7)C(C)C)nn6)cc5)nc4c3F)c12	C61H61F3N12O5S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-SBL98Z	WO2024131777A1_D016A	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C/F)CN(C)CCc5ccc(-c6cn([C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8scnc8C)cc7)C(C)C)nn6)c(Cl)c5)nc4c3F)c12	C62H62ClF3N12O5S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-JYOUJS	WO2024131777A1_D016B	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C\F)CN(C)CCc5ccc(-c6cn([C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8scnc8C)cc7)C(C)C)nn6)c(Cl)c5)nc4c3F)c12	C62H62ClF3N12O5S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-KJLO0T	WO2024131777A1_D017A	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C/F)CN(C)CC(C)(C)c5ccc(-c6cn([C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8scnc8C)cc7)C(C)C)nn6)cc5)nc4c3F)c12	C64H67F3N12O5S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-Y3FSRV	WO2024131777A1_D017B	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C\F)CN(C)CC(C)(C)c5ccc(-c6cn([C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8scnc8C)cc7)C(C)C)nn6)cc5)nc4c3F)c12	C64H67F3N12O5S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-XYTZK5	WO2024131777A1_D018A	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C/F)CNCCc5ccc(-c6cn([C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8ccnn8CC)cc7)C(C)C)nn6)cc5Cl)nc4c3F)c12	C62H63ClF3N13O5	KRAS	P01116	VHL	WO-2024131777-A1
TPD-3UT2KX	WO2024131777A1_D018B	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C\F)CNCCc5ccc(-c6cn([C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8ccnn8CC)cc7)C(C)C)nn6)cc5Cl)nc4c3F)c12	C62H63ClF3N13O5	KRAS	P01116	VHL	WO-2024131777-A1
TPD-SA2DPW	WO2024131777A1_D019A	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](C(C)C)n2cc(-c3ccc(CCCN(C)C/C(=C\F)COc4nc(N5CC6CCC(C5)N6)c5cnc(-c6cc(O)cc7cccc(Cl)c67)c(F)c5n4)cc3)nn2)cc1	C61H65ClF2N12O5S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-0I8E1X	WO2024131777A1_D019B	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](C(C)C)n2cc(-c3ccc(CCCN(C)C/C(=C/F)COc4nc(N5CC6CCC(C5)N6)c5cnc(-c6cc(O)cc7cccc(Cl)c67)c(F)c5n4)cc3)nn2)cc1	C61H65ClF2N12O5S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-8LO4GB	WO2024131777A1_D020	.	CCc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC(=CF)CN(C)CCCc5ccc(-c6cn([C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)c7ccc(-c8scnc8C)cc7)C(C)C)nn6)cc5)nc4c3F)c12	C63H69F3N12O5S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-H35RF4	WO2024131777A1_D021A	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C/F)CN5CCC(Oc6cc(C(C(=O)N7C[C@H](O)C[C@H]7C(=O)NCc7ccc(-c8scnc8C)cc7)C(C)C)on6)CC5)nc4c3F)c12	C58H59F3N10O7S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-AZZVWC	WO2024131777A1_D021B	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C\F)CN5CCC(Oc6cc(C(C(=O)N7C[C@H](O)C[C@H]7C(=O)NCc7ccc(-c8scnc8C)cc7)C(C)C)on6)CC5)nc4c3F)c12	C58H59F3N10O7S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-PKZ723	WO2024131777A1_D022	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC(=CF)CN5CCC(COc6cc(C(C(=O)N7C[C@H](O)C[C@H]7C(=O)NCc7ccc(-c8scnc8C)cc7)C(C)C)on6)CC5)nc4c3F)c12	C59H61F3N10O7S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-WBHYYQ	WO2024131777A1_D023	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC(=CF)CNCC5CCC(COc6cc(C(C(=O)N7C[C@H](O)C[C@H]7C(=O)NCc7ccc(-c8scnc8C)cc7)C(C)C)on6)CC5)nc4c3F)c12	C61H65F3N10O7S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-WHSUSK	WO2024131777A1_D024	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC(=CF)CN(C)CC5CCC(Oc6cc(C(C(=O)N7C[C@H](O)C[C@H]7C(=O)NCc7ccc(-c8scnc8C)cc7)C(C)C)on6)CC5)nc4c3F)c12	C61H65F3N10O7S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-QK8TU9	WO2024131777A1_D025	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC(=CF)CN(C)Cc5ccc(COc6cc(C(C(=O)N7C[C@H](O)C[C@H]7C(=O)NCc7ccc(-c8scnc8C)cc7)C(C)C)on6)cc5)nc4c3F)c12	C62H61F3N10O7S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-F4X1X5	WO2024131777A1_E001	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)C)c(OCCCCCCN(C)CC(=CF)COc2nc(N3CC4CCC(C3)N4)c3cnc(-c4cc(O)cc5ccc(F)c(C)c45)c(F)c3n2)c1	C61H72F4N10O7S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-JNYXT4	WO2024131777A1_E002	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC(=CF)CN(C)CCCCCCCOc5cc(-c6scnc6C)ccc5CNC(=O)[C@@H]5C[C@@H](O)CN5C(=O)[C@@H](NC(O)C5(F)CC5)C(C)(C)C)nc4c3F)c12	C63H74F4N10O7S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-IH2TT1	WO2024131777A1_E003	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC(=CF)CN(C)CCCCCCCCOc5cc(-c6scnc6C)ccc5CNC(=O)[C@@H]5C[C@@H](O)CN5C(=O)[C@@H](NC(=O)C5(F)CC5)C(C)(C)C)nc4c3F)c12	C64H74F4N10O7S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-10FQ4Q	WO2024131777A1_E004	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC(=CF)CN5CCC(OCCOc6cc(-c7scnc7C)ccc6CNC(=O)[C@@H]6C[C@@H](O)CN6C(=O)C(NC(=O)C6(F)CC6)C(C)(C)C)CC5)nc4c3F)c12	C62H68F4N10O8S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-AA8BER	WO2024131777A1_E005A	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C/F)CN(C)C[C@H]5CC[C@H](COc6cc(-c7scnc7C)ccc6CNC(=O)[C@@H]6C[C@@H](O)CN6C(=O)[C@@H](NC(=O)C6(F)CC6)C(C)(C)C)CC5)nc4c3F)c12	C64H72F4N10O7S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-GDQ6S9	WO2024131777A1_E005B	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C\F)CN(C)C[C@H]5CC[C@H](COc6cc(-c7scnc7C)ccc6CNC(=O)[C@@H]6C[C@@H](O)CN6C(=O)[C@@H](NC(=O)C6(F)CC6)C(C)(C)C)CC5)nc4c3F)c12	C64H72F4N10O7S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-IU0GWX	WO2024131777A1_E006A	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C/F)CN(C)CC5CC(COc6cc(-c7scnc7C)ccc6CNC(=O)[C@@H]6C[C@@H](O)CN6C(=O)[C@@H](NC(=O)C6(F)CC6)C(C)(C)C)C5)nc4c3F)c12	C62H68F4N10O7S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-AOJUMY	WO2024131777A1_E006B	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C\F)CN(C)CC5CC(COc6cc(-c7scnc7C)ccc6CNC(=O)[C@@H]6C[C@@H](O)CN6C(=O)[C@@H](NC(=O)C6(F)CC6)C(C)(C)C)C5)nc4c3F)c12	C62H68F4N10O7S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-DQJL5Z	WO2024131777A1_E007	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC(=CF)CNC5CC6(C5)CC(Oc5cc(-c7scnc7C)ccc5CNC(=O)[C@@H]5C[C@@H](O)CN5C(=O)[C@@H](NC(=O)C5(F)CC5)C(C)(C)C)C6)nc4c3F)c12	C62H66F4N10O7S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-QXFQ20	WO2024131777A1_E008A	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C/F)CN(C)Cc5ccc(COc6cc(-c7scnc7C)ccc6CNC(=O)[C@@H]6C[C@@H](O)CN6C(=O)[C@@H](NC(=O)C6(F)CC6)C(C)(C)C)cc5)nc4c3F)c12	C64H66F4N10O7S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-G5XURZ	WO2024131777A1_E008B	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C\F)CN(C)Cc5ccc(COc6cc(-c7scnc7C)ccc6CNC(=O)[C@@H]6C[C@@H](O)CN6C(=O)[C@@H](NC(=O)C6(F)CC6)C(C)(C)C)cc5)nc4c3F)c12	C64H66F4N10O7S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-FJN1DQ	WO2024131777A1_E009A	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C/F)CN(C)C[C@H]5CC[C@H](COc6cc(-c7scnc7C)ccc6[C@H](C)NC(=O)[C@@H]6C[C@@H](O)CN6C(=O)C(NC(=O)C6(N)CC6)C(C)(C)C)CC5)nc4c3F)c12	C65H76F3N11O7S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-2164OC	WO2024131777A1_E009B	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C\F)CN(C)C[C@H]5CC[C@H](COc6cc(-c7scnc7C)ccc6[C@H](C)NC(=O)[C@@H]6C[C@@H](O)CN6C(=O)C(NC(=O)C6(N)CC6)C(C)(C)C)CC5)nc4c3F)c12	C65H76F3N11O7S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-MBDGO9	WO2024131777A1_E010A	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C/F)CN(C)Cc5ccc(COc6cc(-c7scnc7C)ccc6[C@H](C)NC(=O)[C@@H]6C[C@@H](O)CN6C(=O)[C@@H](n6cc(C7CC7)nn6)C(C)(C)C)cc5)nc4c3F)c12	C66H69F3N12O6S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-CB6JCT	WO2024131777A1_E010B	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C\F)CN(C)Cc5ccc(COc6cc(-c7scnc7C)ccc6[C@H](C)NC(=O)[C@@H]6C[C@@H](O)CN6C(=O)[C@@H](n6cc(C7CC7)nn6)C(C)(C)C)cc5)nc4c3F)c12	C66H69F3N12O6S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-S82SSA	WO2024131777A1_E011A	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C/F)CN(C)Cc5ccc(COc6cc(-c7scnc7C)ccc6[C@H](C)NC(=O)[C@@H]6C[C@@H](O)CN6C(=O)C(c6cc(C)no6)C(C)C)cc5)nc4c3F)c12	C64H65F3N10O7S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-94750V	WO2024131777A1_E011B	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C\F)CN(C)Cc5ccc(COc6cc(-c7scnc7C)ccc6[C@H](C)NC(=O)[C@@H]6C[C@@H](O)CN6C(=O)C(c6cc(C)no6)C(C)C)cc5)nc4c3F)c12	C64H65F3N10O7S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-HKF22F	WO2024131777A1_E012A	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C/F)CN(C)CCc5ccc(COc6cc(-c7scnc7C)ccc6[C@H](C)NC(=O)[C@@H]6C[C@@H](O)CN6C(=O)[C@@H](NC(=O)C6(F)CC6)C(C)(C)C)cc5)nc4c3F)c12	C66H70F4N10O7S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-XNKG1A	WO2024131777A1_E012B	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C\F)CN(C)CCc5ccc(COc6cc(-c7scnc7C)ccc6[C@H](C)NC(=O)[C@@H]6C[C@@H](O)CN6C(=O)[C@@H](NC(=O)C6(F)CC6)C(C)(C)C)cc5)nc4c3F)c12	C66H70F4N10O7S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-X6X66K	WO2024131777A1_E013A	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C/F)CN(C)Cc5ccc(COc6cc(-c7scnc7C)ccc6[C@H](C)NC(=O)[C@@H]6C[C@@H](O)CN6C(=O)[C@@H](NC(=O)C6(F)CC6)C(C)(C)C)cn5)nc4c3F)c12	C64H67F4N11O7S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-KHPS8G	WO2024131777A1_E013B	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C\F)CN(C)Cc5ccc(COc6cc(-c7scnc7C)ccc6[C@H](C)NC(=O)[C@@H]6C[C@@H](O)CN6C(=O)[C@@H](NC(=O)C6(F)CC6)C(C)(C)C)cn5)nc4c3F)c12	C64H67F4N11O7S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-IO0CXE	WO2024131777A1_E014A	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C/F)CN(C)Cc5ccc(COc6cc(-c7scnc7C)ccc6[C@H](C)NC(=O)[C@@H]6C[C@@H](O)CN6C(=O)[C@@H](NC(=O)C6(F)CC6)C(C)(C)C)cc5F)nc4c3F)c12	C65H67F5N10O7S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-7FDSRH	WO2024131777A1_E014B	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C\F)CN(C)Cc5ccc(COc6cc(-c7scnc7C)ccc6[C@H](C)NC(=O)[C@@H]6C[C@@H](O)CN6C(=O)[C@@H](NC(=O)C6(F)CC6)C(C)(C)C)cc5F)nc4c3F)c12	C65H67F5N10O7S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-HEBQTJ	WO2024131777A1_E015A	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C/F)CN(C)Cc5ccc(COc6cc(-c7scnc7C)ccc6[C@H](C)NC(=O)[C@@H]6C[C@@H](O)CN6C(=O)[C@@H](NC(=O)C6(F)CC6)C(C)(C)C)c(F)c5)nc4c3F)c12	C65H67F5N10O7S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-HPS0B9	WO2024131777A1_E015B	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C\F)CN(C)Cc5ccc(COc6cc(-c7scnc7C)ccc6[C@H](C)NC(=O)[C@@H]6C[C@@H](O)CN6C(=O)[C@@H](NC(=O)C6(F)CC6)C(C)(C)C)c(F)c5)nc4c3F)c12	C65H67F5N10O7S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-W79GRG	WO2024131777A1_E016A	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C/F)CN(C)Cc5ccc(COc6cc(-c7scnc7C)ccc6[C@H](C)NC(=O)[C@@H]6C[C@@H](O)CN6C(=O)[C@@H](NC(=O)C6(F)CC6)C(C)(C)C)cc5Cl)nc4c3F)c12	C65H67ClF4N10O7S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-HZ7OAI	WO2024131777A1_E016B	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C\F)CN(C)Cc5ccc(COc6cc(-c7scnc7C)ccc6[C@H](C)NC(=O)[C@@H]6C[C@@H](O)CN6C(=O)[C@@H](NC(=O)C6(F)CC6)C(C)(C)C)cc5Cl)nc4c3F)c12	C65H67ClF4N10O7S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-6CLDXE	WO2024131777A1_E017A	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C/F)CN(C)Cc5ccc(COc6cc(-c7scnc7C)ccc6CNC(=O)[C@@H]6C[C@@H](O)CN6C(=O)[C@@H](NC(=O)C6(F)CC6)C(C)(C)C)c(F)c5)nc4c3F)c12	C64H65F5N10O7S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-GK0E1H	WO2024131777A1_E017B	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C\F)CN(C)Cc5ccc(COc6cc(-c7scnc7C)ccc6CNC(=O)[C@@H]6C[C@@H](O)CN6C(=O)[C@@H](NC(=O)C6(F)CC6)C(C)(C)C)c(F)c5)nc4c3F)c12	C64H65F5N10O7S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-15GBAG	WO2024131777A1_E018	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC(=CF)CN(C)Cc5ccc(COc6cc(-c7scnc7C)ccc6CNC(=O)[C@@H]6C[C@@H](O)CN6C(=O)[C@@H](n6cc(C7CC7)nn6)C(C)(C)C)cc5)nc4c3F)c12	C65H67F3N12O6S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-N2QDDH	WO2024131777A1_E019A	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C/F)CN(C)Cc5ccc(COc6cc(-c7scnc7C)ccc6[C@H](C)NC(=O)[C@@H]6C[C@@H](O)CN6C(=O)[C@@H](NC(=O)C6(F)CC6)C(C)(C)C)cc5)nc4c3F)c12	C65H68F4N10O7S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-FMM4S6	WO2024131777A1_E019B	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C\F)CN(C)Cc5ccc(COc6cc(-c7scnc7C)ccc6[C@H](C)NC(=O)[C@@H]6C[C@@H](O)CN6C(=O)[C@@H](NC(=O)C6(F)CC6)C(C)(C)C)cc5)nc4c3F)c12	C65H68F4N10O7S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-5N8P3F	WO2024131777A1_E020	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC(=CF)CN(C)Cc5ccc(COc6cc(-c7c(F)cccc7F)ccc6[C@H](C)NC(=O)[C@@H]6C[C@@H](O)CN6C(=O)[C@@H](NC(=O)C6(F)CC6)C(C)(C)C)cc5)nc4c3F)c12	C67H67F6N9O7	KRAS	P01116	VHL	WO-2024131777-A1
TPD-J4R8YR	WO2024131777A1_E021	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC(=CF)CN(C)Cc5ccc(COc6cc(-c7scnc7C)ccc6CNC(=O)[C@@H]6C[C@@H](O)CN6C(=O)[C@@H](NC(=O)C6(F)CC6)C(C)(C)C)c(Cl)c5)nc4c3F)c12	C64H65ClF4N10O7S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-HAV3RA	WO2024131777A1_E022	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC(=CF)CN(C)Cc5ccc(COc6cc(-c7scnc7C)ccc6CNC(=O)[C@@H]6C[C@@H](O)CN6C(=O)[C@@H](NC(=O)C6(F)CC6)C(C)(C)C)cc5)nc4c3F)c12	C64H66F4N10O7S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-06RZMM	WO2024131777A1_F001	.	Cc1ncsc1-c1ccc([C@H](CO)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](C(C)C)n2cc(-c3ccc(COc4c(-c5c(C)c(F)cc6[nH]ncc56)c(C5CC5)cc5c(N6CC7CCC(C6)N7)nc(OCC(=CF)CN(C)C)nc45)cc3)nn2)cc1	C62H69F2N13O6S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-MTSESW	WO2024131777A1_G001A	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C/F)CN(C)Cc5ccc(CSC(C)(C)[C@H](NC(=O)C6(F)CC6)C(=O)N6C[C@H](O)C[C@H]6C(=O)NCc6ccc(-c7scnc7C)cc6)cc5)nc4c3F)c12	C63H64F4N10O6S2	KRAS	P01116	VHL	WO-2024131777-A1
TPD-J0YAEQ	WO2024131777A1_G001B	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C\F)CN(C)Cc5ccc(CSC(C)(C)[C@H](NC(=O)C6(F)CC6)C(=O)N6C[C@H](O)C[C@H]6C(=O)NCc6ccc(-c7scnc7C)cc6)cc5)nc4c3F)c12	C63H64F4N10O6S2	KRAS	P01116	VHL	WO-2024131777-A1
TPD-I0D1O7	WO2024131777A1_G002A	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C/F)CN(C)C[C@H]5CC[C@H](CSC(C)(C)[C@H](NC(=O)C6(F)CC6)C(=O)N6C[C@H](O)C[C@H]6C(=O)NCc6ccc(-c7scnc7C)cc6)CC5)nc4c3F)c12	C63H70F4N10O6S2	KRAS	P01116	VHL	WO-2024131777-A1
TPD-O0G6DJ	WO2024131777A1_G002B	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C\F)CN(C)C[C@H]5CC[C@H](CSC(C)(C)[C@H](NC(=O)C6(F)CC6)C(=O)N6C[C@H](O)C[C@H]6C(=O)NCc6ccc(-c7scnc7C)cc6)CC5)nc4c3F)c12	C63H70F4N10O6S2	KRAS	P01116	VHL	WO-2024131777-A1
TPD-U0KKZF	WO2024131777A1_H001A	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C/F)CN(C)CCC(=O)NC[C@H](NC(=O)[C@@H]5C[C@@H](O)CN5C(=O)[C@@H](NC(=O)C5(F)CC5)C(C)(C)C)c5ccc(-c6scnc6C)cc5)nc4c3F)c12	C60H65F4N11O7S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-QLYX7R	WO2024131777A1_H001B	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC/C(=C\F)CN(C)CCC(=O)NC[C@H](NC(=O)[C@@H]5C[C@@H](O)CN5C(=O)[C@@H](NC(=O)C5(F)CC5)C(C)(C)C)c5ccc(-c6scnc6C)cc5)nc4c3F)c12	C60H65F4N11O7S	KRAS	P01116	VHL	WO-2024131777-A1
TPD-IWF3XD	SCHEMBL30971903	1-[4-[5-[(1R)-1-(3,5-dichloropyridin-4-yl)ethoxy]-1H-indazol-3-yl]benzoyl]-N-[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]piperidine-4-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3CCN(C(=O)C4=CC=C(C5=NNC6=C5C=C(O[C@H](C)C5=C(Cl)C=NC=C5Cl)C=C6)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C50H54Cl2N8O6S	FGFR3	P22607	VHL	WO-2024137742-A1
TPD-ADNGPX	WO2024137742A1_2	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CC(C)(C)CNC(=O)C3=CC=C(C4=NNC5=C4C=C(O[C@H](C)C4=C(Cl)C=NC=C4Cl)C=C5)C=C3)C(C)(C)C)C=C2)SC=N1	C50H56Cl2N8O6S	FGFR3	P22607	VHL	WO-2024137742-A1
TPD-XGHYQA	WO2024137742A1_3	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCNC(=O)C3=CC=C(C4=NNC5=C4C=C(O[C@H](C)C4=C(Cl)C=NC=C4Cl)C=C5)C=C3)C(C)(C)C)C=C2)SC=N1	C52H60Cl2N8O6S	FGFR3	P22607	VHL	WO-2024137742-A1
TPD-Q1CH9W	WO2024137742A1_4	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOCCOCCNC(=O)C3=CC=C(C4=NNC5=C4C=C(O[C@H](C)C4=C(Cl)C=NC=C4Cl)C=C5)C=C3)C(C)(C)C)C=C2)SC=N1	C56H68Cl2N8O11S	FGFR3	P22607	VHL	WO-2024137742-A1
TPD-4ZQKJP	WO2024137742A1_5	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCCCNC(=O)C3=CC=C(C4=NNC5=C4C=C(O[C@H](C)C4=C(Cl)C=NC=C4Cl)C=C5)C=C3)C(C)(C)C)C=C2)SC=N1	C54H64Cl2N8O6S	FGFR3	P22607	VHL	WO-2024137742-A1
TPD-W4XA96	WO2024137742A1_6	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCNC(=O)C3=CC=C(C4=NNC5=C4C=C(O[C@H](C)C4=C(Cl)C=NC=C4Cl)C=C5)C=C3)C(C)(C)C)C=C2)SC=N1	C50H56Cl2N8O6S	FGFR3	P22607	VHL	WO-2024137742-A1
TPD-VNER47	WO2024137742A1_7	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCNC(=O)C3=CC=C(C4=NNC5=C4C=C(O[C@H](C)C4=C(Cl)C=NC=C4Cl)C=C5)C=C3)C(C)(C)C)C=C2)SC=N1	C48H52Cl2N8O7S	FGFR3	P22607	VHL	WO-2024137742-A1
TPD-DXKP1A	WO2024137742A1_8	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCNC(=O)C3=CC=C(C4=NNC5=C4C=C(O[C@H](C)C4=C(Cl)C=NC=C4Cl)C=C5)C=C3)C(C)(C)C)C=C2)SC=N1	C48H52Cl2N8O6S	FGFR3	P22607	VHL	WO-2024137742-A1
TPD-CTODPZ	WO2024137742A1_9	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCCCCCNC(=O)C3=CC=CC(C4=NNC5=C4C=C(O[C@H](C)C4=C(Cl)C=NC=C4Cl)C=C5)=C3)C(C)(C)C)C=C2)SC=N1	C56H68Cl2N8O6S	FGFR3	P22607	VHL	WO-2024137742-A1
TPD-7K8VFN	WO2024137742A1_10	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCNC(=O)C3=CC=C(C4=NNC5=C4C=C(O[C@H](C)C4=C(Cl)C=NC=C4Cl)C=C5)C=C3)C(C)(C)C)C=C2)SC=N1	C49H54Cl2N8O6S	FGFR3	P22607	VHL	WO-2024137742-A1
TPD-HQTFT4	WO2024137742A1_11	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOCCNC(=O)C3=CC=C(C4=NNC5=C4C=C(O[C@H](C)C4=C(Cl)C=NC=C4Cl)C=C5)C=C3)C(C)(C)C)C=C2)SC=N1	C54H64Cl2N8O10S	FGFR3	P22607	VHL	WO-2024137742-A1
TPD-1PBKGK	WO2024137742A1_12	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCNC(=O)C3=CC=C(C4=NNC5=C4C=C(O[C@H](C)C4=C(Cl)C=NC=C4Cl)C=C5)C=C3)C(C)(C)C)C=C2)SC=N1	C50H56Cl2N8O8S	FGFR3	P22607	VHL	WO-2024137742-A1
TPD-ITOU8S	SCHEMBL30971822	(2S,4R)-N-[[2-[2-[2-[2-[[4-[5-[(1R)-1-(3,5-dichloropyridin-4-yl)ethoxy]-1H-indazol-3-yl]benzoyl]amino]ethoxy]ethoxy]ethoxy]-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-1-[(2S)-2-[(1-fluorocyclopropanecarbonyl)amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide; SCHEMBL30971823	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3(F)CC3)C(C)(C)C)C(OCCOCCOCCNC(=O)C3=CC=C(C4=NNC5=C4C=C(O[C@H](C)C4=C(Cl)C=NC=C4Cl)C=C5)C=C3)=C2)SC=N1	C53H59Cl2FN8O9S	FGFR3	P22607	VHL	WO-2024137742-A1
TPD-G7E3JD	WO2024137742A1_14	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3(F)CC3)C(C)(C)C)C(OCCCCNC(=O)C3=CC=C(C4=NNC5=C4C=C(O[C@H](C)C4=C(Cl)C=NC=C4Cl)C=C5)C=C3)=C2)SC=N1	C51H55Cl2FN8O7S	FGFR3	P22607	VHL	WO-2024137742-A1
TPD-RMH490	WO2024137742A1_15	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3(F)CC3)C(C)(C)C)C(OCCCCCCNC(=O)C3=CC=C(C4=NNC5=C4C=C(O[C@H](C)C4=C(Cl)C=NC=C4Cl)C=C5)C=C3)=C2)SC=N1	C53H59Cl2FN8O7S	FGFR3	P22607	VHL	WO-2024137742-A1
TPD-ZAH07I	WO2024137742A1_16	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3(F)CC3)C(C)(C)C)C(OCCOCCNC(=O)C3=CC=C(C4=NNC5=C4C=C(O[C@H](C)C4=C(Cl)C=NC=C4Cl)C=C5)C=C3)=C2)SC=N1	C51H55Cl2FN8O8S	FGFR3	P22607	VHL	WO-2024137742-A1
TPD-EBL4OH	WO2024137742A1_17	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3(F)CC3)C(C)(C)C)C(OCCCNC(=O)C3=CC=C(C4=NNC5=C4C=C(O[C@H](C)C4=C(Cl)C=NC=C4Cl)C=C5)C=C3)=C2)SC=N1	C50H53Cl2FN8O7S	FGFR3	P22607	VHL	WO-2024137742-A1
TPD-AW9YU8	WO2024137742A1_18	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3(F)CC3)C(C)(C)C)C(OCCCCCCCNC(=O)C3=CC=C(C4=NNC5=C4C=C(O[C@H](C)C4=C(Cl)C=NC=C4Cl)C=C5)C=C3)=C2)SC=N1	C54H61Cl2FN8O7S	FGFR3	P22607	VHL	WO-2024137742-A1
TPD-C2V1Y7	WO2024137742A1_19	.	CC1=CN=CC(Cl)=C1[C@@H](C)OC1=CC2=C(C=C1)NN=C2C1=CC=C(CNC(=O)COCCOC2=CC(C3=C(C)N=CS3)=CC=C2CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)C)C=C1	C52H58ClFN8O8S	FGFR3	P22607	VHL	WO-2024137742-A1
TPD-7AAF5Q	WO2024137742A1_20	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3(F)CC3)C(C)(C)C)C(OCCCC(=O)NCC3=CC=C(C4=NNC5=C4C=C(O[C@H](C)C4=C(Cl)C=NC=C4Cl)C=C5)C=C3)=C2)SC=N1	C51H55Cl2FN8O7S	FGFR3	P22607	VHL	WO-2024137742-A1
TPD-9H0VIN	WO2024137742A1_21	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3(F)CC3)C(C)(C)C)C(OCCOCCOCC(=O)NCC3=CC=C(C4=NNC5=C4C=C(O[C@H](C)C4=C(Cl)C=NC=C4Cl)C=C5)C=C3)=C2)SC=N1	C53H59Cl2FN8O9S	FGFR3	P22607	VHL	WO-2024137742-A1
TPD-5BALAS	WO2024137742A1_22	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOCCOCC(=O)NCC3=CC=C(C4=NNC5=C4C=C(O[C@H](C)C4=C(Cl)C=NC=C4Cl)C=C5)C=C3)C(C)(C)C)C=C2)SC=N1	C56H68Cl2N8O11S	FGFR3	P22607	VHL	WO-2024137742-A1
TPD-UNPJ9C	WO2024137742A1_23	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOCC(=O)NCC3=CC=C(C4=NNC5=C4C=C(O[C@H](C)C4=C(Cl)C=NC=C4Cl)C=C5)C=C3)C(C)(C)C)C=C2)SC=N1	C54H64Cl2N8O10S	FGFR3	P22607	VHL	WO-2024137742-A1
TPD-9QFC0O	WO2024137742A1_24	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCC(=O)NCC3=CC=C(C4=NNC5=C4C=C(O[C@H](C)C4=C(Cl)C=NC=C4Cl)C=C5)C=C3)C(C)(C)C)C=C2)SC=N1	C52H60Cl2N8O6S	FGFR3	P22607	VHL	WO-2024137742-A1
TPD-ID01JZ	WO2024137742A1_25	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCC(=O)NCC3=CC=C(C4=NNC5=C4C=C(O[C@H](C)C4=C(Cl)C=NC=C4Cl)C=C5)C=C3)C(C)(C)C)C=C2)SC=N1	C50H56Cl2N8O6S	FGFR3	P22607	VHL	WO-2024137742-A1
TPD-R7UJ38	WO2024137742A1_26	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCC(=O)NCC3=CC=C(C4=NNC5=C4C=C(O[C@H](C)C4=C(Cl)C=NC=C4Cl)C=C5)C=C3)C(C)(C)C)C=C2)SC=N1	C48H52Cl2N8O6S	FGFR3	P22607	VHL	WO-2024137742-A1
TPD-853TQQ	WO2024137742A1_27	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCC(=O)NCC3=CC=C(C4=NNC5=C4C=C(O[C@H](C)C4=C(Cl)C=NC=C4Cl)C=C5)C=C3)C(C)(C)C)C=C2)SC=N1	C49H54Cl2N8O6S	FGFR3	P22607	VHL	WO-2024137742-A1
TPD-HZI0RC	WO2024137742A1_28	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3(F)CC3)C(C)(C)C)C(OCCCCCC(=O)NCC3=CC=C(C4=NNC5=C4C=C(O[C@H](C)C4=C(Cl)C=NC=C4Cl)C=C5)C=C3)=C2)SC=N1	C53H59Cl2FN8O7S	FGFR3	P22607	VHL	WO-2024137742-A1
TPD-GFQJC7	SCHEMBL30971950	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[2-[[3-[5-[(1R)-1-(3,5-dichloropyridin-4-yl)ethoxy]-1H-indazol-3-yl]phenyl]methylamino]-2-oxoethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCC(=O)NCC3=CC=CC(C4=NNC5=C4C=C(O[C@H](C)C4=C(Cl)C=NC=C4Cl)C=C5)=C3)C(C)(C)C)C=C2)SC=N1	C52H60Cl2N8O9S	FGFR3	P22607	VHL	WO-2024137742-A1
TPD-LIEC0C	WO2024137742A1_30	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOCCOCC(=O)NCC3=CC=CC(C4=NNC5=C4C=C(O[C@H](C)C4=C(Cl)C=NC=C4Cl)C=C5)=C3)C(C)(C)C)C=C2)SC=N1	C56H68Cl2N8O11S	FGFR3	P22607	VHL	WO-2024137742-A1
TPD-8NZKCX	WO2024137742A1_31	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCC(=O)NCC3=CC=CC(C4=NNC5=C4C=C(O[C@H](C)C4=C(Cl)C=NC=C4Cl)C=C5)=C3)C(C)(C)C)C=C2)SC=N1	C50H56Cl2N8O6S	FGFR3	P22607	VHL	WO-2024137742-A1
TPD-778UXY	WO2024137742A1_32	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCC(=O)NCC3=CC=CC(C4=NNC5=C4C=C(O[C@H](C)C4=C(Cl)C=NC=C4Cl)C=C5)=C3)C(C)(C)C)C=C2)SC=N1	C49H54Cl2N8O6S	FGFR3	P22607	VHL	WO-2024137742-A1
TPD-Y53DIH	WO2024137742A1_33	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCC(=O)NCC3=CC=CC(C4=NNC5=C4C=C(O[C@H](C)C4=C(Cl)C=NC=C4Cl)C=C5)=C3)C(C)(C)C)C=C2)SC=N1	C52H60Cl2N8O6S	FGFR3	P22607	VHL	WO-2024137742-A1
TPD-B4BZOQ	WO2024137742A1_34	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOCC(=O)NCC3=CC=CC(C4=NNC5=C4C=C(O[C@H](C)C4=C(Cl)C=NC=C4Cl)C=C5)=C3)C(C)(C)C)C=C2)SC=N1	C54H64Cl2N8O10S	FGFR3	P22607	VHL	WO-2024137742-A1
TPD-BXYB7G	SCHEMBL27395620	(2S,4R)-1-[(2S)-2-[[6-[4-[5-[5-[(1R)-1-(3,5-dichloropyridin-4-yl)ethoxy]-1H-indazol-3-yl]pyridin-2-yl]piperazin-1-yl]-6-oxohexanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCC(=O)N3CCN(C4=NC=C(C5=NNC6=C5C=C(O[C@H](C)C5=C(Cl)C=NC=C5Cl)C=C6)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C52H60Cl2N10O6S	FGFR3	P22607	VHL	WO-2024137742-A1
TPD-L73W4P	WO2024137742A1_36	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCC(=O)N3CCN(C4=NC=C(C5=NNC6=C5C=C(O[C@H](C)C5=C(Cl)C=NC=C5Cl)C=C6)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C54H64Cl2N10O6S	FGFR3	P22607	VHL	WO-2024137742-A1
TPD-1XJTV8	WO2024137742A1_37	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCCC(=O)N3CCN(C4=NC=C(C5=NNC6=C5C=C(O[C@H](C)C5=C(Cl)C=NC=C5Cl)C=C6)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C56H68Cl2N10O6S	FGFR3	P22607	VHL	WO-2024137742-A1
TPD-GX5806	WO2024137742A1_38	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCC(=O)N3CCN(C4=NC=C(C5=NNC6=C5C=C(O[C@H](C)C5=C(Cl)C=NC=C5Cl)C=C6)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C54H64Cl2N10O9S	FGFR3	P22607	VHL	WO-2024137742-A1
TPD-WN8CII	WO2024137742A1_39	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOCC(=O)N3CCN(C4=NC=C(C5=NNC6=C5C=C(O[C@H](C)C5=C(Cl)C=NC=C5Cl)C=C6)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C56H68Cl2N10O10S	FGFR3	P22607	VHL	WO-2024137742-A1
TPD-AKW2AO	WO2024137742A1_40	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCC(=O)N3CCN(C4=NC=C(C5=NNC6=C5C=C(O[C@H](C)C5=C(Cl)C=NC=C5Cl)C=C6)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C50H56Cl2N10O6S	FGFR3	P22607	VHL	WO-2024137742-A1
TPD-E3T5S9	WO2024137742A1_41	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOCCOCC(=O)N3CCN(C4=NC=C(C5=NNC6=C5C=C(O[C@H](C)C5=C(Cl)C=NC=C5Cl)C=C6)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C58H72Cl2N10O11S	FGFR3	P22607	VHL	WO-2024137742-A1
TPD-9EUCF1	SCHEMBL30971853	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[3-[5-[(1R)-1-(3,5-dichloropyridin-4-yl)ethoxy]-1H-indazol-3-yl]phenoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOC3=CC=CC(C4=NNC5=C4C=C(O[C@H](C)C4=C(Cl)C=NC=C4Cl)C=C5)=C3)C(C)(C)C)C=C2)SC=N1	C49H55Cl2N7O8S	FGFR3	P22607	VHL	WO-2024137742-A1
TPD-H5FST4	WO2024137742A1_43	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOC3=CC=CC(C4=NNC5=C4C=C(O[C@H](C)C4=C(Cl)C=NC=C4Cl)C=C5)=C3)C(C)(C)C)C=C2)SC=N1	C51H59Cl2N7O9S	FGFR3	P22607	VHL	WO-2024137742-A1
TPD-BL563T	SCHEMBL30971875	(2S,4R)-1-[(2S)-2-[[2-[4-[5-[5-[(1R)-1-(3,5-dichloropyridin-4-yl)ethoxy]-1H-indazol-3-yl]pyridin-2-yl]piperazin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCN(C4=NC=C(C5=NNC6=C5C=C(O[C@H](C)C5=C(Cl)C=NC=C5Cl)C=C6)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C48H54Cl2N10O5S	FGFR3	P22607	VHL	WO-2024137742-A1
TPD-IO0FHR	SCHEMBL30971880	(2S,4R)-1-[(2S)-2-[[3-[2-[5-[5-[(1R)-1-(3,5-dichloropyridin-4-yl)ethoxy]-1H-indazol-3-yl]pyrimidin-2-yl]-2,8-diazaspiro[3.5]nonan-8-yl]-3-oxopropanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CC(=O)N3CCCC4(C3)CN(C3=NC=C(C5=NNC6=C5C=C(O[C@H](C)C5=C(Cl)C=NC=C5Cl)C=C6)C=N3)C4)C(C)(C)C)C=C2)SC=N1	C51H57Cl2N11O6S	FGFR3	P22607	VHL	WO-2024137742-A1
TPD-C09V2Z	WO2024137742A1_46	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCC(=O)N3CCCC4(C3)CN(C3=NC=C(C5=NNC6=C5C=C(O[C@H](C)C5=C(Cl)C=NC=C5Cl)C=C6)C=N3)C4)C(C)(C)C)C=C2)SC=N1	C52H59Cl2N11O6S	FGFR3	P22607	VHL	WO-2024137742-A1
TPD-RDOX1K	WO2024137742A1_48	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCN3C=C(C4=NNC5=C4C=C(O[C@H](C)C4=C(Cl)C=NC=C4CI)C=C5)C=N3)C(C)(C)C)C=C2)SC=N1	C47H55ClIN9O7S	FGFR3	P22607	VHL	WO-2024137742-A1
TPD-CXCH4T	WO2024137742A1_49	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCN3C=C(C4=NNC5=C4C=C(O[C@H](C)C4=C(Cl)C=NC=C4CI)C=C5)C=N3)C(C)(C)C)C=C2)SC=N1	C47H55ClIN9O5S	FGFR3	P22607	VHL	WO-2024137742-A1
TPD-OE5PG4	WO2024137742A1_50	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCN3C=C(C4=NNC5=CC=C(O[C@H](C)C6=C(Cl)C=NC=C6Cl)C=C54)C=N3)C(C)(C)C)C=C2)SC=N1	C43H47Cl2N9O5S	FGFR3	P22607	VHL	WO-2024137742-A1
TPD-18OLFO	WO2024137742A1_51	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCN3C=C(C4=NNC5=C4C=C(O[C@H](C)C4=C(Cl)C=NC=C4Cl)C=C5)C=N3)C(C)(C)C)C=C2)SC=N1	C47H55Cl2N9O5S	FGFR3	P22607	VHL	WO-2024137742-A1
TPD-4MDVGV	SCHEMBL27396453	5-[5-[(1R)-1-(3,5-dichloropyridin-4-yl)ethoxy]-1H-indazol-3-yl]-N-[4-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2,2-dimethyl-4-oxobutyl]pyridine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CC(C)(C)CNC(=O)C3=CC=C(C4=NNC5=C4C=C(O[C@H](C)C4=C(Cl)C=NC=C4Cl)C=C5)C=N3)C(C)(C)C)C=C2)SC=N1	C49H55Cl2N9O6S	FGFR3	P22607	VHL	WO-2024137742-A1
TPD-VYBHI0	SCHEMBL27396517	(2S,4R)-1-[(2S)-2-[[2-[1-[[[4-[5-[(1R)-1-(3,5-dichloropyridin-4-yl)ethoxy]-1H-indazol-3-yl]benzoyl]amino]methyl]cyclopentyl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CC3(CNC(=O)C4=CC=C(C5=NNC6=C5C=C(O[C@H](C)C5=C(Cl)C=NC=C5Cl)C=C6)C=C4)CCCC3)C(C)(C)C)C=C2)SC=N1	C52H58Cl2N8O6S	FGFR3	P22607	VHL	WO-2024137742-A1
TPD-1US7QU	SCHEMBL30971844	3-cyano-5-[5-[(1R)-1-(3,5-dichloropyridin-4-yl)ethoxy]-1H-indazol-3-yl]-N-[4-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2,2-dimethyl-4-oxobutyl]pyridine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CC(C)(C)CNC(=O)C3=NC=C(C4=NNC5=C4C=C(O[C@H](C)C4=C(Cl)C=NC=C4Cl)C=C5)C=C3C#N)C(C)(C)C)C=C2)SC=N1	C50H54Cl2N10O6S	FGFR3	P22607	VHL	WO-2024137742-A1
TPD-JD6YBJ	SCHEMBL30971857	(2S,4R)-1-[(2S)-2-[[2-[1-[[[4-[5-[(1R)-1-(3,5-dichloropyridin-4-yl)ethoxy]-1H-indazol-3-yl]benzoyl]amino]methyl]cyclobutyl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CC3(CNC(=O)C4=CC=C(C5=NNC6=C5C=C(O[C@H](C)C5=C(Cl)C=NC=C5Cl)C=C6)C=C4)CCC3)C(C)(C)C)C=C2)SC=N1	C51H56Cl2N8O6S	FGFR3	P22607	VHL	WO-2024137742-A1
TPD-6AKPBJ	SCHEMBL30971840	(2S,4R)-1-[(2S)-2-[[2-[1-[[[4-[5-[(1R)-1-(3,5-dichloropyridin-4-yl)ethoxy]-1H-indazol-3-yl]benzoyl]amino]methyl]cyclohexyl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CC3(CNC(=O)C4=CC=C(C5=NNC6=C5C=C(O[C@H](C)C5=C(Cl)C=NC=C5Cl)C=C6)C=C4)CCCCC3)C(C)(C)C)C=C2)SC=N1	C53H60Cl2N8O6S	FGFR3	P22607	VHL	WO-2024137742-A1
TPD-ANOAL3	SCHEMBL30971891	(2S,4R)-1-[(2S)-2-[[2-[1-[[[4-[5-[(1R)-1-(3,5-dichloropyridin-4-yl)ethoxy]-1H-indazol-3-yl]-2-methylbenzoyl]amino]methyl]cyclopentyl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C(=O)NCC2(CC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](C)C3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)CCCC2)C=CC(C2=NNC3=C2C=C(O[C@H](C)C2=C(Cl)C=NC=C2Cl)C=C3)=C1	C53H60Cl2N8O6S	FGFR3	P22607	VHL	WO-2024137742-A1
TPD-Z0GUAL	SCHEMBL27396875	(2S,4R)-1-[(2S)-2-[[2-[1-[[[2-acetamido-4-[5-[(1R)-1-(3,5-dichloropyridin-4-yl)ethoxy]-1H-indazol-3-yl]benzoyl]amino]methyl]cyclopentyl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL30971877	CC(=O)NC1=C(C(=O)NCC2(CC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](C)C3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)CCCC2)C=CC(C2=NNC3=C2C=C(O[C@H](C)C2=C(Cl)C=NC=C2Cl)C=C3)=C1	C54H61Cl2N9O7S	FGFR3	P22607	VHL	WO-2024137742-A1
TPD-C5HQ1X	SCHEMBL27396957	(2S,4R)-1-[(2S)-2-[[2-[4-[5-[5-[(1R)-1-(3,5-dichloropyridin-4-yl)ethoxy]-1H-indazol-3-yl]pyridin-2-yl]piperazin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-N-[(1S)-1-[4-(2,4-dimethyl-1,3-thiazol-5-yl)phenyl]ethyl]-4-hydroxypyrrolidine-2-carboxamide; SCHEMBL30971855	CC1=NC(C)=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCN(C4=NC=C(C5=NNC6=C5C=C(O[C@H](C)C5=C(Cl)C=NC=C5Cl)C=C6)C=C4)CC3)C(C)(C)C)C=C2)S1	C49H56Cl2N10O5S	FGFR3	P22607	VHL	WO-2024137742-A1
TPD-5VTC28	WO2024141052A1_1	3-[6-[4-[[(1S,2S)-2-[[4-[4-(6-methoxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl)phenyl]piperazin-1-yl]methyl]cyclohexyl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	COc1ccc2c(c1)CCC(c1ccccc1)C2c1ccc(N2CCN(C[C@H]3CCCC[C@@H]3CN3CCN(c4ccc5c(c4)CN(C4CCC(=O)NC4=O)C5=O)CC3)CC2)cc1	C52H62N6O4	ERα	P03372	CRBN	WO-2024141052-A1
TPD-09JN6J	WO2024141052A1_11	.	O=C1CCC(N2C(=O)c3ccc(N4CCN(C[C@H]5CCCC[C@@H]5CN5CCC(N6CCN(c7ccc([C@@H]8c9ccc(O)cc9CC[C@@H]8c8ccccc8)cc7)CC6)CC5)CC4)cc3C2=O)C(=O)N1	C56H67N7O5	ERα	P03372	CRBN	WO-2024141052-A1
TPD-C1YFKL	WO2024141052A1_12	.	O=C1CCC(N2Cc3cc(N4CCN(C[C@H]5CCCC[C@@H]5CN5CCC(N6CCN(c7ccc([C@@H]8c9ccc(O)cc9CC[C@@H]8c8ccccc8)cc7)CC6)CC5)CC4)ccc3C2=O)C(=O)N1	C56H69N7O4	ERα	P03372	CRBN	WO-2024141052-A1
TPD-YK6R4W	WO2024141052A1_13	.	O=C1CCC(N2Cc3c(NC4CN(C[C@H]5CCCC[C@@H]5CN5CCN(C6CCN(c7ccc([C@@H]8c9ccc(O)cc9CC[C@@H]8c8ccccc8)cc7)CC6)CC5)C4)cccc3C2=O)C(=O)N1	C55H67N7O4	ERα	P03372	CRBN	WO-2024141052-A1
TPD-9MSJLI	WO2024141052A1_14	.	O=C1CCC(N2Cc3c(NC4CCN(C[C@H]5CCCC[C@@H]5CN5CCN(C6CCN(c7ccc([C@@H]8c9ccc(O)cc9CC[C@@H]8c8ccccc8)cc7)CC6)CC5)CC4)cccc3C2=O)C(=O)N1	C57H71N7O4	ERα	P03372	CRBN	WO-2024141052-A1
TPD-TMV7SY	WO2024141052A1_15	3-[6-[4-[4-[[(1R,2R)-2-[[4-[1-[4-(6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl)phenyl]piperidin-4-yl]piperazin-1-yl]methyl]cyclohexyl]methyl]piperazin-1-yl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2Cc3cc(N4CCC(N5CCN(C[C@@H]6CCCC[C@H]6CN6CCN(C7CCN(c8ccc(C9c%10ccc(O)cc%10CCC9c9ccccc9)cc8)CC7)CC6)CC5)CC4)ccc3C2=O)C(=O)N1	C61H78N8O4	ERα	P03372	CRBN	WO-2024141052-A1
TPD-KLQQVF	WO2024141052A1_16	3-[6-[4-[[(1R,2R)-2-[[4-[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]piperazin-1-yl]methyl]cyclohexyl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2Cc3cc(N4CCN(C[C@@H]5CCCC[C@H]5CN5CCN(C6CCN(c7ccc([C@@H]8c9ccc(O)cc9CC[C@@H]8c8ccccc8)cc7)CC6)CC5)CC4)ccc3C2=O)C(=O)N1	C56H69N7O4	ERα	P03372	CRBN	WO-2024141052-A1
TPD-8BKXAS	WO2024141052A1_17	.	O=C1CCC(N2Cc3cc(C4CCN(C[C@@H]5CCCC[C@H]5CN5CCN(C6CCN(c7ccc([C@@H]8c9ccc(O)cc9CC[C@@H]8c8ccccc8)cc7)CC6)CC5)CC4)ccc3C2=O)C(=O)N1	C57H70N6O4	ERα	P03372	CRBN	WO-2024141052-A1
TPD-EWBJVK	WO2024141052A1_18	3-[6-[4-[4-[[(1S,2S)-2-[[4-[1-[4-(6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl)phenyl]piperidin-4-yl]piperazin-1-yl]methyl]cyclohexyl]methyl]piperazin-1-yl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2Cc3cc(N4CCC(N5CCN(C[C@H]6CCCC[C@@H]6CN6CCN(C7CCN(c8ccc(C9c%10ccc(O)cc%10CCC9c9ccccc9)cc8)CC7)CC6)CC5)CC4)ccc3C2=O)C(=O)N1	C61H78N8O4	ERα	P03372	CRBN	WO-2024141052-A1
TPD-IX1H3W	WO2024141052A1_19	.	O=C1CCC(N2Cc3cc(N4CCN(C[C@@H]5CCCC[C@H]5CN5CC6(CCN(c7ccc(C8c9ccc(O)cc9CCC8c8ccccc8)cc7)CC6)C5)CC4)ccc3C2=O)C(=O)N1	C54H64N6O4	ERα	P03372	CRBN	WO-2024141052-A1
TPD-KZYGOD	WO2024141052A1_2	3-[6-[4-[[(1S,2S)-2-[[4-[4-(6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl)phenyl]piperazin-1-yl]methyl]cyclohexyl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2Cc3cc(N4CCN(C[C@H]5CCCC[C@@H]5CN5CCN(c6ccc(C7c8ccc(O)cc8CCC7c7ccccc7)cc6)CC5)CC4)ccc3C2=O)C(=O)N1	C51H60N6O4	ERα	P03372	CRBN	WO-2024141052-A1
TPD-FWV4XY	WO2024141052A1_20	3-[6-[4-[[(1R,2R)-2-[[3-[4-(6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl)phenyl]-3,9-diazaspiro[5.5]undecan-9-yl]methyl]cyclohexyl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2Cc3cc(N4CCN(C[C@@H]5CCCC[C@H]5CN5CCC6(CC5)CCN(c5ccc(C7c8ccc(O)cc8CCC7c7ccccc7)cc5)CC6)CC4)ccc3C2=O)C(=O)N1	C56H68N6O4	ERα	P03372	CRBN	WO-2024141052-A1
TPD-QJ51VA	WO2024141052A1_21	3-[6-[4-[[(1S,2S)-2-[[3-[4-(6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl)phenyl]-3,9-diazaspiro[5.5]undecan-9-yl]methyl]cyclohexyl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2Cc3cc(N4CCN(C[C@H]5CCCC[C@@H]5CN5CCC6(CC5)CCN(c5ccc(C7c8ccc(O)cc8CCC7c7ccccc7)cc5)CC6)CC4)ccc3C2=O)C(=O)N1	C56H68N6O4	ERα	P03372	CRBN	WO-2024141052-A1
TPD-CU6GIS	WO2024141052A1_22	.	O=C1CCC(N2Cc3cc(N4CCN(C[C@@H]5CCCC[C@H]5CN5CCN(C6CN(c7ccc([C@@H]8c9ccc(O)cc9CC[C@@H]8c8ccccc8)cc7)C6)CC5)CC4)ccc3C2=O)C(=O)N1	C54H65N7O4	ERα	P03372	CRBN	WO-2024141052-A1
TPD-2736PA	WO2024141052A1_23	3-[7-[[(1S,2S)-2-[[4-[4-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperazin-1-yl]piperidin-1-yl]methyl]cyclohexyl]methylamino]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2Cc3c(NC[C@H]4CCCC[C@@H]4CN4CCC(N5CCN(c6ccc([C@@H]7c8ccc(O)cc8CC[C@@H]7c7ccccc7)cc6)CC5)CC4)cccc3C2=O)C(=O)N1	C52H62N6O4	ERα	P03372	CRBN	WO-2024141052-A1
TPD-3NAB72	WO2024141052A1_24	3-[6-[4-[4-[[(1S,2S)-2-[[4-[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]piperazin-1-yl]methyl]cyclohexyl]methyl]piperazin-1-yl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2Cc3cc(N4CCC(N5CCN(C[C@H]6CCCC[C@@H]6CN6CCN(C7CCN(c8ccc([C@@H]9c%10ccc(O)cc%10CC[C@@H]9c9ccccc9)cc8)CC7)CC6)CC5)CC4)ccc3C2=O)C(=O)N1	C61H78N8O4	ERα	P03372	CRBN	WO-2024141052-A1
TPD-WTR4K4	WO2024141052A1_25	3-[6-[4-[4-[[(1R,2R)-2-[[4-[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]piperazin-1-yl]methyl]cyclohexyl]methyl]piperazin-1-yl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2Cc3cc(N4CCC(N5CCN(C[C@@H]6CCCC[C@H]6CN6CCN(C7CCN(c8ccc([C@@H]9c%10ccc(O)cc%10CC[C@@H]9c9ccccc9)cc8)CC7)CC6)CC5)CC4)ccc3C2=O)C(=O)N1	C61H78N8O4	ERα	P03372	CRBN	WO-2024141052-A1
TPD-R9RW9X	WO2024141052A1_26	.	O=C1CCC(N2Cc3cc(N4CCN(C[C@@H]5CCCC[C@H]5CN5CC(N6CCC(c7ccc(C8c9ccc(O)cc9CCC8c8ccccc8)cc7)CC6)C5)CC4)ccc3C2=O)C(=O)N1	C55H66N6O4	ERα	P03372	CRBN	WO-2024141052-A1
TPD-S7H23B	WO2024141052A1_27	.	O=C1CCC(N2Cc3cc(N4CCN(C[C@H]5CCCC[C@@H]5CN5CCC(c6ccc([C@@H]7c8ccc(O)cc8CC[C@@H]7c7ccccc7)cc6)CC5)CC4)ccc3C2=O)C(=O)N1	C52H61N5O4	ERα	P03372	CRBN	WO-2024141052-A1
TPD-J2DYV0	WO2024141052A1_28	.	O=C1CCC(N2Cc3cc(N4CCN(C[C@H]5CCCC[C@@H]5CN5CCN(c6ccc([C@@H]7c8ccc(O)cc8CC[C@@H]7c7ccccc7)cc6)CC5)CC4)ccc3C2=O)C(=O)N1	C51H60N6O4	ERα	P03372	CRBN	WO-2024141052-A1
TPD-41X2Y1	WO2024141052A1_29	.	O=C1CCC(N2C(=O)c3ccc(N4CCN(C[C@H]5CCCC[C@@H]5CN5CCN(C6CCN(c7ccc([C@@H]8c9ccc(O)cc9CC[C@@H]8c8ccccc8)cc7)CC6)CC5)CC4)cc3C2=O)C(=O)N1	C56H67N7O5	ERα	P03372	CRBN	WO-2024141052-A1
TPD-ABTP9W	WO2024141052A1_3	3-[6-[4-[[(1R,2R)-2-[[4-[4-(6-methoxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl)phenyl]piperazin-1-yl]methyl]cyclohexyl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	COc1ccc2c(c1)CCC(c1ccccc1)C2c1ccc(N2CCN(C[C@@H]3CCCC[C@H]3CN3CCN(c4ccc5c(c4)CN(C4CCC(=O)NC4=O)C5=O)CC3)CC2)cc1	C52H62N6O4	ERα	P03372	CRBN	WO-2024141052-A1
TPD-MR94BC	WO2024141052A1_30	.	O=C1CCC(N2Cc3cc(N4CCN(C[C@H]5CCCC[C@@H]5CNC5CCN(c6ccc([C@@H]7c8ccc(O)cc8CC[C@@H]7c7ccccc7)cc6)CC5)CC4)ccc3C2=O)C(=O)N1	C52H62N6O4	ERα	P03372	CRBN	WO-2024141052-A1
TPD-SEXNU8	WO2024141052A1_31	3-[6-[4-[[(1R,2R)-2-[[(3S)-4-[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]-3-methylpiperazin-1-yl]methyl]cyclohexyl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C[C@H]1CN(C[C@@H]2CCCC[C@H]2CN2CCN(c3ccc4c(c3)CN(C3CCC(=O)NC3=O)C4=O)CC2)CCN1C1CCN(c2ccc([C@@H]3c4ccc(O)cc4CC[C@@H]3c3ccccc3)cc2)CC1	C57H71N7O4	ERα	P03372	CRBN	WO-2024141052-A1
TPD-1E917X	WO2024141052A1_32	3-[4-[4-[[(1R,2R)-2-[[4-[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]piperazin-1-yl]methyl]cyclohexyl]methyl]piperazin-1-yl]anilino]piperidine-2,6-dione	O=C1CCC(Nc2ccc(N3CCN(C[C@@H]4CCCC[C@H]4CN4CCN(C5CCN(c6ccc([C@@H]7c8ccc(O)cc8CC[C@@H]7c7ccccc7)cc6)CC5)CC4)CC3)cc2)C(=O)N1	C54H69N7O3	ERα	P03372	CRBN	WO-2024141052-A1
TPD-MNGW3U	WO2024141052A1_33	3-[6-[4-[(1R,2R)-2-[4-[[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperazine-1-carbonyl]cyclohexanecarbonyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2Cc3cc(N4CCN(C(=O)[C@@H]5CCCC[C@H]5C(=O)N5CCN(CC6CCN(c7ccc([C@@H]8c9ccc(O)cc9CC[C@@H]8c8ccccc8)cc7)CC6)CC5)CC4)ccc3C2=O)C(=O)N1	C57H67N7O6	ERα	P03372	CRBN	WO-2024141052-A1
TPD-XX0XVD	WO2024141052A1_34	3-[6-[4-[(1S,2S)-2-[4-[[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperazine-1-carbonyl]cyclohexanecarbonyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2Cc3cc(N4CCN(C(=O)[C@H]5CCCC[C@@H]5C(=O)N5CCN(CC6CCN(c7ccc([C@@H]8c9ccc(O)cc9CC[C@@H]8c8ccccc8)cc7)CC6)CC5)CC4)ccc3C2=O)C(=O)N1	C57H67N7O6	ERα	P03372	CRBN	WO-2024141052-A1
TPD-5ZGYQO	WO2024141052A1_35	3-[6-[4-[[(1S,2S)-2-[[4-[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]piperazin-1-yl]methyl]cyclohexyl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2Cc3cc(N4CCN(C[C@H]5CCCC[C@@H]5CN5CCN(C6CCN(c7ccc([C@@H]8c9ccc(O)cc9CC[C@@H]8c8ccccc8)cc7)CC6)CC5)CC4)ccc3C2=O)C(=O)N1	C56H69N7O4	ERα	P03372	CRBN	WO-2024141052-A1
TPD-OQ86YJ	WO2024141052A1_37	.	O=C1CCC(N2Cc3cc(C4CN(C[C@@H]5CCCC[C@H]5CN5CCN(c6ccc([C@@H]7c8ccc(O)cc8CC[C@@H]7c7ccccc7)cc6)CC5)C4)ccc3C2=O)C(=O)N1	C50H57N5O4	ERα	P03372	CRBN	WO-2024141052-A1
TPD-LXXUF9	WO2024141052A1_38	3-[6-[1-[[(1R,2R)-2-[[4-[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]piperazin-1-yl]methyl]cyclohexyl]methyl]azetidin-3-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2Cc3cc(C4CN(C[C@@H]5CCCC[C@H]5CN5CCN(C6CCN(c7ccc([C@@H]8c9ccc(O)cc9CC[C@@H]8c8ccccc8)cc7)CC6)CC5)C4)ccc3C2=O)C(=O)N1	C55H66N6O4	ERα	P03372	CRBN	WO-2024141052-A1
TPD-11VRPW	WO2024141052A1_39	3-[7-[[1-[[(1S,2S)-2-[[4-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperazin-1-yl]methyl]cyclohexyl]methyl]piperidin-4-yl]amino]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2Cc3c(NC4CCN(C[C@H]5CCCC[C@@H]5CN5CCN(c6ccc([C@@H]7c8ccc(O)cc8CC[C@@H]7c7ccccc7)cc6)CC5)CC4)cccc3C2=O)C(=O)N1	C52H62N6O4	ERα	P03372	CRBN	WO-2024141052-A1
TPD-U2LML7	WO2024141052A1_4	3-[6-[4-[[(1R,2R)-2-[[4-[4-(6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl)phenyl]piperazin-1-yl]methyl]cyclohexyl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2Cc3cc(N4CCN(C[C@@H]5CCCC[C@H]5CN5CCN(c6ccc(C7c8ccc(O)cc8CCC7c7ccccc7)cc6)CC5)CC4)ccc3C2=O)C(=O)N1	C51H60N6O4	ERα	P03372	CRBN	WO-2024141052-A1
TPD-QYTBKU	WO2024141052A1_40	3-[7-[[(1S,2S)-2-[[4-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperazin-1-yl]methyl]cyclohexyl]methylamino]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2Cc3c(NC[C@H]4CCCC[C@@H]4CN4CCN(c5ccc([C@@H]6c7ccc(O)cc7CC[C@@H]6c6ccccc6)cc5)CC4)cccc3C2=O)C(=O)N1	C47H53N5O4	ERα	P03372	CRBN	WO-2024141052-A1
TPD-8LNAIG	WO2024141052A1_41	3-[6-[1-[[(1S,2S)-2-[[4-[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]piperazin-1-yl]methyl]cyclohexyl]methyl]piperidin-4-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2Cc3cc(C4CCN(C[C@H]5CCCC[C@@H]5CN5CCN(C6CCN(c7ccc([C@@H]8c9ccc(O)cc9CC[C@@H]8c8ccccc8)cc7)CC6)CC5)CC4)ccc3C2=O)C(=O)N1	C57H70N6O4	ERα	P03372	CRBN	WO-2024141052-A1
TPD-S243FS	WO2024141052A1_42	2-(2,6-dioxopiperidin-3-yl)-5-[1-[[(1R,2R)-2-[[4-[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]piperazin-1-yl]methyl]cyclohexyl]methyl]piperidin-4-yl]isoindole-1,3-dione	O=C1CCC(N2C(=O)c3ccc(C4CCN(C[C@@H]5CCCC[C@H]5CN5CCN(C6CCN(c7ccc([C@@H]8c9ccc(O)cc9CC[C@@H]8c8ccccc8)cc7)CC6)CC5)CC4)cc3C2=O)C(=O)N1	C57H68N6O5	ERα	P03372	CRBN	WO-2024141052-A1
TPD-DFD1QK	WO2024141052A1_43	.	COc1ccc(C2CCc3cc(O)ccc3C2c2ccc(N3CCN(C[C@@H]4CCCC[C@H]4CN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)CC3)cc2)cc1	C52H62N6O5	ERα	P03372	CRBN	WO-2024141052-A1
TPD-2OQ13N	WO2024141052A1_44	.	O=C1CCC(N2Cc3cc(C4CCN(C[C@@H]5CCCC[C@H]5CN5CCN(c6ccc([C@@H]7c8ccc(O)cc8CC[C@@H]7c7ccccc7)cc6)CC5)CC4)ccc3C2=O)C(=O)N1	C52H61N5O4	ERα	P03372	CRBN	WO-2024141052-A1
TPD-0IMXLG	WO2024141052A1_45	.	O=C1CCC(N2Cc3cc(N4CCN(C[C@@H]5CCCC[C@H]5CN5CCN(c6ccc(C7c8ccc(O)cc8CCC7c7ccc(C(F)(F)F)cc7)cc6)CC5)CC4)ccc3C2=O)C(=O)N1	C52H59F3N6O4	ERα	P03372	CRBN	WO-2024141052-A1
TPD-A8UMBU	WO2024141052A1_46	.	COc1cc(N2CCN(C[C@@H]3CCCC[C@H]3CN3CCN(c4ccc([C@@H]5c6ccc(O)cc6CC[C@@H]5c5ccccc5)cc4)CC3)CC2)ccc1N1CCC(=O)NC1=O	C49H60N6O4	ERα	P03372	CRBN	WO-2024141052-A1
TPD-13XH1V	WO2024141052A1_47	.	O=C1CCC(N2Cc3cc(N4CCN(C[C@H]5CCCC[C@@H]5CN5CCC(N6CCC(c7ccc([C@@H]8c9ccc(O)cc9CC[C@@H]8c8ccccc8)cc7)CC6)CC5)CC4)ccc3C2=O)C(=O)N1	C57H70N6O4	ERα	P03372	CRBN	WO-2024141052-A1
TPD-GNY64Z	WO2024141052A1_48	1-[4-[4-[[(1R,2R)-2-[[4-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperazin-1-yl]methyl]cyclohexyl]methyl]piperazin-1-yl]phenyl]-1,3-diazinane-2,4-dione	O=C1CCN(c2ccc(N3CCN(C[C@@H]4CCCC[C@H]4CN4CCN(c5ccc([C@@H]6c7ccc(O)cc7CC[C@@H]6c6ccccc6)cc5)CC4)CC3)cc2)C(=O)N1	C48H58N6O3	ERα	P03372	CRBN	WO-2024141052-A1
TPD-5D75WM	WO2024141052A1_49	1-[4-[1-[[(1R,2R)-2-[[4-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperazin-1-yl]methyl]cyclohexyl]methyl]piperidin-4-yl]phenyl]-1,3-diazinane-2,4-dione	O=C1CCN(c2ccc(C3CCN(C[C@@H]4CCCC[C@H]4CN4CCN(c5ccc([C@@H]6c7ccc(O)cc7CC[C@@H]6c6ccccc6)cc5)CC4)CC3)cc2)C(=O)N1	C49H59N5O3	ERα	P03372	CRBN	WO-2024141052-A1
TPD-GQXWKR	WO2024141052A1_5	3-[6-[4-[[(1R,2R)-2-[[4-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperazin-1-yl]methyl]cyclohexyl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2Cc3cc(N4CCN(C[C@@H]5CCCC[C@H]5CN5CCN(c6ccc([C@@H]7c8ccc(O)cc8CC[C@@H]7c7ccccc7)cc6)CC5)CC4)ccc3C2=O)C(=O)N1	C51H60N6O4	ERα	P03372	CRBN	WO-2024141052-A1
TPD-LMHLFU	WO2024141052A1_50	.	Cc1cc(N2CCN(C[C@@H]3CCCC[C@H]3CN3CCN(c4ccc([C@@H]5c6ccc(O)cc6CC[C@@H]5c5ccccc5)cc4)CC3)CC2)ccc1N1CCC(=O)NC1=O	C49H60N6O3	ERα	P03372	CRBN	WO-2024141052-A1
TPD-FD6EDN	WO2024141052A1_52	.	O=C1CCC(N2Cc3cc(N4CCN(C[C@@H]5CCCC[C@H]5CN5CCC(N6CCN(c7ccc([C@@H]8c9ccc(O)cc9CC[C@@H]8c8ccccc8)cc7)CC6)CC5)CC4)ccc3C2=O)C(=O)N1	C56H69N7O4	ERα	P03372	CRBN	WO-2024141052-A1
TPD-UFLWQK	WO2024141052A1_53	3-[6-[4-[[(1R,2R)-2-[[4-[4-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-1-yl]piperidin-1-yl]methyl]cyclohexyl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2Cc3cc(N4CCN(C[C@@H]5CCCC[C@H]5CN5CCC(N6CCC(c7ccc([C@@H]8c9ccc(O)cc9CC[C@@H]8c8ccccc8)cc7)CC6)CC5)CC4)ccc3C2=O)C(=O)N1	C57H70N6O4	ERα	P03372	CRBN	WO-2024141052-A1
TPD-AXR5UW	WO2024141052A1_54	.	O=C1CCC(N2Cc3cc(N4CCN(C[C@@H]5CCCC[C@H]5CN5CCN(c6ccc(C7c8ccc(O)cc8CCC7c7ccccc7)cc6F)CC5)CC4)ccc3C2=O)C(=O)N1	C51H59FN6O4	ERα	P03372	CRBN	WO-2024141052-A1
TPD-6CUNEY	WO2024141052A1_55	.	Cc1cc(C2CCN(C[C@H]3CCCC[C@@H]3CN3CCN(c4ccc([C@@H]5c6ccc(O)cc6CC[C@@H]5c5ccccc5)cc4)CC3)CC2)ccc1N1CCC(=O)NC1=O	C50H61N5O3	ERα	P03372	CRBN	WO-2024141052-A1
TPD-878IJ7	WO2024141052A1_56	.	CCc1cc(N2CCN(C[C@@H]3CCCC[C@H]3CN3CCN(c4ccc([C@@H]5c6ccc(O)cc6CC[C@@H]5c5ccccc5)cc4)CC3)CC2)ccc1N1CCC(=O)NC1=O	C50H62N6O3	ERα	P03372	CRBN	WO-2024141052-A1
TPD-SBJ191	WO2024141052A1_57	.	O=C1CCN(c2ccc(N3CCN(C[C@@H]4CCCC[C@H]4CN4CCN(c5ccc([C@@H]6c7ccc(O)cc7CC[C@@H]6c6ccccc6)cc5)CC4)CC3)c3ccccc23)C(=O)N1	C52H60N6O3	ERα	P03372	CRBN	WO-2024141052-A1
TPD-Q8AYRP	WO2024141052A1_58	.	O=C1CCC(N2Cc3cc(N4CCN(C(=O)[C@H]5CCCN5CC5CCN(c6ccc(C7c8ccc(O)cc8CCC7c7ccccc7)cc6)CC5)CC4)ccc3C2=O)C(=O)N1	C50H56N6O5	ERα	P03372	CRBN	WO-2024141052-A1
TPD-PCEIJP	WO2024141052A1_59	.	O=C1CCC(N2C(=O)c3ccc(N4CCN(C[C@@H]5CCCC[C@H]5CN5CCN(C6CCN(c7ccc([C@@H]8c9ccc(O)cc9CC[C@@H]8c8ccccc8)cc7)CC6)CC5)CC4)cc3C2=O)C(=O)N1	C56H67N7O5	ERα	P03372	CRBN	WO-2024141052-A1
TPD-EV0R3W	WO2024141052A1_6	(3R)-3-[6-[4-[[(1R,2R)-2-[[4-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperazin-1-yl]methyl]cyclohexyl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CC[C@@H](N2Cc3cc(N4CCN(C[C@@H]5CCCC[C@H]5CN5CCN(c6ccc([C@@H]7c8ccc(O)cc8CC[C@@H]7c7ccccc7)cc6)CC5)CC4)ccc3C2=O)C(=O)N1	C51H60N6O4	ERα	P03372	CRBN	WO-2024141052-A1
TPD-QFA2CM	WO2024141052A1_60	.	O=C1CCC(N2C(=O)c3ccc(N4CCN(C[C@@H]5CCCC[C@H]5CN5CCC(N6CCN(c7ccc([C@@H]8c9ccc(O)cc9CC[C@@H]8c8ccccc8)cc7)CC6)CC5)CC4)cc3C2=O)C(=O)N1	C56H67N7O5	ERα	P03372	CRBN	WO-2024141052-A1
TPD-4CB17O	WO2024141052A1_61	.	Cc1cc(N2CCN(C(=O)[C@@H]3CCCC[C@H]3C(=O)N3CCN(CC4CCN(c5ccc([C@@H]6c7ccc(O)cc7CC[C@@H]6c6ccccc6)cc5)CC4)CC3)CC2)ccc1N1CCC(=O)NC1=O	C55H67N7O5	ERα	P03372	CRBN	WO-2024141052-A1
TPD-LZUCUZ	WO2024141052A1_62	.	COc1ccc(C2CCc3cc(O)ccc3C2c2ccc(N3CCN(C[C@@H]4CCCC[C@H]4CN4CCN(c5ccc(C6CCC(=O)NC6=O)cc5)CC4)CC3)cc2)cc1	C50H61N5O4	ERα	P03372	CRBN	WO-2024141052-A1
TPD-VQ4QTK	WO2024141052A1_63	3-[4-[4-[[(1R,2R)-2-[[4-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperazin-1-yl]methyl]cyclohexyl]methyl]piperazin-1-yl]phenyl]piperidine-2,6-dione	O=C1CCC(c2ccc(N3CCN(C[C@@H]4CCCC[C@H]4CN4CCN(c5ccc([C@@H]6c7ccc(O)cc7CC[C@@H]6c6ccccc6)cc5)CC4)CC3)cc2)C(=O)N1	C49H59N5O3	ERα	P03372	CRBN	WO-2024141052-A1
TPD-P33RW5	WO2024141052A1_64	.	O=C1CCC(N2Cc3cc(N4CCC(NC[C@H]5CCCC[C@@H]5CN5CCN(c6ccc([C@@H]7c8ccc(O)cc8CC[C@@H]7c7ccccc7)cc6)CC5)CC4)ccc3C2=O)C(=O)N1	C52H62N6O4	ERα	P03372	CRBN	WO-2024141052-A1
TPD-TQSWGE	WO2024141052A1_65	.	C[C@@H]1CN(C2CCN(c3ccc([C@@H]4c5ccc(O)cc5CC[C@@H]4c4ccccc4)cc3)CC2)CCN1C[C@@H]1CCCC[C@H]1CN1CCN(c2ccc3c(c2)CN(C2CCC(=O)NC2=O)C3=O)CC1	C57H71N7O4	ERα	P03372	CRBN	WO-2024141052-A1
TPD-XWGYR5	WO2024141052A1_66	.	Cc1cc(N2CCN(C[C@@H]3CCCC[C@H]3CN3CCN(c4ccc([C@@H]5c6ccc(O)cc6CC[C@@H]5c5ccccc5)cc4)CC3)CC2)ccc1C1CCC(=O)NC1=O	C50H61N5O3	ERα	P03372	CRBN	WO-2024141052-A1
TPD-M8NHYO	WO2024141052A1_67	.	Cc1cc(C2CCN(C[C@@H]3CCCC[C@H]3CN3CCN(c4ccc([C@@H]5c6ccc(O)cc6CC[C@@H]5c5ccccc5)cc4)CC3)CC2)ccc1N1CCC(=O)NC1=O	C50H61N5O3	ERα	P03372	CRBN	WO-2024141052-A1
TPD-A51K3O	WO2024141052A1_7	(3S)-3-[6-[4-[[(1R,2R)-2-[[4-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperazin-1-yl]methyl]cyclohexyl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CC[C@H](N2Cc3cc(N4CCN(C[C@@H]5CCCC[C@H]5CN5CCN(c6ccc([C@@H]7c8ccc(O)cc8CC[C@@H]7c7ccccc7)cc6)CC5)CC4)ccc3C2=O)C(=O)N1	C51H60N6O4	ERα	P03372	CRBN	WO-2024141052-A1
TPD-E3BLQ3	WO2024141052A1_8	.	O=C1CCC(N2Cc3cc(N4CCN(C[C@H]5CCCC[C@@H]5CN5CC(N6CCN(c7ccc(C8c9ccc(O)cc9CCC8c8ccccc8)cc7)CC6)C5)CC4)ccc3C2=O)C(=O)N1	C54H65N7O4	ERα	P03372	CRBN	WO-2024141052-A1
TPD-UZ0IDN	WO2024141052A1_9	.	O=C1CCC(N2Cc3cc(N4CCN(C(=O)[C@H]5CCCCN5CC5CCN(c6ccc([C@@H]7c8ccc(O)cc8CC[C@@H]7c7ccccc7)cc6)CC5)CC4)ccc3C2=O)C(=O)N1	C51H58N6O5	ERα	P03372	CRBN	WO-2024141052-A1
TPD-HR3U8W	WO2024141052A1_II1	3-[6-[4-[[(1S,2S)-2-[[4-[5-[(1R,3R)-2-(2-fluoro-2-methylpropyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyrimidin-2-yl]piperazin-1-yl]methyl]cyclohexyl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C[C@@H]1Cc2c([nH]c3ccccc23)[C@@H](c2cnc(N3CCN(C[C@H]4CCCC[C@@H]4CN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)CC3)nc2)N1CC(C)(C)F	C49H63FN10O3	ERα	P03372	CRBN	WO-2024141052-A1
TPD-C2RTHR	WO2024141052A1_II10	.	C[C@@H]1Cc2c(ccc3[nH]ncc23)[C@@H](c2ccc(N3CCN(C[C@H]4CCCC[C@@H]4CN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)CC3)cn2)N1CC(F)(F)F	C47H57F3N10O3	ERα	P03372	CRBN	WO-2024141052-A1
TPD-VZNOM6	WO2024141052A1_II11	.	C[C@@H]1Cc2c([nH]c3ccccc23)[C@@H](c2c(F)cc(N3CCN(C4CCN(C[C@@H]5CCCC[C@H]5CN5CCN(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC5)CC4)CC3)cc2F)N1CC(C)(C)F	C56H72F3N9O3	ERα	P03372	CRBN	WO-2024141052-A1
TPD-ZHGHDM	WO2024141052A1_II12	.	C[C@@H]1Cc2c([nH]c3ccccc23)[C@@H](c2c(F)cc(N3CCN(C4CCN(C[C@H]5CCCC[C@@H]5CN5CCN(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC5)CC4)CC3)cc2F)N1CC(C)(C)F	C56H72F3N9O3	ERα	P03372	CRBN	WO-2024141052-A1
TPD-JQHLPQ	WO2024141052A1_II13	.	C[C@@H]1Cc2c(ccc3[nH]ncc23)[C@@H](c2ccc(N3CCN(C4CCN(C[C@@H]5CCCC[C@H]5CN5CCN(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC5)CC4)CC3)cn2)N1CC(F)(F)F	C52H66F3N11O3	ERα	P03372	CRBN	WO-2024141052-A1
TPD-FRMDUL	WO2024141052A1_II14	.	C[C@@H]1Cc2c(ccc3[nH]ncc23)[C@@H](c2ccc(N3CCN(C4CCN(C[C@H]5CCCC[C@@H]5CN5CCN(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC5)CC4)CC3)cn2)N1CC(F)(F)F	C52H66F3N11O3	ERα	P03372	CRBN	WO-2024141052-A1
TPD-GBQTNK	WO2024141052A1_II2	3-[6-[4-[[(1R,2R)-2-[[4-[4-[[2-[2-(1,1-difluoroethyl)-4-fluorophenyl]-6-methoxy-1-benzothiophen-3-yl]oxy]phenyl]piperazin-1-yl]methyl]cyclohexyl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	COc1ccc2c(Oc3ccc(N4CCN(C[C@@H]5CCCC[C@H]5CN5CCN(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3)c(-c3ccc(F)cc3C(C)(F)F)sc2c1	C52H57F3N6O5S	ERα	P03372	CRBN	WO-2024141052-A1
TPD-CYKGHO	WO2024141052A1_II3	3-[6-[4-[[(1S,2S)-2-[[4-[4-[[2-[2-(1,1-difluoroethyl)-4-fluorophenyl]-6-methoxy-1-benzothiophen-3-yl]oxy]phenyl]piperazin-1-yl]methyl]cyclohexyl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	COc1ccc2c(Oc3ccc(N4CCN(C[C@H]5CCCC[C@@H]5CN5CCN(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3)c(-c3ccc(F)cc3C(C)(F)F)sc2c1	C52H57F3N6O5S	ERα	P03372	CRBN	WO-2024141052-A1
TPD-O89L7A	WO2024141052A1_II4	3-[6-[4-[[(1S,2S)-2-[[4-[4-[[2-[2-(1,1-difluoroethyl)-4-fluorophenyl]-6-hydroxy-1-benzothiophen-3-yl]oxy]phenyl]piperazin-1-yl]methyl]cyclohexyl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CC(F)(F)c1cc(F)ccc1-c1sc2cc(O)ccc2c1Oc1ccc(N2CCN(C[C@H]3CCCC[C@@H]3CN3CCN(c4ccc5c(c4)CN(C4CCC(=O)NC4=O)C5=O)CC3)CC2)cc1	C51H55F3N6O5S	ERα	P03372	CRBN	WO-2024141052-A1
TPD-J3GPM3	WO2024141052A1_II5	3-[6-[4-[[(1R,2R)-2-[[4-[4-[[2-[2-(1,1-difluoroethyl)-4-fluorophenyl]-6-hydroxy-1-benzothiophen-3-yl]oxy]phenyl]piperazin-1-yl]methyl]cyclohexyl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CC(F)(F)c1cc(F)ccc1-c1sc2cc(O)ccc2c1Oc1ccc(N2CCN(C[C@@H]3CCCC[C@H]3CN3CCN(c4ccc5c(c4)CN(C4CCC(=O)NC4=O)C5=O)CC3)CC2)cc1	C51H55F3N6O5S	ERα	P03372	CRBN	WO-2024141052-A1
TPD-MZ5U3I	WO2024141052A1_II6	3-[6-[4-[[(1R,2R)-2-[[4-[5-[(1R,3R)-2-(2-fluoro-2-methylpropyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]pyrimidin-2-yl]piperazin-1-yl]methyl]cyclohexyl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C[C@@H]1Cc2c([nH]c3ccccc23)[C@@H](c2cnc(N3CCN(C[C@@H]4CCCC[C@H]4CN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)CC3)nc2)N1CC(C)(C)F	C49H63FN10O3	ERα	P03372	CRBN	WO-2024141052-A1
TPD-JR28GN	WO2024141052A1_II7	.	C[C@@H]1Cc2c([nH]c3ccccc23)[C@@H](c2c(F)cc(N3CCN(C[C@@H]4CCCC[C@H]4CN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)CC3)cc2F)N1CC(C)(C)F	C51H63F3N8O3	ERα	P03372	CRBN	WO-2024141052-A1
TPD-IC9LGU	WO2024141052A1_II8	.	C[C@@H]1Cc2c([nH]c3ccccc23)[C@@H](c2c(F)cc(N3CCN(C[C@H]4CCCC[C@@H]4CN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)CC3)cc2F)N1CC(C)(C)F	C51H63F3N8O3	ERα	P03372	CRBN	WO-2024141052-A1
TPD-47XPOR	WO2024141052A1_II9	.	C[C@@H]1Cc2c(ccc3[nH]ncc23)[C@@H](c2ccc(N3CCN(C[C@@H]4CCCC[C@H]4CN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)CC3)cn2)N1CC(F)(F)F	C47H57F3N10O3	ERα	P03372	CRBN	WO-2024141052-A1
TPD-9VF2WB	WO2024148257A1_YX-2-14	.	CC(C)(C)C1=CC=C(C2=N[C@](C)(C3=CC=C(Cl)C=C3)[C@@](C)(C3=CC=C(Cl)C=C3)N2C(=O)N2CCN(CC(=O)NCCOCCOCCOCCNC(=O)CN3CCN(C(=O)N4C(C5=CC=C(C(C)(C)C)C=C5O)=N[C@](C)(C5=CC=C(Cl)C=C5)[C@@]4(C)C4=CC=C(Cl)C=C4)CC3)CC2)C(O)=C1	C76H92Cl4N10O9	MDM2	Q00987	MDM2	WO-2024148257-A1
TPD-INWUCR	WO2024148257A1_YX-2-18	.	CCOC1=CC(C(C)(C)C)=CC=C1C1=N[C@@](C)(C2=CC=C(Cl)C=C2)[C@](C)(C2=CC=C(Cl)C=C2)N1C(=O)N1CCN(CC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)CC1	C58H70Cl2N8O6S	MDM2	Q00987	VHL	WO-2024148257-A1
TPD-4PJWQY	WO2024148257A1_YX-2-20	.	CCOC1=CC(C(C)(C)C)=CC=C1C1=N[C@](C)(C2=CC=C(Cl)C=C2)[C@@](C)(C2=CC=C(Cl)C=C2)N1C(=O)N1CCN(CC(=O)NCCCNC(=O)COC2=CC3=C(C=C2)C[C@H](C(=O)N[C@H]2CCCC4=C2C=CC=C4)N(C(=O)[C@@H](NC(=O)[C@@H](C)NC)C(C)(C)C)C3)CC1	C71H90Cl2N10O8	MDM2	Q00987	MDM2	WO-2024148257-A1
TPD-PRWZ85	WO2024148257A1_YX-2-228	.	CCOC1=CC(C(C)(C)C)=CC=C1C1=N[C@](C)(C2=CC=C(Cl)C=C2)[C@@](C)(C2=CC=C(Cl)C=C2)N1C(=O)N1CCN(CC(=O)NCCOCCOCCNC(=O)CN2CCN(C(=O)N3C(C4=CC=C(C(C)(C)C)C=C4OCC)=N[C@](C)(C4=CC=C(Cl)C=C4)[C@@]3(C)C3=CC=C(Cl)C=C3)CC2)CC1	C78H96Cl4N10O8	MDM2	Q00987	MDM2	WO-2024148257-A1
TPD-HL0E7N	WO2024148257A1_YX-2-230	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCNC(=O)CN3CCN(C(=O)N4C(C5=C(O)C=C(C(C)(C)C)C=C5)=N[C@](C)(C5=CC=C(Cl)C=C5)[C@](C)(CC5=CC=C(Cl)C=C5)[C@H]4C4=CC=C(Cl)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C72H88Cl3N9O10S	MDM2	Q00987	VHL	WO-2024148257-A1
TPD-ZCZGGA	SCHEMBL24718329	2-[6-[[5-chloro-2-[4-[[(5S)-2-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]-2,7-diazaspiro[4.4]nonan-7-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894122	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CC[C@]6(CCN(C7=CC=C8C(=O)N([C@H]9CCC(=O)NC9=O)CC8=C7)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H53ClN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-ENVV2V	WO2024151557A1_2	.	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CC[C@@]6(CCN(C7=CC=C8C(=O)N([C@@H]9CCC(=O)NC9=O)CC8=C7)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H53ClN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-E9B1F7	SCHEMBL24717908	2-[6-[[5-chloro-2-[7-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]-2,7-diazaspiro[4.4]nonan-2-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894151	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC5(CCN(CC6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7)CC6)C5)C4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H53ClN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-X0UBK6	SCHEMBL24717907	2-[6-[[5-chloro-2-[7-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]-2,7-diazaspiro[4.4]nonan-2-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894231	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC5(CCN(CC6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)C5)C4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H51ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-FV61A7	SCHEMBL24717637	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-1-ethyl-2-oxoquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30798354	CCN1C(=O)C(OCC(=O)NC)=CC2=C1C=CC(NC1=NC(N3CCC(O[C@H]4C[C@@H](N5CCC(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)C4)CC3)=NC=C1Cl)=C2	C45H50ClN9O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-YNHRDP	SCHEMBL27219533	2-[6-[[5-chloro-2-[4-[[7-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894221	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCN(CC5CC6(CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H53ClN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-46OIAB	SCHEMBL24717868	2-[6-[[5-chloro-2-[4-[[7-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894335	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCN(CC5CC6(CCN(C7=C8CN(C9CCC(=O)NC9=O)C(=O)C8=CC=C7)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H53ClN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-6P75IM	SCHEMBL24717828	2-[6-[[5-chloro-2-[4-[2-[7-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]-2,7-diazaspiro[3.5]nonan-2-yl]propan-2-yl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894139	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(C(C)(C)N5CC6(CCN(C7=C8CN(C9CCC(=O)NC9=O)C(=O)C8=CC=C7)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H57ClN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-1DE2PO	SCHEMBL24717829	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-5-methoxy-1,3-dioxoisoindol-4-yl]-2-azaspiro[3.5]nonan-7-yl]methyl]piperazin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894216	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCN(CC5CCC6(CC5)CN(C5=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C5OC)C6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H53ClN10O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-85JAGC	SCHEMBL24717827	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-6-methoxy-1,3-dioxoisoindol-4-yl]-2-azaspiro[3.5]nonan-7-yl]methyl]piperazin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894121	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCN(CC5CCC6(CC5)CN(C5=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC(OC)=C5)C6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H53ClN10O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-CUSBL2	SCHEMBL24718335	2-[6-[[5-chloro-2-[7-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperidin-4-yl]methyl]-2,7-diazaspiro[4.4]nonan-2-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC5(CCN(CC6CCN(C7=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=CC=C7)CC6)C5)C4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H51ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-GKNZTV	SCHEMBL24718337	2-[6-[[5-chloro-2-[7-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]piperidin-4-yl]methyl]-2,7-diazaspiro[4.4]nonan-2-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894403	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC5(CCN(CC6CCN(C7=C8CN(C9CCC(=O)NC9=O)C(=O)C8=CC=C7)CC6)C5)C4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H53ClN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-0VSVY2	SCHEMBL24717356	2-[6-[[5-chloro-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]propan-2-yl]piperazin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30798496	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCN(C(C)(C)C5CCN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)CC5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C44H53ClN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-3505DC	SCHEMBL24718738	2-[6-[[5-chloro-2-[2-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]piperazin-1-yl]methyl]-7-azaspiro[3.5]nonan-7-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894178	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC5(CC4)CC(CN4CCN(C6=C7CN(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)CC4)C5)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H53ClN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-JK0RV5	SCHEMBL24717990	2-[6-[[5-chloro-2-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30798458	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCN(CC5CCN(C6=CC7=C(C=C6F)C(=O)N(C6CCC(=O)NC6=O)C7)CC5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C42H48ClFN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-6I1QD5	SCHEMBL24717575	2-[6-[[5-chloro-2-[2-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperidin-4-yl]ethyl]-5-oxa-2,8-diazaspiro[3.5]nonan-8-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894377	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCOC5(CN(CCC6CCN(C7=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=CC=C7)CC6)C5)C4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H51ClN10O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-QWEMXN	SCHEMBL24718142	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-2,7-diazaspiro[4.4]nonan-7-yl]methyl]-4-fluoropiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894086	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(F)(CN5CCC6(CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H52ClFN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-B7NPCC	SCHEMBL24717675	2-[6-[[5-chloro-2-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-7-fluoro-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30798512	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCN(CC5CCN(C6=CC7=C(C(=O)N(C8CCC(=O)NC8=O)C7)C(F)=C6)CC5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C42H48ClFN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-HEO6KV	SCHEMBL24718136	2-[6-[[5-chloro-2-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]piperidine-1-carbonyl]-7-azaspiro[3.5]nonan-7-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894365	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC5(CC4)CC(C(=O)N4CCC(C6=CC=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)CC4)C5)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H52ClN9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-HRVH0Y	SCHEMBL24718336	2-[6-[[5-chloro-2-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-4-methoxy-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30798578	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCN(CC5CCN(C6=C(OC)C7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)CC5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C43H51ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-80YIXN	SCHEMBL24717389	2-[6-[[5-chloro-2-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-6-methoxy-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894145	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCN(CC5CCN(C6=CC7=C(C=C6OC)C(=O)N(C6CCC(=O)NC6=O)C7)CC5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C43H51ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-W2BTFH	SCHEMBL24718340	2-[6-[[5-chloro-2-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]piperidine-4-carbonyl]-2,7-diazaspiro[3.5]nonan-7-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894284	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC5(CC4)CN(C(=O)C4CCN(C6=C7CN(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)CC4)C5)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H51ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-1YT3K8	WO2024151557A1_23	.	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCN(C[C@H]5C[C@H](N6CCC(C7=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=CC=C7)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H53ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-W2ILN4	WO2024151557A1_24	.	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCN(C[C@H]5C[C@@H](N6CCC(C7=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=CC=C7)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H53ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-XMRTTM	SCHEMBL24717984	2-[6-[[5-chloro-2-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-4-fluoro-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894374	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCN(CC5CCN(C6=C(F)C7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)CC5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C42H48ClFN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-2VG43V	SCHEMBL24717679	2-[6-[[5-chloro-2-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30798475	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCN(CC5CCN(C6=CC7=C(C(=O)N(C8CCC(=O)NC8=O)C7)C(OC)=C6)CC5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C43H51ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-CH3JM6	SCHEMBL24718342	2-[6-[[5-chloro-2-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]piperazine-1-carbonyl]-7-azaspiro[3.5]nonan-7-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894225	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC5(CC4)CC(C(=O)N4CCN(C6=C7CN(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)CC4)C5)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H51ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-RXDVKA	SCHEMBL23267964	2-[6-[[5-chloro-2-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894381	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(OC5CCN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)CC5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C42H48ClN9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-K1A9QF	SCHEMBL24717896	2-[6-[(5-chloro-2-piperidin-1-ylpyrimidin-4-yl)amino]-1-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxyethyl]-2-oxoquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894166	CNC(=O)COC1=CC2=C(C=CC(NC3=C(Cl)C=NC(N4CCCCC4)=N3)=C2)N(CCOC2=CC=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=C2)C1=O	C36H35ClN8O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-3LZ4OY	SCHEMBL24717894	2-[6-[[5-chloro-2-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxycyclohexyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27231376; SCHEMBL30894188	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5CC[C@@H](OC6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C43H47ClN8O9	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-LSIYBS	SCHEMBL24717893	2-[6-[[5-chloro-2-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxycyclohexyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27232702; SCHEMBL30894089	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5CC[C@@H](OC6=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)CC5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C43H47ClN8O9	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-ZS6OLJ	SCHEMBL24718132	2-[6-[(5-chloro-2-pyrrolidin-1-ylpyrimidin-4-yl)amino]-1-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxyethyl]-2-oxoquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894233	CNC(=O)COC1=CC2=C(C=CC(NC3=C(Cl)C=NC(N4CCCC4)=N3)=C2)N(CCOC2=CC=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=C2)C1=O	C35H33ClN8O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-6EAOBC	SCHEMBL24718133	2-[6-[[5-chloro-2-(2,6-dimethylmorpholin-4-yl)pyrimidin-4-yl]amino]-1-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxyethyl]-2-oxoquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894192	CNC(=O)COC1=CC2=C(C=CC(NC3=C(Cl)C=NC(N4CC(C)OC(C)C4)=N3)=C2)N(CCOC2=CC=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=C2)C1=O	C37H37ClN8O9	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-DFB10G	SCHEMBL24718134	2-[6-[[5-chloro-2-[2-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]piperazin-1-yl]propan-2-yl]-7-azaspiro[3.5]nonan-7-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894375	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC5(CC4)CC(C(C)(C)N4CCN(C6=C7CN(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)CC4)C5)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H57ClN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-4IVAJJ	SCHEMBL24717899	2-[6-[[5-chloro-2-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-5-fluoro-1,3-dioxoisoindol-4-yl]piperidin-4-yl]methyl]piperazin-1-yl]pyrimidin-4-yl]amino]-1-methyl-2-oxoquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30798359	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCN(CC5CCN(C6=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C6F)CC5)CC4)=NC=C3Cl)=C2)N(C)C1=O	C40H42ClFN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-MGJF31	SCHEMBL24717904	2-[6-[[5-chloro-2-[2-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]piperidin-4-yl]propan-2-yl]-2,7-diazaspiro[3.5]nonan-7-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894180	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC5(CC4)CN(C(C)(C)C4CCN(C6=C7CN(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)CC4)C5)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H57ClN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-3AH2MN	SCHEMBL24717901	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-2,7-diazaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-1-(2-methoxyethyl)-2-oxoquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894293	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CCC6(CC5)CN(C5=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C5)C6)CC4)=NC=C3Cl)=C2)N(CCOC)C1=O	C45H51ClN10O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-YQ1Z7S	SCHEMBL24718719	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-5,5-difluoro-2,7-diazaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894224	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CCC6(CN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)C6)C(F)(F)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H49ClF2N10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-SC5Z93	SCHEMBL24718720	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-3-oxo-2,7-diazaspiro[4.4]nonan-7-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894330	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CCC6(CC(=O)N(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H51ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-RJ6C93	WO2024151557A1_40	.	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCN(C[C@H]5C[C@H](N6CCC(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H53ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-B925NW	WO2024151557A1_41	.	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCN(C[C@H]5C[C@@H](N6CCC(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H53ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-8C7AU1	SCHEMBL24718730	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-1-yl]cyclopentyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894108	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(OC5CCC(N6CCC(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H54ClN9O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-KO40X7	SCHEMBL24718732	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-2,7-diazaspiro[3.5]nonan-7-yl]methyl]-4-fluoropiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894115	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(F)(CN5CCC6(CC5)CN(C5=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C5)C6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H50ClFN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-980U9T	SCHEMBL24718731	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]-2,7-diazaspiro[3.5]nonan-7-yl]methyl]-4-fluoropiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894237	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(F)(CN5CCC6(CC5)CN(C5=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C5)C6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H50ClFN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-2RWAO5	SCHEMBL24717838	2-[6-[[5-chloro-2-[4-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-2,7-diazaspiro[3.5]nonan-7-yl]propan-2-yl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL31225217	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(C(C)(C)N5CCC6(CC5)CN(C5=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C5)C6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H55ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-BKGK32	SCHEMBL24717835	2-[6-[[5-chloro-2-[4-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]-2,7-diazaspiro[3.5]nonan-7-yl]propan-2-yl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894264	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(C(C)(C)N5CCC6(CC5)CN(C5=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C5)C6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H55ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-O5Y64L	SCHEMBL27219547	2-[6-[[5-chloro-2-[4-[7-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-2,7-diazaspiro[4.4]nonane-2-carbonyl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894254	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(C(=O)N5CCC6(CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H51ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-4KK1CJ	SCHEMBL24717839	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-1-oxo-2,7-diazaspiro[4.4]nonan-7-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894318	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CCC6(CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7)C6=O)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H51ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-KLBTNU	SCHEMBL24718317	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-2-azaspiro[3.5]nonan-7-yl]oxy]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894417	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(OC5CCC6(CC5)CN(C5=CC7=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C7)C6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H52ClN9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-E9DEG4	SCHEMBL24718316	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-2,7-diazaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-1-cyclopropyl-2-oxoquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894117	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CCC6(CC5)CN(C5=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C5)C6)CC4)=NC=C3Cl)=C2)N(C2CC2)C1=O	C45H49ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-LV0ZO0	SCHEMBL24718318	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-2,7-diazaspiro[3.5]nonan-7-yl]methyl]-4-fluoropiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894092	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(F)(CN5CCC6(CC5)CN(C5=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C5)C6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H52ClFN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-J450WO	SCHEMBL24718315	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]-2,7-diazaspiro[3.5]nonan-7-yl]methyl]-4-fluoropiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894399	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(F)(CN5CCC6(CC5)CN(C5=C7CN(C8CCC(=O)NC8=O)C(=O)C7=CC=C5)C6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H52ClFN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-1NI98R	SCHEMBL27219598	2-[6-[[5-chloro-2-[4-[2-[7-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-2,7-diazaspiro[4.4]nonan-2-yl]propan-2-yl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL31225103	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(C(C)(C)N5CCC6(CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H57ClN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-3UQWBZ	SCHEMBL27219639	2-[6-[[5-chloro-2-[4-[[7-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-3-oxo-2,7-diazaspiro[4.4]nonan-2-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894120	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CC6(CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7)C6)CC5=O)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H51ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-ISEK0K	SCHEMBL27219529	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-2,7-diazaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N,N-dimethylacetamide; SCHEMBL30894212	CC(C)N1C(=O)C(OCC(=O)N(C)C)=CC2=C1C=CC(NC1=NC(N3CCC(CN4CCC5(CC4)CN(C4=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C4)C5)CC3)=NC=C1Cl)=C2	C46H53ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-6G1DUD	SCHEMBL27219595	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-2,7-diazaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-ethylacetamide; SCHEMBL30894200	CCNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CCC6(CC5)CN(C5=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C5)C6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H53ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-T1T0VO	SCHEMBL27219532	2-[6-[[2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-2,7-diazaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]-5-fluoropyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894305	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CCC6(CC5)CN(C5=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C5)C6)CC4)=NC=C3F)=C2)N(C(C)C)C1=O	C45H51FN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-B3XGAP	SCHEMBL27219583	2-[6-[[5-chloro-2-[4-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-2,7-diazaspiro[3.5]nonan-7-yl]propan-2-yl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894336	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(C(C)(C)N5CCC6(CC5)CN(C5=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C5)C6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H57ClN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-HTGDS0	SCHEMBL24718333	2-[6-[[5-chloro-2-[4-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]-2,7-diazaspiro[3.5]nonan-7-yl]propan-2-yl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894148	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(C(C)(C)N5CCC6(CC5)CN(C5=C7CN(C8CCC(=O)NC8=O)C(=O)C7=CC=C5)C6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H57ClN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-F0VA1Y	SCHEMBL24718334	2-[6-[[5-chloro-2-[4-[[7-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-1-oxo-2,7-diazaspiro[4.4]nonan-2-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894271	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CCC6(CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7)C6)C5=O)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H51ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-IGZEEE	SCHEMBL24717548	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]-2-azaspiro[3.5]nonan-7-yl]oxy]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894386	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(OC5CCC6(CC5)CN(C5=C7CN(C8CCC(=O)NC8=O)C(=O)C7=CC=C5)C6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H52ClN9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-623ZPA	SCHEMBL24717547	2-[6-[[5-chloro-2-[4-[[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]-3,9-diazaspiro[5.5]undecan-9-yl]methyl]-4-fluoropiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894227	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(F)(CN5CCC6(CC5)CCN(C5=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C5)CC6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H54ClFN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-2OUMB8	SCHEMBL24717546	2-[6-[[5-chloro-2-[9-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]-4-fluoropiperidin-4-yl]methyl]-3,9-diazaspiro[5.5]undecan-3-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894201	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC5(CCN(CC6(F)CCN(C7=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=CC=C7)CC6)CC5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H54ClFN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-1U7858	SCHEMBL24718119	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1-oxo-3H-isoindol-5-yl]-2,7-diazaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894385	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CCC6(CC5)CN(C5=C(F)C=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C5)C6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H52ClFN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-KLEWZ8	SCHEMBL24718118	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-3-oxo-2,7-diazaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894356	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CCC6(CC5)CN(C5=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C5)C6=O)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H49ClN10O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-YEV0MC	SCHEMBL24718117	2-[6-[[5-chloro-2-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-2-azaspiro[4.4]nonane-8-carbonyl]piperazin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894304	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCN(C(=O)C5CCC6(CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H51ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-BCZZPY	SCHEMBL24718120	2-[6-[[5-chloro-2-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]pyrimidin-4-yl]amino]-1-methyl-2-oxoquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894272	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCN(CC5CCN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)CC5)CC4)=NC=C3Cl)=C2)N(C)C1=O	C40H45ClN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-XT864L	SCHEMBL24717682	2-[6-[[5-chloro-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]propan-2-yl]piperazin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894280	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCN(C(C)(C)C5CCN(C6=CC7=C(C=C6F)C(=O)N(C6CCC(=O)NC6=O)C7)CC5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C44H52ClFN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-J4QK7F	SCHEMBL24718353	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-3-oxo-1H-isoindol-5-yl]-2-azaspiro[3.5]nonan-7-yl]oxy]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894299	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(OC5CCC6(CC5)CN(C5=CC=C7CN(C8CCC(=O)NC8=O)C(=O)C7=C5)C6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H52ClN9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-HS7H32	SCHEMBL27219584	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-3-oxo-1H-isoindol-4-yl]-2-azaspiro[3.5]nonan-7-yl]oxy]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(OC5CCC6(CC5)CN(C5=C7C(=O)N(C8CCC(=O)NC8=O)CC7=CC=C5)C6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H52ClN9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-R3AAJS	SCHEMBL24718325	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-4-fluoro-1-oxo-3H-isoindol-5-yl]-2,7-diazaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894172	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CCC6(CC5)CN(C5=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C5F)C6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H52ClFN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-I6INRI	SCHEMBL24717755	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-4-methoxy-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30798478	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCC(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7OC)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H56ClN9O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-UQCWP3	SCHEMBL24718326	2-[6-[[5-chloro-2-[4-[[3-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1-oxo-3H-isoindol-4-yl]-3,9-diazaspiro[5.5]undecan-9-yl]methyl]-4-fluoropiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894297	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(F)(CN5CCC6(CC5)CCN(C5=C7CN(C8CCC(=O)NC8=O)C(=O)C7=CC(F)=C5)CC6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H55ClF2N10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-OBS45N	SCHEMBL24717565	2-[6-[[5-chloro-2-[4-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-2-azaspiro[4.4]nonan-8-yl]propan-2-yl]piperazin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894294	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCN(C(C)(C)C5CCC6(CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H57ClN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-FOS5BN	SCHEMBL27219650	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-2-azaspiro[4.4]nonan-8-yl]methyl]piperazin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894125	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCN(CC5CCC6(CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H53ClN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-W84M2M	SCHEMBL24717567	2-[6-[[5-chloro-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-7-fluoro-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]propan-2-yl]piperazin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894245	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCN(C(C)(C)C5CCN(C6=CC7=C(C(=O)N(C8CCC(=O)NC8=O)C7)C(F)=C6)CC5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C44H52ClFN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-8JBDWG	SCHEMBL24717566	2-[6-[[5-chloro-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]propan-2-yl]piperazin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894249	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCN(C(C)(C)C5CCN(C6=CC7=C(C(=O)N(C8CCC(=O)NC8=O)C7)C(OC)=C6)CC5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H55ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-EG7DDB	SCHEMBL24717744	2-[6-[[5-chloro-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-4-methoxy-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]propan-2-yl]piperazin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894101	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCN(C(C)(C)C5CCN(C6=C(OC)C7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)CC5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H55ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-05CAQE	SCHEMBL24717985	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCC(C7=C(F)C=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H53ClFN9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-75W03K	SCHEMBL24718745	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-7-fluoro-1-oxo-3H-isoindol-5-yl]-2,7-diazaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894085	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CCC6(CC5)CN(C5=CC(F)=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C5)C6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H52ClFN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-VDGI9P	WO2024151557A1_81	.	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCC(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7F)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H53ClFN9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-122814	SCHEMBL24718148	2-[6-[[5-chloro-2-[4-[[3-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]-3,9-diazaspiro[5.5]undecan-9-yl]methyl]-4-fluoropiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894285	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(F)(CN5CCC6(CC5)CCN(C5=C7CN(C8CCC(=O)NC8=O)C(=O)C7=CC=C5)CC6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H56ClFN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-K4WQZW	SCHEMBL24718144	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1,3-dioxoisoindol-5-yl]-2,7-diazaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894088	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CCC6(CC5)CN(C5=CC(OC)=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C5)C6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H53ClN10O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-9GIKQV	SCHEMBL24718141	2-[6-[[5-chloro-2-[4-[[7-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1-oxo-3H-isoindol-5-yl]-2,7-diazaspiro[3.5]nonan-2-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894329	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CC6(CCN(C7=CC8=C(C=C7F)C(=O)N(C7CCC(=O)NC7=O)C8)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H52ClFN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-OKYSDT	SCHEMBL24718156	2-[6-[[5-chloro-2-[4-[[7-[2-(2,6-dioxopiperidin-3-yl)-6-methoxy-1-oxo-3H-isoindol-5-yl]-2,7-diazaspiro[3.5]nonan-2-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894243	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CC6(CCN(C7=CC8=C(C=C7OC)C(=O)N(C7CCC(=O)NC7=O)C8)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H55ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-KP1LAM	SCHEMBL24718150	2-[6-[[5-chloro-2-[4-[[7-[2-(2,6-dioxopiperidin-3-yl)-7-fluoro-1-oxo-3H-isoindol-5-yl]-2,7-diazaspiro[3.5]nonan-2-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894119	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CC6(CCN(C7=CC8=C(C(=O)N(C9CCC(=O)NC9=O)C8)C(F)=C7)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H52ClFN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-6L8R0C	SCHEMBL24718152	2-[6-[[5-chloro-2-[4-[[7-[2-(2,6-dioxopiperidin-3-yl)-4-fluoro-1-oxo-3H-isoindol-5-yl]-2,7-diazaspiro[3.5]nonan-2-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894413	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CC6(CCN(C7=C(F)C8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H52ClFN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-Q2D6HT	SCHEMBL24718155	2-[6-[[5-chloro-2-[4-[[7-[2-(2,6-dioxopiperidin-3-yl)-4-methoxy-1-oxo-3H-isoindol-5-yl]-2,7-diazaspiro[3.5]nonan-2-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894357	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CC6(CCN(C7=C(OC)C8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H55ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-IWJYH0	SCHEMBL24717977	2-[6-[[5-chloro-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-4-fluoro-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]propan-2-yl]piperazin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894186	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCN(C(C)(C)C5CCN(C6=C(F)C7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)CC5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C44H52ClFN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-C9GX26	SCHEMBL27219644	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-5,5-difluoro-2,7-diazaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894259	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CCC6(CN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7)C6)C(F)(F)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H51ClF2N10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-JZ7NIL	SCHEMBL24718350	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]-5,5-difluoro-2,7-diazaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894402	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CCC6(CN(C7=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=CC=C7)C6)C(F)(F)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H49ClF2N10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-Z4V9C7	SCHEMBL24718668	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-7-fluoro-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCC(C7=CC(F)=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H53ClFN9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-QMIESH	SCHEMBL27219612	2-[6-[[5-chloro-2-[4-[[3-[2-(2,6-dioxopiperidin-3-yl)-5-fluoro-3-oxo-1H-isoindol-4-yl]-3,9-diazaspiro[5.5]undecan-9-yl]methyl]-4-fluoropiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(F)(CN5CCC6(CC5)CCN(C5=C7C(=O)N(C8CCC(=O)NC8=O)CC7=CC=C5F)CC6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H55ClF2N10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-EJKLDC	SCHEMBL24718346	2-[6-[[5-chloro-2-[9-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]-4-fluoropiperidin-4-yl]methyl]-3,9-diazaspiro[5.5]undecan-3-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894269	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC5(CCN(CC6(F)CCN(C7=C8CN(C9CCC(=O)NC9=O)C(=O)C8=CC=C7)CC6)CC5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H56ClFN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-MG9U11	SCHEMBL24718351	2-[6-[[5-chloro-2-[9-[[1-[2-(2,6-dioxopiperidin-3-yl)-5-fluoro-1-oxo-3H-isoindol-4-yl]-4-fluoropiperidin-4-yl]methyl]-3,9-diazaspiro[5.5]undecan-3-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894290	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC5(CCN(CC6(F)CCN(C7=C8CN(C9CCC(=O)NC9=O)C(=O)C8=CC=C7F)CC6)CC5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H55ClF2N10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-013SZ0	SCHEMBL24718348	2-[6-[[5-chloro-2-[4-[[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-1-yl]azetidin-1-yl]methyl]-4-fluoropiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=C(Cl)C=NC(N4CCC(F)(CN5CC(N6CCC(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)C5)CC4)=N3)=C2)N(C(C)C)C1=O	C46H52ClFN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-JNTTF2	SCHEMBL24717890	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-2-azaspiro[4.4]nonan-8-yl]oxy]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894099	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(OC5CCC6(CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H52ClN9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-MJC0FN	SCHEMBL24717892	2-[6-[[5-chloro-2-[4-[[7-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]-2,7-diazaspiro[3.5]nonan-2-yl]methyl]-4-fluoropiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL31225148	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(F)(CN5CC6(CCN(C7=C8CN(C9CCC(=O)NC9=O)C(=O)C8=CC=C7)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H52ClFN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-ZYRH37	SCHEMBL24717891	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1-oxo-3H-isoindol-5-yl]-5,5-difluoro-2,7-diazaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894384	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CCC6(CN(C7=C(F)C=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7)C6)C(F)(F)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H50ClF3N10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-GR6QXQ	SCHEMBL24717889	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-5-yl]-5,5-difluoro-2,7-diazaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894137	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CCC6(CN(C7=CC(OC)=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7)C6)C(F)(F)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H53ClF2N10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-GWXARH	SCHEMBL27219534	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]-5,5-difluoro-2,7-diazaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CCC6(CN(C7=C8CN(C9CCC(=O)NC9=O)C(=O)C8=CC=C7)C6)C(F)(F)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H51ClF2N10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-Y5ERNT	SCHEMBL24717704	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27231361	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCC(C7=CC(OC)=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H56ClN9O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-7YMXZU	SCHEMBL24717834	2-[6-[[5-chloro-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]piperidin-4-yl]propan-2-yl]piperazin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894105	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCN(C(C)(C)C5CCN(C6=C7CN(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)CC5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C44H53ClN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-0EUZDT	SCHEMBL24717771	2-[6-[[5-chloro-2-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1-oxo-3H-isoindol-4-yl]piperidin-4-yl]methyl]piperazin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894314	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCN(CC5CCN(C6=CC(F)=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)CC5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C42H48ClFN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-W7MINT	SCHEMBL24717886	2-[6-[[5-chloro-2-[4-[[7-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1-oxo-3H-isoindol-5-yl]-2,7-diazaspiro[3.5]nonan-2-yl]methyl]-4-fluoropiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL31225118	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(F)(CN5CC6(CCN(C7=CC8=C(C=C7F)C(=O)N(C7CCC(=O)NC7=O)C8)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H51ClF2N10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-JVXMXE	SCHEMBL24717888	2-[6-[[5-chloro-2-[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]-methylamino]cyclohexyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27231483; SCHEMBL30894313	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5CC[C@@H](N(C)C6CN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)C6)CC5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H55ClN10O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-R9KUWZ	SCHEMBL24717902	2-[6-[[5-chloro-2-[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]azetidin-3-yl]-methylamino]cyclohexyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27231638; SCHEMBL30894236	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5CC[C@@H](N(C)C6CN(C7=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=CC=C7)C6)CC5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H55ClN10O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-JJPRKE	SCHEMBL24717898	2-[6-[[5-chloro-2-[9-[[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1-oxo-3H-isoindol-4-yl]-4-fluoropiperidin-4-yl]methyl]-3,9-diazaspiro[5.5]undecan-3-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894242	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC5(CCN(CC6(F)CCN(C7=C8CN(C9CCC(=O)NC9=O)C(=O)C8=CC(F)=C7)CC6)CC5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H55ClF2N10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-21QL7Z	SCHEMBL24717903	2-[6-[[5-chloro-2-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-1-yl]cyclohexyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27219606; SCHEMBL30894146	CNC(=O)COC1=CC2=C(C=CC(NC3=C(Cl)C=NC(N4CCC(O[C@H]5CC[C@@H](N6CCC(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)CC5)CC4)=N3)=C2)N(C(C)C)C1=O	C48H56ClN9O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-B9E442	SCHEMBL27219632	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-2,7-diazaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-8-fluoro-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894389	CNC(=O)COC1=CC2=C(C(F)=CC(NC3=NC(N4CCC(CN5CCC6(CC5)CN(C5=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C5)C6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H50ClFN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-VNGR1F	SCHEMBL24717385	2-[6-[[5-chloro-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-6-methoxy-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]propan-2-yl]piperazin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894147	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCN(C(C)(C)C5CCN(C6=CC7=C(C=C6OC)C(=O)N(C6CCC(=O)NC6=O)C7)CC5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H55ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-TDC94S	SCHEMBL24717897	2-[6-[[5-chloro-2-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-4-fluoropiperidin-4-yl]methyl]piperazin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30798311	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCN(CC5(F)CCN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)CC5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C42H48ClFN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-8T6B6P	SCHEMBL24717582	2-[6-[[5-chloro-2-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]-4-fluoropiperidin-4-yl]methyl]piperazin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30798364	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCN(CC5(F)CCN(C6=C7CN(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)CC5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C42H48ClFN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-5VNN4R	SCHEMBL24717587	2-[6-[[5-chloro-2-[4-[[7-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-5-yl]-2,7-diazaspiro[3.5]nonan-2-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894361	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CC6(CCN(C7=CC8=C(C(=O)N(C9CCC(=O)NC9=O)C8)C(OC)=C7)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H55ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-238BYM	SCHEMBL24717585	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-4,6-difluoro-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCC(C7=C(F)C=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7F)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H52ClF2N9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-FKEV1J	SCHEMBL24718003	2-[6-[[5-chloro-2-[4-[3-[(3S,4R)-4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-3-fluoropiperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27231487	CNC(=O)COC1=CC2=C(C=CC(NC3=C(Cl)C=NC(N4CCC(O[C@H]5C[C@H](N6CC[C@H](C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)[C@H](F)C6)C5)CC4)=N3)=C2)N(C(C)C)C1=O	C46H51ClFN9O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-9XEVOB	SCHEMBL24718704	2-[6-[[5-chloro-2-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-6-methoxy-1-oxo-3H-isoindol-4-yl]piperidin-4-yl]methyl]piperazin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894370	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCN(CC5CCN(C6=CC(OC)=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)CC5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C43H51ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-R4YG10	SCHEMBL24718347	2-[6-[[5-chloro-2-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-7-fluoro-1-oxo-3H-isoindol-4-yl]piperidin-4-yl]methyl]piperazin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894291	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCN(CC5CCN(C6=CC=C(F)C7=C6CN(C6CCC(=O)NC6=O)C7=O)CC5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C42H48ClFN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-F57PLA	SCHEMBL24718343	2-[6-[[5-chloro-2-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-4-yl]piperidin-4-yl]methyl]piperazin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894167	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCN(CC5CCN(C6=CC=C(OC)C7=C6CN(C6CCC(=O)NC6=O)C7=O)CC5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C43H51ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-PECDYH	SCHEMBL24718344	2-[6-[[5-chloro-2-[4-[[7-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-2,7-diazaspiro[3.5]nonan-2-yl]methyl]-4-fluoropiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894220	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(F)(CN5CC6(CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H52ClFN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-5IZ7MV	SCHEMBL24718151	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1-oxo-3H-isoindol-5-yl]-2-azaspiro[3.5]nonan-7-yl]oxy]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894153	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(OC5CCC6(CC5)CN(C5=C(F)C=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C5)C6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H51ClFN9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-Z9K02Z	SCHEMBL24718154	2-[6-[[5-chloro-2-[4-[[7-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]-5,5-difluoro-2,7-diazaspiro[3.5]nonan-2-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894310	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CC6(CCN(C7=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=CC=C7)CC6(F)F)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H49ClF2N10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-3TH9AS	SCHEMBL27219549	2-[6-[[5-chloro-2-[4-[[7-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]-5,5-difluoro-2,7-diazaspiro[3.5]nonan-2-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CC6(CCN(C7=C8CN(C9CCC(=O)NC9=O)C(=O)C8=CC=C7)CC6(F)F)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H51ClF2N10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-7M1E5E	SCHEMBL24717919	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-5,5-difluoro-2,7-diazaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-1-(2-methoxyethyl)-2-oxoquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894368	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CCC6(CN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)C6)C(F)(F)C5)CC4)=NC=C3Cl)=C2)N(CCOC)C1=O	C45H49ClF2N10O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-V8CACZ	SCHEMBL24717921	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-5,5-difluoro-2,7-diazaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-1-methyl-2-oxoquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894369	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CCC6(CN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)C6)C(F)(F)C5)CC4)=NC=C3Cl)=C2)N(C)C1=O	C43H45ClF2N10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-OMYO3Q	SCHEMBL24717920	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-7-fluoro-4-methoxy-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCC(C7=C(OC)C8=C(C(=O)N(C9CCC(=O)NC9=O)C8)C(F)=C7)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H55ClFN9O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-JWTVQE	SCHEMBL24717849	2-[6-[[5-chloro-2-[9-[[1-[2-(2,6-dioxopiperidin-3-yl)-7-fluoro-1-oxo-3H-isoindol-4-yl]-4-fluoropiperidin-4-yl]methyl]-3,9-diazaspiro[5.5]undecan-3-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894303	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC5(CCN(CC6(F)CCN(C7=C8CN(C9CCC(=O)NC9=O)C(=O)C8=C(F)C=C7)CC6)CC5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H55ClF2N10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-76W4G1	SCHEMBL24717851	2-[6-[[5-chloro-2-[9-[[1-[2-(2,6-dioxopiperidin-3-yl)-7-fluoro-3-oxo-1H-isoindol-4-yl]-4-fluoropiperidin-4-yl]methyl]-3,9-diazaspiro[5.5]undecan-3-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894340	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC5(CCN(CC6(F)CCN(C7=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C(F)C=C7)CC6)CC5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H55ClF2N10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-RIU2KN	SCHEMBL24717850	2-[6-[[5-chloro-2-[4-[3-[(3S,4R)-4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-3-fluoropiperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27231731	CNC(=O)COC1=CC2=C(C=CC(NC3=C(Cl)C=NC(N4CCC(O[C@H]5C[C@H](N6CC[C@H](C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8)[C@H](F)C6)C5)CC4)=N3)=C2)N(C(C)C)C1=O	C46H53ClFN9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-OPYDE5	SCHEMBL24718009	2-[6-[[5-chloro-2-[4-[3-[(3S,4R)-4-[2-(2,6-dioxopiperidin-3-yl)-3-oxo-1H-isoindol-5-yl]-3-fluoropiperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27231401	CNC(=O)COC1=CC2=C(C=CC(NC3=C(Cl)C=NC(N4CCC(O[C@H]5C[C@H](N6CC[C@H](C7=CC8=C(C=C7)CN(C7CCC(=O)NC7=O)C8=O)[C@H](F)C6)C5)CC4)=N3)=C2)N(C(C)C)C1=O	C46H53ClFN9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-O1HUVQ	SCHEMBL27219552	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-3,3-dimethyl-2,7-diazaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894252	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CCC6(CC5)CN(C5=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C5)C6(C)C)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H55ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-JKGVK7	SCHEMBL24717911	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-5-fluoro-2,7-diazaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894266	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CCC6(CN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)C6)C(F)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H50ClFN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-GR0QII	SCHEMBL24717909	2-[6-[[5-chloro-2-[4-[[7-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-5,5-difluoro-2,7-diazaspiro[3.5]nonan-2-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894234	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CC6(CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6(F)F)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H49ClF2N10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-44BTGO	SCHEMBL24717912	2-[6-[[5-chloro-2-[4-[[7-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-5,5-difluoro-2,7-diazaspiro[3.5]nonan-2-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894244	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CC6(CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7)CC6(F)F)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H51ClF2N10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-IN77SI	SCHEMBL24717388	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-3,3-difluoropiperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27232646	CNC(=O)COC1=CC2=C(C=CC(NC3=C(Cl)C=NC(N4CCC(O[C@H]5C[C@H](N6CCC(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)C(F)(F)C6)C5)CC4)=N3)=C2)N(C(C)C)C1=O	C46H50ClF2N9O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-NWOZ60	SCHEMBL24717910	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-4-yl]-2,7-diazaspiro[4.4]nonan-7-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894387	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CCC6(CCN(C7=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=CC(F)=C7)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H50ClFN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-6Q25EW	SCHEMBL24718130	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-5-fluoro-1,3-dioxoisoindol-4-yl]-2,7-diazaspiro[4.4]nonan-7-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894096	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CCC6(CCN(C7=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=CC=C7F)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H50ClFN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-AZRTYJ	SCHEMBL24718126	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-1-ethyl-2-oxoquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27231718	CCN1C(=O)C(OCC(=O)NC)=CC2=C1C=CC(NC1=NC(N3CCC(O[C@H]4C[C@@H](N5CCC(C6=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)CC5)C4)CC3)=NC=C1Cl)=C2	C45H50ClN9O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-Q4Y4TO	SCHEMBL24718125	2-[6-[[5-chloro-2-[(3S)-3-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxymethyl]piperidin-1-yl]pyrimidin-4-yl]amino]-1-[2-(dimethylamino)ethyl]-2-oxoquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894328	CNC(=O)COC1=CC2=C(C=CC(NC3=C(Cl)C=NC(N4CCC[C@H](COC5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)C4)=N3)=C2)N(CCN(C)C)C1=O	C39H42ClN9O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-KE5DI8	SCHEMBL24717576	2-[6-[[5-chloro-2-[2-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]-5-oxa-2,8-diazaspiro[3.5]nonan-8-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894241	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCOC5(CN(CC6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)C5)C4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C44H49ClN10O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-N0Q7HI	SCHEMBL24717574	2-[6-[[5-chloro-2-[2-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperidin-4-yl]methyl]-5-oxa-2,8-diazaspiro[3.5]nonan-8-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894087	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCOC5(CN(CC6CCN(C7=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=CC=C7)CC6)C5)C4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C44H49ClN10O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-VN8A5Y	SCHEMBL24717816	2-[6-[[5-chloro-2-[2-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]ethyl]-5-oxa-2,8-diazaspiro[3.5]nonan-8-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894298	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCOC5(CN(CCC6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)C5)C4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H51ClN10O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-3BEUDD	WO2024151557A1_146	.	[2H]C1=NC(NC2=CC3=C(C=C2)N(CCOC2=CC=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C2)C(=O)C(OCC(=O)NC)=C3)=C(Cl)C=N1	C31H26ClN7O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-1NROM0	SCHEMBL24717814	2-[6-[(5-chloro-2-methylpyrimidin-4-yl)amino]-1-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxyethyl]-2-oxoquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894235	CNC(=O)COC1=CC2=C(C=CC(NC3=C(Cl)C=NC(C)=N3)=C2)N(CCOC2=CC=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=C2)C1=O	C32H28ClN7O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-SV2S3W	SCHEMBL24717906	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperidin-1-yl]cyclopentyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL31225143	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(OC5CCC(N6CCC(C7=CC=CC8=C7C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H54ClN9O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-YV9AAS	SCHEMBL24717900	2-[6-[(5-chloro-2-pyrazol-1-ylpyrimidin-4-yl)amino]-1-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxyethyl]-2-oxoquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894309	CNC(=O)COC1=CC2=C(C=CC(NC3=C(Cl)C=NC(N4C=CC=N4)=N3)=C2)N(CCOC2=CC=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=C2)C1=O	C34H28ClN9O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-D51WWS	SCHEMBL24717905	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-7-azaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894323	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CCC6(CC5)CC(C5=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C5)C6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H52ClN9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-6XFWF0	SCHEMBL24717579	2-[6-[[5-chloro-2-[4-[[3-[2-(2,6-dioxopiperidin-3-yl)-5-fluoro-1-oxo-3H-isoindol-4-yl]-3,9-diazaspiro[5.5]undecan-9-yl]methyl]-4-fluoropiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894217	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(F)(CN5CCC6(CC5)CCN(C5=C7CN(C8CCC(=O)NC8=O)C(=O)C7=CC=C5F)CC6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H55ClF2N10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-8ARNRU	SCHEMBL24717580	2-[6-[[5-chloro-2-[9-[[1-[2-(2,6-dioxopiperidin-3-yl)-5-fluoro-3-oxo-1H-isoindol-4-yl]-4-fluoropiperidin-4-yl]methyl]-3,9-diazaspiro[5.5]undecan-3-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894355	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC5(CCN(CC6(F)CCN(C7=C8C(=O)N(C9CCC(=O)NC9=O)CC8=CC=C7F)CC6)CC5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H55ClF2N10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-52LP5O	SCHEMBL23250131	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL23250132; SCHEMBL24717577	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCC(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H52ClN9O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-8UUVBC	SCHEMBL24718147	2-[6-[[5-chloro-2-[2-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]piperidin-1-yl]propan-2-yl]-7-azaspiro[3.5]nonan-7-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894226	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC5(CC4)CC(C(C)(C)N4CCC(C6=CC=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)CC4)C5)=NC=C3Cl)=C2)N(C(C)C)C1=O	C48H58ClN9O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-KP6HTG	SCHEMBL24718145	2-[6-[[5-chloro-2-[4-[[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-3-azabicyclo[3.1.0]hexan-6-yl]methyl]piperazin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=C(Cl)C=NC(N4CCN(CC5C6CN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC56)CC4)=N3)=C2)N(C(C)C)C1=O	C42H45ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-QZD7YR	SCHEMBL24718146	2-[6-[[5-chloro-2-[4-[[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]-3-azabicyclo[3.1.0]hexan-6-yl]methyl]piperazin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=C(Cl)C=NC(N4CCN(CC5C6CN(C7=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=CC=C7)CC56)CC4)=N3)=C2)N(C(C)C)C1=O	C42H45ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-R3LLDJ	SCHEMBL24717922	2-[6-[[5-chloro-2-[6-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]-3-azabicyclo[3.1.0]hexan-3-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=C(Cl)C=NC(N4CC5C(CN6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)C5C4)=N3)=C2)N(C(C)C)C1=O	C42H45ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-4JO0UG	SCHEMBL24717923	2-[6-[[5-chloro-2-[6-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperazin-1-yl]methyl]-3-azabicyclo[3.1.0]hexan-3-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=C(Cl)C=NC(N4CC5C(CN6CCN(C7=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=CC=C7)CC6)C5C4)=N3)=C2)N(C(C)C)C1=O	C42H45ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-G052SR	SCHEMBL24717436	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-6-propan-2-yloxyisoindol-5-yl]piperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL29152564	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CCC(C7=CC8=C(C=C7OC(C)C)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C49H58ClN9O9	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-D9H1P2	SCHEMBL27219543	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-6-methoxy-1,3-dioxoisoindol-5-yl]piperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27231467	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCC(C7=C(OC)C=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H54ClN9O9	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-H2D29U	SCHEMBL24717687	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-2,7-diazaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-5-fluoro-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30798304	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CCC6(CC5)CN(C5=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C5)C6)CC4)=NC=C3Cl)=C2F)N(C(C)C)C1=O	C45H52ClFN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-LQ8RXY	SCHEMBL24717790	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-4-fluoro-1-oxo-3H-isoindol-5-yl]-3,3-dimethyl-2,7-diazaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30798451	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CCC6(CC5)CN(C5=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C5F)C6(C)C)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H56ClFN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-ESTGRO	SCHEMBL24717788	2-[6-[[5-chloro-2-[4-[3-[4-[4-chloro-2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL29152536	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCC(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7Cl)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H53Cl2N9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-MXM1MF	SCHEMBL24717434	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-4-fluoro-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27231359	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCN(C7=C(F)C8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H52ClFN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-2Y4C94	SCHEMBL24717692	2-[6-[[5-chloro-2-[4-[1-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]cyclohexyl]azetidin-3-yl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL24718251; SCHEMBL30798418	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(OC5CN([C@H]6CC[C@H](C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H54ClN9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-87YYGM	SCHEMBL24718693	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-4-methyl-1,3-dioxoisoindol-5-yl]piperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL29152515	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCC(C7=C(C)C8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H54ClN9O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-0VGTLD	SCHEMBL24718697	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-2,9-diazadispiro[3.1.56.14]dodecan-9-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30798447	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CCC6(CC5)CC5(CN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7)C5)C6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C48H57ClN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-7XNTLF	SCHEMBL27219618	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]-2-azaspiro[3.5]nonan-7-yl]methyl]piperazin-1-yl]pyrimidin-4-yl]amino]-5-fluoro-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCN(CC5CCC6(CC5)CN(C5=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C5)C6)CC4)=NC=C3Cl)=C2F)N(C(C)C)C1=O	C45H50ClFN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-ZCEBEW	SCHEMBL29337974	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-3,3-dimethylpiperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CCN(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8)C(C)(C)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H57ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-Z8KETS	SCHEMBL27219607	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-5,5-difluoro-2,7-diazaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-5-fluoro-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894412	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CCC6(CN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7)C6)C(F)(F)C5)CC4)=NC=C3Cl)=C2F)N(C(C)C)C1=O	C45H50ClF3N10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-JH2FYY	SCHEMBL27219633	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-5-fluoro-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27231634	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CCC(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)C5)CC4)=NC=C3Cl)=C2F)N(C(C)C)C1=O	C46H51ClFN9O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-HSWGWI	SCHEMBL24718158	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-4-fluoro-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-5-fluoro-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27220384	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CCC(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7F)CC6)C5)CC4)=NC=C3Cl)=C2F)N(C(C)C)C1=O	C46H52ClF2N9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-CUBR2Y	SCHEMBL24717738	2-[6-[[5-chloro-2-[4-[3-[(3S,5R)-4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-3,5-dimethylpiperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27231404; SCHEMBL30798573	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6C[C@@H](C)N(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8)[C@@H](C)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H57ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-BALPBB	SCHEMBL27219616	2-[6-[[5-chloro-2-[4-[3-[(3R)-4-[2-(2,6-dioxopiperidin-3-yl)-4-fluoro-1-oxo-3H-isoindol-5-yl]-3-methylpiperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27231629	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7F)[C@H](C)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H54ClFN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-YWCF3E	SCHEMBL24717571	2-[6-[[5-chloro-2-[4-[3-[(3S)-4-[2-(2,6-dioxopiperidin-3-yl)-4-fluoro-1-oxo-3H-isoindol-5-yl]-3-methylpiperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27220358	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7F)[C@@H](C)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H54ClFN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-MLMQXE	SCHEMBL24717791	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-4-methyl-1,3-dioxoisoindol-5-yl]piperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27231351	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7C)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H53ClN10O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-ZX954Y	SCHEMBL27219564	2-[6-[[5-chloro-2-[4-[3-[(2S)-4-[2-(2,6-dioxopiperidin-3-yl)-4-fluoro-1-oxo-3H-isoindol-5-yl]-2-methylpiperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27231427	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7F)C[C@@H]6C)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H54ClFN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-IW41CB	SCHEMBL27219559	2-[6-[[5-chloro-2-[4-[3-[(3R,5R)-4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-3,5-dimethylpiperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27231593	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6C[C@@H](C)N(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8)[C@H](C)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H57ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-MMKIYV	SCHEMBL29338092	2-[6-[[5-chloro-2-[4-[3-[(3S,5S)-4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-3,5-dimethylpiperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6C[C@H](C)N(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8)[C@@H](C)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H57ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-4BPL78	SCHEMBL24717752	2-[6-[[5-chloro-2-[4-[3-[4-[4-chloro-2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7Cl)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H52Cl2N10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-5WZ4G5	SCHEMBL24718767	2-[6-[[5-chloro-2-[4-[3-[(2R)-4-[2-(2,6-dioxopiperidin-3-yl)-4-fluoro-1-oxo-3H-isoindol-5-yl]-2-methylpiperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27232797	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7F)C[C@H]6C)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H54ClFN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-35H4O3	SCHEMBL27219614	2-[6-[[5-chloro-2-[4-[1-[4-[2-(2,6-dioxopiperidin-3-yl)-4-fluoro-1-oxo-3H-isoindol-5-yl]cyclohexyl]azetidin-3-yl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27219649; SCHEMBL27231371; SCHEMBL30894187	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(OC5CN([C@H]6CC[C@@H](C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7F)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H53ClFN9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-I6LKO0	SCHEMBL27219588	2-[6-[[5-chloro-2-[4-[1-[4-[4-chloro-2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]cyclohexyl]azetidin-3-yl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27231384; SCHEMBL29338130; SCHEMBL30894127	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(OC5CN([C@H]6CC[C@@H](C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7Cl)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H53Cl2N9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-J2RYDY	SCHEMBL24718265	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-4-fluoro-1-oxo-3H-isoindol-5-yl]-3,3-dimethylpiperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCC(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7F)C(C)(C)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C48H57ClFN9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-CG6Y2F	SCHEMBL24717925	2-[6-[[5-chloro-2-[4-[3-[4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-4,7-difluoro-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30798476	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCC(C7=C(F)C8=C(C(=O)N([C@H]9CCC(=O)NC9=O)C8)C(F)=C7)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H52ClF2N9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-80X2Y9	SCHEMBL24717784	2-[6-[[5-chloro-2-[4-[3-[4-[6-(2,6-dioxopiperidin-3-yl)-5-oxo-7H-pyrrolo[3,4-b]pyridin-2-yl]piperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27092892	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=N7)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C44H52ClN11O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-V1ULIC	SCHEMBL24717449	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-4-fluoro-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-1-cyclobutyl-2-oxoquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCC(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7F)CC6)C5)CC4)=NC=C3Cl)=C2)N(C2CCC2)C1=O	C47H53ClFN9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-1CIZZZ	SCHEMBL24717924	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-4-fluoro-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-1-cyclopentyl-2-oxoquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCC(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7F)CC6)C5)CC4)=NC=C3Cl)=C2)N(C2CCCC2)C1=O	C48H55ClFN9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-E6IWGZ	SCHEMBL29338244	2-[6-[[5-chloro-2-[4-[3-[(3S)-4-[6-(2,6-dioxopiperidin-3-yl)-5-oxo-7H-pyrrolo[3,4-b]pyridin-2-yl]-3-methylpiperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=N7)[C@@H](C)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H54ClN11O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-VA983A	SCHEMBL24718710	2-[6-[[5-chloro-2-[4-[3-[(3R)-4-[2-(2,6-dioxopiperidin-3-yl)-4-methyl-1,3-dioxoisoindol-5-yl]-3-methylpiperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27092900	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7C)[C@H](C)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H55ClN10O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-ZJW1V0	SCHEMBL27219635	2-[6-[[5-chloro-2-[4-[3-[(2S)-4-[2-(2,6-dioxopiperidin-3-yl)-4-methyl-1,3-dioxoisoindol-5-yl]-2-methylpiperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27231379	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7C)C[C@@H]6C)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H55ClN10O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-VXNA6E	SCHEMBL24717916	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-4-methyl-1,3-dioxoisoindol-5-yl]piperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-5-fluoro-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27231733	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7C)CC6)C5)CC4)=NC=C3Cl)=C2F)N(C(C)C)C1=O	C46H52ClFN10O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-TTVH4R	SCHEMBL27219544	2-[6-[[5-chloro-2-[4-[3-[(3S)-4-[4-chloro-2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-3-ethylpiperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27231658	CC[C@H]1CN([C@H]2C[C@H](OC3CCN(C4=NC=C(Cl)C(NC5=CC6=C(C=C5)N(C(C)C)C(=O)C(OCC(=O)NC)=C6)=N4)CC3)C2)CCN1C1=CC=C2C(=O)N(C3CCC(=O)NC3=O)CC2=C1Cl	C47H56Cl2N10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-JLQS0Y	SCHEMBL27219553	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-4-methyl-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27231426	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CCC(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7C)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H56ClN9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-IHY50H	SCHEMBL27219561	2-[6-[[5-chloro-2-[4-[3-[(3R)-4-[6-(2,6-dioxopiperidin-3-yl)-5-oxo-7H-pyrrolo[3,4-b]pyridin-2-yl]-3-methylpiperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27219636	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=N7)[C@H](C)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H54ClN11O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-9R6DRC	SCHEMBL27219626	2-[6-[[5-chloro-2-[4-[3-[(3R)-4-[2-(2,6-dioxopiperidin-3-yl)-4-methyl-1,3-dioxoisoindol-5-yl]-3-methylpiperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-5-fluoro-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27231665	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7C)[C@H](C)C6)C5)CC4)=NC=C3Cl)=C2F)N(C(C)C)C1=O	C47H54ClFN10O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-SVLXO6	SCHEMBL24717840	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-4-ethyl-1,3-dioxoisoindol-5-yl]piperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27220377	CCC1=C2C(=O)N(C3CCC(=O)NC3=O)C(=O)C2=CC=C1N1CCN([C@H]2C[C@H](OC3CCN(C4=NC=C(Cl)C(NC5=CC6=C(C=C5)N(C(C)C)C(=O)C(OCC(=O)NC)=C6)=N4)CC3)C2)CC1	C47H55ClN10O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-QQRHNB	SCHEMBL27219581	2-[6-[[5-chloro-2-[4-[3-[(3R,4S)-4-[2-(2,6-dioxopiperidin-3-yl)-4-fluoro-1-oxo-3H-isoindol-5-yl]-3-fluoropiperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27232590	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CC[C@@H](C7=C(F)C8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8)[C@@H](F)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H52ClF2N9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-B2WFU0	SCHEMBL27219613	2-[6-[[5-chloro-2-[4-[3-[(3R)-4-[4-chloro-2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-3-methylpiperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27231348	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7Cl)[C@H](C)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H54Cl2N10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-F3SWD0	SCHEMBL24718267	2-[6-[[5-chloro-2-[4-[3-[(3R)-4-[6-(2,6-dioxopiperidin-3-yl)-7-methyl-5-oxo-7H-pyrrolo[3,4-b]pyridin-2-yl]-3-methylpiperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL29152534	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(C)C8=N7)[C@H](C)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H56ClN11O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-6W0O9F	SCHEMBL29338352	2-[6-[[5-chloro-2-[4-[3-[(3S)-4-[6-(2,6-dioxopiperidin-3-yl)-7-methyl-5-oxo-7H-pyrrolo[3,4-b]pyridin-2-yl]-3-methylpiperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(C)C8=N7)[C@@H](C)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H56ClN11O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-GQRZUI	SCHEMBL24718135	2-[6-[[5-chloro-2-[4-[3-[(3R)-4-[4-chloro-2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-3-ethylpiperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CC[C@@H]1CN([C@H]2C[C@H](OC3CCN(C4=NC=C(Cl)C(NC5=CC6=C(C=C5)N(C(C)C)C(=O)C(OCC(=O)NC)=C6)=N4)CC3)C2)CCN1C1=CC=C2C(=O)N(C3CCC(=O)NC3=O)CC2=C1Cl	C47H56Cl2N10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-0NSJXE	SCHEMBL24718124	2-[6-[[5-chloro-2-[4-[3-[(3S)-4-[4-chloro-2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-3-methylpiperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7Cl)[C@@H](C)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H54Cl2N10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-9WCY61	SCHEMBL27219576	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-4-fluoro-7-methyl-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27231355	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCC(C7=CC(C)=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7F)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H55ClFN9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-FVB4T7	SCHEMBL27219623	2-[6-[[5-chloro-2-[4-[3-[(4R)-4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-4-fluoro-1-oxo-3H-isoindol-5-yl]-3,3-dimethylpiperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27232087; SCHEMBL30894408	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CC[C@@H](C7=CC=C8C(=O)N([C@H]9CCC(=O)NC9=O)CC8=C7F)C(C)(C)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C48H57ClFN9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-FR7IH4	SCHEMBL27219565	2-[6-[[5-chloro-2-[4-[3-[(4S)-4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-4-fluoro-1-oxo-3H-isoindol-5-yl]-3,3-dimethylpiperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27231354; SCHEMBL30894181	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CC[C@H](C7=CC=C8C(=O)N([C@H]9CCC(=O)NC9=O)CC8=C7F)C(C)(C)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C48H57ClFN9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-8B1PW8	SCHEMBL24717483	2-[6-[[5-chloro-2-[4-[3-[4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]-3,3-dimethylpiperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30798407	CNC(=O)COC1=CC2=C(C=CC(NC3=C(Cl)C=NC(N4CCC(O[C@H]5C[C@@H](N6CCN(C7=CC8=C(C=C7)C(=O)N([C@H]7CCC(=O)NC7=O)C8)C(C)(C)C6)C5)CC4)=N3)=C2)N(C(C)C)C1=O	C47H57ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-SCXJC4	SCHEMBL24717948	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-6-(trifluoromethyl)-3H-isoindol-5-yl]piperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CCC(C7=C(C(F)(F)F)C=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H53ClF3N9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-TYQJFR	SCHEMBL27219551	2-[6-[[5-chloro-2-[4-[[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-3-fluoropiperidin-1-yl]azetidin-1-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894366	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CC(N6CCC(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)C(F)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H52ClFN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-RLBRXG	SCHEMBL24717945	2-[6-[[5-chloro-2-[4-[3-[4-[6-(2,6-dioxopiperidin-3-yl)-5-oxo-7H-pyrrolo[3,4-b]pyridin-2-yl]piperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCC(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=N7)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H53ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-0U4FWR	SCHEMBL24717583	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-2,7-diazaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]pyridin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30798540	CNC(=O)COC1=CC2=C(C=CC(NC3=CC(N4CCC(CN5CCC6(CC5)CN(C5=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C5)C6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H52ClN9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-7756HU	SCHEMBL24717581	2-[6-[[5-chloro-2-[4-[3-[4-[6-(2,6-dioxopiperidin-3-yl)-7-oxo-5H-pyrrolo[3,4-b]pyridin-3-yl]piperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCC(C7=CN=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H53ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-RXDF3C	SCHEMBL27219597	2-[6-[[5-chloro-2-[4-[[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-3-fluoropiperidin-1-yl]azetidin-1-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894283	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CC(N6CCC(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7)C(F)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H54ClFN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-F8N64E	SCHEMBL24718294	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-3,3-difluoropiperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL29152488	CNC(=O)COC1=CC2=C(C=CC(NC3=C(Cl)C=NC(N4CCC(O[C@H]5C[C@H](N6CCC(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8)C(F)(F)C6)C5)CC4)=N3)=C2)N(C(C)C)C1=O	C46H52ClF2N9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-0F5YUO	SCHEMBL24717845	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-3-oxo-1H-pyrrolo[3,4-c]pyridin-6-yl]piperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCC(C7=NC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H53ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-PQ03EI	SCHEMBL27219641	2-[6-[[5-chloro-2-[4-[6-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]-1,6-diazaspiro[3.3]heptan-1-yl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894334	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(N5CCC56CN(C5CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC5)C6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H54ClN11O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-TFQK0I	SCHEMBL27219628	2-[6-[[5-chloro-2-[4-[6-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]pyrrolidin-3-yl]-1,6-diazaspiro[3.3]heptan-1-yl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894346	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(N5CCC56CN(C5CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)C5)C6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H52ClN11O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-Q5QSKS	SCHEMBL27219554	2-[6-[[5-chloro-2-[4-[6-[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-3-yl]-1,6-diazaspiro[3.3]heptan-1-yl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894255	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(N5CCC56CN(C5CCCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7)C5)C6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H56ClN11O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-JVZAYY	SCHEMBL31225084	2-[6-[[5-chloro-2-[4-[6-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-3-yl]-1,6-diazaspiro[3.3]heptan-1-yl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(N5CCC56CN(C5CCCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)C5)C6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H54ClN11O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-WZJU63	SCHEMBL24718366	2-[6-[[5-chloro-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]-2,7-diazaspiro[3.4]octan-7-yl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894292	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(N5CCC6(C5)CN(C5CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC5)C6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C48H56ClN11O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-EE8UJE	SCHEMBL30798449	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-4-(trideuteriomethoxy)-3H-isoindol-5-yl]-2-azaspiro[3.5]nonan-7-yl]oxy]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	[2H]C([2H])([2H])OC1=C2CN(C3CCC(=O)NC3=O)C(=O)C2=CC=C1N1CC2(CCC(OC3CCN(C4=NC=C(Cl)C(NC5=CC6=C(C=C5)N(C(C)C)C(=O)C(OCC(=O)NC)=C6)=N4)CC3)CC2)C1	C46H54ClN9O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-W7LLNM	SCHEMBL24717595	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-4-(trifluoromethyl)-3H-isoindol-5-yl]piperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCC(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7C(F)(F)F)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H53ClF3N9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-BWKVIA	WO2024151557A1_227	.	[2H]C([2H])([2H])OC1=C2CN(C3CCC(=O)NC3=O)C(=O)C2=CC=C1N1CC2(CCN(CC3CCN(C4=NC=C(Cl)C(NC5=CC6=C(C=C5)N(C(C)C)C(=O)C(OCC(=O)NC)=C6)=N4)CC3)CC2)C1(C)C	C48H59ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-L37QVJ	SCHEMBL27219600	2-[6-[[5-chloro-2-[4-[2-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]-2,7-diazaspiro[3.4]octan-7-yl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894372	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(N5CCC6(CN(CC7CCN(C8=CC=C9C(=O)N(C%10CCC(=O)NC%10=O)C(=O)C9=C8)CC7)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C49H58ClN11O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-MJZWXG	SCHEMBL27219656	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-4-fluoro-1-oxo-3H-isoindol-5-yl]-3,3-dimethyl-2,7-diazaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]pyridin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894240	CNC(=O)COC1=CC2=C(C=CC(NC3=CC(N4CCC(CN5CCC6(CC5)CN(C5=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C5F)C6(C)C)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C48H57ClFN9O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-W8A049	SCHEMBL27219655	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-4-methoxy-1-oxo-3H-isoindol-5-yl]-3,3-dimethyl-2,7-diazaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]pyridin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894302	CNC(=O)COC1=CC2=C(C=CC(NC3=CC(N4CCC(CN5CCC6(CC5)CN(C5=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C5OC)C6(C)C)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C49H60ClN9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-W0WTK9	SCHEMBL27219538	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-5,5-difluoro-2,7-diazaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]pyridin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30798519	CNC(=O)COC1=CC2=C(C=CC(NC3=CC(N4CCC(CN5CCC6(CN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7)C6)C(F)(F)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H52ClF2N9O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-1T0O8S	SCHEMBL24717600	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-4-methoxy-1-oxo-3H-isoindol-5-yl]-5,5-difluoro-2,7-diazaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]pyridin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894274	CNC(=O)COC1=CC2=C(C=CC(NC3=CC(N4CCC(CN5CCC6(CN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7OC)C6)C(F)(F)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H54ClF2N9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-WMYR2W	SCHEMBL24717603	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-3,3-dimethyl-2,7-diazaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]pyridin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30798638	CNC(=O)COC1=CC2=C(C=CC(NC3=CC(N4CCC(CN5CCC6(CC5)CN(C5=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C5)C6(C)C)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C48H58ClN9O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-QN5HG0	SCHEMBL27219660	2-[6-[[5-chloro-2-[4-[6-[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]pyrrolidin-3-yl]-1,6-diazaspiro[3.3]heptan-1-yl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894287	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(N5CCC56CN(C5CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7)C5)C6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H54ClN11O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-M1H692	SCHEMBL24718359	2-[6-[[5-chloro-2-[4-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]-2,7-diazaspiro[3.4]octan-7-yl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894107	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(N5CCC6(C5)CN(C5CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7)CC5)C6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C48H58ClN11O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-QBZ51Y	SCHEMBL27219527	2-[6-[[5-chloro-2-[4-[2-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]-2,7-diazaspiro[3.4]octan-7-yl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894116	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(N5CCC6(CN(CC7CCN(C8=CC=C9C(=O)N(C%10CCC(=O)NC%10=O)CC9=C8)CC7)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C49H60ClN11O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-75723W	SCHEMBL27219605	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-4-fluoro-1-oxo-3H-isoindol-5-yl]-5,5-difluoro-2,7-diazaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]pyridin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894251	CNC(=O)COC1=CC2=C(C=CC(NC3=CC(N4CCC(CN5CCC6(CN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7F)C6)C(F)(F)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H51ClF3N9O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-AWO8QP	SCHEMBL27219562	2-[6-[[5-chloro-2-[4-[6-[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]-1,6-diazaspiro[3.3]heptan-1-yl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894325	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(N5CCC56CN(C5CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7)CC5)C6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H56ClN11O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-A2HHW9	SCHEMBL24717936	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-6,6-dimethyl-2,7-diazaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894157	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CCC6(CN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)C6)CC5(C)C)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H55ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-GHI7WS	SCHEMBL24717944	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-3,3-dimethyl-2,7-diazaspiro[3.5]nonan-7-yl]methyl]-4-fluoropiperidin-1-yl]pyridin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894193	CNC(=O)COC1=CC2=C(C=CC(NC3=CC(N4CCC(F)(CN5CCC6(CC5)CN(C5=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C5)C6(C)C)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C48H57ClFN9O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-TSE223	SCHEMBL27219643	2-[6-[[5-chloro-2-[4-[[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]azetidin-1-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894123	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CC(N6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H52ClN11O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-LPSSV1	SCHEMBL27219630	2-[6-[[5-chloro-2-[4-[[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]azetidin-1-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894143	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CC(N6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H54ClN11O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-6XTPF9	SCHEMBL27219659	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyridin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27231382	CNC(=O)COC1=CC2=C(C=CC(NC3=CC(N4CCC(O[C@H]5C[C@H](N6CCC(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H53ClN8O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-H1O9CX	SCHEMBL27219563	2-[6-[[5-chloro-2-[4-[3-[(3R,5S)-4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-3,5-dimethylpiperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27220359	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6C[C@@H](C)N(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)[C@@H](C)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H55ClN10O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-E3AEKG	SCHEMBL27219652	2-[6-[[5-chloro-2-[4-[3-[(3R,5R)-4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-3,5-dimethylpiperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27232209	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6C[C@@H](C)N(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)[C@H](C)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H55ClN10O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-6L9OX5	SCHEMBL24717824	2-[6-[[5-chloro-2-[4-[3-[(3S,5S)-4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-3,5-dimethylpiperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6C[C@H](C)N(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)[C@@H](C)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H55ClN10O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-7FA4MD	SCHEMBL24717823	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]-2-azaspiro[3.5]nonan-7-yl]methyl]piperazin-1-yl]pyridin-4-yl]amino]-5-fluoro-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894347	CNC(=O)COC1=CC2=C(C=CC(NC3=CC(N4CCN(CC5CCC6(CC5)CN(C5=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C5)C6)CC4)=NC=C3Cl)=C2F)N(C(C)C)C1=O	C46H51ClFN9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-L6YTHA	SCHEMBL27219601	2-[6-[[5-chloro-2-[4-[3-[(2R,6R)-4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-2,6-dimethylpiperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27220380	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6[C@H](C)CN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)C[C@H]6C)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H55ClN10O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-ULM7SS	SCHEMBL24717463	2-[6-[[5-chloro-2-[4-[3-[(2R,6S)-4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-2,6-dimethylpiperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30798472	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6[C@H](C)CN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)C[C@@H]6C)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H55ClN10O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-659O3F	WO2024151557A1_250	.	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6[C@H](C)CN(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8)C[C@@H]6C)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H57ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-2MWN5U	SCHEMBL27219590	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-5,5-difluoro-2,7-diazaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]pyridin-4-yl]amino]-5-fluoro-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30798550	CNC(=O)COC1=CC2=C(C=CC(NC3=CC(N4CCC(CN5CCC6(CN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7)C6)C(F)(F)C5)CC4)=NC=C3Cl)=C2F)N(C(C)C)C1=O	C46H51ClF3N9O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-8JZTLX	SCHEMBL24717926	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-4-fluoro-1-oxo-3H-isoindol-5-yl]-5,5-difluoro-2,7-diazaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]pyridin-4-yl]amino]-5-fluoro-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894174	CNC(=O)COC1=CC2=C(C=CC(NC3=CC(N4CCC(CN5CCC6(CN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7F)C6)C(F)(F)C5)CC4)=NC=C3Cl)=C2F)N(C(C)C)C1=O	C46H50ClF4N9O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-6K79ZK	SCHEMBL24717927	2-[6-[[5-chloro-2-[4-[3-[(2S,6S)-4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-2,6-dimethylpiperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6[C@@H](C)CN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)C[C@@H]6C)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H55ClN10O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-KMRB6U	SCHEMBL24718751	2-[6-[[5-chloro-2-[4-[3-[(2S,6S)-4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-2,6-dimethylpiperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6[C@@H](C)CN(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8)C[C@@H]6C)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H57ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-UF6D7L	SCHEMBL27219579	2-[6-[[5-chloro-2-[4-[[(6S,8S)-2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-6,8-dimethyl-2,7-diazaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894382	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5[C@@H](C)CC6(C[C@@H]5C)CN(C5=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C5)C6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H55ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-6BT6VM	SCHEMBL27219541	2-[6-[[5-chloro-2-[4-[3-[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]pyrrolidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27231424	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCC(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H50ClN9O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-W00L0G	SCHEMBL27219540	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-4-fluoro-1-oxo-3H-isoindol-5-yl]-3,3-dimethyl-2,7-diazaspiro[3.5]nonan-7-yl]methyl]-4-fluoropiperidin-1-yl]pyridin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894203	CNC(=O)COC1=CC2=C(C=CC(NC3=CC(N4CCC(F)(CN5CCC6(CC5)CN(C5=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C5F)C6(C)C)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C48H56ClF2N9O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-1LE0IL	SCHEMBL24717939	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-4-fluoro-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyridin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=CC(N4CCC(O[C@H]5C[C@H](N6CCC(C7=C(F)C8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H54ClFN8O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-DF22RL	SCHEMBL24718356	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-4-fluoro-1-oxo-3H-isoindol-5-yl]-2,7-diazaspiro[3.5]nonan-7-yl]methyl]-4-fluoropiperidin-1-yl]pyridin-4-yl]amino]-5-fluoro-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894229	CNC(=O)COC1=CC2=C(C=CC(NC3=CC(N4CCC(F)(CN5CCC6(CC5)CN(C5=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C5F)C6)CC4)=NC=C3Cl)=C2F)N(C(C)C)C1=O	C46H51ClF3N9O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-7LE55C	SCHEMBL24718357	2-[6-[[5-chloro-2-[4-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-4-fluoro-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]azetidin-3-yl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30798582	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(OC5CN(C6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7F)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H52ClFN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-IX8QAU	SCHEMBL24717797	2-[6-[[5-chloro-2-[4-[3-[(2S)-4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-2-methylpiperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)C[C@@H]6C)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H53ClN10O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-Z0I2IH	SCHEMBL27219535	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-2,7-diazaspiro[3.5]nonan-7-yl]methyl]-4-fluoropiperidin-1-yl]pyridin-4-yl]amino]-5-fluoro-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894248	CNC(=O)COC1=CC2=C(C=CC(NC3=CC(N4CCC(F)(CN5CCC6(CC5)CN(C5=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C5)C6)CC4)=NC=C3Cl)=C2F)N(C(C)C)C1=O	C46H52ClF2N9O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-LR1YQQ	SCHEMBL24718776	2-[6-[[5-chloro-2-[4-[3-[(2R)-4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-2-methylpiperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)C[C@H]6C)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H53ClN10O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-RQ9QZK	SCHEMBL24718777	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-4-fluoro-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxyacetic acid	CC(C)N1C(=O)C(OCC(=O)O)=CC2=C1C=CC(NC1=NC(N3CCC(O[C@H]4C[C@@H](N5CCC(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6F)CC5)C4)CC3)=NC=C1Cl)=C2	C45H50ClFN8O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-CG6OI3	SCHEMBL27219627	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-4-fluoro-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-hydroxy-N-methylacetamide; SCHEMBL27231736	CC(C)N1C(=O)C(OCC(=O)N(C)O)=CC2=C1C=CC(NC1=NC(N3CCC(O[C@H]4C[C@H](N5CCC(C6=C(F)C7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)CC5)C4)CC3)=NC=C1Cl)=C2	C46H53ClFN9O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-LU2VT3	SCHEMBL27219637	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-6-methoxy-4-methyl-1,3-dioxoisoindol-5-yl]piperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27232756	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCN(C7=C(OC)C=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7C)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H55ClN10O9	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-NH1HR7	SCHEMBL24718715	2-[6-[[5-chloro-2-[4-[3-[(3R)-4-[4-chloro-2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]-3-methylpiperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30798591	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCN(C7=CC=C8C(=O)N([C@H]9CCC(=O)NC9=O)CC8=C7Cl)[C@H](C)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H54Cl2N10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-8PFOQK	SCHEMBL24718713	2-[6-[[5-chloro-2-[4-[3-[(3R)-4-[4-chloro-2-[(3R)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]-3-methylpiperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30798521	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCN(C7=CC=C8C(=O)N([C@@H]9CCC(=O)NC9=O)CC8=C7Cl)[C@H](C)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H54Cl2N10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-KL8HGW	SCHEMBL24718055	2-[6-[[5-chloro-2-[4-[3-[(3R)-4-[6-chloro-2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]-3-methylpiperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30798329	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCN(C7=C(Cl)C=C8C(=O)N([C@H]9CCC(=O)NC9=O)CC8=C7)[C@H](C)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H54Cl2N10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-6XV12C	SCHEMBL27219531	2-[6-[[5-chloro-2-[4-[3-[(3R)-4-[(3S)-2-[(3S)-2,6-dioxopiperidin-3-yl]-4-fluoro-3-methyl-1-oxo-3H-isoindol-5-yl]-3-methylpiperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27231959; SCHEMBL30894363	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCN(C7=C(F)C8=C(C=C7)C(=O)N([C@H]7CCC(=O)NC7=O)[C@H]8C)[C@H](C)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H56ClFN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-26OREK	SCHEMBL24718149	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-4-propan-2-yl-3H-isoindol-5-yl]-2,7-diazaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30798579	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CCC6(CC5)CN(C5=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C5C(C)C)C6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C48H59ClN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-PHWXQU	SCHEMBL24718157	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-4,7-difluoro-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCN(C7=CC(F)=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7F)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H51ClF2N10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-6MY257	SCHEMBL27219642	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-6,7-difluoro-3-oxo-1H-isoindol-4-yl]piperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27231472	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCN(C7=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C(F)C(F)=C7)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H51ClF2N10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-I1V9QZ	SCHEMBL24717860	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-4-hydroxypiperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CCC(O)(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H52ClN9O9	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-0Z8MXG	SCHEMBL24718297	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-4-fluoropiperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CCC(F)(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H51ClFN9O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-4F914I	SCHEMBL27219575	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-4-fluoro-1-oxo-3H-isoindol-5-yl]-4-hydroxypiperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27231770	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CCC(O)(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7F)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H53ClFN9O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-6UB4GD	SCHEMBL27219653	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-4-fluoro-1-oxo-3H-isoindol-5-yl]-4-fluoropiperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27232885	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CCC(F)(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7F)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H52ClF2N9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-F9LL99	WO2024151557A1_279	.	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CC[C@@H](C7=C(F)C8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8)[C@H](OC)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H55ClFN9O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-L2PZCN	SCHEMBL24718714	2-[6-[[5-chloro-2-[4-[3-[6-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-3-azabicyclo[4.1.0]heptan-3-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CCC7(C8=CC=C9C(=O)N(C%10CCC(=O)NC%10=O)C(=O)C9=C8)CC7C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H52ClN9O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-FLHX0V	SCHEMBL24718362	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-7-fluoro-3-oxo-1H-isoindol-5-yl]-3-fluoropiperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCC(C7=CC8=C(CN(C9CCC(=O)NC9=O)C8=O)C(F)=C7)C(F)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H52ClF2N9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-LYQNLP	SCHEMBL27219525	2-[6-[[5-chloro-2-[4-[3-[(3S,4R)-4-[2-(2,6-dioxopiperidin-3-yl)-4-fluoro-1-oxo-3H-isoindol-5-yl]-3-hydroxypiperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27231360	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CC[C@H](C7=C(F)C8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8)[C@H](O)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H53ClFN9O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-H3ODWD	SCHEMBL27219566	2-[6-[[5-chloro-2-[4-[3-[6-[2-(2,6-dioxopiperidin-3-yl)-4-fluoro-1-oxo-3H-isoindol-5-yl]-3-azabicyclo[4.1.0]heptan-3-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27232648	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CCC7(C8=CC=C9C(=O)N(C%10CCC(=O)NC%10=O)CC9=C8F)CC7C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H53ClFN9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-ESTUOS	SCHEMBL27219604	2-[6-[[5-chloro-2-[4-[3-[(3R,4R)-4-[2-(2,6-dioxopiperidin-3-yl)-4-fluoro-1-oxo-3H-isoindol-5-yl]-3-hydroxypiperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27220383	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CC[C@H](C7=C(F)C8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8)[C@@H](O)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H53ClFN9O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-F1NURR	SCHEMBL27219560	2-[6-[[5-chloro-2-[4-[[3-[4-[2-(2,6-dioxopiperidin-3-yl)-4-fluoro-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]azetidin-1-yl]methyl]-4-fluoropiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894170	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(F)(CN5CC(N6CCC(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7F)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H53ClF2N10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-FSCI40	SCHEMBL24717870	2-[6-[[5-chloro-2-[4-[3-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-4-fluoro-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CCN(CC7CCN(C8=CC=C9C(=O)N(C%10CCC(=O)NC%10=O)CC9=C8F)CC7)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C51H63ClFN11O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-Y91YXC	SCHEMBL27219585	2-[6-[[5-chloro-2-[4-[3-[(3R)-4-[2-(2,6-dioxopiperidin-3-yl)-4-methyl-1,3-dioxoisoindol-5-yl]-3-ethylpiperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27231620	CC[C@@H]1CN([C@H]2C[C@H](OC3CCN(C4=NC=C(Cl)C(NC5=CC6=C(C=C5)N(C(C)C)C(=O)C(OCC(=O)NC)=C6)=N4)CC3)C2)CCN1C1=CC=C2C(=O)N(C3CCC(=O)NC3=O)C(=O)C2=C1C	C48H57ClN10O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-J2RQMV	SCHEMBL27219567	2-[6-[[5-chloro-2-[4-[3-[4-[(3R)-2-[(3S)-2,6-dioxopiperidin-3-yl]-4-fluoro-3-methyl-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27231345; SCHEMBL30894104	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCC(C7=C(F)C8=C(C=C7)C(=O)N([C@H]7CCC(=O)NC7=O)[C@@H]8C)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H55ClFN9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-WI52CS	SCHEMBL27219647	2-[6-[[5-chloro-2-[4-[3-[4-[(3R)-2-(2,6-dioxopiperidin-3-yl)-4-fluoro-3-methyl-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27232609	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCC(C7=C(F)C8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)[C@@H]8C)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H55ClFN9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-7VTX2H	SCHEMBL27219528	2-[6-[[5-chloro-2-[4-[3-[4-[(3S)-2-[(3S)-2,6-dioxopiperidin-3-yl]-4-fluoro-3-methyl-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27231364; SCHEMBL30894222	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCC(C7=CC=C8C(=O)N([C@H]9CCC(=O)NC9=O)[C@@H](C)C8=C7F)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H55ClFN9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-TZMUIJ	SCHEMBL27219609	2-[6-[[5-chloro-2-[4-[3-[4-[(3S)-2-(2,6-dioxopiperidin-3-yl)-4-fluoro-3-methyl-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27231533	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCC(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)[C@@H](C)C8=C7F)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H55ClFN9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-YZOYOG	SCHEMBL27219631	2-[6-[[5-chloro-2-[4-[3-[(2S,4R)-4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-4-fluoro-1-oxo-3H-isoindol-5-yl]-2-methylpiperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27231356; SCHEMBL30894410	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CC[C@@H](C7=CC=C8C(=O)N([C@H]9CCC(=O)NC9=O)CC8=C7F)C[C@@H]6C)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H55ClFN9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-HSVLOC	SCHEMBL27219624	2-[6-[[5-chloro-2-[4-[3-[(2S,4S)-4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-4-fluoro-1-oxo-3H-isoindol-5-yl]-2-methylpiperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27232331; SCHEMBL30894211	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CC[C@H](C7=CC=C8C(=O)N([C@H]9CCC(=O)NC9=O)CC8=C7F)C[C@@H]6C)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H55ClFN9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-FVKKS3	SCHEMBL27219620	2-[6-[[5-chloro-2-[4-[3-[(2R,4R)-4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-4-fluoro-1-oxo-3H-isoindol-5-yl]-2-methylpiperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27232856; SCHEMBL30894343	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CC[C@@H](C7=CC=C8C(=O)N([C@H]9CCC(=O)NC9=O)CC8=C7F)C[C@H]6C)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H55ClFN9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-3L3Q5S	SCHEMBL27219572	2-[6-[[5-chloro-2-[4-[3-[(2R,4S)-4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-4-fluoro-1-oxo-3H-isoindol-5-yl]-2-methylpiperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27231940; SCHEMBL30894091	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CC[C@H](C7=CC=C8C(=O)N([C@H]9CCC(=O)NC9=O)CC8=C7F)C[C@H]6C)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H55ClFN9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-M0KLYQ	SCHEMBL24717941	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-4-fluoro-7-methyl-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCN(C7=CC(C)=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7F)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H54ClFN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-TRFV2X	SCHEMBL24717862	2-[6-[[5-chloro-2-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-5-fluoro-1-oxo-3H-isoindol-4-yl]piperidin-4-yl]methyl]piperazin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894205	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCN(CC5CCN(C6=C7CN(C8CCC(=O)NC8=O)C(=O)C7=CC=C6F)CC5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C42H48ClFN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-3ZBW4S	SCHEMBL24717863	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-5-fluoro-1-oxo-3H-isoindol-4-yl]-2-azaspiro[3.5]nonan-7-yl]oxy]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894230	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(OC5CCC6(CC5)CN(C5=C7CN(C8CCC(=O)NC8=O)C(=O)C7=CC=C5F)C6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H51ClFN9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-EMFBX9	SCHEMBL24718165	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1-oxo-3H-isoindol-4-yl]-2-azaspiro[3.5]nonan-7-yl]oxy]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894189	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(OC5CCC6(CC5)CN(C5=C7CN(C8CCC(=O)NC8=O)C(=O)C7=CC(F)=C5)C6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H51ClFN9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-7P3JJS	SCHEMBL27219629	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-5-methoxy-1-oxo-3H-isoindol-4-yl]-2-azaspiro[3.5]nonan-7-yl]oxy]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(OC5CCC6(CC5)CN(C5=C7CN(C8CCC(=O)NC8=O)C(=O)C7=CC=C5OC)C6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H54ClN9O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-DJ8366	SCHEMBL27219548	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-6-methoxy-1-oxo-3H-isoindol-4-yl]-2-azaspiro[3.5]nonan-7-yl]oxy]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(OC5CCC6(CC5)CN(C5=C7CN(C8CCC(=O)NC8=O)C(=O)C7=CC(OC)=C5)C6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H54ClN9O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-JNVJOD	SCHEMBL24718367	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-4-methoxy-1-oxo-3H-isoindol-5-yl]-2,7-diazaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894401	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CCC6(CC5)CN(C5=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C5OC)C6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H55ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-5M1QZ6	SCHEMBL27219537	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-3,6-dihydro-2H-pyridin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27232733	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CC=C(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H50ClN9O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-4DP8CH	SCHEMBL27219625	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-4-yl]-2-azaspiro[3.5]nonan-7-yl]oxy]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(OC5CCC6(CC5)CN(C5=C7CN(C8CCC(=O)NC8=O)C(=O)C7=C(OC)C=C5)C6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H54ClN9O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-QOGLOA	SCHEMBL27219638	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-2-azaspiro[3.5]nonan-7-yl]methyl]piperazin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894279	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCN(CC5CCC6(CC5)CN(C5=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C5)C6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H53ClN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-OKTTR7	SCHEMBL27219555	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1-oxo-3H-isoindol-5-yl]-2-azaspiro[3.5]nonan-7-yl]methyl]piperazin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894160	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCN(CC5CCC6(CC5)CN(C5=C(F)C=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C5)C6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H52ClFN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-4O98LG	SCHEMBL24717604	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-4-fluoro-1-oxo-3H-isoindol-5-yl]-2-azaspiro[3.5]nonan-7-yl]methyl]piperazin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894268	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCN(CC5CCC6(CC5)CN(C5=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C5F)C6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H52ClFN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-3GRK8D	SCHEMBL24717606	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-2-azaspiro[3.5]nonan-7-yl]-methylamino]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894169	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(N(C)C5CCC6(CC5)CN(C5=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C5)C6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H53ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-TH2T03	SCHEMBL27219646	2-[6-[[5-chloro-2-[4-[3-[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-1,6-diazaspiro[3.3]heptan-6-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27231425	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CC7(CCN7C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H53ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-LQIO4K	WO2024151557A1_310	2-[6-[[5-chloro-2-[4-[3-[1-[2-(2,6-dioxopiperidin-3-yl)-3-oxo-1H-isoindol-4-yl]-1,6-diazaspiro[3.3]heptan-6-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CC7(CCN7C7=C8C(=O)N(C9CCC(=O)NC9=O)CC8=CC=C7)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H53ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-IGWMR9	SCHEMBL27219539	2-[6-[[5-chloro-2-[4-[3-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-2,6-diazaspiro[3.3]heptan-6-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27231366	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CC7(CN(C8=CC=C9C(=O)N(C%10CCC(=O)NC%10=O)C(=O)C9=C8)C7)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H51ClN10O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-BS029P	SCHEMBL29339269	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-7-fluoro-1-oxo-3H-isoindol-4-yl]-2-azaspiro[3.5]nonan-7-yl]oxy]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894133	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(OC5CCC6(CC5)CN(C5=C7CN(C8CCC(=O)NC8=O)C(=O)C7=C(F)C=C5)C6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H51ClFN9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-I4JGJ9	SCHEMBL24717949	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]-2-azaspiro[3.5]nonan-7-yl]methyl]piperazin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894262	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCN(CC5CCC6(CC5)CN(C5=C7CN(C8CCC(=O)NC8=O)C(=O)C7=CC=C5)C6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H53ClN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-0T7PL3	SCHEMBL24717877	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-5-fluoro-1-oxo-3H-isoindol-4-yl]-2-azaspiro[3.5]nonan-7-yl]methyl]piperazin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894159	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCN(CC5CCC6(CC5)CN(C5=C7CN(C8CCC(=O)NC8=O)C(=O)C7=CC=C5F)C6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H52ClFN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-VGDP78	SCHEMBL27219556	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1-oxo-3H-isoindol-4-yl]-2-azaspiro[3.5]nonan-7-yl]methyl]piperazin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCN(CC5CCC6(CC5)CN(C5=C7CN(C8CCC(=O)NC8=O)C(=O)C7=CC(F)=C5)C6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H52ClFN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-4C13R6	SCHEMBL27219648	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-7-fluoro-1-oxo-3H-isoindol-4-yl]-2-azaspiro[3.5]nonan-7-yl]methyl]piperazin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCN(CC5CCC6(CC5)CN(C5=C7CN(C8CCC(=O)NC8=O)C(=O)C7=C(F)C=C5)C6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H52ClFN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-HHOBLE	WO2024151557A1_317	2-[6-[[5-chloro-2-[4-[3-[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]-1,6-diazaspiro[3.3]heptan-6-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CC7(CCN7C7=C8CN(C9CCC(=O)NC9=O)C(=O)C8=CC=C7)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H53ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-7ANWSV	SCHEMBL27219587	2-[6-[[5-chloro-2-[4-[[7-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1-oxo-3H-isoindol-5-yl]-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894312	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCN(CC5CC6(CCN(C7=C(F)C=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H52ClFN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-Y1J7C7	SCHEMBL27219603	2-[6-[[5-chloro-2-[4-[[7-[2-(2,6-dioxopiperidin-3-yl)-4-fluoro-1-oxo-3H-isoindol-5-yl]-7-azaspiro[3.5]nonan-2-yl]methyl]piperazin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894349	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCN(CC5CC6(CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7F)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H52ClFN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-8477GD	SCHEMBL24717558	2-[6-[(5-chloro-2-piperidin-1-ylpyrimidin-4-yl)amino]-1-[2-[2-(1-methyl-2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxyethyl]-2-oxoquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894332	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCCCC4)=NC=C3Cl)=C2)N(CCOC2=CC=C3C(=O)N(C4CCC(=O)N(C)C4=O)C(=O)C3=C2)C1=O	C37H37ClN8O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-AVIPRW	SCHEMBL24717557	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-2,7-diazaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]pyridin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894348	CNC(=O)COC1=CC2=C(C=CC(NC3=CC(N4CCC(CN5CCC6(CC5)CN(C5=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C5)C6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H54ClN9O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-KPZP71	SCHEMBL24717858	2-[6-[[5-chloro-2-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-4-fluoro-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894278	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CCN(C6=C(F)C7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)CC5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C42H48ClFN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-2XMX5G	SCHEMBL24717856	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-3,6-dihydro-2H-pyridin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27231659	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CC=C(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H52ClN9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-VE45EE	SCHEMBL24717859	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-4,6-difluoro-1-oxo-3H-isoindol-5-yl]-2-azaspiro[3.5]nonan-7-yl]oxy]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894311	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(OC5CCC6(CC5)CN(C5=C(F)C=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C5F)C6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H50ClF2N9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-U8KAIJ	SCHEMBL27219545	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]-5-fluoro-2,7-diazaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CCC6(CN(C7=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=CC=C7)C6)C(F)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H50ClFN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-H1MWCI	SCHEMBL24717878	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]-5-fluoro-2,7-diazaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894300	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CCC6(CN(C7=C8CN(C9CCC(=O)NC9=O)C(=O)C8=CC=C7)C6)C(F)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H52ClFN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-2OPF11	SCHEMBL24717876	2-[6-[[5-chloro-2-[4-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-5-methoxy-1-oxo-3H-isoindol-4-yl]-2,7-diazaspiro[3.5]nonan-7-yl]propan-2-yl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894380	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(C(C)(C)N5CCC6(CC5)CN(C5=C7CN(C8CCC(=O)NC8=O)C(=O)C7=CC=C5OC)C6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C48H59ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-KCET3P	SCHEMBL27219577	2-[6-[[5-chloro-2-[4-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-6-methoxy-1-oxo-3H-isoindol-4-yl]-2,7-diazaspiro[3.5]nonan-7-yl]propan-2-yl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(C(C)(C)N5CCC6(CC5)CN(C5=C7CN(C8CCC(=O)NC8=O)C(=O)C7=CC(OC)=C5)C6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C48H59ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-Q22ORC	SCHEMBL24717589	2-[6-[[5-chloro-2-[4-[3-[4-[6-chloro-2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27219657	CNC(=O)COC1=CC2=C(C=CC(NC3=C(Cl)C=NC(N4CCC(O[C@H]5C[C@@H](N6CCC(C7=CC8=C(C=C7Cl)C(=O)N(C7CCC(=O)NC7=O)C8)CC6)C5)CC4)=N3)=C2)N(C(C)C)C1=O	C46H53Cl2N9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-3HVZU6	WO2024151557A1_330	2-[6-[[5-chloro-2-[4-[3-[1-[2-(2,6-dioxopiperidin-3-yl)-3-oxo-1H-isoindol-5-yl]-1,6-diazaspiro[3.3]heptan-6-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CC7(CCN7C7=CC=C8CN(C9CCC(=O)NC9=O)C(=O)C8=C7)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H53ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-PO78F2	SCHEMBL24717616	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-4-methoxy-1-oxo-3H-isoindol-5-yl]-2-azaspiro[3.5]nonan-7-yl]methyl]piperazin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894362	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCN(CC5CCC6(CC5)CN(C5=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C5OC)C6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H55ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-RRW38K	SCHEMBL24717617	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-4-fluoro-1-oxo-3H-isoindol-5-yl]-5,5-difluoro-2,7-diazaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894109	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CCC6(CN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7F)C6)C(F)(F)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H50ClF3N10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-QX7MO4	SCHEMBL24718786	2-[6-[[5-chloro-2-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]-1,7-diazaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894353	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CCC6(CC5)CCN6C5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H51ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-27TKHX	SCHEMBL24718785	2-[6-[[5-chloro-2-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]-1,7-diazaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894182	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CCC6(CC5)CCN6C5=C6CN(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H53ClN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-WGA8QK	SCHEMBL24717622	2-[6-[[5-chloro-2-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-1,7-diazaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894184	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CCC6(CC5)CCN6C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H51ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-4Q4C04	SCHEMBL24717623	2-[6-[[5-chloro-2-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-1,7-diazaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894128	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CCC6(CC5)CCN6C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)CC6=C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H53ClN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-8D7TSO	SCHEMBL24717914	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]-3,3-dimethyl-2,7-diazaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894344	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CCC6(CC5)CN(C5=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C5)C6(C)C)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H55ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-PYHZFP	SCHEMBL24717913	2-[6-[[5-chloro-2-[4-[3-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-2,7-diazaspiro[3.4]octan-7-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CCC7(CN(C8=CC=C9C(=O)N(C%10CCC(=O)NC%10=O)C(=O)C9=C8)C7)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H53ClN10O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-DBW0IB	SCHEMBL24717915	2-[6-[[5-chloro-2-[4-[3-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-2,7-diazaspiro[4.4]nonan-7-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27220372	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CCC7(CCN(C8=CC=C9C(=O)N(C%10CCC(=O)NC%10=O)C(=O)C9=C8)C7)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C48H55ClN10O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-WXF0WR	SCHEMBL24718139	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-4-methoxy-1-oxo-3H-isoindol-5-yl]-3,3-dimethyl-2,7-diazaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894414	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CCC6(CC5)CN(C5=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C5OC)C6(C)C)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C48H59ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-WSNYYW	SCHEMBL24718143	2-[6-[[5-chloro-2-[4-[1-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]cyclohexyl]azetidin-3-yl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894416	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(OC5CN([C@H]6CC[C@H](C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H52ClN9O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-TD76CV	SCHEMBL24718778	2-[6-[[5-chloro-2-[4-[[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]cyclobutyl]methyl]piperazin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCN(C[C@H]5C[C@@H](N6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H54ClN11O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-M4X58N	SCHEMBL24718779	2-[6-[[5-chloro-2-[4-[3-[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-3,9-diazaspiro[5.5]undecan-9-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCC7(CCN(C8=CC=C9C(=O)N(C%10CCC(=O)NC%10=O)C(=O)C9=C8)CC7)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C50H59ClN10O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-DCHLGC	SCHEMBL24717929	2-[6-[[5-chloro-2-[4-[3-[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-2,7-diazaspiro[3.4]octan-7-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CCC7(CN(C8=CC=C9C(=O)N(C%10CCC(=O)NC%10=O)CC9=C8)C7)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H55ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-NEZKXU	SCHEMBL24717930	2-[6-[[5-chloro-2-[4-[3-[2-[2-(2,6-dioxopiperidin-3-yl)-3-oxo-1H-isoindol-5-yl]-2,7-diazaspiro[3.4]octan-7-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CCC7(CN(C8=CC=C9CN(C%10CCC(=O)NC%10=O)C(=O)C9=C8)C7)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H55ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-6BZYY5	SCHEMBL24717931	2-[6-[[5-chloro-2-[4-[3-[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-2,7-diazaspiro[4.4]nonan-7-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CCC7(CCN(C8=CC9=C(C=C8)C(=O)N(C8CCC(=O)NC8=O)C9)C7)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C48H57ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-4KUJE7	SCHEMBL24717610	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-2,7-diazaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-5-fluoro-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30798501	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CCC6(CC5)CN(C5=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C5)C6)CC4)=NC=C3Cl)=C2F)N(C(C)C)C1=O	C45H50ClFN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-0ZKTE9	SCHEMBL24717614	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-6-methoxy-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27219571	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCC(C7=C(OC)C=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H56ClN9O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-IRUIQK	SCHEMBL24718768	2-[6-[[5-chloro-2-[4-[3-[3-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-3,9-diazaspiro[5.5]undecan-9-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCC7(CCN(C8=CC=C9C(=O)N(C%10CCC(=O)NC%10=O)CC9=C8)CC7)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C50H61ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-U5PV99	SCHEMBL24718765	2-[6-[[5-chloro-2-[4-[3-[7-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-2,7-diazaspiro[3.4]octan-2-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CC7(CCN(C8=CC=C9C(=O)N(C%10CCC(=O)NC%10=O)C(=O)C9=C8)C7)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H53ClN10O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-JRM5LM	SCHEMBL29339819	2-[6-[[5-chloro-2-[4-[3-[7-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-2,7-diazaspiro[3.4]octan-2-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CC7(CCN(C8=CC9=C(C=C8)C(=O)N(C8CCC(=O)NC8=O)C9)C7)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H55ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-IY4XDB	SCHEMBL27219658	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-4-methoxy-1-oxo-3H-isoindol-5-yl]-5,5-difluoro-2,7-diazaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894333	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CCC6(CN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7OC)C6)C(F)(F)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H53ClF2N10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-HWR1BT	WO2024151557A1_353	2-[6-[[5-chloro-2-[4-[3-[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-2,6-diazaspiro[3.3]heptan-6-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CC7(CN(C8=CC=C9C(=O)N(C%10CCC(=O)NC%10=O)CC9=C8)C7)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H53ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-T9R4WO	SCHEMBL24718364	2-[6-[[5-chloro-2-[4-[3-[7-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-2,7-diazaspiro[4.5]decan-2-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27231955	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CCC7(CCCN(C8=CC9=C(C=C8)C(=O)N(C8CCC(=O)NC8=O)C9)C7)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C49H59ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-CGTCM2	SCHEMBL24718368	2-[6-[[5-chloro-2-[4-[3-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-2,9-diazaspiro[4.5]decan-9-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CCCC7(CCN(C8=CC=C9C(=O)N(C%10CCC(=O)NC%10=O)C(=O)C9=C8)C7)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C49H57ClN10O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-I6OOKW	SCHEMBL24718791	2-[6-[[5-chloro-2-[4-[3-[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-2,9-diazaspiro[4.5]decan-9-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CCCC7(CCN(C8=CC=C9C(=O)N(C%10CCC(=O)NC%10=O)CC9=C8)C7)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C49H59ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-0C939W	SCHEMBL29339850	2-[6-[[5-chloro-2-[4-[3-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-2,7-diazaspiro[3.5]nonan-7-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CCC7(CC6)CN(C6=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C6)C7)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C48H55ClN10O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-0Z5XRQ	SCHEMBL27219550	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-4-methyl-1,3-dioxoisoindol-5-yl]-2,7-diazaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894404	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CCC6(CC5)CN(C5=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C5C)C6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H53ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-6SBTA7	SCHEMBL24718377	2-[6-[[5-chloro-2-[4-[3-[7-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-2,7-diazaspiro[4.5]decan-2-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCC7(CCCN(C8=CC=C9C(=O)N(C%10CCC(=O)NC%10=O)C(=O)C9=C8)C7)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C49H57ClN10O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-XW56M4	SCHEMBL24718375	2-[6-[[5-chloro-2-[4-[3-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-2,8-diazaspiro[4.5]decan-8-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27220361	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CCC7(CCN(C8=CC=C9C(=O)N(C%10CCC(=O)NC%10=O)C(=O)C9=C8)C7)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C49H57ClN10O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-3L9IGE	SCHEMBL24717549	2-[6-[[5-chloro-2-[4-[3-[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-2,8-diazaspiro[4.5]decan-8-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CCC7(CCN(C8=CC=C9C(=O)N(C%10CCC(=O)NC%10=O)CC9=C8)C7)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C49H59ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-ZUPB4T	SCHEMBL24717551	2-[6-[[5-chloro-2-[4-[3-[8-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-2,8-diazaspiro[4.5]decan-2-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CCC7(CCN(C8=CC=C9C(=O)N(C%10CCC(=O)NC%10=O)C(=O)C9=C8)CC7)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C49H57ClN10O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-ML88OY	SCHEMBL24717550	2-[6-[[5-chloro-2-[4-[3-[8-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-2,8-diazaspiro[4.5]decan-2-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27231372	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CCC7(CCN(C8=CC9=C(C=C8)C(=O)N(C8CCC(=O)NC8=O)C9)CC7)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C49H59ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-2MNUTY	SCHEMBL24718137	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-4-ethoxy-1-oxo-3H-isoindol-5-yl]-2-azaspiro[3.5]nonan-7-yl]oxy]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894168	CCOC1=C2CN(C3CCC(=O)NC3=O)C(=O)C2=CC=C1N1CC2(CCC(OC3CCN(C4=NC=C(Cl)C(NC5=CC6=C(C=C5)N(C(C)C)C(=O)C(OCC(=O)NC)=C6)=N4)CC3)CC2)C1	C47H56ClN9O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-3S6O63	SCHEMBL24718138	2-[6-[[5-chloro-2-[4-[3-[7-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-2,7-diazaspiro[3.5]nonan-2-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30798264	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CC7(CCN(C8=CC=C9C(=O)N(C%10CCC(=O)NC%10=O)C(=O)C9=C8)CC7)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C48H55ClN10O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-HBQV8Z	SCHEMBL24718140	2-[6-[[5-chloro-2-[4-[3-[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-2,7-diazaspiro[3.5]nonan-7-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CCC7(CC6)CN(C6=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C6)C7)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C48H57ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-5U12XN	SCHEMBL24718331	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-3,3-dimethylpiperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)C(C)(C)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H55ClN10O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-PSRX18	SCHEMBL24718332	2-[6-[[5-chloro-2-[4-[3-[3-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6C7CCC6CN(C6=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C6)C7)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H55ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-1PF800	SCHEMBL24718758	2-[6-[[5-chloro-2-[4-[3-[7-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-2,7-diazaspiro[3.5]nonan-2-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27231739	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CC7(CCN(C8=CC9=C(C=C8)C(=O)N(C8CCC(=O)NC8=O)C9)CC7)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C48H57ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-V4T1LG	SCHEMBL24718759	2-[6-[[5-chloro-2-[4-[3-[8-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-3,8-diazabicyclo[3.2.1]octan-3-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27220366	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CC7CCC(C6)N7C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H53ClN10O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-YF8838	SCHEMBL24718789	2-[6-[[5-chloro-2-[4-[3-[8-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-3,8-diazabicyclo[3.2.1]octan-3-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27231350	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CC7CCC(C6)N7C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H55ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-TGXKRX	SCHEMBL24718788	2-[6-[[5-chloro-2-[4-[3-[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27231624	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6C7CCC6CN(C6=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C6)C7)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H53ClN10O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-KG68KZ	WO2024151557A1_373	.	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CCC6(CC5)CC5(CN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)C5)C6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C48H55ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-UWTOCD	SCHEMBL30894337	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]-2,9-diazadispiro[3.1.56.14]dodecan-9-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CCC6(CC5)CC5(CN(C7=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=CC=C7)C5)C6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C48H55ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-UQDPAY	SCHEMBL27219546	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-3,3-dimethyl-2,7-diazaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-5-fluoro-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894238	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CCC6(CC5)CN(C5=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C5)C6(C)C)CC4)=NC=C3Cl)=C2F)N(C(C)C)C1=O	C47H54ClFN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-2A5RHV	SCHEMBL27219558	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-4-fluoro-1-oxo-3H-isoindol-5-yl]-5,5-difluoro-2,7-diazaspiro[3.5]nonan-7-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-5-fluoro-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894204	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CCC6(CN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7F)C6)C(F)(F)C5)CC4)=NC=C3Cl)=C2F)N(C(C)C)C1=O	C45H49ClF4N10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-JC35MA	SCHEMBL27219569	2-[6-[[5-chloro-2-[4-[3-[7-[2-(2,6-dioxopiperidin-3-yl)-3-oxo-1H-isoindol-5-yl]-2,7-diazaspiro[3.5]nonan-2-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27231445	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CC7(CCN(C8=CC9=C(C=C8)CN(C8CCC(=O)NC8=O)C9=O)CC7)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C48H57ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-IEDJSS	SCHEMBL24718780	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-7-methyl-1,3-dioxoisoindol-5-yl]piperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27219594	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CCN(C7=CC(C)=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H53ClN10O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-PDSZDD	SCHEMBL24718781	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1,3-dioxoisoindol-5-yl]piperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27219596	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCN(C7=CC(OC)=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H53ClN10O9	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-U9LA73	SCHEMBL24717609	2-[6-[[5-chloro-2-[4-[3-[4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-4-fluoro-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-5-fluoro-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27219634; SCHEMBL30894296	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCC(C7=CC=C8C(=O)N([C@H]9CCC(=O)NC9=O)CC8=C7F)CC6)C5)CC4)=NC=C3Cl)=C2F)N(C(C)C)C1=O	C46H52ClF2N9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-OAMCGO	SCHEMBL24717608	2-[6-[[5-chloro-2-[4-[3-[4-[2-[(3R)-2,6-dioxopiperidin-3-yl]-4-fluoro-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-5-fluoro-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27219580; SCHEMBL30894322	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCC(C7=CC=C8C(=O)N([C@@H]9CCC(=O)NC9=O)CC8=C7F)CC6)C5)CC4)=NC=C3Cl)=C2F)N(C(C)C)C1=O	C46H52ClF2N9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-T39GSV	SCHEMBL24718376	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-3,3-dimethyl-2,7-diazaspiro[3.5]nonan-7-yl]methyl]-4-fluoropiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894288	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(F)(CN5CCC6(CC5)CN(C5=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C5)C6(C)C)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H56ClFN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-UI2CUM	SCHEMBL24718378	2-[6-[[5-chloro-2-[4-[[2-[4-chloro-2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-2-azaspiro[3.5]nonan-7-yl]oxy]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894110	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(OC5CCC6(CC5)CN(C5=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C5Cl)C6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H51Cl2N9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-HDTLTB	SCHEMBL27219574	2-[6-[[5-chloro-2-[4-[3-[4-[2-[(3R)-2,6-dioxopiperidin-3-yl]-4-fluoro-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL29340161; SCHEMBL30798479	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CCC(C7=C(F)C8=C(C=C7)C(=O)N([C@@H]7CCC(=O)NC7=O)C8)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H53ClFN9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-N0ITWS	SCHEMBL27219602	2-[6-[[5-chloro-2-[4-[3-[4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-4-fluoro-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL29340162; SCHEMBL30894095	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CCC(C7=C(F)C8=C(C=C7)C(=O)N([C@H]7CCC(=O)NC7=O)C8)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H53ClFN9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-GL51CZ	SCHEMBL24717605	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-4,6-difluoro-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCN(C7=C(F)C=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7F)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H51ClF2N10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-QIATLE	SCHEMBL27219610	2-[6-[[5-chloro-2-[4-[3-[(3R)-4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-3-methylpiperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)[C@H](C)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H53ClN10O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-M0QV7C	SCHEMBL27219542	2-[6-[[5-chloro-2-[4-[3-[4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-4-fluoro-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894185	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CCN(C7=C(F)C8=C(C=C7)C(=O)N([C@H]7CCC(=O)NC7=O)C8)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H52ClFN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-29GENP	SCHEMBL24718113	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-2,7-diazaspiro[3.5]nonan-7-yl]methyl]-4-fluoropiperidin-1-yl]pyrimidin-4-yl]amino]-5-fluoro-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894094	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(F)(CN5CCC6(CC5)CN(C5=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C5)C6)CC4)=NC=C3Cl)=C2F)N(C(C)C)C1=O	C45H51ClF2N10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-3XNKDH	SCHEMBL24718114	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-4-fluoro-1-oxo-3H-isoindol-5-yl]-2,7-diazaspiro[3.5]nonan-7-yl]methyl]-4-fluoropiperidin-1-yl]pyrimidin-4-yl]amino]-5-fluoro-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894258	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(F)(CN5CCC6(CC5)CN(C5=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C5F)C6)CC4)=NC=C3Cl)=C2F)N(C(C)C)C1=O	C45H50ClF3N10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-813Y0B	SCHEMBL27219619	2-[6-[[5-chloro-2-[4-[3-[(3S)-4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-3-methylpiperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27231378	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)[C@@H](C)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H53ClN10O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-V19B5V	SCHEMBL27219651	2-[6-[[5-chloro-2-[4-[3-[4-[2-[(3R)-2,6-dioxopiperidin-3-yl]-4-fluoro-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30798604	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CCN(C7=C(F)C8=C(C=C7)C(=O)N([C@@H]7CCC(=O)NC7=O)C8)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H52ClFN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-QAOVAM	SCHEMBL24717627	2-[6-[[5-chloro-2-[4-[3-[7-[2-(2,6-dioxopiperidin-3-yl)-4-fluoro-1-oxo-3H-isoindol-5-yl]-2,7-diazaspiro[3.5]nonan-2-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27231724	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CC7(CCN(C8=CC=C9C(=O)N(C%10CCC(=O)NC%10=O)CC9=C8F)CC7)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C48H56ClFN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-TAUCZM	SCHEMBL24717943	2-[6-[[5-chloro-2-[4-[3-[(3R)-4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-4-fluoro-1-oxo-3H-isoindol-5-yl]-3-methylpiperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27220367; SCHEMBL30894286	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCN(C7=CC=C8C(=O)N([C@H]9CCC(=O)NC9=O)CC8=C7F)[C@H](C)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H54ClFN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-1TG13F	SCHEMBL24717951	2-[6-[[5-chloro-2-[4-[3-[(3R)-4-[2-[(3R)-2,6-dioxopiperidin-3-yl]-4-fluoro-1-oxo-3H-isoindol-5-yl]-3-methylpiperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27231389; SCHEMBL30894126	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCN(C7=CC=C8C(=O)N([C@@H]9CCC(=O)NC9=O)CC8=C7F)[C@H](C)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H54ClFN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-MTNYJR	SCHEMBL24717952	2-[6-[[5-chloro-2-[4-[3-[(4R)-4-[2-[(3R)-2,6-dioxopiperidin-3-yl]-4-fluoro-1-oxo-3H-isoindol-5-yl]-3,3-dimethylpiperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27232200; SCHEMBL30894097	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CC[C@@H](C7=CC=C8C(=O)N([C@@H]9CCC(=O)NC9=O)CC8=C7F)C(C)(C)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C48H57ClFN9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-81DMFP	SCHEMBL27219582	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-4-fluoro-6-methyl-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCC(C7=C(C)C=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7F)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H55ClFN9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-7PFNFT	WO2024151557A1_398	.	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CCC(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7F)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H53ClFN9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-ETC24X	SCHEMBL27219536	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-3,3-dimethylpiperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27231429	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCC(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)C(C)(C)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C48H56ClN9O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-O9XCVG	SCHEMBL24717633	2-[6-[[5-chloro-2-[4-[3-[7-[2-(2,6-dioxopiperidin-3-yl)-4-fluoro-1-oxo-3H-isoindol-5-yl]-2,7-diazaspiro[3.4]octan-2-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27232664	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CC7(CCN(C8=C(F)C9=C(C=C8)C(=O)N(C8CCC(=O)NC8=O)C9)C7)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H54ClFN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-PRGJYM	SCHEMBL24717634	2-[6-[[5-chloro-2-[4-[3-[2-[2-(2,6-dioxopiperidin-3-yl)-4-fluoro-1-oxo-3H-isoindol-5-yl]-2,9-diazaspiro[4.5]decan-9-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27231625	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CCCC7(CCN(C8=C(F)C9=C(C=C8)C(=O)N(C8CCC(=O)NC8=O)C9)C7)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C49H58ClFN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-YTI99Q	SCHEMBL24717632	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-4-methyl-1-oxo-3H-isoindol-5-yl]-2-azaspiro[3.5]nonan-7-yl]oxy]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894195	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(OC5CCC6(CC5)CN(C5=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C5C)C6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H54ClN9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-V4LD6W	SCHEMBL24717635	2-[6-[[5-chloro-2-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-4-methyl-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894179	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6C)CC5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C43H49ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-X4X88E	SCHEMBL23267947	2-[6-[[5-chloro-2-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894373	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C42H47ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-0UNKT0	SCHEMBL24717636	2-[6-[[5-chloro-2-[4-[3-[2-[2-(2,6-dioxopiperidin-3-yl)-4-fluoro-1-oxo-3H-isoindol-5-yl]-2,7-diazaspiro[3.4]octan-7-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27231370	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CCC7(CN(C8=C(F)C9=C(C=C8)C(=O)N(C8CCC(=O)NC8=O)C9)C7)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H54ClFN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-RDDHER	SCHEMBL24718163	2-[6-[[5-chloro-2-[4-[3-[3-[2-(2,6-dioxopiperidin-3-yl)-4-fluoro-1-oxo-3H-isoindol-5-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6C7CCC6CN(C6=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C6F)C7)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H54ClFN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-VK1PBU	SCHEMBL24718170	2-[6-[[5-chloro-2-[4-[3-[4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-4-fluoro-7-methoxy-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894132	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCC(C7=C(F)C8=C(C(=O)N([C@H]9CCC(=O)NC9=O)C8)C(OC)=C7)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H55ClFN9O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-Q4XXD1	SCHEMBL27219557	2-[6-[[5-chloro-2-[4-[3-[(3R)-4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]-3-methylpiperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCN(C7=C(F)C=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)[C@H](C)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H52ClFN10O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-47LJKH	SCHEMBL27219573	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-4-fluoro-6-methoxy-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCC(C7=C(OC)C=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7F)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H55ClFN9O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-DSNQYW	SCHEMBL24718168	2-[6-[[5-chloro-2-[4-[3-[2-[2-(2,6-dioxopiperidin-3-yl)-4-fluoro-1-oxo-3H-isoindol-5-yl]-2,7-diazaspiro[3.5]nonan-7-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CCC7(CC6)CN(C6=C(F)C8=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C8)C7)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C48H56ClFN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-68V941	SCHEMBL27219568	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-4-fluoro-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-1-cyclohexyl-2-oxoquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CCC(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7F)CC6)C5)CC4)=NC=C3Cl)=C2)N(C2CCCCC2)C1=O	C49H57ClFN9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-3WOFCD	SCHEMBL27219592	2-[6-[[5-chloro-2-[4-[3-[4-[4-chloro-2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7Cl)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H50Cl2N10O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-8DQMAI	SCHEMBL24718167	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-4-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7F)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C45H50ClFN10O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-JLGGZY	SCHEMBL24717928	2-[6-[[5-chloro-2-[4-[3-[2-[2-(2,6-dioxopiperidin-3-yl)-4-methyl-1,3-dioxoisoindol-5-yl]-2,7-diazaspiro[3.5]nonan-7-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27231387	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CCC7(CC6)CN(C6=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C6C)C7)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C49H57ClN10O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-EMELG9	SCHEMBL27219645	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-4-methyl-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7C)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H55ClN10O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-67SVLJ	SCHEMBL24717628	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-4-methyl-1,3-dioxoisoindol-5-yl]-1,4-diazepan-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27232825	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CCCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7C)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H55ClN10O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-RODNPI	SCHEMBL24717629	2-[6-[[5-chloro-2-[4-[3-[7-[2-(2,6-dioxopiperidin-3-yl)-4-methyl-1,3-dioxoisoindol-5-yl]-2,7-diazaspiro[3.5]nonan-2-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CC7(CCN(C8=CC=C9C(=O)N(C%10CCC(=O)NC%10=O)C(=O)C9=C8C)CC7)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C49H57ClN10O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-S0CW8L	SCHEMBL24717631	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-4-methyl-1,3-dioxoisoindol-5-yl]piperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-5-fluoro-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCC(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7C)CC6)C5)CC4)=NC=C3Cl)=C2F)N(C(C)C)C1=O	C47H53ClFN9O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-DUBIFI	SCHEMBL27219621	2-[6-[[5-chloro-2-[4-[3-[2-[2-(2,6-dioxopiperidin-3-yl)-4-methyl-1,3-dioxoisoindol-5-yl]-2,6-diazaspiro[3.3]heptan-6-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27231416	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CC7(CN(C8=CC=C9C(=O)N(C%10CCC(=O)NC%10=O)C(=O)C9=C8C)C7)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C47H53ClN10O8	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-AE7GUF	SCHEMBL27219524	2-[6-[[5-chloro-2-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-2,9-diazadispiro[3.1.56.14]dodecan-9-yl]methyl]piperidin-1-yl]pyrimidin-4-yl]amino]-5-fluoro-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL30894315	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CCC6(CC5)CC5(CN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7)C5)C6)CC4)=NC=C3Cl)=C2F)N(C(C)C)C1=O	C48H56ClFN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-1YUDUB	SCHEMBL24717885	2-[6-[[5-chloro-2-[4-[3-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-4-fluoro-1-oxo-3H-isoindol-5-yl]azetidin-3-yl]piperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27231344	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CCN(C7CN(C8=CC=C9C(=O)N(C%10CCC(=O)NC%10=O)CC9=C8F)C7)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C48H57ClFN11O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-A1PE52	SCHEMBL27219570	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-6-methoxy-1,3-dioxoisoindol-5-yl]piperazin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCN(C7=C(OC)C=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H53ClN10O9	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-JF3UEK	SCHEMBL27219591	2-[1-butan-2-yl-6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-4-fluoro-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxoquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27231358	CCC(C)N1C(=O)C(OCC(=O)NC)=CC2=C1C=CC(NC1=NC(N3CCC(O[C@H]4C[C@@H](N5CCC(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6F)CC5)C4)CC3)=NC=C1Cl)=C2	C47H55ClFN9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-2D2ESN	SCHEMBL27219615	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-4-fluoro-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-1-(2-methylpropyl)-2-oxoquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27231409	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CCC(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7F)CC6)C5)CC4)=NC=C3Cl)=C2)N(CC(C)C)C1=O	C47H55ClFN9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-G2ZGNT	SCHEMBL27219526	2-[6-[[5-chloro-2-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-4-fluoro-1-oxo-3H-isoindol-5-yl]-3,6-dihydro-2H-pyridin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CC=C(C7=C(F)C8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H51ClFN9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-E8P8S0	WO2024151557A1_427	.	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(CN5CCC6(CC5)CC5(CN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7F)C5)C6)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C48H56ClFN10O6	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-EDML2F	SCHEMBL29340483	2-[6-[[5-chloro-2-[4-[3-[4-[4-chloro-2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]-3,6-dihydro-2H-pyridin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CC=C(C7=CC=C8C(=O)N([C@H]9CCC(=O)NC9=O)CC8=C7Cl)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H51Cl2N9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-NG8QWO	SCHEMBL27219608	2-[6-[[5-chloro-2-[4-[3-[4-[4-chloro-2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-3,6-dihydro-2H-pyridin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27231362	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CC=C(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7Cl)CC6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C46H51Cl2N9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-UG4N89	SCHEMBL24717841	2-[6-[[5-chloro-2-[4-[3-[(4R)-4-[2-(2,6-dioxopiperidin-3-yl)-4-fluoro-1-oxo-3H-isoindol-5-yl]-3,3-dimethylpiperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27231670	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@H](N6CC[C@@H](C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7F)C(C)(C)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C48H57ClFN9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-8CBTHM	SCHEMBL24717842	2-[6-[[5-chloro-2-[4-[3-[(4S)-4-[2-(2,6-dioxopiperidin-3-yl)-4-fluoro-1-oxo-3H-isoindol-5-yl]-3,3-dimethylpiperidin-1-yl]cyclobutyl]oxypiperidin-1-yl]pyrimidin-4-yl]amino]-2-oxo-1-propan-2-ylquinolin-3-yl]oxy-N-methylacetamide; SCHEMBL27231689	CNC(=O)COC1=CC2=C(C=CC(NC3=NC(N4CCC(O[C@H]5C[C@@H](N6CC[C@H](C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7F)C(C)(C)C6)C5)CC4)=NC=C3Cl)=C2)N(C(C)C)C1=O	C48H57ClFN9O7	BCL6	P41182	CRBN	WO-2024151557-A1
TPD-5O91BA	WO2024153025A1_1	.	O=C1CC[C@H](N2Cc3cc(N4CCN(CC5CCN(c6ccc7c(c6)C6COCCC6C6=C7c7ccc(O)cc7CCC6)CC5)CC4)ccc3C2=O)C(=O)N1	C45H51N5O5	ERα	P03372	CRBN	WO-2024153025-A1
TPD-CUDB84	WO2024153025A1_2	.	O=C1CC[C@H](N2Cc3cc(N4CCN(CC5CCN(c6ccc(C7=C(C8CCC(F)(F)CC8)CCCc8cc(O)ccc87)cc6)CC5)CC4)ccc3C2=O)C(=O)N1	C46H53F2N5O4	ERα	P03372	CRBN	WO-2024153025-A1
TPD-96PY1Q	WO2024153025A1_3	.	O=C1CC[C@H](N2Cc3cc(N4CCN(CC5CCN(c6ccc7c(c6)C6CCCCC6C6=C7c7ccc(O)cc7CCC6)CC5)CC4)ccc3C2=O)C(=O)N1	C46H53N5O4	ERα	P03372	CRBN	WO-2024153025-A1
TPD-B5SZSC	WO2024165050A1_1	.	CC1(C)[C@H](NC(=O)C2=CC=C(C(=O)NCCOCCOCCC(=O)NCC3=CC=C(S(=O)(=O)N4CCN(C5=NC=CC(C(F)(F)F)=C5)CC4)C=C3)C=C2)C(C)(C)[C@@H]1OC1=CC=C(C#N)C(Cl)=C1	C47H53ClF3N7O8S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-7A97F8	WO2024165050A1_2	.	CC1(C)C(NC(=O)C2=CC=C(C(=O)NCCCCCCN3CCN(CC4=CC=C(S(=O)(=O)N5CCN(C6=NC=CC(C(F)(F)F)=C6)CC5)C=C4)CC3)C=C2)C(C)(C)C1OC1=CC=C(C#N)C(Cl)=C1	C50H60ClF3N8O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-CZK1IG	WO2024165050A1_3	.	CC1(C)[C@H](NC(=O)C2=CC=C(C(=O)NCCOCCOCCC(=O)NCC3=CC=C(S(=O)(=O)N4CCN(C5=CC(C#N)=CC(C(F)(F)F)=C5)CC4)C=C3)C=C2)C(C)(C)[C@@H]1OC1=CC=C(C#N)C(Cl)=C1	C49H53ClF3N7O8S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-RJTBJO	WO2024165050A1_4	.	CC1[C@H](NC(=O)C2=CC=C(C(=O)NCCOCCOCCN3CCC4=C(C=CC(S(=O)(=O)N5CCN(C6=NC=CC(C(F)(F)F)=C6)CC5)=C4)C3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C47H53ClF3N7O7S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-59DVDH	WO2024165050A1_5	.	CC(=O)C1=CC=C(OC2C(C)(C)C(NC(=O)C3=CC=C(N4CCN(CCOCCOCCC(=O)NCC5=CC=C(S(=O)(=O)N6CCN(C7=NC=CC(C(F)(F)F)=C7)CC6)C=C5)CC4)C=C3)C2(C)C)C=C1Cl	C51H63ClF3N7O8S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-J0O32U	WO2024165050A1_6	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCN(CCCCCCC(=O)NCC4=CC=C(S(=O)(=O)N5CCC(C6=NC=CC(C(F)(F)F)=C6)CC5)C=C4)CC3)C=C2)C(C)(C)[C@@H]1OC1=CC=C(C#N)C(Cl)=C1	C51H61ClF3N7O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-X9G04Z	WO2024165050A1_7	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCN(CCCCCCC(=O)NCC4=CC=C(S(=O)(=O)N5CCN(C6=CC=CC(C(F)(F)F)=C6)CC5)C=C4)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C51H61ClF3N7O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-WPGRFO	WO2024165050A1_8	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCN(CCCCCCC(=O)NCC4=CC=C(S(=O)(=O)N5CCN(C6=NC=CC(C(F)(F)F)=C6)CC5)C=N4)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C49H59ClF3N9O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-KVR17M	WO2024165050A1_9	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCN(CCCCCCC(=O)NCC4=CC=C(S(=O)(=O)N5CCN(C6=NC=CC(C(F)(F)F)=C6)CC5)C=C4)CC3)C=C2)C(C)(C)[C@@H]1OC1=CC=C(C#N)C(Cl)=C1	C50H60ClF3N8O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-6OB3ZR	WO2024165050A1_10	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCN(CCCCCCC(=O)N4CCC(S(=O)(=O)N5CCN(C6=NC=CC(C(F)(F)F)=C6)CC5)CC4)CC3)C=C2)C(C)(C)[C@@H]1OC1=CC=C(C#N)C(Cl)=C1	C48H62ClF3N8O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-H1HFWJ	WO2024165050A1_11	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCN(CCCCCCC(=O)NCCCS(=O)(=O)N4CCN(C5=NC=CC(C(F)(F)F)=C5)CC4)CC3)C=C2)C(C)(C)[C@@H]1OC1=CC=C(C#N)C(Cl)=C1	C46H60ClF3N8O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-437CDF	WO2024165050A1_12	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCN(CCCCCCC(=O)NCC4=CC=C(C(=O)N5CCN(C6=NC=CC(C(F)(F)F)=C6)CC5)C=C4)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C51H60ClF3N8O4	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-VC9ZVO	WO2024165050A1_13	.	CC(=O)C1=CC=C(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCN(CCCCCCC(=O)NCC5CCC(S(=O)(=O)N6CCN(C7=NC=CC(C(F)(F)F)=C7)CC6)CC5)CC4)C=C3)C2(C)C)C=C1Cl	C51H69ClF3N7O6S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-X338IL	WO2024165050A1_14	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCN(CCCCC(=O)NCC4=CC=C(S(=O)(=O)N5CCN(C6=NC=CC(C(F)(F)F)=C6)CC5)C=C4)CC3)C=C2)C(C)(C)[C@@H]1OC1=CC=C(C#N)C(Cl)=C1	C48H56ClF3N8O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-8G09RL	WO2024165050A1_15	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCN(CCC(=O)NCC4=CC=C(S(=O)(=O)N5CCN(C6=NC=CC(C(F)(F)F)=C6)CC5)C=C4)CC3)C=C2)C(C)(C)[C@@H]1OC1=CC=C(C#N)C(Cl)=C1	C46H52ClF3N8O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-C3VKKU	WO2024165050A1_16	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCN(CCCCCCC(=O)NCC4CC(S(=O)(=O)N5CCN(C6=NC=CC(C(F)(F)F)=C6)CC5)C4)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C48H62ClF3N8O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-PUB39B	WO2024165050A1_17	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCN(CCCCCCC(=O)NCC4=CC=C(S(=O)(=O)N5CC(C6=NC=CC(C(F)(F)F)=C6)C5)C=C4)CC3)C=C2)C(C)(C)[C@@H]1OC1=CC=C(C#N)C(Cl)=C1	C49H57ClF3N7O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-2ECBWP	WO2024165050A1_18	.	CC(=O)C1=CC=C(O[C@H]2C(C)(C)[C@@H](NC(=O)C3=CC=C(N4CCN(CCCCCCC(=O)NCC5=CC=C(S(=O)(=O)N6CCN(C7=NC=CC(C(F)(F)F)=C7)C6)C=C5)CC4)C=C3)C2(C)C)C=C1Cl	C50H61ClF3N7O6S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-J7L0VF	WO2024165050A1_19	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCN(CCCCCCC(=O)NCC4=CC=C(S(=O)(=O)N5CCN(C6=NC=C(C(F)(F)F)C=C6)CC5)C=C4)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C50H60ClF3N8O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-3UETE1	WO2024165050A1_20	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCN(CCCCCCC(=O)NCC4=CC=C(S(=O)(=O)N5CCN(C6=NC(C(F)(F)F)=CC=C6)CC5)C=C4)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C50H60ClF3N8O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-FLNNNN	WO2024165050A1_21	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCN(CCCCCCC(=O)NCC4=CC=C(S(=O)(=O)N5CCN(C6=NC=CC=C6C(F)(F)F)CC5)C=C4)CC3)C=C2)C(C)(C)[C@@H]1OC1=CC=C(C#N)C(Cl)=C1	C50H60ClF3N8O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-XJYUBB	WO2024165050A1_22	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCN(CCCCCCC(=O)NCC4=CC=C(S(=O)(=O)N5CCN(C6=CN=CC(C(F)(F)F)=C6)CC5)C=C4)CC3)C=C2)C(C)(C)[C@@H]1OC1=CC=C(C#N)C(Cl)=C1	C50H60ClF3N8O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-YQKZ5G	WO2024165050A1_23	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCN(CCCCCCC(=O)NCC4=CC=C(S(=O)(=O)N5CCN(C6=CC=NC(C(F)(F)F)=C6)CC5)C=C4)CC3)C=C2)C(C)(C)[C@@H]1OC1=CC=C(C#N)C(Cl)=C1	C50H60ClF3N8O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-FE1H10	WO2024165050A1_28	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCN(CCCCCCC(=O)N4CCN(C5=NC=CC(C(F)(F)F)=C5)CC4)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C43H53ClF3N7O3	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-IBFG50	WO2024165050A1_29	.	CC1(C)[C@H](NC(=O)C2=CC=C(C(=O)NCCOCCNCC3=CC=C(S(=O)(=O)N4CCN(C5=NC=CC(C(F)(F)F)=C5)CC4)C=C3)C=C2)C(C)(C)[C@@H]1OC1=CC=C(C#N)C(Cl)=C1	C44H49ClF3N7O6S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-G5JXTF	WO2024165050A1_30	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCN(CCCCCCC(=O)NCC4=CC=C(S(=O)(=O)C5CCN(C6=CN=CC(C(F)(F)F)=C6)CC5)C=C4)CC3)C=C2)C(C)(C)[C@@H]1OC1=CC=C(C#N)C(Cl)=C1	C51H61ClF3N7O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-D5D0RX	WO2024165050A1_31	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCN(CCCCCCCN4CCC(S(=O)(=O)N5CCN(C6=CN=CC(C(F)(F)F)=C6)CC5)CC4)CC3)C=C2)C(C)(C)[C@@H]1OC1=CC=C(C#N)C(Cl)=C1	C48H64ClF3N8O4S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-CMMBHW	WO2024165050A1_32	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCN(CCCCCCCNCCCS(=O)(=O)N4CCN(C5=CN=CC(C(F)(F)F)=C5)CC4)CC3)C=C2)C(C)(C)[C@@H]1OC1=CC=C(C#N)C(Cl)=C1	C46H62ClF3N8O4S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-WQON8E	WO2024165050A1_33	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCN(CCOCCNCC4=CC=C(S(=O)(=O)N5CCN(C6=CN=CC(C(F)(F)F)=C6)CC5)C=C4)CC3)C=C2)C(C)(C)[C@@H]1OC1=CC=C(C#N)C(Cl)=C1	C47H56ClF3N8O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-N382CP	WO2024165050A1_34	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCN(CCOCCCNCCCS(=O)(=O)N4CCN(C5=CN=CC(C(F)(F)F)=C5)CC4)CC3)C=C2)C(C)(C)[C@@H]1OC1=CC=C(C#N)C(Cl)=C1	C44H58ClF3N8O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-JLRWQN	WO2024165050A1_35	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCN(CCOCCCS(=O)(=O)N4CCN(C5=CN=CC(C(F)(F)F)=C5)CC4)CC3)C=C2)C(C)(C)[C@@H]1OC1=CC=C(C#N)C(Cl)=C1	C41H51ClF3N7O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-43SQL9	WO2024165050A1_36	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCN(CCCC(=O)NCCCS(=O)(=O)N4CCN(C5=CC(C(F)(F)F)=CC=N5)CC4)CC3)C=C2)C(C)(C)[C@@H]1OC1=CC=C(C#N)C(Cl)=C1	C43H54ClF3N8O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-BBSGSH	WO2024165050A1_37	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCN(CCC(=O)NCCCS(=O)(=O)N4CCN(C5=CC(C(F)(F)F)=CC=N5)CC4)CC3)C=C2)C(C)(C)[C@@H]1OC1=CC=C(C#N)C(Cl)=C1	C42H52ClF3N8O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-UQVL71	WO2024165050A1_38	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCN(CC(=O)NCCCS(=O)(=O)N4CCN(C5=CN=CC(C(F)(F)F)=C5)CC4)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C41H50ClF3N8O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-2SA4KG	WO2024165050A1_39	.	N#CC1=CC=C(O[C@H]2CC[C@H](C(=O)NC3=CC=C(N4CCN(CCOCCCS(=O)(=O)N5CCN(C6=CN=CC(C(F)(F)F)=C6)CC5)CC4)N=N3)CC2)C=C1Cl	C37H45ClF3N9O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-HN5I4C	WO2024165050A1_40	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(CN4CCC(S(=O)(=O)N5CCN(C6=CN=CC(C(F)(F)F)=C6)CC5)CC4)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C43H53ClF3N7O4S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-6W8KHC	WO2024165050A1_41	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCN(CC4CCN(S(=O)(=O)N5CCN(C6=CC(C(F)(F)F)=CN=C6)CC5)CC4)CC3)C=C2)C(C)(C)[C@@H]1OC1=CC=C(C#N)C(Cl)=C1	C42H52ClF3N8O4S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-DDTC92	WO2024165050A1_42	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCN(CCN4CC(S(=O)(=O)N5CCN(C6=CN=CC(C(F)(F)F)=C6)CC5)C4)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C41H50ClF3N8O4S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-MCHKPD	WO2024165050A1_43	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(CN4CCC(S(=O)(=O)N5CCC(C6=CC(C(F)(F)F)=CN=C6)CC5)CC4)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C44H54ClF3N6O4S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-YC5F4J	WO2024165050A1_44	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCN(CCN4CCC(S(=O)(=O)N5CCN(C6=CC(C(F)(F)F)=CN=C6)CC5)CC4)CC3)C=C2)C(C)(C)[C@@H]1OC1=CC=C(C#N)C(Cl)=C1	C43H54ClF3N8O4S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-3WHUQZ	WO2024165050A1_45	.	N#CC1=CC=C(O[C@H]2CC[C@@H](NC(=O)C3=CC=C(N4CCN(CCOCCCS(=O)(=O)N5CCN(C6=CN=CC(C(F)(F)F)=C6)CC5)CC4)N=N3)CC2)C=C1Cl	C37H45ClF3N9O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-F38UGC	WO2024165050A1_46	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(CN4CCC(CS(=O)(=O)N5CCN(C6=CN=CC(C(F)(F)F)=C6)CC5)CC4)CC3)C=C2)C(C)(C)[C@@H]1OC1=CC=C(C#N)C(Cl)=C1	C44H55ClF3N7O4S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-5CGFWU	WO2024165050A1_47	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(CN4CC(CS(=O)(=O)N5CCN(C6=CN=CC(C(F)(F)F)=C6)CC5)C4)CC3)C=C2)C(C)(C)[C@@H]1OC1=CC=C(C#N)C(Cl)=C1	C42H51ClF3N7O4S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-7O5D0O	WO2024165050A1_48	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(N4CCN(CCS(=O)(=O)N5CCN(C6=CN=CC(C(F)(F)F)=C6)CC5)CC4)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C43H54ClF3N8O4S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-6ITJYU	WO2024165050A1_49	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=CC=C(N4CCN(CCCS(=O)(=O)N5CCN(C6=CN=CC(C(F)(F)F)=C6)CC5)CC4)N=N3)CC2)C=C1Cl	C35H41ClF3N9O4S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-PFCQOU	WO2024165050A1_53	.	N#CC1=CC=C(O[C@H]2CC[C@H](C(=O)NC3=CC=C(N4CCN(CCCOCCCS(=O)(=O)N5CCN(C6=CN=CC(C(F)(F)F)=C6)CC5)CC4)N=N3)CC2)C=C1Cl	C38H47ClF3N9O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-CCYPYI	WO2024165050A1_54	.	CC1(C)[C@H](NC(=O)C2=CN(CCOCCCS(=O)(=O)N3CCN(C4=CC(C(F)(F)F)=CN=C4)CC3)N=C2)C(C)(C)[C@@H]1OC1=CC(Cl)=C(C#N)C=C1	C34H41ClF3N7O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-RZLI6W	WO2024165050A1_55	.	CN1CCN(S(=O)(=O)CCCNC(=O)CCCCCCN2CCN(C3=CC=C(C(=O)N[C@H]4C(C)(C)[C@H](OC5=CC=C(C#N)C(Cl)=C5)C4(C)C)C=C3)CC2)CC1	C41H60ClN7O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-DQTZ66	WO2024165050A1_56	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCN(CCCCCCC(=O)NCCCS(=O)(=O)N4CCN(C5=NC=CC=C5)CC4)CC3)C=C2)C(C)(C)[C@@H]1OC1=CC=C(C#N)C(Cl)=C1	C45H61ClN8O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-8XFQYH	WO2024165050A1_57	.	N#CC1=CC=C(O[C@H]2CC[C@@H](C(=O)NC3=CC=C(C4CCN(CCCOCCS(=O)(=O)N5CCN(C6=CN=CC(C(F)(F)F)=C6)CC5)CC4)N=N3)CC2)C=C1Cl	C38H46ClF3N8O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-EE4RUB	WO2024165050A1_58	.	N#CC1=CC=C(O[C@H]2CC[C@H](C(=O)NC3=CC=C(N4CCN(CCOCCN5CCC(S(=O)(=O)N6CCN(C7=CC(C(F)(F)F)=CC=N7)CC6)C5)CC4)N=N3)CC2)C=C1Cl	C40H50ClF3N10O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-CP6JJ0	WO2024165050A1_59	.	N#CC1=CC=C(O[C@H]2CC[C@H](C(=O)NC3=NN=C(C4CCN(CCN5CCC(CS(=O)(=O)N6CCN(C7=CC(C(F)(F)F)=CN=C7)CC6)C5)CC4)C=C3)CC2)C=C1Cl	C40H49ClF3N9O4S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-74ICJ6	WO2024165050A1_60	.	N#CC1=CC=C(O[C@H]2CC[C@@H](C(=O)NC3=CC=C(C4CCC(OCCN5CCC(S(=O)(=O)N6CCN(C7=CN=CC(C(F)(F)F)=C7)CC6)C5)CC4)N=N3)CC2)C=C1Cl	C40H48ClF3N8O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-GAUI8M	WO2024165050A1_61	.	N#CC1=CC=C(OC2CCC(C(=O)NC3=CC=C(C4CCC(CCN5CCC(CS(=O)(=O)C6CCN(C7=NC=CC(C(F)(F)F)=C7)CC6)C5)CC4)N=N3)CC2)C=C1Cl	C42H51ClF3N7O4S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-15ZEGH	WO2024165050A1_62	.	N#CC1=CC=C(OC2CCC(C(=O)NC3=CC=C(C4CCN(CCOCCS(=O)(=O)N5CCN(C6=NC=CC(C(F)(F)F)=C6)CC5)CC4)N=N3)CC2)C=C1Cl	C37H44ClF3N8O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-X7NG9E	WO2024165050A1_63	.	CC1(C)[C@H](NC(=O)C2=CC=C(C3CCN(CCOCCCS(=O)(=O)N4CCN(C5=CC(C(F)(F)F)=CN=C5)CC4)CC3)N=N2)C(C)(C)[C@@H]1OC1=CC=C(C#N)C(Cl)=C1	C40H50ClF3N8O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-LP6I55	WO2024165050A1_64	.	N#CC1=CC=C(O[C@H]2CC[C@@H](C(=O)NC3=NN=C(N4CCN(CCCOCCS(=O)(=O)N5CCN(C6=CN=CC(C(F)(F)F)=C6)CC5)CC4)C=C3)CC2)C=C1Cl	C37H45ClF3N9O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-IIWCIL	WO2024165050A1_65	.	N#CC1=CC=C(O[C@H]2CC[C@H](C(=O)NC3=CC=C(C4CCN(CCOCCS(=O)(=O)N5CCN(C6=CN=CC(C(F)(F)F)=C6)CC5)CC4)N=N3)CC2)C=C1Cl	C37H44ClF3N8O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-TARBHZ	WO2024165050A1_66	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCN(CCOCCCS(=O)(=O)N4CCN(C5=CN=CC(C(F)(F)F)=C5)CC4)CC3)N=N2)C(C)(C)[C@@H]1OC1=CC=C(C#N)C(Cl)=C1	C39H49ClF3N9O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-DX0XP2	WO2024165050A1_67	.	CC1(C)[C@H](NC(=O)C2=NN=C(N3CCN(CCCOCCS(=O)(=O)N4CCN(C5=NN=CC(C(F)(F)F)=C5)CC4)CC3)C=C2)C(C)(C)[C@@H]1OC1=CC=C(C#N)C(Cl)=C1	C38H48ClF3N10O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-Q51CKH	WO2024165050A1_68	.	CC1(C)[C@H](NC(=O)C2=NN=C(CN3CCN(CCOCCS(=O)(=O)N4CCN(C5=NN=CC(C(F)(F)F)=C5)CC4)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C38H48ClF3N10O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-9KOY6I	WO2024165050A1_69	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCN(CCOCCCS(=O)(=O)N4CCN(C5=NN=CC(C(F)(F)F)=C5)CC4)CC3)C=C2)C(C)(C)[C@@H]1OC1=CC=C(C#N)C(Cl)=C1	C40H50ClF3N8O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-7SRF41	WO2024165050A1_70	.	N#CC1=CC=C(O[C@H]2CC[C@@H](NC(=O)C3=NN=C(N4CCN(CCOCCS(=O)(=O)N5CCN(C6=CN=CC(C(F)(F)F)=C6)CC5)CC4)C=C3)CC2)C=C1Cl	C36H43ClF3N9O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-9DPMHD	WO2024165050A1_71	.	CC1(C)C(NC(=O)C2=CC=C(N3CCN(CCOCCS(=O)(=O)N4CCN(C5=CN=CC(C(F)(F)F)=C5)CC4)CC3)N=N2)C(C)(C)C1OC1=CC=C(C#N)C(Cl)=C1	C38H47ClF3N9O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-VSU1I4	WO2024165050A1_72	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=CC=C(C4CCN(CCOCCS(=O)(=O)N5CCN(C6=NN=CC(C(F)(F)F)=C6)CC5)CC4)N=N3)CC2)C=C1Cl	C36H43ClF3N9O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-K6UZK1	WO2024165050A1_73	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=CC=C(C4CCN(CCOCCS(=O)(=O)N5CCN(C6=NC=CC(C(F)(F)F)=C6)CC5)CC4)N=N3)CC2)C=C1Cl	C37H44ClF3N8O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-J5KTYF	WO2024165050A1_74	.	N#CC1=CC=C(O[C@H]2CC[C@H](C(=O)NC3=CC=C(N4CCN(CCOCCS(=O)(=O)N5CCN(C6=NC=CC(C(F)(F)F)=C6)CC5)CC4)N=N3)CC2)C=C1Cl	C36H43ClF3N9O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-OFLD9F	WO2024165050A1_75	.	N#CC1=CC=C(O[C@H]2CC[C@H](C(=O)NC3=CC=C(C4CCN(CCOCCS(=O)(=O)N5CCN(C6=NC=CC(C(F)(F)F)=N6)CC5)CC4)N=N3)CC2)C=C1Cl	C36H43ClF3N9O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-Z8J3ZW	WO2024165050A1_76	.	N#CC1=CC=C(O[C@H]2CC[C@@H](C(=O)NC3=CC=C(C4CCN(CCOCCS(=O)(=O)N5CCN(C6=NC=CC=C6)CC5)CC4)N=N3)CC2)C=C1Cl	C36H45ClN8O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-1VDMKT	WO2024165050A1_77	.	N#CC1=CC=C(O[C@H]2CC[C@H](C(=O)NC3=CC=C(C4CCN(CCOCCS(=O)(=O)N5CCN(C6=NC=CC(Cl)=C6)CC5)CC4)N=N3)CC2)C=C1Cl	C36H44Cl2N8O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-81JLEL	WO2024165050A1_78	.	CS(=O)(=O)C1=CC(N2CCN(S(=O)(=O)CCOCCN3CCC(C4=CC=C(NC(=O)[C@H]5CC[C@H](OC6=CC=C(C#N)C(Cl)=C6)CC5)N=N4)CC3)CC2)=NC=C1	C37H47ClN8O7S2	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-3IG5YV	WO2024165050A1_79	.	CCC1=CC(N2CCN(S(=O)(=O)CCOCCN3CCC(C4=CC=C(NC(=O)[C@H]5CC[C@H](OC6=CC(Cl)=C(C#N)C=C6)CC5)N=N4)CC3)CC2)=NC=C1	C38H49ClN8O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-U1IT2Q	WO2024165050A1_80	.	CC(C)C1=CC(N2CCN(S(=O)(=O)CCOCCN3CCC(C4=CC=C(NC(=O)[C@H]5CC[C@H](OC6=CC(Cl)=C(C#N)C=C6)CC5)N=N4)CC3)CC2)=NC=C1	C39H51ClN8O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-VQS0YY	WO2024165050A1_81	.	N#CC1=C(Cl)C=C(O[C@H]2CC[C@H](C(=O)NC3=CC=C(C4CCN(CCOCCS(=O)(=O)N5CCN(C6=NC=CC(F)=C6)CC5)CC4)N=N3)CC2)C=C1	C36H44ClFN8O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-2CR71L	WO2024165050A1_82	.	N#CC1=CC(N2CCN(S(=O)(=O)CCOCCN3CCC(C4=CC=C(NC(=O)[C@H]5CC[C@H](OC6=CC(Cl)=C(C#N)C=C6)CC5)N=N4)CC3)CC2)=NC=C1	C37H44ClN9O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-RN7UE3	WO2024165050A1_83	.	N#CC1=C(Cl)C=C(O[C@H]2CC[C@H](C(=O)NC3=CC=C(C4CCN(CCOCCS(=O)(=O)N5CCN(C6=CC=CC(=O)N6)CC5)CC4)N=N3)CC2)C=C1	C36H45ClN8O6S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-CD841H	WO2024165050A1_84	.	CC1=CC(N2CCN(S(=O)(=O)CCOCCN3CCN(C4=CC=C(NC(=O)[C@H]5CC[C@H](OC6=CC(Cl)=C(C#N)C=C6)CC5)N=N4)CC3)CC2)=NC=C1	C36H46ClN9O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-8FX5FV	WO2024165050A1_85	.	COC1=CC(N2CCN(S(=O)(=O)CCOCCN3CCC(C4=CC=C(NC(=O)[C@H]5CC[C@H](OC6=CC(Cl)=C(C#N)C=C6)CC5)N=N4)CC3)CC2)=NC=C1	C37H47ClN8O6S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-Q3SMAE	WO2024165050A1_86	.	N#CC1=C(Cl)C=C(OC2CCC(C(=O)NC3=CC=C(C4CCN(CCOCCS(=O)(=O)N5CCN(C6=NC=CC([N+](=O)[O-])=C6)CC5)CC4)N=N3)CC2)C=C1	C36H44ClN9O7S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-Z0BMUW	WO2024165050A1_87	.	CC1CC(C2=CC=C(NC(=O)[C@H]3CC[C@H](OC4=CC(Cl)=C(C#N)C=C4)CC3)N=N2)CCN1CCOCCS(=O)(=O)N1CCN(C2=NC=CC(C(F)(F)F)=C2)CC1	C38H46ClF3N8O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-WVOY8Z	WO2024165050A1_88	.	N#CC1=CC=C(OC2CCC(C(=O)NC3=CC=C(N4CCN(CCOCCCS(=O)(=O)C5CCN(C6=CN=CC(C(F)(F)F)=C6)CC5)CC4)N=N3)CC2)C=C1Cl	C38H46ClF3N8O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-JTDJFM	WO2024165050A1_89	.	N#CC1=CC=C(OC2CCC(C(=O)NC3=CC=C(N4CCN(CCNCCCS(=O)(=O)N5CCN(C6=CN=CC(C(F)(F)F)=C6)CC5)CC4)N=N3)CC2)C=C1Cl	C37H46ClF3N10O4S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-H75DYE	WO2024165050A1_90	.	N#CC1=CC=C(O[C@H]2CC[C@H](C(=O)NC3=CC=C(NCCOCCN4CCC(S(=O)(=O)N5CCN(C6=NC=CC(C(F)(F)F)=C6)CC5)C4)N=N3)CC2)C=C1Cl	C36H43ClF3N9O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-902YL8	WO2024165050A1_91	.	COC1=NC(N2CCN(S(=O)(=O)CCOCCN3CCC(C4=CC=C(NC(=O)[C@H]5CC[C@@H](OC6=CC(Cl)=C(C#N)C=C6)CC5)N=N4)CC3)CC2)=CC=C1	C37H47ClN8O6S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-KNZSZ0	WO2024165050A1_92	.	N#CC1=C(Cl)C=C(O[C@H]2CC[C@H](C(=O)NC3=CC=C(C4CCN(CCOCCS(=O)(=O)N5CCN(C6=NC=CC(C(F)(F)F)=C6)CC5)CC4(F)F)C=C3)CC2)C=C1	C39H44ClF5N6O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-5ZPEHG	WO2024165050A1_93	.	N#CC1=C(Cl)C=C(O[C@H]2CC[C@@H](C(=O)NC3=CC=C(C4CCN(CCOCCS(=O)(=O)N5CCN(C6=NC=CC(C(F)(F)F)=C6)CC5)CC4(F)F)C=N3)CC2)C=C1	C38H43ClF5N7O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-KEX5B1	WO2024165050A1_94	.	N#CC1=CC=C(O[C@H]2CC[C@H](C(=O)NC3=CC=C(C4CCN(CCOCCS(=O)(=O)N5CCN(C6=NC=CC(CF)=C6)CC5)CC4(F)F)C=C3)CC2)C=C1Cl	C39H46ClF3N6O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-YD5FO0	WO2024165050A1_95	.	N#CC1=CC=C(O[C@H]2CC[C@H](C(=O)NC3=CC=C(C4CCN(CCOCCS(=O)(=O)N5CCN(C6=NC=CC(C(F)F)=C6)CC5)CC4(F)F)C=C3)CC2)C=C1Cl	C39H45ClF4N6O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-WGSAHB	WO2024165050A1_96	.	N#CC1=CC=C(OC2CCC(C(=O)NC3=CC=C(C4CN(CCOCCS(=O)(=O)N5CCN(C6=NC=CC(C(F)(F)F)=C6)CC5)C4)N=N3)CC2)C=C1Cl	C35H40ClF3N8O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-BVHFL3	WO2024165050A1_98	.	N#CC1=CC=C(OC2CCC(NC(=O)C3=NN(C4CCC(CCOCCS(=O)(=O)N5CCN(C6=CC(C(F)(F)F)=CC=N6)CC5)CC4)C=C3)CC2)C=C1Cl	C37H45ClF3N7O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-JPR16S	WO2024165050A1_99	.	CC1(C)C(NC(=O)C2=CC=C(N3CCC(CCOCCS(=O)(=O)N4CCN(C5=NC=CC(C(F)(F)F)=C5)CC4)CC3)C=C2)C(C)(C)C1OC1=CC=C(C#N)C(Cl)=C1	C41H50ClF3N6O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-SYS3QK	WO2024165050A1_100	.	N#CC1=CC=C(OC2CCC(NC(=O)C3=CC=C(C4CCC(CN5CCC(S(=O)(=O)N6CCN(C7=CC(C(F)(F)F)=CC=N7)CC6)CC5)CC4)N=N3)CC2)C=C1Cl	C40H48ClF3N8O4S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-9EBPOH	WO2024165050A1_101	.	CN(CCC1CCN(C2=CC=C(C(=O)NC3CCC(OC4=CC=C(C#N)C(Cl)=C4)CC3)N=N2)CC1)CCS(=O)(=O)N1CCN(C2=NC=CC(C(F)(F)F)=C2)CC1	C38H47ClF3N9O4S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-WQEG5F	WO2024165050A1_102	.	COC1=CC(OC2C(C)(C)C(NC(=O)C3=CC=C(N4CCC(CN5CCC(S(=O)(=O)N6CCN(C7=CC(C(F)(F)F)=CC=N7)CC6)CC5)CC4)C=C3)C2(C)C)=CC=C1C#N	C44H56F3N7O5S	AR;CDC20	P10275/Q12834		WO-2024165050-A1
TPD-QNPMWB	WO2024169871A1_I-1	.	COC1=C(C(=O)NCC2=CC=C(C3=NN(C4CCN(C5CN(CC6CCN(C7=CC=C(N8CCC(=O)NC8=O)C=C7)CC6)C5)CC4)C4=C3C(N)=NC=N4)C=C2)C=C(F)C=C1	C44H50FN11O4	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-QJX8CP	WO2024169871A1_I-10	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=NN(C3=CC=C(N4CCN(CC5CCN(C6=CC(C)=C(C7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)C3=C2C(N)=NC=N3)C=C1	C48H51FN10O4	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-OD31S6	WO2024169871A1_I-11	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=NN(C3=CC=C(C4CCN(CC5CCN(C6=CC(C)=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)C(N)=C2C(N)=O)C=C1	C47H52FN9O5	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-3FYI3N	WO2024169871A1_I-12	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=NN(C3=CN=C(C4CCN(CC5CCN(C6=CC(C)=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)C(N)=C2C(N)=O)C=C1	C46H51FN10O5	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-S5G4LK	WO2024169871A1_I-13	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=NN(C3=CC(F)=C(N4CCN(CC5CCN(C6=CC(C)=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)C(N)=C2C(N)=O)C=C1	C46H50F2N10O5	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-BP9YY6	WO2024169871A1_I-14	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=NN(C3=CC(F)=C(N4CCN(CC5CCN(C6=CC(C)=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)C3=C2C(N)=NC=N3)C=C1	C47H49F2N11O4	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-NCJSCK	WO2024169871A1_I-15	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=NN(C3=CN=C(N4CCN(CC5CCN(C6=CC(C)=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)C3=C2C(N)=NC=C3)C=C1	C47H50FN11O4	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-NDFSJ5	WO2024169871A1_I-16	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(N2N=C(C3=CN=C(N4CCN(CC5CCN(C6=CC(C)=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)C3=C2C(N)=NC=C3)C=C1	C47H50FN11O4	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-K75US1	WO2024169871A1_I-17	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=C3C(N)=NC=CN3C(C3=CC(F)=C(N4CCN(CC5CCN(C6=CC(C)=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)=N2)C=C1	C48H50F2N10O4	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-5MOGFI	WO2024169871A1_I-18	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=C3C(N)=NC=CN3C(C3=CC=C(N4CCN(CC5CCN(C6=CC=C(C7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)=N2)C=C1	C48H50FN9O4	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-F5W02X	WO2024169871A1_I-19	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=C3C(N)=NC=CN3C(C3=CC=C(N4CCN(CC5CCN(C6=CC(C)=C(C7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)=N2)C=C1	C49H52FN9O4	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-RMTKPT	WO2024169871A1_I-2	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=NN(C3=CN=C(N4CCN(CC5CCN(C6=CC(C)=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)C3=C2C(N)=NC=N3)C=C1	C46H49FN12O4	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-FWYPVZ	WO2024169871A1_I-20	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=C3C(N)=NC=CN3C(C3=CC(F)=C(N4CCC(CN5CCN(C6=CC(C)=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)=N2)C=C1	C48H50F2N10O4	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-TCLLLB	WO2024169871A1_I-21	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=C3C(N)=NC=CN3C(C3=CC=C(N4CCC(CN5CCN(C6=CC=C(C7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)=N2)C=C1	C48H50FN9O4	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-MTZMNL	WO2024169871A1_I-22	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=C3C(N)=NC=CN3C(C3=CC=C(N4CCC(CN5CCN(C6=CC(C)=C(C7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)=N2)C=C1	C49H52FN9O4	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-6DBRFJ	WO2024169871A1_I-23	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=C3C(N)=NC=CN3C(C3=CC(F)=C(N4CCN(CC5CCN(C6=CC(C)=C(C7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)=N2)C=C1	C49H51F2N9O4	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-N66OMA	WO2024169871A1_I-24	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=NN(C3=CN=C(C4CCN(CC5CCN(C6=CC=C(C7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)C3=C2C(N)=NC=N3)C=C1	C47H49FN10O4	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-QMVXUS	WO2024169871A1_I-25	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=NN(C3=CC(F)=C(N4CCN(CC5CCN(C6=CC(C)=C(C7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)C3=C2C(N)=NC=C3)C=C1	C49H51F2N9O4	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-1BZUFT	WO2024169871A1_I-26	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(N2C(=O)N(C3=CC(F)=C(N4CCN(CC5CCN(C6=CC(C)=C(C7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)C3=C2C(N)=NC=C3)C=C1	C49H51F2N9O5	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-TAUB9B	WO2024169871A1_I-27	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(N2N=C(C3=CC(F)=C(N4CCN(CC5CCN(C6=CC(C)=C(C7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)C3=C2C(N)=NC=C3)C=C1	C49H51F2N9O4	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-EHAXOP	WO2024169871A1_I-28	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(N2C(=O)N(C3=CC(F)=C(N4CCN(CC5CCN(C6=CC(C)=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)C3=C2C(N)=NC=N3)C=C1	C47H49F2N11O5	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-DVHLE6	WO2024169871A1_I-29	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=NN(C3=CC(F)=C(N4CCN(CC5CCN(C6=CC(C)=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)C3=C2C(N)=NNC3=O)C=C1	C47H49F2N11O5	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-RKR5K7	WO2024169871A1_I-3	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=NN(C3=CN=C(N4CCN(CC5CCN(C6=CC=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)C3=C2C(N)=NC=N3)C=C1	C45H47FN12O4	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-MQ0HXV	WO2024169871A1_I-30	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=C3C(N)=NC=CN3C(C3=CN=C(N4CCN(CC5CCN(C6=CC(C)=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)=N2)C=C1	C47H50FN11O4	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-88ES33	WO2024169871A1_I-31	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=C3C(N)=NC=CN3C(C3=CC(F)=C(C4=CCN(CC5CCN(C6=CC(C)=C(C7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)=N2)C=C1	C50H50F2N8O4	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-50A8O8	WO2024169871A1_I-32	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=NN(C3=CC(F)=C(C4=CCN(CC5CCN(C6=CC(C)=C(C7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)C3=C2C(N)=NC=N3)C=C1	C49H49F2N9O4	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-ACQVQZ	WO2024169871A1_I-33	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=C3C(N)=NC=CN3C(C3=CC(F)=C(N4CCN(CC5CCN(C6=CC=C(C7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)=N2)C=C1	C48H49F2N9O4	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-R8UUYD	WO2024169871A1_I-34	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=NN(C3=CC(F)=C(N4CCN(CC5CCN(C6=CC=C(C7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)C3=C2C(N)=NC=N3)C=C1	C47H48F2N10O4	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-G3BJE8	WO2024169871A1_I-35	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=NN(C3=CC=C(N4CC5CC(C4)N5CC4CCN(C5=CC(C)=C(N6CCC(=O)NC6=O)C=C5)CC4)C=C3)C3=C2C(N)=NC=N3)C=C1	C48H50FN11O4	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-R1U0II	WO2024169871A1_I-36	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=NN(C3=CC=C(N4CC5(CN(CC6CCN(C7=CC(C)=C(N8CCC(=O)NC8=O)C=C7)CC6)C5)C4)C=C3)C3=C2C(N)=NC=N3)C=C1	C48H50FN11O4	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-RE6A7Z	WO2024169871A1_I-37	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=NN(C3=CC=C(N4CCC5(CCN(CC6CCN(C7=CC(C)=C(N8CCC(=O)NC8=O)C=C7)CC6)CC5)CC4)C=C3)C3=C2C(N)=NC=N3)C=C1	C52H58FN11O4	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-ILCH29	WO2024169871A1_I-38	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=NN(C3=CC(F)=C(C4CCN(CC5CCN(C6=CC(C)=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)C(N)=C2C(N)=O)C=C1	C47H51F2N9O5	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-1D4YYZ	WO2024169871A1_I-39	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=NN(C3=CN=C(C4CCN(CC5CCN(C6=CC(C)=C(C7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)C3=C2C(N)=NC=N3)C=C1	C48H51FN10O4	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-39XTD6	WO2024169871A1_I-4	.	COC1=CC=C(F)C=C1C(=O)NCC1=C(C)C=C(C2=NN(C3=CN=C(N4CCN(CC5CCN(C6=CC(C)=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)C3=C2C(N)=NC=N3)C=C1	C47H51FN12O4	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-WD2GFS	WO2024169871A1_I-40	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=C3C(N)=NC=CN3C(C3=CC=C(N4CCN(CC5CCN(C6=CC(C)=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)=N2)C=C1	C48H51FN10O4	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-XNXGQC	WO2024169871A1_I-41	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=NN(C3=CN=C(N4CCN(CC5CCN(C6=CC(C)=C(N7CCC(=O)NC7=O)C=C6)CC5)C[C@H]4C)C=C3)C3=C2C(N)=NC=N3)C=C1	C47H51FN12O4	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-7YS79A	WO2024169871A1_I-42	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=NN(C3=CC=C(N4CCC(CN5CCN(C6=CC(C)=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)C3=C2C(N)=NC=N3)C=C1	C47H50FN11O4	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-CVAUWR	WO2024169871A1_I-43	.	COC1=CC=C(F)C=C1C(=O)NCC1=C(F)C(F)=C(C2=NN(C3=CN=C(N4CCN(CC5CCN(C6=CC(C)=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)C3=C2C(N)=NC=N3)C=C1	C46H47F3N12O4	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-QXVHB4	WO2024169871A1_I-44	.	COC1=CC=C(F)C=C1C(=O)NCC1=C(F)C=C(C2=NN(C3=CC=C(C4CCN(CC5CCN(C6=CC(C)=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)C3=C2C(N)=NC=N3)C=C1	C48H50F2N10O4	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-BMZ8OX	WO2024169871A1_I-45	.	COC1=CC=C(F)C=C1C(=O)NCC1=C(F)C=C(C2=C3C(N)=NC=CN3C(C3=CC=C(N4CCN(CC5CCN(C6=CC(C)=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)=N2)C=C1	C48H50F2N10O4	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-GYAMM5	WO2024169871A1_I-46	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=NN(C3=CC=C(N4CCN(CC5CCN(C6=CC(C)=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)C3=C2C(N)=NC=C3)C=C1	C48H51FN10O4	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-TZFYH1	WO2024169871A1_I-47	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC(F)=C(C2=C3C(N)=NC=CN3C(C3=CC=C(N4CCN(CC5CCN(C6=CC(C)=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)=N2)C=C1	C48H50F2N10O4	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-6WHRDM	WO2024169871A1_I-48	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(N2C(=O)N(C3=CC=C(N4CCN(CC5CCN(C6=CC(C)=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)C3=C2C(N)=NC=C3)C=C1	C48H51FN10O5	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-ZHYZH5	WO2024169871A1_I-49	.	CCC1=C(N2CCN(CC3CCN(C4=CC(C)=C(N5CCC(=O)NC5=O)C=C4)CC3)CC2)C=CC(C2=NC(C3=CC=C(CNC(=O)C4=CC(F)=CC=C4OC)C=C3)=C3C(N)=NC=CN23)=C1	C50H55FN10O4	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-WRUT4H	WO2024169871A1_I-5	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=NN(C3=CC=C(C4CCN(CC5CCN(C6=CC(C)=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)C3=C2C(N)=NC=N3)C=C1	C48H51FN10O4	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-MTBVJ6	WO2024169871A1_I-50	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=C3C(N)=NC=CN3C(C3=CC=C(C4=CCN(CC5CCN(C6=CC(C)=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)=N2)C=C1	C49H50FN9O4	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-D76FB1	WO2024169871A1_I-51	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=C3C(N)=NC=CN3C(C3=CC(OC)=C(N4CCN(CC5CCN(C6=CC(C)=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)=N2)C=C1	C49H53FN10O5	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-Z59TJ8	WO2024169871A1_I-52	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(N2C(=O)N(C3=CN=C(N4CCN(CC5CCN(C6=CC(C)=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)C3=C2C(N)=NC=C3)C=C1	C47H50FN11O5	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-PQLJ6T	WO2024169871A1_I-53	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=C3C(N)=NC=CN3C(C3=CC=C(N4CC5CC(C4)N5CC4CCN(C5=CC(C)=C(N6CCC(=O)NC6=O)C=C5)CC4)C=C3)=N2)C=C1	C49H51FN10O4	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-QIX40W	SCHEMBL31113369	1-[4-[4-[[4-[5-[8-Amino-1-(4-phenoxyphenyl)imidazo[1,5-a]pyrazin-3-yl]pyridin-2-yl]piperazin-1-yl]methyl]piperidin-1-yl]-2-methylphenyl]-1,3-diazinane-2,4-dione	CC1=C(N2CCC(=O)NC2=O)C=CC(N2CCC(CN3CCN(C4=NC=C(C5=NC(C6=CC=C(OC7=CC=CC=C7)C=C6)=C6C(N)=NC=CN56)C=C4)CC3)CC2)=C1	C44H46N10O3	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-H34HBI	WO2024169871A1_I-55	.	CC1=C(N2CCC(=O)NC2=O)C=CC(N2CCC(CN3CCN(C4=CC=C(N5N=C(C6=CC=C(OC7=CC=CC=C7)C=C6)C6=C5N=CN=C6N)C=C4)CC3)CC2)=C1	C44H46N10O3	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-8WLKM1	WO2024169871A1_I-6	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=NN(C3=CC=C(C4CCN(CC5CCN(C6=CC=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)C3=C2C(N)=NC=N3)C=C1	C47H49FN10O4	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-I3NEHJ	SCHEMBL31113518	N-[[4-[4-amino-1-[6-[1-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)-3-methylphenyl]piperidin-4-yl]methyl]piperidin-4-yl]pyridin-3-yl]pyrazolo[3,4-d]pyrimidin-3-yl]phenyl]methyl]-5-fluoro-2-methoxybenzamide	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=NN(C3=CN=C(C4CCN(CC5CCN(C6=CC(C)=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)C3=C2C(N)=NC=N3)C=C1	C47H50FN11O4	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-0CXXUP	WO2024169871A1_I-8	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=NN(C3=CC=C(N4CCN(CC5CCN(C6=CC(C)=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)C(N)=C2C(N)=O)C=C1	C46H51FN10O5	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-RG497H	WO2024169871A1_I-9	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=NN(C3=CC=C(N4CCN(CC5CCN(C6=CC(C)=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)C3=C2C(N)=NC=N3)C=C1	C47H50FN11O4	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-2HWF4W	WO2024169871A1_II-1	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=NN(C3=CN=C(N4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)CC5)CC4)C=C3)C3=C2C(N)=NC=N3)C=C1	C48H49FN12O5	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-3B28BG	WO2024169871A1_II-10	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=NN(C3=CC=C(N4CCN(CC5CCN(C6=CC=C7CN(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C=C3)C(N)=C2C(N)=O)C=C1	C48H51FN10O6	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-E0VORB	WO2024169871A1_II-11	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=NN(C3=CC=C(N4CCN(CC5CCN(C6=CC=C7CN(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C(F)=C3)C(N)=C2C(N)=O)C=C1	C48H50F2N10O6	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-9TA4U3	SCHEMBL31113510	N-[[4-[4-amino-1-[6-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-3-yl]pyrazolo[4,3-c]pyridin-3-yl]phenyl]methyl]-5-fluoro-2-methoxybenzamide	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=NN(C3=CN=C(N4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)CC5)CC4)C=C3)C3=C2C(N)=NC=C3)C=C1	C49H50FN11O5	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-ZMCXUU	WO2024169871A1_II-13	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(N2N=C(C3=CN=C(N4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)CC5)CC4)C=C3)C3=C2C(N)=NC=C3)C=C1	C49H50FN11O5	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-1WPJ9F	WO2024169871A1_II-14	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=C3C(N)=NC=CN3C(C3=CN=C(N4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)CC5)CC4)C=C3)=N2)C=C1	C49H50FN11O5	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-GCQ44B	WO2024169871A1_II-15	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=NN(C3=CN=C(N4CCC(CN5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)CC5)CC4)C=C3)C3=C2C(N)=NC=C3)C=C1	C49H50FN11O5	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-V1SFAD	WO2024169871A1_II-16	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(N2N=C(C3=CN=C(N4CCC(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)CC5)CC4)C=C3)C3=C2C(N)=NC=C3)C=C1	C50H51FN10O5	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-WOKDJ1	WO2024169871A1_II-17	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=C3C(N)=NC=CN3C(C3=CN=C(N4CCC(CN5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)CC5)CC4)C=C3)=N2)C=C1	C49H50FN11O5	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-PVSC2Y	WO2024169871A1_II-18	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=C3C(N)=NC=CN3C(C3=CC(F)=C(N4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)CC5)CC4)C=C3)=N2)C=C1	C50H50F2N10O5	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-3RWM4W	WO2024169871A1_II-19	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=C3C(N)=NC=CN3C(C3=CC=C(N4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)CC5)CC4)C=C3)=N2)C=C1	C50H51FN10O5	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-RYS484	SCHEMBL31113894	N-[[4-[4-amino-1-[6-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-3-yl]pyrazolo[3,4-d]pyrimidin-3-yl]-2-methylphenyl]methyl]-5-fluoro-2-methoxybenzamide	COC1=CC=C(F)C=C1C(=O)NCC1=C(C)C=C(C2=NN(C3=CN=C(N4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)CC5)CC4)C=C3)C3=C2C(N)=NC=N3)C=C1	C49H51FN12O5	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-1D4MML	WO2024169871A1_II-20	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=NN(C3=CC=C(N4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)CC5)CC4)C=C3)C3=C2C(N)=NC=C3)C=C1	C50H51FN10O5	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-E8MH7Y	WO2024169871A1_II-21	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(N2N=C(C3=CC=C(N4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)CC5)CC4)C=C3)C3=C2C(N)=NC=C3)C=C1	C50H51FN10O5	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-4U0QUE	WO2024169871A1_II-22	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=NN(C3=CC=C(N4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)CC5)CC4)C=C3)C3=C2C(N)=NNC3=O)C=C1	C49H50FN11O6	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-GF7HC7	WO2024169871A1_II-23	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(N2C(=O)N(C3=CC=C(N4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)CC5)CC4)C=C3)C3=C2C(N)=NC=N3)C=C1	C49H50FN11O6	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-Z5SU8D	SCHEMBL31113520	N-[[4-[4-amino-1-[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]phenyl]-2-oxoimidazo[4,5-c]pyridin-3-yl]phenyl]methyl]-5-fluoro-2-methoxybenzamide	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(N2C(=O)N(C3=CC=C(N4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)CC5)CC4)C=C3)C3=C2C(N)=NC=C3)C=C1	C50H51FN10O6	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-A90872	WO2024169871A1_II-28	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=NN(C3=CN=C(N4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)CC5)CC4)C=C3)C3=C2C(N)=NNC3=O)C=C1	C48H49FN12O6	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-Q7XYKO	WO2024169871A1_II-29	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(N2C(=O)N(C3=CN=C(N4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)CC5)CC4)C=C3)C3=C2C(N)=NC=N3)C=C1	C48H49FN12O6	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-3X4KFS	WO2024169871A1_II-3	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=NN(C3=CN=C(N4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C=C3)C3=C2C(N)=NC=N3)C=C1	C48H47FN12O6	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-ZFBW2V	WO2024169871A1_II-30	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(N2C(=O)N(C3=CN=C(N4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)CC5)CC4)C=C3)C3=C2C(N)=NC=C3)C=C1	C49H50FN11O6	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-PHOENP	WO2024169871A1_II-31	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=C3C(N)=NC=NN3C(C3=CC=C(N4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)CC5)CC4)C=C3)=C2)C=C1	C50H51FN10O5	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-XY6BZL	WO2024169871A1_II-32	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=NN(C3CCN(CC4CCN(C5=CC=C6CN(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)C3=C2C(N)=NC=N3)C=C1	C44H47FN10O5	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-PKU320	WO2024169871A1_II-33	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=NN(C3CCN(C4CN(CC5CCN(C6=CC=C7CN(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)C4)CC3)C3=C2C(N)=NC=N3)C=C1	C47H52FN11O5	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-ZT6Z2M	WO2024169871A1_II-34	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=NN(C3=CC=C(N4CCN(CC5CCN(C6=CC=C7CN(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)N=C3)C(N)=C2C(N)=O)C=C1	C47H50FN11O6	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-TQQMSZ	WO2024169871A1_II-35	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(N2C(=O)N(C3=CC=C(C4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)CC5)CC4)C=C3)C3=C2C(N)=NC=C3)C=C1	C51H52FN9O6	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-P1T1S0	WO2024169871A1_II-36	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(N2C(=O)N(C3=CC=C(C4=CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)CC5)CC4)C=C3)C3=C2C(N)=NC=C3)C=C1	C51H50FN9O6	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-KU2ZOT	SCHEMBL31113605	5-[4-[[1-[5-[4-Amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]pyridin-2-yl]piperidin-4-yl]methyl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	NC1=NC=NC2=C1C(C1=CC=C(OC3=CC=CC=C3)C=C1)=NN2C1=CC=C(N2CCC(CN3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)N=C1	C45H43N11O5	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-E72EI0	SCHEMBL31113721	N-[[4-[4-amino-1-[6-[(2S)-4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]-2-methylpiperazin-1-yl]pyridin-3-yl]pyrazolo[3,4-d]pyrimidin-3-yl]phenyl]methyl]-5-fluoro-2-methoxybenzamide	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=NN(C3=CN=C(N4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)CC5)C[C@@H]4C)C=C3)C3=C2C(N)=NC=N3)C=C1	C49H51FN12O5	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-253ZXH	WO2024169871A1_II-39	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=NN(C3=CC=C(C4CCN(CC5CCN(C6=CC=C7CN(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C=C3)C(N)=C2C(N)=O)C=C1	C49H52FN9O6	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-V1II6I	SCHEMBL31113749	N-[[4-[4-amino-1-[6-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-3-oxo-1H-isoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]pyridin-3-yl]pyrazolo[3,4-d]pyrimidin-3-yl]phenyl]methyl]-5-fluoro-2-methoxybenzamide	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=NN(C3=CC=C(N4CCC(CN5CCN(C6=CC=C7CN(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)N=C3)C3=C2C(N)=NC=N3)C=C1	C48H49FN12O5	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-YM4J02	SCHEMBL31113686	N-[[4-[4-amino-1-[6-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-3-yl]pyrazolo[3,4-d]pyrimidin-3-yl]-2-fluorophenyl]methyl]-5-fluoro-2-methoxybenzamide	COC1=CC=C(F)C=C1C(=O)NCC1=C(F)C=C(C2=NN(C3=CN=C(N4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)CC5)CC4)C=C3)C3=C2C(N)=NC=N3)C=C1	C48H48F2N12O5	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-XQ42QJ	SCHEMBL31113855	N-[[4-[4-amino-1-[6-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]pyridin-3-yl]pyrazolo[3,4-d]pyrimidin-3-yl]-2-methylphenyl]methyl]-5-fluoro-2-methoxybenzamide	COC1=CC=C(F)C=C1C(=O)NCC1=C(C)C=C(C2=NN(C3=CN=C(N4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C=C3)C3=C2C(N)=NC=N3)C=C1	C49H49FN12O6	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-XHM35C	SCHEMBL31113714	N-[[4-[4-amino-1-[6-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperidin-4-yl]pyridin-3-yl]pyrazolo[3,4-d]pyrimidin-3-yl]phenyl]methyl]-5-fluoro-2-methoxybenzamide	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=NN(C3=CN=C(C4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C=C3)C3=C2C(N)=NC=N3)C=C1	C49H48FN11O6	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-5JE2GJ	WO2024169871A1_II-9	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=NN(C3=CN=C(C4CCN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)CC5)CC4)C=C3)C3=C2C(N)=NC=N3)C=C1	C49H50FN11O5	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-7XBSJQ	WO2024169871A1_III-1	.	COC1=C(C(=O)NCC2=CC=C(C3=NN(C4CCN(C5CCN(C[C@@H]6CCCC[C@H]6CN6CCN(C7=CC=C(N8CCC(=O)NC8=O)C=C7)CC6)CC5)CC4)C4=C3C(N)=NC=N4)C=C2)C=C(F)C=C1	C52H65FN12O4	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-54GZ20	WO2024169871A1_III-10	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=C3C(N)=NC=CN3C(C3=CC=C(N4CCN(C[C@@H]5CCCC[C@H]5CN5CCN(C6=CC(C)=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)=N2)C=C1	C54H62FN11O4	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-0OMZVM	WO2024169871A1_III-11	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=C3C(N)=NC=CN3C(C3=CC(F)=C(N4CCN(C[C@H]5CCCC[C@@H]5CN5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)CC5)CC4)C=C3)=N2)C=C1	C56H61F2N11O5	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-4B8VVH	WO2024169871A1_III-12	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=C3C(N)=NC=CN3C(C3=CC(F)=C(N4CCN(C[C@@H]5CCCC[C@H]5CN5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)CC5)CC4)C=C3)=N2)C=C1	C56H61F2N11O5	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-1PDWGV	WO2024169871A1_III-13	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=C3C(N)=NC=CN3C(C3=CN=C(N4CCN(C[C@@H]5CCCC[C@H]5CN5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)CC5)CC4)C=C3)=N2)C=C1	C55H61FN12O5	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-FDA5UF	WO2024169871A1_III-14	.	COC1=C(C(=O)NCC2=CC=C(C3=NN(C4=CC=C(N5CCN(C[C@H]6CCCC[C@@H]6CN6CCN(C7=CC(C)=C(N8CCC(=O)NC8=O)C=C7)CC6)CC5)N=C4)C4=C3C(N)=NC=N4)C=C2)C=C(F)C=C1	C52H60FN13O4	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-GSNRBS	WO2024169871A1_III-15	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=C3C(N)=NC=CN3C(C3=CC(F)=C(N4CCN(C[C@H]5CCCC[C@@H]5CN5CCN(C6=CC(C)=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)=N2)C=C1	C54H61F2N11O4	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-KC3QKY	WO2024169871A1_III-17	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=C3C(N)=NC=CN3C(C3=CC(F)=C(N4CCN(C[C@@H]5CCCC[C@H]5CN5CCN(C6=CC(C)=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)=N2)C=C1	C54H61F2N11O4	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-S4P7QI	SCHEMBL31113371	3-[6-[4-[[(1R,2R)-2-[[4-[5-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]pyridin-2-yl]piperazin-1-yl]methyl]cyclohexyl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	NC1=NC=NC2=C1C(C1=CC=C(OC3=CC=CC=C3)C=C1)=NN2C1=CN=C(N2CCN(C[C@@H]3CCCC[C@H]3CN3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)CC5=C4)CC3)CC2)C=C1	C51H56N12O4	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-JZIT3E	SCHEMBL31113568	1-[4-[4-[[(1R,2R)-2-[[3-[4-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]azetidin-1-yl]methyl]cyclohexyl]methyl]piperazin-1-yl]phenyl]-1,3-diazinane-2,4-dione	NC1=NC=NC2=C1C(C1=CC=C(OC3=CC=CC=C3)C=C1)=NN2C1CCN(C2CN(C[C@@H]3CCCC[C@H]3CN3CCN(C4=CC=C(N5CCC(=O)NC5=O)C=C4)CC3)C2)CC1	C47H57N11O3	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-3CUGE2	SCHEMBL31113610	1-[4-[4-[[(1R,2R)-2-[[4-[5-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]pyridin-2-yl]piperazin-1-yl]methyl]cyclohexyl]methyl]piperazin-1-yl]-2-methylphenyl]-1,3-diazinane-2,4-dione	CC1=C(N2CCC(=O)NC2=O)C=CC(N2CCN(C[C@@H]3CCCC[C@H]3CN3CCN(C4=NC=C(N5N=C(C6=CC=C(OC7=CC=CC=C7)C=C6)C6=C5N=CN=C6N)C=C4)CC3)CC2)=C1	C49H56N12O3	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-BQ2890	WO2024169871A1_III-3	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=NN(C3CCN(C4CCN(C[C@@H]5CCCC[C@H]5CN5CCN(C6=CC=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)CC3)C(N)=C2C(N)=O)C=C1	C51H66FN11O5	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-J2Y3CE	WO2024169871A1_III-4	.	COC1=C(C(=O)NCC2=CC=C(C3=NN(C4CCN(C5CCN(C[C@@H]6CCCC[C@H]6CN6CCN(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8)CC6)CC5)CC4)C4=C3C(N)=NC=N4)C=C2)C=C(F)C=C1	C55H67FN12O5	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-UACZBC	WO2024169871A1_III-7	.	COC1=C(C(=O)NCC2=CC=C(C3=NN(C4CCN(C5CCN(C[C@H]6CCCC[C@@H]6CN6CCN(C7=CC=C(N8CCC(=O)NC8=O)C=C7)CC6)CC5)CC4)C4=C3C(N)=NC=N4)C=C2)C=C(F)C=C1	C52H65FN12O4	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-B6XWXA	WO2024169871A1_III-8	.	COC1=C(C(=O)NCC2=CC=C(C3=NN(C4CCN(C5CN(C[C@@H]6CCCC[C@H]6CN6CCN(C7=CC=C(N8CCC(=O)NC8=O)C=C7)CC6)C5)CC4)C4=C3C(N)=NC=N4)C=C2)C=C(F)C=C1	C50H61FN12O4	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-DWWIT2	WO2024169871A1_III-9	.	COC1=CC=C(F)C=C1C(=O)NCC1=CC=C(C2=C3C(N)=NC=CN3C(C3=CC=C(N4CCN(C[C@H]5CCCC[C@@H]5CN5CCN(C6=CC(C)=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)=N2)C=C1	C54H62FN11O4	BTK	Q06187	CRBN	WO-2024169871-A1
TPD-8NT8TH	WO2024169976A1_1	.	C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](NC(=O)CCCCCCC(=O)N1CCN(CC[C@H](CSc2ccccc2)Nc2ccc(S(=O)(=O)NC(=O)c3ccc(N4CCN(CC5=C(c6ccc(Cl)cc6)CCC(C)(C)C5)CC4)cc3)cc2S(=O)(=O)C(F)(F)F)CC1)C(C)(C)C)c1ccc(-c2ccnn2C)cc1	C78H99ClF3N11O10S3	BCL2L1	Q07817	VHL	WO-2024169976-A1
TPD-BAX85H	WO2024169976A1_2	.	CCn1nccc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCC(=O)N2CCN(CC[C@H](CSc3ccccc3)Nc3ccc(S(=O)(=O)NC(=O)c4ccc(N5CCN(CC6=C(c7ccc(Cl)cc7)CCC(C)(C)C6)CC5)cc4)cc3S(=O)(=O)C(F)(F)F)CC2)C(C)(C)C)cc1	C79H101ClF3N11O10S3	BCL2L1	Q07817	VHL	WO-2024169976-A1
TPD-FLNLX2	WO2024169976A1_3	.	CCn1nccc1-c1ccc([C@H](CO)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCC(=O)N2CCN(C[C@]3(C)CCC(c4ccc(Cl)cc4)=C(CN4CCN(c5ccc(C(=O)NS(=O)(=O)c6ccc(N[C@H](CCN7CCOCC7)CSc7ccccc7)c(S(=O)(=O)C(F)(F)F)c6)cc5)CC4)C3)CC2)C(C)(C)C)cc1	C83H108ClF3N12O12S3	BCL2L1	Q07817	VHL	WO-2024169976-A1
TPD-IY164P	WO2024169976A1_4	.	Cn1nccc1-c1ccc([C@H](CO)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCC(=O)N2CCN(C[C@]3(C)CCC(c4ccc(Cl)cc4)=C(CN4CCN(c5ccc(C(=O)NS(=O)(=O)c6ccc(N[C@H](CCN7CCOCC7)CSc7ccccc7)c(S(=O)(=O)C(F)(F)F)c6)cc5)CC4)C3)CC2)C(C)(C)C)cc1	C82H106ClF3N12O12S3	BCL2L1	Q07817	VHL	WO-2024169976-A1
TPD-0O13E0	WO2024169976A1_5	.	CCn1nccc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCC(=O)N2CCN(C[C@]3(C)CCC(c4ccc(Cl)cc4)=C(CN4CCN(c5ccc(C(=O)NS(=O)(=O)c6ccc(N[C@H](CCN7CCOCC7)CSc7ccccc7)c(S(=O)(=O)C(F)(F)F)c6)cc5)CC4)C3)CC2)C(C)(C)C)cc1	C83H108ClF3N12O11S3	BCL2L1	Q07817	VHL	WO-2024169976-A1
TPD-OZWVSX	WO2024169976A1_6	.	CCn1nccc1-c1ccc([C@H](CO)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCC(=O)N2CCN(C[C@]3(C)CCC(c4ccc(Cl)cc4)=C(CN4CCN(c5ccc(C(=O)NS(=O)(=O)c6ccc(N[C@H](CCN7CCOCC7)CSc7ccccc7)c(S(=O)(=O)C(F)(F)F)c6)cc5)CC4)C3)CC2)C(C)C)cc1	C82H106ClF3N12O12S3	BCL2L1	Q07817	VHL	WO-2024169976-A1
TPD-V0GOD4	WO2024169976A1_7	.	CC(C)C(NC(=O)CCCCCC(=O)N1CCN(CC[C@H](CSc2ccccc2)Nc2ccc(S(=O)(=O)NC(=O)c3ccc(N4CCN(CC5=C(c6ccc(Cl)cc6)CCC(C)(C)C5)CC4)cc3)cc2S(=O)(=O)C(F)(F)F)CC1)C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](CO)c1ccc(-c2ccnn2C)cc1	C76H95ClF3N11O11S3	BCL2L1	Q07817	VHL	WO-2024169976-A1
TPD-R11CO4	WO2024169976A1_8	.	CCn1nccc1-c1ccc([C@H](CO)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)C(NC(=O)CCCCCC(=O)N2CCN(CC[C@H](CSc3ccccc3)Nc3ccc(S(=O)(=O)NC(=O)c4ccc(N5CCN(CC6=C(c7ccc(Cl)cc7)CCC(C)(C)C6)CC5)cc4)cc3S(=O)(=O)C(F)(F)F)CC2)C(C)C)cc1	C77H97ClF3N11O11S3	BCL2L1	Q07817	VHL	WO-2024169976-A1
TPD-WB3GLV	WO2024169976A1_9	.	Cc1ncsc1-c1ccc([C@H](CO)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)C(NC(=O)CCCCCC(=O)N2CCN(CC[C@H](CSc3ccccc3)Nc3ccc(S(=O)(=O)NC(=O)c4ccc(N5CCN(CC6=C(c7ccc(Cl)cc7)CCC(C)(C)C6)CC5)cc4)cc3S(=O)(=O)C(F)(F)F)CC2)C(C)C)cc1	C76H94ClF3N10O11S4	BCL2L1	Q07817	VHL	WO-2024169976-A1
TPD-FWJ20T	WO2024169976A1_10	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)C(NC(=O)CCCCCCC(=O)N2CCN(CC[C@H](CSc3ccccc3)Nc3ccc(S(=O)(=O)NC(=O)c4ccc(N5CCN(CC6=C(c7ccc(Cl)cc7)CCC(C)(C)C6)CC5)cc4)cc3S(=O)(=O)C(F)(F)F)CC2)C(C)(C)C)cc1	C78H98ClF3N10O10S4	BCL2L1	Q07817	VHL	WO-2024169976-A1
TPD-WSNV7U	WO2024169976A1_11	.	CC(C)C(NC(=O)CCCCCCC(=O)N1CCN(CC[C@H](CSc2ccccc2)Nc2ccc(S(=O)(=O)NC(=O)c3ccc(N4CCN(CC5=C(c6ccc(Cl)cc6)CCC(C)(C)C5)CC4)cc3)cc2S(=O)(=O)C(F)(F)F)CC1)C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)c1ccc(-c2ccnn2C)cc1	C77H97ClF3N11O10S3	BCL2L1	Q07817	VHL	WO-2024169976-A1
TPD-S3Y7U9	WO2024169976A1_12	.	CC(C)C(NC(=O)CCCCCCC(=O)N1CCN(CC[C@H](CSc2ccccc2)Nc2ccc(S(=O)(=O)NC(=O)c3ccc(N4CCN(CC5=C(c6ccc(Cl)cc6)CCC(C)(C)C5)CC4)cc3)cc2S(=O)(=O)C(F)(F)F)CC1)C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](CO)c1ccc(-c2ccnn2C)cc1	C77H97ClF3N11O11S3	BCL2L1	Q07817	VHL	WO-2024169976-A1
TPD-L6XUAR	WO2024169976A1_13	.	CCn1nccc1-c1ccc([C@H](CO)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)C(NC(=O)CCCCCCC(=O)N2CCN(CC[C@H](CSc3ccccc3)Nc3ccc(S(=O)(=O)NC(=O)c4ccc(N5CCN(CC6=C(c7ccc(Cl)cc7)CCC(C)(C)C6)CC5)cc4)cc3S(=O)(=O)C(F)(F)F)CC2)C(C)C)cc1	C78H99ClF3N11O11S3	BCL2L1	Q07817	VHL	WO-2024169976-A1
TPD-VVLEZQ	WO2024169976A1_14	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)C(NC(=O)CCCCCCC(=O)N2CCN(CC[C@H](CSc3ccccc3)Nc3ccc(S(=O)(=O)NC(=O)c4ccc(N5CCN(CC6=C(c7ccc(Cl)cc7)CCC(C)(C)C6)CC5)cc4)cc3S(=O)(=O)C(F)(F)F)CC2)C(C)C)cc1	C77H96ClF3N10O10S4	BCL2L1	Q07817	VHL	WO-2024169976-A1
TPD-P1OGAS	WO2024169976A1_15	.	Cc1ncsc1-c1ccc([C@H](CO)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)C(NC(=O)CCCCCCC(=O)N2CCN(CC[C@H](CSc3ccccc3)Nc3ccc(S(=O)(=O)NC(=O)c4ccc(N5CCN(CC6=C(c7ccc(Cl)cc7)CCC(C)(C)C6)CC5)cc4)cc3S(=O)(=O)C(F)(F)F)CC2)C(C)C)cc1	C77H96ClF3N10O11S4	BCL2L1	Q07817	VHL	WO-2024169976-A1
TPD-97BT5H	WO2024169976A1_16	.	Cn1nccc1-c1ccc([C@H](CO)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCCC(=O)N2CCN(CC[C@H](CSc3ccccc3)Nc3ccc(S(=O)(=O)NC(=O)c4ccc(N5CCN(CC6=C(c7ccc(Cl)cc7)CCC(C)(C)C6)CC5)cc4)cc3S(=O)(=O)C(F)(F)F)CC2)C(C)(C)C)cc1	C79H101ClF3N11O11S3	BCL2L1	Q07817	VHL	WO-2024169976-A1
TPD-19LBHB	WO2024169976A1_17	.	CCn1nccc1-c1ccc([C@H](CO)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCCC(=O)N2CCN(CC[C@H](CSc3ccccc3)Nc3ccc(S(=O)(=O)NC(=O)c4ccc(N5CCN(CC6=C(c7ccc(Cl)cc7)CCC(C)(C)C6)CC5)cc4)cc3S(=O)(=O)C(F)(F)F)CC2)C(C)(C)C)cc1	C80H103ClF3N11O11S3	BCL2L1	Q07817	VHL	WO-2024169976-A1
TPD-23BD7B	WO2024169976A1_18	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCCC(=O)N2CCN(CC[C@H](CSc3ccccc3)Nc3ccc(S(=O)(=O)NC(=O)c4ccc(N5CCN(CC6=C(c7ccc(Cl)cc7)CCC(C)(C)C6)CC5)cc4)cc3S(=O)(=O)C(F)(F)F)CC2)C(C)(C)C)cc1	C79H100ClF3N10O10S4	BCL2L1	Q07817	VHL	WO-2024169976-A1
TPD-6B27FL	WO2024169976A1_19	.	Cc1ncsc1-c1ccc([C@H](CO)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCCC(=O)N2CCN(CC[C@H](CSc3ccccc3)Nc3ccc(S(=O)(=O)NC(=O)c4ccc(N5CCN(CC6=C(c7ccc(Cl)cc7)CCC(C)(C)C6)CC5)cc4)cc3S(=O)(=O)C(F)(F)F)CC2)C(C)(C)C)cc1	C79H100ClF3N10O11S4	BCL2L1	Q07817	VHL	WO-2024169976-A1
TPD-G8XO19	WO2024169976A1_20	.	C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](NC(=O)CCCCCCCC(=O)N1CCN(CC[C@H](CSc2ccccc2)Nc2ccc(S(=O)(=O)NC(=O)c3ccc(N4CCN(CC5=C(c6ccc(Cl)cc6)CCC(C)(C)C5)CC4)cc3)cc2S(=O)(=O)C(F)(F)F)CC1)C(C)(C)C)c1ccc(-c2ccnn2C)cc1	C79H101ClF3N11O10S3	BCL2L1	Q07817	VHL	WO-2024169976-A1
TPD-LT00QR	WO2024169976A1_21	.	CC(C)[C@H](NC(=O)CCCCCCCC(=O)N1CCN(CC[C@H](CSc2ccccc2)Nc2ccc(S(=O)(=O)NC(=O)c3ccc(N4CCN(CC5=C(c6ccc(Cl)cc6)CCC(C)(C)C5)CC4)cc3)cc2S(=O)(=O)C(F)(F)F)CC1)C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](CO)c1ccc(-c2ccnn2C)cc1	C78H99ClF3N11O11S3	BCL2L1	Q07817	VHL	WO-2024169976-A1
TPD-RQJAFT	WO2024169976A1_22	.	CCn1nccc1-c1ccc([C@H](CO)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCCC(=O)N2CCN(CC[C@H](CSc3ccccc3)Nc3ccc(S(=O)(=O)NC(=O)c4ccc(N5CCN(CC6=C(c7ccc(Cl)cc7)CCC(C)(C)C6)CC5)cc4)cc3S(=O)(=O)C(F)(F)F)CC2)C(C)C)cc1	C79H101ClF3N11O11S3	BCL2L1	Q07817	VHL	WO-2024169976-A1
TPD-GE6UT1	WO2024169976A1_23	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCCC(=O)N2CCN(CC[C@H](CSc3ccccc3)Nc3ccc(S(=O)(=O)NC(=O)c4ccc(N5CCN(CC6=C(c7ccc(Cl)cc7)CCC(C)(C)C6)CC5)cc4)cc3S(=O)(=O)C(F)(F)F)CC2)C(C)C)cc1	C78H98ClF3N10O10S4	BCL2L1	Q07817	VHL	WO-2024169976-A1
TPD-T9NKMW	WO2024169976A1_24	.	Cc1ncsc1-c1ccc([C@H](CO)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCCC(=O)N2CCN(CC[C@H](CSc3ccccc3)Nc3ccc(S(=O)(=O)NC(=O)c4ccc(N5CCN(CC6=C(c7ccc(Cl)cc7)CCC(C)(C)C6)CC5)cc4)cc3S(=O)(=O)C(F)(F)F)CC2)C(C)C)cc1	C78H98ClF3N10O11S4	BCL2L1	Q07817	VHL	WO-2024169976-A1
TPD-KJHBI3	WO2024169976A1_25	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](NC(=O)CCCCCC(=O)N2CCN(CC[C@H](CSc3ccccc3)Nc3ccc(S(=O)(=O)NC(=O)c4ccc(N5CCN(CC6=C(c7ccc(Cl)cc7)CCC(C)(C)C6)CC5)cc4)cc3S(=O)(=O)C(F)(F)F)CC2)C(C)C)cc1	C76H94ClF3N10O10S4	BCL2L1	Q07817	VHL	WO-2024169976-A1
TPD-NU2IBB	WO2024169976A1_26	.	Cc1ncsc1-c1ccc([C@H](CO)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCC(=O)N2CCN(CC[C@H](CSc3ccccc3)Nc3ccc(S(=O)(=O)NC(=O)c4ccc(N5CCN(CC6=C(c7ccc(Cl)cc7)CCC(C)(C)C6)CC5)cc4)cc3S(=O)(=O)C(F)(F)F)CC2)C(C)(C)C)cc1	C77H96ClF3N10O11S4	BCL2L1	Q07817	VHL	WO-2024169976-A1
TPD-ZCMPQJ	WO2024169976A1_27	.	CCn1nccc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](NC(=O)CCCCCC(=O)N2CCN(CC[C@H](CSc3ccccc3)Nc3ccc(S(=O)(=O)NC(=O)c4ccc(N5CCN(CC6=C(c7ccc(Cl)cc7)CCC(C)(C)C6)CC5)cc4)cc3S(=O)(=O)C(F)(F)F)CC2)C(C)(C)C)cc1	C78H99ClF3N11O10S3	BCL2L1	Q07817	VHL	WO-2024169976-A1
TPD-3TMLDN	WO2024169976A1_28	.	C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@H](NC(=O)CCCCCC(=O)N1CCN(CC[C@H](CSc2ccccc2)Nc2ccc(S(=O)(=O)NC(=O)c3ccc(N4CCN(CC5=C(c6ccc(Cl)cc6)CCC(C)(C)C5)CC4)cc3)cc2S(=O)(=O)C(F)(F)F)CC1)C(C)(C)C)c1ccc(-c2ccnn2C)cc1	C77H97ClF3N11O10S3	BCL2L1	Q07817	VHL	WO-2024169976-A1
TPD-GY55CE	WO2024169976A1_29	.	CCn1nccc1-c1ccc([C@H](CO)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCC(=O)N2CCN(CC[C@H](CSc3ccccc3)Nc3ccc(S(=O)(=O)NC(=O)c4ccc(N5CCN(CC6=C(c7ccc(Cl)cc7)CCC(C)(C)C6)CC5)cc4)cc3S(=O)(=O)C(F)(F)F)CC2)C(C)(C)C)cc1	C79H101ClF3N11O11S3	BCL2L1	Q07817	VHL	WO-2024169976-A1
TPD-U19L9U	WO2024169976A1_30	.	Cc1ncsc1-c1ccc([C@H](CO)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCC(=O)N2CCN(CC[C@H](CSc3ccccc3)Nc3ccc(S(=O)(=O)NC(=O)c4ccc(N5CCN(CC6=C(c7ccc(Cl)cc7)CCC(C)(C)C6)CC5)cc4)cc3S(=O)(=O)C(F)(F)F)CC2)C(C)(C)C)cc1	C78H98ClF3N10O11S4	BCL2L1	Q07817	VHL	WO-2024169976-A1
TPD-ZPL3T0	WO2024169976A1_31	.	Cn1nccc1-c1ccc([C@H](CO)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCC(=O)N2CCN(CC[C@H](CSc3ccccc3)Nc3ccc(S(=O)(=O)NC(=O)c4ccc(N5CCN(CC6=C(c7ccc(Cl)cc7)CCC(C)(C)C6)CC5)cc4)cc3S(=O)(=O)C(F)(F)F)CC2)C(C)(C)C)cc1	C78H99ClF3N11O11S3	BCL2L1	Q07817	VHL	WO-2024169976-A1
TPD-GC6B11	WO2024169976A1_33	.	CCn1nccc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCCC(=O)N2CCN(CC[C@H](CSc3ccccc3)Nc3ccc(S(=O)(=O)NC(=O)c4ccc(N5CCN(CC6=C(c7ccc(Cl)cc7)CCC(C)(C)C6)CC5)cc4)cc3S(=O)(=O)C(F)(F)F)CC2)C(C)(C)C)cc1	C80H103ClF3N11O10S3	BCL2L1	Q07817	VHL	WO-2024169976-A1
TPD-JKAD8S	WO2024169976A1_34	.	CCn1nccc1-c1ccc([C@H](CO)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](NC(=O)CCCCCC(=O)N2CCN(CC[C@H](CSc3ccccc3)Nc3ccc(S(=O)(=O)NC(=O)c4ccc(N5CCN(CC6=C(c7ccc(Cl)cc7)CCC(C)(C)C6)CC5)cc4)cc3S(=O)(=O)C(F)(F)F)CC2)C(C)(C)C)cc1	C78H99ClF3N11O11S3	BCL2L1	Q07817	VHL	WO-2024169976-A1
TPD-76HCEC	WO2024169976A1_35	.	Cn1nccc1-c1ccc([C@H](CO)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](NC(=O)CCCCCC(=O)N2CCN(CC[C@H](CSc3ccccc3)Nc3ccc(S(=O)(=O)NC(=O)c4ccc(N5CCN(CC6=C(c7ccc(Cl)cc7)CCC(C)(C)C6)CC5)cc4)cc3S(=O)(=O)C(F)(F)F)CC2)C(C)(C)C)cc1	C77H97ClF3N11O11S3	BCL2L1	Q07817	VHL	WO-2024169976-A1
TPD-O71L9D	WO2024169976A1_36	.	C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](NC(=O)CCCCC(=O)N1CCN(CC[C@H](CSc2ccccc2)Nc2ccc(S(=O)(=O)NC(=O)c3ccc(N4CCN(CC5=C(c6ccc(Cl)cc6)CCC(C)(C)C5)CC4)cc3)cc2S(=O)C(F)(F)F)CC1)C(C)(C)C)c1ccc(-c2ccnn2C)cc1	C76H95ClF3N11O9S3	BCL2L1	Q07817	VHL	WO-2024169976-A1
TPD-INLZ6B	WO2024169976A1_37	.	CC(C)[C@H](NC(=O)CCCCC(=O)N1CCN(CC[C@H](CSc2ccccc2)Nc2ccc(S(=O)(=O)NC(=O)c3ccc(N4CCN(CC5=C(c6ccc(Cl)cc6)CCC(C)(C)C5)CC4)cc3)cc2S(=O)C(F)(F)F)CC1)C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)c1ccc(-c2ccnn2C)cc1	C75H93ClF3N11O9S3	BCL2L1	Q07817	VHL	WO-2024169976-A1
TPD-SCCLH5	WO2024169976A1_38	.	CCn1nccc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCC(=O)N2CCN(CC[C@H](CSc3ccccc3)Nc3ccc(S(=O)(=O)NC(=O)c4ccc(N5CCN(CC6=C(c7ccc(Cl)cc7)CCC(C)(C)C6)CC5)cc4)cc3S(=O)C(F)(F)F)CC2)C(C)(C)C)cc1	C77H97ClF3N11O9S3	BCL2L1	Q07817	VHL	WO-2024169976-A1
TPD-5SZRD1	WO2024169976A1_39	.	CCn1nccc1-c1ccc([C@H](CO)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCC(=O)N2CCN(CC[C@H](CSc3ccccc3)Nc3ccc(S(=O)(=O)NC(=O)c4ccc(N5CCN(CC6=C(c7ccc(Cl)cc7)CCC(C)(C)C6)CC5)cc4)cc3S(=O)C(F)(F)F)CC2)C(C)(C)C)cc1	C77H97ClF3N11O10S3	BCL2L1	Q07817	VHL	WO-2024169976-A1
TPD-7LWOLS	WO2024169976A1_40	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCC(=O)N2CCN(CC[C@H](CSc3ccccc3)Nc3ccc(S(=O)(=O)NC(=O)c4ccc(N5CCN(CC6=C(c7ccc(Cl)cc7)CCC(C)(C)C6)CC5)cc4)cc3S(=O)C(F)(F)F)CC2)C(C)(C)C)cc1	C76H94ClF3N10O9S4	BCL2L1	Q07817	VHL	WO-2024169976-A1
TPD-5LTJ5N	WO2024169976A1_41	.	Cc1ncsc1-c1ccc([C@H](CO)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCC(=O)N2CCN(CC[C@H](CSc3ccccc3)Nc3ccc(S(=O)(=O)NC(=O)c4ccc(N5CCN(CC6=C(c7ccc(Cl)cc7)CCC(C)(C)C6)CC5)cc4)cc3S(=O)C(F)(F)F)CC2)C(C)(C)C)cc1	C76H94ClF3N10O10S4	BCL2L1	Q07817	VHL	WO-2024169976-A1
TPD-RCJFHX	WO2024169976A1_42	.	CCn1nccc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCC(=O)N2CCN(CC[C@H](CSc3ccccc3)Nc3ccc(S(=O)(=O)NC(=O)c4ccc(N5CCN(CC6=C(c7ccc(Cl)cc7)CCC(C)(C)C6)CC5)cc4)cc3S(=O)(=O)C(F)(F)F)CC2)C(C)C)cc1	C77H97ClF3N11O10S3	BCL2L1	Q07817	VHL	WO-2024169976-A1
TPD-AOSELF	WO2024169976A1_43	.	CC(C)[C@H](NC(=O)CCCCCC(=O)N1CCN(CC[C@H](CSc2ccccc2)Nc2ccc(S(=O)(=O)NC(=O)c3ccc(N4CCN(CC5=C(c6ccc(Cl)cc6)CCC(C)(C)C5)CC4)cc3)cc2S(=O)(=O)C(F)(F)F)CC1)C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)c1ccc(-c2ccnn2C)cc1	C76H95ClF3N11O10S3	BCL2L1	Q07817	VHL	WO-2024169976-A1
TPD-QNFN45	WO2024169976A1_44	.	CCn1nccc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCC(=O)N2CCN(CC[C@H](CSc3ccccc3)Nc3ccc(S(=O)(=O)NC(=O)c4ccc(N5CCN(CC6=C(c7ccc(Cl)cc7)CCC(C)(C)C6)CC5)cc4)cc3S(=O)(=O)C(F)(F)F)CC2)C(C)C)cc1	C78H99ClF3N11O10S3	BCL2L1	Q07817	VHL	WO-2024169976-A1
TPD-PCRO01	WO2024169976A1_45	.	CCn1nccc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCCC(=O)N2CCN(CC[C@H](CSc3ccccc3)Nc3ccc(S(=O)(=O)NC(=O)c4ccc(N5CCN(CC6=C(c7ccc(Cl)cc7)CCC(C)(C)C6)CC5)cc4)cc3S(=O)(=O)C(F)(F)F)CC2)C(C)C)cc1	C79H101ClF3N11O10S3	BCL2L1	Q07817	VHL	WO-2024169976-A1
TPD-25N1CN	WO2024169976A1_46	.	CCn1nccc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)C(NC(=O)CCCCCCCCC(=O)N2CCN(CC[C@H](CSc3ccccc3)Nc3ccc(S(=O)(=O)NC(=O)c4ccc(N5CCN(CC6=C(c7ccc(Cl)cc7)CCC(C)(C)C6)CC5)cc4)cc3S(=O)(=O)C(F)(F)F)CC2)C(C)C)cc1	C80H103ClF3N11O10S3	BCL2L1	Q07817	VHL	WO-2024169976-A1
TPD-9B3UYA	WO2024169976A1_47	.	Cc1ncsc1-c1ccc([C@H](CO)NC(=O)C2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCC(=O)N2CCN(C[C@]3(C)CCC(c4ccc(Cl)cc4)=C(CN4CCN(c5ccc(C(=O)NS(=O)(=O)c6ccc(N[C@H](CCN7CCOCC7)CSc7ccccc7)c(S(=O)(=O)C(F)(F)F)c6)cc5)CC4)C3)CC2)C(C)(C)C)cc1	C82H105ClF3N11O12S4	BCL2L1	Q07817	VHL	WO-2024169976-A1
TPD-2P9FAR	WO2024169976A1_48	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)C2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCC(=O)N2CCN(C[C@]3(C)CCC(c4ccc(Cl)cc4)=C(CN4CCN(c5ccc(C(=O)NS(=O)(=O)c6ccc(N[C@H](CCN7CCOCC7)CSc7ccccc7)c(S(=O)(=O)C(F)(F)F)c6)cc5)CC4)C3)CC2)C(C)C)cc1	C81H103ClF3N11O11S4	BCL2L1	Q07817	VHL	WO-2024169976-A1
TPD-7WSKKG	WO2024169976A1_49	.	CCn1nccc1-c1ccc([C@H](C)NC(=O)C2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCC(=O)N2CCN(C[C@]3(C)CCC(c4ccc(Cl)cc4)=C(CN4CCN(c5ccc(C(=O)NS(=O)(=O)c6ccc(N[C@H](CCN7CCOCC7)CSc7ccccc7)c(S(=O)(=O)C(F)(F)F)c6)cc5)CC4)C3)CC2)C(C)C)cc1	C82H106ClF3N12O11S3	BCL2L1	Q07817	VHL	WO-2024169976-A1
TPD-RHZNQG	WO2024169976A1_50	.	Cc1ncsc1-c1ccc([C@H](CO)NC(=O)C2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCC(=O)N2CCN(C[C@]3(C)CCC(c4ccc(Cl)cc4)=C(CN4CCN(c5ccc(C(=O)NS(=O)(=O)c6ccc(N[C@H](CCN7CCOCC7)CSc7ccccc7)c(S(=O)(=O)C(F)(F)F)c6)cc5)CC4)C3)CC2)C(C)C)cc1	C81H103ClF3N11O12S4	BCL2L1	Q07817	VHL	WO-2024169976-A1
TPD-CQ6OQD	WO2024175065A1_YJZ1078	.	O=C1CCC(N2C(=O)C3=CC=C(N4C=CC(C(=O)N5CCN(C6=CC=C(N(C(=O)NCC7=CC=CC=C7)[C@H]7CC[C@@H](NC8=NC=C9C=CC=CC9=N8)CC7)C=C6)CC5)=N4)C=C3C2=O)C(=O)N1	C49H47N11O6	CDK12;KIAA1791	Q9NYV4/Q14004	CRBN	WO-2024175065-A1
TPD-9MKUAV	WO2024175065A1_YJZ1090	.	O=C1CCC(N2C(=O)C3=CC=C(OCC(=O)N4CCN(C5=CC=C(N(C(=O)NCC6=CC=CC=C6)[C@H]6CC[C@H](NC7=NC=C8C=CC=CC8=N7)CC6)C=C5)CC4)C=C3C2=O)C(=O)N1	C47H47N9O7	CDK12;KIAA1791	Q9NYV4/Q14004	CRBN	WO-2024175065-A1
TPD-XBRO6Q	WO2024175065A1_YJZ1091	.	O=C1CCC(N2C(=O)C3=CC=C(NCC(=O)N4CCN(C5=CC=C(N(C(=O)NCC6=CC=CC=C6)[C@H]6CC[C@H](NC7=NC=C8C=CC=CC8=N7)CC6)C=C5)CC4)C=C3C2=O)C(=O)N1	C47H48N10O6	CDK12;KIAA1791	Q9NYV4/Q14004	CRBN	WO-2024175065-A1
TPD-CW61OQ	WO2024175065A1_YJZ1094	.	O=C1CCC(N2CC3=CC=C(OCC(=O)N4CCN(C5=CC=C(N(C(=O)NCC6=CC=CC=C6)[C@H]6CC[C@H](NC7=NC=C8C=CC=CC8=N7)CC6)C=C5)CC4)C=C3C2=O)C(=O)N1	C47H49N9O6	CDK12;KIAA1791	Q9NYV4/Q14004	CRBN	WO-2024175065-A1
TPD-DEH1IC	WO2024175065A1_YJZ1095	.	O=C1CCC(N2CC3=CC=C(NCC(=O)N4CCN(C5=CC=C(N(C(=O)NCC6=CC=CC=C6)[C@H]6CC[C@H](NC7=NC=C8C=CC=CC8=N7)CC6)C=C5)CC4)C=C3C2=O)C(=O)N1	C47H50N10O5	CDK12;KIAA1791	Q9NYV4/Q14004	CRBN	WO-2024175065-A1
TPD-IFR6TN	WO2024175065A1_YJZ1096	.	O=C1CCC(N2C(=O)C3=CC=C(N4CCC(N5CCN(C6=CC=C(N(C(=O)NCC7=CC=CC=C7)[C@H]7CC[C@H](NC8=NC=C9C=CC=CC9=N8)CC7)C=C6)CC5)C4)C=C3C2=O)C(=O)N1	C49H52N10O5	CDK12;KIAA1791	Q9NYV4/Q14004	CRBN	WO-2024175065-A1
TPD-YDK41J	WO2024175065A1_YJZ1097	.	O=C1CCC(N2C(=O)C3C=CC(N4CCC(CN5CCN(C6=CCC(N(C(=O)NCC7=CC=CC=C7)C7CCC(NC8=NC=C9C=CC=CC9=N8)CC7)C=C6)CC5)CC4)=CC3C2=O)C(=O)N1	C51H60N10O5	CDK12;KIAA1791	Q9NYV4/Q14004	CRBN	WO-2024175065-A1
TPD-0XHQXR	WO2024175065A1_YJZ1102	.	O=C1CCC(N2C(=O)C3=CC=CC(NCCCCCCCC(=O)NC4=CC(N(C(=O)NCC5=CC=CC=C5)[C@H]5CC[C@@H](NC6=NC=C7C=CC=CC7=N6)CC5)=CC=C4)=C3C2=O)C(=O)N1	C49H53N9O6	CDK12;KIAA1791	Q9NYV4/Q14004	CRBN	WO-2024175065-A1
TPD-7MZA9N	WO2024175065A1_YJZ1103	.	O=C1CCC(N2C(=O)C3C=CC(N4CC(N5CCN(C6=CCC(N(C(=O)NCC7=CCCC=C7)[C@H]7CC[C@H](NC8=NC=C9C=CC=CC9=N8)CC7)C=C6)CC5)C4)=CC3C2=O)C(=O)N1	C48H56N10O5	CDK12;KIAA1791	Q9NYV4/Q14004	CRBN	WO-2024175065-A1
TPD-0H1B75	WO2024175065A1_YJZ1105	.	O=C1CCC(N2C(=O)C3=CC=C(N4CCC(N5CCN(C6=CC=C(N(C(=O)NCC7=CC=CC=C7)[C@H]7CC[C@@H](NC8=NC=C9C=CC=CC9=N8)CC7)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C50H54N10O5	CDK12;KIAA1791	Q9NYV4/Q14004	CRBN	WO-2024175065-A1
TPD-NUAJL5	WO2024175065A1_YJZ1114	.	O=C1CCC(N2C(=O)C3=CC=C(N4CC(C(=O)N5CCN(C6=CC=C(N(C(=O)NCC7=CC=CC=C7)[C@H]7CC[C@H](NC8=NC=C9C=CC=CC9=N8)CC7)C=C6)CC5)C4)C=C3C2=O)C(=O)N1	C49H50N10O6	CDK12;KIAA1791	Q9NYV4/Q14004	CRBN	WO-2024175065-A1
TPD-W89JFV	WO2024175065A1_YJZ1130	.	O=C1CCC(N2C(=O)C3=CC=C(/C=C/C(=O)N4CCN(C5=CC=C(N(C(=O)NCC6=CC=CC=C6)[C@H]6CC[C@H](NC7=NC=C8C=CC=CC8=N7)CC6)C=C5)CC4)C=C3C2=O)C(=O)N1	C48H47N9O6	CDK12;KIAA1791	Q9NYV4/Q14004	CRBN	WO-2024175065-A1
TPD-GV30H6	WO2024175065A1_YJZ1131	.	O=C1CCC(N2C(=O)C3=C(C=C(C4=CC=CC(C(=O)N5CCN(C6=CC=C(N(C(=O)NCC7=CC=CC=C7)[C@H]7CC[C@H](NC8=NC=C9C=CC=CC9=N8)CC7)C=C6)CC5)=C4)C=C3)C2=O)C(=O)N1	C52H49N9O6	CDK12;KIAA1791	Q9NYV4/Q14004	CRBN	WO-2024175065-A1
TPD-XC5D8J	WO2024175065A1_YJZ1201	.	O=C1CCC(N2C(=O)C3=CC(F)=C(N4CCC(N5CCN(C6=CC=C(N(C(=O)NCC7=CCCC=C7)[C@H]7CC[C@@H](NC8=NC=C9C=CC=CC9=N8)CC7)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C50H55FN10O5	CDK12;KIAA1791	Q9NYV4/Q14004	CRBN	WO-2024175065-A1
TPD-WZ2ERV	WO2024175065A1_YJZ1202	.	O=C1CCC(N2C(=O)C3=CC=C(N4CCC(N5CCN(C6=C(F)C=C(N(C(=O)NCC7=CCCC=C7)[C@H]7CC[C@@H](NC8=NC=C9C=CC=CC9=N8)CC7)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C50H55FN10O5	CDK12;KIAA1791	Q9NYV4/Q14004	CRBN	WO-2024175065-A1
TPD-IHWWO1	WO2024175065A1_YJZ1203	.	O=C1CCC(N2C(=O)C3=CC=C(N4CCC(N5CCN(C6=NCC(N(C(=O)NCC7=CC=CC=C7)[C@H]7CC[C@@H](NC8=NC=C9C=CC=CC9=N8)CC7)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C49H55N11O5	CDK12;KIAA1791	Q9NYV4/Q14004	CRBN	WO-2024175065-A1
TPD-UHGEV8	WO2024175065A1_YJZ1204	.	O=C1CCC(N2C(=O)C3=CC=C(N4CCC(N5CCN(C6=CC=C(N(C(=O)NCC7=C(F)C=CC=C7)[C@H]7CC[C@@H](NC8=NC=C9C=CC=CC9=N8)CC7)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C50H53FN10O5	CDK12;KIAA1791	Q9NYV4/Q14004	CRBN	WO-2024175065-A1
TPD-JJ0V5S	WO2024175065A1_YJZ1205	.	O=C1CCC(N2C(=O)C3=CC(F)=C(N4CCC(N5CCN(C6=NCC(N(C(=O)NCC7=CC=CC=C7)[C@H]7CC[C@@H](NC8=NC=C9C=CC=CC9=N8)CC7)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C49H54FN11O5	CDK12;KIAA1791	Q9NYV4/Q14004	CRBN	WO-2024175065-A1
TPD-KBVEZ3	WO2024175065A1_YJZ1206	.	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(C5CCN(C6=CC=C(N(C(=O)NCC7=CCCC=C7)[C@H]7CC[C@H](NC8=NC=C9C=CC=CC9=N8)CC7)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C50H56N10O5	CDK12;KIAA1791	Q9NYV4/Q14004	CRBN	WO-2024175065-A1
TPD-SLKZGX	WO2024175065A1_YJZ9043	.	O=C(COC1=C2C(=O)N(C3CCC(=O)NC3=O)C(=O)C2=CC=C1)NCCCCCN1CCN(C2=CC(N(C(=O)NCC3=CC=CC=C3)[C@H]3CC[C@@H](NC4=NC=C5C=CC=CC5=N4)CC3)=CC=C2)CC1	C52H58N10O7	CDK12;KIAA1791	Q9NYV4/Q14004	CRBN	WO-2024175065-A1
TPD-Z0EHJK	WO2024175065A1_YJZ9047	.	O=C(COC1=CC=CC2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O)NCCCCCCN1CCN(C2=CC(N(C(=O)NCC3=CC=CC=C3)[C@H]3CC[C@@H](NC4=NC=C5C=CC=CC5=N4)CC3)=CC=C2)CC1	C53H60N10O7	CDK12;KIAA1791	Q9NYV4/Q14004	CRBN	WO-2024175065-A1
TPD-GWFU3I	WO2024175065A1_YJZ9048	.	O=C(COC1=C2C(=O)N(C3CCC(=O)NC3=O)C(=O)C2=CC=C1)NCCCCN1CCN(C2=CC(N(C(=O)NCC3=CC=CC=C3)[C@H]3CC[C@H](NC4=NC=C5C=CC=CC5=N4)CC3)=CC=C2)CC1	C51H56N10O7	CDK12;KIAA1791	Q9NYV4/Q14004	CRBN	WO-2024175065-A1
TPD-4IPDMY	WO2024175065A1_YJZ9049	.	CCCN1N=CC2=CN=C(N[C@H]3CC[C@H](N(C(=O)NCC4=CC=CC=C4)C4=CC=C(N5CCN(C(=O)COC6=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)CC5)C=C4)CC3)N=C21	C47H51N11O7	CDK12;KIAA1791	Q9NYV4/Q14004	CRBN	WO-2024175065-A1
TPD-V0C8W4	WO2024175065A1_YJZ9052	.	O=C1CCC(N2C(=O)C3=CC=CC(NCCCC(=O)N4CCN(C5=CC(N(C(=O)NCC6=CC=CC=C6)[C@H]6CC[C@H](NC7=NC=C8C=CC=CC8=N7)CC6)=CC=C5)CC4)=C3C2=O)C(=O)N1	C49H52N10O6	CDK12;KIAA1791	Q9NYV4/Q14004	CRBN	WO-2024175065-A1
TPD-8O91EH	WO2024175065A1_YJZ9053	.	O=C1CCC(N2C(=O)C3=CC=CC(NCCCCCC(=O)N4CCN(C5=CC(N(C(=O)NCC6=CC=CC=C6)[C@H]6CC[C@@H](NC7=NC=C8C=CC=CC8=N7)CC6)=CC=C5)CC4)=C3C2=O)C(=O)N1	C51H56N10O6	CDK12;KIAA1791	Q9NYV4/Q14004	CRBN	WO-2024175065-A1
TPD-WLBS6X	WO2024175065A1_YJZ9058	.	O=C(COC1=C2C(=O)N(C3CCC(=O)NC3=O)C(=O)C2=CC=C1)NCCCCCCCN1CCN(C2=CC(N(C(=O)NCC3=CCCC=C3)[C@H]3CC[C@@H](NC4=NC=C5C=CC=CC5=N4)CC3)=CC=C2)CC1	C54H64N10O7	CDK12;KIAA1791	Q9NYV4/Q14004	CRBN	WO-2024175065-A1
TPD-JQU9M7	WO2024175065A1_YJZ9059	.	O=C1CCC(N2C(=O)C3=CC=CC(NCCCC(=O)NC4=CC(N(C(=O)NCC5=CC=CC=C5)[C@H]5CC[C@@H](NC6=NC=C7C=CC=CC7=N6)CC5)=CC=C4)=C3C2=O)C(=O)N1	C45H45N9O6	CDK12;KIAA1791	Q9NYV4/Q14004	CRBN	WO-2024175065-A1
TPD-BA6GFB	WO2024175065A1_YJZ9062	.	O=C1CCC(N2C(=O)C3=C(C2=O)C(NCCCCCCCCCC(=O)N2CCN(C4=CC(N(C(=O)NCC5=CC=CC=C5)[C@H]5CC[C@@H](NC6=NC=C7C=CC=CC7=N6)CC5)=CC=C4)CC2)=CC=C3)C(=O)N1	C55H64N10O6	CDK12;KIAA1791	Q9NYV4/Q14004	CRBN	WO-2024175065-A1
TPD-KR4S2E	WO2024175065A1_YJZ9069	.	O=C1CCC(N2C(=O)C3=CC=CC(OCC(=O)N4CCN(C5=CC=C(N(C(=O)NCC6=CC=CC=C6)[C@H]6CC[C@@H](NC7=NC=C8C=CC=CC8=N7)CC6)C=C5)CC4)=C3C2=O)C(=O)N1	C47H47N9O7	CDK12;KIAA1791	Q9NYV4/Q14004	CRBN	WO-2024175065-A1
TPD-GRE7DX	WO2024175065A1_YJZ9108	.	CN1C(=O)CCC(N2C(=O)C3=CC=CC(OCC(=O)N4CCN(C5=CC=C(N(C(=O)NCC6=CC=CC=C6)[C@H]6CC[C@H](NC7=NC=C8C=CC=CC8=N7)CC6)C=C5)CC4)=C3C2=O)C1=O	C48H49N9O7	CDK12;KIAA1791	Q9NYV4/Q14004	CRBN	WO-2024175065-A1
TPD-IV0TDA	WO2024175065A1_ZLC4-77	.	N#CC1=CC=C(N[C@H]2CC[C@@H](N(C(=O)NCC3=CCCC=C3)C3=CC=C(N4CCN(CC5CCN(C6=CC7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7C=C6)CC5)CC4)C=C3)CC2)N=C1	C49H58N10O5	CDK12;KIAA1791	Q9NYV4/Q14004	CRBN	WO-2024175065-A1
TPD-PT3UQE	WO2024175065A1_ZLC4-79	.	N#CC1=CC=C(N[C@H]2CC[C@@H](N(C(=O)NCC3=CC=CC=C3)C3=CC=C(N4CCN(C(=O)C5CN(C6=CC7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7C=C6)C5)CC4)C=C3)CC2)N=C1	C47H50N10O6	CDK12;KIAA1791	Q9NYV4/Q14004	CRBN	WO-2024175065-A1
TPD-YWZTVN	WO2024175065A1_ZLC4-91	.	N#CC1=CC=C(NC2CCC(N(C(=O)NCC3=CC=CC=C3)C3=CC=C(N4CC5CN(CC6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)CC5C4)C=C3)CC2)N=C1	C51H56N10O5	CDK12;KIAA1791	Q9NYV4/Q14004	CRBN	WO-2024175065-A1
TPD-9WI5CT	WO2024175065A1_ZLC5-104	.	N#CC1=CN=C(N[C@H]2CC[C@@H](N(C(=O)NCC3=CC=CC=C3)C3=CC=C(N4CCC(CN5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C=C3)CC2)C=C1	C49H54N10O5	CDK12;KIAA1791	Q9NYV4/Q14004	CRBN	WO-2024175065-A1
TPD-R1DMKQ	WO2024175065A1_ZLC5-106	.	N#CC1=CN=C(N[C@H]2CC[C@H](N(C(=O)NCC3=CC=CC=C3)C3=CC=C(N4CCC5(CC4)CN(C4=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C4)C5)C=C3)CC2)C=C1	C46H47N9O5	CDK12;KIAA1791	Q9NYV4/Q14004	CRBN	WO-2024175065-A1
TPD-NQD83I	WO2024175065A1_ZLC5-11	.	N#CC1=CN=C(N[C@H]2CC[C@H](N(C(=O)NCC3=CC=CC=C3)C3=CC=C(N4CCN(C[C@H]5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C3)CC2)C=C1	C48H52N10O5	CDK12;KIAA1791	Q9NYV4/Q14004	CRBN	WO-2024175065-A1
TPD-6VXCT1	WO2024175065A1_ZLC5-15	.	N#CC1=CN=C(N[C@H]2CC[C@@H](N(C(=O)NCC3=CC=CC=C3)C3=CC=C(N4CC(CN5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)C4)C=C3)CC2)C=C1	C47H50N10O5	CDK12;KIAA1791	Q9NYV4/Q14004	CRBN	WO-2024175065-A1
TPD-SAAUHB	WO2024175065A1_ZLC5-20	.	N#CC1=CN=C(N[C@H]2CC[C@@H](N(C(=O)NCC3=CC=CC=C3)C3=CC=C(N4CCC(CN5CC6(C5)CN(C5=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C5)C6)CC4)C=C3)CC2)C=C1	C50H54N10O5	CDK12;KIAA1791	Q9NYV4/Q14004	CRBN	WO-2024175065-A1
TPD-2S8TZ8	WO2024175065A1_ZLC5-31	.	N#CC1=CN=C(N[C@H]2CC[C@@H](N(C(=O)NCC3=CC=CC=C3)C3=CC=C(N4CCN(CC#CC5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)C=C3)CC2)C=C1	C46H45N9O5	CDK12;KIAA1791	Q9NYV4/Q14004	CRBN	WO-2024175065-A1
TPD-R7OEZS	WO2024175065A1_ZLC5-6	.	N#CC1=CN=C(N[C@H]2CC[C@H](N(C(=O)NCC3=CC=CC=C3)C3=CC=C(N4CCN(C[C@@H]5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C3)CC2)C=C1	C48H52N10O5	CDK12;KIAA1791	Q9NYV4/Q14004	CRBN	WO-2024175065-A1
TPD-E6MPB3	3053716-46-1	3-Benzyl-1-[4-[(5-cyanopyridin-2-yl)amino]cyclohexyl]-1-[4-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperazin-1-yl]phenyl]urea; orb2695456; EX-A12409E; 3-BENZYL-1-(TRANS-4-((5-CYANOPYRIDIN-2-YL)AMINO)CYCL OHEXYL)-1-(4-(4-(1-(2-(2,6-DIOXOPIPERIDIN-3-YL)-6-FLUORO -1,3-DIOXOISOINDOLIN-5-YL)PIPERIDIN-4-YL)PIPERAZIN	N#CC1=CC=C(N[C@H]2CC[C@@H](N(C(=O)NCC3=CC=CC=C3)C3=CC=C(N4CCN(C5CCN(C6=C(F)C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C=C3)CC2)N=C1	C48H51FN10O5	CDK12;KIAA1791	Q9NYV4/Q14004	CRBN	WO-2024175065-A1
TPD-O1APV8	WO2024175065A1_ZLC6-101	.	N#CC1=CCC(N[C@H]2CC[C@@H](N(C(=O)NCC3=CCCC=C3)C3C=CC(N4CCN(C5CN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)=CC3)CC2)N=C1	C46H54N10O5	CDK12;KIAA1791	Q9NYV4/Q14004	CRBN	WO-2024175065-A1
TPD-7AWJY3	WO2024175065A1_ZLC6-102	.	N#CC1=CN=C(N[C@H]2CC[C@H](N(C(=O)NCC3=CC=CC=C3)C3=CC=C(N4CCN(C5CCN(C6=CC7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7C=C6)C5)CC4)C=C3)CC2)C=C1	C47H52N10O5	CDK12;KIAA1791	Q9NYV4/Q14004	CRBN	WO-2024175065-A1
TPD-KWNQH3	WO2024175065A1_ZLC6-103	.	N#CC1=CC=C(N[C@H]2CC[C@@H](N(C(=O)NCC3=CC=CC=C3)C3=CC=C(N4CCN(C(=O)C5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C=C3)CC2)N=C1	C49H52N10O6	CDK12;KIAA1791	Q9NYV4/Q14004	CRBN	WO-2024175065-A1
TPD-JB8FB8	WO2024175065A1_ZLC6-35	.	N#CC1=CC=C(N[C@H]2CC[C@H](N(C(=O)NCC3=CC=CC=C3)C3=CC=C(N4CCN(CC5CN(C6=C(F)C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C3)CC2)N=C1	C47H49FN10O5	CDK12;KIAA1791	Q9NYV4/Q14004	CRBN	WO-2024175065-A1
TPD-LH0Z8J	WO2024175065A1_ZLC6-38	.	N#CC1=CC=C(N[C@H]2CC[C@@H](N(C(=O)NCC3=CC=CC=C3)C3=CC=C(N4CCN(CC5CN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)C=C3)CC2)N=C1	C47H50N10O5	CDK12;KIAA1791	Q9NYV4/Q14004	CRBN	WO-2024175065-A1
TPD-7KO2B3	WO2024175065A1_ZLC6-42	.	N#CC1=CC=C(N[C@H]2CC[C@H](N(C(=O)NCC3=CC=CC=C3)C3=CC=C(N4CCC(N5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)C=C3)CC2)N=C1	C48H52N10O5	CDK12;KIAA1791	Q9NYV4/Q14004	CRBN	WO-2024175065-A1
TPD-CJ0941	WO2024175065A1_ZLC7-36	.	N#CC1=CN=C(NC2CCC(N(C(=O)NCC3=CC=CC=C3)C3=CC=C(N4CC(N5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)C4)C=C3)CC2)C=C1	C46H48N10O5	CDK12;KIAA1791	Q9NYV4/Q14004	CRBN	WO-2024175065-A1
TPD-ZHBLOB	WO2024178067A9_D08	.	CCCc1cc(NC2CC[C@@H](NC(=O)c3ccc(-c4ccc(CNc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6=O)cc4)cc3)C2)n2nccc2n1	C41H40N8O5	CDK9	P50750	CRBN	WO-2024178067-A9
TPD-WFTBAC	WO2024178067A9_D19	.	CCCc1cc(NC2CC[C@@H](NC(=O)c3ccc(-c4ccc(COc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6=O)cc4)cc3)C2)n2nccc2n1	C41H39N7O6	CDK9	P50750	CRBN	WO-2024178067-A9
TPD-E4BV8N	WO2024178067A9_D20	.	CCCc1cc(NC2CC[C@@H](NC(=O)c3ccc(-c4ccc(CNc5cccc6c5CN(C5CCC(=O)NC5=O)C6=O)cc4)cc3)C2)n2nccc2n1	C41H42N8O4	CDK9	P50750	CRBN	WO-2024178067-A9
TPD-SBJSNU	WO2024178067A9_D21	.	CCCc1cc(NC2CC[C@@H](NC(=O)c3ccc(N4CCC(CNc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)cc3)C2)n2nccc2n1	C40H45N9O5	CDK9	P50750	CRBN	WO-2024178067-A9
TPD-PEYRV9	WO2024178067A9_D22	.	CCCc1cc(NC2CC[C@@H](NC(=O)c3ccc(-c4ccc(CNc5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)cc4)cc3)C2)n2nccc2n1	C41H40N8O5	CDK9	P50750	CRBN	WO-2024178067-A9
TPD-5T9RB8	WO2024178067A9_D23	.	CCCc1cc(NC2CC[C@@H](NC(=O)c3ccc(N4CCC(COc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)cc3)C2)n2nccc2n1	C40H44N8O6	CDK9	P50750	CRBN	WO-2024178067-A9
TPD-XAG96S	WO2024178067A9_D24	.	CCCc1cc(NC2CC[C@@H](NC(=O)c3ccc(N4CCC(CNc5cccc6c5CN(C5CCC(=O)NC5=O)C6=O)CC4)cc3)C2)n2nccc2n1	C40H47N9O4	CDK9	P50750	CRBN	WO-2024178067-A9
TPD-DCV1UR	WO2024178067A9_D25	.	CCCc1cc(NC2CC[C@@H](NC(=O)c3ccc(CN4CCN(c5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)cc3)C2)n2nccc2n1	C39H43N9O5	CDK9	P50750	CRBN	WO-2024178067-A9
TPD-94OKU3	WO2024178067A9_D26	.	CCCc1cc(NC2CC[C@@H](NC(=O)c3ccc(CCN4CCN(c5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)cc3)C2)n2nccc2n1	C40H45N9O5	CDK9	P50750	CRBN	WO-2024178067-A9
TPD-RZVQJF	WO2024178067A9_D27	.	CCCc1cc(NC2CC[C@@H](NC(=O)C3CCN(c4ccc(CNc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6=O)cc4)CC3)C2)n2nccc2n1	C40H45N9O5	CDK9	P50750	CRBN	WO-2024178067-A9
TPD-64I6K3	WO2024178067A9_D28	.	CCCc1cc(NC2CC[C@@H](NC(=O)c3ccc(N4CCC(C#Cc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)cc3)C2)n2nccc2n1	C41H42N8O5	CDK9	P50750	CRBN	WO-2024178067-A9
TPD-ZJ7LBW	WO2024178067A9_D29	.	CCCc1cc(NC2CC[C@@H](NC(=O)c3ccc(N4CCC(CNc5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)cc3)C2)n2nccc2n1	C40H45N9O5	CDK9	P50750	CRBN	WO-2024178067-A9
TPD-HW0RA6	WO2024178067A9_D30	.	CCCc1cc(NC2CC[C@@H](NC(=O)c3ccc(N4CCC(CCc5cccc6c5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)cc3)C2)n2nccc2n1	C41H46N8O5	CDK9	P50750	CRBN	WO-2024178067-A9
TPD-EGREEY	WO2024178067A9_D32	.	CCCc1cc(NC2CC[C@@H](NC(=O)c3ccc(CN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)cc3)C2)n2nccc2n1	C39H45N9O4	CDK9	P50750	CRBN	WO-2024178067-A9
TPD-JCOCNF	WO2024178067A9_D33	.	CCCc1cc(NC2CC[C@@H](NC(=O)c3ccc(CN4CCN(c5ccc6c(c5)CN(C5CCC(=O)N(C)C5=O)C6=O)CC4)cc3)C2)n2nccc2n1	C40H47N9O4	CDK9	P50750	CRBN	WO-2024178067-A9
TPD-DPQ82D	WO2024179529A1_H-1	.	Cc1ncsc1-c1ccc(CNC(=O)C2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCN(c3ccc4c(c3)CCC43CCN(c4cc(-c5ccccc5O)nnc4N)CC3)CC2)C(C)(C)C)cc1	C51H61N9O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-60M6Z0	WO2024179529A1_H-10	.	Cc1csc(Nc2ccc(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3CCN(c4ccc5c(c4)CCC54CCN(c5cc(-c6ccccc6O)nnc5N)CC4)CC3)C(C)(C)C)cn2)n1	C50H61N11O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-2MZ9CA	WO2024179529A1_H-100	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCNc2ccc3c(c2)CCC32CCN(c3cc(-c4ccccc4O)nnc3N)CC2)C(C)C)cc1	C50H61N9O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-9K1LMF	WO2024179529A1_H-101	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)N2CC3(CCN(c4ccc5c(c4)CCC54CCN(c5cc(-c6ccccc6O)nnc5N)CC4)CC3)C2)C(C)(C)C)cc1	C54H66N10O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-LTTU2Y	WO2024179529A1_H-102	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)N2CCC3(CC2)CCN(c2ccc4c(c2)CCC42CCN(c4cc(-c5ccccc5O)nnc4N)CC2)CC3)C(C)(C)C)cc1	C56H70N10O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-O2UF7C	WO2024179529A1_H-103	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCN(c3ccc4c(c3)C3(CCN(c5cc(-c6ccccc6O)nnc5N)CC3)CN4)CC2)C(C)(C)C)cc1	C51H62N10O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-PGY2XX	WO2024179529A1_H-104	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)N2CCC(c3ccc4c(c3)N(C)CC43CCN(c4cc(-c5ccccc5O)nnc4N)CC3)CC2)C(C)(C)C)cc1	C52H64N10O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-T9Z8DJ	WO2024179529A1_H-105-1,H-105-2	.	Cc1ncsc1-c1ccc(C(CCC(=O)N2CCC(N3CCN(c4ccc5c(c4)N(C)CC54CCN(c5cc(-c6ccccc6O)nnc5N)CC4)CC3)CC2)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)C)cc1	C61H77FN12O6S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-127W1V	WO2024179529A1_H-106	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)C(c2cc(N3CCC(C(=O)N4CCC(CN5CC(Nc6ccc7c(c6)C6(CC7)CCN(c7cc(-c8ccccc8O)nnc7N)CC6)C5)CC4)CC3)no2)C(C)C)cc1	C63H78N12O6S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-PO3GDJ	WO2024179529A1_H-107	.	Cc1ccccc1-c1cc(N2CCC3(CC2)CN(C)c2cc(C4CCN(C5CN(C(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)NCc6ccc(-c7scnc7C)cc6)C(C)(C)C)C5)CC4)ccc23)c(N)nn1	C55H69N11O4S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-LXUNFJ	WO2024179529A1_H-108	.	CCN1CC2(CCN(c3cc(-c4ccccc4O)nnc3N)CC2)c2ccc(N3CCC(C(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)N[C@@H](C)c4ccc(-c5scnc5C)cc4)C(C)(C)C)CC3)cc21	C53H66N10O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-C2EPFS	WO2024179529A1_H-109	.	CC(=O)N1CC2(CCN(c3cc(-c4ccccc4O)nnc3N)CC2)c2ccc(N3CCC(C(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)N[C@@H](C)c4ccc(-c5nc(C)cs5)cc4)C(C)(C)C)CC3)cc21	C53H64N10O6S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-908Y1W	WO2024179529A1_H-11	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)C(c2cc(N3CCC(CN4CCC(N5CCC(Cc6ccc7c(c6)C6(CC7)CCN(c7cc(-c8ccccc8O)nnc7N)CC6)CC5)CC4)CC3)no2)C(C)C)cc1	C65H83N11O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-0G9RQ7	WO2024179529A1_H-110	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)N2CCN(c3ccc4c(c3)N(C)CC43CCN(c4cc(-c5ccccc5O)nnc4N)CC3)CC2)C(C)(C)C)cc1	C51H63N11O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-SSK2N5	WO2024179529A1_H-111	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCN(c3ccc4c(n3)CCC43CCN(c4cc(-c5ccccc5O)nnc4N)CC3)CC2)C(C)(C)C)cc1	C51H62N10O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-LSS9TS	WO2024179529A1_H-112	.	Cc1csc(Nc2ccc([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3CCN(c4ccc5c(c4)N(C)CC54CCN(c5cc(-c6ccccc6O)nnc5N)CC4)CC3)C(C)(C)C)cc2)n1	C52H65N11O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-VW3MHT	WO2024179529A1_H-113	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCN2CCN(c3ccc4c(c3)N(C)CC43CCN(c4cc(-c5ccccc5O)nnc4N)CC3)CC2)C(C)(C)C)cc1	C54H69N11O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-7BTO7B	WO2024179529A1_H-114	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)C2C[C@@H](O)CN2C(=O)C(c2cc(N3CCC(OC4CCN(C[C@H]5C[C@H](Oc6ccc7c(c6)C6(CCN(c8cc(-c9ccccc9O)nnc8N)CC6)CO7)C5)CC4)CC3)no2)C(C)C)cc1	C62H76N10O8S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-XNCWAT	WO2024179529A1_H-115	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCN(CC3CCN(C4CCN(Cc5ccc6c(c5)CCC65CCN(c6cc(-c7ccccc7O)nnc6N)CC5)CC4)CC3)CC2)C(C)(C)C)cc1	C64H85N11O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-N42HLN	WO2024179529A1_H-116	.	CCCN1CC2(CCN(c3cc(-c4ccccc4O)nnc3N)CC2)c2ccc(N3CCC(C(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)N[C@@H](C)c4ccc(-c5scnc5C)cc4)C(C)(C)C)CC3)cc21	C54H68N10O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-308UO9	WO2024179529A1_H-117	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCN(c3ccc4c(c3)N(C(C)C)CC43CCN(c4cc(-c5ccccc5O)nnc4N)CC3)CC2)C(C)(C)C)cc1	C54H68N10O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-A4X07E	WO2024179529A1_H-118	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCN(c3ccc4c(c3)N(C)CC43CCN(c4cc(-c5ccccc5O)nnc4N)CC3)CC2)C(C)C)cc1	C51H62N10O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-D1Z2H8	WO2024179529A1_H-119	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCN(c3ccc4c(c3)CCC43CN(c4cc(-c5ccccc5O)nnc4N)C3)CC2)C(C)(C)C)cc1	C49H57N9O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-IPZHXC	WO2024179529A1_H-12	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)C(c2cc(N3CCC(OC4CCN(C(=O)[C@H]5C[C@H](Oc6ccc7c(c6)C6(CC7)CCN(c7cc(-c8ccccc8O)nnc7N)CC6)C5)CC4)CC3)no2)C(C)C)cc1	C63H76N10O8S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-6HW2C6	WO2024179529A1_H-120	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCN(c3ccc4c(c3)CCC43CCN(c4cc(-c5ccccc5O)nnc4N)C3)CC2)C(C)(C)C)cc1	C51H61N9O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-XSDBKS	WO2024179529A1_H-122	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCN(c3ccc4c(c3)CCC43CN(c4cc(-c5ccccc5O)nnc4N)C3)CC2)C(C)C)cc1	C49H57N9O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-QMZD2K	WO2024179529A1_H-123	.	CC[C@@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](NC(=O)C1CCN(c2ccc3c(c2)N(C)CC32CCN(c3cc(-c4ccccc4O)nnc3N)CC2)CC1)C(C)(C)C)c1ccc(-c2scnc2C)cc1	C53H66N10O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-9VWGU2	WO2024179529A1_H-124	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)C2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)c2ccc(-c3ccc4c(c3)CCC43CN(c4cc(-c5ccccc5O)nnc4N)C3)cc2)C(C)(C)C)cc1	C51H54N8O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-QB16A8	WO2024179529A1_H-125	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCN(c3ccc4c(n3)NCC43CCN(c4cc(-c5ccccc5O)nnc4N)CC3)CC2)C(C)C)cc1	C49H59N11O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-PIV3F1	WO2024179529A1_H-126	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCN(c3ccc4c(c3)NCC43CN(c4cc(-c5ccccc5O)nnc4N)C3)CC2)C(C)(C)C)cc1	C49H58N10O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-FN6HTR	WO2024179529A1_H-127	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCC(c3ccc4c(c3)CCC43CN(c4cc(-c5ccccc5O)nnc4N)C3)CC2)C(C)C)cc1	C50H58N8O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-9M0I9K	WO2024179529A1_H-128	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)C(c2cc(N3CCC(c4ccc5c(c4)CCC54CN(c5cc(-c6ccccc6O)nnc5N)C4)CC3)no2)C(C)C)cc1	C51H57N9O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-HF3D1B	WO2024179529A1_H-129	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)N2CC(N3CCC(c4ccc5c(c4)CCC54CN(c5cc(-c6ccccc6O)nnc5N)C4)CC3)C2)C(C)(C)C)cc1	C53H64N10O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-HSOOTC	WO2024179529A1_H-13	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)C(NC(=O)C2CCC(c3ccc4c(c3)CCC43CCN(c4cc(-c5ccccc5O)nnc4N)CC3)CC2)C(C)(C)C)cc1	C52H62N8O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-6CRFAK	WO2024179529A1_H-130	.	Cc1ncsc1-c1ccc([C@H](O)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CC3(C2)CN(c2ccc4c(n2)N(C)CC42CCN(c4cc(-c5ccccc5O)nnc4N)CC2)C3)C(C)(C)C)cc1	C51H61N11O6S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-EDP7ZW	WO2024179529A1_H-131	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CC3(C2)CN(c2ccc4c(n2)N(C)CC42CCN(c4cc(-c5ccccc5O)nnc4N)CC2)C3)C(C)C)cc1	C51H61N11O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-PKDTLN	WO2024179529A1_H-132	.	Cc1ccccc1-c1cc(N2CC3(CCc4cc(N5CCC6(CC5)CC(C(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)c5ccc(-c7scnc7C)cc5)C(C)(C)C)C6)ccc43)C2)c(N)nn1	C54H65N9O4S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-VQ194E	WO2024179529A1_H-133	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCC(Nc3ccc4c(c3)CCC43CN(c4cc(-c5ccccc5O)nnc4N)C3)CC2)C(C)(C)C)cc1	C51H61N9O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-PS27VP	WO2024179529A1_H-134-1,H-134-2	.	Cc1ncsc1-c1ccc(C(CCC(=O)N2CCC(N3CCC(c4ccc5c(c4)CCC54CN(c5cc(-c6ccccc6O)nnc5N)C4)CC3)CC2)NC(=O)C2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)C)cc1	C60H73FN10O6S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-3RGSOT	WO2024179529A1_H-135-1,H-135-2	.	Cc1ncsc1-c1ccc(C(CCC(=O)N2CCC(c3ccc4c(c3)CCC43CN(c4cc(-c5ccccc5O)nnc4N)C3)CC2)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)C)cc1	C55H64FN9O6S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-3IJFOZ	WO2024179529A1_H-136	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)C)c(OCCNC(=O)C2CCN(c3ccc4c(c3)CCC43CN(c4cc(-c5ccccc5O)nnc4N)C3)CC2)c1	C56H67FN10O7S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-V8A8Q1	WO2024179529A1_H-137	.	Cc1ncsc1-c1ccc(C(CCC(=O)N2CCC(N3CCC(c4ccc5c(c4)N(C)CC54CN(c5cc(-c6ccccc6O)nnc5N)C4)CC3)CC2)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)C)cc1	C60H74FN11O6S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-SX8PA0	WO2024179529A1_H-138	.	Cc1ncsc1-c1ccc(C2CCCN2C(=O)C2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCN(c3ccc4c(c3)CCC43CN(c4cc(-c5ccccc5O)nnc4N)C3)CC2)C(C)(C)C)cc1	C52H61N9O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-J65UL3	WO2024179529A1_H-139	.	CCN1CC2(CN(c3cc(-c4ccccc4O)nnc3N)C2)c2ccc(N3CCC(C(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)N[C@@H](C)c4ccc(-c5scnc5C)cc4)C(C)(C)C)CC3)cc21	C51H62N10O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-6YCESO	WO2024179529A1_H-14-1	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCC(N3CCC(c4ccc5c(c4)CCC54CCN(c5cc(-c6ccccc6O)nnc5N)CC4)CC3)CC2)C(C)(C)C)cc1	C57H71N9O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-N4UCLC	WO2024179529A1_H-14-2	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)[C@H]2CC[C@H](N3CCC(c4ccc5c(c4)CCC54CCN(c5cc(-c6ccccc6O)nnc5N)CC4)CC3)CC2)C(C)(C)C)cc1	C57H71N9O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-RWJ0JU	WO2024179529A1_H-141	.	Cc1nc(N)sc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCN(c3ccc4c(c3)N(C)CC43CCN(c4cc(-c5ccccc5O)nnc4N)CC3)CC2)C(C)(C)C)cc1	C52H65N11O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-Z3QOQE	WO2024179529A1_H-142-1,H-142-2	.	Cc1ncsc1-c1ccc(C(CCC(=O)N2CCC(N3CCC(c4ccc5c(c4)N(C)CC54CCN(c5cc(-c6ccccc6O)nnc5N)CC4)CC3)CC2)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)C)cc1	C62H78FN11O6S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-GI46PV	WO2024179529A1_H-144-1,H-144-2	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCC(Nc3ccc4c(c3)NCC43CCN(c4cc(-c5ccccc5O)nnc4N)CC3)CC2)C(C)(C)C)cc1	C52H64N10O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-GIA88D	WO2024179529A1_H-146	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCN(c3ccc4c(c3)NC(=O)C43CCN(c4cc(-c5ccccc5O)nnc4N)CC3)CC2)C(C)C)cc1	C50H58N10O6S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-SA3BYJ	WO2024179529A1_H-147	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)C(c2cc(N3CCC(OC4CCN(C(=O)[C@H]5C[C@H](Nc6ccc7c(c6)C6(CCN(c8cc(-c9ccccc9O)nnc8N)CC6)CN7C)C5)CC4)CC3)no2)C(C)C)cc1	C63H78N12O7S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-4SR26N	WO2024179529A1_H-149	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCN(c3ccc4c(c3)C(=O)NC43CCN(c4cc(-c5ccccc5O)nnc4N)CC3)CC2)C(C)(C)C)cc1	C50H58N10O6S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-A0P8YH	WO2024179529A1_H-15	.	Cc1ncsc1-c1ccc(CNC(=O)C2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCN(Cc3ccc4c(c3)CCC43CCN(c4cc(-c5ccccc5O)nnc4N)CC3)CC2)C(C)(C)C)cc1	C52H63N9O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-LNUCM2	WO2024179529A1_H-151	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CC3CCC(C2)N3c2ccc3c(c2)CCC32CCN(c3cc(-c4ccccc4O)nnc3N)CC2)C(C)(C)C)cc1	C53H63N9O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-W9GJ9N	WO2024179529A1_H-152	.	Cc1csc(Nc2ccc(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3CCN(c4ccc5c(c4)N(C)CC54CCN(c5cc(-c6ccccc6O)nnc5N)CC4)CC3)C(C)(C)C)cn2)n1	C50H62N12O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-T6BZ8P	WO2024179529A1_H-153	.	Cc1ncsc1-c1ccc(C(C)(C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCN(c3ccc4c(c3)N(C)CC43CCN(c4cc(-c5ccccc5O)nnc4N)CC3)CC2)C(C)(C)C)cc1	C53H66N10O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-S3TFZS	WO2024179529A1_H-154	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCN(c3ccc4c(c3)NCC43CCN(c4cc(-c5ccccc5O)nnc4N)CC3)CC2)C(C)(C)C)cc1	C50H60N10O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-U4X8TX	WO2024179529A1_H-155	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCN(c3ccc4c(c3)CNC43CCN(c4cc(-c5ccccc5O)nnc4N)CC3)CC2)C(C)(C)C)cc1	C50H60N10O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-QH8LVQ	WO2024179529A1_H-157	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)C(c2cc(OCCOCCOc3ccc4c(c3)CCC43CCN(c4cc(-c5ccccc5O)nnc4N)CC3)no2)C(C)C)cc1	C52H60N8O8S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-X9BH4S	WO2024179529A1_H-158	.	Cc1ncsc1-c1ccc(C2CCCN2C(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCN(c3ccc4c(c3)N(C)CC43CCN(c4cc(-c5ccccc5O)nnc4N)CC3)CC2)C(C)(C)C)cc1	C54H66N10O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-XCZUUR	WO2024179529A1_H-159	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCN(c3ccc4c(c3)N(C)CC43CN(c4cc(-c5ccccc5O)nnc4N)C3)CC2)C(C)(C)C)cc1	C49H58N10O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-1LZY60	WO2024179529A1_H-16	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)C2C[C@@H](O)CN2C(=O)C(c2cc(OCCCN3CCC(O[C@H]4C[C@H](Oc5ccc6c(c5)C5(CC6)CCN(c6cc(-c7ccccc7O)nnc6N)CC5)C4)CC3)no2)C(C)C)cc1	C60H73N9O8S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-5ZZ43A	WO2024179529A1_H-160	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCN(c3ccc4c(n3)N(C)CC43CCN(c4cc(-c5ccccc5O)nnc4N)CC3)CC2)C(C)(C)C)cc1	C51H63N11O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-FM45P1	WO2024179529A1_H-161	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCN(c3ccc4c(c3)CCC43CN(c4cc(-c5ccccc5O)nnc4N)C3)CC2)C(C)C)cc1	C48H55N9O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-XJIGJ6	WO2024179529A1_H-162	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCN(c3ccc4c(c3)N(C)CC43CN(c4cc(-c5ccccc5O)nnc4N)C3)CC2)C(C)(C)C)cc1	C50H60N10O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-AJX1W3	WO2024179529A1_H-163	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CN(c3ccc4c(c3)CCC43CN(c4cc(-c5ccccc5O)nnc4N)C3)C2)C(C)(C)C)cc1	C48H55N9O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-1GLR47	WO2024179529A1_H-164	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](C)CN2C(=O)[C@@H](NC(=O)N2CCN(c3ccc4c(c3)CCC43CN(c4cc(-c5ccccc5O)nnc4N)C3)CC2)C(C)(C)C)cc1	C50H60N10O4S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-7Q5TYN	WO2024179529A1_H-165	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CN(C)CCNc2ccc3c(c2)CCC32CN(c3cc(-c4ccccc4O)nnc3N)C2)C(C)C)cc1	C48H58N10O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-VOK0YC	WO2024179529A1_H-166	.	Cc1ncsc1-c1ccc(C(C)(C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCN(c3ccc4c(c3)CCC43CN(c4cc(-c5ccccc5O)nnc4N)C3)CC2)C(C)(C)C)cc1	C51H61N9O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-AYTFS1	WO2024179529A1_H-167	.	Cc1ncsc1-c1ccc([C@H](NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCN(c3ccc4c(c3)N(C)CC43CCN(c4cc(-c5ccccc5O)nnc4N)CC3)CC2)C(C)(C)C)C(C)C)cc1	C54H68N10O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-QLEPDU	WO2024179529A1_H-168	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCNc2ccc3c(c2)CCC32CN(c3cc(-c4ccccc4O)nnc3N)C2)C(C)(C)C)cc1	C47H55N9O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-FVT8QE	WO2024179529A1_H-169	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCNc2ccc3c(c2)CCC32CN(c3cc(-c4ccccc4O)nnc3N)C2)C(C)(C)C)cc1	C48H57N9O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-ZC4DCA	WO2024179529A1_H-17	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)C(c2cc(OC3CCC(CNc4ccc5c(c4)CCC54CCN(c5cc(-c6ccccc6O)nnc5N)CC4)CC3)no2)C(C)C)cc1	C54H63N9O6S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-972WV5	WO2024179529A1_H-170	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCNc2ccc3c(c2)CCC32CN(c3cc(-c4ccccc4O)nnc3N)C2)C(C)(C)C)cc1	C49H59N9O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-16Y7T4	WO2024179529A1_H-171	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CC3(C2)CN(c2ccc4c(n2)N(C)CC42CCN(c4cc(-c5ccccc5O)nnc4N)CC2)C3)C(C)(C)C)cc1	C51H61N11O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-CCYBU1	WO2024179529A1_H-172	.	Cc1ncsc1-c1ccc(C(CCC(=O)N2CC3(C2)CN(c2ccc4c(c2)CCC42CN(c4cc(-c5ccccc5O)nnc4N)C2)C3)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)C)cc1	C55H63FN10O6S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-BI51G0	WO2024179529A1_H-173	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCN2CCN(c3ccc4c(c3)CCC43CN(c4cc(-c5ccccc5O)nnc4N)C3)CC2)C(C)(C)C)cc1	C52H64N10O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-D18XOQ	WO2024179529A1_H-174	.	Cc1ncsc1-c1ccc(C(CCCC(=O)N2CCC(c3ccc4c(c3)CCC43CN(c4cc(-c5ccccc5O)nnc4N)C3)CC2)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)C)cc1	C56H66FN9O6S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-A9OJRH	WO2024179529A1_H-175	.	Cc1ncsc1-c1ccc(C(CCCC(=O)N2CCC(N3CCC(c4ccc5c(c4)N(C)CC54CN(c5cc(-c6ccccc6O)nnc5N)C4)CC3)CC2)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)C)cc1	C61H76FN11O6S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-A4I56R	WO2024179529A1_H-176	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)C)c(OCCNC(=O)C2CCN(c3ccc4c(c3)N(C)CC43CN(c4cc(-c5ccccc5O)nnc4N)C3)CC2)c1	C56H68FN11O7S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-1AK9VN	WO2024179529A1_H-177	.	Cc1ncsc1-c1ccc(C(CCC(=O)N2CC3(C2)CN(c2ccc4c(c2)N(C)CC42CN(c4cc(-c5ccccc5O)nnc4N)C2)C3)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)C)cc1	C55H64FN11O6S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-K5XZQ4	WO2024179529A1_H-178	.	Cc1ncsc1-c1ccc(C(CCCC(=O)N2CCC(N3CCC(c4ccc5c(c4)CCC54CN(c5cc(-c6ccccc6O)nnc5N)C4)CC3)CC2)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)C)cc1	C61H75FN10O6S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-GB5XHV	WO2024179529A1_H-179	.	Cc1ncsc1-c1ccc2c(c1)CCC2NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](NC(=O)C1CCN(c2ccc3c(c2)CCC32CN(c3cc(-c4ccccc4O)nnc3N)C2)CC1)C(C)(C)C	C51H59N9O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-12RJJ7	WO2024179529A1_H-18	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)C(c2cc(OCCN3CCC(O[C@H]4C[C@H](Oc5ccc6c(c5)C5(CC6)CCN(c6cc(-c7ccccc7O)nnc6N)CC5)C4)CC3)no2)C(C)C)cc1	C59H71N9O8S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-H4AV9L	WO2024179529A1_H-180	.	Cc1ncsc1-c1ccc(C(CCC(=O)N2CCC(c3ccc4c(c3)N(C)CC43CN(c4cc(-c5ccccc5O)nnc4N)C3)CC2)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)C)cc1	C55H65FN10O6S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-0WNNBM	WO2024179529A1_H-181	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCN(c3ccc4c(c3)CCC43CN(c4cc(-c5cccc(F)c5O)nnc4N)C3)CC2)C(C)(C)C)cc1	C50H58FN9O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-59077R	WO2024179529A1_H-182	.	Cc1ncsc1-c1ccc([C@@H](C)NC(=O)[C@H]2C[C@H](C)CN2C(=O)[C@H](NC(=O)C2CCN(C(=O)[C@H]3C[C@H](Nc4cccc5c4C4(CC5)CCN(c5cc(-c6ccccc6O)nnc5N)CC4)C3)CC2)C(C)(C)C)cc1	C58H72N10O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-2D388L	WO2024179529A1_H-183	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCN(c3ccc4c(c3)CCC43CCN(c4cc(-c5c(O)cccc5Cl)nnc4N)CC3)CC2)C(C)(C)C)cc1	C52H62ClN9O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-7SIDM2	WO2024179529A1_H-184	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCN(C(=O)[C@H]3C[C@H](Nc4ccc5c(c4)CCC54CCN(c5cc(-c6ccccc6O)nnc5N)CC4)C3)CC2)C(C)(C)C)cc1	C57H70N10O6S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-1PBE0Z	WO2024179529A1_H-185	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCN(C(=O)[C@H]3C[C@H](Nc4cccc5c4CCC54CCN(c5cc(-c6ccccc6O)nnc5N)CC4)C3)CC2)C(C)(C)C)cc1	C57H70N10O6S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-00E926	WO2024179529A1_H-19	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)C(NC(=O)C2CCC(N3CCC(c4ccc5c(c4)CCC54CCN(c5cc(-c6ccccc6O)nnc5N)CC4)CC3)CC2)C(C)C)cc1	C56H69N9O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-XRNYLI	WO2024179529A1_H-2	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)C(c2cc(N3CCC(OC4CCN(C[C@H]5C[C@H](Oc6ccc7c(c6)C6(CC7)CCN(c7cc(-c8ccccc8O)nnc7N)CC6)C5)CC4)CC3)no2)C(C)C)cc1	C63H78N10O7S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-JLPQF1	WO2024179529A1_H-20	.	CC(C)C(C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)c1ccc(C#N)cc1)c1cc(OCC#Cc2ncc(O[C@H]3C[C@H](Oc4ccc5c(c4)C4(CC5)CCN(c5cc(-c6ccccc6O)nnc5N)CC4)C3)cn2)no1	C56H58N10O8	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-XJ5CAF	WO2024179529A1_H-21	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CN(c3ccc4c(c3)CCC43CCN(c4cc(-c5ccccc5O)nnc4N)CC3)C2)C(C)(C)C)cc1	C49H57N9O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-CRKNM1	WO2024179529A1_H-22	.	Cc1ncsc1-c1ccc(C(C)(C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCN(c3ccc4c(c3)CCC43CCN(c4cc(-c5ccccc5O)nnc4N)CC3)CC2)C(C)(C)C)cc1	C53H65N9O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-ZYV9I8	WO2024179529A1_H-23	.	Cc1ncsc1-c1ccc(C(CCC(=O)N2CCC(c3ccc4c(c3)CCC43CCN(c4cc(-c5ccccc5O)nnc4N)CC3)CC2)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)C)cc1	C57H68FN9O6S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-UUT41F	WO2024179529A1_H-24	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)C(c2cc(N3CCC(c4ccc5c(c4)CCC54CCN(c5cc(-c6ccccc6O)nnc5N)CC4)CC3)no2)C(C)C)cc1	C52H59N9O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-FXH2GZ	WO2024179529A1_H-25	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CC3(C2)CN(c2ccc4c(c2)CCC42CCN(c4cc(-c5ccccc5O)nnc4N)CC2)C3)C(C)(C)C)cc1	C52H61N9O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-50GC2F	WO2024179529A1_H-26	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)C(c2cc(N3CCC(OC4CCN(C(=O)[C@H]5C[C@H](Nc6ccc7c(c6)C6(CC7)CCN(c7cc(-c8ccccc8O)nnc7N)CC6)C5)CC4)CC3)no2)C(C)C)cc1	C63H77N11O7S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-DKGORZ	WO2024179529A1_H-27	.	Cc1n[nH]c(C)c1-c1ccc([C@H](C)NC(=O)C2C[C@@H](O)CN2C(=O)C(c2cc(OCCN3CCC(O[C@H]4C[C@H](Oc5ccc6c(c5)C5(CC6)CCN(c6cc(-c7ccccc7O)nnc6N)CC5)C4)CC3)no2)C(C)C)cc1	C60H74N10O8	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-QYT06W	WO2024179529A1_H-28	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCN(C(=O)N3CCC(Cc4ccc5c(c4)C4(CC5)CCN(c5cc(-c6ccccc6O)nnc5N)CC4)CC3)CC2)C(C)(C)C)cc1	C58H72N10O6S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-JXPRTM	WO2024179529A1_H-29	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)N2C3CCC2CN(c2ccc4c(c2)CCC42CCN(c4cc(-c5ccccc5O)nnc4N)CC2)C3)C(C)(C)C)cc1	C52H62N10O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-PZI1P7	WO2024179529A1_H-3	.	Cc1ncsc1-c1ccc(C(CCCCCN2CCC(c3ccc4c(c3)CCC43CCN(c4cc(-c5ccccc5O)nnc4N)CC3)CC2)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)C)cc1	C59H74FN9O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-E79TB9	WO2024179529A1_H-30	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCC(N3CCC(c4ccc5c(c4)C(F)(F)CC54CCN(c5cc(-c6ccccc6O)nnc5N)CC4)CC3)CC2)C(C)(C)C)cc1	C57H69F2N9O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-0HNC1U	WO2024179529A1_H-31	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)c2ccc(N3CCC(c4ccc5c(c4)CCC54CCN(c5cc(-c6ccccc6O)nnc5N)CC4)CC3)cc2)C(C)(C)C)cc1	C57H65N9O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-8HBERC	WO2024179529A1_H-32	.	Cc1ncsc1-c1ccc(CNC(=O)C2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)N2CCC(N3CCN(c4ccc5c(c4)CCC54CCN(c5cc(-c6ccccc6O)nnc5N)CC4)CC3)CC2)C(C)(C)C)cc1	C55H69N11O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-BYAKDK	WO2024179529A1_H-34	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCN2CCC(OC3CCN(C(=O)[C@H]4CCN(c5ccc6c(c5)C5(CC6)CCN(c6cc(-c7ccccc7O)nnc6N)CC5)C4)CC3)CC2)C(C)(C)C)cc1	C64H83N11O7S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-LYM1Q8	WO2024179529A1_H-35	.	Cc1ncsc1-c1ccc(CNC(=O)C2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CN2CC3CN(c4ccc5c(c4)CCC54CCN(c5cc(-c6ccccc6O)nnc5N)CC4)CC3C2)C(C)(C)C)cc1	C53H64N10O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-E9DAA7	WO2024179529A1_H-36	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(CNC3CCN(c4ccc5c(c4)CCC54CCN(c5cc(-c6ccccc6O)nnc5N)CC4)CC3)CC2)C(C)(C)C)cc1	C55H68N10O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-PM65CF	WO2024179529A1_H-37	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCN(C(=O)C3(CNc4ccc5c(c4)CCC54CCN(c5cc(-c6ccccc6O)nnc5N)CC4)CC3)CC2)C(C)(C)C)cc1	C56H68N10O6S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-7VHPGA	WO2024179529A1_H-38	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)[C@H]2CCN(C(=O)C3CCN(c4ccc5c(c4)CCC54CCN(c5cc(-c6ccccc6O)nnc5N)CC4)CC3)C2)C(C)(C)C)cc1	C56H68N10O6S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-7CXM3N	WO2024179529A1_H-39	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCN(C(=O)C3CCN(C4CCN(Cc5ccc6c(c5)CCC65CCN(c6cc(-c7ccccc7O)nnc6N)CC5)CC4)CC3)CC2)C(C)(C)C)cc1	C64H83N11O6S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-3FW1SE	WO2024179529A1_H-4	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)N2CC(N3CCC(c4ccc5c(c4)CCC54CCN(c5cc(-c6ccccc6O)nnc5N)CC4)CC3)C2)C(C)(C)C)cc1	C54H66N10O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-8OYUNT	WO2024179529A1_H-40	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(O)CCN(c3ccc4c(c3)CCC43CCN(c4cc(-c5ccccc5O)nnc4N)CC3)CC2)C(C)(C)C)cc1	C51H61N9O6S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-4XJNXW	WO2024179529A1_H-41	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)C(c2cc(N3CCC(OC4CCN(O[C@H]5C[C@H](Oc6ccc7c(c6)CCC76CCN(c7cc(-c8ccccc8O)nnc7N)CC6)C5)CC4)CC3)no2)C(C)C)cc1	C62H76N10O8S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-WBN7DR	WO2024179529A1_H-42	.	Cc1cc(-c2ccc(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3CCN(c4ccc5c(c4)CCC54CCN(c5cc(-c6ccccc6O)nnc5N)CC4)CC3)C(C)(C)C)cc2)ccn1	C53H63N9O5	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-KAH2E8	WO2024179529A1_H-43	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCN2CCC(c3ccc4c(c3)CCC43CCN(c4cc(-c5ccccc5O)nnc4N)CC3)CC2)C(C)C)cc1	C53H65N9O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-N2ELOC	WO2024179529A1_H-44	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CN2CCC(OC3CCN(C[C@H]4C[C@H](Oc5ccc6c(c5)C5(CC6)CCN(c6cc(-c7ccccc7O)nnc6N)CC5)C4)CC3)CC2)C(C)(C)C)cc1	C63H82N10O7S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-X0UQKE	WO2024179529A1_H-45-1,H-45-2	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CC(N3CCC(c4ccc5c(c4)CCC54CCN(c5cc(-c6ccccc6O)nnc5N)CC4)CC3)C2)C(C)(C)C)cc1	C55H67N9O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-GXCD3Q	WO2024179529A1_H-47	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)N2CCC(N3CCC(c4ccc5c(c4)CCC54CCN(c5cc(-c6ccccc6O)nnc5N)CC4)CC3)CC2)C(C)(C)C)cc1	C56H70N10O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-C1HJZK	WO2024179529A1_H-48	.	Cc1nccn1-c1ccc([C@H](C)NC(=O)C2C[C@@H](O)CN2C(=O)C(c2cc(OCCN3CCC(O[C@H]4C[C@H](Oc5ccc6c(c5)C5(CC6)CCN(c6cc(-c7ccccc7O)nnc6N)CC5)C4)CC3)no2)C(C)C)cn1	C58H71N11O8	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-44DTFK	WO2024179529A1_H-49	.	CC(C)c1ncsc1-c1ccc(CNC(=O)C2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCC(N3CCC(c4ccc5c(c4)CCC54CCN(c5cc(-c6ccccc6O)nnc5N)CC4)CC3)CC2)C(C)(C)C)cc1	C59H75N9O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-N0W3YH	WO2024179529A1_H-5	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)C(c2cc(N3CCN(CCN4CCC(O[C@H]5C[C@H](Oc6ccc7c(c6)C6(CC7)CCN(c7cc(-c8ccccc8O)nnc7N)CC6)C5)CC4)CC3)no2)C(C)C)cc1	C63H79N11O7S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-0MSP4H	WO2024179529A1_H-50	.	Cc1ncsc1-c1ccc(C(CCC(=O)N2CCC(c3ccc4c(c3)C3(CC4)CCN(c4cc(-c5ccccc5O)nnc4N)CC3)CC2)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)C)cc1	C57H68FN9O6S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-68TIAU	WO2024179529A1_H-51	.	Cc1ncsc1-c1ccc(C(CCC(=O)Nc2ccc3c(c2)CCC32CCN(c3cc(-c4ccccc4O)nnc3N)CC2)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)C)cc1	C52H60FN9O6S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-DQHVUV	WO2024179529A1_H-52	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(CNc3ccc4c(c3)CCC43CCN(c4cc(-c5ccccc5O)nnc4N)CC3)CC2)C(C)(C)C)cc1	C50H59N9O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-X6DHE3	WO2024179529A1_H-53	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)C(c2cc(OCC#Cc3ncc(O[C@H]4C[C@H](Oc5ccc6c(c5)C5(CC6)CCN(c6cc(-c7ccccc7O)nnc6N)CC5)C4)cn3)no2)C(C)C)cc1	C59H62N10O8S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-XTGWB9	WO2024179529A1_H-54	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)C2(NC(=O)C3CCN(c4ccc5c(c4)CCC54CCN(c5cc(-c6ccccc6O)nnc5N)CC4)CC3)CC2)cc1	C50H57N9O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-D5ECYD	WO2024179529A1_H-55	.	CCC(CC)(C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)c1ccc(-c2scnc2C)cc1)c1cc(N2CCC(OC3CCN(C[C@H]4C[C@H](Oc5ccc6c(c5)C5(CC6)CCN(C(/C=C(\N=N)c6ccccc6O)=C(/C)N)CC5)C4)CC3)CC2)no1	C65H84N10O7S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-FAKESI	WO2024179529A1_H-56	.	CC(C)(C)[C@H](NC(=O)C1CCN(c2ccc3c(c2)CCC32CCN(c3cc(-c4ccccc4O)nnc3N)CC2)CC1)C(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1ccc(-c2nn[nH]n2)cc1	C48H58N12O5	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-H67ENL	WO2024179529A1_H-57	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)C2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCN(CC3CCN(CC4CCN(c5ccc6c(c5)CCC65CCN(c6cc(-c7ccccc7O)nnc6N)CC5)CC4)CC3)CC2)C(C)C)cc1	C63H83N11O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-L7YN02	WO2024179529A1_H-58	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CN(C)CCNc2ccc3c(c2)CCC32CCN(c3cc(-c4ccccc4O)nnc3N)CC2)C(C)C)cc1	C50H62N10O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-08SI05	WO2024179529A1_H-59	.	Cc1csc(Nc2ccc(CNC(=O)C3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3CCN(c4ccc5c(c4)CCC54CCN(c5cc(-c6ccccc6O)nnc5N)CC4)CC3)C(C)(C)C)cc2)n1	C51H62N10O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-P3XP0B	WO2024179529A1_H-60	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCN(c3cnc4c(c3)CCC43CCN(c4cc(-c5ccccc5O)nnc4N)CC3)CC2)C(C)(C)C)cc1	C51H62N10O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-5QHNM8	WO2024179529A1_H-61	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CC3(C2)CN(c2cnc4c(c2)CCC42CCN(c4cc(-c5ccccc5O)nnc4N)CC2)C3)C(C)(C)C)cc1	C52H62N10O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-SF5NVU	WO2024179529A1_H-62	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CC3(C2)CN(c2ccc4c(n2)CCC42CCN(c4cc(-c5ccccc5O)nnc4N)CC2)C3)C(C)(C)C)cc1	C52H62N10O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-J9N6J2	WO2024179529A1_H-63	.	C/C(N)=C(\C=C(/N=N)c1ccccc1O)N1CCC2(CCc3cc(N4CC5(CC(C(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)c6ccc(-c7scnc7C)cc6)C(C)(C)C)C5)C4)ncc32)CC1	C53H66N10O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-GSW519	WO2024179529A1_H-64	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)C2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCN(c3ccc4c(c3)CCC43CN(c4cc(-c5ccccc5O)nnc4N)C3)CC2)C(C)(C)C)cc1	C50H59N9O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-66BYQ1	WO2024179529A1_H-65	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)C(c2cc(N3CCC(OC4CCN(C[C@H]5C[C@H](Oc6ccc7c(c6)C6(CCN(c8cc(-c9ccccc9O)nnc8N)CC6)C(=O)N7)C5)CC4)CC3)no2)C(C)C)cc1	C62H75N11O8S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-PCC4P3	WO2024179529A1_H-66	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCN(c3ccc4c(c3)N(C)C(=O)C43CCN(c4cc(-c5ccccc5O)nnc4N)CC3)CC2)C(C)(C)C)cc1	C52H62N10O6S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-DRJBCZ	WO2024179529A1_H-67-1,H-67-2	.	Cc1ncsc1-c1ccc(C(CCC(=O)N2CCC(N3CCN(c4ccc5c(c4)CCC54CCN(c5cc(-c6ccccc6O)nnc5N)CC4)CC3)CC2)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)C)cc1	C61H76FN11O6S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-29MOBN	WO2024179529A1_H-68-1,H-68-2	.	Cc1ncsc1-c1ccc(C(CCC(=O)N2CCC(N3CCC(c4ccc5c(c4)C4(CCN(c6cc(-c7ccccc7O)nnc6N)CC4)CN5C)CC3)CC2)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)C)cc1	C62H78FN11O6S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-FMTR83	WO2024179529A1_H-69	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCN(c3ccc4c(c3)N(C)CC43CCN(c4cc(-c5ccccc5O)nnc4N)CC3)CC2)C(C)(C)C)cc1	C52H64N10O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-A5TAJD	WO2024179529A1_H-7	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)[C@H]2CCN(Cc3ccc4c(c3)CCC43CCN(c4cc(-c5ccccc5O)nnc4N)CC3)C2)C(C)(C)C)cc1	C51H61N9O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-98CDJA	WO2024179529A1_H-70	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCN(c3ccc4c(c3)N(C)C(=O)C43CCN(c4cc(-c5ccccc5O)nnc4N)CC3)CC2)C(C)C)cc1	C51H60N10O6S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-BSEH5Y	WO2024179529A1_H-73	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCN(c3ccc4c(c3)C=CC43CCN(c4cc(-c5ccccc5O)nnc4N)CC3)CC2)C(C)(C)C)cc1	C52H61N9O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-MH8ICL	WO2024179529A1_H-74	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCN(c3ccc4c(c3)OCC43CCN(c4cc(-c5ccccc5O)nnc4N)CC3)CC2)C(C)(C)C)cc1	C51H61N9O6S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-3AIJG8	WO2024179529A1_H-75	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)C)c(OCCC2CCN(C3CCN(c4ccc5c(c4)CCC54CCN(c5cc(-c6ccccc6O)nnc5N)CC4)CC3)CC2)c1	C62H79FN10O6S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-68NNDS	WO2024179529A1_H-76	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)C(c2cc(N3CCC(CN4CCC(O[C@H]5CC[C@H](Nc6ccc7c(c6)C6(CC7)CCN(c7cc(-c8ccccc8O)nnc7N)CC6)CC5)CC4)CC3)no2)C(C)C)cc1	C65H83N11O6S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-7HM2KM	WO2024179529A1_H-77	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCN(c3cc4c(cn3)C3(CC4)CCN(c4cc(-c5ccccc5O)nnc4N)CC3)CC2)C(C)(C)C)cc1	C51H62N10O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-8ZG2G5	WO2024179529A1_H-78	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCN(c3ccc4c(c3)NS(=O)(=O)C43CCN(c4cc(-c5ccccc5O)nnc4N)CC3)CC2)C(C)(C)C)cc1	C50H60N10O7S2	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-J76Z2W	WO2024179529A1_H-79	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCN(c3ccc4c(c3)NC(=O)OC43CCN(c4cc(-c5ccccc5O)nnc4N)CC3)CC2)C(C)(C)C)cc1	C51H60N10O7S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-7TIV4S	WO2024179529A1_H-8	.	Cc1ncsc1-c1ccc(C(CCC(=O)N2CCC(N3CCC(c4ccc5c(c4)CCC54CCN(c5cc(-c6ccccc6O)nnc5N)CC4)CC3)CC2)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)C)cc1	C62H77FN10O6S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-BJF284	WO2024179529A1_H-80	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCN(c3ccc4c(c3)C(=O)NC43CCN(c4cc(-c5ccccc5O)nnc4N)CC3)CC2)C(C)(C)C)cc1	C51H60N10O6S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-4Z040H	WO2024179529A1_H-81	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)C(c2cc(N3CCC(OC4CCN(Cc5ccc6c(c5)C5(CC6)CCN(c6cc(-c7ccccc7O)nnc6N)CC5)CC4)CC3)no2)C(C)C)cc1	C59H72N10O6S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-51ABQO	WO2024179529A1_H-82	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)C)c(OCCNC(=O)C2CCN(c3ccc4c(c3)CCC43CCN(c4cc(-c5ccccc5O)nnc4N)CC3)CC2)c1	C58H71FN10O7S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-4G2H8J	WO2024179529A1_H-83	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)C(c2cc(N3CCC(OC4CCN(C[C@H]5C[C@H](Oc6ccc7c(c6)C6(CCN(c8cc(-c9ccccc9O)nnc8N)CC6)CN7)C5)CC4)CC3)no2)C(C)C)cc1	C62H77N11O7S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-6GE7PR	WO2024179529A1_H-84	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)C(c2cc(N3CCC(OC4CCN(C[C@H]5C[C@H](Oc6ccc7c(c6)C6(CCN(c8cc(-c9ccccc9O)nnc8N)CC6)CN7C)C5)CC4)CC3)no2)C(C)C)cc1	C63H79N11O7S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-HJIX61	WO2024179529A1_H-85	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)C(c2cc(N3CCC(C(=O)N4CCC(CN5CC(Oc6ccc7c(c6)C6(CC7)CCN(c7cc(-c8ccccc8O)nnc7N)CC6)C5)CC4)CC3)no2)C(C)C)cc1	C63H77N11O7S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-FYS3AZ	WO2024179529A1_H-86	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)C(c2cc(N3CCC(OC4CCN(C(=O)[C@@H]5C[C@@H](Oc6ccc7c(c6)C6(CC7)CCN(c7cc(-c8ccccc8O)nnc7N)CC6)CN5)CC4)CC3)no2)C(C)C)cc1	C63H77N11O8S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-44SAQO	WO2024179529A1_H-87	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)C(c2cc(N3CCC(CN4CCC(OCCCOc5ccc6c(c5)C5(CC6)CCN(c6cc(-c7ccccc7O)nnc6N)CC5)CC4)CC3)no2)C(C)C)cc1	C62H78N10O7S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-PNX2SL	WO2024179529A1_H-88	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)C(c2cc(N3CCC(CN4CCC(O[C@H]5C[C@H](Oc6ccc7c(c6)C6(CC7)CCN(c7cc(-c8ccccc8O)nnc7N)CC6)C5)CC4)CC3)no2)C(C)C)cc1	C63H78N10O7S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-AB3FIY	WO2024179529A1_H-89	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)C(c2cc(N3CCC(OC4CCN(C[C@H]5C[C@H](Nc6ccc7c(c6)C6(CC7)CCN(c7cc(-c8ccccc8O)nnc7N)CC6)C5)CC4)CC3)no2)C(C)C)cc1	C63H79N11O6S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-56DMYN	WO2024179529A1_H-9	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCN(c3ccc4c(c3)CCC43CCN(c4cc(-c5ccccc5O)nnc4N)CC3)CC2)C(C)(C)C)cc1	C52H63N9O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-3X4GZD	WO2024179529A1_H-90-1,H-90-2	.	Cc1ncsc1-c1ccc(C(CCC(=O)N2CCC(N3CCC(c4ccc5c(c4)C4(CC5)CCN(c5cc(-c6ccccc6O)nnc5N)CC4)CC3)CC2)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)C)cc1	C62H77FN10O6S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-MZY0HC	WO2024179529A1_H-91-1,H-91-2	.	Cc1ncsc1-c1ccc(C(CCC(=O)N2CCC(OC3CCN(c4ccc5c(c4)CCC54CCN(c5cc(-c6ccccc6O)nnc5N)CC4)CC3)CC2)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)C)cc1	C62H77FN10O7S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-VGZOQN	WO2024179529A1_H-92	.	Cc1ncsc1-c1ccc(C(CCC(=O)N2CCC(C(=O)N3CCC(c4ccc5c(c4)CCC54CCN(c5cc(-c6ccccc6O)nnc5N)CC4)CC3)CC2)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)C)cc1	C63H77FN10O7S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-IG7SJJ	WO2024179529A1_H-93	.	Cc1ncsc1-c1ccc(C(CCC(=O)N2CC(C(=O)N3CCC(N4CCC(c5ccc6c(c5)CCC65CCN(c6cc(-c7ccccc7O)nnc6N)CC5)CC4)CC3)C2)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2(F)CC2)C(C)(C)C)cc1	C66H82FN11O7S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-8N6BGB	WO2024179529A1_H-94	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)N2CCC3(CCN(c4ccc5c(c4)CCC54CCN(c5cc(-c6ccccc6O)nnc5N)CC4)CC3)C2)C(C)(C)C)cc1	C55H68N10O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-NUZ7BP	WO2024179529A1_H-95	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)C(c2cc(OCCN3CCC(C(=O)N4CC(Oc5ccc6c(c5)C5(CC6)CCN(c6cc(-c7ccccc7O)nnc6N)CC5)C4)CC3)no2)C(C)C)cc1	C59H70N10O8S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-XCH1IA	WO2024179529A1_H-96	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CC3(CCN(c4ccc5c(c4)CCC54CCN(c5cc(-c6ccccc6O)nnc5N)CC4)CC3)C2)C(C)(C)C)cc1	C55H67N9O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-S2IU4D	WO2024179529A1_H-97	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCN(c3ccc4c(c3)CCC43CCN(c4cc(-c5ccc(F)cc5O)nnc4N)CC3)CC2)C(C)(C)C)cc1	C52H62FN9O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-OL0NF0	WO2024179529A1_H-98	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)C(c2cc(N3CCC(CN4CCC(N5CC(Nc6ccc7c(c6)C6(CC7)CCN(c7cc(-c8ccccc8O)nnc7N)CC6)C5)CC4)CC3)no2)C(C)C)cc1	C62H78N12O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-K7AXTH	WO2024179529A1_H-99	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C2CCN(CC3CCN(CC4CCN(Cc5ccc6c(c5)CCC65CCN(c6cc(-c7ccccc7O)nnc6N)CC5)CC4)CC3)CC2)C(C)(C)C)cc1	C65H87N11O5S	SMARCA4	P51532	VHL	WO-2024179529-A1
TPD-KAWSGW	SCHEMBL29313748	(2S,4R)-1-[(2S)-2-[[7-[3-[(3R)-3-[4-[[4-[4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]benzoyl]sulfamoyl]-2-(trifluoromethylsulfonyl)anilino]-4-phenylsulfanylbutyl]-3,8-diazabicyclo[3.2.1]octan-8-yl]-7-oxoheptanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL30286304	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCC(=O)N3C4CCC3CN(CC[C@H](CSC3=CC=CC=C3)NC3=CC=C(S(=O)(=O)NC(=O)C5=CC=C(N6CCN(CC7=C(C8=CC=C(Cl)C=C8)CCC(C)(C)C7)CC6)C=C5)C=C3S(=O)(=O)C(F)(F)F)C4)C(C)(C)C)C=C2)SC=N1	C79H98ClF3N10O10S4	BCL2L1;BCL-2	Q07817/P10415	VHL	WO-2024179577-A1
TPD-1HKY9T	SCHEMBL29219165	(2S,4R)-1-[(2S)-2-[[7-[5-[(3R)-3-[4-[[4-[4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]benzoyl]sulfamoyl]-2-(trifluoromethylsulfonyl)anilino]-4-phenylsulfanylbutyl]-2,5-diazabicyclo[2.2.1]heptan-2-yl]-7-oxoheptanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCC(=O)N3CC4CC3CN4CC[C@H](CSC3=CC=CC=C3)NC3=CC=C(S(=O)(=O)NC(=O)C4=CC=C(N5CCN(CC6=C(C7=CC=C(Cl)C=C7)CCC(C)(C)C6)CC5)C=C4)C=C3S(=O)(=O)C(F)(F)F)C(C)(C)C)C=C2)SC=N1	C78H96ClF3N10O10S4	BCL2L1;BCL-2	Q07817/P10415	VHL	WO-2024179577-A1
TPD-BEZ147	SCHEMBL29219149	(2S,4R)-1-[(2S)-2-[[7-[4-[(3R)-3-[4-[[4-[1-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperidin-4-yl]benzoyl]sulfamoyl]-2-(trifluoromethylsulfonyl)anilino]-4-phenylsulfanylbutyl]piperazin-1-yl]-7-oxoheptanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCC(=O)N3CCN(CC[C@H](CSC4=CC=CC=C4)NC4=CC=C(S(=O)(=O)NC(=O)C5=CC=C(C6CCN(CC7=C(C8=CC=C(Cl)C=C8)CCC(C)(C)C7)CC6)C=C5)C=C4S(=O)(=O)C(F)(F)F)CC3)C(C)(C)C)C=C2)SC=N1	C78H97ClF3N9O10S4	BCL2L1;BCL-2	Q07817/P10415	VHL	WO-2024179577-A1
TPD-O40T67	SCHEMBL29313539	(2S,4R)-1-[(2S)-2-[[7-[4-[(3R)-3-[4-[[4-[4-[[2-(4-cyanophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]benzoyl]sulfamoyl]-2-(trifluoromethylsulfonyl)anilino]-4-phenylsulfanylbutyl]piperazin-1-yl]-7-oxoheptanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL30286313	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCC(=O)N3CCN(CC[C@H](CSC4=CC=CC=C4)NC4=CC=C(S(=O)(=O)NC(=O)C5=CC=C(N6CCN(CC7=C(C8=CC=C(C#N)C=C8)CCC(C)(C)C7)CC6)C=C5)C=C4S(=O)(=O)C(F)(F)F)CC3)C(C)(C)C)C=C2)SC=N1	C78H96F3N11O10S4	BCL2L1;BCL-2	Q07817/P10415	VHL	WO-2024179577-A1
TPD-1D9X6D	SCHEMBL29219135	(2S,4R)-1-[(2S)-2-[[7-[4-[(3R)-3-[4-[[4-[4-[[4-(4-chlorophenyl)-3,6-dihydro-2H-pyran-5-yl]methyl]piperazin-1-yl]benzoyl]sulfamoyl]-2-(trifluoromethylsulfonyl)anilino]-4-phenylsulfanylbutyl]piperazin-1-yl]-7-oxoheptanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCC(=O)N3CCN(CC[C@H](CSC4=CC=CC=C4)NC4=CC=C(S(=O)(=O)NC(=O)C5=CC=C(N6CCN(CC7=C(C8=CC=C(Cl)C=C8)CCOC7)CC6)C=C5)C=C4S(=O)(=O)C(F)(F)F)CC3)C(C)(C)C)C=C2)SC=N1	C74H90ClF3N10O11S4	BCL2L1;BCL-2	Q07817/P10415	VHL	WO-2024179577-A1
TPD-H3JM9I	SCHEMBL31346491	(2S,4R)-1-[(2S)-2-[[7-[4-[(3R)-3-[4-[[4-[4-[[2-(4-chlorophenyl)cyclohepten-1-yl]methyl]piperazin-1-yl]benzoyl]sulfamoyl]-2-(trifluoromethylsulfonyl)anilino]-4-phenylsulfanylbutyl]piperazin-1-yl]-7-oxoheptanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCC(=O)N3CCN(CC[C@H](CSC4=CC=CC=C4)NC4=CC=C(S(=O)(=O)NC(=O)C5=CC=C(N6CCN(CC7=C(C8=CC=C(Cl)C=C8)CCCCC7)CC6)C=C5)C=C4S(=O)(=O)C(F)(F)F)CC3)C(C)(C)C)C=C2)SC=N1	C76H94ClF3N10O10S4	BCL2L1;BCL-2	Q07817/P10415	VHL	WO-2024179577-A1
TPD-A2AVWD	SCHEMBL29219139	6-[4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[(2R)-4-[4-[7-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-7-oxoheptanoyl]piperazin-1-yl]-1-phenylsulfanylbutan-2-yl]amino]-3-(trifluoromethylsulfonyl)phenyl]sulfonylpyridine-3-carboxamide; SCHEMBL29219147	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCC(=O)N3CCN(CC[C@H](CSC4=CC=CC=C4)NC4=CC=C(S(=O)(=O)NC(=O)C5=CN=C(N6CCN(CC7=C(C8=CC=C(Cl)C=C8)CCC(C)(C)C7)CC6)C=C5)C=C4S(=O)(=O)C(F)(F)F)CC3)C(C)(C)C)C=C2)SC=N1	C76H95ClF3N11O10S4	BCL2L1;BCL-2	Q07817/P10415	VHL	WO-2024179577-A1
TPD-IWL6VC	SCHEMBL29314137	(2S,4R)-1-[(2S)-2-[[7-[(3aS,6aR)-2-[(3R)-3-[4-[[4-[4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]benzoyl]sulfamoyl]-2-(trifluoromethylsulfonyl)anilino]-4-phenylsulfanylbutyl]-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-5-yl]-7-oxoheptanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	[H][C@@]12CN(CC[C@H](CSC3=CC=CC=C3)NC3=CC=C(S(=O)(=O)NC(=O)C4=CC=C(N5CCN(CC6=C(C7=CC=C(Cl)C=C7)CCC(C)(C)C6)CC5)C=C4)C=C3S(=O)(=O)C(F)(F)F)C[C@]1([H])CN(C(=O)CCCCCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C3=C(C)N=CS3)C=C1)C(C)(C)C)C2	C79H98ClF3N10O10S4	BCL2L1;BCL-2	Q07817/P10415	VHL	WO-2024179577-A1
TPD-3NE6HJ	SCHEMBL29314366	(2S,4R)-1-[(2S)-2-[[7-[2-[(3R)-3-[4-[[4-[4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]benzoyl]sulfamoyl]-2-(trifluoromethylsulfonyl)anilino]-4-phenylsulfanylbutyl]-2,7-diazaspiro[3.5]nonan-7-yl]-7-oxoheptanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL30977249	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCC(=O)N3CCC4(CC3)CN(CC[C@H](CSC3=CC=CC=C3)NC3=CC=C(S(=O)(=O)NC(=O)C5=CC=C(N6CCN(CC7=C(C8=CC=C(Cl)C=C8)CCC(C)(C)C7)CC6)C=C5)C=C3S(=O)(=O)C(F)(F)F)C4)C(C)(C)C)C=C2)SC=N1	C80H100ClF3N10O10S4	BCL2L1;BCL-2	Q07817/P10415	VHL	WO-2024179577-A1
TPD-1F9VQT	SCHEMBL29313915	(2S,4R)-1-[(2S)-2-[[7-[(1R,4R)-5-[(3R)-3-[4-[[4-[4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]benzoyl]sulfamoyl]-2-(trifluoromethylsulfonyl)anilino]-4-phenylsulfanylbutyl]-2,5-diazabicyclo[2.2.1]heptan-2-yl]-7-oxoheptanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL30286132	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCC(=O)N3C[C@H]4C[C@@H]3CN4CC[C@H](CSC3=CC=CC=C3)NC3=CC=C(S(=O)(=O)NC(=O)C4=CC=C(N5CCN(CC6=C(C7=CC=C(Cl)C=C7)CCC(C)(C)C6)CC5)C=C4)C=C3S(=O)(=O)C(F)(F)F)C(C)(C)C)C=C2)SC=N1	C78H96ClF3N10O10S4	BCL2L1;BCL-2	Q07817/P10415	VHL	WO-2024179577-A1
TPD-E30RXY	SCHEMBL29313244	(2S,4R)-1-[(2S)-2-[[7-[4-[(3R)-3-[4-[[4-[4-[[6-(4-chlorophenyl)spiro[2.5]oct-6-en-7-yl]methyl]piperazin-1-yl]benzoyl]sulfamoyl]-2-(trifluoromethylsulfonyl)anilino]-4-phenylsulfanylbutyl]piperazin-1-yl]-7-oxoheptanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL30286275	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCC(=O)N3CCN(CC[C@H](CSC4=CC=CC=C4)NC4=CC=C(S(=O)(=O)NC(=O)C5=CC=C(N6CCN(CC7=C(C8=CC=C(Cl)C=C8)CCC8(CC8)C7)CC6)C=C5)C=C4S(=O)(=O)C(F)(F)F)CC3)C(C)(C)C)C=C2)SC=N1	C77H94ClF3N10O10S4	BCL2L1;BCL-2	Q07817/P10415	VHL	WO-2024179577-A1
TPD-SDG9UP	SCHEMBL29219105	(2S,4R)-1-[(2S)-2-[[7-[4-[(3R)-3-[4-[[4-[4-[[2-(4-chloro-2-fluorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]benzoyl]sulfamoyl]-2-(trifluoromethylsulfonyl)anilino]-4-phenylsulfanylbutyl]piperazin-1-yl]-7-oxoheptanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCC(=O)N3CCN(CC[C@H](CSC4=CC=CC=C4)NC4=CC=C(S(=O)(=O)NC(=O)C5=CC=C(N6CCN(CC7=C(C8=CC=C(Cl)C=C8F)CCC(C)(C)C7)CC6)C=C5)C=C4S(=O)(=O)C(F)(F)F)CC3)C(C)(C)C)C=C2)SC=N1	C77H95ClF4N10O10S4	BCL2L1;BCL-2	Q07817/P10415	VHL	WO-2024179577-A1
TPD-EVA7WV	SCHEMBL29313847	(2S,4R)-1-[(2S)-2-[[7-[(1S,4S)-5-[(3R)-3-[4-[[4-[4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]benzoyl]sulfamoyl]-2-(trifluoromethylsulfonyl)anilino]-4-phenylsulfanylbutyl]-2,5-diazabicyclo[2.2.1]heptan-2-yl]-7-oxoheptanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL30286226	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCC(=O)N3C[C@@H]4C[C@H]3CN4CC[C@H](CSC3=CC=CC=C3)NC3=CC=C(S(=O)(=O)NC(=O)C4=CC=C(N5CCN(CC6=C(C7=CC=C(Cl)C=C7)CCC(C)(C)C6)CC5)C=C4)C=C3S(=O)(=O)C(F)(F)F)C(C)(C)C)C=C2)SC=N1	C78H96ClF3N10O10S4	BCL2L1;BCL-2	Q07817/P10415	VHL	WO-2024179577-A1
TPD-YV9IQL	SCHEMBL29314186	(2S,4R)-1-[(2S)-2-[[7-[(3aS,6aR)-2-[(3R)-3-[4-[[4-[4-[[2-(4-chloro-2-fluorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]benzoyl]sulfamoyl]-2-(trifluoromethylsulfonyl)anilino]-4-phenylsulfanylbutyl]-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-5-yl]-7-oxoheptanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	[H][C@@]12CN(CC[C@H](CSC3=CC=CC=C3)NC3=CC=C(S(=O)(=O)NC(=O)C4=CC=C(N5CCN(CC6=C(C7=CC=C(Cl)C=C7F)CCC(C)(C)C6)CC5)C=C4)C=C3S(=O)(=O)C(F)(F)F)C[C@]1([H])CN(C(=O)CCCCCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C3=C(C)N=CS3)C=C1)C(C)(C)C)C2	C79H97ClF4N10O10S4	BCL2L1;BCL-2	Q07817/P10415	VHL	WO-2024179577-A1
TPD-7IIQAU	SCHEMBL29314276	(2S,4R)-1-[(2S)-2-[[5-[(3aR,6aS)-2-[(3R)-3-[4-[[4-[4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]benzoyl]sulfamoyl]-2-(trifluoromethylsulfonyl)anilino]-4-phenylsulfanylbutyl]-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-5-yl]-5-oxopentanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	[H][C@@]12CN(CC[C@H](CSC3=CC=CC=C3)NC3=CC=C(S(=O)(=O)NC(=O)C4=CC=C(N5CCN(CC6=C(C7=CC=C(Cl)C=C7)CCC(C)(C)C6)CC5)C=C4)C=C3S(=O)(=O)C(F)(F)F)C[C@]1([H])CN(C(=O)CCCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C3=C(C)N=CS3)C=C1)C(C)(C)C)C2	C77H94ClF3N10O10S4	BCL2L1;BCL-2	Q07817/P10415	VHL	WO-2024179577-A1
TPD-FRPPZO	SCHEMBL30977250	(2S,4R)-1-[(2S)-2-[[9-[(3aS,6aR)-2-[(3R)-3-[4-[[4-[4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]benzoyl]sulfamoyl]-2-(trifluoromethylsulfonyl)anilino]-4-phenylsulfanylbutyl]-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-5-yl]-9-oxononanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	[H][C@@]12CN(CC[C@H](CSC3=CC=CC=C3)NC3=CC=C(S(=O)(=O)NC(=O)C4=CC=C(N5CCN(CC6=C(C7=CC=C(Cl)C=C7)CCC(C)(C)C6)CC5)C=C4)C=C3S(=O)(=O)C(F)(F)F)C[C@]1([H])CN(C(=O)CCCCCCCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C3=C(C)N=CS3)C=C1)C(C)(C)C)C2	C81H102ClF3N10O10S4	BCL2L1;BCL-2	Q07817/P10415	VHL	WO-2024179577-A1
TPD-FLR7M4	SCHEMBL30977256	(2S,4R)-1-[(2S)-2-[[8-[(3aS,6aR)-2-[(3R)-3-[4-[[4-[4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]benzoyl]sulfamoyl]-2-(trifluoromethylsulfonyl)anilino]-4-phenylsulfanylbutyl]-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-5-yl]-8-oxooctanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	[H][C@@]12CN(CC[C@H](CSC3=CC=CC=C3)NC3=CC=C(S(=O)(=O)NC(=O)C4=CC=C(N5CCN(CC6=C(C7=CC=C(Cl)C=C7)CCC(C)(C)C6)CC5)C=C4)C=C3S(=O)(=O)C(F)(F)F)C[C@]1([H])CN(C(=O)CCCCCCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C3=C(C)N=CS3)C=C1)C(C)(C)C)C2	C80H100ClF3N10O10S4	BCL2L1;BCL-2	Q07817/P10415	VHL	WO-2024179577-A1
TPD-C5OHZZ	WO2024179577A1_18	(2S,4R)-1-[(2S)-2-[[7-[(3aS,6aR)-2-[(3R)-3-[4-[[4-[4-[[6-(4-chlorophenyl)spiro[2.5]oct-6-en-7-yl]methyl]piperazin-1-yl]benzoyl]sulfamoyl]-2-(trifluoromethylsulfonyl)anilino]-4-phenylsulfanylbutyl]-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-5-yl]-7-oxoheptanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	[H][C@@]12CN(CC[C@H](CSC3=CC=CC=C3)NC3=CC=C(S(=O)(=O)NC(=O)C4=CC=C(N5CCN(CC6=C(C7=CC=C(Cl)C=C7)CCC7(CC7)C6)CC5)C=C4)C=C3S(=O)(=O)C(F)(F)F)C[C@]1([H])CN(C(=O)CCCCCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C3=C(C)N=CS3)C=C1)C(C)(C)C)C2	C79H96ClF3N10O10S4	BCL2L1;BCL-2	Q07817/P10415	VHL	WO-2024179577-A1
TPD-CPAOEZ	SCHEMBL29313921	(2S,4R)-1-[(2S)-2-[[7-[(1R,4R)-5-[(3R)-3-[4-[[4-[4-[[6-(4-chlorophenyl)spiro[2.5]oct-6-en-7-yl]methyl]piperazin-1-yl]benzoyl]sulfamoyl]-2-(trifluoromethylsulfonyl)anilino]-4-phenylsulfanylbutyl]-2,5-diazabicyclo[2.2.1]heptan-2-yl]-7-oxoheptanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL30286172	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCC(=O)N3C[C@H]4C[C@@H]3CN4CC[C@H](CSC3=CC=CC=C3)NC3=CC=C(S(=O)(=O)NC(=O)C4=CC=C(N5CCN(CC6=C(C7=CC=C(Cl)C=C7)CCC7(CC7)C6)CC5)C=C4)C=C3S(=O)(=O)C(F)(F)F)C(C)(C)C)C=C2)SC=N1	C78H94ClF3N10O10S4	BCL2L1;BCL-2	Q07817/P10415	VHL	WO-2024179577-A1
TPD-Z0J57E	SCHEMBL29313862	(2S,4R)-1-[(2S)-2-[[7-[(1S,4S)-5-[(3R)-3-[4-[[4-[4-[[2-(4-chloro-2-fluorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]benzoyl]sulfamoyl]-2-(trifluoromethylsulfonyl)anilino]-4-phenylsulfanylbutyl]-2,5-diazabicyclo[2.2.1]heptan-2-yl]-7-oxoheptanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL30286201	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCC(=O)N3C[C@@H]4C[C@H]3CN4CC[C@H](CSC3=CC=CC=C3)NC3=CC=C(S(=O)(=O)NC(=O)C4=CC=C(N5CCN(CC6=C(C7=CC=C(Cl)C=C7F)CCC(C)(C)C6)CC5)C=C4)C=C3S(=O)(=O)C(F)(F)F)C(C)(C)C)C=C2)SC=N1	C78H95ClF4N10O10S4	BCL2L1;BCL-2	Q07817/P10415	VHL	WO-2024179577-A1
TPD-VED43R	SCHEMBL29314193	(2S,4R)-1-[(2S)-2-[[7-[(3aS,6aR)-2-[(3R)-3-[4-[[4-[4-[[6-(4-chloro-2-fluorophenyl)spiro[2.5]oct-6-en-7-yl]methyl]piperazin-1-yl]benzoyl]sulfamoyl]-2-(trifluoromethylsulfonyl)anilino]-4-phenylsulfanylbutyl]-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-5-yl]-7-oxoheptanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL30977246	[H][C@@]12CN(CC[C@H](CSC3=CC=CC=C3)NC3=CC=C(S(=O)(=O)NC(=O)C4=CC=C(N5CCN(CC6=C(C7=CC=C(Cl)C=C7F)CCC7(CC7)C6)CC5)C=C4)C=C3S(=O)(=O)C(F)(F)F)C[C@]1([H])CN(C(=O)CCCCCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C3=C(C)N=CS3)C=C1)C(C)(C)C)C2	C79H95ClF4N10O10S4	BCL2L1;BCL-2	Q07817/P10415	VHL	WO-2024179577-A1
TPD-QBG5K9	SCHEMBL31346503	(2S,4R)-1-[(2S)-2-[[8-[(3aS,6aR)-2-[(3R)-3-[4-[[4-[4-[[6-(4-chlorophenyl)spiro[2.5]oct-6-en-7-yl]methyl]piperazin-1-yl]benzoyl]sulfamoyl]-2-(trifluoromethylsulfonyl)anilino]-4-phenylsulfanylbutyl]-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-5-yl]-8-oxooctanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	[H][C@@]12CN(CC[C@H](CSC3=CC=CC=C3)NC3=CC=C(S(=O)(=O)NC(=O)C4=CC=C(N5CCN(CC6=C(C7=CC=C(Cl)C=C7)CCC7(CC7)C6)CC5)C=C4)C=C3S(=O)(=O)C(F)(F)F)C[C@]1([H])CN(C(=O)CCCCCCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C3=C(C)N=CS3)C=C1)C(C)(C)C)C2	C80H98ClF3N10O10S4	BCL2L1;BCL-2	Q07817/P10415	VHL	WO-2024179577-A1
TPD-DB28MO	WO2024179577A1_23	(2S,4R)-1-[(2S)-2-[[8-[(3aS,6aR)-2-[(3R)-3-[4-[[4-[4-[[6-(4-chloro-2-fluorophenyl)spiro[2.5]oct-6-en-7-yl]methyl]piperazin-1-yl]benzoyl]sulfamoyl]-2-(trifluoromethylsulfonyl)anilino]-4-phenylsulfanylbutyl]-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-5-yl]-8-oxooctanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	[H][C@@]12CN(CC[C@H](CSC3=CC=CC=C3)NC3=CC=C(S(=O)(=O)NC(=O)C4=CC=C(N5CCN(CC6=C(C7=C(F)C=C(Cl)C=C7)CCC7(CC7)C6)CC5)C=C4)C=C3S(=O)(=O)C(F)(F)F)C[C@]1([H])CN(C(=O)CCCCCCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C3=C(C)N=CS3)C=C1)C(C)(C)C)C2	C80H97ClF4N10O10S4	BCL2L1;BCL-2	Q07817/P10415	VHL	WO-2024179577-A1
TPD-UX2JQP	SCHEMBL29219119	(2S,4R)-1-[(2S)-2-[[8-[4-[(3R)-3-[4-[[4-[4-[[2-(4-chloro-2-fluorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]benzoyl]sulfamoyl]-2-(trifluoromethylsulfonyl)anilino]-4-phenylsulfanylbutyl]piperazin-1-yl]-8-oxooctanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCC(=O)N3CCN(CC[C@H](CSC4=CC=CC=C4)NC4=CC=C(S(=O)(=O)NC(=O)C5=CC=C(N6CCN(CC7=C(C8=C(F)C=C(Cl)C=C8)CCC(C)(C)C7)CC6)C=C5)C=C4S(=O)(=O)C(F)(F)F)CC3)C(C)(C)C)C=C2)SC=N1	C78H97ClF4N10O10S4	BCL2L1;BCL-2	Q07817/P10415	VHL	WO-2024179577-A1
TPD-IJ1NXU	SCHEMBL30286130	(2S,4R)-1-[(2S)-2-[[8-[(1S,4S)-5-[(3R)-3-[4-[[4-[4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]benzoyl]sulfamoyl]-2-(trifluoromethylsulfonyl)anilino]-4-phenylsulfanylbutyl]-2,5-diazabicyclo[2.2.1]heptan-2-yl]-8-oxooctanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCC(=O)N3C[C@@H]4C[C@H]3CN4CC[C@H](CSC3=CC=CC=C3)NC3=CC=C(S(=O)(=O)NC(=O)C4=CC=C(N5CCN(CC6=C(C7=CC=C(Cl)C=C7)CCC(C)(C)C6)CC5)C=C4)C=C3S(=O)(=O)C(F)(F)F)C(C)(C)C)C=C2)SC=N1	C79H98ClF3N10O10S4	BCL2L1;BCL-2	Q07817/P10415	VHL	WO-2024179577-A1
TPD-MJ402P	SCHEMBL29314140	(2S,4R)-1-[(2S)-2-[[7-[(3aR,6aS)-2-[(3R)-3-[4-[[4-[4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]benzoyl]sulfamoyl]-2-(trifluoromethylsulfonyl)anilino]-4-phenylsulfanylbutyl]-3a,6a-dimethyl-1,3,4,6-tetrahydropyrrolo[3,4-c]pyrrol-5-yl]-7-oxoheptanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCC(=O)N3C[C@]4(C)CN(CC[C@H](CSC5=CC=CC=C5)NC5=CC=C(S(=O)(=O)NC(=O)C6=CC=C(N7CCN(CC8=C(C9=CC=C(Cl)C=C9)CCC(C)(C)C8)CC7)C=C6)C=C5S(=O)(=O)C(F)(F)F)C[C@]4(C)C3)C(C)(C)C)C=C2)SC=N1	C81H102ClF3N10O10S4	BCL2L1;BCL-2	Q07817/P10415	VHL	WO-2024179577-A1
TPD-FOPI0N	SCHEMBL29313858	(2S,4R)-1-[(2S)-2-[[7-[(1S,4S)-5-[(3R)-3-[4-[[4-[4-[[6-(4-chlorophenyl)spiro[2.5]oct-6-en-7-yl]methyl]piperazin-1-yl]benzoyl]sulfamoyl]-2-(trifluoromethylsulfonyl)anilino]-4-phenylsulfanylbutyl]-2,5-diazabicyclo[2.2.1]heptan-2-yl]-7-oxoheptanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL30285953	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCC(=O)N3C[C@@H]4C[C@H]3CN4CC[C@H](CSC3=CC=CC=C3)NC3=CC=C(S(=O)(=O)NC(=O)C4=CC=C(N5CCN(CC6=C(C7=CC=C(Cl)C=C7)CCC7(CC7)C6)CC5)C=C4)C=C3S(=O)(=O)C(F)(F)F)C(C)(C)C)C=C2)SC=N1	C78H94ClF3N10O10S4	BCL2L1;BCL-2	Q07817/P10415	VHL	WO-2024179577-A1
TPD-FCTEBM	WO2024179577A1_28	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(NC(=O)CCCCCCC(=O)N3C[C@@H]4C[C@H]3CN4CC[C@H](CSC3=CC=CC=C3)NC3=CC=C(S(=O)(=O)NC(=O)C4=CC=C(N5CCN(CC6=C(C7=CC=C(Cl)C=C7)CCC7(CC7)C6)CC5)C=C4)C=C3S(=O)(=O)C(F)(F)F)C(C)(C)C)C=C2)SC=N1	C79H96ClF3N10O10S4	BCL2L1;BCL-2	Q07817/P10415	VHL	WO-2024179577-A1
TPD-AJJZRF	WO2024179577A1_29	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCC(=O)N3C[C@H]4C[C@@H]3CN4CC[C@H](CSC3=CC=CC=C3)NC3=CC=C(S(=O)(=O)NC(=O)C4=CC=C(N5CCN(CC6=C(C7=CC=C(Cl)C=C7F)CCC7(CC7)C6)CC5)C=C4)C=C3S(=O)(=O)C(F)(F)F)C(C)(C)C)C=C2)SC=N1	C78H93ClF4N10O10S4	BCL2L1;BCL-2	Q07817/P10415	VHL	WO-2024179577-A1
TPD-Q7U5OQ	WO2024179577A1_30	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(NC(=O)CCCCCCC(=O)N3C[C@@H]4C[C@H]3CN4CC[C@H](CSC3=CC=CC=C3)NC3=CC=C(S(=O)(=O)NC(=O)C4=CC=C(N5CCN(CC6=C(C7=CC=C(Cl)C=C7F)CCC7(CC7)C6)CC5)C=C4)C=C3S(=O)(=O)C(F)(F)F)C(C)(C)C)C=C2)SC=N1	C79H95ClF4N10O10S4	BCL2L1;BCL-2	Q07817/P10415	VHL	WO-2024179577-A1
TPD-JPE8HM	SCHEMBL29313324	(2S,4R)-1-[(2S)-2-[[7-[4-[(3R)-3-[4-[[4-[4-[[6-(4-chloro-2-fluorophenyl)spiro[2.5]oct-6-en-7-yl]methyl]piperazin-1-yl]benzoyl]sulfamoyl]-2-(trifluoromethylsulfonyl)anilino]-4-phenylsulfanylbutyl]piperazin-1-yl]-7-oxoheptanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL30286159	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCC(=O)N3CCN(CC[C@H](CSC4=CC=CC=C4)NC4=CC=C(S(=O)(=O)NC(=O)C5=CC=C(N6CCN(CC7=C(C8=CC=C(Cl)C=C8F)CCC8(CC8)C7)CC6)C=C5)C=C4S(=O)(=O)C(F)(F)F)CC3)C(C)(C)C)C=C2)SC=N1	C77H93ClF4N10O10S4	BCL2L1;BCL-2	Q07817/P10415	VHL	WO-2024179577-A1
TPD-WDK7TD	WO2024179577A1_32	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(NC(=O)CCCCCCC(=O)N3CCN(CC[C@H](CSC4=CC=CC=C4)NC4=CC=C(S(=O)(=O)NC(=O)C5=CC=C(N6CCN(CC7=C(C8=CC=C(Cl)C=C8F)CCC8(CC8)C7)CC6)C=C5)C=C4S(=O)(=O)C(F)(F)F)CC3)C(C)(C)C)C=C2)SC=N1	C78H95ClF4N10O10S4	BCL2L1;BCL-2	Q07817/P10415	VHL	WO-2024179577-A1
TPD-FY7YI0	SCHEMBL29320579	(2S,4R)-1-[(2S)-2-[[7-[(1S,4S)-5-[(3R)-3-[4-[[4-[4-[[2-(4-chlorophenyl)cyclohepten-1-yl]methyl]piperazin-1-yl]benzoyl]sulfamoyl]-2-(trifluoromethylsulfonyl)anilino]-4-phenylsulfanylbutyl]-2,5-diazabicyclo[2.2.1]heptan-2-yl]-7-oxoheptanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL30286243	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCC(=O)N3C[C@@H]4C[C@H]3CN4CC[C@H](CSC3=CC=CC=C3)NC3=CC=C(S(=O)(=O)NC(=O)C4=CC=C(N5CCN(CC6=C(C7=CC=C(Cl)C=C7)CCCCC6)CC5)C=C4)C=C3S(=O)(=O)C(F)(F)F)C(C)(C)C)C=C2)SC=N1	C77H94ClF3N10O10S4	BCL2L1;BCL-2	Q07817/P10415	VHL	WO-2024179577-A1
TPD-NDL75O	WO2024179577A1_34	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(NC(=O)CCCCCCC(=O)N3C[C@@H]4C[C@H]3CN4CC[C@H](CSC3=CC=CC=C3)NC3=CC=C(S(=O)(=O)NC(=O)C4=CC=C(N5CCN(CC6=C(C7=CC=C(Cl)C=C7)CCCCC6)CC5)C=C4)C=C3S(=O)(=O)C(F)(F)F)C(C)(C)C)C=C2)SC=N1	C78H96ClF3N10O10S4	BCL2L1;BCL-2	Q07817/P10415	VHL	WO-2024179577-A1
TPD-E2JS40	SCHEMBL29219122	(2S,4R)-1-[(2S)-2-[[7-[4-[(3R)-3-[4-[[4-[4-[[2-(4-chloro-2-fluorophenyl)cyclohepten-1-yl]methyl]piperazin-1-yl]benzoyl]sulfamoyl]-2-(trifluoromethylsulfonyl)anilino]-4-phenylsulfanylbutyl]piperazin-1-yl]-7-oxoheptanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCC(=O)N3CCN(CC[C@H](CSC4=CC=CC=C4)NC4=CC=C(S(=O)(=O)NC(=O)C5=CC=C(N6CCN(CC7=C(C8=C(F)C=C(Cl)C=C8)CCCCC7)CC6)C=C5)C=C4S(=O)(=O)C(F)(F)F)CC3)C(C)(C)C)C=C2)SC=N1	C76H93ClF4N10O10S4	BCL2L1;BCL-2	Q07817/P10415	VHL	WO-2024179577-A1
TPD-987WK0	WO2024179577A1_36	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(NC(=O)CCCCCCC(=O)N3CCN(CC[C@H](CSC4=CC=CC=C4)NC4=CC=C(S(=O)(=O)NC(=O)C5=CC=C(N6CCN(CC7=C(C8=C(F)C=C(Cl)C=C8)CCCCC7)CC6)C=C5)C=C4S(=O)(=O)C(F)(F)F)CC3)C(C)(C)C)C=C2)SC=N1	C77H95ClF4N10O10S4	BCL2L1;BCL-2	Q07817/P10415	VHL	WO-2024179577-A1
TPD-WBJBNV	SCHEMBL29320847	(2S,4R)-1-[(2S)-2-[[7-[(1S,4S)-5-[(3R)-3-[4-[[4-[4-[[2-(4-chloro-2-fluorophenyl)cyclohepten-1-yl]methyl]piperazin-1-yl]benzoyl]sulfamoyl]-2-(trifluoromethylsulfonyl)anilino]-4-phenylsulfanylbutyl]-2,5-diazabicyclo[2.2.1]heptan-2-yl]-7-oxoheptanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL30286219	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCC(=O)N3C[C@@H]4C[C@H]3CN4CC[C@H](CSC3=CC=CC=C3)NC3=CC=C(S(=O)(=O)NC(=O)C4=CC=C(N5CCN(CC6=C(C7=C(F)C=C(Cl)C=C7)CCCCC6)CC5)C=C4)C=C3S(=O)(=O)C(F)(F)F)C(C)(C)C)C=C2)SC=N1	C77H93ClF4N10O10S4	BCL2L1;BCL-2	Q07817/P10415	VHL	WO-2024179577-A1
TPD-BDBOF2	WO2024179577A1_38	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(NC(=O)CCCCCCC(=O)N3C[C@@H]4C[C@H]3CN4CC[C@H](CSC3=CC=CC=C3)NC3=CC=C(S(=O)(=O)NC(=O)C4=CC=C(N5CCN(CC6=C(C7=C(F)C=C(Cl)C=C7)CCCCC6)CC5)C=C4)C=C3S(=O)(=O)C(F)(F)F)C(C)(C)C)C=C2)SC=N1	C78H95ClF4N10O10S4	BCL2L1;BCL-2	Q07817/P10415	VHL	WO-2024179577-A1
TPD-8M3Q8L	SCHEMBL29316178	(2S,4R)-1-[(2S)-2-[[7-[(3aS,6aR)-2-[(3R)-3-[4-[[4-[4-[[2-(4-chloro-2-fluorophenyl)cyclohepten-1-yl]methyl]piperazin-1-yl]benzoyl]sulfamoyl]-2-(trifluoromethylsulfonyl)anilino]-4-phenylsulfanylbutyl]-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-5-yl]-7-oxoheptanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	[H][C@@]12CN(CC[C@H](CSC3=CC=CC=C3)NC3=CC=C(S(=O)(=O)NC(=O)C4=CC=C(N5CCN(CC6=C(C7=C(F)C=C(Cl)C=C7)CCCCC6)CC5)C=C4)C=C3S(=O)(=O)C(F)(F)F)C[C@]1([H])CN(C(=O)CCCCCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C3=C(C)N=CS3)C=C1)C(C)(C)C)C2	C78H95ClF4N10O10S4	BCL2L1;BCL-2	Q07817/P10415	VHL	WO-2024179577-A1
TPD-VINPBP	WO2024179577A1_40	.	[H][C@@]12CN(CC[C@H](CSC3=CC=CC=C3)NC3=CC=C(S(=O)(=O)NC(=O)C4=CC=C(N5CCN(CC6=C(C7=C(F)C=C(Cl)C=C7)CCCCC6)CC5)C=C4)C=C3S(=O)(=O)C(F)(F)F)C[C@]1([H])CN(C(=O)CCCCCCC(=O)NC(C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C3=C(C)N=CS3)C=C1)C(C)(C)C)C2	C79H97ClF4N10O10S4	BCL2L1;BCL-2	Q07817/P10415	VHL	WO-2024179577-A1
TPD-XZ2W6E	SCHEMBL29316197	(2S,4R)-1-[(2S)-2-[[7-[(3aS,6aR)-2-[(3R)-3-[4-[[4-[4-[[2-(4-chlorophenyl)cyclohepten-1-yl]methyl]piperazin-1-yl]benzoyl]sulfamoyl]-2-(trifluoromethylsulfonyl)anilino]-4-phenylsulfanylbutyl]-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-5-yl]-7-oxoheptanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	[H][C@@]12CN(CC[C@H](CSC3=CC=CC=C3)NC3=CC=C(S(=O)(=O)NC(=O)C4=CC=C(N5CCN(CC6=C(C7=CC=C(Cl)C=C7)CCCCC6)CC5)C=C4)C=C3S(=O)(=O)C(F)(F)F)C[C@]1([H])CN(C(=O)CCCCCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C3=C(C)N=CS3)C=C1)C(C)(C)C)C2	C78H96ClF3N10O10S4	BCL2L1;BCL-2	Q07817/P10415	VHL	WO-2024179577-A1
TPD-0O0VVZ	WO2024179577A1_42	.	[H][C@@]12CN(CC[C@H](CSC3=CC=CC=C3)NC3=CC=C(S(=O)(=O)NC(=O)C4=CC=C(N5CCN(CC6=C(C7=CC=C(Cl)C=C7)CCCCC6)CC5)C=C4)C=C3S(=O)(=O)C(F)(F)F)C[C@]1([H])CN(C(=O)CCCCCCC(=O)NC(C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C3=C(C)N=CS3)C=C1)C(C)(C)C)C2	C79H98ClF3N10O10S4	BCL2L1;BCL-2	Q07817/P10415	VHL	WO-2024179577-A1
TPD-NEPFQD	SCHEMBL29219145	[(3R,5S)-1-[(2S)-2-[[7-[4-[(3R)-3-[4-[[4-[4-[[2-(4-chlorophenyl)cyclohepten-1-yl]methyl]piperazin-1-yl]benzoyl]sulfamoyl]-2-(trifluoromethylsulfonyl)anilino]-4-phenylsulfanylbutyl]piperazin-1-yl]-7-oxoheptanoyl]amino]-3,3-dimethylbutanoyl]-5-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-3-yl] acetate	CC(=O)O[C@@H]1C[C@@H](C(=O)N[C@@H](C)C2=CC=C(C3=C(C)N=CS3)C=C2)N(C(=O)[C@@H](NC(=O)CCCCCC(=O)N2CCN(CC[C@H](CSC3=CC=CC=C3)NC3=CC=C(S(=O)(=O)NC(=O)C4=CC=C(N5CCN(CC6=C(C7=CC=C(Cl)C=C7)CCCCC6)CC5)C=C4)C=C3S(=O)(=O)C(F)(F)F)CC2)C(C)(C)C)C1	C78H96ClF3N10O11S4	BCL2L1;BCL-2	Q07817/P10415	VHL	WO-2024179577-A1
TPD-ZDBSKJ	WO2024180157A1_02C-N	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3(F)CC3)C(C)(C)C)C(OCCCCCCNC(=O)CN3C=C(C4=CC=C5C(=C4)[C@H](F)C[C@@]54NC(=O)N(CC(=O)N(CC5=CC=C(F)C=C5)[C@@H](C)C(F)(F)F)C4=O)C=N3)=C2)SC=N1	C60H68F6N10O9S	P300	Q09472	CRBN	WO-2024180157-A1
TPD-VMZ80U	WO2024180157A1_02C	.	C[C@H](N(CC1=CC=C(F)C=C1)C(=O)CN1C(=O)N[C@@]2(C[C@H](F)C3=CC(C4=CN(CC(=O)NCCCCCCCNC5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)N=C4)=CC=C32)C1=O)C(F)(F)F	C48H48F5N9O8	P300	Q09472	CRBN	WO-2024180157-A1
TPD-TZBVTP	WO2024180157A1_02D	.	C[C@H](N(CC1=CC=C(F)C=C1)C(=O)CN1C(=O)N[C@]2(C[C@@H](F)C3=CC(C4=CN(CC(=O)NCCCNC5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)N=C4)=CC=C32)C1=O)C(F)(F)F	C44H40F5N9O8	P300	Q09472	CRBN	WO-2024180157-A1
TPD-GVL9OS	WO2024180157A1_02E	.	C[C@H](N(CC1=CC=C(F)C=C1)C(=O)CN1C(=O)N[C@@]2(C[C@@H](F)C3=CC(C4=CN(CC(=O)N5CCC(CN6CCN(C7=C(F)C=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)CC5)N=C4)=CC=C32)C1=O)C(F)(F)F	C51H50F6N10O8	P300	Q09472	CRBN	WO-2024180157-A1
TPD-RCE97E	WO2024180157A1_02F	.	C[C@H](N(CC1=CC=C(F)C=C1)C(=O)CN1C(=O)N[C@@]2(C[C@@H](F)C3=CC(C4=CN(CC(=O)N5CCC(CN6CCN(C7=CC=C(N8CCC(=O)NC8=O)C=C7)CC6)CC5)N=C4)=CC=C32)C1=O)C(F)(F)F	C48H51F5N10O6	P300	Q09472	CRBN	WO-2024180157-A1
TPD-SGOCIQ	WO2024180157A1_02G	.	C[C@H](N(CC1=CC=C(F)C=C1)C(=O)CN1C(=O)N[C@@]2(C[C@@H](F)C3=CC(C4=CN(CC(=O)N5CCC(CN6CCN(C7=CC=C(NC8CCC(=O)NC8=O)C=C7)CC6)CC5)N=C4)=CC=C32)C1=O)C(F)(F)F	C49H53F5N10O6	P300	Q09472	CRBN	WO-2024180157-A1
TPD-WHY4U1	WO2024180157A1_02H	.	C[C@H](N(CC1=CC=C(F)C=C1)C(=O)CN1C(=O)N[C@@]2(C[C@@H](F)C3=CC(C4=CN(CC(=O)N5CCC(CN6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)CC5)N=C4)=CC=C32)C1=O)C(F)(F)F	C51H51F5N10O8	P300	Q09472	CRBN	WO-2024180157-A1
TPD-ASUQ6E	WO2024180157A1_02I	.	C[C@H](N(CC1=CC=C(F)C=C1)C(=O)CN1C(=O)N[C@@]2(C[C@@H](F)C3=CC(C4=CN(CC(=O)NCCCCCCCNC5=CC=C6C(=O)N(C7CCC(=O)N(C)C7=O)C(=O)C6=C5)N=C4)=CC=C32)C1=O)C(F)(F)F	C49H50F5N9O8	P300	Q09472	VHL	WO-2024180157-A1
TPD-Y3YM7D	WO2024180157A1_02J	N-[5-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]pentyl]-2-[4-[(1S,3R)-3-fluoro-1'-[2-[(4-fluorophenyl)methyl-[(2S)-1,1,1-trifluoropropan-2-yl]amino]-2-oxoethyl]-2',5'-dioxospiro[2,3-dihydroindene-1,4'-imidazolidine]-5-yl]pyrazol-1-yl]acetamide	C[C@H](N(CC1=CC=C(F)C=C1)C(=O)CN1C(=O)N[C@]2(C[C@@H](F)C3=CC(C4=CN(CC(=O)NCCCCCNC5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)N=C4)=CC=C32)C1=O)C(F)(F)F	C46H44F5N9O8	P300	Q09472	VHL	WO-2024180157-A1
TPD-GQCKLZ	WO2024180157A1_02K	.	C[C@H](N(CC1=CC=C(F)C=C1)C(=O)CN1C(=O)N[C@@]2(C[C@@H](F)C3=CC(C4=CN(CC(=O)NCCCCCCCNC5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)N=C4)=CC=C32)C1=O)C(F)(F)F	C48H48F5N9O8	P300	Q09472	VHL	WO-2024180157-A1
TPD-LTKVV8	WO2024180157A1_02L	N-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethyl]-2-[4-[(1S,3R)-3-fluoro-1'-[2-[(4-fluorophenyl)methyl-[(2S)-1,1,1-trifluoropropan-2-yl]amino]-2-oxoethyl]-2',5'-dioxospiro[2,3-dihydroindene-1,4'-imidazolidine]-5-yl]pyrazol-1-yl]acetamide	C[C@H](N(CC1=CC=C(F)C=C1)C(=O)CN1C(=O)N[C@]2(C[C@@H](F)C3=CC(C4=CN(CC(=O)NCCOCCNC5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)N=C4)=CC=C32)C1=O)C(F)(F)F	C45H42F5N9O9	P300	Q09472	VHL	WO-2024180157-A1
TPD-52QJHW	WO2024180157A1_02M	.	C[C@H](N(CC1=CC=C(F)C=C1)C(=O)CN1C(=O)N[C@@]2(C[C@@H](F)C3=CC(C4=CN(CC(=O)NCCOCCOCCOCCNC5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)N=C4)=CC=C32)C1=O)C(F)(F)F	C49H50F5N9O11	P300	Q09472	VHL	WO-2024180157-A1
TPD-ZGXA8C	WO2024180157A1_02N	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCNC(=O)CN3C=C(C4=CC=C5C(=C4)[C@H](F)C[C@@]54NC(=O)N(CC(=O)N(CC5=CC=C(F)C=C5)[C@@H](C)C(F)(F)F)C4=O)C=N3)C(C)(C)C)C=C2)SC=N1	C53H57F5N10O8S	P300	Q09472	VHL	WO-2024180157-A1
TPD-Q56JQ9	WO2024180157A1_02O	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCNC(=O)CN3C=C(C4=CC=C5C(=C4)[C@H](F)C[C@@]54NC(=O)N(CC(=O)N(CC5=CC=C(F)C=C5)[C@@H](C)C(F)(F)F)C4=O)C=N3)C(C)(C)C)C=C2)SC=N1	C55H61F5N10O8S	P300	Q09472	VHL	WO-2024180157-A1
TPD-FCO3HB	WO2024180157A1_02P	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3(F)CC3)C(C)(C)C)C(OCCCCNC(=O)CN3C=C(C4=CC=C5C(=C4)[C@H](C)C[C@@]54NC(=O)N(CC(=O)N(CC5=CC=C(F)C=C5)[C@@H](C)C(F)(F)F)C4=O)C=N3)=C2)SC=N1	C59H67F5N10O9S	P300	Q09472	VHL	WO-2024180157-A1
TPD-TGN2WG	WO2024183650A1_1	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CCOCCN3CCC4(CC3)CC(n3cc(NC(=O)c5cnn6ccc(N7CCOCC7)nc56)c(C(F)F)n3)C4)c21	C41H45F2N11O6	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-S3G434	WO2024183650A1_2	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CCOCCCN3CCC4(CC3)CC(n3cc(NC(=O)c5cnn6ccc(N7C[C@H]8C[C@@H]7CO8)nc56)c(C(F)F)n3)C4)c21	C43H47F2N11O6	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-5IUI2C	WO2024183650A1_3	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CCN3CCC(CN4CCC5(CC4)CC(n4cc(NC(=O)c6cnn7ccc(N8C[C@H]9C[C@@H]8CO9)nc67)c(C(F)F)n4)C5)CC3)c21	C46H52F2N12O5	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-1W9OWM	WO2024183650A1_4	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CCOCCCCN3CCC4(CC3)CC(n3cc(NC(=O)c5cnn6ccc(N7C[C@H]8C[C@@H]7CO8)nc56)c(C(F)F)n3)C4)c21	C44H49F2N11O6	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-72HDPW	WO2024183650A1_5	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CCOCC(C)(C)C(=O)N3CCC4(CC3)CC(n3cc(NC(=O)c5cnn6ccc(N7C[C@H]8C[C@@H]7CO8)nc56)c(C(F)F)n3)C4)c21	C45H49F2N11O7	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-6FQNEE	WO2024183650A1_6	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CCOCC3(CN4CCC5(CC4)CC(n4cc(NC(=O)c6cnn7ccc(N8C[C@H]9C[C@@H]8CO9)nc67)c(C(F)F)n4)C5)CC3)c21	C45H49F2N11O6	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-RDUOVC	WO2024183650A1_7	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CCOCC3(C(=O)N4CCC5(CC4)CC(n4cc(NC(=O)c6cnn7ccc(N8C[C@H]9C[C@@H]8CO9)nc67)c(C(F)F)n4)C5)CC3)c21	C45H47F2N11O7	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-CACG1S	WO2024183650A1_8	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CCOCCC(=O)N3CCC4(CC3)CC(n3cc(NC(=O)c5cnn6ccc(N7C[C@H]8C[C@@H]7CO8)nc56)c(C(F)F)n3)C4)c21	C43H45F2N11O7	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-1N19AC	WO2024183650A1_9	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CCOCC3CC(N4CCC5(CC4)CC(n4cc(NC(=O)c6cnn7ccc(N8C[C@H]9C[C@@H]8CO9)nc67)c(C(F)F)n4)C5)C3)c21	C45H49F2N11O6	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-6Y96IV	WO2024183650A1_10	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CCOC(C)(C)C(=O)N3CCC4(CC3)CC(n3cc(NC(=O)c5cnn6ccc(N7C[C@H]8C[C@@H]7CO8)nc56)c(C(F)F)n3)C4)c21	C44H47F2N11O7	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-HBYALR	WO2024183650A1_11	.	CC(OCC#Cc1cccc2c1n(C)c(=O)n2C1CCC(=O)NC1=O)C(=O)N1CCC2(CC1)CC(n1cc(NC(=O)c3cnn4ccc(N5C[C@H]6C[C@@H]5CO6)nc34)c(C(F)F)n1)C2	C43H45F2N11O7	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-K8OU97	WO2024183650A1_12	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CCOCC(=O)N3CCC4(CC3)CC(n3cc(NC(=O)c5cnn6ccc(N7C[C@H]8C[C@@H]7CO8)nc56)c(C(F)F)n3)C4)c21	C42H43F2N11O7	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-0U8NNZ	WO2024183650A1_13	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CCOC3CCN(C(=O)N4CCC5(CC4)CC(n4cc(NC(=O)c6cnn7ccc(N8C[C@H]9C[C@@H]8CO9)nc67)c(C(F)F)n4)C5)CC3)c21	C46H50F2N12O7	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-3Y1AOE	WO2024183650A1_14	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CCOC3CN(C(=O)N4CCC5(CC4)CC(n4cc(NC(=O)c6cnn7ccc(N8C[C@H]9C[C@@H]8CO9)nc67)c(C(F)F)n4)C5)C3)c21	C44H46F2N12O7	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-WIL7M2	WO2024183650A1_15	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CCCCCN3CCC4(CC3)CC(n3cc(NC(=O)c5cnn6ccc(N7C[C@H]8C[C@@H]7CO8)nc56)c(C(F)F)n3)C4)c21	C43H47F2N11O5	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-HZ5MA1	WO2024183650A1_16	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CCCOC(=O)N3CCC4(CC3)CC(n3cc(NC(=O)c5cnn6ccc(N7C[C@H]8C[C@@H]7CO8)nc56)c(C(F)F)n3)C4)c21	C42H43F2N11O7	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-P9VVR9	WO2024183650A1_17	.	O=C1CCC(n2c(=O)[nH]c3c(C#CCCCN4CCC5(CC4)CC(n4cc(NC(=O)c6cnn7ccc(N8CCOCC8)nc67)c(C(F)F)n4)C5)cccc32)C(=O)N1	C40H43F2N11O5	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-WHD175	WO2024183650A1_18	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CCO[C@@H]3CCN(C(=O)N4CCC5(CC4)CC(n4cc(NC(=O)c6cnn7ccc(N8C[C@H]9C[C@@H]8CO9)nc67)c(C(F)F)n4)C5)C3)c21	C45H48F2N12O7	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-LFZ3YH	WO2024183650A1_20	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CCO[C@H]3C[C@@H](C(=O)N4CCC5(CC4)CC(n4cc(NC(=O)c6cnn7ccc(N8CCOCC8)nc67)c(C(F)F)n4)C5)C3)c21	C44H47F2N11O7	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-Q9QO7Z	WO2024183650A1_21	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CCOC(=O)N3CC(N4CCC5(CC4)CC(n4cc(NC(=O)c6cnn7ccc(N8C[C@H]9C[C@@H]8CO9)nc67)c(C(F)F)n4)C5)C3)c21	C44H46F2N12O7	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-XU5YAA	WO2024183650A1_22	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CCCN3CCC4(CC3)CC(n3cc(NC(=O)c5cnn6ccc(N7C[C@H]8C[C@@H]7CO8)nc56)c(C(F)F)n3)C4)c21	C41H43F2N11O5	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-SBYH3Z	WO2024183650A1_23	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CCOC(=O)N3CCC4(CC3)CC(n3cc(NC(=O)c5cnn6ccc(N7CCOCC7)nc56)c(C(F)F)n3)C4)c21	C40H41F2N11O7	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-ZQKSW5	WO2024183650A1_24	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CCCC(=O)N3CCC4(CC3)CC(n3cc(NC(=O)c5cnn6ccc(N7C[C@H]8C[C@@H]7CO8)nc56)c(C(F)F)n3)C4)c21	C42H43F2N11O6	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-9RZ5QK	WO2024183650A1_25	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CCCCC(=O)N3CCC4(CC3)CC(n3cc(NC(=O)c5cnn6ccc(N7C[C@H]8C[C@@H]7CO8)nc56)c(C(F)F)n3)C4)c21	C43H45F2N11O6	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-6WKI6K	WO2024183650A1_26	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CCC3CN(C(=O)N4CCC5(CC4)CC(n4cc(NC(=O)c6cnn7ccc(N8C[C@H]9C[C@@H]8CO9)nc67)c(C(F)F)n4)C5)C3)c21	C44H46F2N12O6	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-8S937U	WO2024183650A1_27	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CCC3CCN(C(=O)N4CCC5(CC4)CC(n4cc(NC(=O)c6cnn7ccc(N8C[C@H]9C[C@@H]8CO9)nc67)c(C(F)F)n4)C5)CC3)c21	C46H50F2N12O6	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-V3TE14	WO2024183650A1_28	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CCN3CC[C@H](CN4CCC5(CC4)CC(n4cc(NC(=O)c6cnn7ccc(N8C[C@H]9C[C@@H]8CO9)nc67)c(C(F)F)n4)C5)C3)c21	C45H50F2N12O5	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-96ZT5D	WO2024183650A1_29	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CCO[C@H]3C[C@H](CN4CCC5(CC4)CC(n4cc(NC(=O)c6cnn7ccc(N8C[C@H]9C[C@@H]8CO9)nc67)c(C(F)F)n4)C5)C3)c21	C45H49F2N11O6	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-QKCJ16	WO2024183650A1_30	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CCO[C@H]3C[C@@H](CN4CCC5(CC4)CC(n4cc(NC(=O)c6cnn7ccc(N8C[C@H]9C[C@@H]8CO9)nc67)c(C(F)F)n4)C5)C3)c21	C45H49F2N11O6	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-OYKGFL	WO2024183650A1_31	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CCOC3CCC(CN4CCC5(CC4)CC(n4cc(NC(=O)c6cnn7ccc(N8C[C@H]9C[C@@H]8CO9)nc67)c(C(F)F)n4)C5)CC3)c21	C47H53F2N11O6	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-2NUT7S	WO2024183650A1_32	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CCO[C@H]3CC[C@@H](CN4CCC5(CC4)CC(n4cc(NC(=O)c6cnn7c6NC(N6C[C@H]8C[C@@H]6CO8)C=C7)c(C(F)F)n4)C5)CC3)c21	C47H55F2N11O6	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-1PRG54	WO2024183650A1_33	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CCOC3CCC(N4CCC5(CC4)CC(n4cc(NC(=O)c6cnn7ccc(N8C[C@H]9C[C@@H]8CO9)nc67)c(C(F)F)n4)C5)CC3)c21	C46H51F2N11O6	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-NTU385	WO2024183650A1_34	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CC(C)(C)N3CCC(CN4CCC5(CC4)CC(n4cc(NC(=O)c6cnn7ccc(N8C[C@H]9C[C@@H]8CO9)nc67)c(C(F)F)n4)C5)CC3)c21	C48H56F2N12O5	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-WU2I8A	WO2024183650A1_35	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CCC3CCC(N4CCC5(CC4)CC(n4cc(NC(=O)c6cnn7ccc(N8C[C@H]9C[C@@H]8CO9)nc67)c(C(F)F)n4)C5)CC3)c21	C46H51F2N11O5	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-OAUODU	WO2024183650A1_36	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CCO[C@H]3C[C@H](C(=O)N4CCC5(CC4)CC(n4cc(NC(=O)c6cnn7ccc(N8CCOCC8)nc67)c(C(F)F)n4)C5)C3)c21	C44H47F2N11O7	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-GNJ79Q	WO2024183650A1_37	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CCOCCN3CCC4(CCC(n5cc(NC(=O)c6cnn7ccc(N8C[C@H]9C[C@@H]8CO9)nc67)c(C(F)F)n5)CC4)CC3)c21	C44H49F2N11O6	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-HV4BFM	WO2024183650A1_38	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CCOC3CC(N4CCC5(CCC(n6cc(NC(=O)c7cnn8c7NC(N7C[C@H]9C[C@@H]7CO9)C=C8)c(C(F)F)n6)CC5)CC4)C3)c21	C46H53F2N11O6	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-XLVW5F	WO2024183650A1_39	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CCOC3CN(C(=O)N4CCC5(CCC(n6cc(NC(=O)c7cnn8ccc(N9CCOCC9)nc78)c(C(F)F)n6)CC5)CC4)C3)c21	C45H50F2N12O7	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-QUIA54	WO2024183650A1_40	.	Cc1c(C(=O)Nc2cn(C3CCC4(CC3)CCN(CC3CC(OCC#Cc5cccc6c5n(C)c(=O)n6C5CCC(=O)NC5=O)C3)CC4)nc2C(F)F)cnn1/C=C\C(=N)N1C[C@H]2C[C@@H]1CO2	C48H57F2N11O6	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-622MQW	WO2024183650A1_41	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CCOC3CCN(C(=O)N4CC5(CCC(n6cc(NC(=O)c7cnn8ccc(N9C[C@H]%10C[C@@H]9CO%10)nc78)c(C(F)F)n6)CC5)C4)CC3)c21	C46H50F2N12O7	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-8K2RFE	WO2024183650A1_42	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CCOC3CN(C(=O)N4CC5(CCC(n6cc(NC(=O)c7cnn8ccc(N9C[C@H]%10C[C@@H]9CO%10)nc78)c(C(F)F)n6)CC5)C4)C3)c21	C44H46F2N12O7	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-FCKU8I	WO2024183650A1_43	.	Cn1c(=O)n(C2CCC(=O)NC2O)c2cccc(C#CCOC3CCN(C(=O)N4CCC5(CCC(n6cc(NC(=O)c7cnn8ccc(N9C[C@H]%10C[C@@H]9CO%10)nc78)c(C(F)F)n6)CC5)CC4)CC3)c21	C48H56F2N12O7	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-KO6OAU	WO2024183650A1_44	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CCOC[C@H]3C[C@H]3CN3CCC4(CC3)CC(n3cc(NC(=O)c5cnn6ccc(N7C[C@H]8C[C@@H]7CO8)nc56)c(C(F)F)n3)C4)c21	C45H49F2N11O6	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-L3M1OQ	WO2024183650A1_45	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CCOC3CC(NC(=O)N4CC5(CCC(n6cc(NC(=O)c7cnn8ccc(N9C[C@H]%10C[C@@H]9CO%10)nc78)c(C(F)F)n6)CC5)C4)C3)c21	C45H48F2N12O7	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-V8CJU4	WO2024183650A1_46	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CCOC3CCC(CN4CCC5(CCC(N6C=C(NC(=O)c7cnn8ccc(N9C[C@H]%10C[C@@H]9CO%10)nc78)C(C(F)F)N6)CC5)CC4)CC3)c21	C49H59F2N11O6	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-FW8ANC	WO2024183650A1_47	.	COc1cc2nn(C3CCC4(CC3)CCN(CC3CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC3)CC4)cc2cc1C(=O)Nc1cnc2cccnn12	C44H48N10O6	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-XFFQEA	WO2024183650A1_48	.	COc1cc2nn(C3CCC4(CC3)CCN(CC3CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC3)CC4)cc2cc1NC(=O)c1cnn2cccnc12	C44H48N10O6	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-9L41C3	WO2024183650A1_50	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CC(C)(C)N3CC(C(=O)N4CCC5(CC4)CC(n4cc(NC(=O)c6cnn7ccc(N8C[C@H]9C[C@@H]8CO9)nc67)c(C(F)F)n4)C5)C3)c21	C46H50F2N12O6	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-QUU8B4	WO2024183650A1_51	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CCOC34CCC(C(=O)N5CCC6(CC5)CC(n5cc(NC(=O)c7cnn8ccc(N9C[C@H]%10C[C@@H]9CO%10)nc78)c(C(F)F)n5)C6)(CC3)CC4)c21	C49H53F2N11O7	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-LEV2CT	WO2024183650A1_52	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CCOC34CCC(CN5CCC6(CC5)CC(N5C=C(NC(=O)c7cnn8ccc(N9C[C@H]%10C[C@@H]9CO%10)nc78)C(C(F)F)N5)C6)(CC3)CC4)c21	C49H57F2N11O6	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-2904TH	WO2024183650A1_53	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CC(C)(C)N3CC[C@H](CN4CCC5(CC4)CC(n4cc(NC(=O)c6cnn7ccc(N8C[C@H]9C[C@@H]8CO9)nc67)c(C(F)F)n4)C5)C3)c21	C47H54F2N12O5	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-0Z029K	WO2024183650A1_54	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CC(C)(C)N3CCC(N4CCC5(CC4)CC(n4cc(NC(=O)C6=C7N=C(N8C[C@H]9C[C@@H]8CO9)C=CN7NC6)c(C(F)F)n4)C5)C3)c21	C46H54F2N12O5	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-KT3FD6	WO2024183650A1_55	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CC(C)(C)N3CC[C@H](C(=O)N4CCC5(CC4)CC(n4cc(NC(=O)c6cnn7ccc(N8C[C@H]9C[C@@H]8CO9)nc67)c(C(F)F)n4)C5)C3)c21	C47H52F2N12O6	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-ZEQEKV	WO2024183650A1_56	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CC(C)(C)N3CCC(C(=O)N4CCC5(CC4)CC(n4cc(NC(=O)c6cnn7ccc(N8CCOCC8)nc67)c(C(F)F)n4)C5)CC3)c21	C47H54F2N12O6	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-1MFS6Y	WO2024183650A1_57	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CCOc3ccc(CN4CCC5(CC4)CC(n4cc(NC(=O)c6cnn7ccc(N8C[C@H]9C[C@@H]8CO9)nc67)c(C(F)F)n4)C5)cc3)c21	C47H47F2N11O6	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-QA11OR	WO2024183650A1_58	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CCN3CC(C(=O)N4CCC5(CC4)CC(n4cc(NC(=O)c6cnn7ccc(N8C[C@H]9C[C@@H]8CO9)nc67)c(C(F)F)n4)C5)C3)c21	C44H46F2N12O6	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-AXZ8HP	WO2024183650A1_59	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CCN3CC[C@H](C(=O)N4CCC5(CC4)CC(n4cc(NC(=O)c6cnn7ccc(N8C[C@H]9C[C@@H]8CO9)nc67)c(C(F)F)n4)C5)C3)c21	C45H48F2N12O6	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-80O7RH	WO2024183650A1_60	.	Cn1c(=O)n(C2CCCNC2=O)c2cccc(C#CCN3CC[C@@H](C(=O)N4CCC5(CC4)CC(n4cc(NC(=O)c6cnn7ccc(N8C[C@H]9C[C@@H]8CO9)nc67)c(C(F)F)n4)C5)C3)c21	C45H50F2N12O5	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-USAHDW	WO2024183650A1_61	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CCOC3CCN(CC4CCC5(CC4)CC(n4cc(NC(=O)c6cnn7ccc(N8CCOCC8)nc67)c(C(F)F)n4)C5)CC3)c21	C46H53F2N11O6	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-EXATTH	WO2024183650A1_62	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CCN3CCC(CN4CCC5(CC4)CC(n4cc(NC(=O)c6cnn7ccc(N8C[C@H]9C[C@@H]8CO9)nc67)c(C(F)F)n4)C5)CC3=O)c21	C46H50F2N12O6	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-8HREA3	WO2024183650A1_63	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CCN3CC[C@@H](CN4CCC5(CC4)CC(n4cc(NC(=O)c6cnn7ccc(N8C[C@H]9C[C@@H]8CO9)nc67)c(C(F)F)n4)C5)C3)c21	C45H50F2N12O5	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-F70OGS	WO2024183650A1_64	.	COc1cc2nn(C3CCC4(CC3)CCN(C3CC(OCC#Cc5cccc6c5n(C)c(=O)n6C5CCC(=O)NC5=O)C3)CC4)cc2cc1C(=O)Nc1cnc2cccnn12	C45H48N10O6	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-3G0PPV	WO2024183650A1_65	.	COc1cc2nn(C3CC4(CCN(CC5CC(OCC#Cc6cccc7c6n(C)c(=O)n7C6CCC(=O)NC6=O)C5)CC4)C3)cc2cc1C(=O)Nc1cnc2cccnn12	C44H46N10O6	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-8ALXZD	WO2024183650A1_66	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CCO[C@H]3CC[C@@H](CN4CC5(CCC(n6cc(NC(=O)c7cnn8ccc(N9C[C@H]%10C[C@@H]9CO%10)nc78)c(C(F)F)n6)CC5)C4)CC3)c21	C47H53F2N11O6	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-9QFEDL	WO2024183650A1_67	.	COc1cc2nn(C3CCC4(CC3)CCN(CC3CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC3)CC4)cc2cc1NC(=O)c1cnc2cccnn12	C44H48N10O6	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-5V7WDZ	WO2024183650A1_68	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CCOC3CCN(CC4CCC5(CC4)CCC(n4cc(NC(=O)c6cnn7ccc(N8C[C@H]9C[C@@H]8CO9)nc67)c(C(F)F)n4)CC5)CC3)c21	C49H57F2N11O6	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-DHP1PL	WO2024183650A1_69	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CCOCC3CCC4(CC3)CCC(n3cc(NC(=O)c5cnn6ccc(N7C[C@H]8C[C@@H]7CO8)nc56)c(C(F)F)n3)CC4)c21	C44H48F2N10O6	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-QUS6ER	WO2024183650A1_70	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CC(C)(C)C(=O)N3CCC4(CC3)CC(n3cc(NC(=O)c5cnn6ccc(N7C[C@H]8C[C@@H]7CO8)nc56)c(C(F)F)n3)C4)c21	C43H45F2N11O6	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-C6L6BV	WO2024183650A1_71	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CCOC3CCC(C(=O)N4CCC5(CC4)CC(n4cc(NC(=O)c6cnn7ccc(N8C[C@H]9C[C@@H]8CO9)nc67)c(C(F)F)n4)C5)CC3)c21	C47H51F2N11O7	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-TLDHBB	WO2024183650A1_72	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CCO[C@H]3CC[C@@H](C(=O)N4CCC5(CC4)CC(n4cc(NC(=O)c6cnn7ccc(N8C[C@H]9C[C@@H]8CO9)nc67)c(C(F)F)n4)C5)CC3)c21	C47H51F2N11O7	IRAK4	Q9NWZ3	CRBN	WO-2024183650-A1
TPD-XBKJLP	WO2024188281A1_2B	.	CCCC1=C(C2=C(C)C(F)=CC3=C2C=NN3)C(OC(C)(C)C2=CC=C(C3=CN([C@H](C(=O)N4C[C@H](O)CC4C(=O)N[C@@H](CO)C4=CC=C(C5=C(C)N=CS5)C=C4)C(C)C)NN3)C=C2)=C2N=C(O[C@@H]3CCN(C(C)=O)C3)N=C(N3C[C@@H]4C[C@H]3CN4)C2=C1	C63H74FN13O7S	KRAS	P01116	VHL	WO-2024188281-A1
TPD-OAO512	WO2024188281A1_3B	.	CC1=C(C2=CC=C([C@H](CO)NC(=O)C3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C(C4=CC=C(C5(C)CC6=C(C7=C(C=C6F)NN=C7)C6=C(C7CC7)C=C7C(N8C[C@@H]9C[C@H]8CN9)=NC(OC[C@H](C)N(C)O)=NC7=C6O5)C=C4)N=N3)C=C2)SC=N1	C60H66FN13O7S	KRAS	P01116	VHL	WO-2024188281-A1
TPD-D533FA	WO2024188281A1_5B	.	CON(C)C[C@@H](C)OC1=NC2=C(OCC3=CC=C(C4=CN([C@H](C(=O)N5C[C@H](O)CC5C(=O)N[C@@H](CO)C5=CC=C(C6=C(C)N=C[Se]6)C=C5)C(C)C)NN4)C=C3)C(C3=C(C)C(F)=CC4=C3C=NN4)=C(C3CC3)C=C2C(N2C[C@@H]3C[C@H]2CN3)=N1	C60H70FN13O7Se	KRAS	P01116	VHL	WO-2024188281-A1
TPD-XNR1WZ	WO2024188906A1_595	.	CC1=NN(CCCCCCCCNC2=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=CC=C2)C2=CC(C(=O)NC3=CN4C=C(C5CCCN5C)N=C4C=N3)=CC=C21	C41H46N10O5	MLLT3;MLLT1	P42568/Q03111	CRBN	WO-2024188906-A1
TPD-2H42ST	WO2024188906A1_599	.	CN1CCCC1C1=CN2C=C(NC(=O)CCCCCCCC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)N=CC2=N1	C32H37N7O5	MLLT3;MLLT1	P42568/Q03111	CRBN	WO-2024188906-A1
TPD-AWV6MF	WO2024188906A1_600	.	CN1N=C(N2CCC(CN3CCN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5)CC3)CC2)C2=CC(C(=O)NC3=CN4C=C(C5CCCN5C)N=C4C=N3)=CC=C21	C43H50N12O4	MLLT3;MLLT1	P42568/Q03111	CRBN	WO-2024188906-A1
TPD-81XV3P	WO2024188906A1_603	.	CC1=NN(CCCCCCCCNC2=C3C(=O)N(C4CCC(=O)NC4=O)C(=N)C3=CC=C2)C2=C1C=C(F)C(C(=O)NC1=CN3C=C(C4CCCN4)N=C3C=N1)=C2	C40H44FN11O4	MLLT3;MLLT1	P42568/Q03111	CRBN	WO-2024188906-A1
TPD-BLVGCE	WO2024188906A1_604	.	CC1=NN(CCCCCCCCOC2=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=CC=C2)C2=C1C=CC(C(=O)NC1=CN3C=C(C4CCCN4C)N=C3C=N1)=C2	C41H45N9O6	MLLT3;MLLT1	P42568/Q03111	CRBN	WO-2024188906-A1
TPD-3C8H0Q	WO2024188906A1_605	.	CC1=NN(CCCCCCNC2=CC3=C(C=C2)C(=O)N([C@@H]2CCC(=N)NC2=O)C3=O)C2=CC(C(=O)NC3=CN4C=C(C5CCCN5C)N=C4C=N3)=CC=C21	C39H43N11O4	MLLT3;MLLT1	P42568/Q03111	CRBN	WO-2024188906-A1
TPD-BL1SSF	WO2024188906A1_606	.	CN1CCCC1C1=CN2C=C(NC(=O)C3=CC=C(C4=CN(CCCC5CCN(C6=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)CC5)N=C4)C=C3)N=CC2=N1	C42H44N10O5	MLLT3;MLLT1	P42568/Q03111	CRBN	WO-2024188906-A1
TPD-IFKJSA	WO2024188906A1_607	.	CN1CCCC1C1=CN2C=C(NC(=O)C3=CC=C(C4=CN(CCCC5CCN(C6=C7CN(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)CC5)N=C4)C=C3)N=CC2=N1	C42H46N10O4	MLLT3;MLLT1	P42568/Q03111	CRBN	WO-2024188906-A1
TPD-8VL3PL	WO2024188906A1_608	.	CC1=NN(CCCCCC#CC2=CC=CC3=C2CN(C2CCC(=O)NC2=O)C3=O)C2=C1C=CC(C(=O)NC1=CN3C=C(C4CCCN4)N=C3C=N1)=C2	C39H39N9O4	MLLT3;MLLT1	P42568/Q03111	CRBN	WO-2024188906-A1
TPD-NJMI53	WO2024188906A1_609	.	CC1=NN(CCCCCCCC#CC2=C3CN(C4CCC(=O)NC4=O)C(=O)C3=CC=C2)C2=CC(C(=O)NC3=CN4C=C(C5CCCN5C)N=C4C=N3)=CC=C21	C42H45N9O4	MLLT3;MLLT1	P42568/Q03111	CRBN	WO-2024188906-A1
TPD-0310NA	WO2024188906A1_610	.	CC1=NN(CCOCCCCC#CC2=CC=CC3=C2CN(C2CCC(=O)NC2=O)C3=O)C2=CC(C(=O)NC3=CN4C=C(C5CCCN5C)N=C4C=N3)=CC=C21	C41H43N9O5	MLLT3;MLLT1	P42568/Q03111	CRBN	WO-2024188906-A1
TPD-GX0X56	SCHEMBL31198664	4-chloro-7-[4-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-1H-indole-3-carbonitrile	N#Cc1c[nH]c2c(N3CCC(c4ccc(N5CCC(CN6CCN(c7ccc8c(c7)CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)cc4)CC3)ccc(Cl)c12	C43H47ClN8O3	AR	P10275	CRBN	WO-2024189488-A1
TPD-5BIFAJ	SCHEMBL31198529	7-[4-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-4-fluoro-1H-indole-3-carbonitrile	N#Cc1c[nH]c2c(N3CCC(c4ccc(N5CCC(CN6CCN(c7ccc8c(c7)CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)cc4)CC3)ccc(F)c12	C43H47FN8O3	AR	P10275	CRBN	WO-2024189488-A1
TPD-FSLBHX	SCHEMBL31198657	4-chloro-7-[4-[4-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-1H-indole-3-carbonitrile	N#Cc1c[nH]c2c(N3CCC(c4ccc(N5CCC(CN6CCC(n7ccc8c(N9CCC(=O)NC9=O)cccc87)CC6)CC5)cc4)CC3)ccc(Cl)c12	C43H47ClN8O2	AR	P10275	CRBN	WO-2024189488-A1
TPD-QJHUV8	SCHEMBL31198706	7-[4-[4-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-4-fluoro-1H-indole-3-carbonitrile	N#Cc1c[nH]c2c(N3CCC(c4ccc(N5CCC(CN6CCC(n7ccc8c(N9CCC(=O)NC9=O)cccc87)CC6)CC5)cc4)CC3)ccc(F)c12	C43H47FN8O2	AR	P10275	CRBN	WO-2024189488-A1
TPD-BY67MM	SCHEMBL31198687	4-chloro-7-[4-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-1H-indole-3-carbonitrile	COc1cc(N2CCN(CC3CCN(c4ccc(C5CCN(c6ccc(Cl)c7c(C#N)c[nH]c67)CC5)cc4)CC3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C44H49ClN8O4	AR	P10275	CRBN	WO-2024189488-A1
TPD-6TDBQ9	SCHEMBL31198690	7-[4-[4-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-4-methyl-1H-indole-3-carbonitrile	Cc1ccc(N2CCC(c3ccc(N4CCC(CN5CCC(n6ccc7c(N8CCC(=O)NC8=O)cccc76)CC5)CC4)cc3)CC2)c2[nH]cc(C#N)c12	C44H50N8O2	AR	P10275	CRBN	WO-2024189488-A1
TPD-DYSPUB	WO2024189488A1_9	.	N#Cc1n[nH]c2c(N3CCCC(c4ccc(N5CCC(CN6CCC(n7ccc8c(N9CCC(=O)NC9=O)cccc87)CC6)CC5)cc4)C3)ccc(Cl)c12	C42H46ClN9O2	AR	P10275	CRBN	WO-2024189488-A1
TPD-H683NI	SCHEMBL31198619	4-chloro-7-[(3S)-3-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-1H-indazole-3-carbonitrile	N#Cc1n[nH]c2c(N3CCC[C@@H](c4ccc(N5CCC(CN6CCN(c7ccc8c(c7)CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)cc4)C3)ccc(Cl)c12	C42H46ClN9O3	AR	P10275	CRBN	WO-2024189488-A1
TPD-FDKRO1	WO2024189488A1_11	.	N#Cc1c[nH]c2c(N3CCCC(c4ccc(N5CCC(CN6CCC(n7ccc8c(N9CCC(=O)NC9=O)cccc87)CC6)CC5)cc4)C3)ccc(Cl)c12	C43H47ClN8O2	AR	P10275	CRBN	WO-2024189488-A1
TPD-KC9832	SCHEMBL31198608	4-chloro-7-[(3S)-3-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-1H-indole-3-carbonitrile	N#Cc1c[nH]c2c(N3CCC[C@@H](c4ccc(N5CCC(CN6CCN(c7ccc8c(c7)CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)cc4)C3)ccc(Cl)c12	C43H47ClN8O3	AR	P10275	CRBN	WO-2024189488-A1
TPD-A6RRP0	SCHEMBL31198695	4-chloro-7-[(3S)-3-[4-[4-[[4-[6-(2,4-dioxo-1,3-diazinan-1-yl)-1-methylindol-2-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-1H-indole-3-carbonitrile	Cn1c(C2CCN(CC3CCN(c4ccc([C@@H]5CCCN(c6ccc(Cl)c7c(C#N)c[nH]c67)C5)cc4)CC3)CC2)cc2ccc(N3CCC(=O)NC3=O)cc21	C44H49ClN8O2	AR	P10275	CRBN	WO-2024189488-A1
TPD-WRK41H	SCHEMBL31198550	4-chloro-7-[(3S)-3-[4-[4-[[4-[6-(2,4-dioxo-1,3-diazinan-1-yl)-1-methylindol-2-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-1H-indazole-3-carbonitrile; AZD9750; EX-A13467; 3056515-10-4	Cn1c(C2CCN(CC3CCN(c4ccc([C@@H]5CCCN(c6ccc(Cl)c7c(C#N)n[nH]c67)C5)cc4)CC3)CC2)cc2ccc(N3CCC(=O)NC3=O)cc21	C43H48ClN9O2	AR	P10275	CRBN	WO-2024189488-A1
TPD-DD49NA	SCHEMBL31198622	7-[4-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-4-methyl-1H-indole-3-carbonitrile	COc1cc(N2CCN(CC3CCN(c4ccc(C5CCN(c6ccc(C)c7c(C#N)c[nH]c67)CC5)cc4)CC3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C45H52N8O4	AR	P10275	CRBN	WO-2024189488-A1
TPD-CQQ88E	SCHEMBL31198542	4-chloro-7-[4-[4-[4-[[4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-7-methoxy-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-1H-indole-3-carbonitrile	COc1cc(N2CCN(CC3CCN(c4ccc(C5CCN(c6ccc(Cl)c7c(C#N)c[nH]c67)CC5)cc4)CC3)CC2)cc2c1C(=O)N([C@H]1CCC(=O)NC1=O)C2	C44H49ClN8O4	AR	P10275	CRBN	WO-2024189488-A1
TPD-42NQCD	SCHEMBL31198594	4-chloro-7-[4-[4-[4-[[4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-1H-indole-3-carbonitrile	N#Cc1c[nH]c2c(N3CCC(c4ccc(N5CCC(CN6CCN(c7ccc8c(c7)CN([C@H]7CCC(=O)NC7=O)C8=O)CC6)CC5)cc4)CC3)ccc(Cl)c12	C43H47ClN8O3	AR	P10275	CRBN	WO-2024189488-A1
TPD-EBVIK3	SCHEMBL31198614	7-[4-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-4-fluoro-1H-indole-3-carbonitrile	COc1cc(N2CCN(CC3CCN(c4ccc(C5CCN(c6ccc(F)c7c(C#N)c[nH]c67)CC5)cc4)CC3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C44H49FN8O4	AR	P10275	CRBN	WO-2024189488-A1
TPD-1Y1HZ5	SCHEMBL31198626	4-chloro-7-[(3R)-3-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-1H-indole-3-carbonitrile	N#Cc1c[nH]c2c(N3CCC[C@H](c4ccc(N5CCC(CN6CCN(c7ccc8c(c7)CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)cc4)C3)ccc(Cl)c12	C43H47ClN8O3	AR	P10275	CRBN	WO-2024189488-A1
TPD-QNWTZA	SCHEMBL31198629	7-[4-[4-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]phenyl]piperidin-1-yl]-4-fluoro-1H-indole-3-carbonitrile	N#Cc1c[nH]c2c(N3CCC(c4ccc(N5CCN(CC6CCN(c7ccc8c(c7)CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)cc4)CC3)ccc(F)c12	C43H47FN8O3	AR	P10275	CRBN	WO-2024189488-A1
TPD-F7FIFO	SCHEMBL31198675	7-[(3S)-3-[4-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-4-fluoro-1H-indole-3-carbonitrile	N#Cc1c[nH]c2c(N3CCC[C@@H](c4ccc(N5CCC(CN6CCC(n7ccc8c(N9CCC(=O)NC9=O)cccc87)CC6)CC5)cc4)C3)ccc(F)c12	C43H47FN8O2	AR	P10275	CRBN	WO-2024189488-A1
TPD-ZAX8FK	SCHEMBL31198650	7-[(3S)-3-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-4-fluoro-1H-indole-3-carbonitrile	N#Cc1c[nH]c2c(N3CCC[C@@H](c4ccc(N5CCC(CN6CCN(c7ccc8c(c7)CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)cc4)C3)ccc(F)c12	C43H47FN8O3	AR	P10275	CRBN	WO-2024189488-A1
TPD-ZRGZVD	SCHEMBL31198532	4-chloro-7-[(3R)-3-[4-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-1H-indazole-3-carbonitrile	N#Cc1n[nH]c2c(N3CCC[C@H](c4ccc(N5CCC(CN6CCC(n7ccc8c(N9CCC(=O)NC9=O)cccc87)CC6)CC5)cc4)C3)ccc(Cl)c12	C42H46ClN9O2	AR	P10275	CRBN	WO-2024189488-A1
TPD-H5T59G	SCHEMBL31198642	4-chloro-7-[(3R)-3-[4-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-1H-indole-3-carbonitrile	N#Cc1c[nH]c2c(N3CCC[C@H](c4ccc(N5CCC(CN6CCC(n7ccc8c(N9CCC(=O)NC9=O)cccc87)CC6)CC5)cc4)C3)ccc(Cl)c12	C43H47ClN8O2	AR	P10275	CRBN	WO-2024189488-A1
TPD-NJ0FNF	SCHEMBL31198667	7-[4-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]butoxy]phenyl]piperidin-1-yl]-4-methyl-1H-indole-3-carbonitrile	COc1cc(N2CCN(CCCCOc3ccc(C4CCN(c5ccc(C)c6c(C#N)c[nH]c56)CC4)cc3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C43H49N7O5	AR	P10275	CRBN	WO-2024189488-A1
TPD-AXLB88	SCHEMBL31198658	7-[4-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]butoxy]phenyl]piperidin-1-yl]-4-methyl-1H-indole-3-carbonitrile	Cc1ccc(N2CCC(c3ccc(OCCCCN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)cc3)CC2)c2[nH]cc(C#N)c12	C42H47N7O4	AR	P10275	CRBN	WO-2024189488-A1
TPD-OYWEH4	SCHEMBL31198558	7-[4-[4-[4-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]butoxy]phenyl]piperidin-1-yl]-4-methyl-1H-indole-3-carbonitrile	Cc1ccc(N2CCC(c3ccc(OCCCCN4CCC(n5ccc6c(N7CCC(=O)NC7=O)cccc65)CC4)cc3)CC2)c2[nH]cc(C#N)c12	C42H47N7O3	AR	P10275	CRBN	WO-2024189488-A1
TPD-QQ6BXN	SCHEMBL31198674	7-[4-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-4-methoxy-3-oxo-1H-pyrrolo[3,4-c]pyridin-6-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-4-methyl-1H-indole-3-carbonitrile	COc1nc(N2CCN(CC3CCN(c4ccc(C5CCN(c6ccc(C)c7c(C#N)c[nH]c67)CC5)cc4)CC3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C44H51N9O4	AR	P10275	CRBN	WO-2024189488-A1
TPD-7YWMB8	SCHEMBL31198632	7-[4-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-4-methoxy-3-oxo-1H-pyrrolo[3,4-c]pyridin-6-yl]piperazin-1-yl]butoxy]phenyl]piperidin-1-yl]-4-methyl-1H-indole-3-carbonitrile	COc1nc(N2CCN(CCCCOc3ccc(C4CCN(c5ccc(C)c6c(C#N)c[nH]c56)CC4)cc3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C42H48N8O5	AR	P10275	CRBN	WO-2024189488-A1
TPD-ZT2ORX	SCHEMBL31198649	4-chloro-7-[4-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-4-methoxy-3-oxo-1H-pyrrolo[3,4-c]pyridin-6-yl]piperazin-1-yl]butoxy]phenyl]piperidin-1-yl]-1H-indole-3-carbonitrile	COc1nc(N2CCN(CCCCOc3ccc(C4CCN(c5ccc(Cl)c6c(C#N)c[nH]c56)CC4)cc3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C41H45ClN8O5	AR	P10275	CRBN	WO-2024189488-A1
TPD-L81KV8	SCHEMBL31198570	7-[4-[4-[4-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]butoxy]phenyl]piperidin-1-yl]-4-fluoro-1H-indole-3-carbonitrile	N#Cc1c[nH]c2c(N3CCC(c4ccc(OCCCCN5CCC(n6ccc7c(N8CCC(=O)NC8=O)cccc76)CC5)cc4)CC3)ccc(F)c12	C41H44FN7O3	AR	P10275	CRBN	WO-2024189488-A1
TPD-ECFTAM	SCHEMBL31198685	4-chloro-7-[4-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-4-methoxy-3-oxo-1H-pyrrolo[3,4-c]pyridin-6-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-1H-indole-3-carbonitrile	COc1nc(N2CCN(CC3CCN(c4ccc(C5CCN(c6ccc(Cl)c7c(C#N)c[nH]c67)CC5)cc4)CC3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C43H48ClN9O4	AR	P10275	CRBN	WO-2024189488-A1
TPD-Y0JTE7	SCHEMBL31198566	4-chloro-7-[4-[4-[4-[[4-[2-[(3R)-2,6-dioxopiperidin-3-yl]-4-methoxy-3-oxo-1H-pyrrolo[3,4-c]pyridin-6-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-1H-indole-3-carbonitrile	COc1nc(N2CCN(CC3CCN(c4ccc(C5CCN(c6ccc(Cl)c7c(C#N)c[nH]c67)CC5)cc4)CC3)CC2)cc2c1C(=O)N([C@@H]1CCC(=O)NC1=O)C2	C43H48ClN9O4	AR	P10275	CRBN	WO-2024189488-A1
TPD-YYHQ5E	WO2024189488A1_36	.	COc1nc(N2CCN(CC3CCN(c4ccc(C5CCN(c6ccc(Cl)c7c(C#N)c[nH]c67)CC5)cc4)CC3)CC2)cc2c1C(=O)N([C@H]1CCC(=O)NC1=O)C2	C43H48ClN9O4	AR	P10275	CRBN	WO-2024189488-A1
TPD-Y7QO6T	SCHEMBL31198623	7-[4-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-4-methoxy-3-oxo-1H-pyrrolo[3,4-c]pyridin-6-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-4-fluoro-1H-indole-3-carbonitrile	COc1nc(N2CCN(CC3CCN(c4ccc(C5CCN(c6ccc(F)c7c(C#N)c[nH]c67)CC5)cc4)CC3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C43H48FN9O4	AR	P10275	CRBN	WO-2024189488-A1
TPD-GWN0P9	SCHEMBL31198588	4-chloro-7-[(3S)-3-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-4-methoxy-3-oxo-1H-pyrrolo[3,4-c]pyridin-6-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-1H-indole-3-carbonitrile	COc1nc(N2CCN(CC3CCN(c4ccc([C@@H]5CCCN(c6ccc(Cl)c7c(C#N)c[nH]c67)C5)cc4)CC3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C43H48ClN9O4	AR	P10275	CRBN	WO-2024189488-A1
TPD-IOQT0R	WO2024189488A1_40	.	COc1nc(N2CCN(CC3CCN(c4ccc([C@@H]5CCCN(c6ccc(Cl)c7c(C#N)c[nH]c67)C5)cc4)CC3)CC2)cc2c1C(=O)N([C@H]1CCC(=O)NC1=O)C2	C43H48ClN9O4	AR	P10275	CRBN	WO-2024189488-A1
TPD-NCUJI4	SCHEMBL31198615	7-[4-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]-2-fluorophenyl]piperidin-1-yl]-4-methyl-1H-indole-3-carbonitrile	COc1cc(N2CCN(CC3CCN(c4ccc(C5CCN(c6ccc(C)c7c(C#N)c[nH]c67)CC5)c(F)c4)CC3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C45H51FN8O4	AR	P10275	CRBN	WO-2024189488-A1
TPD-X52H79	SCHEMBL31198662	7-[4-[4-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]-2-fluorophenyl]piperidin-1-yl]-4-methyl-1H-indole-3-carbonitrile	Cc1ccc(N2CCC(c3ccc(N4CCC(CN5CCC(n6ccc7c(N8CCC(=O)NC8=O)cccc76)CC5)CC4)cc3F)CC2)c2[nH]cc(C#N)c12	C44H49FN8O2	AR	P10275	CRBN	WO-2024189488-A1
TPD-7BO4UW	SCHEMBL31198659	7-[4-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]-2-fluorophenyl]piperidin-1-yl]-4-methyl-1H-indole-3-carbonitrile	COc1cc(N2CCN(CC3CCN(c4ccc(C5CCN(c6ccc(C)c7c(C#N)c[nH]c67)CC5)c(F)c4)CC3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O	C45H49FN8O5	AR	P10275	CRBN	WO-2024189488-A1
TPD-B99HGC	SCHEMBL31198606	7-[4-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]butoxy]phenyl]piperidin-1-yl]-4-fluoro-1H-indole-3-carbonitrile	N#Cc1c[nH]c2c(N3CCC(c4ccc(OCCCCN5CCN(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC5)cc4)CC3)ccc(F)c12	C41H44FN7O4	AR	P10275	CRBN	WO-2024189488-A1
TPD-LCGG6T	SCHEMBL31198648	4-chloro-7-[4-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]butoxy]phenyl]piperidin-1-yl]-1H-indole-3-carbonitrile	N#Cc1c[nH]c2c(N3CCC(c4ccc(OCCCCN5CCN(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC5)cc4)CC3)ccc(Cl)c12	C41H44ClN7O4	AR	P10275	CRBN	WO-2024189488-A1
TPD-BUJCH4	SCHEMBL31198709	4-chloro-7-[4-[4-[4-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]butoxy]phenyl]piperidin-1-yl]-1H-indole-3-carbonitrile	N#Cc1c[nH]c2c(N3CCC(c4ccc(OCCCCN5CCC(n6ccc7c(N8CCC(=O)NC8=O)cccc76)CC5)cc4)CC3)ccc(Cl)c12	C41H44ClN7O3	AR	P10275	CRBN	WO-2024189488-A1
TPD-N237VU	SCHEMBL31198561	4-chloro-7-[(3R)-3-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-4-methoxy-3-oxo-1H-pyrrolo[3,4-c]pyridin-6-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-1H-indole-3-carbonitrile	COc1nc(N2CCN(CC3CCN(c4ccc([C@H]5CCCN(c6ccc(Cl)c7c(C#N)c[nH]c67)C5)cc4)CC3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C43H48ClN9O4	AR	P10275	CRBN	WO-2024189488-A1
TPD-934CHS	SCHEMBL31198575	7-[4-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1,3-dioxoisoindol-5-yl]piperazin-1-yl]butoxy]phenyl]piperidin-1-yl]-4-methyl-1H-indole-3-carbonitrile	COc1cc(N2CCN(CCCCOc3ccc(C4CCN(c5ccc(C)c6c(C#N)c[nH]c56)CC4)cc3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O	C43H47N7O6	AR	P10275	CRBN	WO-2024189488-A1
TPD-99IJ35	SCHEMBL31198567	4-chloro-7-[4-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-1H-indole-3-carbonitrile	COc1cc(N2CCN(CC3CCN(c4ccc(C5CCN(c6ccc(Cl)c7c(C#N)c[nH]c67)CC5)cc4)CC3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O	C44H47ClN8O5	AR	P10275	CRBN	WO-2024189488-A1
TPD-X2Y0U9	SCHEMBL31198612	7-[4-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]butoxy]phenyl]piperidin-1-yl]-4-methyl-1H-indole-3-carbonitrile	Cc1ccc(N2CCC(c3ccc(OCCCCN4CCN(c5cc6c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)cc3)CC2)c2[nH]cc(C#N)c12	C42H44FN7O5	AR	P10275	CRBN	WO-2024189488-A1
TPD-PTZGVX	SCHEMBL31198603	4-chloro-7-[4-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-1H-indole-3-carbonitrile	N#Cc1c[nH]c2c(N3CCC(c4ccc(N5CCC(CN6CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)cc4)CC3)ccc(Cl)c12	C43H44ClFN8O4	AR	P10275	CRBN	WO-2024189488-A1
TPD-53YT2K	SCHEMBL31198578	7-[4-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-4-fluoro-1H-indole-3-carbonitrile	N#Cc1c[nH]c2c(N3CCC(c4ccc(N5CCC(CN6CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)cc4)CC3)ccc(F)c12	C43H44F2N8O4	AR	P10275	CRBN	WO-2024189488-A1
TPD-0XQLNR	SCHEMBL31198677	4-chloro-7-[(3S)-3-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-1H-indole-3-carbonitrile	N#Cc1c[nH]c2c(N3CCC[C@@H](c4ccc(N5CCC(CN6CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)cc4)C3)ccc(Cl)c12	C43H44ClFN8O4	AR	P10275	CRBN	WO-2024189488-A1
TPD-PEWO50	SCHEMBL31198704	4-chloro-7-[(3R)-3-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-1H-indole-3-carbonitrile	N#Cc1c[nH]c2c(N3CCC[C@H](c4ccc(N5CCC(CN6CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)cc4)C3)ccc(Cl)c12	C43H44ClFN8O4	AR	P10275	CRBN	WO-2024189488-A1
TPD-M3LJ7O	SCHEMBL31198547	4-chloro-7-[4-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-1H-indole-3-carbonitrile	N#Cc1c[nH]c2c(N3CCC(c4ccc(N5CCC(CN6CCN(c7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)cc4)CC3)ccc(Cl)c12	C43H45ClN8O4	AR	P10275	CRBN	WO-2024189488-A1
TPD-Z2VFBG	SCHEMBL31198670	7-[4-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]butoxy]phenyl]piperidin-1-yl]-4-methyl-1H-indole-3-carbonitrile	Cc1ccc(N2CCC(c3ccc(OCCCCN4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)cc3)CC2)c2[nH]cc(C#N)c12	C42H45N7O5	AR	P10275	CRBN	WO-2024189488-A1
TPD-LPY21B	SCHEMBL31198611	7-[4-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]butoxy]phenyl]piperidin-1-yl]-1H-indole-3-carbonitrile	N#Cc1c[nH]c2c(N3CCC(c4ccc(OCCCCN5CCN(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC5)cc4)CC3)cccc12	C41H45N7O4	AR	P10275	CRBN	WO-2024189488-A1
TPD-2KZHNJ	SCHEMBL31198625	7-[4-[4-[4-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]butoxy]phenyl]piperidin-1-yl]-1H-indole-3-carbonitrile	N#Cc1c[nH]c2c(N3CCC(c4ccc(OCCCCN5CCC(n6ccc7c(N8CCC(=O)NC8=O)cccc76)CC5)cc4)CC3)cccc12	C41H45N7O3	AR	P10275	CRBN	WO-2024189488-A1
TPD-RNLTAV	SCHEMBL31198536	7-[4-[4-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-1H-indole-3-carbonitrile	N#Cc1c[nH]c2c(N3CCC(c4ccc(N5CCC(CN6CCC(n7ccc8c(N9CCC(=O)NC9=O)cccc87)CC6)CC5)cc4)CC3)cccc12	C43H48N8O2	AR	P10275	CRBN	WO-2024189488-A1
TPD-ZWYK6R	SCHEMBL31198586	4-chloro-7-[4-[5-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]pyridin-2-yl]piperidin-1-yl]-1H-indole-3-carbonitrile	COc1cc(N2CCN(CC3CCN(c4ccc(C5CCN(c6ccc(Cl)c7c(C#N)c[nH]c67)CC5)nc4)CC3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C43H48ClN9O4	AR	P10275	CRBN	WO-2024189488-A1
TPD-QF5LF4	SCHEMBL31198651	4-chloro-7-[4-[5-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-4-methoxy-3-oxo-1H-pyrrolo[3,4-c]pyridin-6-yl]piperazin-1-yl]methyl]piperidin-1-yl]pyridin-2-yl]piperidin-1-yl]-1H-indole-3-carbonitrile	COc1nc(N2CCN(CC3CCN(c4ccc(C5CCN(c6ccc(Cl)c7c(C#N)c[nH]c67)CC5)nc4)CC3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C42H47ClN10O4	AR	P10275	CRBN	WO-2024189488-A1
TPD-V60PUM	SCHEMBL31198700	4-chloro-7-[4-[5-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridin-2-yl]piperidin-1-yl]-1H-indole-3-carbonitrile	N#Cc1c[nH]c2c(N3CCC(c4ccc(N5CCC(CN6CCC(n7ccc8c(N9CCC(=O)NC9=O)cccc87)CC6)CC5)cn4)CC3)ccc(Cl)c12	C42H46ClN9O2	AR	P10275	CRBN	WO-2024189488-A1
TPD-3SRZEJ	SCHEMBL31198568	4-chloro-7-[4-[6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridazin-3-yl]piperidin-1-yl]-1H-indole-3-carbonitrile	N#Cc1c[nH]c2c(N3CCC(c4ccc(N5CCC(CN6CCC(n7ccc8c(N9CCC(=O)NC9=O)cccc87)CC6)CC5)nn4)CC3)ccc(Cl)c12	C41H45ClN10O2	AR	P10275	CRBN	WO-2024189488-A1
TPD-D910XJ	SCHEMBL31198628	4-chloro-7-[4-[6-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]pyridazin-3-yl]piperidin-1-yl]-1H-indole-3-carbonitrile	N#Cc1c[nH]c2c(N3CCC(c4ccc(N5CCC(CN6CCN(c7ccc8c(c7)CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)nn4)CC3)ccc(Cl)c12	C41H45ClN10O3	AR	P10275	CRBN	WO-2024189488-A1
TPD-C8DVIF	WO2024189488A1_66	.	N#Cc1c[nH]c2c(N3CCC[C@H](c4ccc(N5CCC(CN6CCC(n7ccc8c(N9CCC(=O)NC9=O)cccc87)CC6)CC5)cn4)C3)ccc(Cl)c12	C42H46ClN9O2	AR	P10275	CRBN	WO-2024189488-A1
TPD-YT4TAQ	SCHEMBL31198585	4-chloro-7-[4-[5-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyrazin-2-yl]piperidin-1-yl]-1H-indole-3-carbonitrile	N#Cc1c[nH]c2c(N3CCC(c4cnc(N5CCC(CN6CCC(n7ccc8c(N9CCC(=O)NC9=O)cccc87)CC6)CC5)cn4)CC3)ccc(Cl)c12	C41H45ClN10O2	AR	P10275	CRBN	WO-2024189488-A1
TPD-S8JGK1	SCHEMBL31198616	4-chloro-7-[4-[5-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]pyrazin-2-yl]piperidin-1-yl]-1H-indole-3-carbonitrile	N#Cc1c[nH]c2c(N3CCC(c4cnc(N5CCC(CN6CCN(c7ccc8c(c7)CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)cn4)CC3)ccc(Cl)c12	C41H45ClN10O3	AR	P10275	CRBN	WO-2024189488-A1
TPD-EG4485	SCHEMBL31198702	7-[4-[4-[4-[[4-[[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-4-yl]methyl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-4-methyl-1H-indole-3-carbonitrile	Cc1ccc(N2CCC(c3ccc(N4CCC(CN5CCN(Cc6cccc7c6n(C)c(=O)n7C6CCC(=O)NC6=O)CC5)CC4)cc3)CC2)c2[nH]cc(C#N)c12	C45H53N9O3	AR	P10275	CRBN	WO-2024189488-A1
TPD-4VY0I0	SCHEMBL31198604	4-chloro-7-[4-[4-[4-[[4-[[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-4-yl]methyl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-1H-indole-3-carbonitrile	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(CN3CCN(CC4CCN(c5ccc(C6CCN(c7ccc(Cl)c8c(C#N)c[nH]c78)CC6)cc5)CC4)CC3)c21	C44H50ClN9O3	AR	P10275	CRBN	WO-2024189488-A1
TPD-9NY1AW	SCHEMBL31198630	7-[4-[4-[4-[[4-[[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-4-yl]methyl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-4-fluoro-1H-indole-3-carbonitrile	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(CN3CCN(CC4CCN(c5ccc(C6CCN(c7ccc(F)c8c(C#N)c[nH]c78)CC6)cc5)CC4)CC3)c21	C44H50FN9O3	AR	P10275	CRBN	WO-2024189488-A1
TPD-3BRCEL	SCHEMBL31198599	4-chloro-7-[4-[4-[4-[[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-4-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-1H-indole-3-carbonitrile	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(N3CCN(CC4CCN(c5ccc(C6CCN(c7ccc(Cl)c8c(C#N)c[nH]c78)CC6)cc5)CC4)CC3)c21	C43H48ClN9O3	AR	P10275	CRBN	WO-2024189488-A1
TPD-2A0YIS	SCHEMBL31198680	4-chloro-7-[(3S)-3-[4-[4-[[4-[[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-4-yl]methyl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-1H-indole-3-carbonitrile	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(CN3CCN(CC4CCN(c5ccc([C@@H]6CCCN(c7ccc(Cl)c8c(C#N)c[nH]c78)C6)cc5)CC4)CC3)c21	C44H50ClN9O3	AR	P10275	CRBN	WO-2024189488-A1
TPD-JXBBII	SCHEMBL31198621	7-[(3S)-3-[4-[4-[[4-[[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-4-yl]methyl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-4-fluoro-1H-indole-3-carbonitrile	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(CN3CCN(CC4CCN(c5ccc([C@@H]6CCCN(c7ccc(F)c8c(C#N)c[nH]c78)C6)cc5)CC4)CC3)c21	C44H50FN9O3	AR	P10275	CRBN	WO-2024189488-A1
TPD-HTC439	SCHEMBL31198638	4-chloro-7-[4-[4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-1H-indole-3-carbonitrile	N#Cc1c[nH]c2c(N3CCC(c4ccc(N5CCC(CN6Cc7cc8c(cc7C6)C(=O)N(C6CCC(=O)NC6=O)C8=O)CC5)cc4)CC3)ccc(Cl)c12	C41H40ClN7O4	AR	P10275	CRBN	WO-2024189488-A1
TPD-KNGYEK	SCHEMBL31198593	4-chloro-7-[(3S)-3-[4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-1H-indazole-3-carbonitrile	N#Cc1n[nH]c2c(N3CCC[C@@H](c4ccc(N5CCC(CN6Cc7cc8c(cc7C6)C(=O)N(C6CCC(=O)NC6=O)C8=O)CC5)cc4)C3)ccc(Cl)c12	C40H39ClN8O4	AR	P10275	CRBN	WO-2024189488-A1
TPD-5DCEJV	SCHEMBL31198694	4-chloro-7-[(3S)-3-[4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-1H-indole-3-carbonitrile	N#Cc1c[nH]c2c(N3CCC[C@@H](c4ccc(N5CCC(CN6Cc7cc8c(cc7C6)C(=O)N(C6CCC(=O)NC6=O)C8=O)CC5)cc4)C3)ccc(Cl)c12	C41H40ClN7O4	AR	P10275	CRBN	WO-2024189488-A1
TPD-284Y5X	WO2024189488A1_79	7-[1-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]butoxy]phenyl]piperidin-3-yl]-4-methyl-1H-indole-3-carbonitrile	Cc1ccc(C2CCCN(c3ccc(OCCCCN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)cc3)C2)c2[nH]cc(C#N)c12	C42H47N7O4	AR	P10275	CRBN	WO-2024189488-A1
TPD-4DR899	SCHEMBL31198569	7-[(3S)-1-[3-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]butoxy]phenyl]piperidin-3-yl]-4-methyl-1H-indole-3-carbonitrile	Cc1ccc([C@@H]2CCCN(c3cccc(OCCCCN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)c3)C2)c2[nH]cc(C#N)c12	C42H47N7O4	AR	P10275	CRBN	WO-2024189488-A1
TPD-9UL8LB	WO2024189488A1_83	7-[1-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-3-yl]-4-methyl-1H-indole-3-carbonitrile	Cc1ccc(C2CCCN(c3ccc(N4CCC(CN5CCN(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cc3)C2)c2[nH]cc(C#N)c12	C44H50N8O3	AR	P10275	CRBN	WO-2024189488-A1
TPD-HC14L8	SCHEMBL31198589	4-chloro-7-[4-[4-[4-[[4-[6-(2,4-dioxo-1,3-diazinan-1-yl)-1-methylindol-2-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-1H-indole-3-carbonitrile	Cn1c(C2CCN(CC3CCN(c4ccc(C5CCN(c6ccc(Cl)c7c(C#N)c[nH]c67)CC5)cc4)CC3)CC2)cc2ccc(N3CCC(=O)NC3=O)cc21	C44H49ClN8O2	AR	P10275	CRBN	WO-2024189488-A1
TPD-46JT3C	SCHEMBL31198697	4-chloro-7-[4-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]piperidine-1-carbonyl]phenyl]piperidin-1-yl]-1H-indole-3-carbonitrile	N#Cc1c[nH]c2c(N3CCC(c4ccc(C(=O)N5CCC(CN6CCN(c7ccc8c(c7)CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)cc4)CC3)ccc(Cl)c12	C44H47ClN8O4	AR	P10275	CRBN	WO-2024189488-A1
TPD-07QDLI	SCHEMBL31198587	4-chloro-7-[4-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-4-methoxy-3-oxo-1H-pyrrolo[3,4-c]pyridin-6-yl]piperazin-1-yl]piperidin-1-yl]phenyl]piperidin-1-yl]-1H-indole-3-carbonitrile	COc1nc(N2CCN(C3CCN(c4ccc(C5CCN(c6ccc(Cl)c7c(C#N)c[nH]c67)CC5)cc4)CC3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C42H46ClN9O4	AR	P10275	CRBN	WO-2024189488-A1
TPD-K9SGBX	SCHEMBL31198546	4-chloro-7-[4-[4-[4-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-4-methoxy-3-oxo-1H-pyrrolo[3,4-c]pyridin-6-yl]piperazin-1-yl]ethyl]piperidin-1-yl]phenyl]piperidin-1-yl]-1H-indole-3-carbonitrile	COc1nc(N2CCN(CCC3CCN(c4ccc(C5CCN(c6ccc(Cl)c7c(C#N)c[nH]c67)CC5)cc4)CC3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C44H50ClN9O4	AR	P10275	CRBN	WO-2024189488-A1
TPD-ITUTZ6	SCHEMBL31198554	4-chloro-7-[4-[4-[4-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-4-methoxy-3-oxo-1H-pyrrolo[3,4-c]pyridin-6-yl]piperazin-1-yl]propyl]piperidin-1-yl]phenyl]piperidin-1-yl]-1H-indole-3-carbonitrile	COc1nc(N2CCN(CCCC3CCN(c4ccc(C5CCN(c6ccc(Cl)c7c(C#N)c[nH]c67)CC5)cc4)CC3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C45H52ClN9O4	AR	P10275	CRBN	WO-2024189488-A1
TPD-O4NV86	SCHEMBL31198571	7-[4-[4-[4-[[4-[5-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-4-fluoro-1H-indole-3-carbonitrile	N#Cc1c[nH]c2c(N3CCC(c4ccc(N5CCC(CN6CCC(n7ccc8cc(N9CCC(=O)NC9=O)ccc87)CC6)CC5)cc4)CC3)ccc(F)c12	C43H47FN8O2	AR	P10275	CRBN	WO-2024189488-A1
TPD-G3YD2T	SCHEMBL31198613	4-chloro-7-[4-[4-[4-[[4-[5-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-1H-indole-3-carbonitrile	N#Cc1c[nH]c2c(N3CCC(c4ccc(N5CCC(CN6CCC(n7ccc8cc(N9CCC(=O)NC9=O)ccc87)CC6)CC5)cc4)CC3)ccc(Cl)c12	C43H47ClN8O2	AR	P10275	CRBN	WO-2024189488-A1
TPD-7QPC9C	WO2024189488A1_92	4-chloro-7-[1-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-4-methoxy-3-oxo-1H-pyrrolo[3,4-c]pyridin-6-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-3-yl]-1H-indole-3-carbonitrile	COc1nc(N2CCN(CC3CCN(c4ccc(N5CCCC(c6ccc(Cl)c7c(C#N)c[nH]c67)C5)cc4)CC3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C43H48ClN9O4	AR	P10275	CRBN	WO-2024189488-A1
TPD-5BYWN3	WO2024189488A1_94	4-chloro-7-[1-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-3-yl]-1H-indole-3-carbonitrile	N#Cc1c[nH]c2c(C3CCCN(c4ccc(N5CCC(CN6CCN(c7ccc8c(c7)CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)cc4)C3)ccc(Cl)c12	C43H47ClN8O3	AR	P10275	CRBN	WO-2024189488-A1
TPD-OB2IG5	SCHEMBL31198581	7-[4-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]butoxy]phenyl]piperazin-1-yl]-4-methyl-1H-indole-3-carbonitrile	Cc1ccc(N2CCN(c3ccc(OCCCCN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)cc3)CC2)c2[nH]cc(C#N)c12	C41H46N8O4	AR	P10275	CRBN	WO-2024189488-A1
TPD-HEFDL2	WO2024189488A1_97	.	N#Cc1c[nH]c2c(C3CCCN(c4ccc(C5CCN(CC6CCN(c7ccc8c(c7)CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)cc4)C3)ccc(Cl)c12	C44H48ClN7O3	AR	P10275	CRBN	WO-2024189488-A1
TPD-0UYRNP	WO2024189488A1_98	.	COc1nc(N2CCC(CN3CCC(c4ccc(N5CCCC(c6ccc(Cl)c7c(C#N)c[nH]c67)C5)cc4)CC3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C44H49ClN8O4	AR	P10275	CRBN	WO-2024189488-A1
TPD-GCNKRH	SCHEMBL31198627	4-chloro-7-[4-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidine-1-carbonyl]phenyl]piperidin-1-yl]-1H-indole-3-carbonitrile	N#Cc1c[nH]c2c(N3CCC(c4ccc(C(=O)N5CCC(CN6CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)cc4)CC3)ccc(Cl)c12	C44H44ClFN8O5	AR	P10275	CRBN	WO-2024189488-A1
TPD-O44L43	SCHEMBL31198708	7-[4-[4-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperidin-4-yl]oxyphenyl]piperidin-1-yl]-4-fluoro-1H-indole-3-carbonitrile	N#Cc1c[nH]c2c(N3CCC(c4ccc(OC5CCN(CC6CCN(c7ccc8c(c7)CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)cc4)CC3)ccc(F)c12	C44H48FN7O4	AR	P10275	CRBN	WO-2024189488-A1
TPD-T04RJV	SCHEMBL31198711	4-chloro-7-[4-[4-[4-[[4-[5-(2,4-dioxo-1,3-diazinan-1-yl)-7-methylindol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-1H-indole-3-carbonitrile	Cc1cc(N2CCC(=O)NC2=O)cc2ccn(C3CCN(CC4CCN(c5ccc(C6CCN(c7ccc(Cl)c8c(C#N)c[nH]c78)CC6)cc5)CC4)CC3)c12	C44H49ClN8O2	AR	P10275	CRBN	WO-2024189488-A1
TPD-VXDHIT	SCHEMBL31198656	4-chloro-7-[4-[4-[4-[[4-[6-(2,4-dioxo-1,3-diazinan-1-yl)-1-methylpyrrolo[3,2-b]pyridin-2-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-1H-indole-3-carbonitrile	Cn1c(C2CCN(CC3CCN(c4ccc(C5CCN(c6ccc(Cl)c7c(C#N)c[nH]c67)CC5)cc4)CC3)CC2)cc2ncc(N3CCC(=O)NC3=O)cc21	C43H48ClN9O2	AR	P10275	CRBN	WO-2024189488-A1
TPD-M67VON	SCHEMBL31198602	4-[4-[[1-[4-[(3S)-1-(4-chloro-3-cyano-1H-indol-7-yl)piperidin-3-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-N-(2,6-dioxopiperidin-3-yl)-2-fluorobenzamide	N#Cc1c[nH]c2c(N3CCC[C@@H](c4ccc(N5CCC(CN6CCN(c7ccc(C(=O)NC8CCC(=O)NC8=O)c(F)c7)CC6)CC5)cc4)C3)ccc(Cl)c12	C42H46ClFN8O3	AR	P10275	CRBN	WO-2024189488-A1
TPD-Y4USCF	SCHEMBL31198698	4-[4-[[1-[4-[1-(3-cyano-4-fluoro-1H-indol-7-yl)piperidin-4-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-N-(2,6-dioxopiperidin-3-yl)-2-fluorobenzamide	N#Cc1c[nH]c2c(N3CCC(c4ccc(N5CCC(CN6CCN(c7ccc(C(=O)NC8CCC(=O)NC8=O)c(F)c7)CC6)CC5)cc4)CC3)ccc(F)c12	C42H46F2N8O3	AR	P10275	CRBN	WO-2024189488-A1
TPD-X8TQHK	SCHEMBL31198552	4-[4-[[1-[4-[1-(4-chloro-3-cyano-1H-indol-7-yl)piperidin-4-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-N-(2,6-dioxopiperidin-3-yl)-2-fluorobenzamide	N#Cc1c[nH]c2c(N3CCC(c4ccc(N5CCC(CN6CCN(c7ccc(C(=O)NC8CCC(=O)NC8=O)c(F)c7)CC6)CC5)cc4)CC3)ccc(Cl)c12	C42H46ClFN8O3	AR	P10275	CRBN	WO-2024189488-A1
TPD-LSBPAG	SCHEMBL31198605	7-[4-[4-[[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]methyl]phenyl]piperidin-1-yl]-4-fluoro-1H-indole-3-carbonitrile	N#Cc1c[nH]c2c(N3CCC(c4ccc(CN5CCN(CC6CCN(c7ccc8c(c7)CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)cc4)CC3)ccc(F)c12	C44H49FN8O3	AR	P10275	CRBN	WO-2024189488-A1
TPD-6TLTDB	SCHEMBL31198696	4-chloro-7-[4-[6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridin-3-yl]piperidin-1-yl]-1H-indole-3-carbonitrile	N#Cc1c[nH]c2c(N3CCC(c4ccc(N5CCC(CN6CCC(n7ccc8c(N9CCC(=O)NC9=O)cccc87)CC6)CC5)nc4)CC3)ccc(Cl)c12	C42H46ClN9O2	AR	P10275	CRBN	WO-2024189488-A1
TPD-1JMZE8	SCHEMBL31198682	4-chloro-7-[4-[6-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]pyridin-3-yl]piperidin-1-yl]-1H-indole-3-carbonitrile	N#Cc1c[nH]c2c(N3CCC(c4ccc(N5CCC(CN6CCN(c7ccc8c(c7)CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)nc4)CC3)ccc(Cl)c12	C42H46ClN9O3	AR	P10275	CRBN	WO-2024189488-A1
TPD-M5S3ZW	SCHEMBL31198684	4-chloro-7-[4-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]piperidin-1-yl]phenyl]piperidin-1-yl]-1H-indole-3-carbonitrile	N#Cc1c[nH]c2c(N3CCC(c4ccc(N5CCC(N6CCN(c7ccc8c(c7)CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)cc4)CC3)ccc(Cl)c12	C42H45ClN8O3	AR	P10275	CRBN	WO-2024189488-A1
TPD-MIK67G	SCHEMBL31198572	4-chloro-7-[4-[4-[4-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]piperidin-1-yl]phenyl]piperidin-1-yl]-1H-indole-3-carbonitrile	N#Cc1c[nH]c2c(N3CCC(c4ccc(N5CCC(N6CCC(n7ccc8c(N9CCC(=O)NC9=O)cccc87)CC6)CC5)cc4)CC3)ccc(Cl)c12	C42H45ClN8O2	AR	P10275	CRBN	WO-2024189488-A1
TPD-XDUE1N	SCHEMBL31198610	4-chloro-7-[4-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-1-methylindole-3-carbonitrile	COc1cc(N2CCN(CC3CCN(c4ccc(C5CCN(c6ccc(Cl)c7c(C#N)cn(C)c67)CC5)cc4)CC3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C45H51ClN8O4	AR	P10275	CRBN	WO-2024189488-A1
TPD-1Y5V74	SCHEMBL31198595	4-chloro-7-[4-[3-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-1H-indole-3-carbonitrile	N#Cc1c[nH]c2c(N3CCC(c4cccc(N5CCC(CN6CCN(c7ccc8c(c7)CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)c4)CC3)ccc(Cl)c12	C43H47ClN8O3	AR	P10275	CRBN	WO-2024189488-A1
TPD-I2MO8H	SCHEMBL31198576	4-chloro-7-[(3S)-3-[4-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)-2-methylindol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-1H-indole-3-carbonitrile	Cc1cc2c(N3CCC(=O)NC3=O)cccc2n1C1CCN(CC2CCN(c3ccc([C@@H]4CCCN(c5ccc(Cl)c6c(C#N)c[nH]c56)C4)cc3)CC2)CC1	C44H49ClN8O2	AR	P10275	CRBN	WO-2024189488-A1
TPD-2VK7RF	WO2024189488A1_116	4-chloro-7-[3-[6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridin-3-yl]piperidin-1-yl]-1H-indole-3-carbonitrile	N#Cc1c[nH]c2c(N3CCCC(c4ccc(N5CCC(CN6CCC(n7ccc8c(N9CCC(=O)NC9=O)cccc87)CC6)CC5)nc4)C3)ccc(Cl)c12	C42H46ClN9O2	AR	P10275	CRBN	WO-2024189488-A1
TPD-J3LGIK	WO2024189488A1_117	4-chloro-7-[2-[4-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]morpholin-4-yl]-1H-indole-3-carbonitrile	N#Cc1c[nH]c2c(N3CCOC(c4ccc(N5CCC(CN6CCC(n7ccc8c(N9CCC(=O)NC9=O)cccc87)CC6)CC5)cc4)C3)ccc(Cl)c12	C42H45ClN8O3	AR	P10275	CRBN	WO-2024189488-A1
TPD-KBW29Q	WO2024189488A1_120	.	N#Cc1n[nH]c2c(N3CCOC(c4ccc(N5CCC(CN6CCC(n7ccc8c(N9CCC(=O)NC9=O)cccc87)CC6)CC5)cc4)C3)ccc(Cl)c12	C41H44ClN9O3	AR	P10275	CRBN	WO-2024189488-A1
TPD-ENU68C	SCHEMBL31198618	4-chloro-7-[(3R)-3-[6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridazin-3-yl]piperidin-1-yl]-1H-indole-3-carbonitrile	N#Cc1c[nH]c2c(N3CCC[C@@H](c4ccc(N5CCC(CN6CCC(n7ccc8c(N9CCC(=O)NC9=O)cccc87)CC6)CC5)nn4)C3)ccc(Cl)c12	C41H45ClN10O2	AR	P10275	CRBN	WO-2024189488-A1
TPD-5M8C71	SCHEMBL31198540	4-chloro-7-[4-[4-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)-2-methylindol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-1H-indole-3-carbonitrile	Cc1cc2c(N3CCC(=O)NC3=O)cccc2n1C1CCN(CC2CCN(c3ccc(C4CCN(c5ccc(Cl)c6c(C#N)c[nH]c56)CC4)cc3)CC2)CC1	C44H49ClN8O2	AR	P10275	CRBN	WO-2024189488-A1
TPD-OPGVL5	SCHEMBL31198645	4-chloro-7-[4-[2-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]pyrimidin-5-yl]piperidin-1-yl]-1H-indole-3-carbonitrile	N#Cc1c[nH]c2c(N3CCC(c4cnc(N5CCC(CN6CCN(c7ccc8c(c7)CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)nc4)CC3)ccc(Cl)c12	C41H45ClN10O3	AR	P10275	CRBN	WO-2024189488-A1
TPD-KX25FQ	SCHEMBL31198647	4-chloro-7-[4-[2-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyrimidin-5-yl]piperidin-1-yl]-1H-indole-3-carbonitrile	N#Cc1c[nH]c2c(N3CCC(c4cnc(N5CCC(CN6CCC(n7ccc8c(N9CCC(=O)NC9=O)cccc87)CC6)CC5)nc4)CC3)ccc(Cl)c12	C41H45ClN10O2	AR	P10275	CRBN	WO-2024189488-A1
TPD-MLDFKB	SCHEMBL31198579	7-[4-[4-[(2R)-2-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]morpholin-4-yl]phenyl]piperidin-1-yl]-4-fluoro-1H-indole-3-carbonitrile	N#Cc1c[nH]c2c(N3CCC(c4ccc(N5CCO[C@H](CN6CCN(c7ccc8c(c7)CN(C7CCC(=O)NC7=O)C8=O)CC6)C5)cc4)CC3)ccc(F)c12	C42H45FN8O4	AR	P10275	CRBN	WO-2024189488-A1
TPD-TR2BPA	SCHEMBL31198713	4-chloro-7-[4-[4-[(2R)-2-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]morpholin-4-yl]phenyl]piperidin-1-yl]-1H-indole-3-carbonitrile	N#Cc1c[nH]c2c(N3CCC(c4ccc(N5CCO[C@H](CN6CCN(c7ccc8c(c7)CN(C7CCC(=O)NC7=O)C8=O)CC6)C5)cc4)CC3)ccc(Cl)c12	C42H45ClN8O4	AR	P10275	CRBN	WO-2024189488-A1
TPD-WU45KJ	SCHEMBL31198661	7-[4-[4-[7-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]-2-azaspiro[3.5]nonan-2-yl]phenyl]piperidin-1-yl]-4-fluoro-1H-indole-3-carbonitrile	N#Cc1c[nH]c2c(N3CCC(c4ccc(N5CC6(CCC(CN7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)C5)cc4)CC3)ccc(F)c12	C46H51FN8O3	AR	P10275	CRBN	WO-2024189488-A1
TPD-JFF0OL	SCHEMBL31198653	4-chloro-7-[4-[4-[7-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]-2-azaspiro[3.5]nonan-2-yl]phenyl]piperidin-1-yl]-1H-indole-3-carbonitrile	N#Cc1c[nH]c2c(N3CCC(c4ccc(N5CC6(CCC(CN7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)C5)cc4)CC3)ccc(Cl)c12	C46H51ClN8O3	AR	P10275	CRBN	WO-2024189488-A1
TPD-P3NEY2	SCHEMBL31198636	4-chloro-7-[(3S)-3-[4-[7-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]-2-azaspiro[3.5]nonan-2-yl]phenyl]piperidin-1-yl]-1H-indole-3-carbonitrile	N#Cc1c[nH]c2c(N3CCC[C@@H](c4ccc(N5CC6(CCC(CN7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)C5)cc4)C3)ccc(Cl)c12	C46H51ClN8O3	AR	P10275	CRBN	WO-2024189488-A1
TPD-LG8SQN	SCHEMBL31198565	4-chloro-7-[(3S)-3-[4-[7-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]-2-azaspiro[3.5]nonan-2-yl]phenyl]piperidin-1-yl]-1H-indole-3-carbonitrile	N#Cc1c[nH]c2c(N3CCC[C@@H](c4ccc(N5CC6(CCC(CN7CCC(n8ccc9c(N%10CCC(=O)NC%10=O)cccc98)CC7)CC6)C5)cc4)C3)ccc(Cl)c12	C46H51ClN8O2	AR	P10275	CRBN	WO-2024189488-A1
TPD-KEP7E6	SCHEMBL31198535	4-chloro-7-[(3R)-3-[4-[4-[[4-[6-(2,4-dioxo-1,3-diazinan-1-yl)-1-methylindol-2-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-1H-indazole-3-carbonitrile	Cn1c(C2CCN(CC3CCN(c4ccc([C@H]5CCCN(c6ccc(Cl)c7c(C#N)n[nH]c67)C5)cc4)CC3)CC2)cc2ccc(N3CCC(=O)NC3=O)cc21	C43H48ClN9O2	AR	P10275	CRBN	WO-2024189488-A1
TPD-FJEBEW	SCHEMBL31198634	7-[(3S)-3-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-4-fluoro-1H-indazole-3-carbonitrile	N#Cc1n[nH]c2c(N3CCC[C@@H](c4ccc(N5CCC(CN6CCN(c7ccc8c(c7)CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)cc4)C3)ccc(F)c12	C42H46FN9O3	AR	P10275	CRBN	WO-2024189488-A1
TPD-X22ZTU	SCHEMBL31198699	7-[(3S)-3-[4-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-4-fluoro-1H-indazole-3-carbonitrile	N#Cc1n[nH]c2c(N3CCC[C@@H](c4ccc(N5CCC(CN6CCC(n7ccc8c(N9CCC(=O)NC9=O)cccc87)CC6)CC5)cc4)C3)ccc(F)c12	C42H46FN9O2	AR	P10275	CRBN	WO-2024189488-A1
TPD-L1MFK8	SCHEMBL31198573	7-[4-[4-[7-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]-2-azaspiro[3.5]nonan-2-yl]phenyl]piperidin-1-yl]-4-fluoro-1H-indole-3-carbonitrile	N#Cc1c[nH]c2c(N3CCC(c4ccc(N5CC6(CCC(CN7CCC(n8ccc9c(N%10CCC(=O)NC%10=O)cccc98)CC7)CC6)C5)cc4)CC3)ccc(F)c12	C46H51FN8O2	AR	P10275	CRBN	WO-2024189488-A1
TPD-QOWN8C	SCHEMBL31198562	4-chloro-7-[(3R)-3-[4-[4-[[4-[6-(2,4-dioxo-1,3-diazinan-1-yl)-5-fluoro-1-methylindol-2-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-1H-indole-3-carbonitrile	Cn1c(C2CCN(CC3CCN(c4ccc([C@H]5CCCN(c6ccc(Cl)c7c(C#N)c[nH]c67)C5)cc4)CC3)CC2)cc2cc(F)c(N3CCC(=O)NC3=O)cc21	C44H48ClFN8O2	AR	P10275	CRBN	WO-2024189488-A1
TPD-F8U8P5	SCHEMBL31198557	4-chloro-7-[(3S)-3-[4-[4-[[4-[6-(2,4-dioxo-1,3-diazinan-1-yl)-5-fluoro-1-methylindol-2-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-1H-indole-3-carbonitrile	Cn1c(C2CCN(CC3CCN(c4ccc([C@@H]5CCCN(c6ccc(Cl)c7c(C#N)c[nH]c67)C5)cc4)CC3)CC2)cc2cc(F)c(N3CCC(=O)NC3=O)cc21	C44H48ClFN8O2	AR	P10275	CRBN	WO-2024189488-A1
TPD-5E33NT	SCHEMBL31198660	4-chloro-7-[(3R)-3-[4-[4-[[4-[6-(2,4-dioxo-1,3-diazinan-1-yl)-5-fluoro-1-methylindol-2-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-1H-indazole-3-carbonitrile	Cn1c(C2CCN(CC3CCN(c4ccc([C@H]5CCCN(c6ccc(Cl)c7c(C#N)n[nH]c67)C5)cc4)CC3)CC2)cc2cc(F)c(N3CCC(=O)NC3=O)cc21	C43H47ClFN9O2	AR	P10275	CRBN	WO-2024189488-A1
TPD-8L7OPM	WO2024189488A1_139	.	Cc1ccc(N2CCC[C@@H](c3ccc(N4CCC(CN5CCC(c6cc7cc(F)c(N8CCC(=O)NC8=O)cc7n6C)CC5)CC4)cc3)C2)c2[nH]nc(C#N)c12	C44H50FN9O2	AR	P10275	CRBN	WO-2024189488-A1
TPD-EAHZSA	SCHEMBL31198556	7-[4-[4-[4-[[4-[6-(2,4-dioxo-1,3-diazinan-1-yl)-1-methylindol-2-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-4-fluoro-1H-indazole-3-carbonitrile	Cn1c(C2CCN(CC3CCN(c4ccc(C5CCN(c6ccc(F)c7c(C#N)n[nH]c67)CC5)cc4)CC3)CC2)cc2ccc(N3CCC(=O)NC3=O)cc21	C43H48FN9O2	AR	P10275	CRBN	WO-2024189488-A1
TPD-2AGBTP	SCHEMBL31198600	7-[4-[4-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)-2-methylindol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-4-fluoro-1H-indole-3-carbonitrile	Cc1cc2c(N3CCC(=O)NC3=O)cccc2n1C1CCN(CC2CCN(c3ccc(C4CCN(c5ccc(F)c6c(C#N)c[nH]c56)CC4)cc3)CC2)CC1	C44H49FN8O2	AR	P10275	CRBN	WO-2024189488-A1
TPD-GYVJHW	SCHEMBL31198678	4-chloro-7-[4-[4-[7-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]-2-azaspiro[3.5]nonan-2-yl]phenyl]piperidin-1-yl]-1H-indole-3-carbonitrile	N#Cc1c[nH]c2c(N3CCC(c4ccc(N5CC6(CCC(CN7CCC(n8ccc9c(N%10CCC(=O)NC%10=O)cccc98)CC7)CC6)C5)cc4)CC3)ccc(Cl)c12	C46H51ClN8O2	AR	P10275	CRBN	WO-2024189488-A1
TPD-RA3F8P	SCHEMBL31198637	4-chloro-7-[4-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-4-methoxy-3-oxo-1H-pyrrolo[3,4-c]pyridin-6-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-1H-indazole-3-carbonitrile	COc1nc(N2CCN(CC3CCN(c4ccc(C5CCN(c6ccc(Cl)c7c(C#N)n[nH]c67)CC5)cc4)CC3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C42H47ClN10O4	AR	P10275	CRBN	WO-2024189488-A1
TPD-PL6FTK	SCHEMBL31198534	7-[4-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-4-methoxy-3-oxo-1H-pyrrolo[3,4-c]pyridin-6-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-4-fluoro-1H-indazole-3-carbonitrile	COc1nc(N2CCN(CC3CCN(c4ccc(C5CCN(c6ccc(F)c7c(C#N)n[nH]c67)CC5)cc4)CC3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C42H47FN10O4	AR	P10275	CRBN	WO-2024189488-A1
TPD-AXNGZW	SCHEMBL31198601	7-[4-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-4-fluoro-1H-indazole-3-carbonitrile	N#Cc1n[nH]c2c(N3CCC(c4ccc(N5CCC(CN6CCN(c7ccc8c(c7)CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)cc4)CC3)ccc(F)c12	C42H46FN9O3	AR	P10275	CRBN	WO-2024189488-A1
TPD-4T0FUI	SCHEMBL31198691	4-chloro-7-[4-[4-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-1H-indazole-3-carbonitrile	N#Cc1n[nH]c2c(N3CCC(c4ccc(N5CCC(CN6CCC(n7ccc8c(N9CCC(=O)NC9=O)cccc87)CC6)CC5)cc4)CC3)ccc(Cl)c12	C42H46ClN9O2	AR	P10275	CRBN	WO-2024189488-A1
TPD-A7C8BC	SCHEMBL31198641	7-[4-[4-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-4-fluoro-1H-indazole-3-carbonitrile	N#Cc1n[nH]c2c(N3CCC(c4ccc(N5CCC(CN6CCC(n7ccc8c(N9CCC(=O)NC9=O)cccc87)CC6)CC5)cc4)CC3)ccc(F)c12	C42H46FN9O2	AR	P10275	CRBN	WO-2024189488-A1
TPD-TRZWMX	SCHEMBL31198663	7-[4-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]butoxy]phenyl]piperidin-1-yl]-4-methyl-1H-indazole-3-carbonitrile	COc1cc(N2CCN(CCCCOc3ccc(C4CCN(c5ccc(C)c6c(C#N)n[nH]c56)CC4)cc3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C42H48N8O5	AR	P10275	CRBN	WO-2024189488-A1
TPD-BFH475	SCHEMBL31198555	7-[4-[4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]piperidin-1-yl]-4-methyl-1H-indazole-3-carbonitrile	COc1cc(N2CCN(CC3CCN(c4ccc(C5CCN(c6ccc(C)c7c(C#N)n[nH]c67)CC5)cc4)CC3)CC2)cc2c1C(=O)N(C1CCC(=O)NC1=O)C2	C44H51N9O4	AR	P10275	CRBN	WO-2024189488-A1
TPD-ZJM4H9	WO2024189488A1_151	7-[3-[4-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]butoxy]phenyl]pyrrolidin-1-yl]-4-methyl-1H-indole-3-carbonitrile	Cc1ccc(N2CCC(c3ccc(OCCCCN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)cc3)C2)c2[nH]cc(C#N)c12	C41H45N7O4	AR	P10275	CRBN	WO-2024189488-A1
TPD-CW513M	SCHEMBL31198652	N-[1-(4-chloro-3-cyano-1H-indazol-7-yl)piperidin-4-yl]-4-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]-2-fluorobenzamide	N#Cc1n[nH]c2c(N3CCC(NC(=O)c4ccc(N5CCC(CN6CCC(n7ccc8c(N9CCC(=O)NC9=O)cccc87)CC6)CC5)cc4F)CC3)ccc(Cl)c12	C43H46ClFN10O3	AR	P10275	CRBN	WO-2024189488-A1
TPD-K6YYSC	SCHEMBL31198666	N-[1-(4-chloro-3-cyano-1H-indol-7-yl)piperidin-4-yl]-4-[4-[[4-[5-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]-2-fluorobenzamide	N#Cc1c[nH]c2c(N3CCC(NC(=O)c4ccc(N5CCC(CN6CCC(n7ccc8cc(N9CCC(=O)NC9=O)ccc87)CC6)CC5)cc4F)CC3)ccc(Cl)c12	C44H47ClFN9O3	AR	P10275	CRBN	WO-2024189488-A1
TPD-9BSD54	WO2024189488A1_154	.	N#Cc1c[nH]c2c(N3CCC(NC(=O)c4ccc(N5CCC(CN6CCN(c7ccc(C(=O)NC8CCC(=O)NC8=O)c(F)c7)CC6)CC5)cc4F)CC3)ccc(Cl)c12	C43H46ClF2N9O4	AR	P10275	CRBN	WO-2024189488-A1
TPD-WL5YPK	SCHEMBL31198672	N-[1-(4-chloro-3-cyano-1H-indol-7-yl)piperidin-4-yl]-4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-5,7-dihydropyrrolo[3,4-f]isoindol-6-yl]methyl]piperidin-1-yl]-2-fluorobenzamide	N#Cc1c[nH]c2c(N3CCC(NC(=O)c4ccc(N5CCC(CN6Cc7cc8c(cc7C6)C(=O)N(C6CCC(=O)NC6=O)C8=O)CC5)cc4F)CC3)ccc(Cl)c12	C42H40ClFN8O5	AR	P10275	CRBN	WO-2024189488-A1
TPD-VMA20T	SCHEMBL31198671	N-[1-(4-chloro-3-cyano-1H-indol-7-yl)piperidin-4-yl]-4-[4-[[4-[6-(2,4-dioxo-1,3-diazinan-1-yl)-5-fluoro-1-methylindol-2-yl]piperidin-1-yl]methyl]piperidin-1-yl]-2-fluorobenzamide	Cn1c(C2CCN(CC3CCN(c4ccc(C(=O)NC5CCN(c6ccc(Cl)c7c(C#N)c[nH]c67)CC5)c(F)c4)CC3)CC2)cc2cc(F)c(N3CCC(=O)NC3=O)cc21	C45H48ClF2N9O3	AR	P10275	CRBN	WO-2024189488-A1
TPD-CBKQMB	SCHEMBL31198644	N-[1-(4-chloro-3-cyano-1H-indol-7-yl)piperidin-4-yl]-4-[4-[[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-4-yl]piperazin-1-yl]methyl]piperidin-1-yl]-2-fluorobenzamide	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(N3CCN(CC4CCN(c5ccc(C(=O)NC6CCN(c7ccc(Cl)c8c(C#N)c[nH]c78)CC6)c(F)c5)CC4)CC3)c21	C44H48ClFN10O4	AR	P10275	CRBN	WO-2024189488-A1
TPD-PY2AGN	SCHEMBL31198563	N-[1-(4-chloro-3-cyano-1H-indol-7-yl)piperidin-4-yl]-4-[4-[[4-[6-(2,4-dioxo-1,3-diazinan-1-yl)-1-methylindol-2-yl]piperidin-1-yl]methyl]piperidin-1-yl]-2-fluorobenzamide	Cn1c(C2CCN(CC3CCN(c4ccc(C(=O)NC5CCN(c6ccc(Cl)c7c(C#N)c[nH]c67)CC5)c(F)c4)CC3)CC2)cc2ccc(N3CCC(=O)NC3=O)cc21	C45H49ClFN9O3	AR	P10275	CRBN	WO-2024189488-A1
TPD-FOQ45G	SCHEMBL31198590	N-[1-(4-chloro-3-cyano-1H-indol-7-yl)piperidin-4-yl]-4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]-2-fluorobenzamide	N#Cc1c[nH]c2c(N3CCC(NC(=O)c4ccc(N5CCC(CN6CCN(c7ccc8c(c7)CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)cc4F)CC3)ccc(Cl)c12	C44H47ClFN9O4	AR	P10275	CRBN	WO-2024189488-A1
TPD-F84VOJ	SCHEMBL31198665	N-[1-(4-chloro-3-cyano-1H-indol-7-yl)piperidin-4-yl]-4-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]-2-fluorobenzamide	N#Cc1c[nH]c2c(N3CCC(NC(=O)c4ccc(N5CCC(CN6CCC(n7ccc8c(N9CCC(=O)NC9=O)cccc87)CC6)CC5)cc4F)CC3)ccc(Cl)c12	C44H47ClFN9O3	AR	P10275	CRBN	WO-2024189488-A1
TPD-TI1I8D	SCHEMBL31198676	N-[1-(4-chloro-3-cyano-1H-indol-7-yl)piperidin-4-yl]-4-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]-2-fluorobenzamide	N#Cc1c[nH]c2c(N3CCC(NC(=O)c4ccc(N5CCC(CN6CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)cc4F)CC3)ccc(Cl)c12	C44H44ClF2N9O5	AR	P10275	CRBN	WO-2024189488-A1
TPD-CMPSD6	SCHEMBL31198693	N-[1-(4-chloro-3-cyano-1H-indol-7-yl)piperidin-4-yl]-2-cyano-4-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]benzamide	N#Cc1cc(N2CCC(CN3CCC(n4ccc5c(N6CCC(=O)NC6=O)cccc54)CC3)CC2)ccc1C(=O)NC1CCN(c2ccc(Cl)c3c(C#N)c[nH]c23)CC1	C45H47ClN10O3	AR	P10275	CRBN	WO-2024189488-A1
TPD-LNMCDQ	SCHEMBL31198559	N-[1-(4-chloro-3-cyano-1H-indol-7-yl)piperidin-4-yl]-4-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]-2-fluoro-6-methylbenzamide	Cc1cc(N2CCC(CN3CCC(n4ccc5c(N6CCC(=O)NC6=O)cccc54)CC3)CC2)cc(F)c1C(=O)NC1CCN(c2ccc(Cl)c3c(C#N)c[nH]c23)CC1	C45H49ClFN9O3	AR	P10275	CRBN	WO-2024189488-A1
TPD-H2L85U	SCHEMBL31198583	N-[1-(4-chloro-3-cyano-1H-indol-7-yl)piperidin-4-yl]-4-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]-3-methylbenzamide	Cc1cc(C(=O)NC2CCN(c3ccc(Cl)c4c(C#N)c[nH]c34)CC2)ccc1N1CCC(CN2CCC(n3ccc4c(N5CCC(=O)NC5=O)cccc43)CC2)CC1	C45H50ClN9O3	AR	P10275	CRBN	WO-2024189488-A1
TPD-P1TIIW	SCHEMBL31198707	N-[1-(4-chloro-3-cyano-1H-indol-7-yl)piperidin-4-yl]-3-cyano-4-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]benzamide	N#Cc1cc(C(=O)NC2CCN(c3ccc(Cl)c4c(C#N)c[nH]c34)CC2)ccc1N1CCC(CN2CCC(n3ccc4c(N5CCC(=O)NC5=O)cccc43)CC2)CC1	C45H47ClN10O3	AR	P10275	CRBN	WO-2024189488-A1
TPD-JL0YZE	SCHEMBL31198591	N-[1-(4-chloro-3-cyano-1H-indol-7-yl)piperidin-4-yl]-5-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]piperidin-1-yl]pyridine-2-carboxamide	N#Cc1c[nH]c2c(N3CCC(NC(=O)c4ccc(N5CCC(N6CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)cn4)CC3)ccc(Cl)c12	C42H42ClFN10O5	AR	P10275	CRBN	WO-2024189488-A1
TPD-E9TRCC	SCHEMBL31198673	N-[1-(4-chloro-3-cyano-1H-indol-7-yl)piperidin-4-yl]-5-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridine-2-carboxamide	N#Cc1c[nH]c2c(N3CCC(NC(=O)c4ccc(N5CCC(CN6CCC(n7ccc8c(N9CCC(=O)NC9=O)cccc87)CC6)CC5)cn4)CC3)ccc(Cl)c12	C43H47ClN10O3	AR	P10275	CRBN	WO-2024189488-A1
TPD-33NYNV	SCHEMBL31198577	N-[1-(4-chloro-3-cyano-1H-indol-7-yl)piperidin-4-yl]-5-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]pyridine-2-carboxamide	N#Cc1c[nH]c2c(N3CCC(NC(=O)c4ccc(N5CCC(CN6CCN(c7ccc8c(c7)CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)cn4)CC3)ccc(Cl)c12	C43H47ClN10O4	AR	P10275	CRBN	WO-2024189488-A1
TPD-DRTSW0	SCHEMBL31198669	N-[1-(4-chloro-3-cyano-1H-indol-7-yl)piperidin-4-yl]-5-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]pyridine-2-carboxamide	N#Cc1c[nH]c2c(N3CCC(NC(=O)c4ccc(N5CCC(CN6CCN(c7cc8c(cc7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)cn4)CC3)ccc(Cl)c12	C43H44ClFN10O5	AR	P10275	CRBN	WO-2024189488-A1
TPD-IRSH1L	SCHEMBL31198668	N-[1-(4-chloro-3-cyano-1H-indazol-7-yl)piperidin-4-yl]-5-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridine-2-carboxamide	N#Cc1n[nH]c2c(N3CCC(NC(=O)c4ccc(N5CCC(CN6CCC(n7ccc8c(N9CCC(=O)NC9=O)cccc87)CC6)CC5)cn4)CC3)ccc(Cl)c12	C42H46ClN11O3	AR	P10275	CRBN	WO-2024189488-A1
TPD-D2XR50	SCHEMBL31198639	N-[1-(3-cyano-4-methyl-1H-indol-7-yl)piperidin-4-yl]-5-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]pyridine-2-carboxamide	Cc1ccc(N2CCC(NC(=O)c3ccc(N4CCC(CN5CCN(c6cc7c(cc6F)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cn3)CC2)c2[nH]cc(C#N)c12	C44H47FN10O5	AR	P10275	CRBN	WO-2024189488-A1
TPD-V32RD1	SCHEMBL31198681	N-[1-(3-cyano-4-methyl-1H-indol-7-yl)piperidin-4-yl]-5-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]pyridine-2-carboxamide	Cc1ccc(N2CCC(NC(=O)c3ccc(N4CCC(CN5CCN(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC5)CC4)cn3)CC2)c2[nH]cc(C#N)c12	C44H50N10O4	AR	P10275	CRBN	WO-2024189488-A1
TPD-6Z3J6A	SCHEMBL31198607	N-[1-(4-chloro-3-cyano-1H-indol-7-yl)piperidin-4-yl]-4-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]benzamide	N#Cc1c[nH]c2c(N3CCC(NC(=O)c4ccc(N5CCC(CN6CCC(n7ccc8c(N9CCC(=O)NC9=O)cccc87)CC6)CC5)cc4)CC3)ccc(Cl)c12	C44H48ClN9O3	AR	P10275	CRBN	WO-2024189488-A1
TPD-TFH8QZ	SCHEMBL31198716	N-[4-(4-chloro-3-cyano-1H-indol-7-yl)cyclohexyl]-4-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]-2-fluorobenzamide	N#Cc1c[nH]c2c(C3CCC(NC(=O)c4ccc(N5CCC(CN6CCC(n7ccc8c(N9CCC(=O)NC9=O)cccc87)CC6)CC5)cc4F)CC3)ccc(Cl)c12	C45H48ClFN8O3	AR	P10275	CRBN	WO-2024189488-A1
TPD-SA4TR5	SCHEMBL31198654	N-[1-(4-chloro-3-cyano-1H-indol-7-yl)piperidin-4-yl]-4-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]-2,6-difluorobenzamide	N#Cc1c[nH]c2c(N3CCC(NC(=O)c4c(F)cc(N5CCC(CN6CCC(n7ccc8c(N9CCC(=O)NC9=O)cccc87)CC6)CC5)cc4F)CC3)ccc(Cl)c12	C44H46ClF2N9O3	AR	P10275	CRBN	WO-2024189488-A1
TPD-CGDGS9	SCHEMBL31198640	N-[1-(4-chloro-3-cyano-1H-indol-7-yl)piperidin-4-yl]-5-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyrazine-2-carboxamide	N#Cc1c[nH]c2c(N3CCC(NC(=O)c4cnc(N5CCC(CN6CCC(n7ccc8c(N9CCC(=O)NC9=O)cccc87)CC6)CC5)cn4)CC3)ccc(Cl)c12	C42H46ClN11O3	AR	P10275	CRBN	WO-2024189488-A1
TPD-9J9F83	SCHEMBL31198584	N-[1-(4-chloro-3-cyano-1H-indol-7-yl)piperidin-4-yl]-5-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyrimidine-2-carboxamide	N#Cc1c[nH]c2c(N3CCC(NC(=O)c4ncc(N5CCC(CN6CCC(n7ccc8c(N9CCC(=O)NC9=O)cccc87)CC6)CC5)cn4)CC3)ccc(Cl)c12	C42H46ClN11O3	AR	P10275	CRBN	WO-2024189488-A1
TPD-CA5HUD	SCHEMBL31198548	N-[1-(4-chloro-3-cyano-1H-indol-7-yl)piperidin-4-yl]-4-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]-2-methylbenzamide	Cc1cc(N2CCC(CN3CCC(n4ccc5c(N6CCC(=O)NC6=O)cccc54)CC3)CC2)ccc1C(=O)NC1CCN(c2ccc(Cl)c3c(C#N)c[nH]c23)CC1	C45H50ClN9O3	AR	P10275	CRBN	WO-2024189488-A1
TPD-M0M92M	SCHEMBL31198609	N-[1-(4-chloro-3-cyano-1H-indol-7-yl)piperidin-4-yl]-6-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]methyl]piperidin-1-yl]pyridazine-3-carboxamide	N#Cc1c[nH]c2c(N3CCC(NC(=O)c4ccc(N5CCC(CN6CCC(n7ccc8c(N9CCC(=O)NC9=O)cccc87)CC6)CC5)nn4)CC3)ccc(Cl)c12	C42H46ClN11O3	AR	P10275	CRBN	WO-2024189488-A1
TPD-Q5AEQV	SCHEMBL31198541	N-[(3R)-1-(4-chloro-3-cyano-1H-indol-7-yl)piperidin-3-yl]-5-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]pyridine-2-carboxamide	N#Cc1c[nH]c2c(N3CCC[C@@H](NC(=O)c4ccc(N5CCC(CN6CCN(c7ccc8c(c7)CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)cn4)C3)ccc(Cl)c12	C43H47ClN10O4	AR	P10275	CRBN	WO-2024189488-A1
TPD-5WZBTJ	WO2024189488A1_181	.	N#Cc1c[nH]c2c(N3CCC[C@H](NC(=O)c4ccc(N5CCC(CN6CCN(c7ccc8c(c7)CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)cn4)C3)ccc(Cl)c12	C43H47ClN10O4	AR	P10275	CRBN	WO-2024189488-A1
TPD-N55G3E	WO2024208256A1_16	.	O=C1CCC(N2CC3=C(C=C4CN(C5CCN(C[C@H]6CC[C@H](N7C=C(NC(=O)C8=C9N=C(N%10CCOCC%10)C=CN9N=C8)C(C(F)F)=N7)CC6)CC5)CC4=C3)C2=O)C(=O)N1	C42H49F2N11O5	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-NTS0EE	WO2024208256A1_17	.	O=C1CCC(N2C(=O)C3=C(C=C4CN(C5CCN(C[C@H]6CC[C@H](N7C=C(NC(=O)C8=C9N=C(N%10CCOCC%10)C=CN9N=C8)C(C(F)F)=N7)CC6)CC5)CC4=C3)C2=O)C(=O)N1	C42H47F2N11O6	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-GKNOB2	WO2024208256A1_18	.	CC(C)(O)C1=CC2=NN(C3CCC(CN4CCC(N5CC6=CC7=C(C=C6C5)C(=O)N(C5CCC(=O)NC5=O)C7)CC4)CC3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C44H49F3N8O5	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-4P697X	WO2024208256A1_19	.	O=C1CCC(N2C(=O)C3=C(C=C4CN(C5CCN(CCN6CCC(N7C=C(NC(=O)C8=C9N=C(N%10CCOCC%10)C=CN9N=C8)C(C(F)F)=N7)CC6)CC5)CC4=C3)C2=O)C(=O)N1	C42H48F2N12O6	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-2EYD04	WO2024208256A1_20	.	CC(C)(O)C1=CC2=NN(C3=CC=C(CC4CCN(C5=C(F)C=C(C6CCC(=O)NC6=O)C=C5)CC4)C=C3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C40H38F4N6O4	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-4OCW73	WO2024208256A1_21	.	CC(C)(O)C1=CC2=NN(C3=CC=C(NC(=O)C4CCN(C5=C(F)C=C(C6CCC(=O)NC6=O)C=C5)CC4)C=C3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C40H37F4N7O5	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-Y9D6IU	WO2024208256A1_22	.	CC(C)(O)C1=CC2=NN(C3=CC=C(OC4CC5(CCN(C6=C(F)C=C(C7CCC(=O)NC7=O)C=C6)CC5)C4)C=C3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C42H40F4N6O5	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-2P9XGV	WO2024208256A1_23	.	CC(C)(O)C1=CC2=NN(C3=CC=C(CN4CCC(C5=C(F)C=C(C6CCC(=O)NC6=O)C=C5)CC4)C=C3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C40H38F4N6O4	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-D618MO	WO2024208256A1_24	.	COC1=CC2=NN([C@H]3CC[C@@H](CN4CCC(C5=C(F)C=C(C6CCC(=O)NC6=O)C=C5)CC4)CC3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C38H40F4N6O4	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-NRMGO2	WO2024208256A1_25	.	CC(C)(O)C1=CC2=NN([C@H]3CC[C@@H](CN4CCC(OC5=CC=C(C6CCC(=O)NC6=O)C=C5F)CC4)CC3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C40H44F4N6O5	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-G6OV84	WO2024208256A1_26	.	CC(C)(O)C1=CC2=NN(C3CCN(CCC4CCC(F)(C5=CC=C(C6CCC(=O)NC6=O)C=C5F)CC4)CC3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C41H45F5N6O4	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-2JK6HZ	WO2024208256A1_29	.	COC1=CC2=NN(C3CCN(CC4CC5(CCN(C6=C(F)C=C(C7CCC(=O)NC7=O)C=C6)CC5)C4)CC3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C40H43F4N7O4	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-HRALOM	WO2024208256A1_30	.	COC1(C2=CC=C(C3CCC(=O)NC3=O)C=C2F)CCC(CCN2CCC(N3C=C4C=C(NC(=O)C5=NC(C(F)(F)F)=CC=C5)C(C(C)(C)O)=CC4=N3)CC2)CC1	C42H48F4N6O5	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-PHOPNU	WO2024208256A1_31	.	CC(C)(O)C1=CC2=NN(C3CCN(CCC4CCC(F)(C5=CC=C(NC6CCC(=O)NC6=O)C=C5F)CC4)CC3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C41H46F5N7O4	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-7P90ER	WO2024208256A1_32	.	CC(C)(O)C1=CC2=NN(C3CCN(CC(F)(F)C4CCN(C5=CC=C(C6CCC(=O)NC6=O)C=C5F)CC4)CC3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C40H43F6N7O4	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-K6LV43	WO2024208256A1_33	.	CC(C)(O)C1=CC2=NN(C3CCC(CC(=O)N4CCC(C5=CC=C(NC6CCC(=O)NC6=O)C=C5F)CC4)CC3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C41H45F4N7O5	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-LPLV1G	WO2024208256A1_34	.	CC(C)(O)C1=CC2=NN(C3CCC(CC(=O)N4CCC(C5=CC=C(C6CCC(=O)NC6=O)C=C5F)C(F)(F)C4)CC3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C41H42F6N6O5	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-HF1H6B	WO2024208256A1_35	.	CC(C)(O)C1=CC2=NN(C3CCC(COC4CCN(C5=CC=C(C6CCC(=O)NC6=O)C=C5F)CC4)CC3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C40H44F4N6O5	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-YJMA73	WO2024208256A1_37	.	COC1=CC2=NN(C3CCC(N4CC5(CCC(C6=C(F)C=C(C7CCC(=O)NC7=O)C=C6)CC5)C4)CC3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C40H42F4N6O4	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-93NZUN	WO2024208256A1_38	.	COC1=CC2=NN(C3CCN(CCC4CCN(C5=CC=C(C6CCC(=O)NC6=O)C=C5F)CC4)CC3)C=C2C=C1NC(=O)C1=CC(C(F)(F)F)=CC=C1	C39H42F4N6O4	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-SZHEC5	WO2024208256A1_39	.	CC(C)(O)C1=CC2=NN([C@H]3CC[C@H](CCC4CCN(C5=C(F)C=C(C6CCC(=O)NC6=O)C=C5)CC4(F)F)CC3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C41H44F6N6O4	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-5NENTK	WO2024208256A1_40	.	COC1=CC2=NN(C3CCC4(CC3)CC(N3CCC(C5=C(F)C=C(C6CCC(=O)NC6=O)C=C5)CC3)C4)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C40H42F4N6O4	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-N1UJA1	WO2024208256A1_41	.	COC1=CC2=NN(C3CCC4(CC3)CC(CN3CCC(C5=C(F)C=C(C6CCC(=O)NC6=O)C=C5)C(F)(F)C3)C4)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C41H42F6N6O4	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-DRCRPR	WO2024208256A1_42	.	CC(C)(O)C1=CC2=NN([C@H]3CC[C@@H](CN4CCC(OC5=CC=C(C6CCC(=O)NC6=O)C=C5F)C(F)(F)C4)CC3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C40H42F6N6O5	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-R9TOGF	WO2024208256A1_43	.	COC1=CC2=NN(C3=CC=C(OCC4CCN(C5=CC=C(C6CCC(=O)NC6=O)C=C5F)CC4(F)F)C=C3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C38H32F6N6O5	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-UQT49R	WO2024208256A1_44	.	COC1=CC2=NN([C@H]3CC[C@@H](OC4CC5(CCN(C6=C(F)C=C(C7CCC(=O)NC7=O)C=C6)CC5)C4)CC3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C40H42F4N6O5	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-42MTMB	WO2024208256A1_45	.	CC(C)(O)C1=CC2=NN(C3CCC(COC4CCN(C5=C(F)C=C(C6CCC(=O)NC6=O)C=C5)CC4(F)F)CC3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C40H42F6N6O5	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-WGEXRJ	WO2024208256A1_46	.	COC1=CC2=NN(C3CCC(N4CC5(CCC(C6=C(F)C=C(C7CCC(=O)NC7=O)C=C6)C5)C4)CC3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C39H40F4N6O4	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-XJIM4T	WO2024208256A1_47	.	COC1=CC2=NN([C@H]3CC[C@H](CCN4C=C(C5=CC=C(C6CCC(=O)NC6=O)C=C5F)C=N4)CC3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C37H35F4N7O4	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-ZL4Y6T	WO2024208256A1_48	.	O=C1CCC(C2=CC(F)=C(N3CCC(CC[C@H]4CC[C@@H](N5C=C(NC(=O)C6=CC=CC(C(F)(F)F)=C6)C(C(F)F)=N5)CC4)CC3)C=C2)C(=O)N1	C36H39F6N5O3	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-10384U	WO2024208256A1_49	.	O=C1CCC(C2=CC(F)=C(N3CCC(CCN4CCC(N5C=C(NC(=O)C6=CC=CC(C(F)(F)F)=N6)C(C(F)F)=N5)CC4)CC3)C=C2)C(=O)N1	C34H37F6N7O3	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-I9FM2V	WO2024208256A1_50	.	CC(C)(O)C1=CC2=NN(C3CCC(OCC4CCN(C5=C(F)C=C(C6CCC(=O)NC6=O)C=C5)CC4(F)F)CC3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C40H42F6N6O5	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-SPB9ZC	WO2024208256A1_51	.	COC1=CC2=NN([C@H]3CC[C@H](CN4CC5(CC(C6=C(F)C=C(C7CCC(=O)NC7=O)C=C6)C5)C4)CC3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C39H40F4N6O4	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-WMLR43	WO2024208256A1_52	.	COC1=CC2=NN([C@H]3CC[C@H](CN4CC5(CCC(C6=C(F)C=C(C7CCC(=O)NC7=O)C=C6)C5)C4)CC3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C40H42F4N6O4	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-1NC7S1	WO2024208256A1_53	.	COC1=CN2N=C(C3CCC(CCN4CCC(C5=C(F)C=C(C6CCC(=O)NC6=O)C=C5)C(F)(F)C4)CC3)N=C2C=C1C(=O)NC1=CC=CC(C(F)(F)F)=N1	C38H39F6N7O4	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-A2MGV8	WO2024208256A1_54	.	COC1=CN2N=C(C3CCC(CCN4CCC(C5=C(F)C=C(C6CCC(=O)NC6=O)C=C5)C(F)(F)C4)CC3)C=C2C=C1C(=O)NC1=CC=CC(C(F)(F)F)=N1	C39H40F6N6O4	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-FEJW9O	WO2024208256A1_55	.	O=C1CCC(C2=CC(F)=C(C3CCN(CC[C@H]4CC[C@@H](N5C=C6C=C(C(=O)NC7=CC=CC(C(F)(F)F)=N7)C(C7(O)CCC7)=CC6=N5)CC4)CC3(F)F)C=C2)C(=O)N1	C42H44F6N6O4	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-GSQ6AO	WO2024208256A1_56	.	O=C1CCC(C2=CC(F)=C(C3CCN(CC[C@H]4CC[C@@H](N5C=C6C=C(C(=O)NC7=CC=CC(C(F)(F)F)=N7)C(C7(F)CCC7)=CC6=N5)CC4)CC3(F)F)C=C2)C(=O)N1	C42H43F7N6O3	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-2M72WZ	WO2024208256A1_57	.	O=C1CCC(C2=CC(F)=C(C3CCN(CC[C@H]4CC[C@@H](N5C=C6C=C(C(=O)NC7=CC=CC(C(F)(F)F)=N7)C(C7(O)CC7)=CC6=N5)CC4)CC3(F)F)C=C2)C(=O)N1	C41H42F6N6O4	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-E5HSTG	WO2024208256A1_58	.	O=C1CCC(C2=CC(F)=C(C3CCN(CC[C@H]4CC[C@H](N5C=C6C=C(C(=O)NC7=CC=CC(C(F)(F)F)=N7)C(N7CC8(COC8)C7)=CC6=N5)CC4)CC3(F)F)C=C2)C(=O)N1	C43H45F6N7O4	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-D5Y8J5	WO2024208256A1_59	.	O=C1CCC(C2=CC(F)=C(C3CCN(CC[C@H]4CC[C@@H](N5C=C6C=C(C(=O)NC7=CC=CC(C(F)(F)F)=N7)C(C7COC7)=CC6=N5)CC4)CC3(F)F)C=C2)C(=O)N1	C41H42F6N6O4	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-JKWAQ2	WO2024208256A1_60	.	O=C1CCC(C2=CC(F)=C(C3CCN(CC[C@H]4CC[C@@H](N5C=C6C=C(C(=O)NC7=CC=CC(C(F)(F)F)=N7)C(N7CC[C@@H](F)C7)=CC6=N5)CC4)CC3(F)F)C=C2)C(=O)N1	C42H44F7N7O3	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-LYPY63	WO2024208256A1_61	.	O=C1CCC(C2=CC(F)=C(N3CCC(CCN4CCC(N5C=C(C6CC6(F)F)C(C(=O)NC6=CC=CC(C(F)(F)F)=N6)=N5)CC4)CC3)C=C2)C(=O)N1	C36H39F6N7O3	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-MZ8QFP	WO2024208256A1_62	.	CC(C)CN1C2=CC=C(C3CCN(CCC4CCN(C5=C(F)C=C(C6CCC(=O)NC6=O)C=C5)CC4)CC3)C=C2N=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C41H47F4N7O3	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-WJOLCT	WO2024208256A1_63	.	O=C1CCC(C2=CC(F)=C(N3CCC(CCN4CCC(N5C=C(C(=O)NC6=CC=CC(C(F)(F)F)=N6)C(C6CC6(F)F)=N5)CC4)CC3)C=C2)C(=O)N1	C36H39F6N7O3	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-F8BEWG	WO2024208256A1_64	.	CC(C)OC1=NN(C2CCN(CCC3CCN(C4=C(F)C=C(C5CCC(=O)NC5=O)C=C4)CC3)CC2)C=C1NC(=S)N1CCC2=C1N=C(C(F)(F)F)C=C2	C38H46F4N8O3S	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-RJMG9T	WO2024208256A1_65	.	CC(C)OC1=NN(C2CCN(CCC3CCN(C4=C(F)C=C(C5CCC(=O)NC5=O)C=C4)CC3)CC2)C=C1NC(=O)NC1=CC=CC(C(F)(F)F)=N1	C36H44F4N8O4	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-N0RNEF	WO2024208256A1_66	.	CS(=O)(=O)C1=CC2=NN(C3CCN(CCC4CCN(C5=C(F)C=C(C6CCC(=O)NC6=O)C=C5)CC4)CC3)C=C2C=C1C(=O)NC1=CC=CC(C(F)(F)F)=N1	C38H41F4N7O5S	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-X4P0Q5	WO2024208256A1_67	.	CP(C)(=O)C1=CC2=NN(C3CCN(CCC4CCN(C5=C(F)C=C(C6CCC(=O)NC6=O)C=C5)CC4)CC3)C=C2C=C1C(=O)NC1=CC=CC(C(F)(F)F)=N1	C39H44F4N7O4P	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-GYOPAE	WO2024208256A1_68	.	CP(C)(=O)C1=CC(C(=O)NC2=CC=CC(C(F)(F)F)=N2)=CC2=CN(C3CCN(CCC4CCN(C5=C(F)C=C(C6CCC(=O)NC6=O)C=C5)CC4)CC3)N=C21	C39H44F4N7O4P	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-V0JCH1	WO2024208256A1_69	.	COC1=CC2=NN(C3CCN(CCC4CCN(C5=C(F)C=C(C6CCC(=O)NC6=O)C=C5)CC4)CC3)C=C2C=C1S(=O)(=O)N1CCC2=C1N=C(C(F)(F)F)C=C2	C39H43F4N7O5S	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-SEMIC0	WO2024208256A1_70	.	CC(C)(O)C1=CC2=NN(C3CCN(CCC4CCN(C5=C(F)C=C(C6CCC(=O)NC6=O)C=C5)CC4)CC3)C=C2C=C1S(=O)(=O)N1CC2=C(C1)N=C(C(F)(F)F)C=C2	C41H47F4N7O5S	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-GB4OFC	WO2024208256A1_71	.	O=C1CCC(C2=CC(F)=C(N3CCC(CCN4CCC5C(CC6=C(C(=O)NC7=C8N=CC=CN8N=C7)C(C(F)F)=NN65)C4)CC3)C=C2)C(=O)N1	C35H38F3N9O3	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-8Q0PT3	WO2024208256A1_72	.	COC1=CC2=NN(C3CCC4(CC3)CC4CN3CC4(C3)CN(C3=C(F)C=C(C5CCC(=O)NC5=O)C=C3)C4)C=C2C=C1C(=O)NC1=CC=CC(C(F)(F)F)=N1	C40H41F4N7O4	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-X5EF4N	WO2024208256A1_73	.	COC1=CC2=NN(C3CCC(CCN4CCC(C5=C(F)C=C(C6CC67CCC(=O)NC7=O)C=C5)C(F)(F)C4)CC3)C=C2C=C1C(=O)NC1=CC=CC(C(F)(F)F)=N1	C41H42F6N6O4	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-C9BI3Y	WO2024208256A1_74	.	COC1=CC2=NN(C3CCC(CC4CC45CCN(C4=C(F)C=C(C6CCC(=O)NC6=O)C=C4)CC5)CC3)C=C2C=C1C(=O)NC1=CC=CC(C(F)(F)F)=N1	C40H42F4N6O4	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-HPBSG8	WO2024208256A1_75	.	CC(C)(O)C1=CC2=NN(C3CCN(CCC4CCC(C5=CC=C(C6CCC(=O)NC6=O)C=C5F)CC4)CC3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C41H46F4N6O4	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-4CN6YQ	WO2024208256A1_76	.	CC(C)(O)C1=CC2=NN(C3CCN(CCC4CC=C(C5=CC=C(C6CCC(=O)NC6=O)C=C5F)CC4)CC3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C41H44F4N6O4	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-E3BI1N	WO2024208256A1_77	.	COC1=CC2=NN(C3CCN(C4CC5(CCC(C6=C(F)C=C(C7CCC(=O)NC7=O)C=C6)CC5)C4)CC3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C40H42F4N6O4	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-20LHFM	WO2024208256A1_78	.	COC1=CC2=NN(C3CCN(CC4CC5(CCC(C6=C(F)C=C(C7CCC(=O)NC7=O)C=C6)CC5)C4)CC3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C41H44F4N6O4	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-MOLDCY	WO2024208256A1_79	.	CC(C)(O)C1=CC2=NN(C3CCN(CCC4CCC(C5=C(F)C=C(C6CCC(=O)NC6=O)C=C5)CC4)CC3(F)F)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C41H44F6N6O4	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-RBF4O7	WO2024208256A1_80	.	CC(C)(O)C1=CC2=NN(C3CCN(CC4CCC(OC5=CC=C(C6CCC(=O)NC6=O)C=C5F)CC4)CC3(F)F)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C40H42F6N6O5	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-IFAT23	WO2024208256A1_81	.	COC1=CC2=NN(C3CCC(OC4CC5(CCC(C6=C(F)C=C(C7CCC(=O)NC7=O)C=C6)CC5)C4)CC3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C41H43F4N5O5	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-QALAZT	WO2024208256A1_82	.	COC1=CC2=NN(C3CCC(OC4CC5(CCC(C6=C(F)C=C(C7CCC(=O)NC7=O)C=C6)C5)C4)CC3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C40H41F4N5O5	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-C3IU0A	WO2024208256A1_83	.	CC(C)OC1=CC2=NN(C3CCN(CCC4CCC(C5=C(F)C=C(C6CCC(=O)NC6=O)C=C5)CC4)CC3(F)F)C=C2C=C1C(=O)NC1=C2N=CC=CN2N=C1	C41H45F3N8O4	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-O7S0LY	WO2024208256A1_84	.	CC(C)OC1=CC2=NN(C3CCN(CCC4CCC(C5=C(F)C=C(C6CCC(=O)NC6=O)C=C5)CC4)CC3(F)F)C=C2C=C1C(=O)NC1=CC=CC(C(F)F)=N1	C41H45F5N6O4	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-TC3V5Z	WO2024208256A1_85	.	COC1=CC2=NN(C3=NC=C(COC4CCN(C5=CC=C(C6CCC(=O)NC6=O)C=C5F)CC4(F)F)C=C3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C37H31F6N7O5	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-T3TLX1	WO2024208256A1_86	.	COC1=CC2=NN(C3CCC(CCN4C=C(C5=CC=C(C6CCC(=O)NC6=O)C=C5F)C=N4)CC3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C37H35F4N7O4	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-X2LI2I	WO2024208256A1_87	.	COC1=CC2=NN(C3CCC(CCC4=NN=C(C5=CC=C(C6CCC(=O)NC6=O)C=C5F)O4)CC3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C36H33F4N7O5	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-29M502	WO2024208256A1_88	.	O=C1CCC(C2=CC(F)=C(N3CCC(CCN4CCC(N5C=C(NC(=O)C6=C7N=CC=CN7N=C6)C(C(F)F)=N5)CC4)CC3)C=C2)C(=O)N1	C34H38F3N9O3	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-NEP8JG	WO2024208256A1_89	.	O=C1CCC(C2=CC(F)=C(N3CCC(CCN4CCC(N5C=C(C(=O)NC6=C7N=CC=CN7N=C6)C(C(F)F)=N5)CC4)CC3)C=C2)C(=O)N1	C34H38F3N9O3	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-D6UZSC	WO2024208256A1_90	.	CC(C)OC1=CC2=NN(C3CCN(CCC4(O)CCN(C5=C(F)C=C(C6=NNC(=O)CC6)C(F)=C5)CC4)CC3)C=C2C=C1C(=O)NC1=NC(C(F)F)=CC=C1	C39H44F4N8O4	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-RVS5JB	WO2024208256A1_91	.	CC(C)OC1=CC2=NN(C3CCC(CCN4CCC(C5=C(F)C=C(C6=NNC(=O)CC6)C=C5)C(F)(F)C4)CC3)C=C2C=C1C(=O)NC1=CC=CC(C(F)F)=N1	C40H44F5N7O3	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-K4NNYX	WO2024208256A1_92	.	CC(C)OC1=CC2=NC(C3CCC(CN(C)C4CCN(C5=CC=C(C6=NNC(=O)C=C6)C=C5F)CC4(F)F)CC3)=CN2C=C1C(=O)NC1=NC(C(F)F)=CC=C1	C40H43F5N8O3	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-NTR33Z	WO2024208256A1_93	.	CC(C)OC1=CC2=NC(C3CCC(COC4CCN(C5=CC=C(C6=NNC(=O)C=C6)C=C5F)CC4(F)F)CC3)=CN2C=C1C(=O)NC1=NC(C(F)F)=CC=C1	C39H40F5N7O4	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-M45JMI	WO2024208256A1_94	.	CC(C)OC1=CC2=NN(C3CCC(CN4CC5(CCC(C6=C(F)C=C(C7=NNC(=O)C=C7)C=C6)CC5)C4)CC3)C=C2C=C1C(=O)NC1=CC=CN([C@@H]2C[C@@H]2F)C1=O	C44H49F2N7O4	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-V8VU63	WO2024208256A1_95	.	CC(C)OC1=CC2=NN(C3CCC(CN4CCC(C5=CC=C(C6=NNC(=O)CC6)C=C5)C(F)(F)C4)CC3)C=C2C=C1C(=O)NC1=CC=CN([C@@H]2C[C@@H]2F)C1=O	C41H46F3N7O4	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-9BY52A	WO2024208256A1_96	.	COC1=CC2=NN(C3CCC(CCN4CCC(C5=C(F)C=C(C6CC7(CCC(=O)NC7=O)C6)C=C5)C(F)(F)C4)CC3)C=C2C=C1C(=O)NC1=CC=CC(C(F)F)=N1	C42H45F5N6O4	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-B3YZ6J	WO2024208256A1_97	.	COC1=CC2=NN(C3C[C@@H]4C(CCN5CCC(C6=NC=C(C7(F)CCC(=O)NC7=O)C=C6)C(F)(F)C5)[C@@H]4C3)C=C2C=C1C(=O)NC1=CC=CC(C(F)(F)F)=N1	C38H37F6N7O4	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-IAQEH8	WO2024208256A1_98	.	CC(C)(O)C1=CC2=NN(C3CCC(CCN4CCC(C5=C(F)C=C(C6CC67CCC(=O)NC7=O)C=C5)C(F)(F)C4)CC3)C=C2C=C1C(=O)NC1=CC=CC(C(F)(F)F)=N1	C43H46F6N6O4	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-CSJLPQ	WO2024208256A1_99	.	COC1=CC2=NN(C3CCC(CCN4CCC(C5=NC=C(C6(F)CCC(=O)NC6=O)C=C5)C(F)(F)C4)CC3)C=C2C=C1C(=O)NC1=CC=CC(C(F)(F)F)=N1	C38H39F6N7O4	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-6D92CL	WO2024208256A1_100	.	COC1=CC2=NN(C3CCC(CCN4CCC(C5=C(F)C=C(N6CCC(=O)NC6=O)C=C5)C(F)(F)C4)CC3)C=C2C=C1C(=O)NC1=CC=CC(C(F)(F)F)=N1	C38H39F6N7O4	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-DZ3J4Z	WO2024208256A1_101	.	COC1=CC2=NN(C3CCC(CCN4CCC(C5=C(F)C=C(N6CCC(=O)NC6=O)C=N5)C(F)(F)C4)CC3)C=C2C=C1C(=O)NC1=CC=CC(C(F)(F)F)=N1	C37H38F6N8O4	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-CJJIKD	WO2024208256A1_104	.	CC(C)(O)C1=CC2=NN([C@H]3CC[C@@H](CN4CCN5C(=CC6=C5CCN(C5CCC(=O)NC5=O)C6)C4)CC3)C=C2C=C1C(=O)NC1=CC=CC(C(F)(F)F)=N1	C39H45F3N8O4	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-NWYBNQ	WO2024208256A1_105	.	CC(C)(O)C1=CC2=NN([C@H]3CC[C@H](CN4CCC5=C(C=C6CN(C7CCC(=O)NC7=O)CCN65)C4)CC3)C=C2C=C1C(=O)NC1=CC=CC(C(F)(F)F)=N1	C39H45F3N8O4	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-JNIGRM	WO2024208256A1_106	.	COC1=C(C(=O)NC2=CC=CC(C(F)(F)F)=N2)C=C2N=C3CC4(CCN3C2=C1)CN(C1CCN(C2=C(F)C=C(C3CCC(=O)NC3=O)C=C2)CC1(F)F)C4	C37H35F6N7O4	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-6NVJGY	WO2024208256A1_107	.	COC1=C(C(=O)NC2=CC=CC(C(F)(F)F)=N2)C=C2N=C3CC4(CCN3C2=C1)CN(CC1CCN(C2=C(F)C=C(C3CCC(=O)NC3=O)C=C2)CC1(F)F)C4	C38H37F6N7O4	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-OLRMNU	WO2024208256A1_110	.	CC(C)(O)C1=CC2=NN([C@H]3CC[C@@H](CN4CCC(C5=C(F)C=C(C6CC7(CCC(=O)NC7=O)C6)C=N5)CC4)CC3)C=C2C=C1C(=O)NC1=CC=CC(C(F)(F)F)=N1	C42H47F4N7O4	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-YFZ6J7	WO2024208256A1_111	.	CC(C)(O)C1=CC2=NN([C@H]3CC[C@H](CN4CCC(C5=CC=C(C6CC67CCC(=O)NC7=O)C=C5)CC4)CC3)C=C2C=C1C(=O)NC1=CC=CC(C(F)(F)F)=N1	C42H47F3N6O4	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-JYVNYE	WO2024208256A1_112	.	COC1=CC2=NN(C3CCN(CC4CCN(C5=C(F)C=C(C6CCC(=O)NC6=O)C=C5)CC4)CC3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C37H39F4N7O4	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-71P6CM	WO2024208256A1_113	.	COC1=CC2=NN([C@H]3CC[C@@H](CN4CCC5(CC4)CCN(C4=C(F)C=C(C6CCC(=O)NC6=O)C=C4)CC5)CC3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C42H47F4N7O4	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-NPSM0Z	WO2024208256A1_114	.	COC1=CC2=NN([C@H]3CC[C@H](CN(C)C4CCN(C5=C(F)C=C(C6CCC(=O)NC6=O)C=C5)CC4)CC3)C=C2C=C1CNC(=O)C1=CC=CC(C(F)(F)F)=N1	C40H45F4N7O4	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-YVIP99	WO2024208256A1_115	.	COC1=CC2=NN([C@H]3CC[C@H](CN(C)C4CCN(C5=C(F)C=C(C6CCC(=O)NC6=O)C=C5)CC4)CC3)C=C2C=C1NC(=O)C(C)(C)C1=CC=CC(C(F)(F)F)=N1	C42H49F4N7O4	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-IQWK6Y	WO2024208256A1_116	.	CN(C[C@H]1CC[C@H](N2C=C(NC(=O)CC3=C4N=C(N5C[C@@H]6C[C@H]5CO6)C=CN4N=C3)C(C(F)F)=N2)CC1)C1CCN(C2=C(F)C=C(C3CCC(=O)NC3=O)C=C2)CC1	C41H49F3N10O4	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-QCM65L	WO2024208256A1_117	.	CN(C[C@H]1CC[C@H](N2C=C(NC(=O)C(F)(F)C3=C4N=C(N5C[C@@H]6C[C@H]5CO6)C=CN4N=C3)C(C(F)F)=N2)CC1)C1CCN(C2=C(F)C=C(C3CCC(=O)NC3=O)C=C2)CC1	C41H47F5N10O4	IRAK4	Q9NWZ3	CRBN	WO-2024208256-A1
TPD-29EDS5	WO2024208300A1_4	.	O=C1CCC(N2C(=O)C3=CC=C(N4CCC(CN5CCC(NC6=CC7=C(C=C6)C6=C(N=NC(C8=C(O)C=CC=C8)=C6)NC7=O)CC5)CC4)C=C3C2=O)C(=O)N1	C41H40N8O6	SMARCA2	P51531	CRBN	WO-2024208300-A1
TPD-RK2TBW	WO2024208300A1_5	.	O=C1CCC(N2C(=O)C3=CC=C(N4CCC(CN5CCN(C(=O)C6=CC7=C(C=C6)C6=C(N=NC(C8=C(O)C=CC=C8)=C6)NC7=O)CC5)CC4)C=C3C2=O)C(=O)N1	C41H38N8O7	SMARCA2	P51531	CRBN	WO-2024208300-A1
TPD-1C2RV0	WO2024208300A1_6	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=C1C1=CC=C(N3CCC(CN4CCC(NC5=CC6=C(C=C5)C5=C(NNC(C7=C(O)C=CC=C7)=C5)NC6=O)CC4)CC3)C=C1C=C2	C45H47N9O5	SMARCA2	P51531	CRBN	WO-2024208300-A1
TPD-CKUU8O	WO2024208300A1_7	.	O=C1CCC(C2=CC=C(C3CCN(CC(=O)N4CCN(C(=O)C5=CC6=C(C=C5)C5=C(N=NC(C7=C(O)C=CC=C7)=C5)NC6=O)CC4)CC3)C=C2)C(=O)N1	C40H39N7O6	SMARCA2	P51531	CRBN	WO-2024208300-A1
TPD-LRZT2K	WO2024208300A1_8	.	O=C1CCC(N2C(=O)C3=CC=C(N4CCC(CN5CCN(C6=CC=C7C(=C6)C(=O)NC6=NN=C(C8=C(O)C=CC=C8)C=C76)CC5)CC4)C=C3C2=O)C(=O)N1	C40H38N8O6	SMARCA2	P51531	CRBN	WO-2024208300-A1
TPD-PSOU1B	WO2024214019A1_1	3-[6-[1-[1-(4-bromo-7-cyclopentyl-5-oxobenzimidazolo[1,2-a]quinazolin-9-yl)piperidin-4-yl]piperidin-4-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(C4CCN(C5CCN(C6=CC7=C(C=C6)N6C8=CC=CC(Br)=C8C(=O)N=C6N7C6CCCC6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C42H44BrN7O4	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024214019-A1
TPD-3OKFU2	WO2024214019A1_2	3-[4-[1-[1-(4-Bromo-7-cyclopentyl-5-oxobenzimidazolo[1,2-a]quinazolin-9-yl)piperidin-4-yl]piperidin-4-yl]phenoxy]piperidine-2,6-dione	O=C1CCC(OC2=CC=C(C3CCN(C4CCN(C5=CC6=C(C=C5)N5C7=CC=CC(Br)=C7C(=O)N=C5N6C5CCCC5)CC4)CC3)C=C2)C(=O)N1	C40H43BrN6O4	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024214019-A1
TPD-HPVDWL	WO2024214019A1_3	3-[4-[1-[1-(4-Bromo-7-cyclopentyl-5-oxobenzimidazolo[1,2-a]quinazolin-9-yl)piperidin-4-yl]piperidin-4-yl]-3-fluoroanilino]piperidine-2,6-dione	O=C1CCC(NC2=CC(F)=C(C3CCN(C4CCN(C5=CC6=C(C=C5)N5C7=CC=CC(Br)=C7C(=O)N=C5N6C5CCCC5)CC4)CC3)C=C2)C(=O)N1	C40H43BrFN7O3	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024214019-A1
TPD-6HPN9T	WO2024214019A1_4	3-[4-[1-[1-(4-Bromo-7-cyclopentyl-5-oxobenzimidazolo[1,2-a]quinazolin-9-yl)piperidin-4-yl]piperidin-4-yl]phenyl]piperidine-2,6-dione	O=C1CCC(C2=CC=C(C3CCN(C4CCN(C5=CC6=C(C=C5)N5C7=CC=CC(Br)=C7C(=O)N=C5N6C5CCCC5)CC4)CC3)C=C2)C(=O)N1	C40H43BrN6O3	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024214019-A1
TPD-221712	WO2024214019A1_5	5-[4-(4-Bromo-7-cyclopentyl-5-oxobenzimidazolo[1,2-a]quinazolin-9-yl)piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC=C(N4CCN(C5=CC6=C(C=C5)N5C7=CC=CC(Br)=C7C(=O)N=C5N6C5CCCC5)CC4)C=C3C2=O)C(=O)N1	C36H32BrN7O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024214019-A1
TPD-NYSJ8Q	WO2024214019A1_6	3-[4-[4-[1-(4-Bromo-7-cyclopentyl-5-oxobenzimidazolo[1,2-a]quinazolin-9-yl)piperidin-4-yl]piperazin-1-yl]phenyl]piperidine-2,6-dione	O=C1CCC(C2=CC=C(N3CCN(C4CCN(C5=CC6=C(C=C5)N5C7=CC=CC(Br)=C7C(=O)N=C5N6C5CCCC5)CC4)CC3)C=C2)C(=O)N1	C39H42BrN7O3	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024214019-A1
TPD-G944Q2	WO2024214019A1_7	3-[6-[1-[1-[1-(4-bromo-7-cyclopentyl-5-oxobenzimidazolo[1,2-a]quinazolin-9-yl)piperidin-4-yl]piperidin-4-yl]piperidin-4-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(C4CCN(C5CCN(C6CCN(C7=CC8=C(C=C7)N7C9=CC=CC(Br)=C9C(=O)N=C7N8C7CCCC7)CC6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C47H53BrN8O4	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024214019-A1
TPD-VR9YFZ	WO2024214019A1_8	3-[6-[1-[1-(4-amino-7-cyclopentyl-5-oxobenzimidazolo[1,2-a]quinazolin-9-yl)piperidin-4-yl]piperidin-4-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	NC1=C2C(=O)N=C3N(C2=CC=C1)C1=C(C=C(N2CCC(N4CCC(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)CC6=C5)CC4)CC2)C=C1)N3C1CCCC1	C42H46N8O4	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024214019-A1
TPD-JT8R5E	WO2024214019A1_9	3-[6-[1-[1-(4-chloro-7-cyclopentyl-5-oxobenzimidazolo[1,2-a]quinazolin-9-yl)piperidin-4-yl]piperidin-4-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(C4CCN(C5CCN(C6=CC7=C(C=C6)N6C8=CC=CC(Cl)=C8C(=O)N=C6N7C6CCCC6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C42H44ClN7O4	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024214019-A1
TPD-P3MRWZ	WO2024214019A1_10	3-[6-[1-[1-(7-cyclopentyl-5-oxobenzimidazolo[1,2-a]quinazolin-9-yl)piperidin-4-yl]piperidin-4-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(C4CCN(C5CCN(C6=CC7=C(C=C6)N6C8=CC=CC=C8C(=O)N=C6N7C6CCCC6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C42H45N7O4	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024214019-A1
TPD-A4M313	WO2024214019A1_11	3-[4-[1-[1-(7-Cyclopentyl-4-methoxy-5-oxobenzimidazolo[1,2-a]quinazolin-9-yl)piperidin-4-yl]piperidin-4-yl]-3-fluoroanilino]piperidine-2,6-dione	COC1=C2C(=O)N=C3N(C2=CC=C1)C1=C(C=C(N2CCC(N4CCC(C5=C(F)C=C(NC6CCC(=O)NC6=O)C=C5)CC4)CC2)C=C1)N3C1CCCC1	C41H46FN7O4	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024214019-A1
TPD-GLQCHK	WO2024214019A1_12	3-[4-[1-[1-(7-Cyclopentyl-4-hydroxy-5-oxobenzimidazolo[1,2-a]quinazolin-9-yl)piperidin-4-yl]piperidin-4-yl]-3-fluoroanilino]piperidine-2,6-dione	O=C1CCC(NC2=CC(F)=C(C3CCN(C4CCN(C5=CC6=C(C=C5)N5C7=CC=CC(O)=C7C(=O)N=C5N6C5CCCC5)CC4)CC3)C=C2)C(=O)N1	C40H44FN7O4	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024214019-A1
TPD-G8E9O2	WO2024214019A1_13	3-[4-[1-[1-[7-Cyclopentyl-5-oxo-4-(trifluoromethyl)benzimidazolo[1,2-a]quinazolin-9-yl]piperidin-4-yl]piperidin-4-yl]phenyl]piperidine-2,6-dione	O=C1CCC(C2=CC=C(C3CCN(C4CCN(C5=CC6=C(C=C5)N5C7=CC=CC(C(F)(F)F)=C7C(=O)N=C5N6C5CCCC5)CC4)CC3)C=C2)C(=O)N1	C41H43F3N6O3	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024214019-A1
TPD-AXNOEH	WO2024214019A1_14	3-[6-[1-[1-(4-bromo-7-methyl-5-oxobenzimidazolo[1,2-a]quinazolin-9-yl)piperidin-4-yl]piperidin-4-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CN1C2=NC(=O)C3=C(Br)C=CC=C3N2C2=C1C=C(N1CCC(N3CCC(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)CC5=C4)CC3)CC1)C=C2	C38H38BrN7O4	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024214019-A1
TPD-S8G5SZ	WO2024214019A1_15	3-[6-[1-[1-(4-amino-7-methyl-5-oxobenzimidazolo[1,2-a]quinazolin-9-yl)piperidin-4-yl]piperidin-4-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CN1C2=NC(=O)C3=C(N)C=CC=C3N2C2=C1C=C(N1CCC(N3CCC(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)CC5=C4)CC3)CC1)C=C2	C38H40N8O4	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024214019-A1
TPD-9YV8U7	WO2024214019A1_16	3-[4-[1-[1-(4-Bromo-7-methyl-5-oxobenzimidazolo[1,2-a]quinazolin-9-yl)piperidin-4-yl]piperidin-4-yl]-3-fluoroanilino]piperidine-2,6-dione	CN1C2=NC(=O)C3=C(Br)C=CC=C3N2C2=C1C=C(N1CCC(N3CCC(C4=C(F)C=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC1)C=C2	C36H37BrFN7O3	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024214019-A1
TPD-BR7ZZW	WO2024214019A1_17	3-[4-[1-[1-(4-Bromo-7-methyl-5-oxobenzimidazolo[1,2-a]quinazolin-9-yl)piperidin-4-yl]piperidin-4-yl]phenyl]piperidine-2,6-dione	CN1C2=NC(=O)C3=C(Br)C=CC=C3N2C2=C1C=C(N1CCC(N3CCC(C4=CC=C(C5CCC(=O)NC5=O)C=C4)CC3)CC1)C=C2	C36H37BrN6O3	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024214019-A1
TPD-MD4GIX	WO2024214019A1_18	3-[4-[1-[1-(4-Amino-7-methyl-5-oxobenzimidazolo[1,2-a]quinazolin-9-yl)piperidin-4-yl]piperidin-4-yl]phenyl]piperidine-2,6-dione	CN1C2=NC(=O)C3=C(N)C=CC=C3N2C2=C1C=C(N1CCC(N3CCC(C4=CC=C(C5CCC(=O)NC5=O)C=C4)CC3)CC1)C=C2	C36H39N7O3	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024214019-A1
TPD-9VN333	WO2024214019A1_19	3-[6-[1-[1-(11-cyclopentyl-8-oxo-1,5,9,11-tetrazatetracyclo[8.7.0.02,7.012,17]heptadeca-2(7),3,5,9,12(17),13,15-heptaen-14-yl)piperidin-4-yl]piperidin-4-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(C4CCN(C5CCN(C6=CC7=C(C=C6)N6C8=CC=NC=C8C(=O)N=C6N7C6CCCC6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C41H44N8O4	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024214019-A1
TPD-XI8KVQ	WO2024214019A1_21	3-[4-[1-[1-(4-Amino-5-oxo-7-propan-2-ylbenzimidazolo[1,2-a]quinazolin-9-yl)piperidin-4-yl]piperidin-4-yl]phenyl]piperidine-2,6-dione	CC(C)N1C2=NC(=O)C3=C(N)C=CC=C3N2C2=C1C=C(N1CCC(N3CCC(C4=CC=C(C5CCC(=O)NC5=O)C=C4)CC3)CC1)C=C2	C38H43N7O3	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024214019-A1
TPD-77JWUD	WO2024214019A1_22	3-[4-[1-[1-(4-Chloro-7-cyclopentyl-5-oxobenzimidazolo[1,2-a]quinazolin-9-yl)piperidin-4-yl]piperidin-4-yl]phenyl]piperidine-2,6-dione	O=C1CCC(C2=CC=C(C3CCN(C4CCN(C5=CC6=C(C=C5)N5C7=CC=CC(Cl)=C7C(=O)N=C5N6C5CCCC5)CC4)CC3)C=C2)C(=O)N1	C40H43ClN6O3	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024214019-A1
TPD-STYHS1	WO2024214019A1_23	3-[4-[1-[1-(4-Chloro-7-cyclopentyl-5-oxobenzimidazolo[1,2-a]quinazolin-9-yl)piperidin-4-yl]piperidin-4-yl]-3-fluoroanilino]piperidine-2,6-dione	O=C1CCC(NC2=CC(F)=C(C3CCN(C4CCN(C5=CC6=C(C=C5)N5C7=CC=CC(Cl)=C7C(=O)N=C5N6C5CCCC5)CC4)CC3)C=C2)C(=O)N1	C40H43ClFN7O3	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024214019-A1
TPD-W3AAU9	WO2024214019A1_24	3-[4-[1-[1-(11-Cyclopentyl-8-oxo-1,6,9,11-tetrazatetracyclo[8.7.0.02,7.012,17]heptadeca-2(7),3,5,9,12(17),13,15-heptaen-14-yl)piperidin-4-yl]piperidin-4-yl]phenyl]piperidine-2,6-dione	O=C1CCC(C2=CC=C(C3CCN(C4CCN(C5=CC6=C(C=C5)N5C7=CC=CN=C7C(=O)N=C5N6C5CCCC5)CC4)CC3)C=C2)C(=O)N1	C39H43N7O3	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024214019-A1
TPD-ZAZ4Q4	WO2024214019A1_25	3-[4-[1-[1-(4-Amino-7-cyclopentyl-5-oxobenzimidazolo[1,2-a]quinazolin-9-yl)piperidin-4-yl]piperidin-4-yl]phenyl]piperidine-2,6-dione	NC1=C2C(=O)N=C3N(C2=CC=C1)C1=C(C=C(N2CCC(N4CCC(C5=CC=C(C6CCC(=O)NC6=O)C=C5)CC4)CC2)C=C1)N3C1CCCC1	C40H45N7O3	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024214019-A1
TPD-M7CKYX	WO2024214019A1_26	3-[4-[4-[1-(4-Amino-7-cyclopentyl-5-oxobenzimidazolo[1,2-a]quinazolin-9-yl)piperidin-4-yl]piperazin-1-yl]phenyl]piperidine-2,6-dione	NC1=C2C(=O)N=C3N(C2=CC=C1)C1=C(C=C(N2CCC(N4CCN(C5=CC=C(C6CCC(=O)NC6=O)C=C5)CC4)CC2)C=C1)N3C1CCCC1	C39H44N8O3	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024214019-A1
TPD-L38XHY	WO2024214019A1_27	3-[6-[1-[1-(4-chloro-7-methyl-5-oxobenzimidazolo[1,2-a]quinazolin-9-yl)piperidin-4-yl]piperidin-4-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CN1C2=NC(=O)C3=C(Cl)C=CC=C3N2C2=C1C=C(N1CCC(N3CCC(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)CC5=C4)CC3)CC1)C=C2	C38H38ClN7O4	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024214019-A1
TPD-88ROJG	WO2024214019A1_28	3-[6-[1-[1-(4-chloro-5-oxo-7-propan-2-ylbenzimidazolo[1,2-a]quinazolin-9-yl)piperidin-4-yl]piperidin-4-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CC(C)N1C2=NC(=O)C3=C(Cl)C=CC=C3N2C2=C1C=C(N1CCC(N3CCC(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)CC5=C4)CC3)CC1)C=C2	C40H42ClN7O4	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024214019-A1
TPD-W8OAWK	WO2024214019A1_29	3-[4-[1-[1-(4-Chloro-5-oxo-7-propan-2-ylbenzimidazolo[1,2-a]quinazolin-9-yl)piperidin-4-yl]piperidin-4-yl]-3-fluoroanilino]piperidine-2,6-dione	CC(C)N1C2=NC(=O)C3=C(Cl)C=CC=C3N2C2=C1C=C(N1CCC(N3CCC(C4=C(F)C=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC1)C=C2	C38H41ClFN7O3	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024214019-A1
TPD-27Q6Z0	WO2024214019A1_30	3-[6-[4-[1-(4-chloro-7-cyclopentyl-5-oxobenzimidazolo[1,2-a]quinazolin-9-yl)piperidin-4-yl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(N4CCN(C5CCN(C6=CC7=C(C=C6)N6C8=CC=CC(Cl)=C8C(=O)N=C6N7C6CCCC6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C41H43ClN8O4	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024214019-A1
TPD-FC8OVC	WO2024214019A1_31	.	NC1=C2C(=O)N=C3NC4=C(C=CC(N5CCC(N6CCC(C7=CC=C(C8CCC(=O)NC8=O)C=C7)CC6)CC5)=C4)N3C2=CC=C1	C35H37N7O3	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024214019-A1
TPD-7AV07V	WO2024214019A1_32	3-[4-[4-[1-(4-Amino-7-methyl-5-oxobenzimidazolo[1,2-a]quinazolin-9-yl)piperidin-4-yl]piperazin-1-yl]phenyl]piperidine-2,6-dione	CN1C2=NC(=O)C3=C(N)C=CC=C3N2C2=C1C=C(N1CCC(N3CCN(C4=CC=C(C5CCC(=O)NC5=O)C=C4)CC3)CC1)C=C2	C35H38N8O3	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024214019-A1
TPD-JTPGCG	WO2024214019A1_33	3-[4-[1-[1-(7-Cyclopentyl-4-methyl-5-oxobenzimidazolo[1,2-a]quinazolin-9-yl)piperidin-4-yl]piperidin-4-yl]-3-fluoroanilino]piperidine-2,6-dione	CC1=C2C(=O)N=C3N(C2=CC=C1)C1=C(C=C(N2CCC(N4CCC(C5=C(F)C=C(NC6CCC(=O)NC6=O)C=C5)CC4)CC2)C=C1)N3C1CCCC1	C41H46FN7O3	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024214019-A1
TPD-E071S5	WO2024214019A1_34	3-[4-[1-[1-(4-bromo-5-oxo-6H-benzimidazolo[1,2-a]quinazolin-9-yl)piperidin-4-yl]piperidin-4-yl]-3-fluoroanilino]piperidine-2,6-dione	O=C1CCC(NC2=CC(F)=C(C3CCN(C4CCN(C5=CC6=C(C=C5)N5C7=CC=CC(Br)=C7C(=O)N=C5N6)CC4)CC3)C=C2)C(=O)N1	C35H35BrFN7O3	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024214019-A1
TPD-ZNJ1AL	WO2024214019A1_35	3-[4-[4-[1-(4-Chloro-7-cyclopentyl-5-oxobenzimidazolo[1,2-a]quinazolin-9-yl)piperidin-4-yl]piperazin-1-yl]-3-fluoroanilino]piperidine-2,6-dione	O=C1CCC(NC2=CC(F)=C(N3CCN(C4CCN(C5=CC6=C(C=C5)N5C7=CC=CC(Cl)=C7C(=O)N=C5N6C5CCCC5)CC4)CC3)C=C2)C(=O)N1	C39H42ClFN8O3	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024214019-A1
TPD-6UH7L6	WO2024214019A1_36	3-[4-[1-[1-(4-Chloro-7-methyl-5-oxobenzimidazolo[1,2-a]quinazolin-9-yl)piperidin-4-yl]piperidin-4-yl]-3-fluoroanilino]piperidine-2,6-dione	CN1C2=NC(=O)C3=C(Cl)C=CC=C3N2C2=C1C=C(N1CCC(N3CCC(C4=C(F)C=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC1)C=C2	C36H37ClFN7O3	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024214019-A1
TPD-9SUQ4D	WO2024214019A1_37	.	NC1=C2C(=O)N=C3N(C2=CC=C1)C1=C(C=C(N2CCC(N4CCN(C5=C(F)C=C(NC6CCC(=O)NC6=O)C=C5)CC4)CC2)C=C1)N3C1CC1	C37H40FN9O3	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024214019-A1
TPD-KFR2OQ	WO2024214019A1_39	4-[1-[1-(4-chloro-7-cyclopentyl-5-oxobenzimidazolo[1,2-a]quinazolin-9-yl)piperidin-4-yl]piperidin-4-yl]-N-(2,6-dioxopiperidin-3-yl)-2-fluorobenzamide	O=C1CCC(NC(=O)C2=C(F)C=C(C3CCN(C4CCN(C5=CC6=C(C=C5)N5C7=CC=CC(Cl)=C7C(=O)N=C5N6C5CCCC5)CC4)CC3)C=C2)C(=O)N1	C41H43ClFN7O4	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024214019-A1
TPD-C6BD54	WO2024214019A1_40	3-[4-[4-[1-(4-Amino-7-methyl-5-oxobenzimidazolo[1,2-a]quinazolin-9-yl)piperidin-4-yl]piperazin-1-yl]-3-fluoroanilino]piperidine-2,6-dione	CN1C2=NC(=O)C3=C(N)C=CC=C3N2C2=C1C=C(N1CCC(N3CCN(C4=C(F)C=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC1)C=C2	C35H38FN9O3	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024214019-A1
TPD-IV83JA	WO2024214019A1_41	1-[6-[4-[1-(4-Amino-7-methyl-5-oxobenzimidazolo[1,2-a]quinazolin-9-yl)piperidin-4-yl]piperazin-1-yl]-5-fluoro-1-methylindazol-3-yl]-1,3-diazinane-2,4-dione	CN1N=C(N2CCC(=O)NC2=O)C2=C1C=C(N1CCN(C3CCN(C4=CC5=C(C=C4)N4C6=CC=CC(N)=C6C(=O)N=C4N5C)CC3)CC1)C(F)=C2	C36H38FN11O3	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024214019-A1
TPD-92DGPY	WO2024214019A1_42	3-[6-[4-[1-(4-amino-7-methyl-5-oxobenzimidazolo[1,2-a]quinazolin-9-yl)piperidin-4-yl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CN1C2=NC(=O)C3=C(N)C=CC=C3N2C2=C1C=C(N1CCC(N3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)CC5=C4)CC3)CC1)C=C2	C37H39N9O4	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024214019-A1
TPD-AGTN8J	WO2024214019A1_43	3-[6-[4-[[4-(4-amino-7-methyl-5-oxobenzimidazolo[1,2-a]quinazolin-9-yl)piperazin-1-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CN1C2=NC(=O)C3=C(N)C=CC=C3N2C2=C1C=C(N1CCN(CC3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)CC5=C4)CC3)CC1)C=C2	C38H41N9O4	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024214019-A1
TPD-B1BX2H	WO2024214019A1_44	3-[4-[4-[1-(4-Amino-5-oxo-7-propan-2-ylbenzimidazolo[1,2-a]quinazolin-9-yl)piperidin-4-yl]piperazin-1-yl]phenyl]piperidine-2,6-dione	CC(C)N1C2=NC(=O)C3=C(N)C=CC=C3N2C2=C1C=C(N1CCC(N3CCN(C4=CC=C(C5CCC(=O)NC5=O)C=C4)CC3)CC1)C=C2	C37H42N8O3	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024214019-A1
TPD-7N9OT7	WO2024214019A1_45	5-[3-[4-(4-Amino-7-methyl-5-oxobenzimidazolo[1,2-a]quinazolin-9-yl)piperazin-1-yl]azetidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN1C2=NC(=O)C3=C(N)C=CC=C3N2C2=C1C=C(N1CCN(C3CN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)C3)CC1)C=C2	C35H33N9O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024214019-A1
TPD-UMPQ21	WO2024214019A1_46	3-[4-[4-[1-(4-Chloro-7-methyl-5-oxobenzimidazolo[1,2-a]quinazolin-9-yl)piperidin-4-yl]piperazin-1-yl]-3-fluoroanilino]piperidine-2,6-dione	CN1C2=NC(=O)C3=C(Cl)C=CC=C3N2C2=C1C=C(N1CCC(N3CCN(C4=C(F)C=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC1)C=C2	C35H36ClFN8O3	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024214019-A1
TPD-S7XSN3	WO2024214019A1_47	3-[4-[4-[1-(4-Chloro-5-oxo-7-propan-2-ylbenzimidazolo[1,2-a]quinazolin-9-yl)piperidin-4-yl]piperazin-1-yl]-3-fluoroanilino]piperidine-2,6-dione	CC(C)N1C2=NC(=O)C3=C(Cl)C=CC=C3N2C2=C1C=C(N1CCC(N3CCN(C4=C(F)C=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC1)C=C2	C37H40ClFN8O3	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024214019-A1
TPD-O7DDGQ	WO2024214019A1_48	3-[6-[4-[1-(4-chloro-5-oxo-7-propan-2-ylbenzimidazolo[1,2-a]quinazolin-9-yl)piperidin-4-yl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CC(C)N1C2=NC(=O)C3=C(Cl)C=CC=C3N2C2=C1C=C(N1CCC(N3CCN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5)CC3)CC1)C=C2	C39H41ClN8O4	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024214019-A1
TPD-RCZRKN	WO2024214019A1_49	3-[4-[4-[4-(4-Amino-7-methyl-5-oxobenzimidazolo[1,2-a]quinazolin-9-yl)phenyl]piperazin-1-yl]-3-fluoroanilino]piperidine-2,6-dione	CN1C2=NC(=O)C3=C(N)C=CC=C3N2C2=C1C=C(C1=CC=C(N3CCN(C4=C(F)C=C(NC5CCC(=O)NC5=O)C=C4)CC3)C=C1)C=C2	C36H33FN8O3	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024214019-A1
TPD-TI9OIZ	SCHEMBL31170907	3-[4-[4-[4-(4-Chloro-5-oxo-7-propan-2-ylbenzimidazolo[1,2-a]quinazolin-9-yl)phenyl]piperazin-1-yl]-3-fluoroanilino]piperidine-2,6-dione	CC(C)N1C2=NC(=O)C3=C(Cl)C=CC=C3N2C2=C1C=C(C1=CC=C(N3CCN(C4=C(F)C=C(NC5CCC(=O)NC5=O)C=C4)CC3)C=C1)C=C2	C38H35ClFN7O3	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024214019-A1
TPD-7M1JSX	WO2024217481A1_1-1	.	COc1cc(N2CCC(N3CCN(CCc4cc(F)c([C@H]5CCC(=O)NC5=O)c(F)c4)CC3)CC2)c(-c2cnn(C)c2)cc1Nc1ncc(Br)c(Nc2ccc3ccccc3c2P(C)(C)=O)n1	C49H54BrF2N10O4P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-5RL0LT	WO2024217481A1_1-2	.	COc1cc(N2CCC(N3CCN(CCc4cc(F)c([C@@H]5CCC(=O)NC5=O)c(F)c4)CC3)CC2)c(-c2cnn(C)c2)cc1Nc1ncc(Br)c(Nc2ccc3ccccc3c2P(C)(C)=O)n1	C49H54BrF2N10O4P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-IWDNUJ	SCHEMBL31155379	(3S)-3-[4-[2-[4-[1-[4-[[5-bromo-4-[(1-dimethylphosphorylnaphthalen-2-yl)amino]pyrimidin-2-yl]amino]-5-(cyclopropylmethoxy)-2-(1-methylpyrazol-4-yl)phenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2,6-difluorophenyl]piperidine-2,6-dione	Cn1cc(-c2cc(Nc3ncc(Br)c(Nc4ccc5ccccc5c4P(C)(C)=O)n3)c(OCC3CC3)cc2N2CCC(N3CCN(CCc4cc(F)c([C@@H]5CCC(=O)NC5=O)c(F)c4)CC3)CC2)cn1	C52H58BrF2N10O4P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-ORYW3V	WO2024217481A1_10-2	.	Cn1cc(-c2cc(Nc3ncc(Br)c(Nc4ccc5ccccc5c4P(C)(C)=O)n3)c(OCC3CC3)cc2N2CCC(N3CCN(CCc4cc(F)c([C@H]5CCC(=O)NC5=O)c(F)c4)CC3)CC2)cn1	C52H58BrF2N10O4P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-R3OP72	WO2024217481A1_11-1	.	Cn1cc(-c2cc(Nc3ncc(Br)c(Nc4ccc5ccccc5c4P(C)(C)=O)n3)c(OC3CC3)cc2N2CCC(N3CCN(CCc4cc(F)c([C@H]5CCC(=O)NC5=O)c(F)c4)CC3)CC2)cn1	C51H56BrF2N10O4P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-H5F9N4	WO2024217481A1_11-2	.	Cn1cc(-c2cc(Nc3ncc(Br)c(Nc4ccc5ccccc5c4P(C)(C)=O)n3)c(OC3CC3)cc2N2CCC(N3CCN(CCc4cc(F)c([C@@H]5CCC(=O)NC5=O)c(F)c4)CC3)CC2)cn1	C51H56BrF2N10O4P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-60O6BC	SCHEMBL31155577	(3R)-3-[4-[2-[4-[1-[4-[[5-bromo-4-[(4-dimethylphosphorylquinolin-3-yl)amino]pyrimidin-2-yl]amino]-5-cyclobutyloxy-2-(1-methylpyrazol-4-yl)phenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2,6-difluorophenyl]piperidine-2,6-dione	Cn1cc(-c2cc(Nc3ncc(Br)c(Nc4cnc5ccccc5c4P(C)(C)=O)n3)c(OC3CCC3)cc2N2CCC(N3CCN(CCc4cc(F)c([C@H]5CCC(=O)NC5=O)c(F)c4)CC3)CC2)cn1	C51H57BrF2N11O4P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-PZYNUP	WO2024217481A1_12-2	.	Cn1cc(-c2cc(Nc3ncc(Br)c(Nc4cnc5ccccc5c4P(C)(C)=O)n3)c(OC3CCC3)cc2N2CCC(N3CCN(CCc4cc(F)c([C@@H]5CCC(=O)NC5=O)c(F)c4)CC3)CC2)cn1	C51H57BrF2N11O4P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-LGUGD5	WO2024217481A1_13	.	Cn1cc(-c2cc(Nc3ncc(Br)c(Nc4ccc5ccccc5c4CP(C)(C)=O)n3)c(OC3CCC3)cc2N2CCC(N3CCN(C(=O)[C@@H]4CCN(c5cc(F)c(C6CCC(=O)NC6=O)c(F)c5)C4)CC3)CC2)cn1	C56H63BrF2N11O5P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-F8MMFM	WO2024217481A1_14	.	Cn1cc(-c2cc(Nc3ncc(Br)c(Nc4ccc5ccccc5c4CP(C)(C)=O)n3)c(OC3CC3)cc2N2CCC(N3CCN(C(=O)[C@@H]4CCN(c5cc(F)c(C6CCC(=O)NC6=O)c(F)c5)C4)CC3)CC2)cn1	C55H61BrF2N11O5P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-GFF2ON	WO2024217481A1_15	.	Cn1cc(-c2cc(Nc3ncc(Br)c(Nc4ccc5cc(F)ccc5c4CP(C)(C)=O)n3)c(OC3CCC3)cc2N2CCC(N3CCN(C(=O)[C@@H]4CCN(c5cc(F)c(C6CCC(=O)NC6=O)c(F)c5)C4)CC3)CC2)cn1	C56H62BrF3N11O5P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-DO4JWN	WO2024217481A1_16	.	Cn1cc(-c2cc(Nc3ncc(Br)c(Nc4ccc5cc(F)ccc5c4CP(C)(C)=O)n3)c(OC3CC3)cc2N2CCC(N3CCN(C(=O)[C@@H]4CCN(c5cc(F)c([C@@H]6CCC(=O)NC6=O)c(F)c5)C4)CC3)CC2)cn1	C55H60BrF3N11O5P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-RR0CEQ	WO2024217481A1_17	.	Cn1cc(-c2cc(Nc3ncc(Br)c(Nc4ccc5cc(F)ccc5c4CP(C)(C)=O)n3)c(OC3CC3)cc2N2CCC(N3CCN(C(=O)[C@@H]4CCN(c5cc(F)c([C@H]6CCC(=O)NC6=O)c(F)c5)C4)CC3)CC2)cn1	C55H60BrF3N11O5P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-3PVJTP	WO2024217481A1_18	.	COc1cc(N2CCC(N3CCN(C(=O)[C@@H]4CCN(c5cc(F)c(C6CCC(=O)NC6=O)c(F)c5)C4)CC3)CC2)c(-c2cnn(C)c2)cc1Nc1ncc(Br)c(Nc2ccc3cc(F)ccc3c2CP(C)(C)=O)n1	C53H58BrF3N11O5P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-21BHXD	WO2024217481A1_20	.	Cn1cc(-c2cc(Nc3ncc(Br)c(Nc4ccc5c(c4CP(C)(C)=O)OCCO5)n3)c(OC3CC3)cc2N2CCC(N3CCN(C(=O)[C@@H]4CCN(c5cc(F)c(C6CCC(=O)NC6=O)c(F)c5)C4)CC3)CC2)cn1	C53H61BrF2N11O7P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-BWEQK9	WO2024217481A1_21	.	Cc1ccc2c(CP(C)(C)=O)c(Nc3nc(Nc4cc(-c5cnn(C)c5)c(N5CCC(N6CCN(C(=O)[C@@H]7CCN(c8cc(F)c(C9CCC(=O)NC9=O)c(F)c8)C7)CC6)CC5)cc4OC4CC4)ncc3Br)ccc2c1	C56H63BrF2N11O5P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-HYLSVQ	WO2024217481A1_22	.	Cn1cc(-c2cc(Nc3ncc(Br)c(Nc4ccc5cc(F)ccc5c4CP(C)(C)=O)n3)c(OC3CC3)cc2N2CCC(N3CCN(C(=O)[C@H]4CCN(c5cc(F)c(C6CCC(=O)NC6=O)c(F)c5)C4)CC3)CC2)cn1	C55H60BrF3N11O5P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-5EU2VQ	SCHEMBL31155519	3-[4-[3-[4-[1-[4-[[5-Bromo-4-(2-dimethylphosphoryl-4-fluoroanilino)pyrimidin-2-yl]amino]-5-cyclopropyloxy-2-(1-methylpyrazol-4-yl)phenyl]piperidin-4-yl]piperazine-1-carbonyl]azetidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	Cn1cc(-c2cc(Nc3ncc(Br)c(Nc4ccc(F)cc4P(C)(C)=O)n3)c(OC3CC3)cc2N2CCC(N3CCN(C(=O)C4CN(c5cc(F)c(C6CCC(=O)NC6=O)c(F)c5)C4)CC3)CC2)cn1	C49H54BrF3N11O5P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-6KLND9	WO2024217481A1_24	.	Cn1cc(-c2cc(Nc3ncc(Br)c(Nc4ccc5ccccc5c4P(C)(C)=O)n3)c(OC3CC3)cc2N2CCC(N3CCN(C(=O)C4CN(c5cc(F)c(C6CCC(=O)NC6=O)c(F)c5)C4)CC3)CC2)cn1	C53H57BrF2N11O5P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-5TICPV	SCHEMBL31155552	(3R)-3-[4-[2-[4-[1-[4-[[5-bromo-4-[(5-dimethylphosphoryl-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-5-cyclopropyloxy-2-(1-methylpyrazol-4-yl)phenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2,6-difluorophenyl]piperidine-2,6-dione	Cc1ccc2c(P(C)(C)=O)c(Nc3nc(Nc4cc(-c5cnn(C)c5)c(N5CCC(N6CCN(CCc7cc(F)c([C@H]8CCC(=O)NC8=O)c(F)c7)CC6)CC5)cc4OC4CC4)ncc3Br)ccc2n1	C51H57BrF2N11O4P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-2ZYEKB	WO2024217481A1_25-2	.	Cc1ccc2c(P(C)(C)=O)c(Nc3nc(Nc4cc(-c5cnn(C)c5)c(N5CCC(N6CCN(CCc7cc(F)c([C@@H]8CCC(=O)NC8=O)c(F)c7)CC6)CC5)cc4OC4CC4)ncc3Br)ccc2n1	C51H57BrF2N11O4P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-GPMFDN	SCHEMBL31155479	(3R)-3-[4-[2-[4-[1-[4-[[5-bromo-4-[(5-dimethylphosphoryl-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-5-cyclobutyloxy-2-(1-methylpyrazol-4-yl)phenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2,6-difluorophenyl]piperidine-2,6-dione	Cc1ccc2c(P(C)(C)=O)c(Nc3nc(Nc4cc(-c5cnn(C)c5)c(N5CCC(N6CCN(CCc7cc(F)c([C@H]8CCC(=O)NC8=O)c(F)c7)CC6)CC5)cc4OC4CCC4)ncc3Br)ccc2n1	C52H59BrF2N11O4P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-0SH5VD	WO2024217481A1_26-2	.	Cc1ccc2c(P(C)(C)=O)c(Nc3nc(Nc4cc(-c5cnn(C)c5)c(N5CCC(N6CCN(CCc7cc(F)c([C@@H]8CCC(=O)NC8=O)c(F)c7)CC6)CC5)cc4OC4CCC4)ncc3Br)ccc2n1	C52H59BrF2N11O4P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-PB6MUW	SCHEMBL31155559	3-[4-[3-[4-[1-[4-[[5-Bromo-4-[(5-dimethylphosphoryl-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-5-cyclopropyloxy-2-(1-methylpyrazol-4-yl)phenyl]piperidin-4-yl]piperazine-1-carbonyl]azetidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	Cc1ccc2c(P(C)(C)=O)c(Nc3nc(Nc4cc(-c5cnn(C)c5)c(N5CCC(N6CCN(C(=O)C7CN(c8cc(F)c(C9CCC(=O)NC9=O)c(F)c8)C7)CC6)CC5)cc4OC4CC4)ncc3Br)ccc2n1	C53H58BrF2N12O5P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-9EAPMG	WO2024217481A1_28-1	.	Cn1cc(-c2cc(Nc3ncc(Br)c(Nc4cnc5ccccc5c4P(C)(C)=O)n3)c(OCC3CC3)cc2N2CCC(N3CCN(CCc4cc(F)c([C@H]5CCC(=O)NC5=O)c(F)c4)CC3)CC2)cn1	C51H57BrF2N11O4P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-KSW4FO	WO2024217481A1_28-2	.	Cn1cc(-c2cc(Nc3ncc(Br)c(Nc4cnc5ccccc5c4P(C)(C)=O)n3)c(OCC3CC3)cc2N2CCC(N3CCN(CCc4cc(F)c([C@@H]5CCC(=O)NC5=O)c(F)c4)CC3)CC2)cn1	C51H57BrF2N11O4P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-WSKGYX	SCHEMBL31155530	(3R)-3-[4-[2-[4-[1-[4-[[5-bromo-4-[(4-dimethylphosphorylquinolin-3-yl)amino]pyrimidin-2-yl]amino]-2-(1-methylpyrazol-4-yl)-5-propan-2-yloxyphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2,6-difluorophenyl]piperidine-2,6-dione	CC(C)Oc1cc(N2CCC(N3CCN(CCc4cc(F)c([C@H]5CCC(=O)NC5=O)c(F)c4)CC3)CC2)c(-c2cnn(C)c2)cc1Nc1ncc(Br)c(Nc2cnc3ccccc3c2P(C)(C)=O)n1	C50H57BrF2N11O4P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-M7JRJL	WO2024217481A1_29-2	.	CC(C)Oc1cc(N2CCC(N3CCN(CCc4cc(F)c([C@@H]5CCC(=O)NC5=O)c(F)c4)CC3)CC2)c(-c2cnn(C)c2)cc1Nc1ncc(Br)c(Nc2cnc3ccccc3c2P(C)(C)=O)n1	C50H57BrF2N11O4P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-YXY8J1	SCHEMBL31155531	(3R)-3-[4-[2-[4-[1-[4-[[5-bromo-4-[(4-dimethylphosphorylquinolin-3-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-(1-methylpyrazol-4-yl)phenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2,6-difluorophenyl]piperidine-2,6-dione	COc1cc(N2CCC(N3CCN(CCc4cc(F)c([C@H]5CCC(=O)NC5=O)c(F)c4)CC3)CC2)c(-c2cnn(C)c2)cc1Nc1ncc(Br)c(Nc2cnc3ccccc3c2P(C)(C)=O)n1	C48H53BrF2N11O4P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-QDTEI4	WO2024217481A1_3-2	.	COc1cc(N2CCC(N3CCN(CCc4cc(F)c([C@@H]5CCC(=O)NC5=O)c(F)c4)CC3)CC2)c(-c2cnn(C)c2)cc1Nc1ncc(Br)c(Nc2cnc3ccccc3c2P(C)(C)=O)n1	C48H53BrF2N11O4P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-7ABVNU	WO2024217481A1_30-1	.	Cn1cc(-c2cc(Nc3ncc(Br)c(Nc4ccc(F)cc4P(C)(C)=O)n3)c(OCC3CC3)cc2N2CCC(N3CCN(CCc4cc(F)c([C@H]5CCC(=O)NC5=O)c(F)c4)CC3)CC2)cn1	C48H55BrF3N10O4P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-8PMQAB	WO2024217481A1_30-2	.	Cn1cc(-c2cc(Nc3ncc(Br)c(Nc4ccc(F)cc4P(C)(C)=O)n3)c(OCC3CC3)cc2N2CCC(N3CCN(CCc4cc(F)c([C@@H]5CCC(=O)NC5=O)c(F)c4)CC3)CC2)cn1	C48H55BrF3N10O4P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-QZMSTJ	SCHEMBL31155483	(3R)-3-[4-[2-[4-[1-[4-[[5-bromo-4-[(5-dimethylphosphorylquinoxalin-6-yl)amino]pyrimidin-2-yl]amino]-5-cyclobutyloxy-2-(1-methylpyrazol-4-yl)phenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2,6-difluorophenyl]piperidine-2,6-dione	Cn1cc(-c2cc(Nc3ncc(Br)c(Nc4ccc5nccnc5c4P(C)(C)=O)n3)c(OC3CCC3)cc2N2CCC(N3CCN(CCc4cc(F)c([C@H]5CCC(=O)NC5=O)c(F)c4)CC3)CC2)cn1	C50H56BrF2N12O4P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-4RCV3E	WO2024217481A1_32-1	.	Cn1cc(-c2cc(Nc3ncc(Br)c(Nc4ccc(-c5ccccc5)cc4P(C)(C)=O)n3)c(OC3CC3)cc2N2CCC(N3CCN(CCc4cc(F)c([C@H]5CCC(=O)NC5=O)c(F)c4)CC3)CC2)cn1	C53H58BrF2N10O4P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-O892UQ	WO2024217481A1_32-2	.	Cn1cc(-c2cc(Nc3ncc(Br)c(Nc4ccc(-c5ccccc5)cc4P(C)(C)=O)n3)c(OC3CC3)cc2N2CCC(N3CCN(CCc4cc(F)c([C@@H]5CCC(=O)NC5=O)c(F)c4)CC3)CC2)cn1	C53H58BrF2N10O4P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-VSG1P0	SCHEMBL31155383	3-[4-[2-[4-[1-[4-[[5-Bromo-4-(2-dimethylphosphorylanilino)pyrimidin-2-yl]amino]-5-cyclobutyloxy-2-(1-methylpyrazol-4-yl)phenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2,6-difluorophenyl]piperidine-2,6-dione	Cn1cc(-c2cc(Nc3ncc(Br)c(Nc4ccccc4P(C)(C)=O)n3)c(OC3CCC3)cc2N2CCC(N3CCN(CCc4cc(F)c(C5CCC(=O)NC5=O)c(F)c4)CC3)CC2)cn1	C48H56BrF2N10O4P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-8D5GP3	SCHEMBL31155403	(3R)-3-[4-[2-[4-[1-[4-[[5-bromo-4-[(4-dimethylphosphorylquinolin-3-yl)amino]pyrimidin-2-yl]amino]-5-cyclopropyloxy-2-(1-methylpyrazol-4-yl)phenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2,6-difluorophenyl]piperidine-2,6-dione	Cn1cc(-c2cc(Nc3ncc(Br)c(Nc4cnc5ccccc5c4P(C)(C)=O)n3)c(OC3CC3)cc2N2CCC(N3CCN(CCc4cc(F)c([C@H]5CCC(=O)NC5=O)c(F)c4)CC3)CC2)cn1	C50H55BrF2N11O4P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-7WGFXE	WO2024217481A1_34-2	.	Cn1cc(-c2cc(Nc3ncc(Br)c(Nc4cnc5ccccc5c4P(C)(C)=O)n3)c(OC3CC3)cc2N2CCC(N3CCN(CCc4cc(F)c([C@@H]5CCC(=O)NC5=O)c(F)c4)CC3)CC2)cn1	C50H55BrF2N11O4P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-F80AZM	SCHEMBL31155428	3-[4-[2-[4-[1-[4-[[5-Bromo-4-[(4-dimethylphosphorylquinolin-3-yl)amino]pyrimidin-2-yl]amino]-2-(1-methylpyrazol-4-yl)-5-(2,2,2-trifluoroethoxy)phenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2,6-difluorophenyl]piperidine-2,6-dione	Cn1cc(-c2cc(Nc3ncc(Br)c(Nc4cnc5ccccc5c4P(C)(C)=O)n3)c(OCC(F)(F)F)cc2N2CCC(N3CCN(CCc4cc(F)c(C5CCC(=O)NC5=O)c(F)c4)CC3)CC2)cn1	C49H52BrF5N11O4P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-IG3ZIZ	WO2024217481A1_36	.	CCOc1cc(N2CCC(N3CCN(CCc4cc(F)c(C5CCC(=O)NC5=O)c(F)c4)CC3)CC2)c(-c2cnn(C)c2)cc1Nc1ncc(Br)c(Nc2cnc3ccccc3c2P(C)(C)=O)n1	C49H55BrF2N11O4P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-MB1J7X	SCHEMBL31155566	(3R)-3-[4-[(3R)-3-[4-[1-[4-[[5-bromo-4-[(5-dimethylphosphorylquinoxalin-6-yl)amino]pyrimidin-2-yl]amino]-5-cyclopropyloxy-2-(1-methylpyrazol-4-yl)phenyl]piperidin-4-yl]piperazine-1-carbonyl]pyrrolidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	Cn1cc(-c2cc(Nc3ncc(Br)c(Nc4ccc5nccnc5c4P(C)(C)=O)n3)c(OC3CC3)cc2N2CCC(N3CCN(C(=O)[C@@H]4CCN(c5cc(F)c([C@H]6CCC(=O)NC6=O)c(F)c5)C4)CC3)CC2)cn1	C52H57BrF2N13O5P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-W8J4D4	WO2024217481A1_37-2	.	Cn1cc(-c2cc(Nc3ncc(Br)c(Nc4ccc5nccnc5c4P(C)(C)=O)n3)c(OC3CC3)cc2N2CCC(N3CCN(C(=O)[C@@H]4CCN(c5cc(F)c([C@@H]6CCC(=O)NC6=O)c(F)c5)C4)CC3)CC2)cn1	C52H57BrF2N13O5P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-VT4XE6	WO2024217481A1_38	.	Cn1cc(-c2cc(Nc3ncc(Br)c(Nc4cnc5ccccc5c4P(C)(C)=O)n3)c(OC3CC3)cc2N2CCC(CN3CCC4(CC3)CN(c3ccc5c(c3)C(=O)N(C3CCC(=O)NC3=O)C5)C4)CC2)cn1	C54H60BrN12O5P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-AFD7JH	WO2024217481A1_39	.	Cc1ncc(Nc2nc(Nc3cc(-c4cnn(C)c4)c(N4CCC(N5CCN(C(=O)[C@@H]6CCN(c7cc(F)c(C8CCC(=O)NC8=O)c(F)c7)C6)CC5)CC4)cc3OC3CC3)ncc2Br)c(P(C)(C)=O)c1C	C51H60BrF2N12O5P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-7ODWH2	SCHEMBL31155516	3-[4-[3-[4-[[1-[4-[[5-Bromo-4-[(4-dimethylphosphorylquinolin-3-yl)amino]pyrimidin-2-yl]amino]-5-cyclopropyloxy-2-(1-methylpyrazol-4-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]azetidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	Cn1cc(-c2cc(Nc3ncc(Br)c(Nc4cnc5ccccc5c4P(C)(C)=O)n3)c(OC3CC3)cc2N2CCC(CN3CCN(C4CN(c5cc(F)c(C6CCC(=O)NC6=O)c(F)c5)C4)CC3)CC2)cn1	C52H58BrF2N12O4P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-UKB00D	SCHEMBL31155522	3-[4-[7-[[1-[4-[[5-Bromo-4-[(4-dimethylphosphorylquinolin-3-yl)amino]pyrimidin-2-yl]amino]-5-cyclopropyloxy-2-(1-methylpyrazol-4-yl)phenyl]piperidin-4-yl]methyl]-2,7-diazaspiro[3.5]nonan-2-yl]-2,6-difluorophenyl]piperidine-2,6-dione	Cn1cc(-c2cc(Nc3ncc(Br)c(Nc4cnc5ccccc5c4P(C)(C)=O)n3)c(OC3CC3)cc2N2CCC(CN3CCC4(CC3)CN(c3cc(F)c(C5CCC(=O)NC5=O)c(F)c3)C4)CC2)cn1	C52H57BrF2N11O4P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-EQ04AZ	WO2024217481A1_42	.	Cn1cc(-c2cc(Nc3ncc(Br)c(Nc4cnc5ccccc5c4P(C)(C)=O)n3)c(OC3CC3)cc2N2CCC(N3CCN(CCc4cccc5c4n(C)c(=O)n5C4CCC(=O)NC4=O)CC3)CC2)cn1	C52H59BrN13O5P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-TWKUXA	WO2024217481A1_43	.	Cn1cc(-c2cc(Nc3ncc(Br)c(Nc4cnc5ccccc5c4P(C)(C)=O)n3)c(OC3CC3)cc2N2CCC(CN3CCC4(CC3)CN(c3ccc5c(c3)C(=O)N(C3CCC(=O)NC3=O)C5=O)C4)CC2)cn1	C54H58BrN12O6P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-HUGJ5P	WO2024217481A1_44-1	.	Cn1cc(-c2cc(Nc3ncc(Br)c(Nc4ccccc4P(C)(C)=O)n3)c(OC3CC3)cc2N2CCC(N3CCN(C(=O)[C@@H]4CCN(c5cc(F)c([C@H]6CCC(=O)NC6=O)c(F)c5)C4)CC3)CC2)cn1	C50H57BrF2N11O5P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-8R1TQR	WO2024217481A1_44-2	.	Cn1cc(-c2cc(Nc3ncc(Br)c(Nc4ccccc4P(C)(C)=O)n3)c(OC3CC3)cc2N2CCC(N3CCN(C(=O)[C@@H]4CCN(c5cc(F)c([C@@H]6CCC(=O)NC6=O)c(F)c5)C4)CC3)CC2)cn1	C50H57BrF2N11O5P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-AIYMUW	WO2024217481A1_45-1	.	Cn1cc(-c2cc(Nc3ncc(Br)c(Nc4ccc(Cl)cc4P(C)(C)=O)n3)c(OC3CC3)cc2N2CCC(N3CCN(C(=O)[C@@H]4CCN(c5cc(F)c([C@H]6CCC(=O)NC6=O)c(F)c5)C4)CC3)CC2)cn1	C50H56BrClF2N11O5P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-WT0BB7	WO2024217481A1_45-2	.	Cn1cc(-c2cc(Nc3ncc(Br)c(Nc4ccc(Cl)cc4P(C)(C)=O)n3)c(OC3CC3)cc2N2CCC(N3CCN(C(=O)[C@@H]4CCN(c5cc(F)c([C@@H]6CCC(=O)NC6=O)c(F)c5)C4)CC3)CC2)cn1	C50H56BrClF2N11O5P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-UVYISQ	SCHEMBL31155638	(3R)-3-[4-[(3R)-3-[4-[1-[4-[[5-bromo-4-(2-dimethylphosphoryl-3,4-dimethylanilino)pyrimidin-2-yl]amino]-5-cyclopropyloxy-2-(1-methylpyrazol-4-yl)phenyl]piperidin-4-yl]piperazine-1-carbonyl]pyrrolidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	Cc1ccc(Nc2nc(Nc3cc(-c4cnn(C)c4)c(N4CCC(N5CCN(C(=O)[C@@H]6CCN(c7cc(F)c([C@H]8CCC(=O)NC8=O)c(F)c7)C6)CC5)CC4)cc3OC3CC3)ncc2Br)c(P(C)(C)=O)c1C	C52H61BrF2N11O5P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-KBWHE8	WO2024217481A1_46-2	.	Cc1ccc(Nc2nc(Nc3cc(-c4cnn(C)c4)c(N4CCC(N5CCN(C(=O)[C@@H]6CCN(c7cc(F)c([C@@H]8CCC(=O)NC8=O)c(F)c7)C6)CC5)CC4)cc3OC3CC3)ncc2Br)c(P(C)(C)=O)c1C	C52H61BrF2N11O5P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-Z0B9VH	SCHEMBL31155455	(3R)-3-[4-[2-[4-[1-[4-[[5-bromo-4-[(4-dimethylphosphoryl-6-phenylpyridin-3-yl)amino]pyrimidin-2-yl]amino]-5-cyclopropyloxy-2-(1-methylpyrazol-4-yl)phenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2,6-difluorophenyl]piperidine-2,6-dione	Cn1cc(-c2cc(Nc3ncc(Br)c(Nc4cnc(-c5ccccc5)cc4P(C)(C)=O)n3)c(OC3CC3)cc2N2CCC(N3CCN(CCc4cc(F)c([C@H]5CCC(=O)NC5=O)c(F)c4)CC3)CC2)cn1	C52H57BrF2N11O4P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-T4B7MY	WO2024217481A1_48	.	CCOc1cc(N2CCC(N3CCN(CCc4cc(F)c(C5(C)CC(C)(C)C(=O)NC5=O)c(F)c4)CC3)CC2)c(-c2cnn(C)c2)cc1Nc1ncc(Br)c(Nc2cnc3ccccc3c2P(C)(C)=O)n1	C52H61BrF2N11O4P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-50N0R6	WO2024217481A1_49	.	Cn1cc(-c2cc(Nc3ncc(Br)c(Nc4cnc5ccccc5c4P(C)(C)=O)n3)c(OC3CC3)cc2N2CCC(N3CCN(CCc4cc(F)c(C5(C)CC(C)(C)C(=O)NC5=O)c(F)c4)CC3)CC2)cn1	C53H61BrF2N11O4P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-TBP744	WO2024217481A1_5-1	.	Cn1cc(-c2cc(Nc3ncc(Br)c(Nc4ccc5ccccc5c4P(C)(C)=O)n3)c(OC3CCC3)cc2N2CCC(N3CCN(CCc4cc(F)c([C@H]5CCC(=O)NC5=O)c(F)c4)CC3)CC2)cn1	C52H58BrF2N10O4P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-9AYZGH	SCHEMBL31155622	(3S)-3-[4-[2-[4-[1-[4-[[5-bromo-4-[(1-dimethylphosphorylnaphthalen-2-yl)amino]pyrimidin-2-yl]amino]-5-cyclobutyloxy-2-(1-methylpyrazol-4-yl)phenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2,6-difluorophenyl]piperidine-2,6-dione	Cn1cc(-c2cc(Nc3ncc(Br)c(Nc4ccc5ccccc5c4P(C)(C)=O)n3)c(OC3CCC3)cc2N2CCC(N3CCN(CCc4cc(F)c([C@@H]5CCC(=O)NC5=O)c(F)c4)CC3)CC2)cn1	C52H58BrF2N10O4P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-72C5GQ	SCHEMBL31155543	3-[4-[2-[4-[1-[4-[[5-Bromo-4-[(4-dimethylphosphorylquinolin-3-yl)amino]pyrimidin-2-yl]amino]-5-cyclopropyloxy-2-(1-methylpyrazol-4-yl)phenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2,6-difluorophenyl]piperidine-2,6-dione	Cn1cc(-c2cc(Nc3ncc(Br)c(Nc4cnc5ccccc5c4P(C)(C)=O)n3)c(OC3CC3)cc2N2CCC(N3CCN(CCc4cc(F)c(C5CCC(=O)NC5=O)c(F)c4)CC3)CC2)cn1	C50H55BrF2N11O4P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-V7VUPS	SCHEMBL31155484	3-[4-[2-[4-[1-[4-[[5-Bromo-4-[(4-dimethylphosphoryl-6-phenylpyridin-3-yl)amino]pyrimidin-2-yl]amino]-5-ethoxy-2-(1-methylpyrazol-4-yl)phenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2,6-difluorophenyl]piperidine-2,6-dione	CCOc1cc(N2CCC(N3CCN(CCc4cc(F)c(C5CCC(=O)NC5=O)c(F)c4)CC3)CC2)c(-c2cnn(C)c2)cc1Nc1ncc(Br)c(Nc2cnc(-c3ccccc3)cc2P(C)(C)=O)n1	C51H57BrF2N11O4P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-3DWONN	WO2024217481A1_52	.	Cc1ncc(Nc2nc(Nc3cc(-c4cnn(C)c4)c(N4CCC(N5CCN(CCc6cc(F)c(C7CCC(=O)NC7=O)c(F)c6)CC5)CC4)cc3OC3CC3)ncc2Br)c(P(C)(C)=O)n1	C46H54BrF2N12O4P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-UO4RVV	WO2024217481A1_53	.	Cn1cc(-c2cc(Nc3ncc(C(F)(F)F)c(Nc4ccc5ccccc5c4P(C)(C)=O)n3)c(OC3CC3)cc2N2CCC(N3CCN(CCc4cc(F)c(C5CCC(=O)NC5=O)c(F)c4)CC3)CC2)cn1	C52H56F5N10O4P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-2YH00J	WO2024217481A1_54	.	Cn1cc(-c2cc(Nc3ncc(Br)c(Nc4ccc5ccccc5c4P(C)(C)=O)n3)c(OC3CC3)cc2N2CCC(N3CCN(CCc4cccc5c4C(C)(C)C(=O)N5C4CCC(=O)NC4=O)CC3)CC2)cn1	C55H63BrN11O5P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-9PJ69C	WO2024217481A1_55	.	CC(C)Oc1cc(N2CCN(C(=O)CN3CCC(c4ccc(NC5CCC(=O)NC5=O)cc4)CC3)CC2)c(-c2cnn(C)c2)cc1Nc1ncc(Br)c(Nc2ccc3nccnc3c2P(C)(C)=O)n1	C49H57BrN13O5P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-J6H39T	SCHEMBL31155490	(3R)-3-[4-[2-[4-[1-[4-[[5-bromo-4-[(4-dimethylphosphorylquinolin-3-yl)amino]pyrimidin-2-yl]amino]-5-cyclopropyloxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2,6-difluorophenyl]piperidine-2,6-dione	Cc1cc(Nc2ncc(Br)c(Nc3cnc4ccccc4c3P(C)(C)=O)n2)c(OC2CC2)cc1N1CCC(N2CCN(CCc3cc(F)c([C@H]4CCC(=O)NC4=O)c(F)c3)CC2)CC1	C47H53BrF2N9O4P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-IHNJLX	WO2024217481A1_56-2	.	Cc1cc(Nc2ncc(Br)c(Nc3cnc4ccccc4c3P(C)(C)=O)n2)c(OC2CC2)cc1N1CCC(N2CCN(CCc3cc(F)c([C@@H]4CCC(=O)NC4=O)c(F)c3)CC2)CC1	C47H53BrF2N9O4P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-PBI8ZF	SCHEMBL31155423	3-[4-[2-[4-[1-[4-[[5-Bromo-4-[(4-dimethylphosphorylquinolin-3-yl)amino]pyrimidin-2-yl]amino]-2-cyclopropyl-5-cyclopropyloxyphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2,6-difluorophenyl]piperidine-2,6-dione	CP(C)(=O)c1c(Nc2nc(Nc3cc(C4CC4)c(N4CCC(N5CCN(CCc6cc(F)c(C7CCC(=O)NC7=O)c(F)c6)CC5)CC4)cc3OC3CC3)ncc2Br)cnc2ccccc12	C49H55BrF2N9O4P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-7XR2BV	WO2024217481A1_58-2	.	COc1cc(N2CCC(N3CCN(CCc4cc(F)c([C@@H]5CCC(=O)NC5=O)c(F)c4)CC3)CC2)c(-c2cnn(C)c2)cc1Nc1ncc(Br)c(Nc2cnc(-c3ccccc3)cc2P(C)(C)=O)n1	C50H55BrF2N11O4P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-H6368K	WO2024217481A1_7-1	.	Cn1cc(-c2cc(Nc3ncc(Br)c(Nc4ccc5cc(F)ccc5c4P(C)(C)=O)n3)c(OC3CCC3)cc2N2CCC(N3CCN(CCc4cc(F)c([C@H]5CCC(=O)NC5=O)c(F)c4)CC3)CC2)cn1	C52H57BrF3N10O4P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-R1JSAF	WO2024217481A1_7-2	.	Cn1cc(-c2cc(Nc3ncc(Br)c(Nc4ccc5cc(F)ccc5c4P(C)(C)=O)n3)c(OC3CCC3)cc2N2CCC(N3CCN(CCc4cc(F)c([C@@H]5CCC(=O)NC5=O)c(F)c4)CC3)CC2)cn1	C52H57BrF3N10O4P	EGFR	P00533	CRBN	WO-2024217481-A1
TPD-C39Q59	WO2024217520A1_A02	.	Cc1c(NC(=O)CN2CCN(C(=O)CCOCCOCCNC(=O)COc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)c[nH]c1/C=C1\C(=O)Nc2ccc(F)cc21	C42H45FN8O11	FLT3	P36888	CRBN	WO-2024217520-A1
TPD-FR0V2A	WO2024217520A1_A03	.	Cc1c(NC(=O)CN2CCN(C(=O)CCOCCNc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)c[nH]c1/C=C1\C(=O)Nc2ccc(F)cc21	C38H39FN8O8	FLT3	P36888	CRBN	WO-2024217520-A1
TPD-VH99FS	WO2024217520A1_A04	.	Cc1c(NC(=O)CN2CCN(C(=O)CCOCCOCCNc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)c[nH]c1/C=C1\C(=O)Nc2ccc(F)cc21	C40H43FN8O9	FLT3	P36888	CRBN	WO-2024217520-A1
TPD-MQK9UG	WO2024217520A1_A05	.	Cc1c(NC(=O)CN2CCN(C(=O)CCOCCOCCOCCNc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)c[nH]c1/C=C1\C(=O)Nc2ccc(F)cc21	C42H47FN8O10	FLT3	P36888	CRBN	WO-2024217520-A1
TPD-09BRXM	WO2024217520A1_A06	.	Cc1c(NC(=O)CC2CCN(CCCCCCCCC(=O)Nc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)c[nH]c1/C=C1\C(=O)Nc2ccc(F)cc21	C43H48FN7O7	FLT3	P36888	CRBN	WO-2024217520-A1
TPD-F9IRKQ	WO2024217520A1_A07	.	Cc1c(NC(=O)CN2CCN(CCCCCCCCCOc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)c[nH]c1/C=C1\C(=O)Nc2ccc(F)cc21	C42H48FN7O7	FLT3	P36888	CRBN	WO-2024217520-A1
TPD-TIO2IQ	WO2024217520A1_A08	.	Cc1c(NC(=O)CN2CCN(C(=O)CCCC(=O)NCCNc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)c[nH]c1/C=C1\C(=O)Nc2ccc(F)cc21	C40H42FN9O8	FLT3	P36888	CRBN	WO-2024217520-A1
TPD-HAL5FZ	WO2024217520A1_A09	.	Cc1c(NC(=O)CN2CCN(C(=O)CCCCC(=O)NCCNc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)c[nH]c1/C=C1\C(=O)Nc2ccc(F)cc21	C41H44FN9O8	FLT3	P36888	CRBN	WO-2024217520-A1
TPD-IEL8Y0	WO2024217520A1_A10	.	Cc1c(NC(=O)CN2CCN(C(=O)CCCCCC(=O)NCCNc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)c[nH]c1/C=C1\C(=O)Nc2ccc(F)cc21	C42H46FN9O8	FLT3	P36888	CRBN	WO-2024217520-A1
TPD-XQ0G76	WO2024217520A1_A11	.	Cc1c(NC(=O)CN2CCN(C(=O)CCCCCCC(=O)NCCN=Nc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)c[nH]c1/C=C1\C(=O)Nc2ccc(F)cc21	C43H47FN10O8	FLT3	P36888	CRBN	WO-2024217520-A1
TPD-X4EOKX	WO2024217520A1_A12	.	Cc1c(NC(=O)CN2CCN(C(=O)CCCCCCCC(=O)NCCNc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)c[nH]c1/C=C1\C(=O)Nc2ccc(F)cc21	C44H50FN9O8	FLT3	P36888	CRBN	WO-2024217520-A1
TPD-7I0ZDB	SCHEMBL31121740	N-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethyl]-10-[4-[2-[[5-[(Z)-(5-fluoro-2-oxo-1H-indol-3-ylidene)methyl]-4-methyl-1H-pyrrol-3-yl]amino]-2-oxoethyl]piperazin-1-yl]-10-oxodecanamide	Cc1c(NC(=O)CN2CCN(C(=O)CCCCCCCCC(=O)NCCNc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)c[nH]c1/C=C1\C(=O)Nc2ccc(F)cc21	C45H52FN9O8	FLT3	P36888	CRBN	WO-2024217520-A1
TPD-2ZNJLR	WO2024217520A1_A14	.	Cc1c(NC(=O)CN2CCN(C(=O)CCCCCNc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)c[nH]c1/C=C1\C(=O)Nc2ccc(F)cc21	C39H41FN8O7	FLT3	P36888	CRBN	WO-2024217520-A1
TPD-TT5YLU	SCHEMBL31121727	2-[4-[7-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]heptanoyl]piperazin-1-yl]-N-[5-[(Z)-(5-fluoro-2-oxo-1H-indol-3-ylidene)methyl]-4-methyl-1H-pyrrol-3-yl]acetamide	Cc1c(NC(=O)CN2CCN(C(=O)CCCCCCNc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)c[nH]c1/C=C1\C(=O)Nc2ccc(F)cc21	C40H43FN8O7	FLT3	P36888	CRBN	WO-2024217520-A1
TPD-552OGS	WO2024217520A1_A16	.	Cc1c(NC(=O)CN2CCN(C(=O)CCCCCCCNc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)c[nH]c1/C=C1\C(=O)Nc2ccc(F)cc21	C41H45FN8O7	FLT3	P36888	CRBN	WO-2024217520-A1
TPD-SQPVON	WO2024217520A1_A17	.	Cc1c(NC(=O)CN2CCN(C(=O)CCCCCCCCCCNc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)c[nH]c1/C=C1\C(=O)Nc2ccc(F)cc21	C44H51FN8O7	FLT3	P36888	CRBN	WO-2024217520-A1
TPD-LYB14X	WO2024217520A1_A18	.	C=c1[nH]c2ccc(F)cc2/c1=C/c1[nH]cc(NC(=O)CN2CCN(C(=O)CCCCCCCCCCCNc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)c1C	C46H55FN8O6	FLT3	P36888	CRBN	WO-2024217520-A1
TPD-8IWSDK	SCHEMBL31121736	2-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperidin-4-yl]methyl]piperazin-1-yl]-N-[5-[(Z)-(5-fluoro-2-oxo-1H-indol-3-ylidene)methyl]-4-methyl-1H-pyrrol-3-yl]acetamide	Cc1c(NC(=O)CN2CCN(CC3CCN(c4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)c[nH]c1/C=C1\C(=O)Nc2ccc(F)cc21	C39H41FN8O6	FLT3	P36888	CRBN	WO-2024217520-A1
TPD-OS4CSI	PROTAC FLT-3 degrader 4	PROTAC FLT-3 degrader 4; orb2564707; SCHEMBL31121739; HY-158325; CS-1052111; 2956722-48-6	Cc1c(NC(=O)CN2CCN(CC3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)c[nH]c1/C=C1\C(=O)Nc2ccc(F)cc21	C39H41FN8O6	FLT3	P36888	CRBN	WO-2024217520-A1
TPD-ZJ66CE	SCHEMBL31121743	2-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]piperazin-1-yl]-N-[5-[(Z)-(5-fluoro-2-oxo-1H-indol-3-ylidene)methyl]-4-methyl-1H-pyrrol-3-yl]acetamide	Cc1c(NC(=O)CN2CCN(C3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)c[nH]c1/C=C1\C(=O)Nc2ccc(F)cc21	C38H39FN8O6	FLT3	P36888	CRBN	WO-2024217520-A1
TPD-OQL8WB	SCHEMBL31121737	2-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]piperazin-1-yl]-N-[5-[(Z)-(5-fluoro-2-oxo-1H-indol-3-ylidene)methyl]-4-methyl-1H-pyrrol-3-yl]acetamide	Cc1c(NC(=O)CN2CCN(C3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)CC2)c[nH]c1/C=C1\C(=O)Nc2ccc(F)cc21	C36H35FN8O6	FLT3	P36888	CRBN	WO-2024217520-A1
TPD-ETES22	WO2024217520A1_A23	.	Cc1c(NC(=O)CN2CCN(C3CC4(CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C3)CC2)c[nH]c1/C=C1\C(=O)Nc2ccc(F)cc21	C41H43FN8O6	FLT3	P36888	CRBN	WO-2024217520-A1
TPD-CMJPNB	SCHEMBL31121728	2-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]methyl]piperazin-1-yl]-N-[5-[(Z)-(5-fluoro-2-oxo-1H-indol-3-ylidene)methyl]-4-methyl-1H-pyrrol-3-yl]acetamide	Cc1c(NC(=O)CN2CCN(CC3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)CC2)c[nH]c1/C=C1\C(=O)Nc2ccc(F)cc21	C37H37FN8O6	FLT3	P36888	CRBN	WO-2024217520-A1
TPD-AK3I39	SCHEMBL31121741	2-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]-N-[5-[(Z)-(5-fluoro-2-oxo-1H-indol-3-ylidene)methyl]-4-methyl-1H-pyrrol-3-yl]acetamide	Cc1c(NC(=O)CN2CCN(CC3CCN(c4cc5c(cc4F)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)c[nH]c1/C=C1\C(=O)Nc2ccc(F)cc21	C39H40F2N8O6	FLT3	P36888	CRBN	WO-2024217520-A1
TPD-RMD1J0	WO2024217520A1_A26	.	Cc1[nH]c(/C=C2\C(=O)Nc3ccc(F)cc32)c(C)c1NC(=O)CN1CCN(CC2CCN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)CC1	C40H43FN8O6	FLT3	P36888	CRBN	WO-2024217520-A1
TPD-1U4Q04	WO2024217520A1_A27	.	Cc1[nH]c(/C=C2\C(=O)Nc3ccc(F)cc32)c(C)c1C(=O)N1CCN(CC2CCN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)CC1	C39H40FN7O6	FLT3	P36888	CRBN	WO-2024217520-A1
TPD-CORC6U	SCHEMBL31121731	N-[2-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]ethyl]-5-[(Z)-(5-fluoro-2-oxo-1H-indol-3-ylidene)methyl]-2,4-dimethyl-1H-pyrrole-3-carboxamide	Cc1[nH]c(/C=C2\C(=O)Nc3ccc(F)cc32)c(C)c1C(=O)NCCN1CCN(CC2CCN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)CC1	C41H45FN8O6	FLT3	P36888	CRBN	WO-2024217520-A1
TPD-YIAEEH	SCHEMBL31121730	N-[3-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]propyl]-5-[(Z)-(5-fluoro-2-oxo-1H-indol-3-ylidene)methyl]-2,4-dimethyl-1H-pyrrole-3-carboxamide	Cc1[nH]c(/C=C2\C(=O)Nc3ccc(F)cc32)c(C)c1C(=O)NCCCN1CCN(CC2CCN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)CC1	C42H47FN8O6	FLT3	P36888	CRBN	WO-2024217520-A1
TPD-52BPZZ	WO2024230647A1_B003	.	CC1=CC(NC2=NC(C[C@@]3(C(=O)O)CCN(CC4=C(F)C(Cl)=CC=C4)[C@H](C)C3)=C(F)C(C#CCCCCCCCOC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)=C2)=NN1	C46H48ClF2N7O7	AURKA	O14965	CRBN	WO-2024230647-A1
TPD-U54D6S	WO2024230647A1_B004	.	CC1=CC(NC2=NC(C[C@@]3(C(=O)NCCOCCOCCNC4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CCN(CC4=CC=CC(Cl)=C4F)[C@H](C)C3)=C(F)C=C2)=NN1	C43H48ClF2N9O7	AURKA	O14965	CRBN	WO-2024230647-A1
TPD-HP6ZOH	WO2024230647A1_B006	.	CC1=CC(NC2=NC(C[C@@]3(C(=O)NCCCCCCNC4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CCN(CC4=C(F)C(Cl)=CC=C4)[C@H](C)C3)=C(F)C=C2)=NN1	C43H48ClF2N9O5	AURKA	O14965	CRBN	WO-2024230647-A1
TPD-W33ZZQ	WO2024230647A1_B007	.	CC1=CC(NC2=NC(C[C@@]3(C(=O)NCCCCCCCNC4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CCN(CC4=C(F)C(C#N)=CC=C4)[C@H](C)C3)=C(F)C=C2)=NN1	C45H50F2N10O5	AURKA	O14965	CRBN	WO-2024230647-A1
TPD-J9T3X2	WO2024230647A1_B008	.	CC1=CC(NC2=NC(C[C@@]3(C(=O)NCCCCCCCCNC4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CCN(CC4=C(F)C(C#N)=CC=C4)[C@H](C)C3)=C(F)C=C2)=NN1	C46H52F2N10O5	AURKA	O14965	CRBN	WO-2024230647-A1
TPD-492LPF	WO2024230647A1_B009	.	CC1=CC(NC2=NC(C[C@@]3(C(=O)NCCCCCCCCCNC4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CCN(CC4=C(F)C(C#N)=CC=C4)[C@H](C)C3)=C(F)C=C2)=NN1	C47H54F2N10O5	AURKA	O14965	CRBN	WO-2024230647-A1
TPD-1LJ84O	WO2024230647A1_B010	.	CC1=CC(NC2=NC(CC3(C(=O)NCCCCCCNC4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CCN(CC4=C(F)C(C#N)=CC=C4)CC3)=C(F)C=C2)=NN1	C43H46F2N10O5	AURKA	O14965	CRBN	WO-2024230647-A1
TPD-5BBZ4O	WO2024230647A1_B011	.	CC1=CC(NC2=NC(CC3(C(=O)NCCCCCCCNC4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CCN(CC4=C(F)C(C#N)=CC=C4)CC3)=C(F)C=C2)=NN1	C44H48F2N10O5	AURKA	O14965	CRBN	WO-2024230647-A1
TPD-UXZY2K	WO2024230647A1_B012	.	CC1=CC(NC2=NC(CC3(C(=O)NCCCCCCCCNC4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CCN(CC4=C(F)C(C#N)=CC=C4)CC3)=C(F)C=C2)=NN1	C45H50F2N10O5	AURKA	O14965	CRBN	WO-2024230647-A1
TPD-ATSDUN	WO2024230647A1_B013	.	CC1=CC(NC2=NC(C[C@@]3(C(=O)NCCCCCCCOC4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CCN(CC4=C(F)C(C#N)=CC=C4)[C@H](C)C3)=C(F)C=C2)=NN1	C45H49F2N9O6	AURKA	O14965	CRBN	WO-2024230647-A1
TPD-3KANGC	WO2024230647A1_B014	.	CC1=CC(NC2=NC(C[C@@]3(C(=O)NCCCCCCC#CC4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CCN(CC4=C(F)C(Cl)=CC=C4)[C@H](C)C3)=C(F)C=C2)=NN1	C45H47ClF2N8O5	AURKA	O14965	CRBN	WO-2024230647-A1
TPD-JO5I36	WO2024230647A1_B015	.	CC1=CC(NC2=NC(C[C@@]3(C(=O)NCCCCCCCCC4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CCN(CC4=C(F)C(Cl)=CC=C4)[C@H](C)C3)=C(F)C=C2)=NN1	C45H51ClF2N8O5	AURKA	O14965	CRBN	WO-2024230647-A1
TPD-FZBZET	WO2024230647A1_B016	.	CC1=CC(NC2=NC(C[C@@]3(C(=O)O)CCN(CC4=C(F)C(C#N)=CC=C4)[C@H](C)C3)=C(F)C(C(=O)NCCN3CCN(C4=CC=C(N5CCC(=O)NC5=O)C=C4)CC3)=C2)=NN1	C42H47F2N11O5	AURKA	O14965	CRBN	WO-2024230647-A1
TPD-CFGB8G	WO2024230647A1_B017	.	CC1=CC(NC2=NC(C[C@@]3(C(=O)O)CCN(CC4=C(F)C(C#N)=CC=C4)[C@H](C)C3)=C(F)C(C(=O)NCCCN3CCN(C4=CC=C(N5CCC(=O)NC5=O)C=C4)CC3)=C2)=NN1	C43H49F2N11O5	AURKA	O14965	CRBN	WO-2024230647-A1
TPD-DTPRRD	WO2024230647A1_B018	.	CC1=CC(NC2=NC(C[C@@]3(C(=O)O)CCN(CC4=C(F)C(Cl)=CC=C4)[C@H](C)C3)=C(F)C(C#CCCN3CCN(C4=CC(N5CCC(=O)NC5=O)=CC=C4)CC3)=C2)=NN1	C42H46ClF2N9O4	AURKA	O14965	CRBN	WO-2024230647-A1
TPD-WRA7XB	WO2024230647A1_B019	.	CC1=CC(NC2=NC(C[C@@]3(C(=O)O)CCN(CC4=C(F)C(Cl)=CC=C4)[C@H](C)C3)=C(F)C(C#CCCN3CCN(C4=CC=C(N5CCC(=O)NC5=O)C=C4)CC3)=C2)=NN1	C42H46ClF2N9O4	AURKA	O14965	CRBN	WO-2024230647-A1
TPD-M4348P	WO2024230647A1_B020	.	CC1=CC(NC2=NC(C[C@@]3(C(=O)O)CCN(CC4=C(F)C(Cl)=CC=C4)[C@H](C)C3)=C(F)C(C#CCN3CCN(C4=CC=C(N5CCC(=O)NC5=O)C=C4)CC3)=C2)=NN1	C41H44ClF2N9O4	AURKA	O14965	CRBN	WO-2024230647-A1
TPD-AAEFA4	WO2024230647A1_B021	.	CC1=CC(NC2=NC(C[C@@]3(C(=O)O)CCN(CC4=C(F)C(Cl)=CC=C4)[C@H](C)C3)=C(F)C(C#CCN3CCN(C4=CC(N5CCC(=O)NC5=O)=CC=C4)CC3)=C2)=NN1	C41H44ClF2N9O4	AURKA	O14965	CRBN	WO-2024230647-A1
TPD-VPR0BG	WO2024230647A1_B022	.	CC1=CC(NC2=NC(C[C@@]3(C(=O)NCCCN4CCN(C5=CC=C(N6CCC(=O)NC6=O)C=C5)CC4)CCN(CC4=CC=CC(Cl)=C4F)[C@H](C)C3)=C(F)C=C2)=NN1	C41H49ClF2N10O3	AURKA	O14965	CRBN	WO-2024230647-A1
TPD-BQEJ7O	WO2024230647A1_B023	.	CC1=CC(NC2=NC(C[C@@]3(C(=O)NCCCCN4CCN(C5=CC=C(N6CCC(=O)NC6=O)C=C5)CC4)CCN(CC4=C(F)C(C#N)=CC=C4)[C@H](C)C3)=C(F)C=C2)=NN1	C43H51F2N11O3	AURKA	O14965	CRBN	WO-2024230647-A1
TPD-580M95	WO2024230647A1_B024	.	CC1=CC(NC2=NC(C[C@@]3(C(=O)NCCCCCN4CCN(C5=CC=C(N6CCC(=O)NC6=O)C=C5)CC4)CCN(CC4=C(F)C(Cl)=CC=C4)[C@H](C)C3)=C(F)C=C2)=NN1	C43H53ClF2N10O3	AURKA	O14965	CRBN	WO-2024230647-A1
TPD-SIHB9J	WO2024230647A1_B025	.	CC1=CC(NC2=NC(C[C@@]3(C(=O)NCCCN4CCN(C5=CC(N6CCC(=O)NC6=O)=CC=C5)CC4)CCN(CC4=C(F)C(C#N)=CC=C4)[C@H](C)C3)=C(F)C=C2)=NN1	C42H49F2N11O3	AURKA	O14965	CRBN	WO-2024230647-A1
TPD-9H5DB7	WO2024230647A1_B026	.	CC1=CC(NC2=NC(C[C@@]3(C(=O)NCCCCCN4CCN(C5=CC(N6CCC(=O)NC6=O)=CC=C5)CC4)CCN(CC4=C(F)C(C#N)=CC=C4)[C@H](C)C3)=C(F)C=C2)=NN1	C44H53F2N11O3	AURKA	O14965	CRBN	WO-2024230647-A1
TPD-JUKUHB	WO2024230647A1_B027	.	CC1=CC(NC2=NC(C[C@@]3(C(=O)NCCCCN4CCN(C5=CC=CC(N6CCC(=O)NC6=O)=C5)CC4)CCN(CC4=C(F)C(Cl)=CC=C4)[C@H](C)C3)=C(F)C=C2)=NN1	C42H51ClF2N10O3	AURKA	O14965	CRBN	WO-2024230647-A1
TPD-LLAAI2	WO2024230647A1_B028	.	CC1=CC(NC2=NC(C[C@@]3(C(=O)NCCCCN4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CCN(CC4=C(F)C(C#N)=CC=C4)[C@H](C)C3)=C(F)C=C2)=NN1	C46H51F2N11O5	AURKA	O14965	CRBN	WO-2024230647-A1
TPD-WMTJ2T	WO2024230647A1_B029	.	CC1=CC(NC2=NC(C[C@@]3(C(=O)NC4CN(CCCCNC5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CCN(CC4=CC=CC(Cl)=C4F)[C@H](C)C3)=C(F)C=C2)=NN1	C44H49ClF2N10O5	AURKA	O14965	CRBN	WO-2024230647-A1
TPD-E3W6SB	WO2024230647A1_B030	.	CC1=CC(NC2=NC(C[C@@]3(C(=O)NC4CCN(C5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC4)CCN(CC4=CC=CC(Cl)=C4F)[C@H](C)C3)=C(F)C=C2)=NN1	C47H53ClF2N10O5	AURKA	O14965	CRBN	WO-2024230647-A1
TPD-VQH39B	WO2024230647A1_B031	.	CC1=CC(NC2=NC(C[C@@]3(C(=O)NC4CN(CC5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)C4)CCN(CC4=CC=CC(Cl)=C4F)[C@H](C)C3)=C(F)C=C2)=NN1	C46H51ClF2N10O5	AURKA	O14965	CRBN	WO-2024230647-A1
TPD-ZIAHXN	WO2024230647A1_B032	.	CC1=CC(NC2=NC(C[C@@]3(C(=O)NCCN4CCN(C5=CC=C(N6CCC(=O)NC6=O)C=C5)CC4)CCN(CC4=C(F)C(C#N)=CC=C4)[C@H](C)C3)=C(F)C=C2)=NN1	C41H47F2N11O3	AURKA	O14965	CRBN	WO-2024230647-A1
TPD-V8630H	WO2024230647A1_B033	.	CC1=CC(NC2=NC(C[C@@]3(C(=O)NC4CN(CC5CN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)C4)CCN(CC4=C(F)C(Cl)=CC=C4)[C@H](C)C3)=C(F)C=C2)=NN1	C44H47ClF2N10O5	AURKA	O14965	CRBN	WO-2024230647-A1
TPD-542PB1	WO2024230647A1_B034	.	CC1=CC(NC2=NC(C[C@@]3(C(=O)NC4CCN(C5CCN(C6=CC=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)CCN(CC4=C(F)C(C#N)=CC=C4)[C@H](C)C3)=C(F)C=C2)=NN1	C45H53F2N11O3	AURKA	O14965	CRBN	WO-2024230647-A1
TPD-VO48OH	WO2024230647A1_B035	.	CC1=CC(NC2=NC(C[C@@]3(C(=O)NC4CN(CC5CN(C6=CC=C(N7CCC(=O)NC7=O)C=C6)C5)C4)CCN(CC4=C(F)C(Cl)=CC=C4)[C@H](C)C3)=C(F)C=C2)=NN1	C41H47ClF2N10O3	AURKA	O14965	CRBN	WO-2024230647-A1
TPD-3VVXM9	WO2024230647A1_B037	.	CC1=CC(NC2=NC(C[C@@]3(C(=O)NC4CN(C5CCN(C6=CC=C(N7CCC(=O)NC7=O)C=C6)CC5)C4)CCN(CC4=C(F)C(C#N)=CC=C4)[C@H](C)C3)=C(F)C=C2)=NN1	C43H49F2N11O3	AURKA	O14965	CRBN	WO-2024230647-A1
TPD-5UF7MP	WO2024230647A1_B038	.	CC1=CC(NC2=NC(CC3(C(=O)O)CCN(CC4=C(F)C(Cl)=CC=C4)CC3)=C(F)C(N3CCN(CC4CCN(C5=CC=C(N6CCC(=O)NC6=O)C=C5)CC4)CC3)=C2)=NN1	C43H51ClF2N10O4	AURKA	O14965	CRBN	WO-2024230647-A1
TPD-KQT5HQ	WO2024230647A1_B039	.	CC1=CC(NC2=NC(C[C@@]3(C(=O)NC4CN(C5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)C4)CCN(CC4=C(F)C(C#N)=CC=C4)[C@H](C)C3)=C(F)C=C2)=NN1	C46H49F2N11O5	AURKA	O14965	CRBN	WO-2024230647-A1
TPD-O45CSF	WO2024230647A1_B040	.	CC1=CC(NC2=NC(CC3(C(=O)O)CCN(CC4=C(F)C(Cl)=CC=C4)CC3)=C(F)C(N3CCN(CC4CN(C5=CC=C(N6CCC(=O)NC6=O)C=C5)C4)CC3)=C2)=NN1	C41H47ClF2N10O4	AURKA	O14965	CRBN	WO-2024230647-A1
TPD-1T7TNR	WO2024230647A1_B041	.	CC1=CC(NC2=NC(CC3(C(=O)O)CCN(CC4=C(F)C(Cl)=CC=C4)CC3)=C(F)C(N3CCN(C4CCN(C5=CC=C(N6CCC(=O)NC6=O)C=C5)CC4)CC3)=C2)=NN1	C42H49ClF2N10O4	AURKA	O14965	CRBN	WO-2024230647-A1
TPD-H6IMFY	WO2024230647A1_B042	.	CC1=CC(NC2=NC(CC3(C(=O)O)CCN(CC4=C(F)C(Cl)=CC=C4)CC3)=C(F)C(N3CCN(C4CN(C5=CC=C(N6CCC(=O)NC6=O)C=C5)C4)CC3)=C2)=NN1	C40H45ClF2N10O4	AURKA	O14965	CRBN	WO-2024230647-A1
TPD-8YYLJH	WO2024230647A1_B043	.	CC1=CC(NC2=NC(CC3(C(=O)O)CCN(CC4=C(F)C(Cl)=CC=C4)CC3)=C(C3=CCN(CC4CCN(C5=CC=C(N6CCC(=O)NC6=O)C=C5)CC4)CC3)C=C2F)=NN1	C44H50ClF2N9O4	AURKA	O14965	CRBN	WO-2024230647-A1
TPD-BZGJHV	WO2024230647A1_B044	.	CC1=CC(NC2=NC(CC3(C(=O)O)CCN(CC4=C(F)C(Cl)=CC=C4)CC3)=C(C3=CCN(CC4CN(C5=CC=C(N6CCC(=O)NC6=O)C=C5)C4)CC3)C=C2F)=NN1	C42H46ClF2N9O4	AURKA	O14965	CRBN	WO-2024230647-A1
TPD-S9Z7Z8	WO2024230647A1_B045	.	CC1=CC(NC2=NC(CC3(C(=O)O)CCN(CC4=C(F)C(Cl)=CC=C4)CC3)=C(F)C(C3CN(CC4CN(C5=CC=C(N6CCC(=O)NC6=O)C=C5)C4)C3)=C2)=NN1	C40H44ClF2N9O4	AURKA	O14965	CRBN	WO-2024230647-A1
TPD-SGMCU9	WO2024230647A1_B046	.	CC1=CC(NC2=NC(CC3(C(=O)O)CCN(CC4=C(F)C(Cl)=CC=C4)CC3)=C(F)C(N3CCC(CN4CCN(C5=CC=C(N6CCC(=O)NC6=O)C=C5)CC4)CC3)=C2)=NN1	C43H51ClF2N10O4	AURKA	O14965	CRBN	WO-2024230647-A1
TPD-AEYYIA	WO2024230647A1_B047	.	CC1=CC(NC2=CC=C(F)C(CC3(C(=O)NC4CN(CC5CN(C6=CC=C(C7CCC(=O)NC7=O)C=C6)C5)C4)CCN(CC4=CC=CC(Cl)=C4F)CC3)=N2)=NN1	C41H46ClF2N9O3	AURKA	O14965	CRBN	WO-2024230647-A1
TPD-T1WPMS	WO2024230647A1_B048	.	CC1=CC(NC2=CC=C(F)C(CC3(C(=O)NC4CN(CC5CN(C6=CC=C(N7CCC(=O)NC7=O)C=C6)C5)C4)CCN(CC4=CC=CC(Cl)=C4F)CC3)=N2)=NN1	C40H45ClF2N10O3	AURKA	O14965	CRBN	WO-2024230647-A1
TPD-K7IS1L	WO2024230647A1_B049	.	CC1=CC(NC2=CC=C(F)C(CC3(C(=O)NC4CN(CC5CN(C6=CC=C(N7CCC(=O)NC7=O)C=N6)C5)C4)CCN(CC4=CC=CC(Cl)=C4F)CC3)=N2)=NN1	C39H44ClF2N11O3	AURKA	O14965	CRBN	WO-2024230647-A1
TPD-6VR4L6	WO2024230647A1_B050	.	CC1=CC(NC2=NC(CC3(C(=O)NCC4CN(C5CN(C6=CC=C(N7CCC(=O)NC7=O)C=C6)C5)C4)CCN(CC4=C(F)C(C#N)=CC=C4)CC3)=C(F)C=C2)=NN1	C41H45F2N11O3	AURKA	O14965	CRBN	WO-2024230647-A1
TPD-FS3DGA	WO2024230647A1_B051	.	CC1=CC(NC2=NC(CC3(C(=O)NC4CN(C5CCN(C6=CC=C(N7CCC(=O)NC7=O)C=C6)CC5)C4)CCN(CC4=CC=CC(Cl)=C4F)CC3)=C(F)C=C2)=NN1	C41H47ClF2N10O3	AURKA	O14965	CRBN	WO-2024230647-A1
TPD-UAG2FJ	WO2024230647A1_B057	.	CC1=CC(NC2=NC(CC3(C(=O)NC4CCN(CCCC#CC5=CC=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)CCN(CC4=C(F)C(Cl)=CC=C4)CC3)=C(F)C=C2)=NN1	C46H50ClF2N9O4	AURKA	O14965	CRBN	WO-2024230647-A1
TPD-SRM991	WO2024230647A1_B058	.	CC1=CC(NC2=NC(CC3(C(=O)O)CCN(CC4=C(F)C(Cl)=CC=C4)CC3)=C(C#CCN3CCN(C4=CC=C(N5CCC(=O)NC5=O)C=C4)CC3)C=C2F)=NN1	C40H42ClF2N9O4	AURKA	O14965	CRBN	WO-2024230647-A1
TPD-UD9HMO	WO2024230647A1_B059	.	CC1=CC(NC2=NC(CC3(C(=O)O)CCN(CC4=C(F)C(Cl)=CC=C4)CC3)=C(C#CCCN3CCN(C4=CC=CC(N5CCC(=O)NC5=O)=C4)CC3)C=C2F)=NN1	C41H44ClF2N9O4	AURKA	O14965	CRBN	WO-2024230647-A1
TPD-49Y098	WO2024230647A1_B061	.	O=C1CCN(C2=CC=C(N3CCN(CCC#CC4=CC(F)=C(NC5=NC=CS5)N=C4CC4(C(=O)O)CCN(CC5=C(F)C(Cl)=CC=C5)CC4)CC3)C=C2)C(=O)N1	C40H41ClF2N8O4S	AURKA	O14965	CRBN	WO-2024230647-A1
TPD-ZPRSHJ	WO2024230647A1_B062	.	O=C1CCN(C2=CC=C(N3CCC(CN4CCN(C5=CC(F)=C(NC6=NC=CS6)N=C5CC5(C(=O)O)CCN(CC6=C(F)C(Cl)=CC=C6)CC5)CC4)CC3)C=C2)C(=O)N1	C42H48ClF2N9O4S	AURKA	O14965	CRBN	WO-2024230647-A1
TPD-IP5TV6	WO2024230647A1_B063	.	CC1=CC(NC2=NC(CC3(C(=O)O)CCN(CC4=C(F)C(Cl)=CC=C4)CC3)=C(C3=CCN(C4CCN(C5=CC=C(N6CCC(=O)NC6=O)C=C5)CC4)CC3)C=C2F)=NN1	C43H48ClF2N9O4	AURKA	O14965	CRBN	WO-2024230647-A1
TPD-F0ODMV	WO2024230647A1_B065	.	CC1=CC(NC2=NC(CC3(C(=O)O)CCN(CC4=C(F)C(Cl)=CC=C4)CC3)=C(C#CCCN3CCN(C4=NC=C(N5CCC(=O)NC5=O)S4)CC3)C=C2F)=NN1	C38H41ClF2N10O4S	AURKA	O14965	CRBN	WO-2024230647-A1
TPD-ERUJK9	WO2024230647A1_B066	.	O=C1CCN(C2=CN=C(N3CCN(CCC#CC4=CC(F)=C(NC5=NC=CS5)N=C4CC4(C(=O)O)CCN(CC5=C(F)C(Cl)=CC=C5)CC4)CC3)S2)C(=O)N1	C37H38ClF2N9O4S2	AURKA	O14965	CRBN	WO-2024230647-A1
TPD-A1FW0J	WO2024230647A1_B067	.	O=C1CCN(C2=CC=C(N3CCN(CCC#CC4=CC(F)=C(NC5=NC=CS5)N=C4CC4(C(=O)O)CCN(CC5=C(F)C(Cl)=CC=C5)CC4)CC3)N=C2)C(=O)N1	C39H40ClF2N9O4S	AURKA	O14965	CRBN	WO-2024230647-A1
TPD-ZXASSR	WO2024230647A1_B068	.	O=C1CCN(C2=CN=C(N3CCN(CCC#CC4=CC(F)=C(NC5=NC=CS5)N=C4CC4(C(=O)N5CCC5)CCN(CC5=C(F)C(Cl)=CC=C5)CC4)CC3)S2)C(=O)N1	C40H43ClF2N10O3S2	AURKA	O14965	CRBN	WO-2024230647-A1
TPD-12XU93	WO2024233747A1_P-1	.	CN1N=C(C2CCC(=O)NC2=O)C2=C1C=C(NC1CCN(C(=O)[C@H]3CC[C@H](N4C=C(NC(=O)C5=C6N=C(N7C[C@H](N)C[C@@H](F)C7)C=CN6N=C5)C(C(F)F)=N4)CC3)CC1)C=C2	C41H48F3N13O4	IRAK4	Q9NWZ3	CRBN	WO-2024233747-A1
TPD-JCYN7N	WO2024233747A1_P-10	5-[(3R,5R)-3-amino-5-fluoropiperidin-1-yl]-N-[3-(difluoromethyl)-1-[4-[2-[4-[3-(2,6-dioxopiperidin-3-yl)-1-methylindazol-6-yl]piperazin-1-yl]ethyl]cyclohexyl]pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide	CN1N=C(C2CCC(=O)NC2=O)C2=CC=C(N3CCN(CC[C@H]4CC[C@H](N5C=C(NC(=O)C6=C7N=C(N8C[C@H](N)C[C@@H](F)C8)C=CN7N=C6)C(C(F)F)=N5)CC4)CC3)C=C21	C41H50F3N13O3	IRAK4	Q9NWZ3	CRBN	WO-2024233747-A1
TPD-7PD554	WO2024233747A1_P-11	5-[(3R,5R)-3-amino-5-fluoropiperidin-1-yl]-N-[3-(difluoromethyl)-1-[4-[2-[4-[3-(2,6-dioxopiperidin-3-yl)-1-methylindazol-7-yl]piperazin-1-yl]ethyl]cyclohexyl]pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide	CN1N=C(C2CCC(=O)NC2=O)C2=C1C(N1CCN(CC[C@H]3CC[C@H](N4C=C(NC(=O)C5=C6N=C(N7C[C@H](N)C[C@@H](F)C7)C=CN6N=C5)C(C(F)F)=N4)CC3)CC1)=CC=C2	C41H50F3N13O3	IRAK4	Q9NWZ3	CRBN	WO-2024233747-A1
TPD-UD1WUV	WO2024233747A1_P-12	.	CN1N=C(C2CCC(=O)NC2=O)C2=C1C=C(NC1CC3(C1)CN(C[C@H]1CC[C@H](N4C=C(NC(=O)C5=C6N=C(N7C[C@H](N)C[C@@H](F)C7)C=CN6N=C5)C(C(F)F)=N4)CC1)C3)C=C2	C42H50F3N13O3	IRAK4	Q9NWZ3	CRBN	WO-2024233747-A1
TPD-ABI2ED	WO2024233747A1_P-13	5-[(3R,5R)-3-amino-5-fluoropiperidin-1-yl]-N-[3-(difluoromethyl)-1-[4-[[3-[[3-(2,6-dioxopiperidin-3-yl)-1-methylindazol-6-yl]amino]azetidin-1-yl]methyl]cyclohexyl]pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide	CN1N=C(C2CCC(=O)NC2=O)C2=C1C=C(NC1CN(C[C@H]3CC[C@H](N4C=C(NC(=O)C5=C6N=C(N7C[C@H](N)C[C@@H](F)C7)C=CN6N=C5)C(C(F)F)=N4)CC3)C1)C=C2	C39H46F3N13O3	IRAK4	Q9NWZ3	CRBN	WO-2024233747-A1
TPD-SDNOYT	WO2024233747A1_P-14	5-[(3R,5R)-3-amino-5-fluoropiperidin-1-yl]-N-[3-(difluoromethyl)-1-[4-[[4-[3-(2,6-dioxopiperidin-3-yl)-1-methylindazol-6-yl]piperazin-1-yl]methyl]cyclohexyl]pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide	CN1N=C(C2CCC(=O)NC2=O)C2=CC=C(N3CCN(C[C@H]4CC[C@H](N5C=C(NC(=O)C6=C7N=C(N8C[C@H](N)C[C@@H](F)C8)C=CN7N=C6)C(C(F)F)=N5)CC4)CC3)C=C21	C40H48F3N13O3	IRAK4	Q9NWZ3	CRBN	WO-2024233747-A1
TPD-1GQCCF	WO2024233747A1_P-15	5-[(3R,5R)-3-amino-5-fluoropiperidin-1-yl]-N-[3-(difluoromethyl)-1-[4-[[[1-[3-(2,6-dioxopiperidin-3-yl)-1-methylindazol-7-yl]piperidin-4-yl]amino]methyl]cyclohexyl]pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide	CN1N=C(C2CCC(=O)NC2=O)C2=C1C(N1CCC(NC[C@H]3CC[C@H](N4C=C(NC(=O)C5=C6N=C(N7C[C@H](N)C[C@@H](F)C7)C=CN6N=C5)C(C(F)F)=N4)CC3)CC1)=CC=C2	C41H50F3N13O3	IRAK4	Q9NWZ3	CRBN	WO-2024233747-A1
TPD-77837I	WO2024233747A1_P-16	5-[(3R,5R)-3-amino-5-fluoropiperidin-1-yl]-N-[3-(difluoromethyl)-1-[4-[2-[4-[[3-(2,6-dioxopiperidin-3-yl)-1-methylindazol-6-yl]amino]piperidin-1-yl]ethyl]cyclohexyl]pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide	CN1N=C(C2CCC(=O)NC2=O)C2=CC=C(NC3CCN(CC[C@H]4CC[C@H](N5C=C(NC(=O)C6=C7N=C(N8C[C@H](N)C[C@@H](F)C8)C=CN7N=C6)C(C(F)F)=N5)CC4)CC3)C=C21	C42H52F3N13O3	IRAK4	Q9NWZ3	CRBN	WO-2024233747-A1
TPD-S7MG7Q	WO2024233747A1_P-17	5-[(3R,5R)-3-amino-5-fluoropiperidin-1-yl]-N-[3-(difluoromethyl)-1-[4-[[4-[3-(2,6-dioxopiperidin-3-yl)-1-methylindazole-6-carbonyl]piperazin-1-yl]methyl]cyclohexyl]pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide	CN1N=C(C2CCC(=O)NC2=O)C2=C1C=C(C(=O)N1CCN(C[C@H]3CC[C@H](N4C=C(NC(=O)C5=C6N=C(N7C[C@H](N)C[C@@H](F)C7)C=CN6N=C5)C(C(F)F)=N4)CC3)CC1)C=C2	C41H48F3N13O4	IRAK4	Q9NWZ3	CRBN	WO-2024233747-A1
TPD-6QI5YL	SCHEMBL31236454	5-[(3S,4S)-3-amino-4-fluoropiperidin-1-yl]-N-[3-(difluoromethyl)-1-[4-[[4-[[3-(2,6-dioxopiperidin-3-yl)-1-methylindazol-6-yl]amino]piperidin-1-yl]methyl]cyclohexyl]pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide	CN1N=C(C2CCC(=O)NC2=O)C2=C1C=C(NC1CCN(C[C@H]3CC[C@H](N4C=C(NC(=O)C5=C6N=C(N7CC[C@H](F)[C@@H](N)C7)C=CN6N=C5)C(C(F)F)=N4)CC3)CC1)C=C2	C41H50F3N13O3	IRAK4	Q9NWZ3	CRBN	WO-2024233747-A1
TPD-EKPCRX	WO2024233747A1_P-19	5-[(3R,5S)-3-amino-5-fluoropiperidin-1-yl]-N-[3-(difluoromethyl)-1-[4-[[4-[[3-(2,6-dioxopiperidin-3-yl)-1-methylindazol-6-yl]amino]piperidin-1-yl]methyl]cyclohexyl]pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide	CN1N=C(C2CCC(=O)NC2=O)C2=C1C=C(NC1CCN(C[C@H]3CC[C@H](N4C=C(NC(=O)C5=C6N=C(N7C[C@H](N)C[C@H](F)C7)C=CN6N=C5)C(C(F)F)=N4)CC3)CC1)C=C2	C41H50F3N13O3	IRAK4	Q9NWZ3	CRBN	WO-2024233747-A1
TPD-16W1SL	SCHEMBL31236445	5-[(3R,5R)-3-amino-5-fluoropiperidin-1-yl]-N-[3-(difluoromethyl)-1-[4-[[4-[[3-(2,6-dioxopiperidin-3-yl)-1-methylindazol-6-yl]amino]piperidin-1-yl]methyl]cyclohexyl]pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide	CN1N=C(C2CCC(=O)NC2=O)C2=C1C=C(NC1CCN(C[C@H]3CC[C@H](N4C=C(NC(=O)C5=C6N=C(N7C[C@H](N)C[C@@H](F)C7)C=CN6N=C5)C(C(F)F)=N4)CC3)CC1)C=C2	C41H50F3N13O3	IRAK4	Q9NWZ3	CRBN	WO-2024233747-A1
TPD-OX2V3Z	WO2024233747A1_P-20	5-[(5R)-5-amino-3,3-difluoropiperidin-1-yl]-N-[3-(difluoromethyl)-1-[4-[[4-[[3-(2,6-dioxopiperidin-3-yl)-1-methylindazol-6-yl]amino]piperidin-1-yl]methyl]cyclohexyl]pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide	CN1N=C(C2CCC(=O)NC2=O)C2=C1C=C(NC1CCN(C[C@H]3CC[C@H](N4C=C(NC(=O)C5=C6N=C(N7C[C@H](N)CC(F)(F)C7)C=CN6N=C5)C(C(F)F)=N4)CC3)CC1)C=C2	C41H49F4N13O3	IRAK4	Q9NWZ3	CRBN	WO-2024233747-A1
TPD-6UWHDK	WO2024233747A1_P-21	5-[(3S,4R)-3-amino-4-fluoropiperidin-1-yl]-N-[3-(difluoromethyl)-1-[4-[[4-[[3-(2,6-dioxopiperidin-3-yl)-1-methylindazol-6-yl]amino]piperidin-1-yl]methyl]cyclohexyl]pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide	CN1N=C(C2CCC(=O)NC2=O)C2=C1C=C(NC1CCN(C[C@H]3CC[C@H](N4C=C(NC(=O)C5=C6N=C(N7CC[C@@H](F)[C@@H](N)C7)C=CN6N=C5)C(C(F)F)=N4)CC3)CC1)C=C2	C41H50F3N13O3	IRAK4	Q9NWZ3	CRBN	WO-2024233747-A1
TPD-T89WUU	WO2024233747A1_P-23	5-[(3R,5R)-3-amino-5-fluoropiperidin-1-yl]-N-[3-(difluoromethyl)-1-[4-[[(3R,4S)-4-[[3-(2,6-dioxopiperidin-3-yl)-1-methylindazol-6-yl]amino]-3-fluoropiperidin-1-yl]methyl]cyclohexyl]pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide	CN1N=C(C2CCC(=O)NC2=O)C2=C1C=C(N[C@H]1CCN(C[C@H]3CC[C@H](N4C=C(NC(=O)C5=C6N=C(N7C[C@H](N)C[C@@H](F)C7)C=CN6N=C5)C(C(F)F)=N4)CC3)C[C@H]1F)C=C2	C41H49F4N13O3	IRAK4	Q9NWZ3	CRBN	WO-2024233747-A1
TPD-2XWAEG	WO2024233747A1_P-24	.	CN1N=C(C2CCC(=O)NC2=O)C2=C1C=C(N[C@@H]1CCN(C[C@H]3CC[C@H](N4C=C(NC(=O)C5=C6N=C(N7C[C@H](N)C[C@@H](F)C7)C=CN6N=C5)C(C(F)F)=N4)CC3)C[C@@H]1F)C=C2	C41H49F4N13O3	IRAK4	Q9NWZ3	CRBN	WO-2024233747-A1
TPD-K3IYGI	WO2024233747A1_P-25	5-[(3R,5R)-3-amino-5-fluoropiperidin-1-yl]-N-[3-(difluoromethyl)-1-[4-[[(3S,4S)-4-[[3-(2,6-dioxopiperidin-3-yl)-1-methylindazol-6-yl]amino]-3-fluoropiperidin-1-yl]methyl]cyclohexyl]pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide	CN1N=C(C2CCC(=O)NC2=O)C2=C1C=C(N[C@H]1CCN(C[C@H]3CC[C@H](N4C=C(NC(=O)C5=C6N=C(N7C[C@H](N)C[C@@H](F)C7)C=CN6N=C5)C(C(F)F)=N4)CC3)C[C@@H]1F)C=C2	C41H49F4N13O3	IRAK4	Q9NWZ3	CRBN	WO-2024233747-A1
TPD-ZXZ398	WO2024233747A1_P-26	.	CN1N=C(C2CCC(=O)NC2=O)C2=C1C=C(OC1CCN(C[C@H]3CC[C@H](N4C=C(NC(=O)C5=C6N=C(N7C[C@H](N)C[C@@H](F)C7)C=CN6N=C5)C(C(F)F)=N4)CC3)CC1)C=C2	C41H49F3N12O4	IRAK4	Q9NWZ3	CRBN	WO-2024233747-A1
TPD-VW4T2P	WO2024233747A1_P-27	N-[3-(difluoromethyl)-1-[4-[[4-[[3-(2,6-dioxopiperidin-3-yl)-1-methylindazol-6-yl]amino]piperidin-1-yl]methyl]cyclohexyl]pyrazol-4-yl]-5-morpholin-4-ylpyrazolo[1,5-a]pyrimidine-3-carboxamide	CN1N=C(C2CCC(=O)NC2=O)C2=C1C=C(NC1CCN(C[C@H]3CC[C@H](N4C=C(NC(=O)C5=C6N=C(N7CCOCC7)C=CN6N=C5)C(C(F)F)=N4)CC3)CC1)C=C2	C40H48F2N12O4	IRAK4	Q9NWZ3	CRBN	WO-2024233747-A1
TPD-EOTCME	SCHEMBL31236412	5-[(3R,5R)-3-amino-5-fluoropiperidin-1-yl]-N-[3-(difluoromethyl)-1-[4-[[[1-[3-(2,6-dioxopiperidin-3-yl)-1-methylindazol-6-yl]piperidin-4-yl]-methylamino]methyl]cyclohexyl]pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide	CN1N=C(C2CCC(=O)NC2=O)C2=CC=C(N3CCC(N(C)C[C@H]4CC[C@H](N5C=C(NC(=O)C6=C7N=C(N8C[C@H](N)C[C@@H](F)C8)C=CN7N=C6)C(C(F)F)=N5)CC4)CC3)C=C21	C42H52F3N13O3	IRAK4	Q9NWZ3	CRBN	WO-2024233747-A1
TPD-FJHZ3P	SCHEMBL31236424	N-[3-(difluoromethyl)-1-[4-[[[1-[3-(2,6-dioxopiperidin-3-yl)-1-methylindazol-6-yl]piperidin-4-yl]-methylamino]methyl]cyclohexyl]pyrazol-4-yl]-5-morpholin-4-ylpyrazolo[1,5-a]pyrimidine-3-carboxamide	CN1N=C(C2CCC(=O)NC2=O)C2=CC=C(N3CCC(N(C)C[C@H]4CC[C@H](N5C=C(NC(=O)C6=C7N=C(N8CCOCC8)C=CN7N=C6)C(C(F)F)=N5)CC4)CC3)C=C21	C41H50F2N12O4	IRAK4	Q9NWZ3	CRBN	WO-2024233747-A1
TPD-F5LAAI	WO2024233747A1_P-3	5-[(3R,5R)-3-amino-5-fluoropiperidin-1-yl]-N-[3-(difluoromethyl)-1-[4-[[4-[[3-(2,6-dioxopiperidin-3-yl)-1-methylindazol-7-yl]amino]piperidin-1-yl]methyl]cyclohexyl]pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide	CN1N=C(C2CCC(=O)NC2=O)C2=C1C(NC1CCN(C[C@H]3CC[C@H](N4C=C(NC(=O)C5=C6N=C(N7C[C@H](N)C[C@@H](F)C7)C=CN6N=C5)C(C(F)F)=N4)CC3)CC1)=CC=C2	C41H50F3N13O3	IRAK4	Q9NWZ3	CRBN	WO-2024233747-A1
TPD-G1GYIK	SCHEMBL31236462	5-[(3R,5R)-3-amino-5-fluoropiperidin-1-yl]-N-[3-(difluoromethyl)-1-[4-[[[1-[3-(2,6-dioxopiperidin-3-yl)-1-methylindazol-7-yl]piperidin-4-yl]-methylamino]methyl]cyclohexyl]pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide	CN1N=C(C2CCC(=O)NC2=O)C2=C1C(N1CCC(N(C)C[C@H]3CC[C@H](N4C=C(NC(=O)C5=C6N=C(N7C[C@H](N)C[C@@H](F)C7)C=CN6N=C5)C(C(F)F)=N4)CC3)CC1)=CC=C2	C42H52F3N13O3	IRAK4	Q9NWZ3	CRBN	WO-2024233747-A1
TPD-J2S35O	WO2024233747A1_P-31	.	CN1N=C(C2CCC(=O)NC2=O)C2=C1C=C(N(C)C1CCN(C[C@H]3CC[C@H](N4C=C(NC(=O)C5=C6N=C(N7C[C@H](N)C[C@@H](F)C7)C=CN6N=C5)C(C(F)F)=N4)CC3)CC1)C=C2	C42H52F3N13O3	IRAK4	Q9NWZ3	CRBN	WO-2024233747-A1
TPD-DFFN7M	WO2024233747A1_P-32	N-[3-(difluoromethyl)-1-[4-[[4-[[3-(2,6-dioxopiperidin-3-yl)-1-methylindazol-6-yl]-methylamino]piperidin-1-yl]methyl]cyclohexyl]pyrazol-4-yl]-5-morpholin-4-ylpyrazolo[1,5-a]pyrimidine-3-carboxamide	CN1N=C(C2CCC(=O)NC2=O)C2=C1C=C(N(C)C1CCN(C[C@H]3CC[C@H](N4C=C(NC(=O)C5=C6N=C(N7CCOCC7)C=CN6N=C5)C(C(F)F)=N4)CC3)CC1)C=C2	C41H50F2N12O4	IRAK4	Q9NWZ3	CRBN	WO-2024233747-A1
TPD-9JXZ7S	WO2024233747A1_P-33	5-[(3R,5R)-3-amino-5-fluoropiperidin-1-yl]-N-[3-(difluoromethyl)-1-[4-[2-[4-[[3-(2,6-dioxopiperidin-3-yl)-1-methylindazol-6-yl]-methylamino]piperidin-1-yl]ethyl]cyclohexyl]pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide	CN1N=C(C2CCC(=O)NC2=O)C2=C1C=C(N(C)C1CCN(CC[C@H]3CC[C@H](N4C=C(NC(=O)C5=C6N=C(N7C[C@H](N)C[C@@H](F)C7)C=CN6N=C5)C(C(F)F)=N4)CC3)CC1)C=C2	C43H54F3N13O3	IRAK4	Q9NWZ3	CRBN	WO-2024233747-A1
TPD-04D8SU	WO2024233747A1_P-34	N-[3-(difluoromethyl)-1-[4-[2-[4-[[3-(2,6-dioxopiperidin-3-yl)-1-methylindazol-6-yl]-methylamino]piperidin-1-yl]ethyl]cyclohexyl]pyrazol-4-yl]-5-morpholin-4-ylpyrazolo[1,5-a]pyrimidine-3-carboxamide	CN1N=C(C2CCC(=O)NC2=O)C2=C1C=C(N(C)C1CCN(CC[C@H]3CC[C@H](N4C=C(NC(=O)C5=C6N=C(N7CCOCC7)C=CN6N=C5)C(C(F)F)=N4)CC3)CC1)C=C2	C42H52F2N12O4	IRAK4	Q9NWZ3	CRBN	WO-2024233747-A1
TPD-GHONSZ	WO2024233747A1_P-35	N-[3-(difluoromethyl)-1-[4-[2-[[1-[3-(2,6-dioxopiperidin-3-yl)-1-methylindazol-7-yl]piperidin-4-yl]-methylamino]ethyl]cyclohexyl]pyrazol-4-yl]-5-morpholin-4-ylpyrazolo[1,5-a]pyrimidine-3-carboxamide	CN1N=C(C2CCC(=O)NC2=O)C2=C1C(N1CCC(N(C)CC[C@H]3CC[C@H](N4C=C(NC(=O)C5=C6N=C(N7CCOCC7)C=CN6N=C5)C(C(F)F)=N4)CC3)CC1)=CC=C2	C42H52F2N12O4	IRAK4	Q9NWZ3	CRBN	WO-2024233747-A1
TPD-M6AH5J	WO2024233747A1_P-36	5-[(3R,5R)-3-amino-5-fluoropiperidin-1-yl]-N-[3-(difluoromethyl)-1-[1-[2-[(3S)-4-[3-(2,6-dioxopiperidin-3-yl)-1-methylindazol-6-yl]-3-methylpiperazin-1-yl]ethyl]piperidin-4-yl]pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide	C[C@H]1CN(CCN2CCC(N3C=C(NC(=O)C4=C5N=C(N6C[C@H](N)C[C@@H](F)C6)C=CN5N=C4)C(C(F)F)=N3)CC2)CCN1C1=CC=C2C(=C1)N(C)N=C2C1CCC(=O)NC1=O	C41H51F3N14O3	IRAK4	Q9NWZ3	CRBN	WO-2024233747-A1
TPD-BL00TC	SCHEMBL31236448	5-[(3R,5R)-3-amino-5-fluoropiperidin-1-yl]-N-[3-(difluoromethyl)-1-[1-[2-[(3R)-4-[3-(2,6-dioxopiperidin-3-yl)-1-methylindazol-6-yl]-3-methylpiperazin-1-yl]ethyl]piperidin-4-yl]pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide	C[C@@H]1CN(CCN2CCC(N3C=C(NC(=O)C4=C5N=C(N6C[C@H](N)C[C@@H](F)C6)C=CN5N=C4)C(C(F)F)=N3)CC2)CCN1C1=CC=C2C(=C1)N(C)N=C2C1CCC(=O)NC1=O	C41H51F3N14O3	IRAK4	Q9NWZ3	CRBN	WO-2024233747-A1
TPD-7TT5TN	WO2024233747A1_P-38	N-[3-(difluoromethyl)-1-[4-[2-[[1-[3-(2,6-dioxopiperidin-3-yl)-1-methylindazol-6-yl]piperidin-4-yl]-methylamino]ethyl]cyclohexyl]pyrazol-4-yl]-5-morpholin-4-ylpyrazolo[1,5-a]pyrimidine-3-carboxamide	CN1N=C(C2CCC(=O)NC2=O)C2=CC=C(N3CCC(N(C)CC[C@H]4CC[C@H](N5C=C(NC(=O)C6=C7N=C(N8CCOCC8)C=CN7N=C6)C(C(F)F)=N5)CC4)CC3)C=C21	C42H52F2N12O4	IRAK4	Q9NWZ3	CRBN	WO-2024233747-A1
TPD-85XUGA	WO2024233747A1_P-39	.	CN1N=C(C2CCC(=O)NC2=O)C2CC=CC(N(C)C3CCN(CC[C@H]4CC[C@H](N5C=C(NC(=O)C6=C7N=C(N8CCOCC8)C=CN7N=C6)C(C(F)F)=N5)CC4)CC3)=C21	C42H54F2N12O4	IRAK4	Q9NWZ3	CRBN	WO-2024233747-A1
TPD-6L5EKX	WO2024233747A1_P-4	5-[(3R,5R)-3-amino-5-fluoropiperidin-1-yl]-N-[3-(difluoromethyl)-1-[4-[[1-[3-(2,6-dioxopiperidin-3-yl)-1-methylindazol-6-yl]piperidin-4-yl]carbamoyl]cyclohexyl]pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide	CN1N=C(C2CCC(=O)NC2=O)C2=C1C=C(N1CCC(NC(=O)[C@H]3CC[C@H](N4C=C(NC(=O)C5=C6N=C(N7C[C@H](N)C[C@@H](F)C7)C=CN6N=C5)C(C(F)F)=N4)CC3)CC1)C=C2	C41H48F3N13O4	IRAK4	Q9NWZ3	CRBN	WO-2024233747-A1
TPD-CUX7I5	WO2024233747A1_P-40	.	CN1N=C(C2CCC(=O)NC2=O)C2CC=CC(N(C)N3CCN(CCN4CCC(N5C=C(NC(=O)C6=C7N=C(N8C[C@H](N)C[C@@H](F)C8)C=CN7N=C6)C(C(F)F)=N5)CC4)CC3)=C21	C41H54F3N15O3	IRAK4	Q9NWZ3	CRBN	WO-2024233747-A1
TPD-E2FDSP	WO2024233747A1_P-41	N-[3-(difluoromethyl)-1-[4-[[[1-[3-(2,6-dioxopiperidin-3-yl)-1-methylindazol-6-yl]piperidin-4-yl]-methylamino]methyl]cyclohexyl]pyrazol-4-yl]-5-(1,3-oxazolidin-3-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide	CN1N=C(C2CCC(=O)NC2=O)C2=CC=C(N3CCC(N(C)C[C@H]4CC[C@H](N5C=C(NC(=O)C6=C7N=C(N8CCOC8)C=CN7N=C6)C(C(F)F)=N5)CC4)CC3)C=C21	C40H48F2N12O4	IRAK4	Q9NWZ3	CRBN	WO-2024233747-A1
TPD-K4FYET	WO2024233747A1_P-42	N-[3-(difluoromethyl)-1-[4-[[[1-[3-(2,6-dioxopiperidin-3-yl)-1-methylindazol-6-yl]piperidin-4-yl]-methylamino]methyl]cyclohexyl]pyrazol-4-yl]-5-[(1R,5S)-8-oxa-3-azabicyclo[3.2.1]octan-3-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide	CN1N=C(C2CCC(=O)NC2=O)C2=CC=C(N3CCC(N(C)C[C@H]4CC[C@H](N5C=C(NC(=O)C6=C7N=C(N8C[C@H]9CC[C@@H](C8)O9)C=CN7N=C6)C(C(F)F)=N5)CC4)CC3)C=C21	C43H52F2N12O4	IRAK4	Q9NWZ3	CRBN	WO-2024233747-A1
TPD-793XT3	WO2024233747A1_P-43	.	CN(C)C1=NC2=C(C(=O)NC3=CN([C@H]4CC[C@H](CN(C)C5CCN(C6=CC=C7C(=C6)N(C)N=C7C6CCC(=O)NC6=O)CC5)CC4)N=C3C(F)F)C=NN2C=C1	C39H48F2N12O3	IRAK4	Q9NWZ3	CRBN	WO-2024233747-A1
TPD-X25JDM	WO2024233747A1_P-44	N-[3-(difluoromethyl)-1-[4-[[[1-[3-(2,6-dioxopiperidin-3-yl)-1-methylindazol-6-yl]piperidin-4-yl]-methylamino]methyl]cyclohexyl]pyrazol-4-yl]-5-(pyridin-2-ylmethylamino)pyrazolo[1,5-a]pyrimidine-3-carboxamide	CN1N=C(C2CCC(=O)NC2=O)C2=CC=C(N3CCC(N(C)C[C@H]4CC[C@H](N5C=C(NC(=O)C6=C7N=C(NCC8=NC=CC=C8)C=CN7N=C6)C(C(F)F)=N5)CC4)CC3)C=C21	C43H49F2N13O3	IRAK4	Q9NWZ3	CRBN	WO-2024233747-A1
TPD-IEB7ER	WO2024233747A1_P-45	5-(2-aminoethylamino)-N-[3-(difluoromethyl)-1-[4-[[[1-[3-(2,6-dioxopiperidin-3-yl)-1-methylindazol-6-yl]piperidin-4-yl]-methylamino]methyl]cyclohexyl]pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide	CN1N=C(C2CCC(=O)NC2=O)C2=CC=C(N3CCC(N(C)C[C@H]4CC[C@H](N5C=C(NC(=O)C6=C7N=C(NCCN)C=CN7N=C6)C(C(F)F)=N5)CC4)CC3)C=C21	C39H49F2N13O3	IRAK4	Q9NWZ3	CRBN	WO-2024233747-A1
TPD-N414WR	WO2024233747A1_P-46	N-[3-(difluoromethyl)-1-[4-[[[1-[3-(2,6-dioxopiperidin-3-yl)-1-methylindazol-6-yl]piperidin-4-yl]-methylamino]methyl]cyclohexyl]pyrazol-4-yl]-5-[(3S)-3-(1-methylpyrazol-3-yl)pyrrolidin-1-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide	CN1C=CC([C@H]2CCN(C3=NC4=C(C(=O)NC5=CN([C@H]6CC[C@H](CN(C)C7CCN(C8=CC=C9C(=C8)N(C)N=C9C8CCC(=O)NC8=O)CC7)CC6)N=C5C(F)F)C=NN4C=C3)C2)=N1	C45H54F2N14O3	IRAK4	Q9NWZ3	CRBN	WO-2024233747-A1
TPD-0O4SU0	WO2024233747A1_P-47	N-[3-(difluoromethyl)-1-[4-[[[1-[3-(2,6-dioxopiperidin-3-yl)-1-methylindazol-6-yl]piperidin-4-yl]-methylamino]methyl]cyclohexyl]pyrazol-4-yl]-5-[(3R)-3-(1-methylpyrazol-3-yl)pyrrolidin-1-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide	CN1C=CC([C@@H]2CCN(C3=NC4=C(C(=O)NC5=CN([C@H]6CC[C@H](CN(C)C7CCN(C8=CC=C9C(=C8)N(C)N=C9C8CCC(=O)NC8=O)CC7)CC6)N=C5C(F)F)C=NN4C=C3)C2)=N1	C45H54F2N14O3	IRAK4	Q9NWZ3	CRBN	WO-2024233747-A1
TPD-RDGLKM	WO2024233747A1_P-48	N-[3-(difluoromethyl)-1-[4-[[[1-[3-(2,6-dioxopiperidin-3-yl)-1-methylindazol-6-yl]piperidin-4-yl]-methylamino]methyl]cyclohexyl]pyrazol-4-yl]-5-[(6-methylpyridin-3-yl)amino]pyrazolo[1,5-a]pyrimidine-3-carboxamide	CC1=CC=C(NC2=NC3=C(C(=O)NC4=CN([C@H]5CC[C@H](CN(C)C6CCN(C7=CC=C8C(=C7)N(C)N=C8C7CCC(=O)NC7=O)CC6)CC5)N=C4C(F)F)C=NN3C=C2)C=N1	C43H49F2N13O3	IRAK4	Q9NWZ3	CRBN	WO-2024233747-A1
TPD-CVJF7Q	WO2024233747A1_P-49	N-[3-(difluoromethyl)-1-[4-[[[1-[3-(2,6-dioxopiperidin-3-yl)-1-methylindazol-6-yl]piperidin-4-yl]-methylamino]methyl]cyclohexyl]pyrazol-4-yl]-5-(1-methyl-4,6-dihydropyrrolo[3,4-c]pyrazol-5-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide	CN1N=C(C2CCC(=O)NC2=O)C2=CC=C(N3CCC(N(C)C[C@H]4CC[C@H](N5C=C(NC(=O)C6=C7N=C(N8CC9=C(C8)N(C)N=C9)C=CN7N=C6)C(C(F)F)=N5)CC4)CC3)C=C21	C43H50F2N14O3	IRAK4	Q9NWZ3	CRBN	WO-2024233747-A1
TPD-EJREOB	WO2024233747A1_P-5	5-[(3R,5R)-3-amino-5-fluoropiperidin-1-yl]-N-[3-(difluoromethyl)-1-[4-[[[1-[3-(2,6-dioxopiperidin-3-yl)-1-methylindazol-6-yl]piperidin-4-yl]amino]methyl]cyclohexyl]pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide	CN1N=C(C2CCC(=O)NC2=O)C2=C1C=C(N1CCC(NC[C@H]3CC[C@H](N4C=C(NC(=O)C5=C6N=C(N7C[C@H](N)C[C@@H](F)C7)C=CN6N=C5)C(C(F)F)=N4)CC3)CC1)C=C2	C41H50F3N13O3	IRAK4	Q9NWZ3	CRBN	WO-2024233747-A1
TPD-59ZO0H	WO2024233747A1_P-50	5-[(3S)-3-cyanopyrrolidin-1-yl]-N-[3-(difluoromethyl)-1-[4-[[[1-[3-(2,6-dioxopiperidin-3-yl)-1-methylindazol-6-yl]piperidin-4-yl]-methylamino]methyl]cyclohexyl]pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide	CN1N=C(C2CCC(=O)NC2=O)C2=CC=C(N3CCC(N(C)C[C@H]4CC[C@H](N5C=C(NC(=O)C6=C7N=C(N8CC[C@H](C#N)C8)C=CN7N=C6)C(C(F)F)=N5)CC4)CC3)C=C21	C42H49F2N13O3	IRAK4	Q9NWZ3	CRBN	WO-2024233747-A1
TPD-FJ1GFF	WO2024233747A1_P-6	5-[(3R,5R)-3-amino-5-fluoropiperidin-1-yl]-N-[3-(difluoromethyl)-1-[4-[[1-[3-(2,6-dioxopiperidin-3-yl)-1-methylindazol-7-yl]piperidin-4-yl]carbamoyl]cyclohexyl]pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide	CN1N=C(C2CCC(=O)NC2=O)C2=C1C(N1CCC(NC(=O)[C@H]3CC[C@H](N4C=C(NC(=O)C5=C6N=C(N7C[C@H](N)C[C@@H](F)C7)C=CN6N=C5)C(C(F)F)=N4)CC3)CC1)=CC=C2	C41H48F3N13O4	IRAK4	Q9NWZ3	CRBN	WO-2024233747-A1
TPD-GHPWEZ	WO2024233747A1_P-7	5-[(3R,5R)-3-amino-5-fluoropiperidin-1-yl]-N-[3-(difluoromethyl)-1-[4-[2-[4-[[3-(2,6-dioxopiperidin-3-yl)-1-methylindazol-7-yl]-methylamino]piperidin-1-yl]ethyl]cyclohexyl]pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide	CN1N=C(C2CCC(=O)NC2=O)C2=CC=CC(N(C)C3CCN(CC[C@H]4CC[C@H](N5C=C(NC(=O)C6=C7N=C(N8C[C@H](N)C[C@@H](F)C8)C=CN7N=C6)C(C(F)F)=N5)CC4)CC3)=C21	C43H54F3N13O3	IRAK4	Q9NWZ3	CRBN	WO-2024233747-A1
TPD-EKGKWL	WO2024233747A1_P-8	5-[(3R,5R)-3-amino-5-fluoropiperidin-1-yl]-N-[3-(difluoromethyl)-1-[4-[[4-[3-(2,6-dioxopiperidin-3-yl)-1-methylindazol-7-yl]piperazin-1-yl]methyl]cyclohexyl]pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide	CN1N=C(C2CCC(=O)NC2=O)C2=C1C(N1CCN(C[C@H]3CC[C@H](N4C=C(NC(=O)C5=C6N=C(N7C[C@H](N)C[C@@H](F)C7)C=CN6N=C5)C(C(F)F)=N4)CC3)CC1)=CC=C2	C40H48F3N13O3	IRAK4	Q9NWZ3	CRBN	WO-2024233747-A1
TPD-UX6XRF	WO2024233747A1_P-9	5-[(3R,5R)-3-amino-5-fluoropiperidin-1-yl]-N-[3-(difluoromethyl)-1-[4-[4-[[3-(2,6-dioxopiperidin-3-yl)-1-methylindazol-7-yl]amino]piperidine-1-carbonyl]cyclohexyl]pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide	CN1N=C(C2CCC(=O)NC2=O)C2=CC=CC(NC3CCN(C(=O)[C@H]4CC[C@H](N5C=C(NC(=O)C6=C7N=C(N8C[C@H](N)C[C@@H](F)C8)C=CN7N=C6)C(C(F)F)=N5)CC4)CC3)=C21	C41H48F3N13O4	IRAK4	Q9NWZ3	CRBN	WO-2024233747-A1
TPD-SP82OO	SCHEMBL25550417	5-[[4-[2-[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynylnaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxyethyl]piperazin-1-yl]methyl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	C#Cc1cccc2cccc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCCN5CCN(Cc6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)nc4c3F)c12	C45H42FN9O5	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-QUXU9U	WO2024233838A1_2	.	CN1C[C@H](N2CCC(C(=O)NCCOCCOc3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)C[C@@H]1COc1nc(N2CC3CCC(C2)N3)c2cnc(-c3cccc4ccccc34)c(F)c2n1	C52H57FN10O8	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-DS8Z49	WO2024233838A1_3	.	C#Cc1cccc2cccc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC[C@H]5C[C@@H](N6CCN(Cc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CN5C)nc4c3F)c12	C49H49FN10O5	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-UFK9OT	WO2024233838A1_4	.	CN1C[C@H](N2CCN(CC3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)C[C@@H]1COc1nc(N2CC3CCC(C2)N3)c2cnc(-c3cc(O)cc4ccccc34)c(F)c2n1	C52H58FN11O6	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-HT2TGC	WO2024233838A1_5	.	CN1C[C@H](N2CCN(CC3CCN(c4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)C[C@@H]1COc1nc(N2CC3CCC(C2)N3)c2cnc(-c3cc(O)cc4ccccc34)c(F)c2n1	C52H58FN11O6	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-0RSC9B	WO2024233838A1_7	.	CN1C[C@H](N2CCN(C(=O)C3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)C[C@@H]1COc1nc(N2CC3CCC(C2)N3)c2cnc(-c3cc(O)cc4ccccc34)c(F)c2n1	C52H56FN11O7	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-PNLDXU	WO2024233838A1_8	.	CN1C[C@H](N2CCN(Cc3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)C[C@@H]1COc1nc(N2CC3CCC(C2)N3)c2cnc(-c3cc(O)cc4ccccc34)c(F)c2n1	C47H49FN10O6	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-XDTEZN	WO2024233838A1_9	.	O=C1CCC(N2C(=O)c3ccc(N4CCC(C(=O)N5CCN(CC6(COc7nc(N8CC9CCC(C8)N9)c8cnc(-c9cc(O)cc%10ccccc9%10)c(F)c8n7)CC6)CC5)CC4)cc3C2=O)C(=O)N1	C51H53FN10O7	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-FM8H26	WO2024233838A1_10	.	O=C1CCC(N2Cc3cc(CN4CCN(CC5(COc6nc(N7CC8CCC(C7)N8)c7cnc(-c8cc(O)cc9ccccc89)c(F)c7n6)CC5)CC4)ccc3C2=O)C(=O)N1	C46H48FN9O5	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-JHO0S6	WO2024233838A1_11	.	O=C1CCC(N2C(=O)c3ccc(CN4CCN(CC5(COc6nc(N7CC8CCC(C7)N8)c7cnc(-c8cc(O)cc9ccccc89)c(F)c7n6)CC5)CC4)cc3C2=O)C(=O)N1	C46H46FN9O6	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-29YCMF	WO2024233838A1_12	.	O=C1CCC(N2C(=O)c3cccc(N4CCC(CN5CCN(CC6(COc7nc(N8CC9CCC(C8)N9)c8cnc(-c9cc(O)cc%10ccccc9%10)c(F)c8n7)CC6)CC5)CC4)c3C2=O)C(=O)N1	C51H55FN10O6	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-1IOKKZ	WO2024233838A1_13	.	O=C1CCC(N2Cc3cc(N4CCC(C(=O)N5CCN(CC6(COc7nc(N8CC9CCC(C8)N9)c8cnc(-c9cc(O)cc%10ccccc9%10)c(F)c8n7)CC6)CC5)CC4)ccc3C2=O)C(=O)N1	C51H55FN10O6	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-TFS64Z	WO2024233838A1_14	.	CN1C[C@H](N2CCN(C(=O)C3CCN(c4ccc5c(c4)CN(C4CCC(=O)NC4=O)C5=O)CC3)CC2)C[C@@H]1COc1nc(N2CC3CCC(C2)N3)c2cnc(-c3cc(O)cc4ccccc34)c(F)c2n1	C52H58FN11O6	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-9ZE1Z3	WO2024233838A1_16	.	CN1C[C@H](N2CCC(C(=O)N3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)C[C@@H]1COc1nc(N2CC3CCC(C2)N3)c2cnc(-c3cc(O)cc4ccccc34)c(F)c2n1	C52H56FN11O7	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-HF37JS	WO2024233838A1_17	.	O=C1CCC(N2C(=O)c3ccc(N4CCC(CN5CCN(CC6(COc7nc(N8CC9CCC(C8)N9)c8cnc(-c9cc(O)cc%10ccccc9%10)c(F)c8n7)CC6)CC5)CC4)cc3C2=O)C(=O)N1	C51H55FN10O6	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-UR682Q	WO2024233838A1_18	.	C#Cc1cccc2cccc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C53H55FN10O5	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-XUKCHJ	WO2024233838A1_19	.	CN1C[C@H](N2CCC(C(=O)Nc3ccc4c(c3)CN(C3CCC(=O)NC3=O)C4=O)CC2)C[C@@H]1COc1nc(N2CC3CCC(C2)N3)c2cnc(-c3cccc4cccc(Cl)c34)c(F)c2n1	C48H50ClFN10O5	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-LWKZJX	WO2024233838A1_20	.	O=C1CCC(N2C(=O)c3ccc(CN4CCN([C@H]5CN6CCC[C@@]6(COc6nc(N7CC8CCC(C7)N8)c7cnc(-c8cc(O)cc9ccccc89)c(F)c7n6)C5)CC4)cc3C2=O)C(=O)N1	C49H51FN10O6	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-R3ABPC	WO2024233838A1_21	.	C#Cc1cccc2cccc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCN(C(=O)C7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C53H55FN10O5	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-YPE1RY	WO2024233838A1_23	.	CN1C[C@H](N2CCC(C(=O)NCCOc3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)C[C@@H]1COc1nc(N2CC3CCC(C2)N3)c2cnc(-c3cc(O)cc4ccccc34)c(F)c2n1	C50H53FN10O8	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-4SVV1T	WO2024233838A1_24	.	CN1C[C@H](N2CCC(C(=O)NCCOCCOc3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)C[C@@H]1COc1nc(N2CC3CCC(C2)N3)c2cnc(-c3cc(O)cc4ccccc34)c(F)c2n1	C52H57FN10O9	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-ELODRZ	WO2024233838A1_25	.	C#Cc1cccc2cccc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC[C@H]5CC[C@@H](CN6CCN(CC7CCN(c8cc9c(cc8F)C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)CC6)N5C)nc4c3F)c12	C55H59F2N11O5	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-PKDI3W	WO2024233838A1_26	.	C#Cc1cccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C53H55FN10O6	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-01E67F	WO2024233838A1_27	.	C#Cc1cccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C53H57FN10O5	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-067XGI	WO2024233838A1_28	5-[4-[[4-[[1-[[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-8-fluoro-7-(8-methylnaphthalen-1-yl)pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperazin-1-yl]methyl]piperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	Cc1cccc2cccc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C52H57FN10O5	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-E2X3VB	SCHEMBL26508548	5-[4-[[4-[[1-[[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperazin-1-yl]methyl]piperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C53H54F2N10O6	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-S9OZN0	WO2024233838A1_30	.	CN1[C@@H](COc2nc(N3CC4CCC(C3)N4)c3cnc(-c4cc(O)cc5ccccc45)c(F)c3n2)CC[C@H]1CN1CCN(CC2CCN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)CC1	C53H60FN11O6	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-X757PQ	WO2024233838A1_31	3-[6-[[4-[[1-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperazin-1-yl]methyl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#Cc1cccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCN(Cc7ccc8c(c7)CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)nc4c3F)c12	C48H48FN9O5	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-6PETRC	WO2024233838A1_32	.	C#Cc1cccc2cccc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC[C@H]5CC[C@@H](CN6CCN(CCC7CCN(c8ccc9c(c8)C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)CC6)N5)nc4c3F)c12	C55H60FN11O5	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-5S8GPQ	WO2024233838A1_33	.	Cc1cccc(-c2ncc3c(N4CC5CCC(C4)N5)nc(OCC4(CN5CCN(CC6CCN(c7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)CC4)nc3c2F)c1C	C49H57FN10O5	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-ICIEL8	WO2024233838A1_34	5-[[4-[[1-[[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperazin-1-yl]methyl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCN(Cc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)nc4c3F)c12	C48H45F2N9O6	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-6FSKTW	WO2024233838A1_35	5-[[4-[[1-[[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperazin-1-yl]methyl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	C#Cc1cccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCN(Cc7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)nc4c3F)c12	C48H46FN9O6	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-R71868	WO2024233838A1_36	.	COc1nc(-c2cc(O)cc3ccccc23)c(F)c2nc(OCC3(CN4CCN(CC5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)CC4)CC3)nc(N3CC4CCC(C3)N4)c12	C52H57FN10O7	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-FRTKUD	WO2024233838A1_37	5-[4-[[[1-[[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynylnaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl-methylamino]methyl]piperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	C#Cc1cccc2cccc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)CC6CCN(c7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)nc4c3F)c12	C50H50FN9O5	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-AADH7A	WO2024233838A1_38	.	C#Cc1cccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC[C@H]5CC[C@@H](CN6CCN(CC7CCN(c8ccc9c(c8)C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)CC6)N5C)nc4c3F)c12	C55H60FN11O6	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-FU3OSA	WO2024233838A1_39	.	C#Cc1cccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC[C@H]5CC[C@@H](CN6CCN(CC7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)N5)nc4c3F)c12	C54H60FN11O5	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-HEOCYU	WO2024233838A1_40	.	O=C1CCC(N2Cc3cc(N4CCC(CN5CCN(CC6(COc7nc(N8CC9CCC(C8)N9)c8cnc(-c9cc(O)cc%10ccccc9%10)c(F)c8n7)CC6)CC5)CC4)ccc3C2=O)C(=O)N1	C51H57FN10O5	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-8LKJXS	WO2024233838A1_41	.	C#Cc1cccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)CN(C8CCC(=O)N(C)C8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C54H59FN10O5	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-C31VQV	WO2024233838A1_42	.	C#Cc1cccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)C(=O)N(C8CCC(=O)N(C)C8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C54H57FN10O6	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-E6B6YH	WO2024233838A1_43	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C53H56F2N10O5	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-JTPEUH	WO2024233838A1_44	5-[4-[2-[4-[(3R,5R)-5-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynylnaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1-methylpyrrolidin-3-yl]piperazin-1-yl]ethyl]piperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	C#Cc1cccc2cccc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC[C@H]5C[C@@H](N6CCN(CCC7CCN(c8ccc9c(c8)C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CN5C)nc4c3F)c12	C55H60FN11O5	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-D0ALGZ	WO2024233838A1_45	.	CN(CC1CCN(c2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)CC1)CC1(COc2nc(N3CC4CCC(C3)N4)c3cnc(-c4cc(O)cc5ccccc45)c(F)c3n2)CC1	C48H50FN9O6	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-3MGHU9	WO2024233838A1_46	.	O=C1CCC(N2C(=O)c3ccc(N4CCN(C(=O)C5CCN(CC6(COc7nc(N8CC9CCC(C8)N9)c8cnc(-c9cc(O)cc%10ccccc9%10)c(F)c8n7)CC6)CC5)CC4)cc3C2=O)C(=O)N1	C51H53FN10O7	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-LTNOLZ	SCHEMBL25446466	5-[[4-[[4-[(3R,5R)-5-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynylnaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1-methylpyrrolidin-3-yl]piperazin-1-yl]methyl]cyclohexyl]amino]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	C#Cc1cccc2cccc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC[C@H]5C[C@@H](N6CCN(C[C@H]7CC[C@H](Nc8ccc9c(c8)C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CN5C)nc4c3F)c12	C55H60FN11O5	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-FWIBTM	WO2024233838A1_48	.	C#Cc1cccc2cc(O)cc(-c3nc(OC)c4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C54H59FN10O6	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-ZU03GE	WO2024233838A1_49	5-[[4-[[4-[[(2S,5R)-5-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynylnaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1-methylpyrrolidin-2-yl]methyl]piperazin-1-yl]methyl]cyclohexyl]amino]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	C#Cc1cccc2cccc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OC[C@H]5CC[C@@H](CN6CCN(CC7CCC(Nc8ccc9c(c8)C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)CC6)N5C)nc4c3F)c12	C56H62FN11O5	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-GNH771	WO2024233838A1_50	.	O=C1CCC(N2Cc3cc(N4CCN(CC5(COc6nc(N7CC8CCC(C7)N8)c7cnc(-c8cccc9cccc(Cl)c89)c(F)c7n6)CC5)CC4)ccc3C2=O)C(=O)N1	C45H45ClFN9O4	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-8K0O8T	WO2024233838A1_51	.	C#Cc1cccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)CN(C)C9=O)CC7)CC6)CC5)nc4c3F)c12	C49H54FN9O3	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-AI4FTL	WO2024233838A1_52	.	C#Cc1cccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCN(CC7CCN(CC(=O)N[C@@H](C(=O)N8C[C@@H](O)C[C@@H]8C(=O)NCc8ccc(-c9scnc9C)cc8)C(C)(C)C)CC7)CC6)CC5)nc4c3F)c12	C64H77FN12O6S	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-PQVQUK	WO2024233838A1_53	.	C#Cc1cccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCN(CC7CCN(CCC(=O)N[C@@H](C(=O)N8C[C@@H](O)C[C@@H]8C(=O)NCc8ccc(-c9scnc9C)cc8)C(C)(C)C)CC7)CC6)CC5)nc4c3F)c12	C65H79FN12O6S	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-GQ7KAX	WO2024233838A1_54	3-[6-[4-[[[1-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl-methylamino]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#Cc1cccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)CC6CCN(c7ccc8c(c7)CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)nc4c3F)c12	C50H52FN9O5	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-ZB5KH5	WO2024233838A1_55	.	C#Cc1cccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(C(=O)N7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C53H55FN10O6	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-QD40BT	WO2024233838A1_56	.	C#Cc1cccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)C(=O)N(C8CCC(=O)NC8=O)C9)CC7)CC6)CC5)nc4c3F)c12	C53H57FN10O5	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-VGPZLG	WO2024233838A1_57	3-[6-[4-[[4-[[1-[[7-(8-ethynyl-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[8-(2,2,2-trifluoroacetyl)-3,8-diazabicyclo[3.2.1]octan-3-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperazin-1-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#Cc1cccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6C(=O)C(F)(F)F)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C55H56F4N10O6	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-DO0EES	WO2024233838A1_58	.	C#Cc1cccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCN(C(=O)N7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C52H54FN11O6	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-UPWG1L	WO2024233838A1_59	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)CC6CCN(c7ccc8c(c7)C(=O)N(C7CCC(=O)NC7=O)C8)CC6)CC5)nc4c3F)c12	C50H51F2N9O5	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-E4TTF8	WO2024233838A1_60	.	C#Cc1cccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCN(CC7CCN(c8cc9c(cc8F)C(=O)N(C8CCC(=O)NC8=O)C9)CC7)CC6)CC5)nc4c3F)c12	C53H56F2N10O5	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-T6TCFY	SCHEMBL25446523	3-[6-[4-[[4-[[1-[[7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-(8-propanoyl-3,8-diazabicyclo[3.2.1]octan-3-yl)pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperazin-1-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6C(=O)CC)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C56H60F2N10O6	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-0D03HI	WO2024233838A1_62	.	C#Cc1c(F)ccc2cc(O)cc(-c3nc(OC)c4c(N5CCN(C(=O)CC)[C@H](CC#N)C5)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C57H61F2N11O7	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-V7I2WM	WO2024233838A1_63	.	C#Cc1c(F)ccc2cc(O)cc(-c3nc(OC)c4c(N5CC6CCC(C5)N6C(=O)C(F)(F)F)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C56H57F5N10O7	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-K56VML	WO2024233838A1_64	.	C#Cc1cccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)n(C)c(=O)n9C8CCC(=O)NC8=O)CC7)CC6)CC5)nc4c3F)c12	C53H58FN11O5	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-6OJA3R	WO2024233838A1_65	3-[4-[4-[[4-[[1-[[4-(3,8-Diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperazin-1-yl]methyl]piperidin-1-yl]anilino]piperidine-2,6-dione	C#Cc1cccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCN(CC7CCN(c8ccc(NC9CCC(=O)NC9=O)cc8)CC7)CC6)CC5)nc4c3F)c12	C51H57FN10O4	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-9FS2K7	WO2024233838A1_66	.	C#Cc1cccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)[C@@H](C7CC7)C6)CC5)nc4c3F)c12	C56H61FN10O5	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-EONF1Z	WO2024233838A1_67	2-[(2S)-4-[2-[[1-[[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]methyl]cyclopropyl]methoxy]-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-4-yl]-1-propanoylpiperazin-2-yl]acetonitrile	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCN(C(=O)CC)[C@@H](CC#N)C5)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C56H59F2N11O6	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-ROJWC3	WO2024233838A1_68	.	CCC(=O)N1CCN(c2nc(OCC3(CN4CCN(CC5CCN(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC5)CC4)CC3)nc3c2CCN(c2cccc4cccc(Cl)c24)C3)C[C@@H]1CC#N	C54H64ClN11O5	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-CB461N	WO2024233838A1_69	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(CN7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C53H56F2N10O5	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-OMKS0Z	WO2024233838A1_70	3-[6-[4-[[4-[[1-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-5-methoxypyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperazin-1-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#Cc1c(F)ccc2cc(O)cc(-c3nc(OC)c4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C54H58F2N10O6	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-6RLL4D	WO2024233838A1_71	.	C#Cc1c(F)ccc2cc(O)cc(-c3nc(O)c4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C53H56F2N10O6	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-O9G3ZB	WO2024233838A1_72	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(C7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C53H55F2N9O5	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-7KZ6LE	WO2024233838A1_73	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCN(CC7CN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)C7)CC6)CC5)nc4c3F)c12	C51H52F2N10O5	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-AKAEQ5	WO2024233838A1_74	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCN(C7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C52H54F2N10O5	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-KVC78Q	WO2024233838A1_75	.	C#Cc1cccc2cc(O)cc(-c3nc(O)c4c(N5CC6CCC(C5)N6C)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C54H59FN10O6	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-V92LVW	WO2024233838A1_76	2-[(2S)-4-[2-[[1-[[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]methyl]cyclopropyl]methoxy]-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-5-methoxypyrido[4,3-d]pyrimidin-4-yl]-1-methylpiperazin-2-yl]acetonitrile	C#Cc1c(F)ccc2cc(O)cc(-c3nc(OC)c4c(N5CCN(C)[C@@H](CC#N)C5)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C55H59F2N11O6	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-Q0GL7U	WO2024233838A1_77	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(N7CCC(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C53H55F2N9O5	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-PPJMKT	WO2024233838A1_78	3-[6-[4-[[4-[[1-[[7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[8-(2,2,2-trifluoroacetyl)-3,8-diazabicyclo[3.2.1]octan-3-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperazin-1-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6C(=O)C(F)(F)F)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C55H55F5N10O6	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-EYU3NW	WO2024233838A1_79	2-[(2S)-4-[2-[[1-[[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]methyl]cyclopropyl]methoxy]-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-4-yl]-1-prop-2-enoylpiperazin-2-yl]acetonitrile	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCN(C(=O)C=C)[C@@H](CC#N)C5)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C56H57F2N11O6	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-143S15	SCHEMBL25446641	3-[3-[2-[[1-[[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]methyl]cyclopropyl]methoxy]-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]-3-oxopropanenitrile	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6C(=O)CC#N)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C56H57F2N11O6	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-HEM71P	SCHEMBL26509200	3-[6-[1-[[1-[[1-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]methyl]piperidin-4-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(CN7CCC(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C54H57F2N9O5	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-R97O5I	WO2024233838A1_82	.	C#Cc1c(F)ccc2cc(O)cc(-c3nc(OC)c4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCN(C7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8)C9=O)CC7)CC6)CC5)nc4c3F)c12	C53H58F2N10O5	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-Q0RUTT	WO2024233838A1_83	.	C#Cc1c(F)ccc2cc(O)cc(C3=NCC4C(N5CC6CCC(C5)N6)=NC(OCC5(CN6CCC(CN7CCC(c8ccc(NC9CCC(=O)NC9=O)cc8)CC7)CC6)CC5)=NC4=C3F)c12	C52H59F2N9O4	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-SUMKXT	WO2024233838A1_84	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC7(CC6)CCN(c6ccc8c(c6)CN(C6CCC(=O)NC6=O)C8=O)CC7)CC5)nc4c3F)c12	C52H53F2N9O5	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-SRTH7F	WO2024233838A1_85	.	C#Cc1c(F)ccc2cc(O)cc(-c3nc(OC)c4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCN(C7CCN(c8ccc9c(c8)C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C53H54F2N10O7	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-E0ZKZ8	WO2024233838A1_86	3-[6-[7-[[1-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]-2,7-diazaspiro[3.5]nonan-2-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC7(CC6)CN(c6ccc8c(c6)CN(C6CCC(=O)NC6=O)C8=O)C7)CC5)nc4c3F)c12	C50H49F2N9O5	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-OS566G	WO2024233838A1_87	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CC7(C6)CN(c6ccc8c(c6)CN(C6CCC(=O)NC6=O)C8=O)C7)CC5)nc4c3F)c12	C48H45F2N9O5	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-Z06K1K	WO2024233838A1_88	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(=O)n(C%10CCC(=O)NC%10=O)ncc9c8)CC7)CC6)CC5)nc4c3F)c12	C53H55F2N11O5	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-QTS3OL	WO2024233838A1_89	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCN(CC#Cc7ccc8c(c7)CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)nc4c3F)c12	C50H47F2N9O5	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-7XE4D9	WO2024233838A1_90	3-[6-[2-[1-[[1-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]azetidin-3-yl]ethynyl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CC(C#Cc7ccc8c(c7)CN(C7CCC(=O)NC7=O)C8=O)C6)CC5)nc4c3F)c12	C48H42F2N8O5	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-E7KXII	WO2024233838A1_91	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(C#Cc7ccc8c(c7)CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)nc4c3F)c12	C50H46F2N8O5	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-H1HNXF	WO2024233838A1_92	3-[6-[3-[4-[[[1-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl-methylamino]methyl]phenyl]azetidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN(C)Cc6ccc(C7CN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)C7)cc6)CC5)nc4c3F)c12	C54H51F2N9O5	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-15O6M1	WO2024233838A1_93	3-[6-[1-[[1-[[1-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]methyl]-3,3-difluoropiperidin-4-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6)nc(OCC5(CN6CCC(CN7CCC(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)C(F)(F)C7)CC6)CC5)nc4c3F)c12	C54H55F4N9O5	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-XZ9YIO	WO2024233838A1_100	2-[3-[2-[[1-[[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]methyl]cyclopropyl]methoxy]-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-5-methoxypyrido[4,3-d]pyrimidin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]acetonitrile	C#Cc1c(F)ccc2cc(O)cc(-c3nc(OC)c4c(N5CC6CCC(C5)N6CC#N)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C56H59F2N11O6	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-BHBZM0	WO2024233838A1_101	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6CC#N)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C55H57F2N11O5	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-3F1Y8E	WO2024233838A1_102	3-[3-[2-[[1-[[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]methyl]cyclopropyl]methoxy]-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-5-methoxypyrido[4,3-d]pyrimidin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]-3-oxopropanenitrile	C#Cc1c(F)ccc2cc(O)cc(-c3nc(OC)c4c(N5CC6CCC(C5)N6C(=O)CC#N)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C57H59F2N11O7	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-6TNDVR	SCHEMBL31158010	3-[(2S)-2-(cyanomethyl)-4-[2-[[1-[[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]methyl]cyclopropyl]methoxy]-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-4-yl]piperazin-1-yl]-3-oxopropanenitrile	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCN(C(=O)CC#N)[C@@H](CC#N)C5)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C56H56F2N12O6	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-EEP9N5	WO2024233838A1_104	.	C#Cc1c(F)ccc2cc(O)cc(-c3nc(OC)c4c(N5CCN(C(=O)CC#N)[C@@H](CC#N)C5)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C57H58F2N12O7	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-9UR93T	WO2024233838A1_105	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCN(C(=O)C(=C)F)[C@@H](CC#N)C5)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C56H56F3N11O6	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-XGMA8X	WO2024233838A1_106	3-[3-[2-[[1-[[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]methyl]cyclopropyl]methoxy]-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]-2,2-dimethyl-3-oxopropanenitrile	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6C(=O)C(C)(C)C#N)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C58H61F2N11O6	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-9VUA4L	WO2024233838A1_107	1-[3-[2-[[1-[[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]methyl]cyclopropyl]methoxy]-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-4-yl]-3,8-diazabicyclo[3.2.1]octane-8-carbonyl]cyclopropane-1-carbonitrile	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6C(=O)C5(C#N)CC5)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C58H59F2N11O6	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-309T50	WO2024233838A1_108	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6C(=O)C(C)C#N)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C57H59F2N11O6	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-P8JCQ3	WO2024233838A1_109	(2S)-3-[3-[2-[[1-[[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]methyl]cyclopropyl]methoxy]-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]-2-methyl-3-oxopropanenitrile	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6C(=O)[C@@H](C)C#N)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C57H59F2N11O6	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-4P1XRB	WO2024233838A1_110	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6C(=O)[C@H](C)C#N)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C57H59F2N11O6	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-MD8Y7Q	WO2024233838A1_111	.	C#Cc1c(F)ccc2cc(O)cc(-c3nc(OC)c4c(N5CC6CCC(C5)N6C(=O)C(C)C#N)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C58H61F2N11O7	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-6U8S7Q	WO2024233838A1_112	.	C#Cc1c(F)ccc2cc(O)cc(-c3nc(OC)c4c(N5CC6CCC(C5)N6C(=O)C(C#N)CC)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C59H63F2N11O7	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-TULPPV	WO2024233838A1_113	.	C#Cc1c(F)ccc2cc(O)cc(-c3nc(OC)c4c(N5CC6CCC(C5)N6C(=O)CC#N)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)n(C)c(=O)n9C8CCC(=O)NC8=O)CC7)CC6)CC5)nc4c3F)c12	C57H60F2N12O7	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-M66T4O	WO2024233838A1_116	.	C#Cc1c(F)ccc2cc(O)cc(-c3nc(OC)c4c(N5CC6CCC(C5)N6C(=O)C(C)CC#N)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C59H63F2N11O7	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-XQJK4T	WO2024233838A1_117	4-[3-[2-[[1-[[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]methyl]cyclopropyl]methoxy]-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-5-methoxypyrido[4,3-d]pyrimidin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]-4-oxobutanenitrile	C#Cc1c(F)ccc2cc(O)cc(-c3nc(OC)c4c(N5CC6CCC(C5)N6C(=O)CCC#N)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C58H61F2N11O7	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-5QTHZJ	WO2024233838A1_118	N-tert-butyl-3-[2-[[1-[[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]methyl]cyclopropyl]methoxy]-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-4-yl]-3,8-diazabicyclo[3.2.1]octane-8-carboxamide	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6C(=O)NC(C)(C)C)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C58H65F2N11O6	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-JNRMOJ	WO2024233838A1_120	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6C(=O)CC(F)(F)F)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C56H57F5N10O6	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-SQB1UT	WO2024233838A1_122	N-(cyanomethyl)-3-[2-[[1-[[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]methyl]cyclopropyl]methoxy]-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-5-methoxypyrido[4,3-d]pyrimidin-4-yl]-3,8-diazabicyclo[3.2.1]octane-8-carboxamide	C#Cc1c(F)ccc2cc(O)cc(-c3nc(OC)c4c(N5CC6CCC(C5)N6C(=O)NCC#N)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C57H60F2N12O7	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-CW46OG	WO2024233838A1_123	3-[2-[[1-[[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]methyl]cyclopropyl]methoxy]-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-5-methoxypyrido[4,3-d]pyrimidin-4-yl]-N-(2,2,2-trifluoroethyl)-3,8-diazabicyclo[3.2.1]octane-8-carboxamide	C#Cc1c(F)ccc2cc(O)cc(-c3nc(OC)c4c(N5CC6CCC(C5)N6C(=O)NCC(F)(F)F)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C57H60F5N11O7	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-3S8EB5	WO2024233838A1_124	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6C(=O)/C(C#N)=C/C5CC5)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C60H61F2N11O6	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-04W7FD	WO2024233838A1_125	.	C#Cc1c(F)ccc2cc(O)cc(-c3nc(OC)c4c(N5CCN(C(=O)C=C)[C@@H](CC#N)C5)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C57H59F2N11O7	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-0XGTYQ	WO2024233838A1_126	2-[3-[2-[[1-[[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]methyl]cyclopropyl]methoxy]-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-5-methoxypyrido[4,3-d]pyrimidin-4-yl]-3,8-diazabicyclo[3.2.1]octane-8-carbonyl]butanedinitrile	C#Cc1c(F)ccc2cc(O)cc(-c3nc(OC)c4c(N5CC6CCC(C5)N6C(=O)C(C#N)CC#N)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C59H60F2N12O7	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-XNFMR6	WO2024233838A1_127	3-[6-[4-[[4-[[1-[[7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-5-methoxy-4-(1,4-oxazepan-4-yl)pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperazin-1-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#Cc1c(F)ccc2cc(O)cc(-c3nc(OC)c4c(N5CCCOCC5)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C53H57F2N9O7	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-U65B4Y	WO2024233838A1_128	N-cyclobutyl-3-[2-[[1-[[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]methyl]cyclopropyl]methoxy]-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-4-yl]-3,8-diazabicyclo[3.2.1]octane-8-carboxamide	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6C(=O)NC5CCC5)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C58H63F2N11O6	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-BISUF9	WO2024233838A1_129	4-[3-[2-[[1-[[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]methyl]cyclopropyl]methoxy]-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]-2-methyl-4-oxobutanenitrile	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6C(=O)CC(C)C#N)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C58H61F2N11O6	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-S5HUN3	WO2024233838A1_130	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6C(=O)CC(C)C#N)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)CN(C8CCC(=O)N(C)C8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C59H63F2N11O6	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-Y9MZG6	WO2024233838A1_131	4-[3-[2-[[1-[[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]methyl]cyclopropyl]methoxy]-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]-2,2-dimethyl-4-oxobutanenitrile	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6C(=O)CC(C)(C)C#N)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C59H63F2N11O6	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-YOYH0Y	WO2024233838A1_132	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6C(=O)CC(C)C#N)nc(OCC5(CN(C)Cc6ccc(C7CN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)C7)cc6)CC5)nc4c3F)c12	C59H56F2N10O6	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-OVMBXF	WO2024233838A1_133	4-[3-[2-[[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperidin-3-yl]methoxy]-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]-2-methyl-4-oxobutanenitrile	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6C(=O)CC(C)C#N)nc(OCC5CCCN(CC6CCN(c7ccc8c(c7)CN(C7CCC(=O)NC7=O)C8=O)CC6)C5)nc4c3F)c12	C55H56F2N10O6	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-29OJEN	WO2024233838A1_134	.	C#CC1c2c(cc(O)cc2-c2ncc3c(N4CCCOCC4)nc(OCC4(CN5CCN(CC6CCN(c7ccc8c(c7)CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)CC4)nc3c2F)C=CC1F	C52H57F2N9O6	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-WAC9PG	WO2024233838A1_135	4-[3-[2-[[1-[[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]methyl]cyclopropyl]methoxy]-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-5-methoxypyrido[4,3-d]pyrimidin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]-2-methyl-4-oxobutanenitrile	C#Cc1c(F)ccc2cc(O)cc(-c3nc(OC)c4c(N5CC6CCC(C5)N6C(=O)CC(C)C#N)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C59H63F2N11O7	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-MR4YN0	WO2024233838A1_136	4-[3-[2-[[1-[[4-[[1-[1-(2,6-Dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]methyl]cyclopropyl]methoxy]-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]-2-methyl-4-oxobutanenitrile	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6C(=O)CC(C)C#N)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)n(C)c(=O)n9C8CCC(=O)NC8=O)CC7)CC6)CC5)nc4c3F)c12	C58H62F2N12O6	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-CTW6A8	WO2024233838A1_137	4-[3-[2-[[1-[[4-[[1-[4-[(2,6-Dioxopiperidin-3-yl)amino]-2-fluorophenyl]piperidin-4-yl]methyl]piperazin-1-yl]methyl]cyclopropyl]methoxy]-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]-2-methyl-4-oxobutanenitrile	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6C(=O)CC(C)C#N)nc(OCC5(CN6CCN(CC7CCN(c8ccc(NC9CCC(=O)NC9=O)cc8F)CC7)CC6)CC5)nc4c3F)c12	C56H60F3N11O5	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-HMZ9PN	WO2024233838A1_139	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CCCOC6CC65)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C53H55F2N9O6	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-JJYI92	WO2024233838A1_140	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6C(=O)CC(C)C#N)nc(OCC5(CN6CC7CC7C6)CC5)nc4c3OCc3ccc(-c4cn([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](CO)c5ccc(-c6ccnn6CC)cc5)C(C)C)nn4)cc3)c12	C72H77FN14O8	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-1WFLW8	WO2024233838A1_141	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6C(=O)Cn5cc(COCCOCCOCCNc6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)nn5)nc(OCC56CCCN5C[C@@H](F)C6)nc4c3F)c12	C57H59F3N12O9	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-LY8IBF	WO2024233838A1_142	.	C#Cc1c(F)ccc2cc(O)cc(-c3nc(OC)c4c(N5CC6CCC(C5)N6C(=O)CC(C)C#N)nc(OCC5(CN6CCN(CC7CCN(c8cccc(NC9CCC(=O)NC9=O)c8)CC7)CC6)CC5)nc4c3F)c12	C57H63F2N11O6	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-UTL4FX	WO2024233838A1_143	.	C#Cc1c(F)ccc2cc(O)cc(-c3nc(OC)c4c(N5CC6CCC(C5)N6C(=O)C[C@@H](C)C#N)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C59H63F2N11O7	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-DC1ARU	WO2024233838A1_144	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6C(=O)CC(C)C#N)nc(OCC5(CN6CC(OC7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)C6)CC5)nc4c3F)c12	C56H56F2N10O7	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-S9MIKG	WO2024233838A1_145	4-[3-[2-[[1-[[(2,6-Dioxopiperidin-3-yl)amino]methyl]cyclopropyl]methoxy]-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-5-methoxypyrido[4,3-d]pyrimidin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]-2-methyl-4-oxobutanenitrile	C#Cc1c(F)ccc2cc(O)cc(-c3nc(OC)c4c(N5CC6CCC(C5)N6C(=O)CC(C)C#N)nc(OCC5(CNC6CCC(=O)NC6=O)CC5)nc4c3F)c12	C41H40F2N8O6	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-TUMITX	WO2024233838A1_146	.	C#Cc1c(F)ccc2cc(O)cc(-c3nc(OC)c4c(N5CC6CCC(C5)N6C(=O)CC(C)C#N)nc(OCC5CCCN(CC6CCN(c7ccc8c(c7)CN(C7CCC(=O)NC7=O)C8=O)CC6)C5)nc4c3F)c12	C56H58F2N10O7	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-8CXGTH	WO2024233838A1_147	4-[3-[2-[[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperidin-3-yl]methoxy]-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-5-methoxypyrido[4,3-d]pyrimidin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]-4-oxobutanenitrile	C#Cc1c(F)ccc2cc(O)cc(-c3nc(OC)c4c(N5CC6CCC(C5)N6C(=O)CCC#N)nc(OCC5CCCN(CC6CCN(c7ccc8c(c7)CN(C7CCC(=O)NC7=O)C8=O)CC6)C5)nc4c3F)c12	C55H56F2N10O7	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-Y4S058	WO2024233838A1_148	.	C#Cc1c(F)ccc2cc(O)cc(-c3ncc4c(N5CC6CCC(C5)N6C(=O)CC(C)C#N)nc(OCC5(CN6CCN(CCOCCC(=O)N[C@@H](C(=O)N7C[C@@H](O)C[C@@H]7C(=O)N[C@H](CO)c7ccc(-c8ccnn8CC)cc7)C(C)C)CC6)CC5)nc4c3C)c12	C68H82FN13O9	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-HXBP2L	WO2024233838A1_149	.	C#Cc1c(F)ccc2cc(O)cc(-c3nc(OC)c4c(N5CC6CCC(C5)N6C(=O)CC(C)C#N)nc(OCc5cn(-c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)nn5)nc4c3F)c12	C47H39F2N11O7	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-CK1WQM	WO2024233838A1_150	.	C#Cc1c(F)ccc2cc(O)cc(-c3nc(OC(F)(F)F)c4c(N5CC6CCC(C5)N6C(=O)CC(C)C#N)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C59H60F5N11O7	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-333E8M	WO2024233838A1_151	.	C#Cc1c(F)ccc2cc(O)cc(-c3nc(OC(F)(F)F)c4c(N5CC6CCC(C5)N6C(=O)CCC#N)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C58H58F5N11O7	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-1U4LSP	WO2024233838A1_152	4-[3-[2-[[1-[[4-[[1-[3-(2,4-Dioxo-1,3-diazinan-1-yl)-1-methylindazol-6-yl]piperidin-4-yl]methyl]piperazin-1-yl]methyl]cyclopropyl]methoxy]-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-5-methoxypyrido[4,3-d]pyrimidin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]-2-methyl-4-oxobutanenitrile	C#Cc1c(F)ccc2cc(O)cc(-c3nc(OC)c4c(N5CC6CCC(C5)N6C(=O)CC(C)C#N)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(N%10CCC(=O)NC%10=O)nn(C)c9c8)CC7)CC6)CC5)nc4c3F)c12	C58H63F2N13O6	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-D9QL1O	WO2024233838A1_153	4-[3-[7-[5-amino-3-chloro-2-(trifluoromethyl)phenyl]-6-chloro-2-[[1-[[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]methyl]cyclopropyl]methoxy]-8-fluoroquinazolin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]-4-oxobutanenitrile	N#CCCC(=O)N1C2CCC1CN(c1nc(OCC3(CN4CCN(CC5CCN(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC5)CC4)CC3)nc3c(F)c(-c4cc(N)cc(Cl)c4C(F)(F)F)c(Cl)cc13)C2	C53H57Cl2F4N11O5	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-1DHMSR	WO2024233838A1_154	.	C#Cc1c(F)ccc2cc(O)cc(-c3nc(OC)c4c(N5CC6CCC(C5)N6C(=O)CC(C)C#N)nc(OCC5(CN6CCN(C[C@H]7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)C[C@@H]7F)CC6)CC5)nc4c3F)c12	C59H62F3N11O7	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-UCEOH7	WO2024233838A1_155	3-[6-[4-[[4-[[1-[[7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[8-(3-fluorobicyclo[1.1.1]pentane-1-carbonyl)-3,8-diazabicyclo[3.2.1]octan-3-yl]-5-methoxypyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperazin-1-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#Cc1c(F)ccc2cc(O)cc(-c3nc(OC)c4c(N5CC6CCC(C5)N6C(=O)C56CC(F)(C5)C6)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C60H63F3N10O7	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-WWGP7Z	WO2024233838A1_156	2'-amino-3-[4-chloro-6-[[1-[[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperazin-1-yl]methyl]cyclopropyl]methoxy]pyrimidin-2-yl]spiro[5,6-dihydro-4H-1,2-benzoxazole-7,4'-6,7-dihydro-5H-1-benzothiophene]-3'-carbonitrile	N#Cc1c(N)sc2c1C1(CCC2)CCCc2c(-c3nc(Cl)cc(OCC4(CN5CCN(CC6CCN(c7ccc8c(c7)CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)CC4)n3)noc21	C47H53ClN10O5S	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-PT2RDC	WO2024233838A1_157	3-[6-[4-[[4-[[1-[[7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-5-methoxy-4-(2-oxa-6-azabicyclo[5.1.0]octan-6-yl)pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperazin-1-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#Cc1c(F)ccc2cc(O)cc(-c3nc(OC)c4c(N5CCCOC6CC65)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C54H57F2N9O7	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-3XXJNZ	WO2024233838A1_158	.	C#Cc1c(F)ccc2cc(O)cc(-c3nc4c5c(nc(OCC6(CN7CCN(CC8CCN(c9ccc%10c(c9)CN(C9CCC(=O)NC9=O)C%10=O)CC8)CC7)CC6)nc5c3F)N(CC(F)F)[C@@H](C)CO4)c12	C52H53F4N9O6	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-H0S66F	WO2024233838A1_159	4-[3-[2-[[1-[[4-[[1-[3-(2,4-Dioxo-1,3-diazinan-1-yl)-1-methylindazol-6-yl]piperidin-4-yl]methyl]piperazin-1-yl]methyl]cyclopropyl]methoxy]-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-5-methoxypyrido[4,3-d]pyrimidin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]-4-oxobutanenitrile	C#Cc1c(F)ccc2cc(O)cc(-c3nc(OC)c4c(N5CC6CCC(C5)N6C(=O)CCC#N)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(N%10CCC(=O)NC%10=O)nn(C)c9c8)CC7)CC6)CC5)nc4c3F)c12	C57H61F2N13O6	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-0MXKYW	WO2024233838A1_160	.	C#Cc1c(F)ccc2cc(O)cc(-c3nc(OC)c4c(N5CC6CCC(C5)N6C(=O)C[C@@H](C)C#N)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(N%10CCC(=O)NC%10=O)nn(C)c9c8)CC7)CC6)CC5)nc4c3F)c12	C58H63F2N13O6	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-Q5E2RA	WO2024233838A1_161	4-[3-[2-[[1-[[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]-3,3-difluoropiperidin-1-yl]methyl]piperidin-1-yl]methyl]cyclopropyl]methoxy]-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-5-methoxypyrido[4,3-d]pyrimidin-4-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]-2-methyl-4-oxobutanenitrile	C#Cc1c(F)ccc2cc(O)cc(-c3nc(OC)c4c(N5CC6CCC(C5)N6C(=O)CC(C)C#N)nc(OCC5(CN6CCC(CN7CCC(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)C(F)(F)C7)CC6)CC5)nc4c3F)c12	C60H62F4N10O7	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-PKL59W	WO2024233838A1_162	.	C#Cc1c(F)ccc2cc(O)cc(-c3nc(OC)c4c(N5CC6CCC(C5)N6C(=O)C[C@@H](C)C#N)nc(OCC5(CN6CCC(CN7CCC(N8Cc9cc%10c(cc9C8)C(=O)N(C8CCC(=O)NC8=O)C%10)CC7)CC6)CC5)nc4c3F)c12	C62H67F2N11O7	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-43SVL5	WO2024233838A1_163	.	C#Cc1c(F)ccc2cc(O)cc(-c3nc(OC)c4c(N5CC6CCC(C5)N6C(=O)CCC#N)nc(OCC5(CN6CCC(CN7CCC(N8Cc9cc%10c(cc9C8)C(=O)N(C8CCC(=O)NC8=O)C%10)CC7)CC6)CC5)nc4c3F)c12	C61H65F2N11O7	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-75GXTH	WO2024233838A1_164	.	C#Cc1c(F)ccc2cc(O)cc(-c3nc(OC)c4c(N5CCCO[C@H]6C[C@H]65)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)CN([C@@H]8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C54H57F2N9O7	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-WVYMT2	WO2024233838A1_165	(3S)-3-[6-[4-[[4-[[1-[[7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-5-methoxy-4-[(1R,7S)-2-oxa-6-azabicyclo[5.1.0]octan-6-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperazin-1-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	C#Cc1c(F)ccc2cc(O)cc(-c3nc(OC)c4c(N5CCCO[C@@H]6C[C@@H]65)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(c8)CN([C@H]8CCC(=O)NC8=O)C9=O)CC7)CC6)CC5)nc4c3F)c12	C54H57F2N9O7	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-1M9RH4	WO2024233838A1_166	.	C#Cc1c(F)ccc2cc(O)cc(-c3nc(OC)c4c(N5CCCOC6CC65)nc(OCC5(CN6CCN(CC7CCN(c8ccc9c(N%10CCC(=O)NC%10=O)nn(C)c9c8)CC7)CC6)CC5)nc4c3F)c12	C53H57F2N11O6	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-0I8BY0	WO2024233838A1_167	.	C#Cc1c(F)ccc2cc(O)cc(-c3nc(OC)c4c(N5CCCOC6CC65)nc(OCC5(CN6CCN(CC7CCN(c8cccc(NC9CCC(=O)NC9=O)c8)CC7)CC6)CC5)nc4c3F)c12	C52H57F2N9O6	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-GIOA4L	WO2024233838A1_168	.	C#Cc1c(F)ccc2cc(O)cc(-c3nc(OC)c4c(N5CCCOC6CC65)nc(OCC5(CN6CCN(C[C@H]7CCN(c8ccc9c(c8)CN(C8CCC(=O)NC8=O)C9=O)C[C@@H]7F)CC6)CC5)nc4c3F)c12	C54H56F3N9O7	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-CIV1MB	WO2024233838A1_169	3-[6-[1-[[1-[[1-[[7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-5-methoxy-4-(2-oxa-6-azabicyclo[5.1.0]octan-6-yl)pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]methyl]piperidin-4-yl]-1-oxo-5,7-dihydro-3H-pyrrolo[3,4-f]isoindol-2-yl]piperidine-2,6-dione	C#Cc1c(F)ccc2cc(O)cc(-c3nc(OC)c4c(N5CCCOC6CC65)nc(OCC5(CN6CCC(CN7CCC(N8Cc9cc%10c(cc9C8)C(=O)N(C8CCC(=O)NC8=O)C%10)CC7)CC6)CC5)nc4c3F)c12	C57H61F2N9O7	KRAS	P01116	CRBN	WO-2024233838-A1
TPD-JIL0UV	WO2024235289A1_T-001	.	CNC(=O)C1=C(NC2=NC(NC3=C(OC)C=C(N4CCN(C(=O)CN5CCC(C6=CC=C(NC7CCC(=O)NC7=O)C=C6)CC5)CC4)C(C4CC4)=C3)=NC=C2Cl)C=CC=C1	C44H51ClN10O5	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-8VLK3T	WO2024235289A1_T-002	.	CNC(=O)C1=C(NC2=NC(NC3=C(OC)C=C(N4CCN(C(=O)CN5CCC(C6=CC=C(NC7CCC(=O)NC7=O)C=C6)CC5)CC4)C(C4CC4)=C3)=NC=C2Br)C=CC=C1	C44H51BrN10O5	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-7HRTKY	WO2024235289A1_T-003	.	C=CC1=CC(NC2=NC=C(Cl)C(NC3=C(C(=O)NC)C=CC=C3)=N2)=C(OC)C=C1N1CCN(C(=O)CN2CCC(C3=CC=C(NC4CCC(=O)NC4=O)C=C3)CC2)CC1	C43H49ClN10O5	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-W0ILH4	WO2024235289A1_T-004	.	C=CC1=CC(NC2=NC=C(Br)C(NC3=C(C(=O)NC)C=CC=C3)=N2)=C(OC)C=C1N1CCN(C(=O)CN2CCC(C3=CC=C(NC4CCC(=O)NC4=O)C=C3)CC2)CC1	C43H49BrN10O5	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-X8YOB6	WO2024235289A1_T-005	.	COC1=C(NC2=NC=C(Cl)C(NC3=C(N4N=CC=N4)C=CC=C3)=N2)C=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C41H45ClN12O4	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-J4X2TB	WO2024235289A1_T-006	.	COC1=C(NC2=NC=C(Br)C(NC3=C(N4N=CC=N4)C=CC=C3)=N2)C=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C41H45BrN12O4	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-5MK0M4	WO2024235289A1_T-007	.	COC1=C(NC2=NC=C(Cl)C(NC3=C(N4C=CN=N4)C=CC=C3)=N2)C=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C41H45ClN12O4	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-5WL54J	WO2024235289A1_T-008	.	COC1=C(NC2=NC=C(Br)C(NC3=C(N4C=CN=N4)C=CC=C3)=N2)C=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C41H45BrN12O4	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-KAB9KM	WO2024235289A1_T-009	.	CCC1=CC(NC2=NC(NC3=C(C(=O)NC)C=CC=C3)=C(Cl)C=N2)=C(OC)C=C1N1CCN(C(=O)CN2CCC(C3=CC=C(NC4CCC(=O)NC4=O)C=C3)C(F)(F)C2)CC1	C43H49ClF2N10O5	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-FVBLYL	WO2024235289A1_T-010	.	CCC1=CC(NC2=NC(NC3=C(C(=O)NC)C=CC=C3)=C(Br)C=N2)=C(OC)C=C1N1CCN(C(=O)CN2CCC(C3=CC=C(NC4CCC(=O)NC4=O)C=C3)C(F)(F)C2)CC1	C43H49BrF2N10O5	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-4B7ZMW	WO2024235289A1_T-011	.	COC1=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=CC=C1NC1=NC=C(Cl)C(NC2=C(C3=NC=CN3)C=CC=C2)=N1	C42H46ClN11O4	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-SNTV64	WO2024235289A1_T-012	.	COC1=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=CC=C1NC1=NC=C(Br)C(NC2=C(C3=NC=CN3)C=CC=C2)=N1	C42H46BrN11O4	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-940T5Q	WO2024235289A1_T-013	.	CCC1=CC(NC2=NC=C(Cl)C(NC3=C(C(=O)NC)C=CC=C3)=N2)=C(OC)C=C1N1CCN(C(=O)CN2CCC(C3=CC=C4C(=C3)N(C)N=C4N3CCC(=O)NC3=O)C(F)(F)C2)CC1	C44H49ClF2N12O5	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-KC44N5	WO2024235289A1_T-014	.	CCC1=CC(NC2=NC=C(Br)C(NC3=C(C(=O)NC)C=CC=C3)=N2)=C(OC)C=C1N1CCN(C(=O)CN2CCC(C3=CC=C4C(=C3)N(C)N=C4N3CCC(=O)NC3=O)C(F)(F)C2)CC1	C44H49BrF2N12O5	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-Z1KQ46	WO2024235289A1_T-015	.	CCC1=CC(NC2=NC=C(Cl)C(NC3=C(C(=O)NC)C=CC=C3)=N2)=C(OC)C=C1N1CCN(C(=O)CC2(O)CCN(C3=CC=C(NC4CCC(=O)NC4=O)CC3)CC2)CC1	C43H53ClN10O6	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-1TSGJP	WO2024235289A1_T-016	.	CCC1=CC(NC2=NC=C(Br)C(NC3=C(C(=O)NC)C=CC=C3)=N2)=C(OC)C=C1N1CCN(C(=O)CC2(O)CCN(C3=CC=C(NC4CCC(=O)NC4=O)CC3)CC2)CC1	C43H53BrN10O6	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-MW7SL6	WO2024235289A1_T-017	.	COC1=C(NC2=NC(NC3=CC=CC=C3C3=NC(C)=CN3)=C(Cl)C=N2)C=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C43H48ClN11O4	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-Z9DX95	WO2024235289A1_T-018	.	COC1=C(NC2=NC(NC3=CC=CC=C3C3=NC(C)=CN3)=C(Br)C=N2)C=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C43H48BrN11O4	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-0YKBVB	WO2024235289A1_T-019	.	COC1=C(NC2=NC(NC3=CC=CC=C3C3=NC(C)=C(C)N3)=C(Cl)C=N2)C=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C44H50ClN11O4	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-E22O63	WO2024235289A1_T-020	.	COC1=C(NC2=NC(NC3=CC=CC=C3C3=NC(C)=C(C)N3)=C(Br)C=N2)C=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C44H50BrN11O4	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-LZHFBW	WO2024235289A1_T-021	.	CNC(=O)C1=C(NC2=NC(NC3=C(OC)C=C(N4CCN(CCN5CCC(C6=CC=C(NC7CCC(=O)NC7=O)C=C6)CC5)CC4)C(C)=C3)=NC=C2Cl)C=CC=C1	C42H51ClN10O4	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-WVFOVM	WO2024235289A1_T-022	.	CNC(=O)C1=C(NC2=NC(NC3=C(OC)C=C(N4CCN(CCN5CCC(C6=CC=C(NC7CCC(=O)NC7=O)C=C6)CC5)CC4)C(C)=C3)=NC=C2Br)C=CC=C1	C42H51BrN10O4	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-LFHD67	WO2024235289A1_T-023	.	CCC1=CC(NC2=NC=C(Cl)C(NC3=C(C(=O)NC)C=CC=C3)=N2)=C(OC)C=C1N1CCN(CCN2CCC(C3=CC=C(NC4CCC(=O)NC4=O)C=C3)CC2)CC1	C43H53ClN10O4	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-FMYIFD	WO2024235289A1_T-024	.	CCC1=CC(NC2=NC=C(Br)C(NC3=C(C(=O)NC)C=CC=C3)=N2)=C(OC)C=C1N1CCN(CCN2CCC(C3=CC=C(NC4CCC(=O)NC4=O)C=C3)CC2)CC1	C43H53BrN10O4	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-BM39VG	WO2024235289A1_T-025	.	CNC(=O)C1=C(NC2=NC(NC3=C(OC)C=C(N4CCN(CCN5CCC(C6=CC=C(NC7CCC(=O)NC7=O)C=C6)CC5)CC4)C(C4CC4)=C3)=NC=C2Cl)C=CC=C1	C44H53ClN10O4	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-SVYSMP	WO2024235289A1_T-026	.	CNC(=O)C1=C(NC2=NC(NC3=C(OC)C=C(N4CCN(CCN5CCC(C6=CC=C(NC7CCC(=O)NC7=O)C=C6)CC5)CC4)C(C4CC4)=C3)=NC=C2Br)C=CC=C1	C44H53BrN10O4	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-O9P7WU	WO2024235289A1_T-027	.	C=CC1=CC(NC2=NC=C(Cl)C(NC3=C(C(=O)NC)C=CC=C3)=N2)=C(OC)C=C1N1CCN(CCN2CCC(C3=CC=C(NC4CCC(=O)NC4=O)C=C3)CC2)CC1	C43H51ClN10O4	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-1AVXSD	WO2024235289A1_T-028	.	C=CC1=CC(NC2=NC=C(Br)C(NC3=C(C(=O)NC)C=CC=C3)=N2)=C(OC)C=C1N1CCN(CCN2CCC(C3=CC=C(NC4CCC(=O)NC4=O)C=C3)CC2)CC1	C43H51BrN10O4	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-GX2GR3	WO2024235289A1_T-029	.	CCC1=CC(NC2=NC=C(Cl)C(NC3=C(C(=O)NC)C=CC=C3)=N2)=C(OC)C=C1N1CCN(C(=O)CN2CCN(C3=C(F)C=C(NC4CCC(=O)NC4=O)C=C3)CC2)CC1	C42H49ClFN11O5	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-0F2UQD	WO2024235289A1_T-030	.	CCC1=CC(NC2=NC=C(Br)C(NC3=C(C(=O)NC)C=CC=C3)=N2)=C(OC)C=C1N1CCN(C(=O)CN2CCN(C3=C(F)C=C(NC4CCC(=O)NC4=O)C=C3)CC2)CC1	C42H49BrFN11O5	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-H90DKB	WO2024235289A1_T-031	.	CNC(=O)C1=C(NC2=NC(NC3=C(OC)C=C(N4CCN(C(=O)CN5CCN(C6=C(F)C=C(NC7CCC(=O)NC7=O)C=C6)CC5)CC4)C(C)=C3)=NC=C2Cl)C=CC=C1	C41H47ClFN11O5	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-8PWOHX	WO2024235289A1_T-032	.	CNC(=O)C1=C(NC2=NC(NC3=C(OC)C=C(N4CCN(C(=O)CN5CCN(C6=C(F)C=C(NC7CCC(=O)NC7=O)C=C6)CC5)CC4)C(C)=C3)=NC=C2Br)C=CC=C1	C41H47BrFN11O5	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-3XI1M3	WO2024235289A1_T-033	.	CNC(=O)C1=C(NC2=NC(NC3=C(OC)C=C(N4CCN(C(=O)CC5(O)CCN(C6=C(F)C=C(NC7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)=NC=C2Cl)C=CC=C1	C41H46ClFN10O6	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-G8U5D3	WO2024235289A1_T-034	.	CNC(=O)C1=C(NC2=NC(NC3=C(OC)C=C(N4CCN(C(=O)CC5(O)CCN(C6=C(F)C=C(NC7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)=NC=C2Br)C=CC=C1	C41H46BrFN10O6	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-VFAKDB	WO2024235289A1_T-035	.	CNC(=O)C1=C(NC2=NC(NC3=C(OC)C=C(N4CCN(C(=O)CC5(O)CCN(C6=C(F)C=C(NC7CCC(=O)NC7=O)C=C6)CC5)CC4)C(C)=C3)=NC=C2Cl)C=CC=C1	C42H48ClFN10O6	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-F7IBOZ	WO2024235289A1_T-036	.	CNC(=O)C1=C(NC2=NC(NC3=C(OC)C=C(N4CCN(C(=O)CC5(O)CCN(C6=C(F)C=C(NC7CCC(=O)NC7=O)C=C6)CC5)CC4)C(C)=C3)=NC=C2Br)C=CC=C1	C42H48BrFN10O6	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-6Y9LSP	WO2024235289A1_T-037	.	CCC1=CC(NC2=NC=C(Cl)C(NC3=C(C(=O)NC)C=CC=C3)=N2)=C(OC)C=C1N1CCN(C(=O)CC2(O)CCN(C3=C(F)C=C(NC4CCC(=O)NC4=O)C=C3)CC2)CC1	C43H50ClFN10O6	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-JAQ6QG	WO2024235289A1_T-038	.	CCC1=CC(NC2=NC=C(Br)C(NC3=C(C(=O)NC)C=CC=C3)=N2)=C(OC)C=C1N1CCN(C(=O)CC2(O)CCN(C3=C(F)C=C(NC4CCC(=O)NC4=O)C=C3)CC2)CC1	C43H50BrFN10O6	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-478SIG	WO2024235289A1_T-039	.	C=CC1=CC(NC2=NC=C(Cl)C(NC3=C(C(=O)NC)C=CC=C3)=N2)=C(OC)C=C1N1CCN(C(=O)CC2(O)CCN(C3=C(F)C=C(NC4CCC(=O)NC4=O)C=C3)CC2)CC1	C43H48ClFN10O6	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-OTW0WJ	WO2024235289A1_T-040	.	C=CC1=CC(NC2=NC=C(Br)C(NC3=C(C(=O)NC)C=CC=C3)=N2)=C(OC)C=C1N1CCN(C(=O)CC2(O)CCN(C3=C(F)C=C(NC4CCC(=O)NC4=O)C=C3)CC2)CC1	C43H48BrFN10O6	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-9BILL7	WO2024235289A1_T-041	.	CNC(=O)C1=C(NC2=NC(NC3=C(OC)C=C(N4CCN(C(=O)CC5(O)CCN(C6=C(F)C=C(NC7CCC(=O)NC7=O)C=C6)CC5)CC4)C(C4CC4)=C3)=NC=C2Cl)C=CC=C1	C44H50ClFN10O6	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-SVSF7O	WO2024235289A1_T-042	.	CNC(=O)C1=C(NC2=NC(NC3=C(OC)C=C(N4CCN(C(=O)CC5(O)CCN(C6=C(F)C=C(NC7CCC(=O)NC7=O)C=C6)CC5)CC4)C(C4CC4)=C3)=NC=C2Br)C=CC=C1	C44H50BrFN10O6	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-Z0H19Q	WO2024235289A1_T-043	.	CCC1=CC(NC2=NC=C(Cl)C(NC3=C(C(=O)NC)C=CC=C3)=N2)=C(OC)C=C1N1CCN(C(=O)CN2CCC(C3=CC=C4C(=C3)N(C)N=C4N3CCC(=O)NC3=O)CC2)CC1	C44H51ClN12O5	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-2ZXBBK	WO2024235289A1_T-044	.	CCC1=CC(NC2=NC=C(Br)C(NC3=C(C(=O)NC)C=CC=C3)=N2)=C(OC)C=C1N1CCN(C(=O)CN2CCC(C3=CC=C4C(=C3)N(C)N=C4N3CCC(=O)NC3=O)CC2)CC1	C44H51BrN12O5	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-ZWVTLW	WO2024235289A1_T-045	.	CCC1=CC(NC2=NC=C(Cl)C(NC3=C(C(=O)NC)C=CC=C3)=N2)=C(OC)C=C1N1CCN(C(=O)CN2CCN(C3=CC=C4C(=C3)N(C)N=C4N3CCC(=O)NC3=O)CC2)CC1	C43H50ClN13O5	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-W93GTI	WO2024235289A1_T-046	.	CCC1=CC(NC2=NC=C(Br)C(NC3=C(C(=O)NC)C=CC=C3)=N2)=C(OC)C=C1N1CCN(C(=O)CN2CCN(C3=CC=C4C(=C3)N(C)N=C4N3CCC(=O)NC3=O)CC2)CC1	C43H50BrN13O5	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-3KD359	WO2024235289A1_T-047	.	CNC(=O)C1=C(NC2=NC(NC3=C(OC)C=C(N4CCN(C(=O)CN5CCC(C6=CC=C7C(=C6)N(C)N=C7N6CCC(=O)NC6=O)C(F)(F)C5)CC4)C=C3)=NC=C2Cl)C=CC=C1	C42H45ClF2N12O5	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-244QZK	WO2024235289A1_T-048	.	CNC(=O)C1=C(NC2=NC(NC3=C(OC)C=C(N4CCN(C(=O)CN5CCC(C6=CC=C7C(=C6)N(C)N=C7N6CCC(=O)NC6=O)C(F)(F)C5)CC4)C=C3)=NC=C2Br)C=CC=C1	C42H45BrF2N12O5	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-ZMY9XK	WO2024235289A1_T-049	.	CNC(=O)C1=C(NC2=NC(NC3=C(OC)C=C(N4CCN(C(=O)CN5CCC(C6=CC=C7C(=C6)N(C)N=C7N6CCC(=O)NC6=O)C(F)(F)C5)CC4)C(C)=C3)=NC=C2Cl)C=CC=C1	C43H47ClF2N12O5	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-6PYA7Y	WO2024235289A1_T-050	.	CNC(=O)C1=C(NC2=NC(NC3=C(OC)C=C(N4CCN(C(=O)CN5CCC(C6=CC=C7C(=C6)N(C)N=C7N6CCC(=O)NC6=O)C(F)(F)C5)CC4)C(C)=C3)=NC=C2Br)C=CC=C1	C43H47BrF2N12O5	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-Q49GQ4	WO2024235289A1_T-051	.	CNC(=O)C1=C(NC2=C(Cl)C=NC(NC3=C(OC)C=C(N4CCN(C(=O)CC5(F)CCN(C6=CC=C(NC7CCC(=O)NC7=O)C=C6)CC5)CC4)C(C)=C3)=N2)C=CC=C1	C42H48ClFN10O5	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-RILX0Y	WO2024235289A1_T-052	.	CNC(=O)C1=C(NC2=C(Br)C=NC(NC3=C(OC)C=C(N4CCN(C(=O)CC5(F)CCN(C6=CC=C(NC7CCC(=O)NC7=O)C=C6)CC5)CC4)C(C)=C3)=N2)C=CC=C1	C42H48BrFN10O5	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-0NTQ74	WO2024235289A1_T-053	.	CCC1=CC(NC2=NC(NC3=C(C(=O)NC)C=CC=C3)=C(Cl)C=N2)=C(OC)C=C1N1CCN(C(=O)CC2(F)CCN(C3=CC=C(NC4CCC(=O)NC4=O)C=C3)CC2)CC1	C43H50ClFN10O5	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-GSK8XG	WO2024235289A1_T-054	.	CCC1=CC(NC2=NC(NC3=C(C(=O)NC)C=CC=C3)=C(Br)C=N2)=C(OC)C=C1N1CCN(C(=O)CC2(F)CCN(C3=CC=C(NC4CCC(=O)NC4=O)C=C3)CC2)CC1	C43H50BrFN10O5	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-E9G9A2	WO2024235289A1_T-055	.	CNC(=O)C1=C(NC2=C(Cl)C=NC(NC3=C(OC)C=C(N4CCN(C(=O)CN5CCC(O)(C6=CC=C(NC7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)=N2)C=CC=C1	C41H47ClN10O6	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-S1CXT9	WO2024235289A1_T-056	.	CNC(=O)C1=C(NC2=C(Br)C=NC(NC3=C(OC)C=C(N4CCN(C(=O)CN5CCC(O)(C6=CC=C(NC7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)=N2)C=CC=C1	C41H47BrN10O6	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-WNUR1Q	WO2024235289A1_T-057	.	CNC(=O)C1=C(NC2=C(Cl)C=NC(NC3=C(OC)C=C(N4CCN(C(=O)CN5CCC(O)(C6=CC=C(NC7CCC(=O)NC7=O)C=C6)CC5)CC4)C(C)=C3)=N2)C=CC=C1	C42H49ClN10O6	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-9NQAAJ	WO2024235289A1_T-058	.	CNC(=O)C1=C(NC2=C(Br)C=NC(NC3=C(OC)C=C(N4CCN(C(=O)CN5CCC(O)(C6=CC=C(NC7CCC(=O)NC7=O)C=C6)CC5)CC4)C(C)=C3)=N2)C=CC=C1	C42H49BrN10O6	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-FKB0F8	WO2024235289A1_T-059	.	CCC1=CC(NC2=NC(NC3=C(C(=O)NC)C=CC=C3)=C(Cl)C=N2)=C(OC)C=C1N1CCN(C(=O)CN2CCC(O)(C3=CC=C(NC4CCC(=O)NC4=O)C=C3)CC2)CC1	C43H51ClN10O6	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-RSAR3A	WO2024235289A1_T-060	.	CCC1=CC(NC2=NC(NC3=C(C(=O)NC)C=CC=C3)=C(Br)C=N2)=C(OC)C=C1N1CCN(C(=O)CN2CCC(O)(C3=CC=C(NC4CCC(=O)NC4=O)C=C3)CC2)CC1	C43H51BrN10O6	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-R1KTE5	WO2024235289A1_T-061	.	CNC(=O)C1=C(NC2=C(Cl)C=NC(NC3=C(OC)C=C(N4CCN(C(=O)CN5CCC(F)(C6=CC=C(NC7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)=N2)C=CC=C1	C41H46ClFN10O5	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-CLSSOW	WO2024235289A1_T-062	.	CNC(=O)C1=C(NC2=C(Br)C=NC(NC3=C(OC)C=C(N4CCN(C(=O)CN5CCC(F)(C6=CC=C(NC7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)=N2)C=CC=C1	C41H46BrFN10O5	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-RN3U6Q	WO2024235289A1_T-063	.	CNC(=O)C1=C(NC2=C(Cl)C=NC(NC3=C(OC)C=C(N4CCN(C(=O)CN5CCC(F)(C6=CC=C(NC7CCC(=O)NC7=O)C=C6)CC5)CC4)C(C)=C3)=N2)C=CC=C1	C42H48ClFN10O5	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-IAEGV8	WO2024235289A1_T-064	.	CNC(=O)C1=C(NC2=C(Br)C=NC(NC3=C(OC)C=C(N4CCN(C(=O)CN5CCC(F)(C6=CC=C(NC7CCC(=O)NC7=O)C=C6)CC5)CC4)C(C)=C3)=N2)C=CC=C1	C42H48BrFN10O5	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-MQKL0I	WO2024235289A1_T-065	.	CCC1=CC(NC2=NC(NC3=C(C(=O)NC)C=CC=C3)=C(Cl)C=N2)=C(OC)C=C1N1CCN(C(=O)CN2CCC(F)(C3=CC=C(NC4CCC(=O)NC4=O)C=C3)CC2)CC1	C43H50ClFN10O5	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-7X4ZED	WO2024235289A1_T-066	.	CCC1=CC(NC2=NC(NC3=C(C(=O)NC)C=CC=C3)=C(Br)C=N2)=C(OC)C=C1N1CCN(C(=O)CN2CCC(F)(C3=CC=C(NC4CCC(=O)NC4=O)C=C3)CC2)CC1	C43H50BrFN10O5	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-EN7LHP	WO2024235289A1_T-067	.	CCC1=CC(NC2=NC(NC3=C(C(=O)NC)C=CC=C3)=C(Cl)C=N2)=C(OC)C=C1N1CCN(C(=O)CN2CCC(C3=CC=C(NC4CCC(=O)NC4=O)C=C3F)CC2)CC1	C43H50ClFN10O5	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-OY8XQI	WO2024235289A1_T-068	.	CCC1=CC(NC2=NC(NC3=C(C(=O)NC)C=CC=C3)=C(Cl)C=N2)=C(OC)C=C1N1CCN(C(=O)CN2CCC(C3=C(F)C=C(NC4CCC(=O)NC4=O)C=C3F)CC2)CC1	C43H49ClF2N10O5	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-1XMXTH	WO2024235289A1_T-069	.	CCC1=CC(NC2=NC(NC3=C(C(=O)NC)C=CC=C3)=C(Cl)C=N2)=C(OC)C=C1N1CCN(C(=O)CN2CCC(C3=CC=C(N(C)C4CCC(=O)NC4=O)C=C3)CC2)CC1	C44H53ClN10O5	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-MLV59J	WO2024235289A1_T-070	.	CCC1=CC(NC2=NC(NC3=C(C(=O)NC)C=CC=C3)=C(Cl)C=N2)=C(OC)C=C1N1CCN(C(=O)CN2CCN(C3=CC=C(NC4CCC(=O)NC4=O)C=C3)CC2)CC1	C42H50ClN11O5	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-3BP977	WO2024235289A1_T-071	.	CCC1=CC(NC2=NC(NC3=C(C(=O)NC)C=CC=C3)=C(Cl)C=N2)=C(OC)C=C1N1CCN(C(=O)CN2CCC(C3=CC=C(NC4CCC(=O)NC4=O)C=C3C#N)CC2)CC1	C44H50ClN11O5	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-PFN3JZ	WO2024235289A1_T-072	.	CCC1=CC(NC2=NC(NC3=C(C(=O)NC)C=CC=C3)=C(Cl)C=N2)=C(OC)C=C1N1CCN(C(=O)CC2CCN(C3=CC=C(NC4CCC(=O)NC4=O)C=C3)CC2)CC1	C43H51ClN10O5	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-62GGKW	WO2024235289A1_T-073	.	CCC1=CC(NC2=NC(NC3=C(C(=O)NC)C=CC=C3)=C(Cl)C=N2)=C(OC)C=C1N1CCN(C(=O)CN2CCC(C3=CC=C(NC4CCC(=O)NC4=O)C=C3C(F)F)CC2)CC1	C44H51ClF2N10O5	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-PWH0TU	WO2024235289A1_T-074	.	CCC1=CC(NC2=NC(NC3=C(C(=O)NC)C=CC=C3)=C(Cl)C=N2)=C(OC)C=C1N1CCN(C(=O)CN2CCC(C3=CC=C(NC4CCC(=O)NC4=O)C=C3C(F)(F)F)CC2)CC1	C44H50ClF3N10O5	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-FU4DF1	WO2024235289A1_T-075	.	CCC1=CC(NC2=NC(NC3=C(C(=O)NC)C=CC=C3)=C(Cl)C=N2)=C(OC)C=C1N1CCN(C(=O)CC2(O)CCN(C3=CC=C(NC4CCC(=O)NC4=O)C=C3C(F)(F)F)CC2)CC1	C44H50ClF3N10O6	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-BEAE6T	WO2024235289A1_T-076	.	CCC1=CC(NC2=NC(NC3=CC=CC4=C3C(=O)NC=N4)=C(Cl)C=N2)=C(OC)C=C1N1CCN(C(=O)CN2CCC(C3=CC=C(NC4CCC(=O)NC4=O)C=C3)CC2)CC1	C43H48ClN11O5	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-0OGC1V	WO2024235289A1_T-077	.	CCC1=CC(NC2=NC(NC3=CC=CC4=C3C(=O)NC=N4)=C(Br)C=N2)=C(OC)C=C1N1CCN(C(=O)CN2CCC(C3=CC=C(NC4CCC(=O)NC4=O)C=C3)CC2)CC1	C43H48BrN11O5	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-8FS99H	WO2024235289A1_T-078	.	CCC1=CC(NC2=NC(NC3=C(C(=O)NC)C=CC=C3)=C(Cl)C=N2)=C(OC)C=C1N1CCN(C(=O)CN2CCC(C3=CC=C(NC4CCC(=O)NC4=O)C=C3)CC2)[C@@H](C)C1	C44H53ClN10O5	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-666KNL	WO2024235289A1_T-079	.	CCC1=CC(NC2=NC(NC3=C(C(=O)NC)C=CC=C3)=C(Cl)C=N2)=C(OC)C=C1N1CCN(C(=O)CN2CCC(C3=CC=C(NC4CCC(=O)NC4=O)C=C3)CC2)[C@H](C)C1	C44H53ClN10O5	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-6VWN41	WO2024235289A1_T-080	.	CCC1=CC(NC2=NC(NC3=C(C(=O)NC)C=CC=C3)=C(Cl)C=N2)=C(OC)C=C1N1CC2(CN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)C2)C1	C44H51ClN10O5	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-1GEWS1	WO2024235289A1_T-082	.	CCC1=CC(NC2=NC=C(Cl)C(NC3=C(C(=O)NC)C=CC=C3)=N2)=C(OC)C=C1N1CCN(C(=O)CC2(O)CCN(C3=CC=C4C(=C3)N(C)N=C4N3CCC(=O)NC3=O)CC2)CC1	C44H51ClN12O6	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-QDP8JY	WO2024235289A1_T-083	.	CCC1=CC(NC2=NC=C(Br)C(NC3=C(C(=O)NC)C=CC=C3)=N2)=C(OC)C=C1N1CCN(C(=O)CC2(O)CCN(C3=CC=C4C(=C3)N(C)N=C4N3CCC(=O)NC3=O)CC2)CC1	C44H51BrN12O6	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-79COC9	WO2024235289A1_T-084	.	CCC1=CC(NC2=NC=C(Cl)C(NC3=C(C(=O)NC)C=CC=C3)=N2)=C(OC)C=C1N1CCN(C(=O)CC2(O)CCN(C3=C(F)C=C4C(=C3)N(C)N=C4N3CCC(=O)NC3=O)CC2)CC1	C44H50ClFN12O6	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-ZTOI8G	WO2024235289A1_T-085	.	CCC1=CC(NC2=NC=C(Br)C(NC3=C(C(=O)NC)C=CC=C3)=N2)=C(OC)C=C1N1CCN(C(=O)CC2(O)CCN(C3=C(F)C=C4C(=C3)N(C)N=C4N3CCC(=O)NC3=O)CC2)CC1	C44H50BrFN12O6	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-TBNA6W	WO2024235289A1_T-086	.	CNC(=O)C1=C(NC2=NC(NC3=C(OC)C=C(N4CCN(C(=O)CC5(O)CCN(C6=CC=C7C(=C6)N(C)N=C7N6CCC(=O)NC6=O)CC5)CC4)C(C)=C3)=NC=C2Cl)C=CC=C1	C43H49ClN12O6	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-JHZRCM	WO2024235289A1_T-087	.	CNC(=O)C1=C(NC2=NC(NC3=C(OC)C=C(N4CCN(C(=O)CC5(O)CCN(C6=CC=C7C(=C6)N(C)N=C7N6CCC(=O)NC6=O)CC5)CC4)C(C)=C3)=NC=C2Br)C=CC=C1	C43H49BrN12O6	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-FWR0LZ	WO2024235289A1_T-088	.	CNC(=O)C1=C(NC2=NC(NC3=C(OC)C=C(N4CCN(C(=O)CC5(O)CCN(C6=C(F)C=C7C(=C6)N(C)N=C7N6CCC(=O)NC6=O)CC5)CC4)C(C)=C3)=NC=C2Cl)C=CC=C1	C43H48ClFN12O6	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-6OTL4U	WO2024235289A1_T-089	.	CNC(=O)C1=C(NC2=NC(NC3=C(OC)C=C(N4CCN(C(=O)CC5(O)CCN(C6=C(F)C=C7C(=C6)N(C)N=C7N6CCC(=O)NC6=O)CC5)CC4)C(C)=C3)=NC=C2Br)C=CC=C1	C43H48BrFN12O6	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-RON8H2	WO2024235289A1_T-090	.	CCC1=CC(NC2=NC(NC3=C(C(=O)NC)C=CC=C3)=C(Cl)C=N2)=C(OC)C=C1N1CCN(C(=O)CN2CCC(C3=CC=C(NC4CCC(=O)NC4=O)C=C3C)CC2)CC1	C44H53ClN10O5	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-8Q2L13	WO2024235289A1_T-091	.	CCC1=CC(NC2=NC(NC3=C(C(=O)NC)C=CC=C3)=C(Br)C=N2)=C(OC)C=C1N1CCN(C(=O)CN2CCC(C3=CC=C(NC4CCC(=O)NC4=O)C=C3C)CC2)CC1	C44H53BrN10O5	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-T3G7KZ	WO2024235289A1_T-092	.	CCC1=CC(NC2=NC(NC3=C(C(=O)NC)C=CC=C3)=C(Cl)C=N2)=C(OC)C=C1N1CCN(C(C)CN2CCC(C3=CC=C(NC4CCC(=O)NC4=O)C=C3)CC2)CC1	C44H55ClN10O4	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-0H6KY7	WO2024235289A1_T-093	.	CCC1=CC(NC2=NC(NC3=C(C(=O)NC)C=CC=C3)=C(Br)C=N2)=C(OC)C=C1N1CCN(C(C)CN2CCC(C3=CC=C(NC4CCC(=O)NC4=O)C=C3)CC2)CC1	C44H55BrN10O4	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-FMQYNI	WO2024235289A1_T-094	.	CCC1=CC(NC2=NC(NC3=C(C(=O)NC)C=CC=C3)=C(Cl)C=N2)=C(OC)C=C1N1CCN(CC(C)N2CCC(C3=CC=C(NC4CCC(=O)NC4=O)C=C3)CC2)CC1	C44H55ClN10O4	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-EA4C0T	WO2024235289A1_T-095	.	CCC1=CC(NC2=NC(NC3=C(C(=O)NC)C=CC=C3)=C(Br)C=N2)=C(OC)C=C1N1CCN(CC(C)N2CCC(C3=CC=C(NC4CCC(=O)NC4=O)C=C3)CC2)CC1	C44H55BrN10O4	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-7RRT82	WO2024235289A1_T-096	.	CCC1=CC(NC2=NC(NC3=C(C(=O)NC)C=CC=C3)=C(Cl)C=N2)=C(OC)C=C1N1CCN(C(C)C(C)N2CCC(C3=CC=C(NC4CCC(=O)NC4=O)C=C3)CC2)CC1	C45H57ClN10O4	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-026RDS	WO2024235289A1_T-097	.	CCC1=CC(NC2=NC(NC3=C(C(=O)NC)C=CC=C3)=C(Br)C=N2)=C(OC)C=C1N1CCN(C(C)C(C)N2CCC(C3=CC=C(NC4CCC(=O)NC4=O)C=C3)CC2)CC1	C45H57BrN10O4	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-N6YLKQ	WO2024235289A1_T-098	.	CNC(=O)C1=C(NC2=C(Cl)C=NC(NC3=C(OC)C=C(N4CCN(C(C)C(C)N5CCC(C6=CC=C(NC7CCC(=O)NC7=O)C=C6)CC5)CC4)C(C)=C3)=N2)C=CC=C1	C44H55ClN10O4	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-5RDGG1	WO2024235289A1_T-099	.	CCC1=CC(NC2=NC(NC3=C(C(=O)NC)C=CC=C3)=C(Cl)C=N2)=C(OC)C=C1N1CCN(C2CC(N3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)C2)CC1	C45H55ClN10O4	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-SMA36Z	WO2024235289A1_T-100	.	CCC1=CC(NC2=NC(NC3=C(C(=O)NC)C=CC=C3)=C(Br)C=N2)=C(OC)C=C1N1CCN(C2CC(N3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)C2)CC1	C45H55BrN10O4	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-1FNR7X	WO2024235289A1_T-101	.	CCC1=CC(NC2=NC(NC3=C(C(=O)NC)C=CC=C3)=C(Cl)C=N2)=C(OC)C=C1N1CCN(C2COCC2N2CCC(C3=CC=C(NC4CCC(=O)NC4=O)C=C3)CC2)CC1	C45H55ClN10O5	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-3P4GJ5	WO2024235289A1_T-102	.	CCC1=CC(NC2=NC(NC3=C(C(=O)NC)C=CC=C3)=C(Br)C=N2)=C(OC)C=C1N1CCN(C2COCC2N2CCC(C3=CC=C(NC4CCC(=O)NC4=O)C=C3)CC2)CC1	C45H55BrN10O5	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-AWT1GW	WO2024235289A1_T-103	.	CCC1=CC(NC2=NC(C3=C4C=CC=CN4N=C3)=C(Cl)C=N2)=C(OC)C=C1N1CCN(C(=O)CN2CCC(C3=CC=C(NC4CCC(=O)NC4=O)C=C3)CC2)CC1	C42H47ClN10O4	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-GWQZAJ	WO2024235289A1_T-104	.	CCC1=CC(NC2=NC(C3=C4C=CC=CN4N=C3)=C(Br)C=N2)=C(OC)C=C1N1CCN(C(=O)CN2CCC(C3=CC=C(NC4CCC(=O)NC4=O)C=C3)CC2)CC1	C42H47BrN10O4	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-49VX3B	WO2024235289A1_T-105	.	COC1=C(NC2=NC(C3=C4C=CC=CN4N=C3)=C(Cl)C=N2)C=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C40H43ClN10O4	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-5KPW7M	WO2024235289A1_T-106	.	COC1=C(NC2=NC(C3=C4C=CC=CN4N=C3)=C(Br)C=N2)C=CC(N2CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C40H43BrN10O4	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-JBBG8K	WO2024235289A1_T-107	.	CCC1=CC(NC2=NC(NC3=C(C(=O)NC)C=CC=C3)=C(Cl)C=N2)=C(OC)C=C1N1CC2CC(C1)N2C(=O)CN1CCC(C2=CC=C(NC3CCC(=O)NC3=O)C=C2)CC1	C44H51ClN10O5	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-59KU3P	WO2024235289A1_T-108	.	CCC1=CC(NC2=NC(NC3=C(C(=O)NC)C=CC=C3)=C(Br)C=N2)=C(OC)C=C1N1CC2CC(C1)N2C(=O)CN1CCC(C2=CC=C(NC3CCC(=O)NC3=O)C=C2)CC1	C44H51BrN10O5	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-BLX34H	WO2024235289A1_T-109	.	CCC1=CC(NC2=NC(NC3=C(C(=O)NC)C=CC=C3)=C(Cl)C=N2)=C(OC)C=C1N1CC2CCC(C1)N2C(=O)CN1CCC(C2=CC=C(NC3CCC(=O)NC3=O)C=C2)CC1	C45H53ClN10O5	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-Q5E08L	WO2024235289A1_T-110	.	CCC1=CC(NC2=NC(NC3=C(C(=O)NC)C=CC=C3)=C(Br)C=N2)=C(OC)C=C1N1CC2CCC(C1)N2C(=O)CN1CCC(C2=CC=C(NC3CCC(=O)NC3=O)C=C2)CC1	C45H53BrN10O5	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-HYIS1Y	WO2024235289A1_T-111	.	CCC1=CC(NC2=NC(NC3=C(C(=O)NC)C=CC=C3)=C(Cl)C=N2)=C(OC)C=C1N1CCN([C@H](C)CN2CCC(C3=CC=C(NC4CCC(=O)NC4=O)C=C3)CC2)CC1	C44H55ClN10O4	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-GAJNGH	WO2024235289A1_T-112	.	CCC1=CC(NC2=NC(NC3=C(C(=O)NC)C=CC=C3)=C(Cl)C=N2)=C(OC)C=C1N1CCN([C@@H](C)CN2CCC(C3=CC=C(NC4CCC(=O)NC4=O)C=C3)CC2)CC1	C44H55ClN10O4	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-N9RCW2	WO2024235289A1_T-113	.	CCC1=CC(NC2=NC(NC3=C(C(=O)NC)C=CC=C3)=C(Cl)C=N2)=C(OC)C=C1N1CCN(C[C@@H](C)N2CCC(C3=CC=C(NC4CCC(=O)NC4=O)C=C3)CC2)CC1	C44H55ClN10O4	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-LP2EOJ	WO2024235289A1_T-114	.	CCC1=CC(NC2=NC(NC3=C(C(=O)NC)C=CC=C3)=C(Cl)C=N2)=C(OC)C=C1N1CCN(C[C@H](C)N2CCC(C3=CC=C(NC4CCC(=O)NC4=O)C=C3)CC2)CC1	C44H55ClN10O4	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-7OE2QF	WO2024235289A1_T-115	.	CCC1=CC(NC2=NC(NC3=C(C(=O)NC)C=CC=C3)=C(Cl)C=N2)=C(OC)C=C1N1CCN(C(=O)CN2CCC(C3=CC=C(NC4CCC(=O)NC4=O)C=N3)CC2)CC1	C42H50ClN11O5	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-ZUXTG9	WO2024235289A1_T-116	.	CCC1=CC(NC2=NC(NC3=C(C(=O)NC)C=CC=C3)=C(Br)C=N2)=C(OC)C=C1N1CCN(C(=O)CN2CCC(C3=CC=C(NC4CCC(=O)NC4=O)C=N3)CC2)CC1	C42H50BrN11O5	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-EWA2CK	WO2024235289A1_T-117	.	CCC1=CC(NC2=NC(NC3=C(C(=O)NC)C=CC=C3)=C(Cl)C=N2)=C(OC)C=C1N1CCN(C(=O)CN2CCC(C3=CC=C(OC4CCC(=O)NC4=O)C=C3)CC2)CC1	C43H50ClN9O6	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-HAFL2F	WO2024235289A1_T-118	.	CCC1=CC(NC2=NC(NC3=C(C(=O)NC)C=CC=C3)=C(Br)C=N2)=C(OC)C=C1N1CCN(C(=O)CN2CCC(C3=CC=C(OC4CCC(=O)NC4=O)C=C3)CC2)CC1	C43H50BrN9O6	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-AUSBBH	WO2024235289A1_T-119	.	CNC(=O)C1=C(NC2=C(Cl)C=NC(NC3=C(OC)C=C(N4CCN(C(=O)[C@H](C)N5CCC(C6=CC=C(NC7CCC(=O)NC7=O)C=C6)CC5)CC4)C(C)=C3)=N2)C=CC=C1	C43H51ClN10O5	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-KJ61OC	WO2024235289A1_T-120	.	CNC(=O)C1=C(NC2=C(Cl)C=NC(NC3=C(OC)C=C(N4CCN(C(=O)[C@@H](C)N5CCC(C6=CC=C(NC7CCC(=O)NC7=O)C=C6)CC5)CC4)C(C)=C3)=N2)C=CC=C1	C43H51ClN10O5	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-J00LW3	WO2024235289A1_T-121	.	CNC(=O)C1=C(NC2=C(Br)C=NC(NC3=C(OC)C=C(N4CCN(C(=O)[C@H](C)N5CCC(C6=CC=C(NC7CCC(=O)NC7=O)C=C6)CC5)CC4)C(C)=C3)=N2)C=CC=C1	C43H51BrN10O5	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-8YX9UH	WO2024235289A1_T-122	.	CNC(=O)C1=C(NC2=C(Br)C=NC(NC3=C(OC)C=C(N4CCN(C(=O)[C@@H](C)N5CCC(C6=CC=C(NC7CCC(=O)NC7=O)C=C6)CC5)CC4)C(C)=C3)=N2)C=CC=C1	C43H51BrN10O5	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-3IJ7K2	WO2024235289A1_T-123	.	CNC(=O)C1=C(NC2=C(Br)C=NC(NC3=C(OC)C=C(N4CCN(C(=O)C(C)N5CCC(C6=C(F)C=C(NC7CCC(=O)NC7=O)C=C6)CC5)CC4)C(C)=C3)=N2)C=CC=C1	C43H50BrFN10O5	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-D6VNM6	WO2024235289A1_T-124	.	COC1=C(NC2=NC(C3=C4C=CC=CN4N=C3)=C(Br)C=N2)C=C(C)C(N2CCN(C(=O)C(C)N3CCC(C4=C(F)C=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C42H46BrFN10O4	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-NNPD6Y	WO2024235289A1_T-125	.	COC1=C(NC2=NC(C3=C4C=CC=CN4N=C3)=C(Cl)C=N2)C=CC(N2CCN(C(=O)C(C)N3CCC(C4=C(F)C=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C41H44ClFN10O4	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-5B24HH	WO2024235289A1_T-126	.	COC1=C(NC2=NC(C3=C4C=CC=CN4N=C3)=C(Cl)C=N2)C=CC(N2CCN(C(=O)C(C)N3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)=C1	C41H45ClN10O4	EGFR	P00533	CRBN	WO-2024235289-A1
TPD-MLFDUO	WO2024240268A1_A-P-1	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(N5CC6(CCC7(CC6)COc6c7ccc7c6CN(C6CCC(=O)NC6=O)C7=O)C5)CC4)nn3)CC2)cc1Cl	C45H49ClN8O6	AR	P10275	CRBN	WO-2024240268-A1
TPD-824TTA	WO2024240268A1_A-P-10	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cc3c(cc21)C1(CCN(CC2CCN(c4ccc(C(=O)N[C@H]5CC[C@H](Oc6ccc(C#N)c(Cl)c6)CC5)nn4)CC2)CC1)CO3	C43H48ClN9O6	AR	P10275	CRBN	WO-2024240268-A1
TPD-8G1T2A	WO2024240268A1_A-P-100	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCC(CN5CCN6c7ccc(N[C@H]8CCC(=O)NC8=O)cc7OC[C@@H]6C5)CC4)cc3)C2(C)C)ccc1C#N	C45H55N7O6	AR	P10275	CRBN	WO-2024240268-A1
TPD-T406T5	WO2024240268A1_A-P-101	.	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(CN5CCN6c7cc(NC8CCC(=O)NC8=O)ccc7OCC[C@H]6C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C46H55ClN8O4	AR	P10275	CRBN	WO-2024240268-A1
TPD-L3XM1Q	WO2024240268A1_A-P-102	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCN6c7cc(NC8CCC(=O)NC8=O)ccc7OCC[C@H]6C5)CC4)nn3)CC2)cc1Cl	C41H48ClN9O5	AR	P10275	CRBN	WO-2024240268-A1
TPD-ED2A07	WO2024240268A1_A-P-103	.	COc1cc(N2CC3(CCN(c4ccc(C(=O)N5CCC(CN6CCN7c8cc(NC9CCC(=O)NC9=O)ccc8OCC[C@H]7C6)CC5)cc4)CC3)C[C@@H]2C)ccc1C#N	C47H58N8O5	AR	P10275	CRBN	WO-2024240268-A1
TPD-3OWUWQ	WO2024240268A1_A-P-104	.	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(F)(CN5CCN6c7cc(NC8CCC(=O)NC8=O)ccc7OCC[C@H]6C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C46H54ClFN8O4	AR	P10275	CRBN	WO-2024240268-A1
TPD-TL1FGK	WO2024240268A1_A-P-105	.	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(CN5CCN6c7cc(N(C)C8CCC(=O)NC8=O)ccc7OCC[C@H]6C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C47H57ClN8O4	AR	P10275	CRBN	WO-2024240268-A1
TPD-Q71784	WO2024240268A1_A-P-106	.	C=C(c1ccc(N2CCC3(CC2)C[C@H](C)N(c2ccc(C#N)c(Cl)c2)C3)cc1)N1CCC(CN2CCN3c4ccc(NC5CCC(=O)NC5=O)cc4OCC[C@H]3C2)CC1	C47H57ClN8O3	AR	P10275	CRBN	WO-2024240268-A1
TPD-PVFKT3	WO2024240268A1_A-P-107	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCN6c7ccc(NC8CCC(=O)NC8=O)cc7OCC[C@H]6C5)CC4)nn3)CC2)cc1Cl	C41H48ClN9O5	AR	P10275	CRBN	WO-2024240268-A1
TPD-ECC0CG	WO2024240268A1_A-P-108	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCC(CN5CCN6c7ccc(NC8CCC(=O)NC8=O)cc7OCC[C@H]6C5)CC4)cc3)C2(C)C)ccc1C#N	C46H57N7O6	AR	P10275	CRBN	WO-2024240268-A1
TPD-26QP0Q	WO2024240268A1_A-P-109	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCC(CN5CCN6c7cc(NC8CCC(=O)NC8=O)ccc7OCC[C@H]6C5)CC4)cc3)C2(C)C)ccc1C#N	C46H57N7O6	AR	P10275	CRBN	WO-2024240268-A1
TPD-5U467L	WO2024240268A1_A-P-11	.	COc1cc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC5(CC4)CC(N4CCC6(CC4)COc4cc7c(cc46)n(C)c(=O)n7C4CCC(=O)NC4=O)C5)nn3)CC2)ccc1C#N	C46H53N9O7	AR	P10275	CRBN	WO-2024240268-A1
TPD-MZDDD8	WO2024240268A1_A-P-12	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cc3c(cc21)C1(CCN(C2CC4(CCN(c5ccc(C(=O)N[C@H]6CC[C@H](Oc7ccc(C#N)c(Cl)c7)CC6)nn5)CC4)C2)CC1)CO3	C45H50ClN9O6	AR	P10275	CRBN	WO-2024240268-A1
TPD-XV6OIA	WO2024240268A1_A-P-13	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCC(F)(CN5CCC6(CC5)COc5cc7c(cc56)n(C)c(=O)n7C5CCC(=O)NC5=O)CC4)cc3)C2(C)C)ccc1C#N	C48H56FN7O7	AR	P10275	CRBN	WO-2024240268-A1
TPD-BITELX	WO2024240268A1_A-P-14	.	COc1cc(OC2C(C)(C)C(NC(=O)c3ccc(N4CCC5(CC4)CC(N4CCC6(CC4)COc4cc7c(cc46)n(C)c(=O)n7C4CCC(=O)NC4=O)C5)nn3)C2(C)C)ccc1C#N	C48H57N9O7	AR	P10275	CRBN	WO-2024240268-A1
TPD-EWXDAI	WO2024240268A1_A-P-15	.	COc1cc(OC2C(C)(C)C(NC(=O)c3ccc(N4CCC(CN5CCC6(CC5)COc5cc7c(cc56)n(C)c(=O)n7C5CCC(=O)NC5=O)CC4)cc3)C2(C)C)ccc1C#N	C48H57N7O7	AR	P10275	CRBN	WO-2024240268-A1
TPD-VF8Z3P	WO2024240268A1_A-P-16	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCC(C)(CN5CCC6(CC5)COc5cc7c(cc56)n(C)c(=O)n7C5CCC(=O)NC5=O)CC4)cc3)C2(C)C)ccc1C#N	C49H59N7O7	AR	P10275	CRBN	WO-2024240268-A1
TPD-INYPO2	WO2024240268A1_A-P-17	.	COc1cc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(CN5CCC6(CC5)COc5cc7c(cc56)n(C)c(=O)n7C5CCC(=O)NC5=O)CC4)nn3)CC2)ccc1C#N	C44H51N9O7	AR	P10275	CRBN	WO-2024240268-A1
TPD-GQ2UGM	WO2024240268A1_A-P-18	.	COc1cc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(N5CCC6(CC5)COc5cc7c(cc56)n(C)c(=O)n7C5CCC(=O)NC5=O)CC4)nn3)CC2)ccc1C#N	C43H49N9O7	AR	P10275	CRBN	WO-2024240268-A1
TPD-M8MBMU	WO2024240268A1_A-P-19	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cc3c(cc21)C1(CCN(C2CCN(c4ccc(C(=O)N[C@H]5CC[C@H](Oc6ccc(C#N)c(Cl)c6)CC5)nn4)CC2)CC1)CO3	C42H46ClN9O6	AR	P10275	CRBN	WO-2024240268-A1
TPD-KZ81OM	WO2024240268A1_A-P-2	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCC(N5CC6(CCC7(CC6)COc6c7ccc7c6CN(C6CCC(=O)NC6=O)C7=O)C5)CC4)cc3)C2(C)C)ccc1C#N	C50H58N6O7	AR	P10275	CRBN	WO-2024240268-A1
TPD-D976CA	WO2024240268A1_A-P-20	.	COc1cc(OC2C(C)(C)C(NC(=O)c3ccc(N4CCC(N5CCC6(CC5)COc5cc7c(cc56)n(C)c(=O)n7C5CCC(=O)NC5=O)CC4)cc3)C2(C)C)ccc1C#N	C47H55N7O7	AR	P10275	CRBN	WO-2024240268-A1
TPD-L2M7OD	WO2024240268A1_A-P-21	.	COc1cc(OC2C(C)(C)C(NC(=O)c3ccc(N4CCC5(CC4)CC(N4CCC6(CC4)COc4cc7c(cc46)n(C)c(=O)n7C4CCC(=O)NC4=O)C5)cc3)C2(C)C)ccc1C#N	C50H59N7O7	AR	P10275	CRBN	WO-2024240268-A1
TPD-7GJ4M6	WO2024240268A1_A-P-22	.	COc1cc(O[C@H]2CC[C@H](NC(=O)C3=NNC(N4CCC(CN5CCC6(CC5)COc5c6ccc6c5n(C)c(=O)n6C5CCC(=O)NC5=O)CC4)C=C3)CC2)ccc1C#N	C44H53N9O7	AR	P10275	CRBN	WO-2024240268-A1
TPD-Z221D8	WO2024240268A1_A-P-23	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2ccc3c(c21)OCC31CCN(C2CCN(c3ccc(C(=O)N[C@H]4CC[C@H](Oc5ccc(C#N)c(CI)c5)CC4)nn3)CC2)CC1	C43H48IN9O6	AR	P10275	CRBN	WO-2024240268-A1
TPD-RRGYKX	WO2024240268A1_A-P-24	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2ccc3c(c21)OCC31CCN(CC2CCN(c3ccc(C(=O)N[C@H]4CC[C@H](Oc5ccc(C#N)c(Cl)c5)CC4)nn3)CC2)CC1	C43H48ClN9O6	AR	P10275	CRBN	WO-2024240268-A1
TPD-66YQNW	WO2024240268A1_A-P-25	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2ccc3c(c21)OCC31CCN(C2CC3(CCN(c4ccc(C(=O)N[C@H]5CC[C@H](Oc6ccc(C#N)c(Cl)c6)CC5)nn4)CC3)C2)CC1	C45H50ClN9O6	AR	P10275	CRBN	WO-2024240268-A1
TPD-KTFTYK	WO2024240268A1_A-P-26	.	C[C@H]1CC2(CCN(c3ccc(N4CCC(CN5CCC6(CC5)COc5ccc7c(c56)n(C)c(=O)n7C5CCC(=O)NC5=O)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C47H55ClN8O4	AR	P10275	CRBN	WO-2024240268-A1
TPD-H8QLWE	WO2024240268A1_A-P-27	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCC(CN5CCC6(CC5)COc5c6ccc6c5n(C)c(=O)n6C5CCC(=O)NC5=O)CC4)nn3)C2(C)C)ccc1C#N	C46H55N9O7	AR	P10275	CRBN	WO-2024240268-A1
TPD-57NYNE	WO2024240268A1_A-P-28	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCC(CN5CCC6(CC5)COc5c6ccc6c5n(C)c(=O)n6C5CCC(=O)NC5=O)CC4)cc3)C2(C)C)ccc1C#N	C48H57N7O7	AR	P10275	CRBN	WO-2024240268-A1
TPD-8KOAKK	WO2024240268A1_A-P-29	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCC(N5CCC6(CC5)COc5c6ccc6c5n(C)c(=O)n6C5CCC(=O)NC5=O)CC4)cc3)C2(C)C)ccc1C#N	C47H55N7O7	AR	P10275	CRBN	WO-2024240268-A1
TPD-BI17H4	WO2024240268A1_A-P-3	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCC(CN5CC6(CCC7(CC6)COc6c7ccc7c6CN(C6CCC(=O)NC6=O)C7=O)C5)CC4)cc3)C2(C)C)ccc1C#N	C51H60N6O7	AR	P10275	CRBN	WO-2024240268-A1
TPD-LY4LCY	WO2024240268A1_A-P-30	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCC(CN5CCC6(CCc7cc(C(=O)N[C@H]8CCC(=O)NC8=O)c(F)cc7O6)CC5)CC4)cc3)C2(C)C)ccc1C#N	C48H57FN6O7	AR	P10275	CRBN	WO-2024240268-A1
TPD-4K1D18	WO2024240268A1_A-P-31	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCC(C)(CN5CCC6(CCc7cc(C(=O)N[C@H]8CCC(=O)NC8=O)c(F)cc7O6)CC5)CC4)cc3)C2(C)C)ccc1C#N	C49H59FN6O7	AR	P10275	CRBN	WO-2024240268-A1
TPD-WWHBR1	WO2024240268A1_A-P-32	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(N5CCC6(CC5)CCC5(CC6)COc6c5ccc5c6CC(C6C=CC(=O)NC6=O)C5=O)CC4)nn3)CC2)cc1Cl	C48H52ClN7O6	AR	P10275	CRBN	WO-2024240268-A1
TPD-3ZVLNO	WO2024240268A1_A-P-33	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCC(CN5CCC6(CCc7cc(C(=O)N[C@H]8CCC(=O)NC8=O)c(F)cc7O6)CC5)CC4)nc3)C2(C)C)ccc1C#N	C47H56FN7O7	AR	P10275	CRBN	WO-2024240268-A1
TPD-GWVUR7	WO2024240268A1_A-P-34	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCC(CN5CCC6(CCc7cc(C(=O)N[C@H]8CCC(=O)NC8=O)c(F)cc7O6)CC5)CC4)nn3)C2(C)C)ccc1C#N	C46H55FN8O7	AR	P10275	CRBN	WO-2024240268-A1
TPD-QHMLT7	WO2024240268A1_A-P-35	.	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(CN5CCC6(CCc7cc(C(=O)N[C@H]8CCC(=O)NC8=O)c(F)cc7O6)CC5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C48H55ClFN7O5	AR	P10275	CRBN	WO-2024240268-A1
TPD-17KNTK	WO2024240268A1_A-P-36	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCC(CN5CCC6(CCc7cc(C(=O)N[C@H]8CCC(=O)NC8=O)c(F)cc7O6)CC5)(OC)CC4)cc3)C2(C)C)ccc1C#N	C49H59FN6O8	AR	P10275	CRBN	WO-2024240268-A1
TPD-YOLOP2	WO2024240268A1_A-P-37	.	COCc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCC5(CC4)CC(N4CCC6(CCc7cc(C(=O)N[C@H]8CCC(=O)NC8=O)c(F)cc7O6)CC4)C5)cc3)C2(C)C)ccc1C#N	C51H61FN6O7	AR	P10275	CRBN	WO-2024240268-A1
TPD-JL2PW1	WO2024240268A1_A-P-38	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCC(C)(CN5CCC6(CCc7cc(F)c(C(=O)N[C@H]8CCC(=O)NC8=O)cc7O6)CC5)CC4)cc3)C2(C)C)ccc1C#N	C49H59FN6O7	AR	P10275	CRBN	WO-2024240268-A1
TPD-4KMUUR	WO2024240268A1_A-P-39	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCC(CN5CCC6(CCc7cc(F)c(C(=O)N[C@H]8CCC(=O)NC8=O)cc7O6)CC5)CC4)cc3)C2(C)C)ccc1C#N	C48H57FN6O7	AR	P10275	CRBN	WO-2024240268-A1
TPD-RNRC80	WO2024240268A1_A-P-4	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCC(C)(CN5CC6(CCC7(CC6)COc6c7ccc7c6CN(C6CCC(=O)NC6=O)C7=O)C5)CC4)cc3)C2(C)C)ccc1C#N	C52H62N6O7	AR	P10275	CRBN	WO-2024240268-A1
TPD-DKLW1W	WO2024240268A1_A-P-40	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCC(CN5CCC6(CCc7cc(F)c(C(=O)N[C@H]8CCC(=O)NC8=O)cc7O6)CC5)(OC)CC4)cc3)C2(C)C)ccc1C#N	C49H59FN6O8	AR	P10275	CRBN	WO-2024240268-A1
TPD-Q2GYI6	WO2024240268A1_A-P-41	.	COc1cc(OC2C(C)(C)C(NC(=O)c3ccc(N4CCC(F)(CN5CCC6(CCc7cc(F)c(C(=O)N[C@H]8CCC(=O)NC8=O)cc7O6)CC5)CC4)cc3)C2(C)C)ccc1C#N	C48H56F2N6O7	AR	P10275	CRBN	WO-2024240268-A1
TPD-Y866J5	WO2024240268A1_A-P-42	.	C[C@H]1CC2(CCN(c3ccc(N4CCC(CN5CCC6(CCc7cc(C(=O)N[C@H]8CCC(=O)NC8=O)c(F)cc7O6)CC5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C47H55ClFN7O4	AR	P10275	CRBN	WO-2024240268-A1
TPD-AK6RYG	WO2024240268A1_A-P-43	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCC(C)(CN5CCC6(CCc7cc(C(=O)N[C@H]8CCC(=O)NC8=O)c(F)cc7O6)CC5)CC4)cn3)C2(C)C)ccc1C#N	C48H58FN7O7	AR	P10275	CRBN	WO-2024240268-A1
TPD-752D54	WO2024240268A1_A-P-44	.	N#Cc1cc2c(cc1Cl)OCC1(CCN(C(=O)c3ccc(N4CCC(CN5CCC6(CCc7cc(C(=O)N[C@H]8CCC(=O)NC8=O)c(F)cc7O6)CC5)CC4)cc3)CC1)O2	C45H48ClFN6O7	AR	P10275	CRBN	WO-2024240268-A1
TPD-JKLZBM	WO2024240268A1_A-P-45	.	CC1(C)[C@H](NC(=O)c2ccc(N3CCC(CN4CCC5(CCc6cc(C(=O)N[C@H]7CCC(=O)NC7=O)c(F)cc6O5)CC4)CC3)nc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(C(F)(F)F)c1	C47H53F4N7O6	AR	P10275	CRBN	WO-2024240268-A1
TPD-L3VW0T	WO2024240268A1_A-P-46	.	N#Cc1cc2c(cc1Cl)OC1(CCN(c3ccc(C(=O)N4CCC(CN5CCC6(CCc7cc(C(=O)N[C@H]8CCC(=O)NC8=O)c(F)cc7O6)CC5)CC4)cc3)CC1)CO2	C45H48ClFN6O7	AR	P10275	CRBN	WO-2024240268-A1
TPD-RVCMNF	WO2024240268A1_A-P-47	.	COc1cc2c(cc1C(=O)N[C@H]1CCC(=O)NC1=O)CCC1(CCN(CC3CCN(C(=O)c4ccc(N5CCC6(CC5)C[C@H](C)N(c5ccc(C#N)c(Cl)c5)C6)cc4)CC3)CC1)O2	C49H58ClN7O6	AR	P10275	CRBN	WO-2024240268-A1
TPD-TQIHMG	WO2024240268A1_A-P-48	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCC(C)(CN5CCC6(CCc7cc(C(=O)N[C@H]8CCC(=O)NC8=O)c(F)cc7O6)CC5)CC4)nn3)C2(C)C)ccc1C#N	C47H57FN8O7	AR	P10275	CRBN	WO-2024240268-A1
TPD-IF08QI	WO2024240268A1_A-P-49	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCC(C)(CN5CCC6(CCc7cc(C(=O)N[C@H]8CCC(=O)NC8=O)c(F)cc7O6)CC5)CC4)nc3)C2(C)C)ccc1C#N	C48H58FN7O7	AR	P10275	CRBN	WO-2024240268-A1
TPD-UF4E1Q	WO2024240268A1_A-P-5	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCC(F)(CN5CC6(CCC7(CC6)COc6c7ccc7c6CN(C6CCC(=O)NC6=O)C7=O)C5)CC4)cc3)C2(C)C)ccc1C#N	C51H59FN6O7	AR	P10275	CRBN	WO-2024240268-A1
TPD-4LY02X	WO2024240268A1_A-P-50	.	CC1(C)[C@H](NC(=O)c2ccc(N3CCC(CN4CCC5(CCC6C=C(C(=O)N[C@H]7CCC(=O)NC7=O)C(F)=CC6O5)CC4)CC3)nc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C46H55ClFN7O6	AR	P10275	CRBN	WO-2024240268-A1
TPD-0YK4F9	WO2024240268A1_A-P-51	.	N#Cc1cc2c(cc1Cl)CC1(CCN(c3ccc(C(=O)N4CCC(CN5CCC6(CCc7cc(C(=O)N[C@H]8CCC(=O)NC8=O)c(F)cc7O6)CC5)CC4)cc3)CC1)CO2	C46H50ClFN6O6	AR	P10275	CRBN	WO-2024240268-A1
TPD-KXEE4Z	WO2024240268A1_A-P-52	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCC(F)(CN5CCC6(CCc7cc(C(=O)N[C@H]8CCC(=O)NC8=O)c(F)cc7O6)CC5)CC4)cc3)C2(C)C)ccc1C#N	C48H56F2N6O7	AR	P10275	CRBN	WO-2024240268-A1
TPD-H17CES	WO2024240268A1_A-P-53	.	N#Cc1cc2c(cc1Cl)OC1(CCN(C(=O)c3ccc(N4CCC(CN5CCC6(CCc7cc(C(=O)N[C@H]8CCC(=O)NC8=O)c(F)cc7O6)CC5)CC4)cc3)CC1)CO2	C45H48ClFN6O7	AR	P10275	CRBN	WO-2024240268-A1
TPD-IYFWPH	WO2024240268A1_A-P-54	.	COc1cc2c(cc1C(=O)N[C@H]1CCC(=O)NC1=O)CCC1(CCN(CC3CCN(c4ccc(N5CCC6(CC5)C[C@H](C)N(c5ccc(C#N)c(Cl)c5)C6)cc4)CC3)CC1)O2	C48H58ClN7O5	AR	P10275	CRBN	WO-2024240268-A1
TPD-26UX3J	WO2024240268A1_A-P-55	.	CC1(CN2CCC3(CCc4cc(C(=O)N[C@H]5CCC(=O)NC5=O)c(F)cc4O3)CC2)CCN(c2ccc(C(=O)N[C@H]3C(C)(C)[C@H](Oc4ccc(C#N)c(Cl)c4)C3(C)C)cc2)CC1	C48H56ClFN6O6	AR	P10275	CRBN	WO-2024240268-A1
TPD-R5EDPB	WO2024240268A1_A-P-56	.	COc1cc2c(cc1C(=O)N[C@H]1CCC(=O)NC1=O)CCC1(CCN(CC3CCN(c4ccc(C(=O)N[C@H]5C(C)(C)[C@H](OC6C=C(Cl)C(C#N)=CC6)C5(C)C)cc4)CC3)CC1)O2	C48H59ClN6O7	AR	P10275	CRBN	WO-2024240268-A1
TPD-1ZK0N9	WO2024240268A1_A-P-57	.	C[C@H]1CC2(CCN(c3ccc(N4CCC(CN5CCN6c7ccc(C(=O)N[C@H]8CCC(=O)NC8=O)cc7OC[C@@H]6C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H53ClN8O4	AR	P10275	CRBN	WO-2024240268-A1
TPD-Z2F58H	WO2024240268A1_A-P-58	.	C[C@H]1CC2(CCN(c3ccc(N4CCC(CN5CCN6c7ccc(C(=O)N[C@H]8CCC(=O)NC8=O)cc7OC[C@H]6C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H53ClN8O4	AR	P10275	CRBN	WO-2024240268-A1
TPD-3VKYC0	WO2024240268A1_A-P-59	.	C[C@H]1CC2(CCN(c3ccc(N4CCC(CN5CCN6c7cc(F)c(C(=O)N[C@H]8CCC(=O)NC8=O)cc7OC[C@H]6C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H52ClFN8O4	AR	P10275	CRBN	WO-2024240268-A1
TPD-28UKSX	WO2024240268A1_A-P-6	.	C[C@H]1CC2(CCN(c3ccc(N4CCC(CN5CC6(CCC7(CC6)COc6c7ccc7c6CN(C6CCC(=O)NC6=O)C7=O)C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C50H58ClN7O4	AR	P10275	CRBN	WO-2024240268-A1
TPD-X9XWIU	WO2024240268A1_A-P-60	.	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(CN5CCN6c7cc(F)c(C(=O)N[C@H]8CCC(=O)NC8=O)cc7OC[C@H]6C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C46H52ClFN8O5	AR	P10275	CRBN	WO-2024240268-A1
TPD-T0WFS3	WO2024240268A1_A-P-61	.	C[C@H]1CC2(CCN(c3ccc(N4CCC(CN5CCN6c7ccc(C(=O)N[C@H]8CCC(=O)NC8=O)c(F)c7OC[C@H]6C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C45H52ClFN8O4	AR	P10275	CRBN	WO-2024240268-A1
TPD-XOXIIP	WO2024240268A1_A-P-62	.	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(CN5CCN6c7ccc(C(=O)N[C@H]8CCC(=O)NC8=O)c(F)c7OC[C@H]6C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C46H52ClFN8O5	AR	P10275	CRBN	WO-2024240268-A1
TPD-KUUB56	WO2024240268A1_A-P-63	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCC(CN5CCN6c7cc(F)c(C(=O)N[C@H]8CCC(=O)NC8=O)cc7OC[C@H]6C5)CC4)cc3)C2(C)C)ccc1C#N	C46H54FN7O7	AR	P10275	CRBN	WO-2024240268-A1
TPD-XQEDMW	WO2024240268A1_A-P-64	.	COc1c(C(=O)N[C@H]2CCC(=O)NC2=O)ccc2c1OC[C@H]1CN(CC3CCN(C(=O)c4ccc(N5CCC6(CC5)C[C@H](C)N(c5ccc(C#N)c(Cl)c5)C6)cc4)CC3)CCN21	C47H55ClN8O6	AR	P10275	CRBN	WO-2024240268-A1
TPD-J6YRYX	WO2024240268A1_A-P-65	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCC(CN5CCN6c7cc(OC)c(C(=O)N[C@H]8CCC(=O)NC8=O)cc7COC[C@H]6C5)CC4)cc3)C2(C)C)ccc1C#N	C48H59N7O8	AR	P10275	CRBN	WO-2024240268-A1
TPD-PQDXKD	WO2024240268A1_A-P-66	.	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(CN5CCN6c7ccc(C(=O)N[C@H]8CCC(=O)NC8=O)cc7COC[C@H]6C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C47H55ClN8O5	AR	P10275	CRBN	WO-2024240268-A1
TPD-ZT4S7K	WO2024240268A1_A-P-67	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCC(CN5CCN6c7ccc(C(=O)N[C@H]8CCC(=O)NC8=O)cc7OC[C@@H]6C5)CC4)cc3)C2(C)C)ccc1C#N	C46H55N7O7	AR	P10275	CRBN	WO-2024240268-A1
TPD-3870VB	WO2024240268A1_A-P-68	.	CC1CC2(CCN(c3ccc(C(=O)N4CCC(CN5CCN6c7ccc(C(=O)N[C@H]8CCC(=O)NC8=O)cc7OC[C@H]6C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C46H53ClN8O5	AR	P10275	CRBN	WO-2024240268-A1
TPD-UARODO	WO2024240268A1_A-P-69	.	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(CN5CCN6c7ccc(C(=O)NC8CCC(=O)NC8=O)cc7OC[C@@H]6C5)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C46H53ClN8O5	AR	P10275	CRBN	WO-2024240268-A1
TPD-A79JPV	WO2024240268A1_A-P-7	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC(N5CCC6(CC5)CCC5(CC6)COc6c5ccc5c6CN(C6CCC(=O)NC6=O)C5=O)CC4)nn3)CC2)cc1Cl	C47H53ClN8O6	AR	P10275	CRBN	WO-2024240268-A1
TPD-7E5ESI	WO2024240268A1_A-P-70	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCC(CN5CCN6c7ccc(C(=O)N[C@H]8CCC(=O)NC8=O)cc7OC[C@H]6C5)CC4)cc3)C2(C)C)ccc1C#N	C46H55N7O7	AR	P10275	CRBN	WO-2024240268-A1
TPD-0MAV74	WO2024240268A1_A-P-71	.	COc1cc2c(cc1C(=O)N[C@H]1CCC(=O)NC1=O)N(C)C[C@H]1CN(CC3CCN(C(=O)c4ccc(N5CCC6(CC5)CC(C)N(c5ccc(C#N)c(Cl)c5)C6)cc4)CC3)CCN21	C48H58ClN9O5	AR	P10275	CRBN	WO-2024240268-A1
TPD-3EZS78	WO2024240268A1_A-P-72	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCC(CN5CCN6c7cc(OC)c(C(=O)N[C@H]8CCC(=O)NC8=O)cc7N(C)C[C@H]6C5)CC4)cc3)C2(C)C)ccc1C#N	C48H60N8O7	AR	P10275	CRBN	WO-2024240268-A1
TPD-SEWPMS	WO2024240268A1_A-P-73	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCC(CN5CCN6c7cc(OC)c(C(=O)N[C@H]8CCC(=O)NC8=O)cc7OC[C@H]6C5)CC4)cc3)C2(C)C)ccc1C#N	C47H57N7O8	AR	P10275	CRBN	WO-2024240268-A1
TPD-71D5YL	WO2024240268A1_A-P-75	.	COc1cc2c(cc1C(=O)N[C@H]1CCC(=O)NC1=O)OC[C@H]1CN(CC3CCN(c4ccc(N5CCC6(CC5)C[C@H](C)N(c5ccc(C#N)c(Cl)c5)C6)cc4)CC3)CCN21	C46H55ClN8O5	AR	P10275	CRBN	WO-2024240268-A1
TPD-R727ND	WO2024240268A1_A-P-76	.	COc1cc2c(cc1C(=O)N[C@H]1CCC(=O)NC1=O)OC[C@H]1CN(CC3CCN(C(=O)c4ccc(N5CCC6(CC5)C[C@H](C)N(c5ccc(C#N)c(Cl)c5)C6)cc4)CC3)CCN21	C47H55ClN8O6	AR	P10275	CRBN	WO-2024240268-A1
TPD-37FW84	WO2024240268A1_A-P-77	.	CC1(C)[C@H](NC(=O)c2ccc(N3CCC(CN4CCN5c6ccc(C(=O)N[C@H]7CCC(=O)NC7=O)cc6OC[C@H]5C4)CC3)cc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(Cl)c1	C45H52ClN7O6	AR	P10275	CRBN	WO-2024240268-A1
TPD-S5YGG3	WO2024240268A1_A-P-78	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCC(CN5CCC6(CC5)COc5c6ccc(C(=O)N[C@H]6CCC(=O)NC6=O)c5OC)CC4)cc3)C2(C)C)ccc1C#N	C48H58N6O8	AR	P10275	CRBN	WO-2024240268-A1
TPD-EJ723Q	WO2024240268A1_A-P-79	.	COc1cc2c(cc1C(=O)N[C@H]1CCC(=O)NC1=O)OCC21CCN(CC2CCN(C(=O)c3ccc(N4CCC5(CC4)C[C@H](C)N(c4ccc(C#N)c(Cl)c4)C5)cc3)CC2)CC1	C48H56ClN7O6	AR	P10275	CRBN	WO-2024240268-A1
TPD-P6YOLK	WO2024240268A1_A-P-8	.	C[C@H]1CC2(CCN(c3ccc(N4CCC(CN5CCC6(CC5)CCC5(CC6)COc6c5ccc5c6CN(C6CCC(=O)NC6=O)C5=O)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C52H62ClN7O4	AR	P10275	CRBN	WO-2024240268-A1
TPD-75OIL8	WO2024240268A1_A-P-80	.	COc1cc2c(cc1C(=O)N[C@H]1CCC(=O)NC1=O)OCC21CCN(CC2CCN(c3ccc(N4CCC5(CC4)C[C@H](C)N(c4ccc(C#N)c(Cl)c4)C5)cc3)CC2)CC1	C47H56ClN7O5	AR	P10275	CRBN	WO-2024240268-A1
TPD-N40HX2	WO2024240268A1_A-P-81	.	COc1cc2c(cc1C(=O)N[C@H]1CCC(=O)NC1=O)C1(CCN(CC3CCN(c4ccc(N5CCC6(CC5)C[C@H](C)N(c5ccc(C#N)c(Cl)c5)C6)cc4)CC3)CC1)CO2	C47H56ClN7O5	AR	P10275	CRBN	WO-2024240268-A1
TPD-I1E9NZ	WO2024240268A1_A-P-82	.	COc1cc2c(cc1C(=O)N[C@H]1CCC(=O)NC1=O)C1(CCN(CC3CCN(C(=O)c4ccc(N5CCC6(CC5)C[C@H](C)N(c5ccc(C#N)c(Cl)c5)C6)cc4)CC3)CC1)CO2	C48H56ClN7O6	AR	P10275	CRBN	WO-2024240268-A1
TPD-T8009T	WO2024240268A1_A-P-83	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCC(CN5CCC6(CC5)COc5c6ccc(C(=O)N[C@H]6CCC(=O)NC6=O)c5F)CC4)cc3)C2(C)C)ccc1C#N	C47H55FN6O7	AR	P10275	CRBN	WO-2024240268-A1
TPD-QZODOU	WO2024240268A1_A-P-84	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCC(F)(CN5CCCOc6c(ccc(C(=O)N[C@H]7CCC(=O)NC7=O)c6F)CC5)CC4)cc3)C2(C)C)ccc1C#N	C46H54F2N6O7	AR	P10275	CRBN	WO-2024240268-A1
TPD-4KTJ90	WO2024240268A1_A-P-85	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCC(C)(CN5CCC6(CC5)COc5c6ccc(C(=O)N[C@H]6CCC(=O)NC6=O)c5F)CC4)cc3)C2(C)C)ccc1C#N	C48H57FN6O7	AR	P10275	CRBN	WO-2024240268-A1
TPD-8VWIDM	WO2024240268A1_A-P-86	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCC(CN5CCC6(CC5)COc5c6ccc(C(=O)N[C@H]6CCC(=O)NC6=O)c5F)(OC)CC4)cc3)C2(C)C)ccc1C#N	C48H57FN6O8	AR	P10275	CRBN	WO-2024240268-A1
TPD-F43UH4	WO2024240268A1_A-P-87	.	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(CN5CCC6(CC5)COc5cc(NC7CCC(=O)NC7=O)ccc56)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C46H54ClN7O4	AR	P10275	CRBN	WO-2024240268-A1
TPD-700NPI	WO2024240268A1_A-P-88	.	CC(C)N(CC1(C)CCN(c2ccc(C(=O)N3CCC(C)(CN4CCC5(CC4)COc4cc(NC6CCC(=O)NC6=O)ccc45)CC3)cc2)CC1)c1ccc(C#N)c(Cl)c1	C48H60ClN7O4	AR	P10275	CRBN	WO-2024240268-A1
TPD-NIVCG6	WO2024240268A1_A-P-89	.	COc1cc(N2CC3(CCN(c4ccc(C(=O)N5CCC(CN6CCC7(CC6)COc6cc(NC8CCC(=O)NC8=O)ccc67)CC5)cc4)CC3)C[C@@H]2C)ccc1C#N	C47H57N7O5	AR	P10275	CRBN	WO-2024240268-A1
TPD-A53OUQ	WO2024240268A1_A-P-9	.	N#Cc1ccc(O[C@H]2CC[C@H](NC(=O)c3ccc(N4CCC5(CC4)CCC4(CC5)COc5c4ccc4c5CN(C5CCC(=O)NC5=O)C4=O)nn3)CC2)cc1Cl	C42H44ClN7O6	AR	P10275	CRBN	WO-2024240268-A1
TPD-K7VL87	WO2024240268A1_A-P-90	.	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(O)(CN5CCC6(CC5)COc5cc(NC7CCC(=O)NC7=O)ccc56)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C46H54ClN7O5	AR	P10275	CRBN	WO-2024240268-A1
TPD-LG0N2W	WO2024240268A1_A-P-91	.	COC1(CN2CCC3(CC2)COc2cc(NC4CCC(=O)NC4=O)ccc23)CCN(C(=O)c2ccc(N3CCC4(CC3)C[C@H](C)N(c3ccc(C#N)c(Cl)c3)C4)cc2)CC1	C47H56ClN7O5	AR	P10275	CRBN	WO-2024240268-A1
TPD-4HWO5J	WO2024240268A1_A-P-92	.	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(F)(CN5CCC6(CC5)COc5cc(NC7CCC(=O)NC7=O)ccc56)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C46H53ClFN7O4	AR	P10275	CRBN	WO-2024240268-A1
TPD-5OOIGU	WO2024240268A1_A-P-93	.	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(CN5CCC6(CC5)COc5cc(N(C)C7CCC(=O)NC7=O)ccc56)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C47H56ClN7O4	AR	P10275	CRBN	WO-2024240268-A1
TPD-TBEL7W	WO2024240268A1_A-P-94	.	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(CN5CCC6(CC5)Cc5ccc(NC7CCC(=O)NC7=O)cc5O6)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C46H54ClN7O4	AR	P10275	CRBN	WO-2024240268-A1
TPD-ZNJECX	WO2024240268A1_A-P-95	.	COC1(CN2CCC3(CC2)Cc2ccc(NC4CCC(=O)NC4=O)cc2O3)CCN(C(=O)c2ccc(N3CCC4(CC3)C[C@H](C)N(c3ccc(C#N)c(Cl)c3)C4)cc2)CC1	C47H56ClN7O5	AR	P10275	CRBN	WO-2024240268-A1
TPD-CT4FMM	WO2024240268A1_A-P-96	.	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(C#N)(CN5CCC6(CC5)Cc5ccc(NC7CCC(=O)NC7=O)cc5O6)CC4)cc3)CC2)CN1C1=CC=C(C#N)C(Cl)C1	C47H55ClN8O4	AR	P10275	CRBN	WO-2024240268-A1
TPD-2KMUZ5	WO2024240268A1_A-P-97	.	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(C)(CN5CCC6(CC5)Cc5ccc(NC7CCC(=O)NC7=O)cc5O6)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C47H56ClN7O4	AR	P10275	CRBN	WO-2024240268-A1
TPD-E7F5C7	WO2024240268A1_A-P-98	.	C[C@H]1CC2(CCN(c3ccc(C(=O)N4CCC(CN5CCC6(CC5)COc5ccc(NC7CCC(=O)NC7=O)cc56)CC4)cc3)CC2)CN1c1ccc(C#N)c(Cl)c1	C46H54ClN7O4	AR	P10275	CRBN	WO-2024240268-A1
TPD-8OYK4C	WO2024240268A1_A-P-99	.	COc1cc(N2CC3(CCN(c4ccc(C(=O)N5CCC(CN6CCC7(CC6)COc6ccc(NC8CCC(=O)NC8=O)cc67)CC5)cc4)CC3)C[C@@H]2C)ccc1C#N	C47H57N7O5	AR	P10275	CRBN	WO-2024240268-A1
TPD-NPRH35	WO2024240268A1_ER-P-1	.	O=C1CCC(N2Cc3c(ccc4c3OCC43CCC4(CCN(CC5CCN(c6ccc([C@@H]7c8ccc(O)cc8CC[C@@H]7c7ccccc7)cc6)CC5)CC4)CC3)C2=O)C(=O)N1	C52H58N4O5	ERα	P03372	CRBN	WO-2024240268-A1
TPD-THRX1B	WO2024240268A1_ER-P-10	.	O=C1CCC(N2Cc3c(ccc4c3OCC43CCC4(CC3)CN(C3CCC5(CC3)CN(c3ccc([C@@H]6c7ccc(O)cc7CC[C@@H]6c6ccccc6)cc3)C5)C4)C2=O)C(=O)N1	C52H56N4O5	ERα	P03372	CRBN	WO-2024240268-A1
TPD-G9A2M8	WO2024240268A1_ER-P-11	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cc3c(cc21)C1(CCN(C2CCN(c4ccc([C@@H]5c6ccc(O)cc6CC[C@@H]5c5ccccc5)cc4)CC2)CC1)CO3	C46H49N5O5	ERα	P03372	CRBN	WO-2024240268-A1
TPD-Q2WW0I	WO2024240268A1_ER-P-12	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cc3c(cc21)C1(CCN(C2CC4(CCN(c5ccc([C@@H]6c7ccc(O)cc7CC[C@@H]6c6ccccc6)cc5)CC4)C2)CC1)CO3	C49H53N5O5	ERα	P03372	CRBN	WO-2024240268-A1
TPD-8N0EAX	WO2024240268A1_ER-P-13	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2ccc3c(c21)OCC31CCN(C2CCN(C(=O)C3CCN(c4ccc([C@@H]5c6ccc(O)cc6CC[C@@H]5c5ccccc5)cc4)CC3)CC2)CC1	C52H58N6O6	ERα	P03372	CRBN	WO-2024240268-A1
TPD-0NFO30	WO2024240268A1_ER-P-14	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cc3c(cc21)C1(CCN(C2CCN(C(=O)C4CCN(c5ccc([C@@H]6c7ccc(O)cc7CC[C@@H]6c6ccccc6)cc5)CC4)CC2)CC1)CO3	C52H58N6O6	ERα	P03372	CRBN	WO-2024240268-A1
TPD-4OYO47	WO2024240268A1_ER-P-16	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2C=CC3=C(OCC34CCN(C3CCC5(CC3)CCN(c3ccc([C@@H]6c7ccc(O)cc7CC[C@@H]6c6ccccc6)cc3)CC5)CC4)C21	C51H59N5O5	ERα	P03372	CRBN	WO-2024240268-A1
TPD-TIQ0EW	WO2024240268A1_ER-P-17	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2ccc3c(c21)OCC31CCN(C2CC3(CCN(c4ccc([C@@H]5c6ccc(O)cc6CC[C@@H]5c5ccccc5)cc4)CC3)C2)CC1	C49H53N5O5	ERα	P03372	CRBN	WO-2024240268-A1
TPD-4NSF2V	WO2024240268A1_ER-P-18	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2ccc3c(c21)OCC31CCN(C2CC3(C2)CN(c2ccc([C@@H]4c5ccc(O)cc5CC[C@@H]4c4ccccc4)cc2)C3)CC1	C47H49N5O5	ERα	P03372	CRBN	WO-2024240268-A1
TPD-PMGU7T	WO2024240268A1_ER-P-19	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2ccc3c(c21)C1(CCN(C2CCC4(CC2)CN(c2ccc([C@@H]5c6ccc(O)cc6CC[C@@H]5c5ccccc5)cc2)C4)CC1)CO3	C49H53N5O5	ERα	P03372	CRBN	WO-2024240268-A1
TPD-RQHOTZ	WO2024240268A1_ER-P-2	.	O=C1CCC(N2Cc3c(ccc4c3OCC43CCC4(CCN(C5CCC6(CC5)CN(c5ccc([C@@H]7c8ccc(O)cc8CC[C@@H]7c7ccccc7)cc5)C6)CC4)CC3)C2=O)C(=O)N1	C54H60N4O5	ERα	P03372	CRBN	WO-2024240268-A1
TPD-EUV98X	WO2024240268A1_ER-P-21	.	C[C@@H]1Cc2cc(O)ccc2C(c2c(F)cc(N3CCC4(CCC(N5CC6(CCC7(CC6)COc6c7ccc7c6CN(C6CCC(=O)NC6=O)C7=O)C5)CC4)CC3)cc2F)N1CC(F)F	C50H57F4N5O5	ERα	P03372	CRBN	WO-2024240268-A1
TPD-PDTSFI	WO2024240268A1_ER-P-22	.	C[C@@H]1Cc2cc(O)ccc2C(c2c(F)cc(N3CCC(C(=O)N4CCC(N5CCC6(CC5)COc5cc7c(cc56)n(C)c(=O)n7C5CCC(=O)NC5=O)CC4)CC3)cc2F)N1CC(F)F	C48H55F4N7O6	ERα	P03372	CRBN	WO-2024240268-A1
TPD-CML6OX	WO2024240268A1_ER-P-23	.	O=C1CCC(N2Cc3c(ccc4c3OCC43CCC4(CC3)CN(CC3CCN(c5ccc([C@@H]6c7ccc(O)cc7CC[C@@H]6c6ccccc6)cc5)CC3)C4)C2=O)C(=O)N1	C50H54N4O5	ERα	P03372	CRBN	WO-2024240268-A1
TPD-X923CX	WO2024240268A1_ER-P-24	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cc3c(cc21)C1(CCN(CC2CCN(c4ccc([C@@H]5c6ccc(O)cc6CC[C@@H]5c5ccccc5)cc4)CC2)CC1)CO3	C47H51N5O5	ERα	P03372	CRBN	WO-2024240268-A1
TPD-LRGRIY	WO2024240268A1_ER-P-25	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2ccc3c(c21)OCC31CCN(C(=O)C2CN(CC3CCN(c4ccc([C@@H]5c6ccc(O)cc6CC[C@@H]5c5ccccc5)cc4)CC3)C2)CC1	C51H56N6O6	ERα	P03372	CRBN	WO-2024240268-A1
TPD-HH996P	WO2024240268A1_ER-P-26	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cc3c(cc21)C1(CCN(C(=O)C2CN(CC4CCN(c5ccc([C@@H]6c7ccc(O)cc7CC[C@@H]6c6ccccc6)cc5)CC4)C2)CC1)CO3	C51H56N6O6	ERα	P03372	CRBN	WO-2024240268-A1
TPD-BR21F0	WO2024240268A1_ER-P-27	.	C[C@@H]1Cc2cc(O)ccc2C(c2c(F)cc(N3CCC4(CC3)CC(N3CCC5(CC3)CCC3(CC5)COc5c3ccc3c5CN(C5CCC(=O)NC5=O)C3=O)C4)cc2F)N1CC(F)F	C50H57F4N5O5	ERα	P03372	CRBN	WO-2024240268-A1
TPD-2QLITZ	WO2024240268A1_ER-P-28	.	C[C@@H]1Cc2cc(O)ccc2C(c2c(F)cc(N3CCC4(CC3)CC(N3CC5(CCC6(CC5)COc5c6ccc6c5CN(C5CCC(=O)NC5=O)C6=O)C3)C4)cc2F)N1CC(F)F	C48H53F4N5O5	ERα	P03372	CRBN	WO-2024240268-A1
TPD-X4S0EF	WO2024240268A1_ER-P-29	.	C[C@@H]1Cc2cc(O)ccc2C(c2c(F)cc(N3CCC4(CCC(N5CCC6(CC5)COc5c6ccc6c5n(C)c(=O)n6C5CCC(=O)NC5=O)CC4)CC3)cc2F)N1CC(F)F	C47H54F4N6O5	ERα	P03372	CRBN	WO-2024240268-A1
TPD-1EM6OB	WO2024240268A1_ER-P-3	.	O=C1CCC(N2Cc3c(ccc4c3OCC43CCC4(CCN(C5CC6(CCN(c7ccc([C@@H]8c9ccc(O)cc9CC[C@@H]8c8ccccc8)cc7)CC6)C5)CC4)CC3)C2=O)C(=O)N1	C54H60N4O5	ERα	P03372	CRBN	WO-2024240268-A1
TPD-M1MG4H	WO2024240268A1_ER-P-30	.	C[C@@H]1Cc2cc(O)ccc2C(c2c(F)cc(N3CCC(C(=O)N4CCC(N5CCC6(CC5)COc5c6ccc6c5n(C)c(=O)n6C5CCC(=O)NC5=O)CC4)CC3)cc2F)N1CC(F)F	C48H55F4N7O6	ERα	P03372	CRBN	WO-2024240268-A1
TPD-V5GNMG	WO2024240268A1_ER-P-31	.	O=C1CCC(Nc2ccc3c(c2)OCC32CCN(C[C@H]3CC[C@@H](OC4CCN(c5ccc([C@@H]6c7ccc(O)cc7CCC6c6ccccc6)cc5)CC4)CC3)CC2)C(=O)N1	C51H60N4O5	ERα	P03372	CRBN	WO-2024240268-A1
TPD-NKFEVA	WO2024240268A1_ER-P-32	.	CN(c1ccc2c(c1)OCC21CCN(C[C@H]2CC[C@@H](OC3CCN(c4ccc([C@@H]5c6ccc(O)cc6CC[C@@H]5c5ccccc5)cc4)CC3)CC2)CC1)C1CCC(=O)NC1=O	C52H62N4O5	ERα	P03372	CRBN	WO-2024240268-A1
TPD-E7PSVO	WO2024240268A1_ER-P-33	.	O=C1CCC(Nc2ccc3c(c2)OC2(CC3)CN(C[C@H]3CC[C@@H](OC4CCN(c5ccc([C@@H]6c7ccc(O)cc7CC[C@@H]6c6ccccc6)cc5)CC4)CC3)C2)C(=O)N1	C50H58N4O5	ERα	P03372	CRBN	WO-2024240268-A1
TPD-TJYVJ7	WO2024240268A1_ER-P-35	.	O=C1CCC(Nc2ccc3c(c2)OC[C@@H]2CN(C4CC5(CCN(c6ccc([C@@H]7c8ccc(O)cc8CC[C@@H]7c7ccccc7)cc6)CC5)C4)CCN32)C(=O)N1	C46H51N5O4	ERα	P03372	CRBN	WO-2024240268-A1
TPD-J3JAH3	WO2024240268A1_ER-P-36	.	O=C1CCC(Nc2ccc3c(c2)OC[C@@H]2CN(C4CCC5(CC4)CN(c4ccc([C@@H]6c7ccc(O)cc7CC[C@@H]6c6ccccc6)cc4)C5)CCN32)C(=O)N1	C46H51N5O4	ERα	P03372	CRBN	WO-2024240268-A1
TPD-95A80P	WO2024240268A1_ER-P-37	.	O=C1CC[C@H](NC(=O)c2ccc3c(c2F)OCC32CCN(C3CC4(CCN(c5ccc([C@@H]6c7ccc(O)cc7CC[C@@H]6c6ccccc6)cc5)CC4)C3)CC2)C(=O)N1	C48H51FN4O5	ERα	P03372	CRBN	WO-2024240268-A1
TPD-ITNZUV	WO2024240268A1_ER-P-38	.	O=C1CC[C@H](NC(=O)c2ccc3c(c2F)OCC32CCN(C3CCC4(CC3)CN(c3ccc([C@@H]5c6ccc(O)cc6CC[C@@H]5c5ccccc5)cc3)C4)CC2)C(=O)N1	C48H51FN4O5	ERα	P03372	CRBN	WO-2024240268-A1
TPD-02LF4N	WO2024240268A1_ER-P-39	.	O=C1CC[C@H](NC(=O)c2ccc3c(c2F)OCC32CCN(C3CCC4(CC3)CCN(c3ccc([C@@H]5c6ccc(O)cc6CC[C@@H]5c5ccccc5)cc3)CC4)CC2)C(=O)N1	C50H55FN4O5	ERα	P03372	CRBN	WO-2024240268-A1
TPD-SHBHAG	WO2024240268A1_ER-P-4	.	O=C1CCC(N2Cc3c(ccc4c3OCC43CCC4(CC3)CN(C(=O)C3CCN(c5ccc([C@@H]6c7ccc(O)cc7CC[C@@H]6c6ccccc6)cc5)CC3)C4)C2=O)C(=O)N1	C50H52N4O6	ERα	P03372	CRBN	WO-2024240268-A1
TPD-J0JWPM	WO2024240268A1_ER-P-40	.	CN(C(=O)CN1CCC2(CC1)COc1c2ccc(F)c1C(=O)N[C@H]1CCC(=O)NC1=O)C1CCC2(CC1)CN(c1ccc([C@@H]3c4ccc(O)cc4CC[C@@H]3c3ccccc3)cc1)C2	C51H56FN5O6	ERα	P03372	CRBN	WO-2024240268-A1
TPD-B0ZBVP	WO2024240268A1_ER-P-41	.	O=C1CCC(Nc2ccc3c(c2)OCC2(CCN(C[C@H]4CC[C@@H](OC5CCN(c6ccc([C@@H]7c8ccc(O)cc8CC[C@@H]7c7ccccc7)cc6)CC5)CC4)CC2)C3)C(=O)N1	C52H62N4O5	ERα	P03372	CRBN	WO-2024240268-A1
TPD-KSXJBC	WO2024240268A1_ER-P-42	.	O=C1CC[C@H](NC(=O)c2ccc3c(c2F)OCC32CCN(CC3CCN(c4ccc([C@@H]5c6ccc(O)cc6CC[C@@H]5c5ccccc5)cc4)CC3)CC2)C(=O)N1	C46H49FN4O5	ERα	P03372	CRBN	WO-2024240268-A1
TPD-KUHSMY	WO2024240268A1_ER-P-43	.	O=C1CCC(Nc2ccc3c(c2)OC2(CC3)CCN(C[C@H]3CC[C@@H](OC4CCN(c5ccc([C@@H]6c7ccc(O)cc7CC[C@@H]6c6ccccc6)cc5)CC4)CC3)CC2)C(=O)N1	C52H62N4O5	ERα	P03372	CRBN	WO-2024240268-A1
TPD-EHULFJ	WO2024240268A1_ER-P-45	.	O=C1CC[C@H](NC(=O)c2ccc3c(c2)OCC[C@H]2CN(CC4CCC(OC5CCN(c6ccc([C@@H]7c8ccc(O)cc8CC[C@@H]7c7ccccc7)cc6)CC5)CC4)CCN32)C(=O)N1	C52H61N5O6	ERα	P03372	CRBN	WO-2024240268-A1
TPD-0XLKDI	WO2024240268A1_ER-P-46	.	COc1cc2c(cc1C(=O)N[C@H]1CCC(=O)NC1=O)OCC[C@H]1CN(C[C@H]3CC[C@@H](OC4CCN(c5ccc([C@@H]6c7ccc(O)cc7CC[C@@H]6c6ccccc6)cc5)CC4)CC3)CCN21	C53H63N5O7	ERα	P03372	CRBN	WO-2024240268-A1
TPD-95O9NI	WO2024240268A1_ER-P-47	.	O=C1CC[C@H](NC(=O)c2ccc3c(c2)OC[C@@H]2CN(C[C@H]4CC[C@@H](OC5CCN(c6ccc([C@@H]7c8ccc(O)cc8CC[C@@H]7c7ccccc7)cc6)CC5)CC4)CCN32)C(=O)N1	C51H59N5O6	ERα	P03372	CRBN	WO-2024240268-A1
TPD-BP5JK0	WO2024240268A1_ER-P-48	.	COc1c(C(=O)N[C@H]2CCC(=O)NC2=O)ccc2c1OC[C@H]1CN(C[C@H]3CC[C@@H](OC4CCN(c5ccc([C@@H]6c7ccc(O)cc7CC[C@@H]6c6ccccc6)cc5)CC4)CC3)CCN21	C52H61N5O7	ERα	P03372	CRBN	WO-2024240268-A1
TPD-UHT665	WO2024240268A1_ER-P-49	.	COc1cc2c(cc1C(=O)N[C@H]1CCC(=O)NC1=O)N(C)C[C@H]1CN(C[C@H]3CC[C@@H](OC4CCN(c5ccc([C@@H]6c7ccc(O)cc7CC[C@@H]6c6ccccc6)cc5)CC4)CC3)CCN21	C53H64N6O6	ERα	P03372	CRBN	WO-2024240268-A1
TPD-1SLO08	WO2024240268A1_ER-P-5	.	O=C1CCC(N2Cc3c(ccc4c3OCC43CCC4(CCN(C5CCN(C(=O)C6CCN(c7ccc([C@@H]8c9ccc(O)cc9CC[C@@H]8c8ccccc8)cc7)CC6)CC5)CC4)CC3)C2=O)C(=O)N1	C57H65N5O6	ERα	P03372	CRBN	WO-2024240268-A1
TPD-N0RZCW	WO2024240268A1_ER-P-50	.	O=C1CCC(Nc2ccc3c(c2)COC[C@H]2CN(CC4CCC(OC5CCN(c6ccc([C@@H]7c8ccc(O)cc8CC[C@@H]7c7ccccc7)cc6)CC5)CC4)CCN32)C(=O)N1	C51H61N5O5	ERα	P03372	CRBN	WO-2024240268-A1
TPD-LPHFME	WO2024240268A1_ER-P-52	.	CN(c1ccc2c(c1)COC[C@H]1CN(CC3CCC(OC4CCN(c5ccc([C@@H]6c7ccc(O)cc7CC[C@@H]6c6ccccc6)cc5)CC4)CC3)CCN21)C1CCC(=O)NC1=O	C52H63N5O5	ERα	P03372	CRBN	WO-2024240268-A1
TPD-H8PVB3	WO2024240268A1_ER-P-54	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2ccc3c(c21)OCC31CCN(C[C@H]2CC[C@@H](OC3CCN(c4ccc([C@@H]5c6ccc(O)cc6CC[C@@H]5c5ccccc5)cc4)CC3)CC2)CC1	C53H61N5O6	ERα	P03372	CRBN	WO-2024240268-A1
TPD-4QWL6Z	WO2024240268A1_ER-P-55	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cc3c(cc21)C1(CCN(C[C@H]2CC[C@@H](OC4CCN(c5ccc([C@@H]6c7ccc(O)cc7CC[C@@H]6c6ccccc6)cc5)CC4)CC2)CC1)CO3	C53H61N5O6	ERα	P03372	CRBN	WO-2024240268-A1
TPD-LVHC1P	WO2024240268A1_ER-P-56	.	O=C1CCC(n2c(=O)n3c4c(cccc42)N(C[C@H]2CC[C@@H](OC4CCN(c5ccc([C@@H]6c7ccc(O)cc7CC[C@@H]6c6ccccc6)cc5)CC4)CC2)CC3)C(=O)N1	C48H53N5O5	ERα	P03372	CRBN	WO-2024240268-A1
TPD-51P05A	WO2024240268A1_ER-P-57	.	O=C1CCC(N2Cc3c(ccc4c3OCC43CCC4(CCN(C5CCC6(CC5)CCN(c5ccc([C@@H]7c8ccc(O)cc8CC[C@@H]7c7ccccc7)cc5)CC6)CC4)CC3)C2=O)C(=O)N1	C56H64N4O5	ERα	P03372	CRBN	WO-2024240268-A1
TPD-DUZTIF	WO2024240268A1_ER-P-58	.	O=C1CCC(N2Cc3c(ccc4c3OCC43CCC4(CCN(C5CCN(c6ccc([C@@H]7c8ccc(O)cc8CC[C@@H]7c7ccccc7)cc6)CC5)CC4)CC3)C2=O)C(=O)N1	C51H56N4O5	ERα	P03372	CRBN	WO-2024240268-A1
TPD-TH3G0Y	WO2024240268A1_ER-P-59	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cc3c(cc21)C1(CCN(C2CCC4(CC2)CN(c2ccc([C@@H]5c6ccc(O)cc6CC[C@@H]5c5ccccc5)cc2)C4)CC1)CO3	C49H53N5O5	ERα	P03372	CRBN	WO-2024240268-A1
TPD-W5AWLP	WO2024240268A1_ER-P-6	.	O=C1CCC(N2Cc3c(ccc4c3OCC43CCC4(CC3)CN(C3CCN(C(=O)C5CCN(c6ccc([C@@H]7c8ccc(O)cc8CC[C@@H]7c7ccccc7)cc6)CC5)CC3)C4)C2=O)C(=O)N1	C55H61N5O6	ERα	P03372	CRBN	WO-2024240268-A1
TPD-W0JIFG	WO2024240268A1_ER-P-60	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cc3c(cc21)C1(CCN(C2CCC4(CC2)CCN(c2ccc([C@@H]5c6ccc(O)cc6CC[C@@H]5c5ccccc5)cc2)CC4)CC1)CO3	C51H57N5O5	ERα	P03372	CRBN	WO-2024240268-A1
TPD-J3IPRA	WO2024240268A1_ER-P-61	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cc3c(cc21)C1(CCN(CC2CCC4(CC2)CN(c2ccc([C@@H]5c6ccc(O)cc6CC[C@@H]5c5ccccc5)cc2)C4)CC1)CO3	C50H55N5O5	ERα	P03372	CRBN	WO-2024240268-A1
TPD-COJFOW	WO2024240268A1_ER-P-62	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cc3c(cc21)C1(CCN(CC2CCC4(CC2)CCN(c2ccc([C@@H]5c6ccc(O)cc6CC[C@@H]5c5ccccc5)cc2)CC4)CC1)CO3	C52H59N5O5	ERα	P03372	CRBN	WO-2024240268-A1
TPD-6ROAYD	WO2024240268A1_ER-P-63	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2ccc3c(c21)OCC31CCN(CC2CCN(C(=O)C3CCN(c4ccc([C@@H]5c6ccc(O)cc6CC[C@@H]5c5ccccc5)cc4)CC3)CC2)CC1	C53H60N6O6	ERα	P03372	CRBN	WO-2024240268-A1
TPD-CQNERX	WO2024240268A1_ER-P-64	.	CN(C(=O)CN1CCC2(CC1)COc1c2ccc2c1n(C)c(=O)n2C1CCC(=O)NC1=O)C1CCC2(CC1)CN(c1ccc([C@@H]3c4ccc(O)cc4CC[C@@H]3c3ccccc3)cc1)C2	C52H58N6O6	ERα	P03372	CRBN	WO-2024240268-A1
TPD-ES3Z8O	WO2024240268A1_ER-P-65	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cc3c(cc21)OC1(CC3)CCN(C[C@H]2CC[C@@H](OC3CCN(c4ccc([C@@H]5c6ccc(O)cc6CC[C@@H]5c5ccccc5)cc4)CC3)CC2)CC1	C54H63N5O6	ERα	P03372	CRBN	WO-2024240268-A1
TPD-BU5CZ2	WO2024240268A1_ER-P-66	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2ccc3c(c21)C1(CCN(C[C@H]2CC[C@@H](OC4CCN(c5ccc([C@@H]6c7ccc(O)cc7CC[C@@H]6c6ccccc6)cc5)CC4)CC2)CC1)CO3	C53H61N5O6	ERα	P03372	CRBN	WO-2024240268-A1
TPD-F90WW8	WO2024240268A1_ER-P-67	.	O=C1CC[C@H](NC(=O)c2cc3c(cc2F)N2CCN(C[C@H]4CC[C@@H](OC5CCN(c6ccc([C@@H]7c8ccc(O)cc8CC[C@@H]7c7ccccc7)cc6)CC5)CC4)C[C@@H]2CO3)C(=O)N1	C51H58FN5O6	ERα	P03372	CRBN	WO-2024240268-A1
TPD-WFO22E	WO2024240268A1_ER-P-68	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2ccc3c(c21)OCC31CCN(C(=O)CN2CCC3(CCN(c4ccc([C@@H]5c6ccc(O)cc6CC[C@@H]5c5ccccc5)cc4)CC3)C2)CC1	C51H56N6O6	ERα	P03372	CRBN	WO-2024240268-A1
TPD-BYKV5F	WO2024240268A1_ER-P-69	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cc3c(cc21)C1(CCN(C(=O)CN2CCC4(CCN(c5ccc([C@@H]6c7ccc(O)cc7CC[C@@H]6c6ccccc6)cc5)CC4)C2)CC1)CO3	C51H56N6O6	ERα	P03372	CRBN	WO-2024240268-A1
TPD-I5YGP3	WO2024240268A1_ER-P-7	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2ccc3c(c21)C1(CCN(C(=O)[C@H]2CC[C@H](CN4CCN(c5ccc([C@@H]6c7ccc(O)cc7CC[C@@H]6c6ccccc6)cc5)CC4)CC2)CC1)CO3	C53H60N6O6	ERα	P03372	CRBN	WO-2024240268-A1
TPD-PSUJ02	WO2024240268A1_ER-P-70	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2ccc3c(c21)OCC31CCN(C2CCN(C3CCN(c4ccc([C@@H]5c6ccc(O)cc6CC[C@@H]5c5ccccc5)cc4)CC3)CC2)CC1	C51H58N6O5	ERα	P03372	CRBN	WO-2024240268-A1
TPD-0R289H	WO2024240268A1_ER-P-71	.	CN(CC(=O)N1CCC2(CC1)CCC1(CC2)COc2c1ccc1c2CN(C2CCC(=O)NC2=O)C1=O)C1CCC2(CC1)CN(c1ccc([C@@H]3c4ccc(O)cc4CC[C@@H]3c3ccccc3)cc1)C2	C57H65N5O6	ERα	P03372	CRBN	WO-2024240268-A1
TPD-4YPGT6	WO2024240268A1_ER-P-72	.	CN(CC(=O)N1CC2(CCC3(CC2)COc2c3ccc3c2CN(C2CCC(=O)NC2=O)C3=O)C1)C1CCC2(CC1)CN(c1ccc([C@@H]3c4ccc(O)cc4CC[C@@H]3c3ccccc3)cc1)C2	C55H61N5O6	ERα	P03372	CRBN	WO-2024240268-A1
TPD-IM5D1N	WO2024240268A1_ER-P-73	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2ccc3c(c21)OCC31CCN(CC2CCN(c3ccc([C@@H]4c5ccc(O)cc5CC[C@@H]4c4ccccc4)cc3)CC2)CC1	C47H51N5O5	ERα	P03372	CRBN	WO-2024240268-A1
TPD-Q27UQM	WO2024240268A1_ER-P-74	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2ccc3c(c21)OCC31CCN(C(=O)C2CCN(CC3CCN(c4ccc([C@@H]5c6ccc(O)cc6CC[C@@H]5c5ccccc5)cc4)CC3)CC2)CC1	C53H60N6O6	ERα	P03372	CRBN	WO-2024240268-A1
TPD-JOM7YL	WO2024240268A1_ER-P-75	.	CN(CC(=O)N1CCC2(CC1)COc1c2ccc2c1n(C)c(=O)n2C1CCC(=O)NC1=O)CC1CCN(c2ccc([C@@H]3c4ccc(O)cc4CC[C@@H]3c3ccccc3)cc2)CC1	C50H56N6O6	ERα	P03372	CRBN	WO-2024240268-A1
TPD-AGJ5HA	WO2024240268A1_ER-P-76	.	O=C1CCC(N2Cc3c(ccc4c3OCC43CCC4(CCN(C(=O)C5CCN(c6ccc([C@@H]7c8ccc(O)cc8CC[C@@H]7c7ccccc7)cc6)CC5)CC4)CC3)C2=O)C(=O)N1	C52H56N4O6	ERα	P03372	CRBN	WO-2024240268-A1
TPD-XUZH8E	WO2024240268A1_ER-P-77	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2ccc3c(c21)C1(CCN(C2CCN(C(=O)C4CCN(c5ccc([C@@H]6c7ccc(O)cc7CC[C@@H]6c6ccccc6)cc5)CC4)CC2)CC1)CO3	C52H58N6O6	ERα	P03372	CRBN	WO-2024240268-A1
TPD-AUKHEE	WO2024240268A1_ER-P-78	.	O=C1CCC(N2Cc3c(ccc4c3OCC43CCC4(CC3)CN(C[C@H]3CC[C@@H](OC5CCN(c6ccc([C@@H]7c8ccc(O)cc8CC[C@@H]7c7ccccc7)cc6)CC5)CC3)C4)C2=O)C(=O)N1	C56H64N4O6	ERα	P03372	CRBN	WO-2024240268-A1
TPD-9WXTDA	WO2024240268A1_ER-P-79	.	O=C1CCC(N2Cc3c(ccc4c3OCC43CCC4(CCN(C[C@H]5CC[C@@H](OC6CCN(c7ccc([C@@H]8c9ccc(O)cc9CC[C@@H]8c8ccccc8)cc7)CC6)CC5)CC4)CC3)C2=O)C(=O)N1	C58H68N4O6	ERα	P03372	CRBN	WO-2024240268-A1
TPD-YWEZCP	WO2024240268A1_ER-P-8	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2ccc3c(c21)OCC31CCN(C2CCN(C3CC4(CCN(c5ccc([C@@H]6c7ccc(O)cc7CC[C@@H]6c6ccccc6)cc5)CC4)C3)C[C@@H]2F)CC1	C54H61FN6O5	ERα	P03372	CRBN	WO-2024240268-A1
TPD-R3BBIN	WO2024240268A1_ER-P-80	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2ccc3c(c21)OCC31CCN(C[C@H]2C[C@@H](OC3CCN(c4ccc([C@@H]5c6ccc(O)cc6CC[C@@H]5c5ccccc5)cc4)CC3)C2)CC1	C51H57N5O6	ERα	P03372	CRBN	WO-2024240268-A1
TPD-OHQ2DX	WO2024240268A1_ER-P-81	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cc3c(cc21)OC1(CC3)CCN(C[C@H]2C[C@@H](OC3CCN(c4ccc([C@@H]5c6ccc(O)cc6CC[C@@H]5c5ccccc5)cc4)CC3)C2)CC1	C52H59N5O6	ERα	P03372	CRBN	WO-2024240268-A1
TPD-4ETDNI	WO2024240268A1_ER-P-82	.	O=C1CC[C@H](NC(=O)c2ccc3c(c2F)OCC32CCN(C[C@H]3CC[C@@H](OC4CCN(c5ccc([C@@H]6c7ccc(O)cc7CC[C@@H]6c6ccccc6)cc5)CC4)CC3)CC2)C(=O)N1	C52H59FN4O6	ERα	P03372	CRBN	WO-2024240268-A1
TPD-N50SO4	WO2024240268A1_ER-P-83	.	O=C1CC[C@H](NC(=O)c2cc3c(cc2F)OCC32CCN(C[C@H]3CC[C@@H](OC4CCN(c5ccc([C@@H]6c7ccc(O)cc7CC[C@@H]6c6ccccc6)cc5)CC4)CC3)CC2)C(=O)N1	C52H59FN4O6	ERα	P03372	CRBN	WO-2024240268-A1
TPD-AG7N90	WO2024240268A1_ER-P-84	.	COc1cc2c(cc1C(=O)N[C@H]1CCC(=O)NC1=O)OCC21CCN(C[C@H]2CC[C@@H](OC3CCN(c4ccc([C@@H]5c6ccc(O)cc6CC[C@@H]5c5ccccc5)cc4)CC3)CC2)CC1	C53H62N4O7	ERα	P03372	CRBN	WO-2024240268-A1
TPD-T1OT9X	WO2024240268A1_ER-P-85	.	O=C1CC[C@H](NC(=O)c2cc3c(cc2F)CCC2(CN(C[C@H]4CC[C@@H](OC5CCN(c6ccc([C@@H]7c8ccc(O)cc8CC[C@@H]7c7ccccc7)cc6)CC5)CC4)C2)O3)C(=O)N1	C51H57FN4O6	ERα	P03372	CRBN	WO-2024240268-A1
TPD-QL7V2P	WO2024240268A1_ER-P-86	.	O=C1CC[C@H](NC(=O)c2c(F)ccc3c2OCC32CCN(C[C@H]3CC[C@@H](OC4CCN(c5ccc([C@@H]6c7ccc(O)cc7CC[C@@H]6c6ccccc6)cc5)CC4)CC3)CC2)C(=O)N1	C52H59FN4O6	ERα	P03372	CRBN	WO-2024240268-A1
TPD-GHL25W	WO2024240268A1_ER-P-87	.	O=C1CC[C@H](NC(=O)c2cc3c(cc2F)C2(CCN(C[C@H]4CC[C@@H](OC5CCN(c6ccc([C@@H]7c8ccc(O)cc8CC[C@@H]7c7ccccc7)cc6)CC5)CC4)CC2)CO3)C(=O)N1	C52H59FN4O6	ERα	P03372	CRBN	WO-2024240268-A1
TPD-C6YOD9	WO2024240268A1_ER-P-88	.	COc1cc2c(cc1C(=O)N[C@H]1CCC(=O)NC1=O)CCC1(CCN(C[C@H]3CC[C@@H](OC4CCN(c5ccc([C@@H]6c7ccc(O)cc7CC[C@@H]6c6ccccc6)cc5)CC4)CC3)CC1)O2	C54H64N4O7	ERα	P03372	CRBN	WO-2024240268-A1
TPD-TTNRSF	WO2024240268A1_ER-P-89	.	O=C1CC[C@H](NC(=O)c2cc3c(cc2F)OC2(CC3)CCN(C[C@H]3CC[C@@H](OC4CCN(c5ccc([C@@H]6c7ccc(O)cc7CC[C@@H]6c6ccccc6)cc5)CC4)CC3)CC2)C(=O)N1	C53H61FN4O6	ERα	P03372	CRBN	WO-2024240268-A1
TPD-T55BEX	WO2024240268A1_ER-P-9	.	O=C1NC(O)CCC1N1Cc2c(ccc3c2OCC32CCC3(CC2)CN(C2CCC4(CC2)CCN(c2ccc([C@@H]5c6ccc(O)cc6CC[C@@H]5c5ccccc5)cc2)CC4)C3)C1=O	C54H62N4O5	ERα	P03372	CRBN	WO-2024240268-A1
TPD-HORUQ7	WO2024240268A1_ER-P-90	.	O=C1CC[C@H](NC(=O)c2cc3c(cc2F)CCC2(CCN(C[C@H]4CC[C@@H](OC5CCN(c6ccc([C@@H]7c8ccc(O)cc8CC[C@@H]7c7ccccc7)cc6)CC5)CC4)CC2)O3)C(=O)N1	C53H61FN4O6	ERα	P03372	CRBN	WO-2024240268-A1
TPD-HE8VL9	WO2024240268A1_ER-P-91	.	COc1cc2c(cc1C(=O)N[C@H]1CCC(=O)NC1=O)C1(CCN(C[C@H]3CC[C@@H](OC4CCN(c5ccc([C@@H]6c7ccc(O)cc7CC[C@@H]6c6ccccc6)cc5)CC4)CC3)CC1)CO2	C53H62N4O7	ERα	P03372	CRBN	WO-2024240268-A1
TPD-CUVUAV	WO2024240268A1_ER-P-92	.	O=C1CCC(Nc2ccc3c(c2)OCC32CCN(C[C@H]3C[C@@H](OC4CCN(c5ccc([C@@H]6c7ccc(O)cc7CC[C@@H]6c6ccccc6)cc5)CC4)C3)CC2)C(=O)N1	C49H56N4O5	ERα	P03372	CRBN	WO-2024240268-A1
TPD-9JUTQL	WO2024240268A1_SM-P-1	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cc3c(cc21)OC1(CC3)CCN(C2CC3(CCC(C#Cc4cc(-c5ccccc5O)nnc4N)CC3)C2)CC1	C41H45N7O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024240268-A1
TPD-BXNMB2	WO2024240268A1_SM-P-10	.	COc1cc(N2CCN(C3CC4(CCC(C#Cc5cc(-c6ccccc6O)nnc5N)CC4)C3)CC2)ccc1C(=O)N[C@H]1CCC(=O)NC1=O	C38H43N7O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024240268-A1
TPD-8E0AXW	WO2024240268A1_SM-P-11	.	COc1cc2c(cc1C(=O)N[C@H]1CCC(=O)NC1=O)OCC[C@H]1CN(C3CC4(CCC(C#Cc5cc(-c6ccccc6O)nnc5N)CC4)C3)CCN21	C40H45N7O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024240268-A1
TPD-II2ACF	WO2024240268A1_SM-P-12	.	Nc1nnc(-c2ccccc2O)cc1C#CC1CCC2(CC1)CC(N1CCC3(CCc4cc(F)c(C(=O)N[C@H]5CCC(=O)NC5=O)cc4O3)CC1)C2	C40H43FN6O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024240268-A1
TPD-X7IR5Q	WO2024240268A1_SM-P-13	.	Nc1nnc(-c2ccccc2O)cc1C#CC1CCC2(CC1)CC(N1CCN3c4ccc(C(=O)N[C@H]5CCC(=O)NC5=O)cc4OCC[C@H]3C1)C2	C39H43N7O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024240268-A1
TPD-NX3I36	WO2024240268A1_SM-P-14	.	COc1cc2c(cc1C(=O)N[C@H]1CCC(=O)NC1=O)C1(CCN(C3CC4(CCC(C#Cc5cc(-c6ccccc6O)nnc5N)CC4)C3)CC1)CO2	C40H44N6O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024240268-A1
TPD-3W86DZ	WO2024240268A1_SM-P-15	.	COc1c(C(=O)N[C@H]2CCC(=O)NC2=O)ccc2c1OC[C@H]1CN(C3CC4(CCC(C#Cc5cc(-c6ccccc6O)nnc5N)CC4)C3)CCN21	C39H43N7O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024240268-A1
TPD-DJILN0	WO2024240268A1_SM-P-16	.	Nc1nnc(-c2ccccc2O)cc1C#CC1CCC2(CC1)CC(N1CCC3(CC1)COc1c3ccc(C(=O)N[C@H]3CCC(=O)NC3=O)c1F)C2	C39H41FN6O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024240268-A1
TPD-QW4DKZ	WO2024240268A1_SM-P-17	.	Nc1nnc(-c2ccccc2O)cc1C#CC1CCC2(CC1)CC(N1CCN3c4cc(NC5CCC(=O)NC5=O)ccc4OCC[C@H]3C1)C2	C38H43N7O4	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024240268-A1
TPD-OA1U8M	WO2024240268A1_SM-P-18	.	CN(C(=O)c1ccc2c(c1)OC[C@H]1CN(C3CC4(CCC(C#Cc5cc(-c6ccccc6O)nnc5N)CC4)C3)CCN21)[C@H]1CCC(=O)NC1=O	C39H43N7O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024240268-A1
TPD-QY6361	WO2024240268A1_SM-P-19	.	Nc1nnc(-c2ccccc2O)cc1C#CC1CCC2(CC1)CC(N1CCC3(CC1)COc1c3ccc(F)c1C(=O)N[C@H]1CCC(=O)NC1=O)C2	C39H41FN6O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024240268-A1
TPD-6AK343	WO2024240268A1_SM-P-2	.	Nc1nnc(-c2ccccc2O)cc1C#CC1CCC2(CC1)CC(N1CCC3(CC1)CCC1(CC3)COc3c1ccc1c3CN(C3CCC(=O)NC3=O)C1=O)C2	C45H50N6O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024240268-A1
TPD-XFWYLA	WO2024240268A1_SM-P-20	.	Nc1nnc(-c2ccccc2O)cc1C#CC1CCC2(CC1)CC(N1CCN3c4ccc(C(=O)N[C@H]5CCC(=O)NC5=O)cc4OC[C@@H]3C1)C2	C38H41N7O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024240268-A1
TPD-VG7RQM	WO2024240268A1_SM-P-21	.	Nc1nnc(-c2ccccc2O)cc1C#CC1CCC2(CC1)CC(N1CCC3(CC1)COc1cc(F)c(C(=O)N[C@H]4CCC(=O)NC4=O)cc13)C2	C39H41FN6O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024240268-A1
TPD-AGIIKO	WO2024240268A1_SM-P-22	.	Nc1nnc(-c2ccccc2O)cc1C#CC1CCC2(CC1)CC(N1CCN3c4ccc(C(=O)N[C@H]5CCC(=O)NC5=O)c(F)c4OC[C@H]3C1)C2	C38H40FN7O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024240268-A1
TPD-0PG7S0	WO2024240268A1_SM-P-23	.	Nc1nnc(-c2ccccc2O)cc1C#CC1CCC2(CC1)CC(N1CCC3(CC1)COc1cc(NC4CCC(=O)NC4=O)ccc1C3)C2	C39H44N6O4	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024240268-A1
TPD-Y7VTIX	WO2024240268A1_SM-P-24	.	Nc1nnc(-c2ccccc2O)cc1C#CC1CCC2(CC1)CC(N1CCC3(CCc4ccc(NC5CCC(=O)NC5=O)cc4O3)CC1)C2	C39H44N6O4	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024240268-A1
TPD-A3VGPO	WO2024240268A1_SM-P-25	.	Nc1nnc(-c2ccccc2O)cc1C#CC1CCC2(CC1)CC(N1CCC3(CC1)Cc1ccc(NC4CCC(=O)NC4=O)cc1O3)C2	C38H42N6O4	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024240268-A1
TPD-KNVIIL	WO2024240268A1_SM-P-26	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2ccc3c(c21)OCC31CCN(C2CC3(CCC(C#Cc4cc(-c5ccccc5O)nnc4N)CC3)C2)CC1	C40H43N7O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024240268-A1
TPD-WM6QGA	WO2024240268A1_SM-P-27	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2ccc3c(c21)OCC31CCN(C(=O)[C@H]2CC[C@H](Cn3cc(-c4cc(-c5ccccc5O)nnc4N)cn3)CC2)CC1	C40H43N9O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024240268-A1
TPD-9B0HNK	WO2024240268A1_SM-P-28	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cc3c(cc21)C1(CCN(C(=O)[C@H]2CC[C@H](Cn4cc(-c5cc(-c6ccccc6O)nnc5N)cn4)CC2)CC1)CO3	C40H43N9O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024240268-A1
TPD-XZ4BQZ	WO2024240268A1_SM-P-29	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2ccc3c(c21)OCC31CCN(C[C@H]2CC[C@H](Cn3cc(-c4cc(-c5ccccc5O)nnc4N)cn3)CC2)CC1	C40H45N9O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024240268-A1
TPD-LVUGMB	WO2024240268A1_SM-P-3	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2ccc3c(c21)C1(CCN(C2CC4(CCC(C#Cc5cc(-c6ccccc6O)nnc5N)CC4)C2)CC1)CO3	C40H43N7O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024240268-A1
TPD-KF32DE	WO2024240268A1_SM-P-30	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cc3c(cc21)C1(CCN(C[C@H]2CC[C@H](Cn4cc(-c5cc(-c6ccccc6O)nnc5N)cn4)CC2)CC1)CO3	C40H45N9O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024240268-A1
TPD-F7EUUB	WO2024240268A1_SM-P-31	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2ccc3c(c21)OCC31CCN(C(=O)[C@H]2CC[C@H](n3cc(-c4cc(-c5ccccc5O)nnc4N)cn3)CC2)CC1	C39H41N9O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024240268-A1
TPD-9VWF25	WO2024240268A1_SM-P-32	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2ccc3c(c21)OCC31CCN(C2CCN(C(=O)[C@H]3CC[C@H](n4cc(-c5cc(-c6ccccc6O)nnc5N)cn4)CC3)CC2)CC1	C44H50N10O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024240268-A1
TPD-9CWZDL	WO2024240268A1_SM-P-33	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cc3c(cc21)C1(CCN(C(=O)[C@H]2CC[C@H](n4cc(-c5cc(-c6ccccc6O)nnc5N)cn4)CC2)CC1)CO3	C39H41N9O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024240268-A1
TPD-2RZ30Q	WO2024240268A1_SM-P-34	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cc3c(cc21)C1(CCN(C2CCN(C(=O)[C@H]4CC[C@H](n5cc(-c6cc(-c7ccccc7O)nnc6N)cn5)CC4)CC2)CC1)CO3	C44H50N10O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024240268-A1
TPD-9HPNJ4	WO2024240268A1_SM-P-35	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2ccc3c(c21)OCC31CCN(C[C@H]2CC[C@H](n3cc(-c4cc(-c5ccccc5O)nnc4N)cn3)CC2)CC1	C39H43N9O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024240268-A1
TPD-0GR38M	WO2024240268A1_SM-P-36	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cc3c(cc21)C1(CCN(C[C@H]2CC[C@H](n4cc(-c5cc(-c6ccccc6O)nnc5N)cn4)CC2)CC1)CO3	C39H43N9O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024240268-A1
TPD-5ET94M	WO2024240268A1_SM-P-37	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2ccc3c(c21)OCC31CCN(C2CN(c3cc(-c4ccccc4O)nnc3N)C2)CC1	C32H34N8O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024240268-A1
TPD-RR0X9K	WO2024240268A1_SM-P-38	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cc3c(cc21)C1(CCN(C2CN(c4cc(-c5ccccc5O)nnc4N)C2)CC1)CO3	C32H34N8O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024240268-A1
TPD-ZDKK01	WO2024240268A1_SM-P-4	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cc3c(cc21)C1(CCN(C2CC4(CCC(C#Cc5cc(-c6ccccc6O)nnc5N)CC4)C2)CC1)CO3	C40H43N7O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024240268-A1
TPD-3S9IT6	WO2024240268A1_SM-P-5	.	Nc1nnc(-c2ccccc2O)cc1C#CC1CCC2(CC1)CC(N1CCN3c4ccc(NC5CCC(=O)NC5=O)cc4OCC[C@H]3C1)C2	C38H43N7O4	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024240268-A1
TPD-D6B4MJ	WO2024240268A1_SM-P-6	.	Nc1nnc(-c2ccccc2O)cc1C#CC1CCC2(CC1)CC(N1CCN3c4cc(F)c(C(=O)N[C@H]5CCC(=O)NC5=O)cc4OC[C@H]3C1)C2	C38H40FN7O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024240268-A1
TPD-XOCOG4	WO2024240268A1_SM-P-7	.	Nc1nnc(-c2ccccc2O)cc1C#CC1CCC2(CC1)CC(N1CCC3(CCc4cc(C(=O)N[C@H]5CCC(=O)NC5=O)c(F)cc4O3)CC1)C2	C40H43FN6O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024240268-A1
TPD-KX9MET	WO2024240268A1_SM-P-8	.	Nc1nnc(-c2ccccc2O)cc1C#CC1CCC2(CC1)CC(N1CCC3(CC1)COc1cc(C(=O)N[C@H]4CCC(=O)NC4=O)c(F)cc13)C2	C39H41FN6O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024240268-A1
TPD-PYB6UH	WO2024240268A1_SM-P-9	.	Nc1nnc(-c2ccccc2O)cc1C#CC1CCC2(CC1)CC(N1CC3(CCc4cc(F)c(C(=O)N[C@H]5CCC(=O)NC5=O)cc4O3)C1)C2	C38H39FN6O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2024240268-A1
TPD-D7MP6X	SCHEMBL31232461	2-[2-[2-[2-[2-[2-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperazin-1-yl]ethoxy]ethoxy]ethoxymethyl]-3-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]-2-methylpropoxy]ethoxy]ethoxy]ethyl 2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetate	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCC(C)(COCCOCCOCCOC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)COCCOCCOCCN2CCN(c3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)C(C)(C)C)cc1	C77H97ClN12O17S2	BRD2;BRD3	P25440/Q15059	VHL	WO-2024241046-A1
TPD-9S08G9	SCHEMBL31232504	2-[2-[2-[2-[2-[2-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]ethoxy]ethoxy]ethoxymethyl]-3-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]-2-methylpropoxy]ethoxy]ethoxy]ethyl 2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetate	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCC(C)(COCCOCCOCCOC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)COCCOCCOCCN2CCN(c3cc4c(cc3F)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)C(C)(C)C)cc1	C77H96ClFN12O17S2	BRD2;BRD3	P25440/Q15059	VHL	WO-2024241046-A1
TPD-G6GT0I	SCHEMBL31232372	2-[2-[2-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxymethyl]-3-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]-2-methylpropoxy]ethoxy]ethoxy]ethyl 2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetate	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCC(C)(COCCOCCOCCNc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)COCCOCCOCCOC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)C(C)(C)C)cc1	C73H90ClN11O17S2	BRD2;BRD3	P25440/Q15059	VHL	WO-2024241046-A1
TPD-OIT9CX	SCHEMBL31232445	2-[2-[2-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]amino]ethoxy]ethoxy]ethoxymethyl]-3-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]-2-methylpropoxy]ethoxy]ethoxy]ethyl 2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetate	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCC(C)(COCCOCCOCCNc2cc3c(cc2F)C(=O)N(C2CCC(=O)NC2=O)C3=O)COCCOCCOCCOC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)C(C)(C)C)cc1	C73H89ClFN11O17S2	BRD2;BRD3	P25440/Q15059	VHL	WO-2024241046-A1
TPD-UW0529	WO2024241046A1_AB3064	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCC(C)(COCCOCCOCCNc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)COCCOCCOC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)C(C)(C)C)cc1	C71H86ClN11O16S2	BRD2;BRD3	P25440/Q15059	VHL	WO-2024241046-A1
TPD-EHRTPE	WO2024241046A1_AB3065	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCC(C)(COCCOCCOCCNc2cc3c(cc2F)C(=O)N(C2CCC(=O)NC2=O)C3=O)COCCOCCOC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)C(C)(C)C)cc1	C71H85ClFN11O16S2	BRD2;BRD3	P25440/Q15059	VHL	WO-2024241046-A1
TPD-NQJU0G	SCHEMBL31232498	2-[2-[2-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxymethyl]-3-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]-2-methylpropoxy]ethoxy]ethoxy]ethyl 2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetate	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCC(C)(COCCOCCOCCNc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)COCCOCCOCCOC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)C(C)(C)C)cc1	C74H92ClN11O17S2	BRD2;BRD3	P25440/Q15059	VHL	WO-2024241046-A1
TPD-TG0UGL	orb2945747	2-[2-[2-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]amino]ethoxy]ethoxy]ethoxymethyl]-3-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]-2-methylpropoxy]ethoxy]ethoxy]ethyl 2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetate; SCHEMBL31232422; HY-170390	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCC(C)(COCCOCCOCCNc2cc3c(cc2F)C(=O)N(C2CCC(=O)NC2=O)C3=O)COCCOCCOCCOC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)C(C)(C)C)cc1	C74H91ClFN11O17S2	BRD2;BRD3	P25440/Q15059	VHL	WO-2024241046-A1
TPD-TFU3O9	WO2024241046A1_AB3124	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCC(COCCOCCOCCNc2cc3c(cc2F)C(=O)N(C2CCC(=O)NC2=O)C3=O)(COCCOCCOCCOC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)COCCOCCOCCOC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)C(C)(C)C)cc1	C98H116Cl2FN15O22S3	BRD2;BRD3	P25440/Q15059	VHL	WO-2024241046-A1
TPD-8VXCBE	WO2024241046A1_AB3125	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCC(C)(COCCOCCNc2cc3c(cc2F)C(=O)N(C2CCC(=O)NC2=O)C3=O)COCCOCCOC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)C(C)(C)C)cc1	C70H83ClFN11O15S2	BRD2;BRD3	P25440/Q15059	VHL	WO-2024241046-A1
TPD-PDQYHZ	WO2024241046A1_AB3126	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCC(C)(COCCOCCNc2cc3c(cc2F)C(=O)N(C2CCC(=O)NC2=O)C3=O)COCCOCCOCCOC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)C(C)(C)C)cc1	C72H87ClFN11O16S2	BRD2;BRD3	P25440/Q15059	VHL	WO-2024241046-A1
TPD-JOKTIJ	SCHEMBL31232349	2-[2-[2-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]amino]ethoxy]ethoxy]ethoxymethyl]-3-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]-2-methylpropoxy]ethoxy]ethoxy]ethyl (2R)-2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]butanoate	CC[C@@H](C(=O)OCCOCCOCCOCC(C)(COCCOCCOCCNc1cc2c(cc1F)C(=O)N(C1CCC(=O)NC1=O)C2=O)COCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)c1ccc(-c2scnc2C)cc1)C(C)(C)C)[C@@H]1N=C(c2ccc(Cl)cc2)c2c(sc(C)c2C)-n2c(C)nnc21	C76H95ClFN11O17S2	BRD2;BRD3	P25440/Q15059	VHL	WO-2024241046-A1
TPD-9QQGP7	WO2024241046A1_MN666	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCC(C)(COCCOCCNC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)COCCOCCNc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)C(C)(C)C)cc1	C69H83ClN12O14S2	BRD2;BRD3	P25440/Q15059	VHL	WO-2024241046-A1
TPD-W8B0P5	WO2024241046A1_MN675	.	Cc1ncsc1-c1ccc(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)COCC(C)(COCCOCCOCCNC(=O)C[C@@H]2N=C(c3ccc(Cl)cc3)c3c(sc(C)c3C)-n3c(C)nnc32)COCCOCCOCCNc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)C(C)(C)C)cc1	C73H91ClN12O16S2	BRD2;BRD3	P25440/Q15059	VHL	WO-2024241046-A1
TPD-8TVQX2	WO2024244888A1_1	.	CN1CCN([C@@H]2CCCN(C3=NC(NC4=CC=C(N5CCN(CC6CCN(C7=CC=C(N8CCC(=O)NC8=O)C=C7)CC6)CC5)C=C4)=C4N=CNC4=N3)C2)C1=O	C40H51N13O3	BTK	Q06187	CRBN	WO-2024244888-A1
TPD-ARZGB1	WO2024244888A1_2	1-[2-methyl-4-[4-[[4-[4-[(2-piperidin-1-yl-7H-purin-6-yl)amino]phenyl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]-1,3-diazinane-2,4-dione	CC1=CC(N2CCC(CN3CCN(C4=CC=C(NC5=C6N=CNC6=NC(N6CCCCC6)=N5)C=C4)CC3)CC2)=CC=C1N1CCC(=O)NC1=O	C37H47N11O2	BTK	Q06187	CRBN	WO-2024244888-A1
TPD-N0VVCU	WO2024244888A1_3	1-[2-methyl-4-[4-[[4-[4-[[2-[(3R)-3-(3-methyl-2-oxoimidazolidin-1-yl)piperidin-1-yl]-7H-purin-6-yl]amino]phenyl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]-1,3-diazinane-2,4-dione	CC1=CC(N2CCC(CN3CCN(C4=CC=C(NC5=C6N=CNC6=NC(N6CCC[C@@H](N7CCN(C)C7=O)C6)=N5)C=C4)CC3)CC2)=CC=C1N1CCC(=O)NC1=O	C41H53N13O3	BTK	Q06187	CRBN	WO-2024244888-A1
TPD-JL0SHJ	WO2024244888A1_4	.	CN1CCN([C@@H]2CCCN(C3=CC4=NC=NN4C(NC4=CC=C(N5CCN(CC6CCN(C7=CC=C(N8CCC(=O)NC8=O)C=C7)CC6)CC5)C=C4)=N3)C2)C1=O	C40H51N13O3	BTK	Q06187	CRBN	WO-2024244888-A1
TPD-ZXCKNN	WO2024244888A1_6	1-[4-[4-[[4-[4-[[9-methyl-2-[(3R)-3-(3-methyl-2-oxoimidazolidin-1-yl)piperidin-1-yl]purin-6-yl]amino]phenyl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]-1,3-diazinane-2,4-dione	CN1C=NC2=C(NC3=CC=C(N4CCN(CC5CCN(C6=CC=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)C=C3)N=C(N3CCC[C@@H](N4CCN(C)C4=O)C3)N=C21	C41H53N13O3	BTK	Q06187	CRBN	WO-2024244888-A1
TPD-ANOIP9	WO2024244888A1_7	.	CN1CCN([C@@H]2CCCN(C3=NC(NC4=CC=C(N5CCN(CC6CCN(C7=CC=C(N8CCC(=O)NC8=O)C=C7)CC6)CC5)C=C4)=C4N=CSC4=N3)C2)C1=O	C40H50N12O3S	BTK	Q06187	CRBN	WO-2024244888-A1
TPD-A3ZVGR	WO2024244888A1_8	.	CN1CCN([C@@H]2CCCN(C3=NC(NC4=CC=C(N5CCN(CC6CCN(C7=CC=C(N8CCC(=O)NC8=O)C=C7)CC6)CC5)C=C4)=C4NN=CC4=N3)C2)C1=O	C40H51N13O3	BTK	Q06187	CRBN	WO-2024244888-A1
TPD-AG47Z5	WO2024244888A1_9	1-[4-[4-[[4-[2-fluoro-4-[[2-[(3R)-3-(3-methyl-2-oxoimidazolidin-1-yl)piperidin-1-yl]-7H-purin-6-yl]amino]phenyl]piperazin-1-yl]methyl]piperidin-1-yl]-2-methylphenyl]-1,3-diazinane-2,4-dione	CC1=CC(N2CCC(CN3CCN(C4=CC=C(NC5=C6N=CNC6=NC(N6CCC[C@@H](N7CCN(C)C7=O)C6)=N5)C=C4F)CC3)CC2)=CC=C1N1CCC(=O)NC1=O	C41H52FN13O3	BTK	Q06187	CRBN	WO-2024244888-A1
TPD-4QE74E	WO2024244888A1_10	.	C=C1N(C)CCN1[C@@H]1CCCN(C2=NC(NC3=CC=C(N4CCN(CC5CCN(C6=CC=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)C(F)=C3)=C3N=CCC3=N2)C1	C42H53FN12O2	BTK	Q06187	CRBN	WO-2024244888-A1
TPD-K2GEBV	WO2024245169A1_1	.	CC1(C)CC(=C(c2ccc(N3CCN(CC4CN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)CC3)cc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C44H48FN7O5	ERα	P03372	CRBN	WO-2024245169-A1
TPD-ORH35Y	WO2024245169A1_2	.	CC1(C)CC(=C(c2ccc(N3CCN(C4CN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)CC3)cc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C43H46FN7O5	ERα	P03372	CRBN	WO-2024245169-A1
TPD-72NPI1	WO2024245169A1_3	.	CC1(C)CC(=C(c2ccc3[nH]nc(F)c3c2)c2c(F)cc(N3CCN(C4CN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)CC3)cc2F)CC(C)(C)O1	C43H44F3N7O5	ERα	P03372	CRBN	WO-2024245169-A1
TPD-Y64NZY	WO2024245169A1_4	.	CC1(C)CC(=C(c2ccc(N3CCN(CC4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C45H51FN8O5	ERα	P03372	CRBN	WO-2024245169-A1
TPD-CNANTR	WO2024245169A1_5	.	CC1(C)CC(=C(c2ccc(N3CCC(CN4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)cc2)c2ccc3[nH]ncc3c2)CC(C)(C)O1	C46H53N7O5	ERα	P03372	CRBN	WO-2024245169-A1
TPD-SMIWCX	WO2024245169A1_6	.	CC1(C)CC(=C(c2ccc(N3CCC(CN4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)cc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C46H52FN7O5	ERα	P03372	CRBN	WO-2024245169-A1
TPD-O3VO1B	WO2024245169A1_7	.	CC1(C)CC(=C(c2ccc(OC3CN(CC4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C3)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C44H48FN7O6	ERα	P03372	CRBN	WO-2024245169-A1
TPD-NWMI6I	WO2024245169A1_8	.	CC1(C)CC(=C(c2ccc(OC3CN(CC4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C3)cc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C45H49FN6O6	ERα	P03372	CRBN	WO-2024245169-A1
TPD-HXSC2V	WO2024245169A1_9	.	CC1(C)CC(=C(c2ccc3[nH]nc(F)c3c2)c2c(F)cc(N3CCN(CC4CN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)CC3)cc2F)CC(C)(C)O1	C44H46F3N7O5	ERα	P03372	CRBN	WO-2024245169-A1
TPD-L8CMSB	WO2024245169A1_10	.	CC1(C)CC(=C(c2ccc3[nH]nc(F)c3c2)c2c(F)cc(N3CCN(C4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)cc2F)CC(C)(C)O1	C45H48F3N7O5	ERα	P03372	CRBN	WO-2024245169-A1
TPD-151O2G	WO2024245169A1_11	.	CC1(C)CC(=C(c2ccc3[nH]nc(F)c3c2)c2c(F)cc(N3CCC(N4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)cc2F)CC(C)(C)O1	C45H48F3N7O5	ERα	P03372	CRBN	WO-2024245169-A1
TPD-0N433H	WO2024245169A1_12	.	CC1(C)CC(=C(c2ccc3[nH]nc(F)c3c2)c2c(F)cc(N3CCC(CN4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)cc2F)CC(C)(C)O1	C46H50F3N7O5	ERα	P03372	CRBN	WO-2024245169-A1
TPD-GUIKIK	WO2024245169A1_13	.	CC1(C)CC(=C(c2ccc(N3CC(N4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C3)cc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C43H46FN7O5	ERα	P03372	CRBN	WO-2024245169-A1
TPD-5A2TDQ	WO2024245169A1_14	.	CC1(C)CC(=C(c2ccc3[nH]nc(F)c3c2)c2c(F)cc(OC3CN(C4CN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)C3)cc2F)CC(C)(C)O1	C42H41F3N6O6	ERα	P03372	CRBN	WO-2024245169-A1
TPD-775V6L	WO2024245169A1_15	.	CC1(C)CC(=C(c2ccc3[nH]nc(F)c3c2)c2c(F)cc(N3CC(CN4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C3)cc2F)CC(C)(C)O1	C44H46F3N7O5	ERα	P03372	CRBN	WO-2024245169-A1
TPD-GB3K30	WO2024245169A1_16	.	CC1(C)CC(=C(c2ccc(OCCN3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)cc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C42H45FN6O6	ERα	P03372	CRBN	WO-2024245169-A1
TPD-RJ64QJ	WO2024245169A1_17	.	CC1(C)CC(=C(c2ccc(N3CC(CN4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C3)cc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C44H48FN7O5	ERα	P03372	CRBN	WO-2024245169-A1
TPD-6DTOCX	WO2024245169A1_18	.	CC1(C)CC(=C(c2ccc(OC3CN(C4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C3)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C43H46FN7O6	ERα	P03372	CRBN	WO-2024245169-A1
TPD-1Z7024	WO2024245169A1_19	.	CC1(C)CC(=C(c2ccc(OC3CN(C4CN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)C3)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C41H42FN7O6	ERα	P03372	CRBN	WO-2024245169-A1
TPD-U5VGPR	WO2024245169A1_20	.	CC1(C)CC(=C(c2ccc(OC3CN(C4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C3)cc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C44H47FN6O6	ERα	P03372	CRBN	WO-2024245169-A1
TPD-QBSANH	WO2024245169A1_21	.	CC1(C)CC(=C(c2ccc(OC3CN(C4CN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)C3)cc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C42H43FN6O6	ERα	P03372	CRBN	WO-2024245169-A1
TPD-7NFSSH	WO2024245169A1_22	.	CC1(C)CC(=C(c2ccc(N3CCN(C4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)cc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C45H50FN7O5	ERα	P03372	CRBN	WO-2024245169-A1
TPD-9ZHE1D	WO2024245169A1_23	.	CC1(C)CC(=C(c2ccc3[nH]nc(F)c3c2)c2c(F)cc(OCCN3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)cc2F)CC(C)(C)O1	C42H43F3N6O6	ERα	P03372	CRBN	WO-2024245169-A1
TPD-IFCL4V	WO2024245169A1_24	.	CC1(C)CC(=C(c2ccc3[nH]nc(F)c3c2)c2c(F)cc(OC3CN(CC4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C3)cc2F)CC(C)(C)O1	C45H47F3N6O6	ERα	P03372	CRBN	WO-2024245169-A1
TPD-ZRPZKQ	WO2024245169A1_25	.	CC1(C)CC(=C(c2ccc3[nH]nc(F)c3c2)c2c(F)cc(OC3CN(C4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C3)cc2F)CC(C)(C)O1	C44H45F3N6O6	ERα	P03372	CRBN	WO-2024245169-A1
TPD-D15Z7B	WO2024245169A1_26	.	CC1(C)CC(=C(c2ccc3[nH]nc(F)c3c2)c2c(F)cc(OC3CN(CC4CN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)C3)cc2F)CC(C)(C)O1	C43H43F3N6O6	ERα	P03372	CRBN	WO-2024245169-A1
TPD-KJLMTT	WO2024245169A1_27	.	CC1(C)CC(=C(c2ccc(N3CC(CN4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C3)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C43H47FN8O5	ERα	P03372	CRBN	WO-2024245169-A1
TPD-ZHE74P	WO2024245169A1_28	.	CC1(C)CC(=C(c2ccc(OCCN3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C41H44FN7O6	ERα	P03372	CRBN	WO-2024245169-A1
TPD-3LXFAR	WO2024245169A1_29	.	CC1(C)CC(=C(c2ccc3[nH]nc(F)c3c2)c2c(F)cc(N3CC(N4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C3)cc2F)CC(C)(C)O1	C43H44F3N7O5	ERα	P03372	CRBN	WO-2024245169-A1
TPD-XEO3TK	WO2024245169A1_30	.	CC1(C)CC(=C(c2ccc(OC3CN(CC4CN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)C3)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C42H44FN7O6	ERα	P03372	CRBN	WO-2024245169-A1
TPD-G4LF0X	WO2024245169A1_31	.	CC1(C)CC(=C(c2ccc(N3CCC(N4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)cc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C45H50FN7O5	ERα	P03372	CRBN	WO-2024245169-A1
TPD-N6UHI7	WO2024245169A1_32	.	CC1(C)CC(=C(c2ccc(OC3CN(CC4CN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)C3)cc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C43H45FN6O6	ERα	P03372	CRBN	WO-2024245169-A1
TPD-6QC97K	WO2024245169A1_33	.	CC1(C)CC(=C(c2ccc(N3CCN(CC4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)cc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C46H52FN7O5	ERα	P03372	CRBN	WO-2024245169-A1
TPD-RS4QU9	WO2024245169A1_34	.	CC1(C)CC(=C(c2ccc(N3CCC(CN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)CC3)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C45H53FN8O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-KEGLL7	WO2024245169A1_35	.	CC1(C)CC(=C(c2ccc(N3CCC4(CC3)CC(N3CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC3)C4)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C47H55FN8O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-C09DZY	WO2024245169A1_36	.	CC1(C)CC(=C(c2ccc(N3CCC(O)(CN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)CC3)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C45H53FN8O5	ERα	P03372	CRBN	WO-2024245169-A1
TPD-DA54T7	WO2024245169A1_37	.	CC1(C)CC(=C(c2ccc(N3CCC(N4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)CC3)cc2)c2ccc3[nH]ncc3c2)CC(C)(C)O1	C45H53N7O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-HEEGM4	WO2024245169A1_38	.	CC1(C)CC(=C(c2ccc3[nH]nc(F)c3c2)c2c(F)cc(N3CCC(N4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)CC3)cc2F)CC(C)(C)O1	C45H50F3N7O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-2I7K4O	WO2024245169A1_39	.	CC1(C)CC(=C(c2ccc(N3CCC(CN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)CC3)nc2)c2ccc3[nH]ncc3c2)CC(C)(C)O1	C45H54N8O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-PMY7DE	WO2024245169A1_40	.	CC1(C)CC(=C(c2ccc(N3CC(CN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)C3)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C43H49FN8O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-UJXKNL	WO2024245169A1_41	.	CC1(C)CC(=C(c2ccc(N3CCC(CN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)CC3)cc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C46H54FN7O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-3JF3PB	WO2024245169A1_42	.	CC1(C)CC(=C(c2ccc(N3CCN(C4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)CC3)cc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C45H52FN7O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-IOQBVX	WO2024245169A1_43	.	CC1(C)CC(=C(c2ccc(N3CCC4(CC3)CC(N3CC5(CN(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)C5)C3)C4)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C48H55FN8O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-HGFP89	WO2024245169A1_44	.	CC1(C)CC(=C(c2ccc(N3CCC(CNC4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)CC3)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C46H55FN8O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-G6L47J	WO2024245169A1_45	.	CN(CC1CCN(c2ccc(C(=C3CC(C)(C)OC(C)(C)C3)c3ccc4[nH]nc(F)c4c3)cn2)CC1)C1CCN(c2ccc3c(c2)CN(C2CCC(=O)NC2=O)C3=O)CC1	C47H57FN8O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-FAVOB6	WO2024245169A1_46	.	CC1(C)CC(=C(c2ccc(N3CC4(CCN(C5CCN(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC5)CC4)C3)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C47H55FN8O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-AIKZBS	WO2024245169A1_47	.	CC1(C)CC(=C(c2ccc(N3CCC4(CC3)CN(C3CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC3)C4)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C47H55FN8O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-6U8DPO	WO2024245169A1_49	.	CC1(C)CC(=C(c2ccc(N3CCC4(CC(N5CCN(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC5)C4)C3)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C46H53FN8O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-C7QV47	WO2024245169A1_50	.	CC1(C)CC(=C(c2ccc(N3CC4(CC(N5CCN(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC5)C4)C3)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C45H51FN8O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-A3QL35	WO2024245169A1_51	.	CC1(C)CC(=C(c2ccc(N3C[C@@H]4[C@@H](CN5CCN(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC5)[C@@H]4C3)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C45H51FN8O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-B9Y7KM	WO2024245169A1_52	.	CC1(C)CC(=C(c2ccc(N3CCN(C[C@@H]4[C@H]5CN(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)C[C@@H]45)CC3)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C45H51FN8O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-SVVDJJ	WO2024245169A1_53	.	CC1(C)CC(=C(c2ccc(N3CCN(C4CC5(CCN(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)C5)C4)CC3)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C46H53FN8O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-F3RV2B	WO2024245169A1_54	.	CC1(C)CC(=C(C2=CC3C(F)=NNC3C=C2)c2ccc(N3CCC4(CC3)CC(CN3CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC3)C4)nc2)CC(C)(C)O1	C48H59FN8O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-75WTUK	WO2024245169A1_55	.	CC1(C)CC(=C(c2ccc3[nH]nc(F)c3c2)c2c(F)cc(N3CCC(CN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)CC3)cc2F)CC(C)(C)O1	C46H52F3N7O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-LPOWRY	WO2024245169A1_56	.	CC1(C)CC(=C(c2ccc(N3CCC(CN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)CC3)cc2)c2ccc3[nH]ncc3c2)CC(C)(C)O1	C46H55N7O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-8HXJND	WO2024245169A1_57	.	CC1(C)CC(=C(c2ccc(N3CCC(CNC4CN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)C4)CC3)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C44H51FN8O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-S4P839	WO2024245169A1_58	.	CC1(C)CC(C(c2ccc(N3CCC(N4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)CC3)cc2)c2ccc3[nH]ncc3c2)CC(C)(C)O1	C45H55N7O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-PQFQ0N	WO2024245169A1_60	.	CC1(C)CC(=C(c2ccc(OC3CCN(C4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)CC3)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C45H52FN7O5	ERα	P03372	CRBN	WO-2024245169-A1
TPD-O5LSFY	WO2024245169A1_61	.	CC1(C)CC(=C(c2ccc(N3CCC(F)(CNC4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)CC3)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C46H54F2N8O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-Q2JV75	WO2024245169A1_62	.	CC1(C)CC(=C(c2ccc(N3CCC4(CC3)CC(N3CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC3)C4)cc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C48H56FN7O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-M39BDS	WO2024245169A1_63	.	CC1(C)CC(=C(c2ccc(N3CCC4(CC3)CC(N3CCC(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC3)C4)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C48H56FN7O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-NBPKXM	WO2024245169A1_64	.	CC1(C)CC(=C(c2ccc(N3CCC(N4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)CC3)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C44H51FN8O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-E8D80K	WO2024245169A1_65	.	CC1(C)CC(=C(c2ccc(N3CCN(C(=O)C4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)CC3)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C45H51FN8O5	ERα	P03372	CRBN	WO-2024245169-A1
TPD-MU9G5F	WO2024245169A1_66	.	CC1(C)CC(=C(c2ccc(N3CCN(C4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)CC3)cc2)c2ccc3[nH]ncc3c2)CC(C)(C)O1	C45H53N7O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-U2Z09R	WO2024245169A1_67	.	CC1(C)CC(=C(c2ccc(N3CCN(C4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)CC3)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C44H51FN8O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-9I4H3Y	WO2024245169A1_68	.	CC1(C)CC(=C(c2ccc(N3CCC4(CC3)CC(OCC#Cc3ccc5c(c3)CN(C3CCC(=O)NC3=O)C5=O)C4)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C46H49FN6O5	ERα	P03372	CRBN	WO-2024245169-A1
TPD-KOHXA3	WO2024245169A1_69	.	CC1(C)CC(=C(c2ccc(N3CCC(CN4CCC(N5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7)CC4)CC3)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C48H57FN8O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-909TOM	WO2024245169A1_70	.	CC1(C)CC(=C(c2ccc(N3CCC4(CC3)CN(C(=O)CN3Cc5cc6c(cc5C3)C(=O)N(C3CCC(=O)NC3=O)C6)C4)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C46H51FN8O5	ERα	P03372	CRBN	WO-2024245169-A1
TPD-LRCTDS	WO2024245169A1_71	.	CC1(C)CC(=C(c2ccc(N3CC4(CCN(C(=O)CN5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7)C4)C3)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C45H49FN8O5	ERα	P03372	CRBN	WO-2024245169-A1
TPD-5BW355	WO2024245169A1_72	.	CC1(C)CC(=C(c2ccc(N3CCC4(CN(C(=O)CN5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7)C4)C3)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C45H49FN8O5	ERα	P03372	CRBN	WO-2024245169-A1
TPD-C2FWOJ	WO2024245169A1_73	.	CC1(C)CC(=C(c2ccc(N3CC4(CCN(C(=O)CN5Cc6cc7c(cc6C5)C(=O)N(C5CCC(=O)NC5=O)C7)CC4)C3)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C46H51FN8O5	ERα	P03372	CRBN	WO-2024245169-A1
TPD-GK92F1	WO2024245169A1_74	.	CC1(C)CC(=C(c2ccc(N3CCC4(CC3)CN(C(=O)CN3Cc5cc6c(cc5C3)C(=O)N(C3CCC(=O)NC3=O)C6=O)C4)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C46H49FN8O6	ERα	P03372	CRBN	WO-2024245169-A1
TPD-NNUVW1	WO2024245169A1_75	.	CC1(C)CC(=C(c2ccc(N3CCC(CN4CCN(c5cccc(N6CCC(=O)NC6=O)c5)CC4)CC3)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C42H51FN8O3	ERα	P03372	CRBN	WO-2024245169-A1
TPD-GKCVA4	WO2024245169A1_76	.	CC1(C)CC(=C(c2ccc(N3CCC(CN4CCN(c5ccc(N6CCC(=O)NC6=O)cc5)CC4)CC3)cc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C43H52FN7O3	ERα	P03372	CRBN	WO-2024245169-A1
TPD-6CFG28	WO2024245169A1_77	.	CC1(C)CC(=C(c2ccc(N3CCC(CN4CCN(c5ccc(N6CCC(=O)NC6=O)cc5)CC4)CC3)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C42H51FN8O3	ERα	P03372	CRBN	WO-2024245169-A1
TPD-XWFF3B	WO2024245169A1_78	.	CC1(C)CC(=C(c2ccc(N3CCC(N4CCN(c5ccc(N6CCC(=O)NC6=O)cc5)CC4)CC3)cc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C42H50FN7O3	ERα	P03372	CRBN	WO-2024245169-A1
TPD-Q1YH6K	WO2024245169A1_79	.	CC1(C)CC(=C(c2ccc(N3CCC(CN4CCN(c5ccc(N6CCC(=O)NC6=O)c(F)c5)CC4)CC3)cc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C43H51F2N7O3	ERα	P03372	CRBN	WO-2024245169-A1
TPD-6KBG3X	WO2024245169A1_80	.	CC1(C)CC(=C(c2ccc(N3CCC(CN4CCN(c5ccc(N6CCC(=O)NC6=O)c(F)c5)CC4)CC3)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C42H50F2N8O3	ERα	P03372	CRBN	WO-2024245169-A1
TPD-BU0LDB	WO2024245169A1_81	.	CC1(C)CC(=C(c2ccc(N3CCN(C4CCN(c5ccc(N6CCC(=O)NC6=O)cc5)CC4)CC3)cc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C42H50FN7O3	ERα	P03372	CRBN	WO-2024245169-A1
TPD-IV4IJI	WO2024245169A1_82	.	CC1(C)CC(=C(c2ccc(N3CCN(C4CN(c5ccc(N6CCC(=O)NC6=O)cc5)C4)CC3)cc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C40H46FN7O3	ERα	P03372	CRBN	WO-2024245169-A1
TPD-FPABXZ	WO2024245169A1_83	.	CC1(C)CC(=C(c2ccc(N3CCC(CN4CCN(c5ccc(F)c(NC6CCC(=O)NC6=O)c5)CC4)CC3)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C43H52F2N8O3	ERα	P03372	CRBN	WO-2024245169-A1
TPD-8OMM0K	WO2024245169A1_84	.	CC1(C)CC(=C(c2ccc(N3CC4(CN(C(=O)CN5CCC(c6ccc(NC7CCC(=O)NC7=O)cc6F)CC5)C4)C3)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C45H52F2N8O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-OQTO8F	WO2024245169A1_85	.	CC1(C)CC(=C(c2ccc(N3CC4(CN(C(=O)CN5CCC(c6ccc(NC7CCC(=O)NC7=O)cc6)CC5)C4)C3)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C45H53FN8O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-WSP8PA	WO2024245169A1_86	.	CC1(C)CC(=C(c2ccc(N3CCC(N4CCN(c5ccc(NC6CCC(=O)NC6=O)cc5)CC4)CC3)cc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C43H52FN7O3	ERα	P03372	CRBN	WO-2024245169-A1
TPD-1PRF32	WO2024245169A1_87	.	CC1(C)CC(=C(c2ccc(N3CCC(CN4CCN(c5ccc(NC6CCC(=O)NC6=O)cc5)CC4)CC3)cc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C44H54FN7O3	ERα	P03372	CRBN	WO-2024245169-A1
TPD-SLIM7R	WO2024245169A1_88	.	CC1(C)CC(=C(c2ccc(N3CCC(CN4CCN(c5ccc(NC6CCC(=O)NC6=O)cc5)CC4)CC3)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C43H53FN8O3	ERα	P03372	CRBN	WO-2024245169-A1
TPD-NE4VW3	WO2024245169A1_89	.	CC1(C)CC(=C(c2ccc(N3CCC(CN4CCN(c5ccc(NC6CCC(=O)NC6=O)c(F)c5)CC4)CC3)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C43H52F2N8O3	ERα	P03372	CRBN	WO-2024245169-A1
TPD-CEVA9Q	WO2024245169A1_90	.	CC1(C)CC(=C(c2ccc(N3CCC(CN4CCN(c5cccc(NC6CCC(=O)NC6=O)c5)CC4)CC3)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C43H53FN8O3	ERα	P03372	CRBN	WO-2024245169-A1
TPD-X42FJ5	WO2024245169A1_91	.	CC1(C)CC(=C(c2ccc(N3CCN(C4CCN(c5ccc(NC6CCC(=O)NC6=O)cc5)CC4)CC3)cc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C43H52FN7O3	ERα	P03372	CRBN	WO-2024245169-A1
TPD-RDNHCJ	WO2024245169A1_92	.	Cn1nc(N2CCC(=O)NC2=O)c2ccc(C3CCN(CC(=O)N4CCN(c5ccc(C(=C6CC(C)(C)OC(C)(C)C6)c6ccc7[nH]nc(F)c7c6)cn5)CC4)CC3)cc21	C45H53FN10O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-F1NLKE	WO2024245169A1_93	.	Cn1nc(N2CCC(=O)NC2=O)c2ccc(C3CCN(CC(=O)N4CCN(c5ccc(C(C6=CC7C(F)=NNC7C=C6)=C6CC(C)(C)OC(C)(C)C6)cn5)CC4)CC3(F)F)cc21	C45H53F3N10O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-W027Z8	WO2024245169A1_94	.	Cn1nc(N2CCC(=O)NC2=O)c2ccc(C3CCN(CC(=O)N4CC5(C4)CN(c4ccc(C(=C6CC(C)(C)OC(C)(C)C6)c6ccc7[nH]nc(F)c7c6)cn4)C5)CC3(F)F)cc21	C46H51F3N10O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-5IOIAO	WO2024245169A1_95	.	Cn1nc(N2CCC(=O)NC2=O)c2ccc(C3CCN(CC(=O)N4CC5(C4)CN(c4ccc(C(=C6CC(C)(C)OC(C)(C)C6)c6ccc7[nH]nc(F)c7c6)cn4)C5)CC3)cc21	C46H53FN10O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-QX8UKP	WO2024245169A1_96	.	CC1(C)CC(=C(c2ccc(N3CCC(CN4CCN(c5cccn6c(N7CCC(=O)NC7=O)cnc56)CC4)CC3)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C43H51FN10O3	ERα	P03372	CRBN	WO-2024245169-A1
TPD-02MMWJ	WO2024245169A1_97	.	CN(CC1CCN(c2ccc(C(=C3CC(C)(C)OC(C)(C)C3)c3ccc4[nH]nc(F)c4c3)cn2)CC1)C1CCN(c2cccn3c(N4CCC(=O)NC4=O)cnc23)CC1	C45H55FN10O3	ERα	P03372	CRBN	WO-2024245169-A1
TPD-44BTXE	WO2024245169A1_98	.	CN(CC1CCN(c2ccc(C(=C3CC(C)(C)OC(C)(C)C3)C3C=Cc4[nH]nc(F)c4C3)cn2)CC1)C1CCN(c2ccn3c(N4CCC(=O)NC4=O)cnc3c2)CC1	C45H57FN10O3	ERα	P03372	CRBN	WO-2024245169-A1
TPD-AB171K	WO2024245169A1_99	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C3CCN(CC4CCN(c5ccc(C(=C6CC(C)(C)OC(C)(C)C6)c6ccc7[nH]nc(F)c7c6)cn5)CC4)CC3)c21	C46H55FN8O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-DCG357	WO2024245169A1_100	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CCOC3CCN(c4ccc(C(=C5CC(C)(C)OC(C)(C)C5)c5ccc6[nH]nc(F)c6c5)cn4)CC3)c21	C43H46FN7O5	ERα	P03372	CRBN	WO-2024245169-A1
TPD-U6X6TJ	WO2024245169A1_101	.	Cn1c(=O)n(C2CCC(=O)NC2=O)c2cccc(C#CCN3CCN(c4ccc(C(=C5CC(C)(C)OC(C)(C)C5)c5ccc6[nH]nc(F)c6c5)cn4)CC3)c21	C42H45FN8O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-IT958P	WO2024245169A1_102	.	Cc1cc(N2CCN(CC3CCN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)cc(F)c1C(=C1CC(C)(C)OC(C)(C)C1)c1ccc2[nH]nc(F)c2c1	C47H53F2N7O5	ERα	P03372	CRBN	WO-2024245169-A1
TPD-OY2ZL9	WO2024245169A1_103	.	CC1(C)CC(=C(c2ccc(N3CCC(CN4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C45H51FN8O5	ERα	P03372	CRBN	WO-2024245169-A1
TPD-O3QHHC	WO2024245169A1_104	.	CC1(C)CC(=C(c2ccc(N3CCC(N4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C44H49FN8O5	ERα	P03372	CRBN	WO-2024245169-A1
TPD-HU6XO5	WO2024245169A1_105	.	CC1(C)CC(=C(c2ccc(N3CCN(C4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C44H49FN8O5	ERα	P03372	CRBN	WO-2024245169-A1
TPD-AGVWWK	WO2024245169A1_106	.	CC1(C)CC(=C(c2ccc(N3CCN(C4CN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)CC3)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C42H45FN8O5	ERα	P03372	CRBN	WO-2024245169-A1
TPD-IA4KEY	WO2024245169A1_107	.	CC1(C)CC(=C(c2ccc(N3CCC(CN4CCN(c5cccc(NC6CCC(=O)NC6=O)c5)CC4)CC3)cc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C44H54FN7O3	ERα	P03372	CRBN	WO-2024245169-A1
TPD-5BU0KF	WO2024245169A1_108	.	CC1(C)CC(=C(c2ccc(N3CCN(C4CCN(c5cccc(NC6CCC(=O)NC6=O)c5)CC4)CC3)cc2)c2ccc3[nH]ncc3c2)CC(C)(C)O1	C43H53N7O3	ERα	P03372	CRBN	WO-2024245169-A1
TPD-QXXCVT	WO2024245169A1_109	.	CC1(C)CC(=C(c2ccc(N3CC4(CCC(N5CCN(c6ccc7c(c6)CN(C6CCC(=O)NC6=O)C7=O)CC5)CC4)C3)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C47H55FN8O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-9PN5DB	WO2024245169A1_110	.	CC1(C)CC(=C(c2ccc(N3CCC(CN4CCN(c5ccc6c(c5)CN([C@H]5CCC(=O)NC5=O)C6=O)CC4)CC3)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C45H53FN8O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-0SPKV6	WO2024245169A1_112	.	CC1(C)CC(C(c2ccc(N3CCC(CN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)CC3)nc2)c2ccc3c(F)n[nH]c3c2)CC(C)(C)O1	C45H55FN8O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-2AF2O9	WO2024245169A1_113	.	CC1(C)CC(=C(c2ccc(N3CCC(CN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)CC3)nc2)c2ccc3cncn3c2)CC(C)(C)O1	C45H54N8O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-N5KPCG	WO2024245169A1_114	.	CC1(C)CC(=C(c2ccc(N3CCC(CN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)CC3)nc2)C2C=CC=C(O)C2)CC(C)(C)O1	C44H56N6O5	ERα	P03372	CRBN	WO-2024245169-A1
TPD-NYJJOZ	WO2024245169A1_115	.	CC1(C)CC(=C(c2ccc(N3CCC(CN4CCN(c5ccc(NC6CCC(=O)NC6=O)c(F)c5)CC4)CC3)cc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C44H53F2N7O3	ERα	P03372	CRBN	WO-2024245169-A1
TPD-95PYGN	WO2024245169A1_116	.	CC1(C)CC(=C(c2ccc(N)nc2)c2ccc(N3CCC(CN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)CC3)nc2)CC(C)(C)O1	C43H54N8O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-FQPLO0	WO2024245169A1_117	.	CC1(C)CC(=C(c2ccc(N3CCC(F)(CN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)CC3)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C45H52F2N8O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-88S6EB	WO2024245169A1_118	.	CC1(C)CC(=C(c2ccc(N3CCC(CN4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6)CC4)CC3)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C45H53FN8O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-TKI4QK	WO2024245169A1_119	.	CC1(C)CC(=C(c2ccc(N3CCC(CN4CCN(c5ccc6c(c5)CN([C@@H]5CCC(=O)NC5=O)C6=O)CC4)CC3)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C45H53FN8O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-TWTLGN	WO2024245169A1_120	.	CC1(C)CC(=C(c2ccc(N3CCC4(CC3)CC(N3CCN(c5ccc6c(c5)CN([C@H]5CCC(=O)NC5=O)C6=O)CC3)C4)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C47H55FN8O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-05O45I	WO2024245169A1_121	.	CC1(C)CC(=C(c2ccc(N3CCC4(CC3)CC(N3CCN(c5ccc6c(c5)CN([C@@H]5CCC(=O)NC5=O)C6=O)CC3)C4)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C47H55FN8O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-U3OHF6	WO2024245169A1_122	.	CC1(C)CC(=C(c2ccc(N3CCC(CN4CCN(c5ccc(C(=O)N[C@H]6CCC(=O)NC6=O)c(F)c5)CC4)CC3)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C44H52F2N8O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-GKDLPB	WO2024245169A1_123	.	CC1(C)CC(=C(c2ccc(N3CCC4(CC3)CC(N3CCN(c5ccc(C(=O)N[C@H]6CCC(=O)NC6=O)c(F)c5)CC3)C4)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C46H54F2N8O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-ABOIAQ	WO2024245169A1_124	.	Cn1nc(N2CCC(=O)NC2=O)c2cc(F)c(N3CCN(CC4CCN(c5ccc(C(=C6CC(C)(C)OC(C)(C)C6)c6ccc7[nH]nc(F)c7c6)cn5)CC4)CC3)cc21	C44H52F2N10O3	ERα	P03372	CRBN	WO-2024245169-A1
TPD-JPCVN4	WO2024245169A1_125	.	Cn1nc(N2CCC(=O)NC2=O)c2cc(F)c(N3CCN(C4CC5(CCN(c6ccc(C(=C7CC(C)(C)OC(C)(C)C7)c7ccc8[nH]nc(F)c8c7)cn6)CC5)C4)CC3)cc21	C46H54F2N10O3	ERα	P03372	CRBN	WO-2024245169-A1
TPD-TPPHQK	WO2024245169A1_126	.	CC1(C)CC(=C(c2ccc(N3CCC(CN4CCN(c5ccc(C(=O)N[C@H]6CCC(=O)NC6=O)cc5)CC4)CC3)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C44H53FN8O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-DIQXGJ	WO2024245169A1_127	.	CC1(C)CC(=C(c2ccc(N3CCC4(CC3)CC(N3CCN(C5=CC=C(C(=O)N[C@H]6CCC(=O)NC6=O)CC5)CC3)C4)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C46H57FN8O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-UXMM8R	WO2024245169A1_128	.	CC1(C)CC(=C(c2ccc(N3CCC(CN4CCN(c5ccc(C(=O)N[C@H]6CCC(=O)NC6=O)nc5)CC4)CC3)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C43H52FN9O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-2ZVEEG	WO2024245169A1_129	.	CC1(C)CC(=C(c2ccc(N3CCC4(CC3)CC(N3CCN(c5ccc(C(=O)N[C@H]6CCC(=O)NC6=O)nc5)CC3)C4)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C45H54FN9O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-S479CS	WO2024245169A1_130	.	CC1(C)CC(=C(c2ccc(N3CCC(CN4CCN(c5ccc6c(c5)C(=O)N([C@@H]5CCC(=O)NC5=O)C6=O)CC4)CC3)cc2)c2ccc3[nH]ncc3c2)CC(C)(C)O1	C46H53N7O5	ERα	P03372	CRBN	WO-2024245169-A1
TPD-DCBQGH	WO2024245169A1_131	.	CC1(C)CC(=C(c2ccc(N3CCC(CN4CCN(c5ccc6c(c5)C(=O)N([C@H]5CCC(=O)NC5=O)C6=O)CC4)CC3)cc2)c2ccc3[nH]ncc3c2)CC(C)(C)O1	C46H53N7O5	ERα	P03372	CRBN	WO-2024245169-A1
TPD-2QVHGR	WO2024245169A1_132	.	CC1(C)CC(=C(c2ccc(N3CCC(O)(CN4CCN(c5ccc6c(c5)CN([C@@H]5CCC(=O)NC5=O)C6=O)CC4)CC3)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C45H53FN8O5	ERα	P03372	CRBN	WO-2024245169-A1
TPD-HLNBVW	WO2024245169A1_133	.	CC1(C)CC(=C(c2ccc(N3CCC(O)(CN4CCN(c5ccc6c(c5)CN([C@H]5CCC(=O)NC5=O)C6=O)CC4)CC3)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C45H53FN8O5	ERα	P03372	CRBN	WO-2024245169-A1
TPD-2DINR9	WO2024245169A1_134	.	CC1(C)CC(=C(c2ccc(N3CCC(N4CCN(c5ccc6c(c5)CN([C@@H]5CCC(=O)NC5=O)C6=O)CC4)CC3)cc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C45H52FN7O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-7OOYXU	WO2024245169A1_135	.	CC1(C)CC(=C(c2ccc(N3CCC(N4CCN(c5ccc6c(c5)CN([C@H]5CCC(=O)NC5=O)C6=O)CC4)CC3)cc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C45H52FN7O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-RI03YA	WO2024245169A1_136	.	CC1(C)CC(=C(c2ccc(N3CCC(CN4CCN(c5ccc6c(c5)CN([C@@H]5CCC(=O)NC5=O)C6=O)CC4)CC3)nc2)c2ccc3[nH]ncc3c2)CC(C)(C)O1	C45H54N8O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-P74NPC	WO2024245169A1_137	.	CC1(C)CC(=C(c2ccc(N3CCC(CN4CCN(c5ccc6c(c5)CN([C@H]5CCC(=O)NC5=O)C6=O)CC4)CC3)nc2)c2ccc3[nH]ncc3c2)CC(C)(C)O1	C45H54N8O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-UW72HH	WO2024245169A1_138	.	CC1(C)CC(=C(c2ccc(N3CC4(CCN(C5CCN(c6ccc7c(c6)CN([C@@H]6CCC(=O)NC6=O)C7=O)CC5)CC4)C3)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C47H55FN8O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-T523PH	WO2024245169A1_139	.	CC1(C)CC(=C(c2ccc(N3CC4(CCN(C5CCN(c6ccc7c(c6)CN([C@H]6CCC(=O)NC6=O)C7=O)CC5)CC4)C3)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C47H55FN8O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-23D30O	WO2024245169A1_140	.	CC1(C)CC(=C(c2ccc(N3CCC4(CC3)CN(C3CCN(c5ccc6c(c5)CN([C@@H]5CCC(=O)NC5=O)C6=O)CC3)C4)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C47H55FN8O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-E5QBVA	WO2024245169A1_141	.	CC1(C)CC(=C(c2ccc(N3CCC4(CC3)CN(C3CCN(c5ccc6c(c5)CN([C@H]5CCC(=O)NC5=O)C6=O)CC3)C4)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C47H55FN8O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-18X2TX	WO2024245169A1_142	.	CC1(C)CC(=C(c2ccc(N3CCC(F)(CNC4CCN(c5ccc6c(c5)CN([C@@H]5CCC(=O)NC5=O)C6=O)CC4)CC3)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C46H54F2N8O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-021U2D	WO2024245169A1_143	.	CC1(C)CC(=C(c2ccc(N3CCC(F)(CNC4CCN(c5ccc6c(c5)CN([C@H]5CCC(=O)NC5=O)C6=O)CC4)CC3)nc2)c2ccc3[nH]nc(F)c3c2)CC(C)(C)O1	C46H54F2N8O4	ERα	P03372	CRBN	WO-2024245169-A1
TPD-YRXZMA	WO2024245312A1_2	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCC(=O)N3CCN(CC[C@H](CSC4=CC=CC=C4)NC4=CC=C(S(=O)(=O)NC5=CC=C(N6CCN(C7=CC(C8=C(C9=CC=C(F)C=C9)N(C)C(C)=C8S(C)(=O)=O)=CC(F)=C7)CC6)C=C5)C=C4S(=O)(=O)C(F)(F)F)CC3)C(C)(C)C)C=C2)SC=N1	C80H94F5N11O11S5	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-HBU2AJ	WO2024245312A1_3	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCC(=O)N3CCN(CC[C@H](CSC4=CC=CC=C4)NC4=CC=C(S(=O)(=O)NC5=CC=C(N6CCN(C7=CC(F)=CC(C8=C(C9=CC=C(F)C=C9)N(C9CC9)C(C)=C8S(C)(=O)=O)=C7)CC6)C=C5)C=C4S(=O)(=O)C(F)(F)F)CC3)C(C)(C)C)C=C2)SC=N1	C82H96F5N11O11S5	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-NYKDPE	WO2024245312A1_4	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C([N+](=O)[O-])=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(Cl)C=C1	C80H96ClFN12O11S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-HU8H03	WO2024245312A1_5	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(NC(CCN6CCN(CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C(S(=O)(=O)C(F)(F)F)=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C80H96F5N11O10S5	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-8T4QDY	WO2024245312A1_6	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(NC(CCN6CCN(CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)NC7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C(S(=O)(=O)C(F)(F)F)=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C78H92F5N11O10S5	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-BEPSZI	WO2024245312A1_7	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(NC(CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)NC7(C8=CC=C(C9=C(C)N=CS9)C=C8)CC7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C(S(=O)(=O)C(F)(F)F)=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C82H96F5N11O11S5	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-DPIYL8	WO2024245312A1_8	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)NC7(C8=CC=C(C9=C(C)N=CS9)C=C8)CC7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C(S(=O)(=O)C(F)(F)F)=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(Cl)C=C1	C82H96ClF4N11O11S5	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-VDUQQS	WO2024245312A1_9	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCC(=O)N3CCN(CC[C@H](CSC4=CC=CC=C4)NC4=CC=C(S(=O)(=O)NC5=CC=C(N6CCN(C7=CC(F)=CC(C8=C(C9=CC=C(F)C=C9)N(C(C)C)C(C)=C8S(C)(=O)=O)=C7)CC6)C=C5)C=C4[N+](=O)[O-])CC3)C(C)(C)C)C=C2)SC=N1	C81H98F2N12O11S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-2BQHXL	WO2024245312A1_10	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@@H](CCN6CCN(CCCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C([N+](=O)[O-])=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C80H98F2N12O10S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-184NCX	WO2024245312A1_11	.	C=NC1=CC(S(=O)(=O)NC2=CC=C(N3CCN(C4=CC(F)=CC(C5=C(C6=CC=C(F)C=C6)N(CC)C(C)=C5S(C)(=O)=O)=C4)CC3)C=C2)=CC=C1N[C@H](CCN1CCN(C(=O)CCOCCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)CC1)CSC1=CC=CC=C1	C80H96F2N12O10S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-UMMCE1	WO2024245312A1_12	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(NC(CCN6CCN(CCOCCOCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSSC6=CC=CC=C6)C(OC)=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C81H101F2N11O11S5	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-L5NC1J	WO2024245312A1_13	.	C=[SH](=O)C1=CC(S(=O)(=O)NC2=CC=C(N3CCN(C4=CC(F)=CC(C5=C(C6=CC=C(F)C=C6)N(CC)C(C)=C5S(C)(=O)=O)=C4)CC3)C=C2)=CC=C1NC(CCN1CCC(C)(CN(C)C(=O)CCCCCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)CC1)CSC1=CC=CC=C1	C85H107F2N11O10S5	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-P1INIC	WO2024245312A1_14	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(F)=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(CCCCCOCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C(S(=O)(=O)C(F)(F)F)=C5)C=C4)CC3)=C2)=C1C1=CC=C(F)C=C1	C81H98F5N11O11S5	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-E49KWV	WO2024245312A1_15	.	C=NC1=CC(S(=O)(=O)NC2=CC=C(N3CCN(C4=CC(F)=CC(C5=C(C6=CC=C(F)C=C6)N(CC)C(C)=C5S(C)(=O)=O)=C4)CC3)C=C2)=CC=C1NC(CSC1=CC=CC=C1)CSC1CCN(C(=O)CCCCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)CC1	C80H95F2N11O9S5	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-UMHEN9	WO2024245312A1_16	.	C=N/N=C\C(CCN1CCN(C(=O)CCCCCCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)CC1)NC1=CC=C(S(=O)(=O)NC2=CC=C(N3CCN(C4=CC(F)=CC(C5=C(C6=CC=C(F)C=C6)N(CC)C(C)=C5S(C)(=O)=O)=C4)CC3)C=C2)C=C1N=C	C77H96F2N14O9S3	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-A66OLQ	WO2024245312A1_17	.	CCN1C(C)=C(C(=O)N2CCN(C)CC2)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(NC(CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C([As])=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C85H104AsF2N13O8S3	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-SF9QIK	WO2024245312A1_18	.	CCN1C(C)=C(C(=O)NCCN(C)C)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(NC(CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C(S(N)(=O)=O)=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C84H106F2N14O10S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-KSDKSX	WO2024245312A1_19	.	CCN1C(C)=C(C(=O)N2CCN(C)CC2)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C(S(=O)(=O)C(F)(F)F)=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(Cl)C=C1	C86H104ClF4N13O10S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-7JIS22	WO2024245312A1_20	.	CCOC1=CC(S(=O)(=O)NC2=CC=C(N3CCN(C4=CC(F)=CC(C5=C(C6=CC=C(Cl)C=C6)N(CC)C(C)=C5C(=O)NCCN(C)C)=C4)CC3)C=C2)=CC=C1N[C@H](CCN1CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)CC1)CSC1=CC=CC=C1	C86H109ClFN13O9S3	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-4RTXJ7	WO2024245312A1_21	.	CCN1C(C)=C(S(C)(=O)=O)C(CCC2=CC(NS(=O)(=O)C3=CC=C(NC(CCN4CCN(C(=O)CCCOCC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=C(C)N=CS6)C=C5)C(C)(C)C)CC4)CSC4=CC=CC=C4)C([N+](=O)[O-])=C3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C71H86F2N10O12S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-FHNVOR	WO2024245312A1_22	.	CCN1C(C)=C(S(C)(=O)=O)C(CC2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(NC(CCN6CCN(C(=O)CCCCOCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C(S(=O)C(F)(F)F)=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C84H102F5N11O11S5	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-1564WG	WO2024245312A1_23	.	CCN1C(C)=C(S(C)(=O)=O)C(CC2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(NC(CCN6CCN(C(=O)CCOCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C(S(=O)(=O)C(F)(F)F)=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C82H98F5N11O12S5	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-7QOWEZ	WO2024245312A1_24	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(NC(CCN6CCN(CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C([N+](=O)[O-])=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C79H96F2N12O10S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-GGZB1L	WO2024245312A1_25	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C([N+](=O)[O-])=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=CC=C1	C80H97FN12O11S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-EHX5FY	WO2024245312A1_26	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(F)=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(CCCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C(S(=O)(=O)C(F)(F)F)=C5)C=C4)CC3)=C2)=C1C1=CC=CC=C1	C81H99F4N11O10S5	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-CUWYDQ	WO2024245312A1_27	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(NC(CCN6CCN(CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C([NH2+]C)=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(Cl)C=C1	C80H101ClFN12O8S4+	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-3SUJ23	WO2024245312A1_28	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C(S(=O)(=O)C(F)(F)F)=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C80H96F5N11O10S5	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-7LA90M	WO2024245312A1_29	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCC(=O)N3CCN(CCC(CSC4=CC=CC=C4)NC4=CC=C(S(=O)(=O)NC5=CC=C(N6CCN(C7=CC(F)=CC(C8=C(C9=CC=C(F)C=C9)N(C(C)C)C(C)=C8C(=O)NCC8CCOCC8)=C7)CC6)C=C5)C=C4[N+](=O)[O-])CC3)C(C)(C)C)C=C2)SC=N1	C87H107F2N13O11S3	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-8V5SEV	WO2024245312A1_30	.	C=NC1=CC(S(=O)(=O)NC2=CC=C(N3CCN(C4=CC(F)=CC(C5=C(C6=CC=C(F)C=C6)N(CC)C(C)=C5S(C)(=O)=O)=C4)CC3)C=C2)=CC=C1NC(CCN1CCN(CCCCCOCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)CC1)CSC1=CC=CC=C1	C81H100F2N12O9S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-A98YMY	WO2024245312A1_31	.	[C-]#[N+]C1=CC(S(=O)(=O)NCC2=CC=C(N3CCN(C4=CC(F)=CC(C5=C(C6=CC=C(F)C=C6)N(C(C)C)C(C)=C5S(C)(=O)=O)=C4)CC3)C=C2)=CC=C1N[C@H](CCN1CCC2(CCN(CCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](C)C3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)CC2)CC1)CSC1=CC=CC=C1	C84H102F2N12O8S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-GG8H6N	WO2024245312A1_32	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCC(=O)N3CCN(CC[C@H](CSC4=CC=CC=C4)NC4=CC=C(S(=O)(=O)NC5=CC=C(N6CCN(C7=CC(F)=CC(C8=C(C9=CC=C(Cl)C=C9)N(C(C)C)C=C8C(=O)NCCC8CCOCC8)=C7)CC6)C=C5)C=C4[N+](=O)[O-])CC3)C(C)(C)C)C=C2)SC=N1	C87H107ClFN13O11S3	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-22F109	WO2024245312A1_33	.	CCN1C(C)=C(C(=O)N2CCOCC2)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(NC(CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C([N+](=O)[O-])=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(Cl)C=C1	C84H101ClFN13O11S3	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-ZPIXDH	WO2024245312A1_34	.	CCN1C(C)=C(C(=O)N2CC3(CCOCC3)C2)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C(OC(F)(F)F)=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C88H105F5N12O10S3	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-VDMO92	WO2024245312A1_35	.	CCN1C(C)=C(C(=O)NC2CN(C)C2)C(CC2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C([N+](=O)[O-])=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C85H104F2N14O10S3	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-WMT23J	WO2024245312A1_36	.	CCN1C(C)=C(C(=O)NCC2COCCO2)C(CC2=CC=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(NC(CCN6CCN(CCCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C(S(=O)(=O)C(F)(F)F)=C5)C=C4)CC3)=C2)=C1C1=CC=C(F)C=C1	C87H108F4N12O11S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-ZFZ99R	WO2024245312A1_37	.	CCN1C(C)=C(C(=O)N2CC3(CCOCC3)C2)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(CCCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C([N+](=O)[O-])=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C87H107F2N13O10S3	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-BNVST7	WO2024245312A1_38	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCC(=O)N3CCN(CC[C@H](CSC4=CC=CC=C4)NC4=CC=C(S(=O)(=O)NC5=CC=C(N6CCN(C7=CC(F)=CC(C8=C(C9=CC=C(Cl)C=C9)N(C(C)C)C(C)=C8C(=O)N8CCOCC8)=C7)CC6)C=C5)C=C4[N+](=O)[O-])CC3)C(C)(C)C)C=C2)SC=N1	C85H103ClFN13O11S3	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-CQUMCM	WO2024245312A1_39	.	CCN1C(C)=C(C(=O)N2CCOCC2)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C([N+](=O)[O-])=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C84H101F2N13O11S3	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-L6WUR6	WO2024245312A1_40	.	CCN1C(C)=C(C(=O)NCCC2CCOCC2)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7CCC(C8=C(C)N=CS8)CC7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C([N+](=O)[O-])=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C87H113F2N13O11S3	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-FWCHOB	WO2024245312A1_41	.	C=NC1=CC(S(=O)(=O)NC2=CC=C(N3CCN(C4=CC(F)=CC(C5=C(C6=CC=C(F)C=C6)N(CC)C(CCCCCO)=C5C(=O)NCCCCCCO)=C4)CC3)C=C2)=CC=C1N[C@H](CCN1CCN(CCCCCCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2CCC(C3=C(C)N=CS3)CC2)C(C)(C)C)CC1)CSC1=CC=CC=C1	C91H125F2N13O9S3	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-6JMUTZ	WO2024245312A1_42	.	CCN1C(C)=C(C(=O)NC2CCOCC2)C(C2=CC(F)=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(NCCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)C(S(=O)C(F)(F)F)=C5)C=C4)CC3)=C2)=C1C1=CC=C(F)C=C1	C78H95F5N12O10S3	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-8NJFF7	WO2024245312A1_43	.	CCN1C(C)=C(C(=O)N[C@@H](C)C2CCOCC2)C(C2=CC(F)=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(NC(CCN6CCN(CCCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C(S(=O)(=O)C(F)(F)F)=C5)C=C4)CC3)=C2)=C1C1=CC=C(F)C=C1	C88H109F5N12O10S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-ATBX61	WO2024245312A1_44	.	CCN1C(C)=C(C(=O)N2CCOCC2)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(NC(CCN6CCN(CCCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C(S(=O)(=O)C(F)(F)F)=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C85H103F5N12O10S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-V40D8N	WO2024245312A1_45	.	CCN1C(C)=C(S(C)(=O)=O)C(CC2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C(S(=O)(=O)C(F)(F)F)=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C82H98F5N11O11S5	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-7H5YYV	WO2024245312A1_46	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCC(=O)N3CCC4(CCN(CCC(CSC5=CC=CC=C5)NC5=CC=C(S(=O)(=O)NC6=CC=C(N7CCN(C8=CC(C9=C(C%10=CC=C(F)C=C%10)N(C)C(C)=C9S(C)(=O)=O)=CC(F)=C8)CC7)C=C6)C=C5S(=O)(=O)C(F)(F)F)C4)CC3)C(C)(C)C)C=C2)SC=N1	C84H100F5N11O11S5	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-2O7YLO	WO2024245312A1_47	.	CCN1C(C)=C(S(C)(=O)=NC)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C(S(=O)(=O)C(F)(F)F)=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C82H99F5N12O10S5	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-DGQ8SR	WO2024245312A1_48	.	C=NC1=CC(S(=O)(=O)NC2=CC=C(N3CCN(C4=CC(F)=CC(C5=C(C6=CC=C(F)C=C6)N(CC)C(C)=C5S(C)(=O)=O)=C4)CC3)C=C2)=CC=C1NC(CCN1CCC2(CC1)CN(C(=O)CCCCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C3=C(C)N=CS3)C=C1)C(C)(C)C)C2)CSC1=CC=CC=C1	C83H100F2N12O9S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-Q1UJPB	WO2024245312A1_49	.	CCN1C(C)=C(CS(C)(=O)=O)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(NC(CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C(S(=O)(=O)C(F)(F)F)=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C82H98F5N11O11S5	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-AASDLD	WO2024245312A1_50	.	C=[As]C1=CC(S(=O)(=O)NC2=CC=C(N3CCN(C4=CC(F)=CC(C5=C(C6=CC=C(F)C=C6)N(CC)C(C)=C5S(C)(=O)=O)=C4)CC3)C=C2)=CC=C1NC(CCN1CCN(C(=O)COCCOCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)CC1)CSC1=CC=CC=C1	C80H96AsF2N11O11S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-1LB4QO	WO2024245312A1_51	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(F)=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)C7CC8(C7)CN(CC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C9=C(C)N=CS9)C=C7)C(C)(C)C)C8)CC6)CSC6=CC=CC=C6)C(S(=O)(=O)C(F)(F)F)=C5)C=C4)CC3)=C2)=C1C1=CC=C(F)C=C1	C83H97F5N12O11S5	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-G1RWL0	WO2024245312A1_52	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@@H](CCN6CCN(C(=O)NCCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C(N)=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C80H99F2N13O9S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-91HQAP	WO2024245312A1_53	.	CCN1C(C)=C(C(=O)N2CC[C@@H](O)C2)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C(S(=O)(=O)C(F)(F)F)=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C85H101F5N12O11S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-6SQ779	WO2024245312A1_54	.	CCN1C(C)=C(C(=O)N2CC[C@H](O)C2)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C(OC(F)(F)F)=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C85H101F5N12O10S3	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-S9KN8U	WO2024245312A1_55	.	CCN1C(C)=C(C(=O)N(C)C)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C7CC7)CC6)CSC6=CC=CC=C6)C(C(=O)O)=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C82H96F2N12O10S3	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-ON6SHY	WO2024245312A1_56	.	C=[NH+]C1=CC(S(=O)(=O)NC2=CC=C(N3CCN(C4=CC(F)=CC(C5=C(C6=CC=C(F)C=C6)N(CC)C(C)=C5C(=O)N5CCC(C)(O)C5)=C4)CC3)C=C2)=CC=C1N[C@H](CCN1CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)CC1)CSC1=CC=CC=C1	C86H106F2N13O9S3+	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-FYW3FF	WO2024245312A1_57	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)OCCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C([N+](=O)[O-])=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C80H96F2N12O12S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-NGZUD1	WO2024245312A1_58	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)COCCOCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C(OC(F)(F)F)=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C81H96F5N11O12S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-EC39SU	WO2024245312A1_59	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C(N)=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(Cl)C=C1	C80H98ClFN12O9S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-4AILRZ	WO2024245312A1_60	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(F)=CC(N3CCN(C4CCC(NS(=O)(=O)C5=CC=C(NC(CCN(C)CCN(C)C(=O)CCCCCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)(C)C)CSC6=CC=CC=C6)C(S(=O)(=O)C(F)(F)F)=C5)CC4)CC3)=C2)=C1C1=CC=C(F)C=C1	C81H104F5N11O11S5	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-MZILT4	WO2024245312A1_61	.	C=[NH+]C1=CC(S(=O)(=O)NC2=CC=C(N3CCN(C4=CC(F)=CC(C5=C(C6=CC=C(F)C=C6)N(CC)C(C)=C5S(C)(=O)=O)=C4)CC3)C=C2)=CC=C1NC(CCN(C)CCCN(C)CCCN(C)C(=O)CCCCCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=C(C)N=CS2)C=C1)C(C)(C)C)CSC1=CC=CC=C1	C86H112F2N13O9S4+	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-W68C66	WO2024245312A1_62	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)C7CCN(CC(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)C8=CC=C(C9=C(C)N=CS9)C=C8)C(C)(C)C)CC7)CC6)CSC6=CC=CC=C6)C(S(=O)(=O)C(F)(F)F)=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C82H97F5N12O11S5	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-JG3DC8	WO2024245312A1_63	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)C7CCN(CCC(=O)N[C@H](C(=O)N(CCO)[C@@H](C=O)C[C@@H](C)C8=CC=C(C9=C(C)N=CS9)C=C8)C(C)(C)C)CC7)CC6)CSC6=CC=CC=C6)C([As](C)(C)=O)=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C84H106AsF2N11O10S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-A9JVQC	WO2024245312A1_64	.	[C-]#[N+]C1=CC(S(=O)(=O)NC2=CC=C(N3CCN(C4=CC(F)=CC(C5=C(C6=CC=C(F)C=C6)N(CC)C(C)=C5S(C)(=O)=O)=C4)CC3)C=C2)=CC=C1N[C@H](CCN1CCN(C(=O)CCOCCOCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)CC1)CSC1=CC=CC=C1	C81H96F2N12O11S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-YXZFWB	WO2024245312A1_65	.	[C-]#[N+]C1=CC(S(=O)(=O)NC2=CC=C(N3CCN(C4=CC(F)=CC(C5=C(C6=CC=C(F)C=C6)N(CC)C(C)=C5S(C)(=O)=O)=C4)CC3)C=C2)=CC=C1N[C@H](CCN1CC[C@H](NC(=O)CCCCCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)C1)CSC1=CC=CC=C1	C81H96F2N12O9S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-TNCVLU	WO2024245312A1_66	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(F)=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)CCCCOC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C(S(=O)(=O)O)=C5)C=C4)CC3)=C2)=C1C1=CC=C(F)C=C1	C79H95F2N11O13S5	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-IPXL9A	WO2024245312A1_67	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CC3CC4(C3)CC(C(=O)N3CCN(CC[C@H](CSC5=CC=CC=C5)NC5=CC=C(S(=O)(=O)NC6=CC=C(N7CCN(C8=CC(C9=C(C%10=CC=C(F)C=C%10)N(C)C(C)=C9S(C)(=O)=O)=CC(F)=C8)CC7)C=C6)C=C5S(=O)(=O)C(F)(F)F)CC3)C4)C(C)(C)C)C=C2)SC=N1	C83H96F5N11O11S5	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-E4FQ68	WO2024245312A1_68	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(NC(CCN6CCN(C(=O)CCC(C)(C)CCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C([N+](=O)[O-])=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C82H100F2N12O11S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-652ZCD	WO2024245312A1_69	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)CCN7CCC(C(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)C8=CC=C(C9=C(C)N=CS9)C=C8)C(C)(C)C)CC7)CC6)CSC6=CC=CC=C6)C(S(=O)(=O)C(F)(F)F)=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C83H99F5N12O11S5	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-Q9YCT3	WO2024245312A1_70	.	C=NC1=CC(S(=O)(=O)NC2=CC=C(N3CCN(C4=CC(F)=CC(C5=C(C6=CC=C(F)C=C6)N(CC)C(C)=C5S(C)(=O)=O)=C4)CC3)C=C2)=CC=C1NCCCN1CCN(C(=O)CC2CCC(CC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](C)C3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)CC2)CC1	C77H96F2N12O9S3	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-G5R544	WO2024245312A1_71	.	CCN1C(C)=C(C(=O)N2CC[C@](C)(O)C2)C(CC2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(NC(CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C([N+](=O)[O-])=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C86H105F2N13O11S3	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-THGLP7	WO2024245312A1_72	.	CCN1C(C)=C(C(=O)N2CC[C@H](O)C2)C(CC2=CC(F)=CC=C2N2CCN(C3=CC=C(NS(=O)(=O)C4=CC=C(NC(CCN5CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)(C)C)CC5)CSC5=CC=CC=C5)C(OC(F)(F)F)=C4)C=C3)CC2)=C1C1=CC=C(F)C=C1	C86H103F5N12O10S3	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-GQS18G	WO2024245312A1_73	.	CCN1C(C)=C(C(=O)N2CC3COCC3C2)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(NC(CCN6CCN(C(=O)CCCCC(=O)NC(C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)C)CC6)CSC6=CC=CC=C6)C(OC(F)(F)F)=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C85H99F5N12O10S3	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-HH5YWW	WO2024245312A1_74	.	CCN1C(C)=C(C(=O)N2CC[C@@H](F)C2)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(NC(CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C([N+](=O)[O-])=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C84H100F3N13O10S3	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-HE5KOR	WO2024245312A1_75	.	CCN1C(C)=C(C(=O)N2C[C@H](OC)[C@@H](F)C2)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C([N+](=O)[O-])=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C85H102F3N13O11S3	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-UN0QEE	WO2024245312A1_76	.	CCN1C(C)=C(C(=O)N2CC[C@@H](O)C2)C(CC2=CC(F)=C(S(=O)(=O)NC3=CC=C(N4CCN(C5=CC=C(NS(=O)(=O)C6=CC=C(NC(CCN7CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)C8=CC=C(C9=C(C)N=CS9)C=C8)C(C)(C)C)CC7)OC)C(OC(F)(F)F)=C6)C=C5)CC4)C=C3)C=C2C2=CC=C(F)C=C2)=C1C1=CC=C(F)C=C1	C92H107F6N13O13S3	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-SSQRVX	WO2024245312A1_77	.	CCN1C(C)=C(S(=O)(=O)N2CC[C@@H](O)C2)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C([N+](=O)[O-])=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C83H101F2N13O12S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-NCU5O0	WO2024245312A1_78	.	CCOCCCCCCNS(=O)(=O)C1=C(C)N(CC)C(C2=CC=C(F)C=C2)=C1C1=CC(N2CCN(C3CCC(NS(=O)(=O)C4=CC=C(N(C=O)CCN(C)C5CCCC(C6CCCC(N7CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)C8=CC=C(C9=C(C)N=CS9)C=C8)C(C)C)CC7)CC6)CC5)C(N)=C4)CC3)CC2)=CC(F)=C1	C94H136F2N14O11S3	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-HFTVY7	WO2024245312A1_79	.	C=NC1=CC(S(=O)(=O)NC2=CC=C(N3CCN(C4=CC(F)=CC(C5=C(C6=CC=C(F)C=C6)N(CC)C(C)=C5S(=O)(=O)N5C[C@H](O)[C@@H](F)C5)=C4)CC3)C=C2)=CC=C1N[C@H](CCN1CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)CC1)CSC1=CC=CC=C1	C84H102F3N13O10S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-FQ06GO	WO2024245312A1_80	.	CCN1C(C)=C(S(=O)(=O)N2CCN(C)CC2)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C([As])=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C84H104AsF2N13O9S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-7437GD	WO2024245312A1_81	.	CCN1C(C)=C(S(=O)(=O)NCCN(C)C)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C(S(N)(=O)=O)=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C83H106F2N14O11S5	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-I810CT	WO2024245312A1_82	.	CCN1C(C)=C(C(=O)N2C[C@H](O)C(F)[C@@H](O)C2)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C([NH2+]C)=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C86H107F3N13O10S3+	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-W3DMF5	WO2024245312A1_83	.	CCN1C(C)=C(C(=O)N2CC[C@H](F)C2)C(C2=CC=C(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(NC(CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C([N+](=O)[O-])=C5)C=C4)CC3)C=C2)=C1C1=CC=C(F)C=C1	C84H101F2N13O10S3	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-PK51B0	WO2024245312A1_84	.	CCN1C(C)=C(C(=O)N2CCC(S(C)(=O)=O)C2)C(CC2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C([N+](=O)[O-])=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C86H105F2N13O12S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-ZMSFSS	WO2024245312A1_85	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCC(=O)N3CCN(CCC(CSC4=CC=CC=C4)NC4=CC=C(S(=O)(=O)NC5=CC=C(N6CCN(C7=CC(F)=CC(C8=C(C9=CC=C(F)C=C9)N(CC(F)(F)F)C(C)=C8C(=O)N8CC[C@H](O)C8)=C7)CC6)C=C5)C=C4S(=O)(=O)C(F)(F)F)CC3)C(C)(C)C)C=C2)SC=N1	C85H98F8N12O11S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-L5QVXN	WO2024245312A1_86	.	CCN1C(C)=C(C(=O)N2CC[C@@H](OC)C2)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C(S(=O)(=O)C(F)(F)F)=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C86H103F5N12O11S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-QTGYY6	WO2024245312A1_87	.	CCN1C(C)=C(S(=O)(=O)NCC2CCOCC2)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)CCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C(S(C)(=O)=O)=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C85H106F2N12O12S5	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-EA61GY	WO2024245312A1_88	.	C=N/N=C\C(CCN1CCN(C(=O)NCCCCCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)CC1)NC1=CC=C(S(=O)(=O)NC2=CC=C(N3CCN(C4=CC(F)=CC(C5=C(C6=CC=C(F)C=C6)N(CC)C(C)=C5C(=O)N5CC[C@H](O)C5)=C4)CC3)C=C2)C=C1N=C	C80H100F2N16O9S2	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-UWI22M	WO2024245312A1_89	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)NCCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C(S(=O)(=O)C(F)(F)F)=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C81H97F5N12O11S5	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-C3QKHS	WO2024245312A1_90	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCC(=O)N3CCN(CC[C@H](CSC4=CC=CC=C4)NC4=CC=CC(S(=O)(=O)NC5=CC=C(N6CCN(C7=CC(F)=CC(C8=C(C9=CC=C(F)C=C9)N(C)C(C)=C8C(=O)N8CC[C@H](O)C8)=C7)CC6)C=C5)=C4S(=O)C(F)(F)F)CC3)C(C)(C)C)C=C2)SC=N1	C84H99F5N12O10S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-U3TRWX	WO2024245312A1_91	.	[C-]#[N+]C1=CC(S(=O)(=O)NC2=CC=C(N3CCN(C4=CC(F)=CC(C5=C(C6=CC=C(F)C=C6)N(CC)C(C)=C5C(=O)N5CCC(C)(C#N)C5)=C4)CC3)C=C2)=CC=C1N[C@@H](CCN1CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)CC1)CSC1=CC=CC=C1	C87H102F2N14O8S3	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-2PS6G1	WO2024245312A1_92	.	CCN1C(C)=C(C(=O)N2CCC(O)(CF)CC2)C(CC2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C([N+](=O)[O-])=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C87H106F3N13O11S3	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-3RGGBM	WO2024245312A1_93	.	CCN1C(C)=C(S(=O)(=O)N2CC3COCC3C2)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@@H](CCN6CCN(CC(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)C)CC6)CSC6=CC=CC=C6)C(N)=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C85H105F2N13O10S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-T8AA57	WO2024245312A1_94	.	CCN1C(C)=C(S(=O)(=O)N2CC[C@@H](O)C2)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(NC(CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C(S(=O)(=O)C(F)(F)F)=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C84H101F5N12O12S5	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-YDYLJH	WO2024245312A1_95	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCC(=O)N3CCN(CC[C@H](CSC4=CC=CC=C4)NC4=CC=C(S(=O)(=O)NC5=CC=C(N6CCN(C7=CC(C8=C(C9=CC=CC=C9)N(C)C(C)=C8C(=O)N8CC[C@H](O)C8)=CC(F)=C7)CC6)C=C5)C=C4S(=O)(=O)C(F)(F)F)CC3)C(C)(C)C)C=C2)SC=N1	C84H100F4N12O11S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-5SV8EB	WO2024245312A1_96	.	CCN1C(C)=C(S(=O)(=O)N2CCC(S(C)(=O)=O)C2)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(NC(CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C([N+](=O)[O-])=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C84H103F2N13O13S5	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-4VYS4O	WO2024245312A1_97	.	CCN1C(C)=C(C(=O)N2CC(O)C(F)(F)C2)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(NC(CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C([N+](=O)[O-])=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C84H99F4N13O11S3	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-R2MD8B	WO2024245312A1_98	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCC(=O)N3CCN(CC[C@H](CSC4=CC=CC=C4)NC4=CC=C(S(=O)(=O)NC5=CC=C(N6CCN(C7=CC(F)=CC(C8=C(C9=CC=C(F)C=C9)N(C(C)C)C(C)=C8C(=O)N8CCC[C@H](O)C8)=C7)CC6)C=C5)C=C4[N+](=O)[O-])CC3)C(C)(C)C)C=C2)SC=N1	C86H105F2N13O11S3	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-SWC51O	WO2024245312A1_99	.	CCN1C(C)=C(C(=O)N2C[C@H](O)C[C@@H](O)C2)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C([N+](=O)[O-])=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C85H103F2N13O12S3	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-YPKJWF	WO2024245312A1_100	.	CCN1C(C)=C(C(=O)N2CC[C@H](NC(C)=O)C2)C(C2C=C(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C([N+](=O)[O-])=C5)C=C4)CC3)C=C(F)C2)=C1C1=CC=C(F)C=C1	C86H106F2N14O11S3	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-31H1BX	WO2024245312A1_101	.	CCN1C(C)=C(C(=O)N2CC[C@H](O)C2)C(CC2=CC=C(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C([N+](=O)[O-])=C5)C=C4)CC3)C=C2)=C1C1=CC=C(F)C=C1	C85H104FN13O11S3	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-L6DVJQ	WO2024245312A1_102	.	[C-]#[N+]C1=CC(S(=O)(=O)NC2=CC=C(N3CCN(C4=CC=C(CC5=C(C6=CC=C(F)C=C6)N(CC)C(C)=C5C(=O)N5CC[C@@H](NS(C)(=O)=O)C5)C=C4)CC3)C=C2)=CC=C1N[C@H](CCN1CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=C(C)N=CS3)C=C2)C(C)C)CC1)CSC1=CC=CC=C1	C86H105FN14O10S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-NFX5UZ	WO2024245312A1_103	.	C=NC1=CC(S(=O)(=O)NC2=CC=C(N3CCN(C4=CC(F)=CC(C5=C(C6=CC=C(F)C=C6)N(CC)C(C)=C5C(=O)N5C[C@H](O)[C@@H](O)C5)=C4)CC3)C=C2)=CC=C1N[C@@H](CCN1CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)CC1)CSC1=CC=CC=C1	C85H103F2N13O10S3	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-THTT9F	WO2024245312A1_104	.	CCN1C(C)=C(C(=O)N2CC[C@@H](OC)C2)C(CC2=CC=C(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C([N+](=O)[O-])=C5)C=C4)CC3)C=C2)=C1C1=CC=C(F)C=C1	C86H106FN13O11S3	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-T7RSTT	WO2024245312A1_105	.	CCN1C(C)=C(C(=O)N2CC[C@@H](NC(C)=O)C2)C(CC2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C([N+](=O)[O-])=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C87H106F2N14O11S3	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-YU870S	WO2024245312A1_106	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCC(=O)N3CCN(CC[C@H](CSC4=CC=CC=C4)NC4=CC=C(S(=O)(=O)NC5=CC=C(N6CCN(C7=CC(F)=CC(C8=C(C9=CC=C(Cl)C=C9)N(C(C)C)C(C)=C8C(=O)N8CC[C@@H](O)C8)=C7)CC6)C=C5)C=C4S(=O)(=O)C(F)(F)F)CC3)C(C)(C)C)C=C2)SC=N1	C86H103ClF4N12O11S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-F0VT42	WO2024245312A1_107	.	CCCN1C(C)=C(C(=O)NCCN2CCN(C)CC2)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(NC(CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C([N+](=O)[O-])=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C88H111F2N15O10S3	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-KLWJSX	WO2024245312A1_108	.	CCN1C(C)=C(C(=O)N2CC[C@H](O)C2)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(NC(CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C([N+](=O)[O-])=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=CC=C1	C84H102FN13O11S3	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-DH9YI7	WO2024245312A1_110	.	CCN1C(C)=C(C(=O)NCCCCN2CCOCC2)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(NC(CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C(S(=O)(=O)C(F)(F)F)=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C89H110F5N13O11S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-0JFZ3T	WO2024245312A1_111	.	C=NC1=CC(S(=O)(=O)NC2=CC=C(N3CCN(C4=CC(F)=CC(C5=C(C6=CC=C(F)C=C6)N(CC)C(C)=C5S(C)(=O)=O)=C4)C[C@H]3C)C=C2)=CC=C1N[C@H](CCN1CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)CC1)CSC1=CC=CC=C1	C82H100F2N12O9S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-MO3N3R	WO2024245312A1_112	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C(S(=O)(=O)C(F)(F)F)=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C81H96F5N11O11S5	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-45B6IB	WO2024245312A1_113	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(F)=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C([N+](=O)[O-])=C5)C=C4)C[C@@H]3C)=C2)=C1C1=CC=C(F)C=C1	C81H98F2N12O11S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-YWAOUW	WO2024245312A1_115	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3CC4CCC(C3)N4C3=CC=C(NS(=O)(=O)C4=CC=C(N[C@H](CCN5CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)(C)C)CC5)CSC5=CC=CC=C5)C([N+](=O)[O-])=C4)C=C3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C82H98F2N12O11S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-Z8OAU1	WO2024245312A1_116	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3C4CCC3CN(C3=CC=C(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C(S(=O)(=O)C(F)(F)F)=C5)C=C3)C4)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C83H98F5N11O11S5	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-YZ5BIQ	WO2024245312A1_117	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(F)=CC(C3=CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C(S(=O)(=O)C(F)(F)F)=C5)C=C4)CC3)=C2)=C1C1=CC=C(F)C=C1	C82H95F5N10O11S5	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-2098UL	WO2024245312A1_118	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(F)=CC(C3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C(S(=O)(=O)C(F)(F)F)=C5)C=C4)CC3)=C2)=C1C1=CC=C(F)C=C1	C82H97F5N10O11S5	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-KBL6L9	WO2024245312A1_119	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3CCC(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C(S(=O)(=O)C(F)(F)F)=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C82H97F5N10O11S5	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-IFF451	WO2024245312A1_120	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3CCC(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C([N+](=O)[O-])=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C81H97F2N11O11S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-DQ4MR1	WO2024245312A1_121	.	CCN1C(=O)C(/C(=C/C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C([N+](=O)[O-])=C5)C=C4)C[C@@H]3CF)=CC(F)=C2)S(C)(=O)=O)=C1C	C76H94F2N12O12S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-71N0U7	WO2024245312A1_122	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(F)=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C(S(=O)(=O)C(F)(F)F)=C5)C=C4)C[C@H]3CF)=C2)=C1C1=CC=C(F)C=C1	C82H97F6N11O11S5	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-VLZHGK	WO2024245312A1_123	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3CC4(CN(C5=CC=C(NS(=O)(=O)C6=CC=C(NC(CCN7CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)C8=CC=C(C9=C(C)N=CS9)C=C8)C(C)(C)C)CC7)CSC7=CC=CC=C7)C([N+](=O)[O-])=C6)C=C5)C4)C3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C81H96F2N12O11S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-U851UL	WO2024245312A1_124	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3CC(NC4=CC=C(NS(=O)(=O)C5=CC=C(C(=O)N(CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C(N)=C5)C=C4)C3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C79H94F2N12O10S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-HR6WQ1	WO2024245312A1_125	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3CC(OC4=CC=C(NS(=O)(=O)C5=CC=C(NC(CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C([N+](=O)[O-])=C5)C=C4)C3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C79H93F2N11O12S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-4QVW3O	WO2024245312A1_126	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(NC3CN(C4=CC=C(NS(=O)(=O)C5=CC=C(NC(CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C([N+](=O)[O-])=C5)C=C4)C3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C79H94F2N12O11S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-TPGY5O	WO2024245312A1_127	.	C=S(C)(=O)C1=CC(S(=O)(=O)NC2=CC=C(N3CC(OC4=CC(F)=CC(C5=C(C6=CC=C(F)C=C6)N(CC)C(C)=C5S(C)(=O)=O)=C4)C3)C=C2)=CC=C1NC(CCN1CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)CC1)CSC1=CC=CC=C1	C81H98F2N10O11S5	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-3AQC0D	WO2024245312A1_128	.	C=NC1=CC(S(=O)(=O)NC2=CC=C(C#CCNC3=CC(F)=CC(C4=C(C5=CC=C(F)C=C5)N(CC)C(C)=C4S(C)(=O)=O)=C3)C=C2)=CC=C1N[C@H](CCN1CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)CC1)CSC1=CC=CC=C1	C80H93F2N11O9S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-EK7CMM	WO2024245312A1_129	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(OCC#CC3=CC=C(NS(=O)(=O)C4=CC=C(N[C@H](CCN5CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)(C)C)CC5)CSC5=CC=CC=C5)C(N)=C4)C=C3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C79H92F2N10O10S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-7US5T7	WO2024245312A1_130	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(C#CCNC3=CC=C(NS(=O)(=O)C4=CC=C(N[C@H](CCN5CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)(C)C)CC5)CSC5=CC=CC=C5)C(S(=O)(=O)C(F)(F)F)=C4)C=C3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C80H91F5N10O11S5	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-IBGQI0	WO2024245312A1_131	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(F)=CC(C#CCOC3=CC=C(NS(=O)(=O)C4=CC=C(N[C@H](CCN5CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)(C)C)CC5)CSC5=CC=CC=C5)C(S(=O)(=O)C(F)(F)F)=C4)C=C3)=C2)=C1C1=CC=C(F)C=C1	C80H90F5N9O12S5	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-RZXMD0	WO2024245312A1_133	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3CC4CN(C5=CC=C(NS(=O)(=O)C6=CC=C(NC(CCN7CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)C8=CC=C(C9=C(C)N=CS9)C=C8)C(C)(C)C)CC7)CSC7=CC=CC=C7)C(S(C)(=O)=O)=C6)C=C5)CC4C3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C83H101F2N11O11S5	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-E1QCWJ	WO2024245312A1_134	.	C=NC1=CC(S(=O)(=O)NC2=CC=C(N3CCN(C4=CC(F)=CC(C5=C(C6=CC=C(F)C=C6)N(CC)C(C)=C5S(C)(=O)=O)=C4)CC3)N=C2)=CC=C1N[C@H](CCN1CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)CC1)CSC1=CC=CC=C1	C80H97F2N13O9S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-EAIADF	WO2024245312A1_135	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C([N+](=O)[O-])=C5)N=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C79H95F2N13O11S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-HQ09GO	WO2024245312A1_136	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(F)=CC(N3CCN(C4=CN=C(NS(=O)(=O)C5=CC=C(NC(CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C([N+](=O)[O-])=C5)N=C4)CC3)=C2)=C1C1=CC=C(F)C=C1	C78H94F2N14O11S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-5VQYY0	WO2024245312A1_137	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(F)=CC(N3CCN(C4=NC=C(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C([N+](=O)[O-])=C5)N=C4)CC3)=C2)=C1C1=CC=C(F)C=C1	C78H94F2N14O11S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-8ZH73S	WO2024245312A1_138	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C([N+](=O)[O-])=C5)N=N4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C78H94F2N14O11S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-OB3AQP	WO2024245312A1_139	.	CCN(CC1=CC=C(F)C=C1)C(C)C(CC1=CC(N2CCN(C3=NC=C(NS(=O)(=O)C4=CC=C(NC(CCN5CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)(C)C)CC5)CSC5=CC=CC=C5)C([N+](=O)[O-])=C4)C=N3)CC2)=CC(F)=C1)S(C)(=O)=O	C78H100F2N14O11S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-UW03VD	WO2024245312A1_140	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3CCN(C4=NC=C(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C(S(=O)(=O)C(F)(F)F)=C5)S4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C78H93F5N12O11S6	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-U7KRML	WO2024245312A1_141	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3CCN(C4=NC(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C([N+](=O)[O-])=C5)=CS4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C77H93F2N13O11S5	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-A9A6BZ	WO2024245312A1_142	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3CCN(C4=CN=C(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C(S(=O)(=O)C(F)(F)F)=C5)S4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C78H93F5N12O11S6	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-IYG8I6	WO2024245312A1_143	.	CCN1C(C)=C(C(F)(F)F)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C(S(=O)(=O)C(F)(F)F)=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C81H93F8N11O9S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-MBHNO7	WO2024245312A1_144	.	CCN1C(C)=C(CO)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C(S(=O)(=O)C(F)(F)F)=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C81H96F5N11O10S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-SFBHNB	WO2024245312A1_145	.	C=NC1=CC(S(=O)(=O)NC2=CC=C(N3CCN(C4=CC(C5=C(C6=CC=C(F)C=C6)N(CC)C(C)=C5C(C)O)=CC(F)=C4)CC3)C=C2)=CC=C1N[C@H](CCN1CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)CC1)CSC1=CC=CC=C1	C82H100F2N12O8S3	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-A99UP5	WO2024245312A1_147	.	CCN1C(C)=C(C(O)(C(F)(F)F)C(F)(F)F)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C([N+](=O)[O-])=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C82H94F8N12O10S3	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-1457FT	WO2024245312A1_148	.	CCN1C(C)=C(C(=O)O)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C(S(N)(=O)=O)=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C80H96F2N12O11S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-KZGY76	WO2024245312A1_149	.	CCN1C(C)=C(CN(C)C)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C(S(=O)(=O)C(F)(F)F)=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C83H101F5N12O9S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-0QFZYR	WO2024245312A1_150	.	CCN1C(C)=C(C(F)(F)CO)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C(S(=O)(=O)C(F)(F)F)=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C82H96F7N11O10S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-7QJ373	WO2024245312A1_163	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(NC(CCN6CCN(C(=O)CCNC7=NOC([C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)C8=CC=C(C9=C(C)N=CS9)C=C8)C(C)C)=C7)CC6)CSC6=CC=CC=C6)C(OC)=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C79H92F2N12O10S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-BLY5IV	WO2024245312A1_164	.	C=NC1=CC(S(=O)(=O)NC2=CC=C(N3CCN(C4=CC(F)=CC(C5=C(C6=CC=C(F)C=C6)N(CC)C(C)=C5S(C)(=O)=O)=C4)CC3)C=C2)=CC=C1NC(CCN1CCN(CCOC2=CN([C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](C)C3=CC=C(C4=C(C)N=CS4)C=C3)C(C)C)N=N2)CC1)CSC1=CC=CC=C1	C77H90F2N14O8S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-S21ES9	WO2024245312A1_165	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(F)=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(NC(CCN6CCN(C(=O)CCCOC7=NOC([C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)C8=CC=C(C9=C(C)N=CS9)C=C8)C(C)C)=C7)CC6)CSC6=CC=CC=C6)C(S(C)(=O)=O)=C5)C=C4)CC3)=C2)=C1C1=CC=C(F)C=C1	C80H93F2N11O12S5	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-0MULJM	WO2024245312A1_166	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(NC(CCN6CCN(C(=O)CCC7CCN(C8=NOC([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)C9=CC=C(C%10=C(C)N=CS%10)C=C9)C(C)C)=C8)CC7)CC6)CSC6=CC=CC=C6)C([N+](=O)[O-])=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C83H97F2N13O11S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-TVOZDY	WO2024245312A1_167	.	[C-]#[N+]C1=CC(S(=O)(=O)NC2=CC=C(N3CCN(C4=CC(F)=CC(C5=C(C6=CC=C(F)C=C6)N(CC)C(C)=C5S(C)(=O)=O)=C4)CC3)C=C2)=CC=C1N[C@H](CCN1CCN(CC(=O)N2CCN(C3=NOC([C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)N[C@@H](C)C4=CC=C(C5=C(C)N=CS5)C=C4)C(C)C)=C3)CC2)CC1)CSC1=CC=CC=C1	C82H94F2N14O9S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-4S9TCY	WO2024245312A1_168	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)CC7CN(C8=NOC([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)C9=CC=C(C%10=C(C)N=CS%10)C=C9)C(C)C)=C8)C7)CC6)CSC6=CC=CC=C6)C([N+](=O)[O-])=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C80H91F2N13O11S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-OUIAFO	WO2024245312A1_169	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(F)=CC(N3CCN(C4CCC(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C([N+](=O)[O-])=C5)CC4)CC3)=C2)=C1C1=CC=C(F)C=C1	C80H102F2N12O11S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-7CGXWW	WO2024245312A1_170	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(F)=CC(N3CCC(N4CCC(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C([N+](=O)[O-])=C5)CC4)CC3)=C2)=C1C1=CC=C(F)C=C1	C80H102F2N12O11S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-C2UODY	WO2024245312A1_172	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3CCC(NC4CCC(N(N)/C(=C/CN5CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)(C)C)CC5)CSC5CCCCC5)CC4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C75H105F2N11O7S3	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-P50F1B	WO2024245312A1_173	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3CCC(N4CCC(NC5CC(NC6=CC=C(N[C@H](CCN7CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)C8=CC=C(C9=C(C)N=CS9)C=C8)C(C)(C)C)CC7)CSC7=CC=CC=C7)C([N+](=O)[O-])=C6)C5)CC4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C84H109F2N13O9S3	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-MEW03I	WO2024245312A1_174	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3CCC(N4CC5(CC(NS(=O)(=O)C6=CC=C(N[C@H](CCN7CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)C8=CC=C(C9=C(C)N=CS9)C=C8)C(C)(C)C)CC7)CSC7=CC=CC=C7)C(S(=O)(=O)C(F)(F)F)=C6)C5)C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C82H102F5N11O11S5	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-RXZKTG	WO2024245312A1_175	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3CCN(C4CC5(CC(NS(=O)(=O)C6=CC=C(N[C@H](CCN7CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)C8=CC=C(C9=C(C)N=CS9)C=C8)C(C)(C)C)CC7)CSC7=CC=CC=C7)C(S(=O)(=O)C(F)(F)F)=C6)C5)C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C82H102F5N11O11S5	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-XEVHU9	WO2024245312A1_176	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3CCC4(CC3)CC(C(=O)NS(=O)(=O)C3=CC=C(N[C@H](CCN5CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)(C)C)CC5)CSC5=CC=CC=C5)C([N+](=O)[O-])=C3)C4)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C79H97F2N11O12S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-1DSRIS	WO2024245312A1_177	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3CCC4(CC3)CN(CC(=O)NS(=O)(=O)C3=CC=C(N[C@H](CCN5CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)(C)C)CC5)CSC5=CC=CC=C5)C(S(=O)(=O)C(F)(F)F)=C3)C4)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C80H98F5N11O12S5	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-7E3AG6	WO2024245312A1_178	.	[C-]#[N+]C1=CC(S(=O)(=O)NC(=O)CCN2CCN(C3=CC(F)=CC(C4=C(C5=CC=C(F)C=C5)N(CC)C(C)=C4S(C)(=O)=O)=C3)CC2)=CC=C1N[C@H](CCN1CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)CC1)CSC1=CC=CC=C1	C78H96F2N12O10S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-U8VIXD	WO2024245312A1_179	.	[C-]#[N+]C1=CC(S(=O)(=O)NC(=O)C2CCC3(CC2)CCN(C2=CC(F)=CC(C4=C(C5=CC=C(F)C=C5)N(CC)C(C)=C4S(C)(=O)=O)=C2)CC3)=CC=C1N[C@H](CCN1CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)CC1)CSC1=CC=CC=C1	C82H101F2N11O10S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-KSLRP8	WO2024245312A1_180	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(S(=O)(=O)NC3CCC4(CC3)CCN(C3=CC=C(N[C@H](CCN5CCN(C(=O)CCCCCCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)(C)C)CC5)CSC5=CC=CC=C5)C(S(=O)(=O)C(F)(F)F)=C3)CC4)=CC=C2C)=C1C1=CC=C(F)C=C1	C83H106F4N10O11S5	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-MYQ5YT	WO2024245312A1_181	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(F)=CC(C3=CC=C(N4CCC(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C(S(=O)(=O)C(F)(F)F)=C5)CC4)C=C3)=C2)=C1C1=CC=C(F)C=C1	C82H97F5N10O11S5	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-LMAUBO	WO2024245312A1_182	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(F)=CC(C3=CC=C(N4CCC(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C(N=C=O)=C5)CC4)N=C3)=C2)=C1C1=CC=C(F)C=C1	C81H96F2N12O10S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-YHGDKG	WO2024245312A1_183	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(F)=CC(N3CCN(CC(=O)NS(=O)(=O)C4=CC=C(N[C@H](CCN5CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)(C)C)CC5)CSC5=CC=CC=C5)C(S(C)(=O)=O)=C4)CC3)=C2)=C1C1=CC=C(F)C=C1	C77H97F2N11O12S5	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-44VTCP	WO2024245312A1_184	.	C=[SH](=O)C1=CC(S(=O)(=O)NC2CN(CC3CCN(C4=CC(F)=CC(C5=C(C6=CC=C(F)C=C6)N(CC)C(C)=C5S(C)(=O)=O)=C4)CC3)C2)=CC=C1N[C@H](CCN1CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)CC1)CSC1=CC=CC=C1	C80H103F2N11O10S5	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-PDWV7B	WO2024245312A1_185	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3CCN(C4CC(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C(S(=O)(=O)C(F)(F)F)=C5)C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C79H98F5N11O11S5	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-4CK2K6	WO2024245312A1_186	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3CCN(C45CC(NS(=O)(=O)C6=CC=C(N[C@H](CCN7CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)C8=CC=C(C9=C(C)N=CS9)C=C8)C(C)(C)C)CC7)CSC7=CC=CC=C7)C(S(=O)(=O)C(F)(F)F)=C6)(C4)C5)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C80H98F5N11O11S5	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-368GK6	WO2024245312A1_187	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3CCN(C4CC5CC(CNS(=O)(=O)C6=CC=C(N[C@H](CCN7CCN(C(=O)CCCCCCC(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)C8=CC=C(C9=C(C)N=CS9)C=C8)C(C)(C)C)CC7)CSC7CCCCC7)C(S(=O)(=O)C(F)(F)F)=C6)(C5)C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C84H112F5N11O11S5	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-5ML8TB	WO2024245312A1_188	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(NCCNC34CC(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C(S(=O)(=O)C(F)(F)F)=C5)(C3)C4)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C78H96F5N11O11S5	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-TBL3S5	WO2024245312A1_189	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3CCN(C4CCN(S(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C(C)=C5)CC4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C80H103F2N11O9S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-T128WF	WO2024245312A1_190	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3CCC(N4CCN(S(=O)(=O)C5=CC=C(N[C@H](CC[N+]6(C)CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C(C(F)(F)F)=C5)CC4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C81H103F5N11O9S4+	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-J2HCQ4	WO2024245312A1_191	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(C3CCN(C4CCN(S(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C([N+](=O)[O-])=C5)CC4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C80H101F2N11O11S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-P237EV	WO2024245312A1_193	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3CCC(N4CC5(C4)CN(S(=O)(=O)C4=CC=C(NC(CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C(C)=C4)C5)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C81H103F2N11O9S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-1PIJS5	WO2024245312A1_194	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3CCN(CCC4CN(S(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C([N+](=O)[O-])=C5)C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C79H100F2N12O11S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-TGDF4G	WO2024245312A1_195	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(C3=CC=C(N4CCN(S(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C([N+](=O)[O-])=C5)CC4)C=C3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C80H95F2N11O11S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-R3SLHX	WO2024245312A1_196	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(C3=CC=C(N4CCN(S(=O)(=O)C5=CC=C(N(C)[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C(N)=C5)CC4)N=C3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C80H98F2N12O9S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-PTSMPH	WO2024245312A1_198	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(NC(CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)NCC7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C(S(=O)(=O)C(F)(F)F)=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C80H94F5N11O11S5	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-6D90BF	WO2024245312A1_199	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(NC(CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](CO)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C([N+](=O)[O-])=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C80H96F2N12O12S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-NMS5K3	WO2024245312A1_200	.	C=NC[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](NC(=O)CCCCCC(=O)N1CCN(CC[C@H](CSC2=CC=CC=C2)NC2=CC=C(S(=O)(=O)NC3=CC=C(N4CCN(C5=CC(F)=CC(C6=C(C7=CC=C(F)C=C7)N(CC)C(C)=C6S(C)(=O)=O)=C5)CC4)C=C3)C=C2[N+](=O)[O-])CC1)C(C)(C)C)C1=CC=C(C2=C(C)N=CS2)C=C1	C81H97F2N13O11S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-FD474I	WO2024245312A1_201	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(NC(CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)NOC7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C([N+](=O)[O-])=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C78H92F2N12O12S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-EEPIQ2	WO2024245312A1_202	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)CCCC7=CC8=C(C=C7)C(=O)N([C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C9=C(C)N=CS9)C=C7)C(C)C)CC8)CC6)CSC6=CC=CC=C6)C(S(=O)(=O)C(F)(F)F)=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C86H96F5N11O11S5	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-XF9UEE	WO2024245312A1_203	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N7CCCC[C@H]7C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)CC6)CSC6=CC=CC=C6)C(S(=O)(=O)C(F)(F)F)=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C81H94F5N11O11S5	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-6THIYS	WO2024245312A1_204	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(F)=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N7CCOC[C@H]7C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)CC6)CSC6=CC=CC=C6)C(S(=O)(=O)C(F)(F)F)=C5)C=C4)CC3)C2)=C1C1=CC=C(F)C=C1	C80H94F5N11O12S5	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-3CQP0I	WO2024245312A1_205	.	CCN1C(C2=CC=C(F)C=C2)=C(C2=CC(F)=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C(S(=O)(=O)C(F)(F)F)=C5)C=C4)CC3)=C2)C[C@H]1C	C80H96F5N11O9S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-B0084Y	WO2024245312A1_206	.	C=C1CC(C2=CC(F)=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C([N+](=O)[O-])=C5)C=C4)CC3)=C2)=C(C2=CC=C(F)C=C2)N1C(C)C	C80H96F2N12O9S3	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-12IKBU	WO2024245312A1_207	.	CC1=CC(C2=CC(F)=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C([N+](=O)[O-])=C5)C=C4)CC3)=C2)=C(C2=CC=C(Cl)C=C2)N1C(C)C	C80H96ClFN12O9S3	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-42A6NC	WO2024245312A1_208	.	CCN1C(C)=CC(C2=CC(F)=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(NC(CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C([N+](=O)[O-])=C5)C=C4)CC3)=C2)=C1C1=CC=C(Cl)C=C1	C79H94ClFN12O9S3	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-VFLODS	WO2024245312A1_209	.	C=NC1=CC(S(=O)(=O)NC2=CC=C(N3CCN(C4=CC(C5=C(C6=CC=C(F)C=C6)N(CC)C(C)=C5C(=O)O)=CC(F)=C4)CC3)C=C2)=CC=C1NC(CCN1CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)CC1)CSC1=CC=CC=C1	C81H96F2N12O9S3	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-UIMYSB	WO2024245312A1_210	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3CCN(C4=NC=C(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C(N)=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C79H97F2N13O9S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-TTYD5H	WO2024245312A1_211	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C7=NC=C(CCCCC(=O)N[C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)C8=CC=C(C9=C(C)N=CS9)C=C8)C(C)(C)C)C=N7)CC6)CSC6=CC=CC=C6)C(OC)=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(Cl)C=C1	C83H99ClFN13O9S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-NPU78E	WO2024245312A1_212	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3CCN(C4=NC=C(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C(N)=C5)C=N4)CC3)=CC(F)=C2)C1C1=CC=C(F)C=C1	C78H98F2N14O9S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-89KT64	WO2024245312A1_213	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3CCN(C4=CC=C(NS(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C(S(=O)(=O)C(F)(F)F)=C5)C=C4)CC3)=CC(F)=C2)=C1C1=CC=C(Cl)C=N1	C80H95ClF4N12O11S5	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-GHNOV9	WO2024245312A1_214	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3CCC(N4CC5(C4)CN(S(=O)(=O)C4=CC=C(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C(N)=C4)C5)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C80H102F2N12O9S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-TLRZ12	WO2024245312A1_215	.	CCN1C(C)=C(S(C)(=O)=O)C(C2=CC(N3CCC(N4CCN(S(=O)(=O)C5=CC=C(N[C@H](CCN6CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)(C)C)CC6)CSC6=CC=CC=C6)C(N)=C5)CC4)CC3)=CC(F)=C2)=C1C1=CC=C(F)C=C1	C79H102F2N12O9S4	BCL-2;BCL2L1	P10415/Q07817	VHL	WO-2024245312-A1
TPD-096EWX	WO2024245331A1_13	.	CC(C)(O)C1=CC2=NN(C3CCC(CCN4CCN5C6=CC=C(C7CCC(=O)NC7=O)C=C6SCC5C4)CC3)C=C2C=C1C(=O)NC1=CC=CC(C(F)(F)F)=N1	C41H46F3N7O4S	IRAK4	Q9NWZ3	CRBN	WO-2024245331-A1
TPD-SEHSAY	WO2024245331A1_14	.	CC(C)(O)C1=CC2=NN(C3CCC(CCN4CCN5C6=CC=C(C7CCC(=O)NC7=O)C=C6S(=O)(=O)CC5C4)CC3)C=C2C=C1C(=O)NC1=CC=CC(C(F)(F)F)=N1	C41H46F3N7O6S	IRAK4	Q9NWZ3	CRBN	WO-2024245331-A1
TPD-9LGJ50	WO2024245331A1_15	.	COC1=CC2=NN([C@H]3CC[C@@H](CCN4CCN5C6=CC=C(N7CCC(=O)NC7=O)C=C6C(F)(F)CC5C4)CC3)C=C2C=C1NC(=O)C1CC=CC(C(F)(F)F)=N1	C39H43F5N8O4	IRAK4	Q9NWZ3	CRBN	WO-2024245331-A1
TPD-KVU7JL	WO2024245331A1_16	.	COC1=CC2=NN(C3CCC(CCN4CCN5C6=CC=C(C7(F)CCC(=O)NC7=O)C=C6C(F)(F)CC5C4)CC3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C40H41F6N7O4	IRAK4	Q9NWZ3	CRBN	WO-2024245331-A1
TPD-PLPZXW	WO2024245331A1_17	.	COC1=CC2=NN(C3CCC(CCN4CCN5C(=CC6=CC(C7CCC(=O)NC7=O)=CC=C65)C4)CC3)C=C2C=C1NC(=O)C1CC=CC(C(F)(F)F)=N1	C39H42F3N7O4	IRAK4	Q9NWZ3	CRBN	WO-2024245331-A1
TPD-FK4QRQ	WO2024245331A1_18	.	COC1=CC2=NN([C@H]3CC[C@@H](CCN4CCN5C6=CC=C(C7CCC(=O)NC7=O)C=C6C(F)=C5C4)CC3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C39H39F4N7O4	IRAK4	Q9NWZ3	CRBN	WO-2024245331-A1
TPD-9NFMPB	WO2024245331A1_19	.	COC1=CC2=NN([C@H]3CC[C@@H](CCN4CCN5C6=CC=C(C7CCC(=O)NC7=O)C=C6N=C5C4)CC3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C38H39F3N8O4	IRAK4	Q9NWZ3	CRBN	WO-2024245331-A1
TPD-V1Q327	WO2024245331A1_20	.	CC(C)(O)C1=CC2=NN([C@H]3CC[C@@H](CCN4CCN5C6=CC=C(C7CCC(=O)NC7=O)C=C6N=C5C4)CC3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C40H43F3N8O4	IRAK4	Q9NWZ3	CRBN	WO-2024245331-A1
TPD-0WB804	WO2024245331A1_21	.	CC(C)(O)C1=CC2=NN([C@H]3CC[C@@H](CCN4CCN5C(=NC6=CC(C7CCC(=O)NC7=O)=CN=C65)C4)CC3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C39H42F3N9O4	IRAK4	Q9NWZ3	CRBN	WO-2024245331-A1
TPD-JBZ00O	WO2024245331A1_22	.	CC(C)(O)C1=CC2=NN(C3CCC(CCN4CCC5=C(C4)OC4=CC(C6CCC(=O)NC6=O)=CC(F)=C45)CC3)C=C2C=C1NC(=O)C1CC=CC(C(F)(F)F)=N1	C41H44F4N6O5	IRAK4	Q9NWZ3	CRBN	WO-2024245331-A1
TPD-Y2HK3K	WO2024245331A1_23	.	CC(C)(O)C1=CC2=NN(C3CCC(CCN4CCC5=C(C4)SC4=CC(C6CCC(=O)NC6=O)=CC=C45)CC3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C41H43F3N6O4S	IRAK4	Q9NWZ3	CRBN	WO-2024245331-A1
TPD-Z7QWGE	WO2024245331A1_24	.	COC1=CC2=NN([C@H]3CC[C@@H](CN4CC5(CCN6C(=NC7=C6C=CC(C6CCC(=O)NC6=O)=C7)C5)C4)CC3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C40H41F3N8O4	IRAK4	Q9NWZ3	CRBN	WO-2024245331-A1
TPD-I0ROHC	WO2024245331A1_25	.	COC1=CC2=NN([C@H]3CC[C@@H](CCN4CCN5C6=CC=C(C7CCC(=O)NC7=O)C=C6C(=O)C5C4)CC3)C=C2C=C1NC(=O)C1CC=CC(C(F)(F)F)=N1	C39H42F3N7O5	IRAK4	Q9NWZ3	CRBN	WO-2024245331-A1
TPD-5ZTHSP	WO2024245331A1_26	.	COC1=CC2=NN([C@H]3CC[C@H](CCN4CCN5C6=CC=C(C7CCC(=O)NC7=O)C=C6C(C)(O)C5C4)CC3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C40H44F3N7O5	IRAK4	Q9NWZ3	CRBN	WO-2024245331-A1
TPD-0SGKHL	WO2024245331A1_27	.	COC1=CC2=NN([C@H]3CC[C@@H](CCN4CCN5C6=CC=C(C7CCC(=O)NC7=O)C=C6C(O)C5C4)CC3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C39H42F3N7O5	IRAK4	Q9NWZ3	CRBN	WO-2024245331-A1
TPD-582LW7	WO2024245331A1_28	.	COC1=CC2=NN(C3CCC(CCN4CCN5C6=CC=C(C7CCC(=O)NC7=O)C=C6C(F)(F)C5C4)CC3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C39H40F5N7O4	IRAK4	Q9NWZ3	CRBN	WO-2024245331-A1
TPD-GOFOAK	WO2024245331A1_29	.	COC1=CC2=NN([C@H]3CC[C@@H](CCN4CCN5C6=CC=C(C7CCC(=O)NC7=O)C=C6OCCC5C4)CC3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C40H44F3N7O5	IRAK4	Q9NWZ3	CRBN	WO-2024245331-A1
TPD-6UHXWG	WO2024245331A1_30	.	COC1=CC2=NN(C3CCC(CCN4CCN5C6=CC=C(C7CCC(=O)NC7=O)C=C6OC6(CC6)C5C4)CC3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C41H44F3N7O5	IRAK4	Q9NWZ3	CRBN	WO-2024245331-A1
TPD-3EDPL2	WO2024245331A1_31	.	COC1=CC2=NN(C3CCC(CCN4CCN5C6=CC=C(C7CCC(=O)NC7=O)C=C6OCC5C4)CC3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C39H42F3N7O5	IRAK4	Q9NWZ3	CRBN	WO-2024245331-A1
TPD-86V5OE	WO2024245331A1_32	.	CC(C)(O)C1=CC2=NN([C@H]3CC[C@@H](CCN4CC5(CCN6C(=NC7=C6C=CC(C6CCC(=O)NC6=O)=C7)C5)C4)CC3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C43H47F3N8O4	IRAK4	Q9NWZ3	CRBN	WO-2024245331-A1
TPD-ER2BGU	WO2024245331A1_33	.	O=C1CCC(C2=CC=C3C(=C2)OCC2CN(CC[C@H]4CC[C@@H](N5C=C6C=C(C(=O)NC7=CC=CC(C(F)(F)F)=N7)C(C7(O)CC7)=CC6=N5)CC4)CCN32)C(=O)N1	C41H44F3N7O5	IRAK4	Q9NWZ3	CRBN	WO-2024245331-A1
TPD-0765XH	WO2024245331A1_34	.	CP(C)(=O)C1=CC2=NN(C3CCC(CCN4CCN5C6=CC=C(C7CCC(=O)NC7=O)C=C6OCC5C4)CC3)C=C2C=C1NC(=O)C1CC=CC(C(F)(F)F)=N1	C40H47F3N7O5P	IRAK4	Q9NWZ3	CRBN	WO-2024245331-A1
TPD-BT8ZAB	WO2024245331A1_35	.	COC1=CN2N=C([C@H]3CC[C@@H](CCN4CCN5C6=CC=C(C7CCC(=O)NC7=O)C=C6OCC5C4)CC3)C=C2C=C1C(=O)NC1=CC=CC(C(F)(F)F)=N1	C39H42F3N7O5	IRAK4	Q9NWZ3	CRBN	WO-2024245331-A1
TPD-OO3ZXX	WO2024245331A1_36	.	COC1=CN2N=C(C3CCC(CCN4CCN5C6=CC=C(C7CCC(=O)NC7=O)C=C6OCC5C4)CC3)N=C2C=C1C(=O)NC1=CC=CC(C(F)(F)F)=N1	C38H41F3N8O5	IRAK4	Q9NWZ3	CRBN	WO-2024245331-A1
TPD-K6K0QR	WO2024245331A1_37	.	CC(C)OC1=CC2=NC(C3CCC(CCN4CCN5C6=C(C=C(C7CCC(=O)NC7=O)C=C6)OCC5C4)CC3)=CN2C=C1C(=O)NC1=NC(C(F)(F)F)=CC=C1	C41H46F3N7O5	IRAK4	Q9NWZ3	CRBN	WO-2024245331-A1
TPD-UYO718	WO2024245331A1_38	.	CC(C)OC1=CC2=NC([C@H]3CC[C@@H](CCN4CCN5C6=C(C=C(C7CCC(=O)NC7=O)C=C6)OCC5C4)CC3)=CN2C=C1C(=O)NC1=C2N=C3CC(F)(F)CCN3C2=CC=C1	C46H52F2N8O5	IRAK4	Q9NWZ3	CRBN	WO-2024245331-A1
TPD-J3TNAZ	WO2024245331A1_39	.	CC(C)OC1=CC2=NC(C3CCC(CCN4CCN5C6=C(C=C(C7CCC(=O)NC7=O)C=C6)OCC5C4)CC3)=CN2C=C1C(=O)NC1=C2N=C3COCCN3C2=CC=C1	C45H52N8O6	IRAK4	Q9NWZ3	CRBN	WO-2024245331-A1
TPD-7GUFBC	WO2024245331A1_40	.	COC1=CC2=C(C=C1C(=O)NC1=CC=CC(C(F)(F)F)=N1)N=C1CC3(CCN12)CN(CCN1CCN2C4=C(C=C(C5CCC(=O)NC5=O)C=C4)OCC2C1)C3	C39H41F3N8O5	IRAK4	Q9NWZ3	CRBN	WO-2024245331-A1
TPD-23H6UO	WO2024245331A1_41	.	COC1=CC2=NN([C@H]3CC[C@H](CN(C)C4CCN5C6=CC(Cl)=C(C7CCC(=O)NC7=O)C=C6OCC5C4)CC3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C40H43ClF3N7O5	IRAK4	Q9NWZ3	CRBN	WO-2024245331-A1
TPD-UPNGKW	WO2024245331A1_42	.	COC1=CC2=NN([C@H]3CC[C@H](COC4CCN5C6=C(F)C=C(C7CCC(=O)NC7=O)C=C6OCC5C4)CC3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C39H40F4N6O6	IRAK4	Q9NWZ3	CRBN	WO-2024245331-A1
TPD-RYUMQE	WO2024245331A1_43	.	COC1=CC2=NN(C3CCC(CCN4CC(=O)N5C6=CC(Cl)=C(C7CCC(=O)NC7=O)C=C6OCC5C4)CC3)C=C2C=C1NC(=O)C1CC=CC(C(F)(F)F)=N1	C39H41ClF3N7O6	IRAK4	Q9NWZ3	CRBN	WO-2024245331-A1
TPD-53Y2L3	WO2024245331A1_44	.	COC1=CC2=NN(C3CCC(CCN4CCN5C6=CC(Cl)=C(C7CCC(=O)NC7=O)C=C6OCC5C4)CC3)C=C2C=C1C(=O)NC1=CC=CC(C(F)(F)F)=N1	C39H41ClF3N7O5	IRAK4	Q9NWZ3	CRBN	WO-2024245331-A1
TPD-9FX2UX	WO2024245408A1_HANT-312	.	CCOc1c(C#N)cc2c(c1Cl)CCCC2Nc1ccc(OCCCNc2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)nc1	C34H33ClN6O6	AR	P10275	CRBN	WO-2024245408-A1
TPD-O1Q9QU	WO2024245408A1_HANT-314	.	N#Cc1cc2c(c(Cl)c1OCCCl)CCCC2c1cnc(NCCCNc2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)nc1	C33H31Cl2N7O5	AR	P10275	CRBN	WO-2024245408-A1
TPD-7CW0G5	WO2024245408A1_HANT-315-P1	.	N#Cc1cc2c(c(Cl)c1OCCCl)CCC[C@H]2c1cnc(NCCOCCOc2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)nc1	C34H32Cl2N6O7	AR	P10275	CRBN	WO-2024245408-A1
TPD-H5DPHO	WO2024245408A1_HANT-315-P2	.	N#Cc1cc2c(c(Cl)c1OCCCl)CCC[C@@H]2c1cnc(NCCOCCOc2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)nc1	C34H32Cl2N6O7	AR	P10275	CRBN	WO-2024245408-A1
TPD-0H423W	WO2024245408A1_HANT-315	.	N#Cc1cc2c(c(Cl)c1OCCCl)CCCC2c1cnc(NCCOCCOc2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)nc1	C34H32Cl2N6O7	AR	P10275	CRBN	WO-2024245408-A1
TPD-8LTOAG	WO2024245408A1_HANT-328	.	N#Cc1cc2c(c(Cl)c1OCCCl)CCCC2Nc1ccc(OCOCNc2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)nc1	C33H30Cl2N6O7	AR	P10275	CRBN	WO-2024245408-A1
TPD-4GCKT9	WO2024245408A1_HANT-329	.	N#Cc1cc2c(c(Cl)c1OCCCl)CCCC2Nc1ccc(OCNc2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)nc1	C32H28Cl2N6O6	AR	P10275	CRBN	WO-2024245408-A1
TPD-U6MAO0	WO2024245408A1_HANT-331	.	N#Cc1cc2c(c(Cl)c1OCCCl)CCCC2Nc1ccc(OCCCCNc2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)nc1	C35H34Cl2N6O6	AR	P10275	CRBN	WO-2024245408-A1
TPD-LBGDPT	WO2024245408A1_HANT-336	.	N#Cc1cc2c(c(Cl)c1OCCCl)CCCC2c1cnc(NCCCCCOc2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)nc1	C35H34Cl2N6O6	AR	P10275	CRBN	WO-2024245408-A1
TPD-41BOAP	SCHEMBL31294812	4-Chloro-3-(2-chloroethoxy)-8-[6-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxybutoxy]pyridin-3-yl]-5,6,7,8-tetrahydronaphthalene-2-carbonitrile	N#Cc1cc2c(c(Cl)c1OCCCl)CCCC2c1ccc(OCCCCOc2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)nc1	C35H32Cl2N4O7	AR	P10275	CRBN	WO-2024245408-A1
TPD-HM9G03	WO2024245408A1_HANT-339	.	N#Cc1cc2c(c(Cl)c1OCCCl)CCCC2c1ccc(OCCCNc2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)nc1	C34H31Cl2N5O6	AR	P10275	CRBN	WO-2024245408-A1
TPD-3QRO26	SCHEMBL31294892	4-Chloro-3-(2-chloroethoxy)-8-[2-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxyethoxy]piperidin-1-yl]pyrimidin-5-yl]-5,6,7,8-tetrahydronaphthalene-2-carbonitrile	N#Cc1cc2c(c(Cl)c1OCCCl)CCCC2c1cnc(N2CCC(OCCOc3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)nc1	C37H36Cl2N6O7	AR	P10275	CRBN	WO-2024245408-A1
TPD-E1TGBB	WO2024245408A1_HANT-346	.	N#Cc1cc2c(c(Cl)c1OCCCl)CCCC2c1ccc(NCCOCCOc2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)nc1	C35H33Cl2N5O7	AR	P10275	CRBN	WO-2024245408-A1
TPD-CIYW6B	WO2024245408A1_HANT-354	.	CCOc1c(C#N)cc2c(c1Cl)CCCC2c1cnc(NCCOCCOc2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)nc1	C34H33ClN6O7	AR	P10275	CRBN	WO-2024245408-A1
TPD-U8UQNT	WO2024245408A1_HANT-362	.	N#Cc1cc2c(c(Cl)c1OCCCl)CCCC2Nc1ccc(OCOCNc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)nc1	C33H30Cl2N6O7	AR	P10275	CRBN	WO-2024245408-A1
TPD-WSC2XB	WO2024245408A1_HANT-369	.	N#Cc1cc2c(c(Cl)c1OCCCl)CCCC2Nc1ccc(OCNc2cccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)nc1	C32H28Cl2N6O6	AR	P10275	CRBN	WO-2024245408-A1
TPD-54UYH2	SCHEMBL31294769	4-Chloro-3-(2-chloroethoxy)-8-[2-[4-[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]oxypropoxy]piperidin-1-yl]pyrimidin-5-yl]-5,6,7,8-tetrahydronaphthalene-2-carbonitrile	N#Cc1cc2c(c(Cl)c1OCCCl)CCCC2c1cnc(N2CCC(OCCCOc3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)nc1	C38H38Cl2N6O7	AR	P10275	CRBN	WO-2024245408-A1
TPD-BG9E37	WO2024245408A1_HANT-380	.	N#Cc1cc2c(c(Cl)c1OCCCl)CCC2c1ccc(N2CC(OCCOc3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)nc1	C35H31Cl2N5O7	AR	P10275	CRBN	WO-2024245408-A1
TPD-2SAVAW	SCHEMBL31294871	4-Chloro-3-(2-chloroethoxy)-8-[2-[4-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]azetidin-3-yl]oxypiperidin-1-yl]pyrimidin-5-yl]-5,6,7,8-tetrahydronaphthalene-2-carbonitrile	N#Cc1cc2c(c(Cl)c1OCCCl)CCCC2c1cnc(N2CCC(OC3CN(c4ccc5c(c4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)CC2)nc1	C38H37Cl2N7O6	AR	P10275	CRBN	WO-2024245408-A1
TPD-YISZP2	WO2024245408A1_HANT-393	.	N#Cc1cc2c(c(Cl)c1OCCCl)CCCC2c1cnc(N2CCC(OCCNc3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)nc1	C36H35Cl2N7O6	AR	P10275	CRBN	WO-2024245408-A1
TPD-S9CVJ3	WO2024245408A1_HANT-431	.	CCOc1c(C#N)cc2c(c1Cl)CCCC2c1cnc(NCCOC2CN(c3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)nc1	C35H34ClN7O6	AR	P10275	CRBN	WO-2024245408-A1
TPD-A0E14Q	WO2024245408A1_HANT-501	.	N#Cc1cc2c(c(Cl)c1OCCCl)CCCC2Nc1ccc2c(cnn2CCCNc2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)c1	C36H33Cl2N7O5	AR	P10275	CRBN	WO-2024245408-A1
TPD-RZWEUR	WO2024245408A1_HANT-502	.	N#Cc1cc2c(c(Cl)c1OCCCl)CCCC2Nc1ccc2cnn(CCCNc3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)c2c1	C36H33Cl2N7O5	AR	P10275	CRBN	WO-2024245408-A1
TPD-60M6AV	WO2024245408A1_HANT-503	.	N#Cc1cc2c(c(Cl)c1OCCCl)CCCC2Nc1ccc2c(cnn2CCCCNc2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)c1	C37H35Cl2N7O5	AR	P10275	CRBN	WO-2024245408-A1
TPD-BE14UX	WO2024245408A1_HANT-505	.	N#Cc1cc2c(c(Cl)c1OCCCl)CCCC2Nc1ccc2c(cnn2CCCCCNc2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)c1	C38H37Cl2N7O5	AR	P10275	CRBN	WO-2024245408-A1
TPD-LJWEID	WO2024245408A1_HANT-506	.	N#Cc1cc2c(c(Cl)c1OCCCl)CCCC2Nc1ccc2cnn(CCCCCNc3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)c2c1	C38H37Cl2N7O5	AR	P10275	CRBN	WO-2024245408-A1
TPD-NJ059L	WO2024245408A1_HANT-507	.	N#Cc1cc2c(c(Cl)c1OCCCl)CCCC2Nc1ccc2c(cnn2CCOCCNc2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)c1	C37H35Cl2N7O6	AR	P10275	CRBN	WO-2024245408-A1
TPD-BA9T3O	WO2024245408A1_HANT-508	.	N#Cc1cc2c(c(Cl)c1OCCCl)CCCC2Nc1ccc2cnn(CCOCCNc3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)c2c1	C37H35Cl2N7O6	AR	P10275	CRBN	WO-2024245408-A1
TPD-P9RVWN	WO2024245408A1_HANT-509	.	N#Cc1cc2c(c(Cl)c1OCCCl)CCCC2c1ccc(NCCOCCOc2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)cc1	C36H34Cl2N4O7	AR	P10275	CRBN	WO-2024245408-A1
TPD-L75HD8	WO2024245408A1_HANT-510	.	N#Cc1cc2c(c(Cl)c1OCCCl)CCCC2c1ccc(OCCOCCOc2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)cc1	C36H33Cl2N3O8	AR	P10275	CRBN	WO-2024245408-A1
TPD-UCEQ3U	WO2024245408A1_HANT-511	.	N#Cc1cc2c(c(Cl)c1OCCCl)CCCC2c1ccc(N2CCC(OCCOc3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)cc1	C39H38Cl2N4O7	AR	P10275	CRBN	WO-2024245408-A1
TPD-ZI94AJ	WO2024245408A1_HANT-512	.	N#Cc1cc2c(c(Cl)c1OCCCl)CCCC2c1ccc(N2CCC(OCCCOc3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)nc1	C39H39Cl2N5O7	AR	P10275	CRBN	WO-2024245408-A1
TPD-R6LXNX	WO2024245408A1_HANT-513	.	N#Cc1cc2c(c(Cl)c1OCCCl)CCCC2c1ccc(N2CC(OCCOc3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)nc1	C36H33Cl2N5O7	AR	P10275	CRBN	WO-2024245408-A1
TPD-KRQTAN	WO2024245408A1_HANT-514	.	N#Cc1cc2c(c(Cl)c1OCCCl)CCCC2c1ccc(N2CCC(OCCOc3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)nc1	C38H37Cl2N5O7	AR	P10275	CRBN	WO-2024245408-A1
TPD-80PD6W	WO2024245408A1_HANT-515	.	N#Cc1cc2c(c(Cl)c1OCCCl)CCCC2c1cnc2c(cnn2CCOCCOc2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)c1	C36H32Cl2N6O7	AR	P10275	CRBN	WO-2024245408-A1
TPD-D8HR8P	WO2024245408A1_HANT-517	.	N#Cc1cc2c(c(Cl)c1OCCCl)CCCC2c1ccc(OC2CCC(Oc3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)nc1	C37H34Cl2N4O7	AR	P10275	CRBN	WO-2024245408-A1
TPD-8CH8C2	WO2024245408A1_HANT-518	.	N#Cc1cc2c(c(Cl)c1OCCCl)CCCC2c1ccc(OC2CCC(OCCOc3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)nc1	C39H38Cl2N4O8	AR	P10275	CRBN	WO-2024245408-A1
TPD-KD6OL4	WO2024245408A1_HANT-519	.	N#Cc1cc2c(c(Cl)c1OCCCl)CCCC2c1cnc(N2CC(OCCOc3ccc4c(c3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C2)nc1	C35H32Cl2N6O7	AR	P10275	CRBN	WO-2024245408-A1
TPD-EV63EY	WO2024245430A1_1	.	Cc1cc2cc(n1)-c1cnn(C)c1OCC[C@H]1C[C@@H]1CN1/C(=N/C2=O)Nc2ccc(NC3CN(C4CCN(c5cnc(C6CCC(=O)NC6=O)cc5C)CC4)C3)cc21	C43H49N11O4	EGFR	P00533	CRBN	WO-2024245430-A1
TPD-GOGPFR	WO2024245430A1_2	.	Cc1cc2cc(n1)-c1cnn(C)c1OCC[C@H]1C[C@@H]1CN1/C(=N/C2=O)Nc2ccc(N3CCN(C4CCN(c5ccc(C6CCC(=O)NC6=O)nc5C)CC4)C[C@H]3C)cc21	C45H53N11O4	EGFR	P00533	CRBN	WO-2024245430-A1
TPD-LPH8HP	WO2024245430A1_3	.	Cc1cc2cc(n1)-c1cnn(C)c1OCC[C@H]1C[C@@H]1CN1/C(=N/C2=O)Nc2ccc(N3CCN(C4CCN(c5ccc(C6CCC(=O)NC6=O)nc5C)CC4)C[C@@H]3C)cc21	C45H53N11O4	EGFR	P00533	CRBN	WO-2024245430-A1
TPD-N3HQCI	WO2024245430A1_4	.	Cc1cc2cc(n1)-c1cnn(C)c1OCC[C@H]1C[C@@H]1CN1/C(=N/C2=O)Nc2ccc(N3CCC(N4CC5CCC(C4)N5c4ccc(C5CCC(=O)NC5=O)nc4C)CC3)cc21	C46H53N11O4	EGFR	P00533	CRBN	WO-2024245430-A1
TPD-H1EPGN	WO2024245430A1_5	.	Cc1cc2cc(n1)-c1cnn(C)c1OCC[C@H]1C[C@@H]1CN1/C(=N/C2=O)Nc2ccc(N3CCC(N4CC5CCC4CN5c4ccc(C5CCC(=O)NC5=O)nc4C)CC3)cc21	C46H53N11O4	EGFR	P00533	CRBN	WO-2024245430-A1
TPD-GNMIFS	WO2024245430A1_6	.	Cc1cc2cc(n1)-c1cnn(C)c1OCC[C@H]1C[C@@H]1CN1/C(=N/C2=O)Nc2ccc(N3CC4CCC3CN4C3CCN(c4ccc(C5CCC(=O)NC5=O)nc4C)CC3)cc21	C46H53N11O4	EGFR	P00533	CRBN	WO-2024245430-A1
TPD-NRHPG2	WO2024245430A1_7	.	Cc1cc2cc(n1)-c1cnn(C)c1OCC[C@H]1C[C@@H]1CN1/C(=N/C2=O)Nc2ccc(N3C4CCC3CN(C3CCN(c5ccc(C6CCC(=O)NC6=O)nc5C)CC3)C4)cc21	C46H53N11O4	EGFR	P00533	CRBN	WO-2024245430-A1
TPD-Y4ECOE	WO2024245430A1_8	.	Cc1cc2cc(n1)-c1cnn(C)c1OCC[C@H]1C[C@@H]1CN1/C(=N/C2=O)Nc2ccc(N3CCN([C@@H]4CCN(c5ccc(C6CCC(=O)NC6=O)nc5C)CC4(F)F)CC3)cc21	C44H49F2N11O4	EGFR	P00533	CRBN	WO-2024245430-A1
TPD-1C2WMD	WO2024245430A1_9	.	Cc1cc2cc(n1)-c1cnn(C)c1OCC[C@H]1C[C@@H]1CN1/C(=N/C2=O)Nc2ccc(N3CCN(C[C@@H]4CCN(c5ccc(C6CCC(=O)NC6=O)nc5C)C4)CC3)cc21	C44H51N11O4	EGFR	P00533	CRBN	WO-2024245430-A1
TPD-7HG82U	WO2024245430A1_10	.	Cc1cc2cc(n1)-c1cnn(C)c1OCC[C@H]1C[C@@H]1CN1/C(=N/C2=O)Nc2ccc(N3CCN(C4CN(C5CCN(c6cc(F)c([C@H]7CCC(=O)NC7=O)c(F)c6)CC5)C4)CC3)cc21	C47H53F2N11O4	EGFR	P00533	CRBN	WO-2024245430-A1
TPD-ZNDBJ8	WO2024245430A1_11	.	Cc1cc2cc(n1)-c1cnn(C)c1OCC[C@H]1C[C@@H]1CN1/C(=N/C2=O)Nc2ccc(N3CCN([C@H]4CCN(c5cnc(C6CCC(=O)NC6=O)cc5C)C[C@H]4F)CC3)cc21	C44H50FN11O4	EGFR	P00533	CRBN	WO-2024245430-A1
TPD-VGQ6IR	WO2024245430A1_12	.	Cc1cc2cc(n1)-c1cnn(C)c1OCC[C@H]1C[C@@H]1CN1/C(=N/C2=O)Nc2ccc(N3CCN([C@@H]4CCN(c5cnc(C6CCC(=O)NC6=O)cc5C)C[C@@H]4F)CC3)cc21	C44H50FN11O4	EGFR	P00533	CRBN	WO-2024245430-A1
TPD-CEJEWT	WO2024245430A1_13	.	Cc1cc2cc(n1)-c1cnn(C)c1OCC[C@H]1C[C@@H]1CN1/C(=N/C2=O)Nc2ccc(N3CCN(CC4CN(c5ccc6c(c5)C(C)(C)C(=O)N6C5CCC(=O)NC5=O)C4)CC3)cc21	C47H53N11O5	EGFR	P00533	CRBN	WO-2024245430-A1
TPD-X77DPG	WO2024245430A1_14	.	CCc1nc(C2CCC(=O)NC2=O)ccc1N1CCC(N2CCN(c3ccc4c(c3)N3C[C@H]5C[C@@H]5CCOc5c(cnn5C)-c5cc(cc(C)n5)C(=O)/N=C/3N4)CC2)CC1	C45H53N11O4	EGFR	P00533	CRBN	WO-2024245430-A1
TPD-MX1HMM	WO2024245430A1_15	.	Cc1cc2cc(n1)-c1cnn(C)c1OCC[C@H]1C[C@@H]1CN1/C(=N/C2=O)Nc2ccc(N3CCN(C4CCN(c5c(C)cc(C6CCC(=O)NC6=O)nc5C)CC4)CC3)cc21	C45H53N11O4	EGFR	P00533	CRBN	WO-2024245430-A1
TPD-56ED86	WO2024245430A1_16	.	Cc1cc2cc(n1)-c1cnn(C)c1OCC[C@H]1C[C@@H]1CN1/C(=N/C2=O)Nc2ccc(N3CCN(C4CCN(c5cc(F)c(C6CCC(=O)NC6=O)nc5C)CC4)CC3)cc21	C44H50FN11O4	EGFR	P00533	CRBN	WO-2024245430-A1
TPD-ZC8EHP	WO2024245430A1_17	.	Cc1cc2cc(n1)-c1cnn(C)c1OCC[C@]1(C)C[C@H]1CN1/C(=N/C2=O)Nc2ccc(N3CCN(C4CCN(c5cc(F)c([C@H]6CCC(=O)NC6=O)c(F)c5)CC4)CC3)cc21	C45H50F2N10O4	EGFR	P00533	CRBN	WO-2024245430-A1
TPD-CU963J	WO2024245430A1_18	.	Cc1cc2cc(n1)-c1cnn(C)c1OCC[C@H]1C[C@@H]1CN1/C(=N/C2=O)Nc2ccc(N3CCN(C4CCN(c5cccc6c5C(C)(C)C(=O)N6C5CCC(=O)NC5=O)CC4)CC3)cc21	C48H55N11O5	EGFR	P00533	CRBN	WO-2024245430-A1
TPD-2RSL26	WO2024245430A1_19	.	Cc1cc2cc(n1)-c1cnn(C)c1OCC[C@]1(C)C[C@H]1CN1/C(=N/C2=O)Nc2ccc(N3CCN(C4CCN(c5ccc(C6CCC(=O)NC6=O)nc5C)CC4)CC3)cc21	C45H53N11O4	EGFR	P00533	CRBN	WO-2024245430-A1
TPD-EKNBVQ	WO2024245430A1_20	.	Cc1cc2cc(n1)-c1cnn(C)c1OCC[C@H]1C[C@@H]1CN1/C(=N/C2=O)Nc2ccc(N3CCN(C4CN(C5CCN(c6ccc(C7CCC(=O)NC7=O)nc6C)CC5)C4)CC3)cc21	C47H56N12O4	EGFR	P00533	CRBN	WO-2024245430-A1
TPD-STCLEE	WO2024245430A1_21	.	Cc1cc2cc(n1)-c1cnn(C)c1OCC[C@H]1C[C@@H]1CN1/C(=N/C2=O)Nc2ccc(N3CCN(CCc4c(C)cc(C5CCC(=O)NC5=O)nc4C)CC3)cc21	C42H48N10O4	EGFR	P00533	CRBN	WO-2024245430-A1
TPD-UUKAQ5	WO2024245430A1_22	.	Cc1cc2cc(n1)-c1cnn(C)c1OCC[C@H]1C[C@@H]1CN1/C(=N/C2=O)Nc2ccc(N3CCN(C4CN(C5CCN(c6c(C)cc(C7CCC(=O)NC7=O)nc6C)CC5)C4)C[C@@H]3C)cc21	C49H60N12O4	EGFR	P00533	CRBN	WO-2024245430-A1
TPD-Y56URF	WO2024245430A1_24	.	Cc1cc2cc(n1)-c1cnn(C)c1OCC[C@H]1C[C@@H]1CN1/C(=N/C2=O)Nc2ccc(N3CCN(C4CN(C5CCN(c6c(C)cc(C7CCC(=O)NC7=O)nc6C)CC5)C4)C[C@H]3C)cc21	C49H60N12O4	EGFR	P00533	CRBN	WO-2024245430-A1
TPD-96W0DK	WO2024245430A1_25	.	CCc1nc(C2CCC(=O)NC2=O)ccc1N1CCC(N2CCN(c3ccc4c(c3)N3C[C@@H]5C[C@@]5(C)CCOc5c(cnn5C)-c5cc(cc(C)n5)C(=O)/N=C/3N4)CC2)CC1	C46H55N11O4	EGFR	P00533	CRBN	WO-2024245430-A1
TPD-HLVHEG	WO2024245430A1_26	.	COC[C@@H]1CN(c2ccc3c(c2)N2C[C@@H]4C[C@@]4(C)CCOc4c(cnn4C)-c4cc(cc(C)n4)C(=O)/N=C/2N3)CCN1C1CCN(c2cc(F)c([C@H]3CCC(=O)NC3=O)c(F)c2)CC1	C47H54F2N10O5	EGFR	P00533	CRBN	WO-2024245430-A1
TPD-7DCUED	WO2024245430A1_27	.	Cc1cc2cc(n1)-c1cnn(C)c1OCC[C@]1(C)C[C@H]1CN1/C(=N/C2=O)Nc2ccc(N3CCN(C4CN(C5CCN(c6cc(F)c([C@H]7CCC(=O)NC7=O)c(F)c6)CC5)C4)C[C@@H]3C)cc21	C49H57F2N11O4	EGFR	P00533	CRBN	WO-2024245430-A1
TPD-IT3WWO	WO2024245430A1_28	.	Cc1cc2cc(n1)-c1cnn(C)c1OCC[C@H]1C[C@@H]1CN1/C(=N/C2=O)Nc2ccc(N3CC4CCC3CN4C3CN(C4CCN(c5c(C)cc(C6CCC(=O)NC6=O)nc5C)CC4)C3)cc21	C50H60N12O4	EGFR	P00533	CRBN	WO-2024245430-A1
TPD-2LIS5U	WO2024245430A1_29	.	Cc1cc2cc(n1)-c1cnn(C)c1OCC[C@]1(C)C[C@H]1CN1/C(=N/C2=O)Nc2ccc(N3CCC(C(=O)N4CCC(Oc5cc(F)c([C@H]6CCC(=O)NC6=O)c(F)c5)CC4)CC3)cc21	C47H51F2N9O6	EGFR	P00533	CRBN	WO-2024245430-A1
TPD-ZYZU0M	WO2024245430A1_30	.	Cc1cc2cc(n1)-c1cnn(C)c1OCC[C@H]1C[C@@H]1CN1/C(=N/C2=O)Nc2ccc(N3CCN([C@H]4CCN(c5cc(F)c(C6CCC(=O)NC6=O)nc5C)C[C@H]4F)CC3)cc21	C44H49F2N11O4	EGFR	P00533	CRBN	WO-2024245430-A1
TPD-HPEN03	WO2024245430A1_31	.	CCc1nc(C2CCC(=O)NC2=O)ccc1N1CC[C@H](N2CCN(c3ccc4c(c3)N3C[C@H]5C[C@@H]5CCOc5c(cnn5C)-c5cc(cc(C)n5)C(=O)/N=C/3N4)CC2)[C@H](F)C1	C45H52FN11O4	EGFR	P00533	CRBN	WO-2024245430-A1
TPD-MR5DYZ	WO2024245430A1_32	.	CCc1nc(C2CCC(=O)NC2=O)ccc1N1CC[C@@H](N2CCN(c3ccc4c(c3)N3C[C@H]5C[C@@H]5CCOc5c(cnn5C)-c5cc(cc(C)n5)C(=O)/N=C/3N4)CC2)[C@@H](F)C1	C45H52FN11O4	EGFR	P00533	CRBN	WO-2024245430-A1
TPD-RZA5NK	WO2024245430A1_33	.	Cc1cc2cc(n1)-c1cnn(C)c1OCC[C@H]1C[C@@H]1CN1/C(=N/C2=O)Nc2ccc(N3CCN([C@@H]4CCN(c5c(C)cc(C6CCC(=O)NC6=O)nc5C)C[C@@H]4F)CC3)cc21	C45H52FN11O4	EGFR	P00533	CRBN	WO-2024245430-A1
TPD-X8B04R	WO2024245430A1_34	.	Cc1cc2cc(n1)-c1cnn(C)c1OCC[C@H]1C[C@@H]1CN1/C(=N/C2=O)Nc2ccc(N3CCN([C@@H]4CCN(c5cc(F)c(C6CCC(=O)NC6=O)nc5C)C[C@@H]4F)CC3)cc21	C44H49F2N11O4	EGFR	P00533	CRBN	WO-2024245430-A1
TPD-CHMM29	WO2024245430A1_35	.	Cc1cc2cc(n1)-c1cnn(C)c1OCC[C@H]1C[C@@H]1CN1/C(=N/C2=O)Nc2ccc(N3CCN(CCc4cc(F)c([C@H]5CCC(=O)NC5=O)c(F)c4)C(C4CCOC4)C3)cc21	C45H49F2N9O5	EGFR	P00533	CRBN	WO-2024245430-A1
TPD-ZWUGK2	WO2024245430A1_36	.	Cc1cc2cc(n1)-c1cnn(C)c1OCC[C@H]1C[C@@H]1CN1/C(=N/C2=O)Nc2ccc(N3CCN(C4CN(C5CCN(c6ccc(C7CCC(=O)NC7=O)nc6C)CC5)C4)C[C@@H]3C)cc21	C48H58N12O4	EGFR	P00533	CRBN	WO-2024245430-A1
TPD-FV8MT5	WO2024245430A1_37	.	Cc1cc2cc(n1)-c1cnn(C)c1OCC[C@H]1C[C@@H]1CN1/C(=N/C2=O)Nc2ccc(N3CCN(C4CN(C5CCN(c6ccc(C7CCC(=O)NC7=O)nc6C)CC5)C4)C[C@H]3C)cc21	C48H58N12O4	EGFR	P00533	CRBN	WO-2024245430-A1
TPD-9PBZVB	WO2024245430A1_43	.	Cc1cc2cc(n1)-c1cnn(C)c1OCC[C@]1(C)C[C@H]1CN1/C(=N/C2=O)Nc2ccc(N3CCN([C@@H]4CCN(c5cc(F)c(C6CCC(=O)NC6=O)nc5C)C[C@@H]4F)CC3)cc21	C45H51F2N11O4	EGFR	P00533	CRBN	WO-2024245430-A1
TPD-0A3DMJ	WO2024245430A1_49	.	Cc1cc2cc(n1)-c1cnn(C)c1OCC[C@]1(C)C[C@H]1CN1/C(=N/C2=O)Nc2ccc(N3CCN([C@@H]4CCN(c5ccc(C6CCC(=O)NC6=O)nc5C)C[C@@H]4F)CC3)cc21	C45H52FN11O4	EGFR	P00533	CRBN	WO-2024245430-A1
TPD-M3O4WU	WO2024245430A1_54	.	Cc1cc2cc(n1)-c1cnn(C)c1OCC[C@]1(C)C[C@H]1CN1/C(=N/C2=O)Nc2ccc(N3CCN(C4CCN(c5cc(F)c(C6CCC(=O)NC6=O)nc5C)CC4)CC3)cc21	C45H52FN11O4	EGFR	P00533	CRBN	WO-2024245430-A1
TPD-GQQ7G5	WO2024245430A1_57	.	Cc1cc2cc(n1)-c1cnn(C)c1OCC[C@]1(C)C[C@H]1CN1/C(=N/C2=O)Nc2ccc(N3CCN([C@@H]4CCN(c5cccc6c5C(C)(C)C(=O)N6C5CCC(=O)NC5=O)C[C@@H]4F)CC3)cc21	C49H56FN11O5	EGFR	P00533	CRBN	WO-2024245430-A1
TPD-WAR3TD	WO2024245430A1_59	.	Cc1cc2cc(n1)-c1cnn(C)c1OCC[C@]1(C)C[C@H]1CN1/C(=N/C2=O)Nc2ccc(N3CCN([C@@H]4CCN(c5cnc(C6CCC(=O)NC6=O)cc5C)C[C@@H]4F)CC3)cc21	C45H52FN11O4	EGFR	P00533	CRBN	WO-2024245430-A1
TPD-NTYOBD	WO2024245430A1_61	.	Cc1cc2cc(n1)-c1cnn(C)c1OCC[C@]1(C)C[C@H]1CN1/C(=N/C2=O)Nc2ccc(N3CCN([C@H]4CCN(c5cc(F)c(C6CCC(=O)NC6=O)nc5C)C[C@H]4F)CC3)cc21	C45H51F2N11O4	EGFR	P00533	CRBN	WO-2024245430-A1
TPD-OJ34YG	WO2024245430A1_62	.	Cc1cc2cc(n1)-c1cnn(C)c1OCC[C@]1(C)C[C@H]1CN1/C(=N/C2=O)Nc2ccc(N3CCN([C@H]4CCN(c5ccc(C6CCC(=O)NC6=O)nc5C)C[C@H]4F)CC3)cc21	C45H52FN11O4	EGFR	P00533	CRBN	WO-2024245430-A1
TPD-3DP63R	WO2024256569A1_26	.	CC1=NC2=C(F)C=C(C3=C(F)C=NC(NC4=CC=C(N5CCN(C(=O)CCCC(=O)NC6=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)CC5)C=C4)=N3)C=C2N1C(C)C	C43H42F2N10O6	CDK4;CDK6;CDK9	P11802/Q00534/P50750	CRBN	WO-2024256569-A1
TPD-9Z7SSV	WO2024256569A1_28 LOT1	.	CC1=NC2=C(F)C=C(C3=C(F)C=NC(NC4=CC=C(N5CCN(C(=O)CCCC(=O)N6CCN(C7=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=CC=C7)CC6)CC5)C=N4)=N3)C=C2N1C(C)C	C46H48F2N12O6	CDK4;CDK6;CDK9	P11802/Q00534/P50750	CRBN	WO-2024256569-A1
TPD-F3UCDC	WO2024256569A1_29	.	CC1=NC2=C(F)C=C(C3=C(F)C=NC(NC4=NC=C(N5CCN(C(=O)CC(C)(C)CC(=O)N6CCN(C7=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=CC=C7)CC6)CC5)C=C4)=N3)C=C2N1C(C)C	C48H52F2N12O6	CDK4;CDK6;CDK9	P11802/Q00534/P50750	CRBN	WO-2024256569-A1
TPD-C3EKZB	WO2024256569A1_30	.	CC1=NC2=C(F)C=C(C3=C(F)C=NC(NC4=NC=C(N5CCN(C(=O)COCC(=O)N6CCN(C7=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=CC=C7)CC6)CC5)C=C4)=N3)C=C2N1C(C)C	C45H46F2N12O7	CDK4;CDK6;CDK9	P11802/Q00534/P50750	CRBN	WO-2024256569-A1
TPD-6ZMGT6	WO2024256569A1_31	.	CC1=NC2=C(F)C=C(C3=C(F)C=NC(NC4=NC=C(N5CCN(C(=O)CN(C)CC(=O)N6CCN(C7=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=CC=C7)CC6)CC5)C=C4)=N3)C=C2N1C(C)C	C46H49F2N13O6	CDK4;CDK6;CDK9	P11802/Q00534/P50750	CRBN	WO-2024256569-A1
TPD-AANNDZ	WO2024256569A1_32	.	CC1=NC2=C(F)C=C(C3=C(F)C=NC(NC4=NC=C(N5CCN(C(=O)CSCC(=O)N6CCN(C7=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=CC=C7)CC6)CC5)C=C4)=N3)C=C2N1C(C)C	C45H46F2N12O6S	CDK4;CDK6;CDK9	P11802/Q00534/P50750	CRBN	WO-2024256569-A1
TPD-4KO3GZ	WO2024256569A1_33	.	CC1=NC2=C(F)C=C(C3=C(F)C=NC(NC4=NC=C(N5CCN(C(=O)CCCCC(=O)N6CCN(C7=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=CC=C7)CC6)CC5)C=C4)=N3)C=C2N1C(C)C	C47H50F2N12O6	CDK4;CDK6;CDK9	P11802/Q00534/P50750	CRBN	WO-2024256569-A1
TPD-0CAA1N	WO2024256569A1_35	.	CC1=NC2=C(F)C=C(C3=C(F)C=NC(NC4=NC=C(N5CCN(C(=O)/C=C/C(=O)N6CCN(C7=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=CC=C7)CC6)CC5)C=C4)=N3)C=C2N1C(C)C	C45H44F2N12O6	CDK4;CDK6;CDK9	P11802/Q00534/P50750	CRBN	WO-2024256569-A1
TPD-9XZ6PN	WO2024256569A1_36	.	CC1=NC2=C(F)C=C(C3=C(F)C=NC(NC4=CC=C(N5CCN(C(=O)C6CC6C(=O)N6CCN(C7=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=CC=C7)CC6)CC5)C=N4)=N3)C=C2N1C(C)C	C46H46F2N12O6	CDK4;CDK6;CDK9	P11802/Q00534/P50750	CRBN	WO-2024256569-A1
TPD-PYBN6M	WO2024256569A1_37	.	CC1=NC2=C(F)C=C(C3=C(F)C=NC(NC4=NC=C(N5CCN(C(=O)C6C(C(=O)N7CCN(C8=C9C(=O)N(C%10CCC(=O)NC%10=O)C(=O)C9=CC=C8)CC7)C6(C)C)CC5)C=C4)=N3)C=C2N1C(C)C	C48H50F2N12O6	CDK4;CDK6;CDK9	P11802/Q00534/P50750	CRBN	WO-2024256569-A1
TPD-GK80LT	WO2024256569A1_42	.	CC1=NC2=C(F)C=C(C3=C(F)C=NC(NC4=CC=C(N5CCN(C(=O)CCCCC#CC6=CC=C(C(=O)N7CCN(C8=C9C(=O)N(C%10CCC(=O)NC%10=O)C(=O)C9=CC=C8)CC7)C=C6)CC5)C=C4)=N3)C=C2N1C(C)C	C56H55F2N11O6	CDK4;CDK6;CDK9	P11802/Q00534/P50750	CRBN	WO-2024256569-A1
TPD-BEY1CT	WO2024256569A1_47	.	CC1=NC2=C(F)C=C(C3=C(F)C=NC(NC4=CC=C(N5CCN(C(=O)C6C(C(=O)N7CCN(CC8=CC=C(COC9=C%10C(=O)N(C%11CCC(=O)NC%11=O)C(=O)C%10=CC=C9)C=C8)CC7)C6(C)C)CC5)C=N4)=N3)C=C2N1C(C)C	C56H58F2N12O7	CDK4;CDK6;CDK9	P11802/Q00534/P50750	CRBN	WO-2024256569-A1
TPD-6VXXF6	WO2024256569A1_51	.	CC1=NC2=C(F)C=C(C3=C(F)C=NC(NC4=CC=C(N5CCN(C(=O)CCCC(=O)N6CCN(C7=C8C(=O)N(C9CCC(=O)N(C)C9=O)C(=O)C8=CC=C7)CC6)CC5)C=N4)=N3)C=C2N1C(C)C	C47H50F2N12O6	CDK4;CDK6;CDK9	P11802/Q00534/P50750	CRBN	WO-2024256569-A1
TPD-H9CT48	SCHEMBL31297431	[3-(dimethylamino)cyclobutyl] 3-[[6-cyclopropyl-7-(6-fluoro-5-methyl-1H-indazol-4-yl)-8-[[4-[1-[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1R)-2-hydroxy-1-[4-(4-methyl-1,3-oxazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]triazol-4-yl]phenyl]methoxy]-2-[(2S)-2-methoxypropoxy]quinazolin-4-yl]amino]azetidine-1-carboxylate	CO[C@@H](C)COc1nc(NC2CN(C(=O)O[C@H]3C[C@@H](N(C)C)C3)C2)c2cc(C3CC3)c(-c3c(C)c(F)cc4[nH]ncc34)c(OCc3ccc(-c4cn([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](CO)c5ccc(-c6ocnc6C)cc5)C(C)C)nn4)cc3)c2n1	C64H74FN13O10	KRAS	P01116	VHL	WO-2024261256-A1
TPD-Q6W0Q2	SCHEMBL31297428	[3-(dimethylamino)cyclobutyl] 3-[[6-cyclopropyl-7-(6-fluoro-5-methyl-1H-indazol-4-yl)-8-[[4-[1-[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1R)-2-hydroxy-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]triazol-4-yl]phenyl]methoxy]-2-[(2S)-2-methoxypropoxy]quinazolin-4-yl]amino]azetidine-1-carboxylate	CO[C@@H](C)COc1nc(NC2CN(C(=O)O[C@H]3C[C@@H](N(C)C)C3)C2)c2cc(C3CC3)c(-c3c(C)c(F)cc4[nH]ncc34)c(OCc3ccc(-c4cn([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](CO)c5ccc(-n6cncn6)cc5)C(C)C)nn4)cc3)c2n1	C62H72FN15O9	KRAS	P01116	VHL	WO-2024261256-A1
TPD-CLQ0BI	WO2024261256A1_3	.	CO[C@@H](C)COc1nc(NC2CN(C(=O)O[C@H]3C[C@@H](N(C)C)C3)C2)c2cc(C3CC3)c(-c3c(C)c(F)cc4[nH]ncc34)c(OCc3ccc(-c4cn([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](CO)c5ccc(-c6scnc6C)nc5)C(C)C)nn4)cc3)c2n1	C63H73FN14O9S	KRAS	P01116	VHL	WO-2024261256-A1
TPD-M6WSGZ	WO2024261256A1_4	.	CO[C@@H](C)COc1nc(NC2CN(C(=O)O[C@H]3C[C@H](N(C)C)C3)C2)c2cc(C3CC3)c(-c3c(C)c(F)cc4[nH]ncc34)c(OCc3ccc(-c4cn([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](CO)c5ccc(N6CCOC6=O)cc5)C(C)C)nn4)cc3)c2n1	C63H74FN13O11	KRAS	P01116	VHL	WO-2024261256-A1
TPD-R1DCJB	SCHEMBL30753923	(2S,4R)-1-[(2S)-2-[4-[4-[[6-cyclopropyl-4-[1-[3-[(dimethylamino)methyl]azetidine-1-carbonyl]azetidin-3-yl]oxy-7-(6-fluoro-5-methyl-1H-indazol-4-yl)-2-[(2S)-2-methoxypropoxy]quinolin-8-yl]oxymethyl]phenyl]triazol-1-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1R)-2-hydroxy-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CO[C@@H](C)COc1cc(OC2CN(C(=O)N3CC(CN(C)C)C3)C2)c2cc(C3CC3)c(-c3c(C)c(F)cc4[nH]ncc34)c(OCc3ccc(-c4cn([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](CO)c5ccc(-n6cncn6)cc5)C(C)C)nn4)cc3)c2n1	C63H73FN14O9	KRAS	P01116	VHL	WO-2024261256-A1
TPD-DUHUQH	SCHEMBL30753897	(2S,4R)-1-[(2S)-2-[4-[4-[[6-cyclopropyl-4-[1-[3-[(dimethylamino)methyl]azetidine-1-carbonyl]azetidin-3-yl]oxy-7-(6-fluoro-5-methyl-1H-indazol-4-yl)-2-[(2S)-2-methoxypropoxy]quinolin-8-yl]oxymethyl]phenyl]triazol-1-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1R)-2-hydroxy-1-[4-(4-methyl-1,3-oxazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CO[C@@H](C)COc1cc(OC2CN(C(=O)N3CC(CN(C)C)C3)C2)c2cc(C3CC3)c(-c3c(C)c(F)cc4[nH]ncc34)c(OCc3ccc(-c4cn([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](CO)c5ccc(-c6ocnc6C)cc5)C(C)C)nn4)cc3)c2n1	C65H75FN12O10	KRAS	P01116	VHL	WO-2024261256-A1
TPD-F5W89Z	WO2024261256A1_7	.	CO[C@@H](C)COc1cc(OC2CN(C(=O)N3CC[C@@H](N(C)C)C3)C2)c2cc(C3CC3)c(-c3c(C)c(F)cc4[nH]ncc34)c(OCc3ccc(-c4cn([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](CO)c5ccc(-n6cncn6)cc5)C(C)C)nn4)cc3)c2n1	C63H73FN14O9	KRAS	P01116	VHL	WO-2024261256-A1
TPD-3EW600	WO2024261256A1_8	.	CO[C@@H](C)COc1cc(OC2CN(C(=O)N3CC(CN(C)C)C3)C2)c2cc(C3CC3)c(-c3c(C)c(F)cc4[nH]ncc34)c(OCc3ccc(-c4cn([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](CO)c5ccc(N6CCOC6=O)cc5)C(C)C)nn4)cc3)c2n1	C64H75FN12O11	KRAS	P01116	VHL	WO-2024261256-A1
TPD-TLDLIJ	WO2024261256A1_9	.	COC(C)(C)COc1cc(OC2CN(C(=O)N3CC(CN(C)C)C3)C2)c2cc(C3CC3)c(-c3c(C)c(F)cc4[nH]ncc34)c(OCc3ccc(-c4cn([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](CO)c5ccc(-n6cncn6)cc5)C(C)C)nn4)cc3)c2n1	C64H75FN14O9	KRAS	P01116	VHL	WO-2024261256-A1
TPD-NKAAXS	WO2024261256A1_10	.	COC(C)(C)COc1cc(OC2CN(C(=O)N[C@H]3C[C@@H](N(C)C)C3)C2)c2cc(C3CC3)c(-c3c(C)c(F)cc4[nH]ncc34)c(OCc3ccc(-c4cn([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](CO)c5ccc(-n6cncn6)cc5)C(C)C)nn4)cc3)c2n1	C64H75FN14O9	KRAS	P01116	VHL	WO-2024261256-A1
TPD-ZGAWNB	SCHEMBL31297453	[3-(dimethylamino)cyclobutyl] 3-[[6-cyclopropyl-7-(6-fluoro-5-methyl-1H-indazol-4-yl)-8-[[4-[1-[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1R)-2-hydroxy-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]triazol-4-yl]phenyl]methoxy]-2-[(2S)-2-methoxypropoxy]quinazolin-4-yl]amino]azetidine-1-carboxylate	CO[C@@H](C)COc1nc(NC2CN(C(=O)O[C@H]3C[C@@H](N(C)C)C3)C2)c2cc(C3CC3)c(-c3c(C)c(F)cc4[nH]ncc34)c(OCc3ccc(-c4cn([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](CO)c5ccc(-c6scnc6C)cc5)C(C)C)nn4)cc3)c2n1	C64H74FN13O9S	KRAS	P01116	VHL	WO-2024261256-A1
TPD-IUDH3X	SCHEMBL31297449	(2S,4R)-1-[(2S)-2-[4-[4-[[6-cyclopropyl-4-[1-[2-(dimethylamino)ethylcarbamoyl]azetidin-3-yl]oxy-7-(6-fluoro-5-methyl-1H-indazol-4-yl)-2-[(2S)-2-methoxypropoxy]quinolin-8-yl]oxymethyl]phenyl]triazol-1-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1R)-2-hydroxy-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CO[C@@H](C)COc1cc(OC2CN(C(=O)NCCN(C)C)C2)c2cc(C3CC3)c(-c3c(C)c(F)cc4[nH]ncc34)c(OCc3ccc(-c4cn([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](CO)c5ccc(-n6cncn6)cc5)C(C)C)nn4)cc3)c2n1	C61H71FN14O9	KRAS	P01116	VHL	WO-2024261256-A1
TPD-OY7R5J	SCHEMBL31297438	[3-(dimethylamino)cyclobutyl] 3-[6-cyclopropyl-7-(6-fluoro-5-methyl-1H-indazol-4-yl)-8-[[4-[1-[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1R)-2-hydroxy-1-[4-(1,2,4-triazol-1-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]triazol-4-yl]phenyl]methoxy]-2-[(2S)-2-methoxypropoxy]quinolin-4-yl]oxyazetidine-1-carboxylate	CO[C@@H](C)COc1cc(OC2CN(C(=O)O[C@H]3C[C@@H](N(C)C)C3)C2)c2cc(C3CC3)c(-c3c(C)c(F)cc4[nH]ncc34)c(OCc3ccc(-c4cn([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](CO)c5ccc(-n6cncn6)cc5)C(C)C)nn4)cc3)c2n1	C63H72FN13O10	KRAS	P01116	VHL	WO-2024261256-A1
TPD-52LJCU	SCHEMBL30753916	(2S,4R)-1-[(2S)-2-[4-[4-[[6-cyclopropyl-4-[1-[3-[(dimethylamino)methyl]azetidine-1-carbonyl]azetidin-3-yl]oxy-7-(6-fluoro-5-methyl-1H-indazol-4-yl)-2-[(2S)-2-methoxypropoxy]quinolin-8-yl]oxymethyl]phenyl]triazol-1-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1R)-2-hydroxy-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CO[C@@H](C)COc1cc(OC2CN(C(=O)N3CC(CN(C)C)C3)C2)c2cc(C3CC3)c(-c3c(C)c(F)cc4[nH]ncc34)c(OCc3ccc(-c4cn([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](CO)c5ccc(-c6scnc6C)cc5)C(C)C)nn4)cc3)c2n1	C65H75FN12O9S	KRAS	P01116	VHL	WO-2024261256-A1
TPD-ZBTGUM	SCHEMBL31297455	(2S,4R)-1-[(2S)-2-[4-[4-[[6-cyclopropyl-7-(6-fluoro-5-methyl-1H-indazol-4-yl)-2-(oxan-4-yloxy)-4-[(1-pyrimidin-2-ylazetidin-3-yl)amino]quinazolin-8-yl]oxymethyl]phenyl]triazol-1-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1R)-2-hydroxy-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	Cc1ncsc1-c1ccc([C@H](CO)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](C(C)C)n2cc(-c3ccc(COc4c(-c5c(C)c(F)cc6[nH]ncc56)c(C5CC5)cc5c(NC6CN(c7ncccn7)C6)nc(OC6CCOCC6)nc45)cc3)nn2)cc1	C62H65FN14O7S	KRAS	P01116	VHL	WO-2024261256-A1
TPD-7X6L9U	WO2024261256A1_16	.	Cc1ncsc1-c1ccc([C@H](CO)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](C(C)C)n2cc(-c3ccc(COc4c(-c5c(C)c(F)cc6[nH]ncc56)c(C5CC5)cc5c(OC6CN(C(=O)NCCO)C6)nc(OC6CCOCC6)nc45)cc3)nn2)cc1	C61H67FN12O10S	KRAS	P01116	VHL	WO-2024261256-A1
TPD-F7BFOD	WO2024261256A1_17	.	CO[C@@H](C)COc1nc(OC2CN(C(=O)NCCN(C)C)C2)c2cc(C3CC3)c(-c3c(C)c(F)cc4[nH]ncc34)c(OCc3ccc(-c4cn([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](CO)c5ccc(-c6scnc6C)cc5)C(C)C)nn4)cc3)c2n1	C62H72FN13O9S	KRAS	P01116	VHL	WO-2024261256-A1
TPD-IAK9TO	WO2024261256A1_18	.	CNCCNC(=O)N1CC(Oc2nc(OC[C@H](C)OC)nc3c(OCc4ccc(-c5cn([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](CO)c6ccc(-c7scnc7C)cc6)C(C)C)nn5)cc4)c(-c4c(C)c(F)cc5[nH]ncc45)c(C4CC4)cc23)C1	C61H70FN13O9S	KRAS	P01116	VHL	WO-2024261256-A1
TPD-OH1O61	WO2024261256A1_19	.	CO[C@@H](C)COc1nc(N(C)[C@H]2CCN(C(=O)NCCN(C)C)C2)c2cc(C3CC3)c(-c3c(C)c(F)cc4[nH]ncc34)c(OCc3ccc(-c4cn(C(C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](CO)c5ccc(-c6scnc6C)cc5)C(C)C)nn4)cc3)c2n1	C64H77FN14O8S	KRAS	P01116	VHL	WO-2024261256-A1
TPD-GA0CFU	WO2024261256A1_20	.	CO[C@@H](C)COc1nc(N2CC(C#N)C2)c2cc(C3CC3)c(-c3c(C)c(F)cc4[nH]ncc34)c(OCc3ccc(-c4cn([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](CO)c5ccc(-c6scnc6C)cc5)C(C)C)nn4)cc3)c2n1	C58H61FN12O7S	KRAS	P01116	VHL	WO-2024261256-A1
TPD-GAWUIH	WO2024261256A1_22	.	CO[C@@H](C)COc1nc(OC2CN(C(=O)NCCN3CCCC3)C2)c2cc(C3CC3)c(-c3c(C)c(F)cc4[nH]ncc34)c(OCc3ccc(-c4cn([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](CO)c5ccc(-c6scnc6C)cc5)C(C)C)nn4)cc3)c2n1	C64H74FN13O9S	KRAS	P01116	VHL	WO-2024261256-A1
TPD-4AOPRY	WO2024261256A1_23	.	CO[C@@H](C)COc1nc(N[C@H]2C[C@H](OCCN(C)C)C2)c2cc(C3CC3)c(-c3c(C)c(F)cc4[nH]ncc34)c(OCc3ccc(-c4cn([C@H](C(=O)N5C[C@H](O)CC5C(=O)N[C@@H](CO)c5ccc(-c6scnc6C)cc5)C(C)C)nn4)cc3)c2n1	C62H73FN12O8S	KRAS	P01116	VHL	WO-2024261256-A1
TPD-4OXJ24	WO2024261256A1_24	.	CO[C@@H](C)COc1nc(N(C)C2CN(C(=O)CCCN(C)C)C2)c2cc(C3CC3)c(-c3c(C)c(F)cc4[nH]ncc34)c(OCc3ccc(-c4cn([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](CO)c5ccc(-c6scnc6C)cc5)C(C)C)nn4)cc3)c2n1	C64H76FN13O8S	KRAS	P01116	VHL	WO-2024261256-A1
TPD-X1Q2TF	WO2024261256A1_25	.	CO[C@@H](C)COc1nc(NC2CN(C(=O)N3CC(CN(C)C)C3)C2)c2cc(C3CC3)c(-c3c(C)c(F)cc4[nH]ncc34)c(OCc3ccc(-c4cn([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](CO)c5ccc(-c6scnc6C)cc5)C(C)C)nn4)cc3)c2n1	C64H75FN14O8S	KRAS	P01116	VHL	WO-2024261256-A1
TPD-46R3P5	WO2024261256A1_26	.	CO[C@@H](C)COc1nc(NC2CN(C(=S)N3CC(CN(C)C)C3)C2)c2cc(C3CC3)c(-c3c(C)c(F)cc4[nH]ncc34)c(OCc3ccc(-c4cn([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](CO)c5ccc(-n6cncn6)cc5)C(C)C)nn4)cc3)c2n1	C62H73FN16O7S	KRAS	P01116	VHL	WO-2024261256-A1
TPD-WMOFRW	WO2024261256A1_27	.	CO[C@@H](C)COc1nc(NC2CN(C(=O)N3CCN(C)CC3)C2)c2cc(C3CC3)c(-c3c(C)c(F)cc4[nH]ncc34)c(OCc3ccc(-c4cn([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](CO)c5ccc(-n6cncn6)cc5)C(C)C)nn4)cc3)c2n1	C61H71FN16O8	KRAS	P01116	VHL	WO-2024261256-A1
TPD-9M9CA3	SCHEMBL31297430	(2S,4R)-1-[(2S,3S)-2-[4-[4-[[6-cyclopropyl-4-[(3S)-1-[2-(dimethylamino)ethylcarbamoyl]pyrrolidin-3-yl]oxy-7-(6-fluoro-5-methyl-1H-indazol-4-yl)-2-[(2S)-2-methoxypropoxy]quinazolin-8-yl]oxymethyl]phenyl]triazol-1-yl]-3-methylpentanoyl]-4-hydroxy-N-[(1R)-2-hydroxy-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC[C@H](C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](CO)c1ccc(-c2scnc2C)cc1)n1cc(-c2ccc(COc3c(-c4c(C)c(F)cc5[nH]ncc45)c(C4CC4)cc4c(O[C@H]5CCN(C(=O)NCCN(C)C)C5)nc(OC[C@H](C)OC)nc34)cc2)nn1	C64H76FN13O9S	KRAS	P01116	VHL	WO-2024261256-A1
TPD-GP2HI7	WO2024261256A1_29	.	Cc1ncsc1-c1ccc([C@H](CO)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](C(C)C)n2cc(-c3ccc(COc4c(-c5c(C)c(F)cc6[nH]ncc56)c(C5CC5)cc5c(NCc6cccnc6)nc(OC6CCOCC6)nc45)cc3)nn2)cc1	C61H63FN12O7S	KRAS	P01116	VHL	WO-2024261256-A1
TPD-P5T21H	WO2024261256A1_30	.	Cc1c(F)cc2[nH]ncc2c1-c1c(C2CC2)cc2c(OC3CN(C(=O)NCCN(C)C)C3)nc(OC3CCOCC3)nc2c1OCc1ccc(-c2cn([C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](CO)c3ccc(-n4cccn4)cc3)C(C)C)nn2)cc1	C62H71FN14O9	KRAS	P01116	VHL	WO-2024261256-A1
TPD-AX842F	WO2024261256A1_31	.	Cc1ncsc1-c1ccc([C@H](CO)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](C(C)C)n2cc(-c3ccc(COc4c(-c5c(C)c(F)cc6[nH]ncc56)c(C5CC5)cc5c(OC6CN(C(=O)NCCN(C)C)C6)nc(OC6CCN(CC(F)F)CC6)nc45)cc3)nn2)cc1	C65H75F3N14O8S	KRAS	P01116	VHL	WO-2024261256-A1
TPD-ES7ER2	WO2024261256A1_32	.	Cc1c(F)cc2[nH]ncc2c1-c1c(C2CC2)cc2c(NC3CN(C(=O)NCCN(C)C)C3)nc(OC[C@@H]3CCCO3)nc2c1OCc1ccc(-c2cn([C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](CO)c3ccc(-n4cncn4)cc3)C(C)C)nn2)cc1	C61H71FN16O8	KRAS	P01116	VHL	WO-2024261256-A1
TPD-3BHGVV	WO2024261256A1_33	.	Cc1ncsc1C1C=CC([C@H](CO)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)C(C(C)C)n2cc(-c3ccc(COc4c(-c5c(C)c(F)cc6[nH]ncc56)c(C5CC5)cc5c(N(C)C6CN(C(=O)O[C@H]7CCN(C)C7)C6)nc(OC6CCOCC6)nc45)cc3)nn2)=CC1	C65H76FN13O9S	KRAS	P01116	VHL	WO-2024261256-A1
TPD-FH0ZUX	WO2024261256A1_34	.	CO[C@@H](C)COc1nc(NC2CN(C(=O)OCCN(C)C)C2)c2cc(C3CC3)c(-c3c(C)c(F)cc4[nH]ncc34)c(OCc3ccc(-c4cn([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](CO)c5ccc(-c6scnc6C)cc5)C(C)C)nn4)cc3)c2n1	C62H72FN13O9S	KRAS	P01116	VHL	WO-2024261256-A1
TPD-7DFK9S	WO2024261256A1_35	.	Cc1ncsc1-c1ccc([C@H](CO)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](C(C)C)n2cc(-c3ccc(COc4c5c(cc(C6CC6)c4-c4c(C)c(F)cc6[nH]ncc46)C(N4CC[C@H]4C(N)=O)=NC(OC4CCOCC4)N5)cc3)nn2)cc1	C59H65FN12O8S	KRAS	P01116	VHL	WO-2024261256-A1
TPD-2WC6JJ	WO2024261256A1_36	.	Cc1ncsc1-c1ccc([C@H](CO)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](C(C)C)n2cc(-c3ccc(COc4c(-c5c(C)c(F)cc6[nH]ncc56)c(C5CC5)cc5c(OC6CN(C(=O)NCCN(C)C)C6)nc(OCC(C)(C)CN(C)C)nc45)cc3)nn2)cc1	C65H79FN14O8S	KRAS	P01116	VHL	WO-2024261256-A1
TPD-TGAH4H	WO2024261256A1_38	.	Cc1ncsc1-c1ccc([C@H](CO)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](C(C)C)n2cc(-c3ccc(COc4c(-c5c(C)c(F)cc6[nH]ncc56)c(C5CC5)cc5c(N6CC(C#N)C6)nc(OC[C@@H]6CCN(C)C6)nc45)cc3)nn2)cc1	C60H64FN13O6S	KRAS	P01116	VHL	WO-2024261256-A1
TPD-7CO9ZQ	WO2024261256A1_39	.	Cc1ncsc1-c1ccc([C@H](CCO)NC(=O)[C@@H]2CC(=O)CN2C(=O)[C@H](C(C)C)n2cc(-c3ccc(COc4c(-c5c(C)c(F)cc6[nH]ncc56)c(C5CC5)cc5c(OC6CN(C(=O)NCCN(C)C)C6)nc(OC6CCOCC6)nc45)cc3)nn2)cc1	C64H72FN13O9S	KRAS	P01116	VHL	WO-2024261256-A1
TPD-58LXL6	SCHEMBL31613752	(2S,4R)-1-[(2S)-2-[[4-[[6-cyclopropyl-4-[1-[2-(dimethylamino)ethylcarbamoyl]azetidin-3-yl]oxy-7-(6-fluoro-5-methyl-1H-indazol-4-yl)-2-[(2S)-2-methoxypropoxy]quinazolin-8-yl]oxymethyl]benzoyl]amino]-3-methylbutanoyl]-4-hydroxy-N-[(1R)-2-hydroxy-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CO[C@@H](C)COc1nc(OC2CN(C(=O)NCCN(C)C)C2)c2cc(C3CC3)c(-c3c(C)c(F)cc4[nH]ncc34)c(OCc3ccc(C(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)N[C@@H](CO)c4ccc(-c5scnc5C)cc4)C(C)C)cc3)c2n1	C61H72FN11O10S	KRAS	P01116	VHL	WO-2024261256-A1
TPD-ATBWWE	WO2024261256A1_41	.	CO[C@@H](C)COc1cc(OC2CN(C(=O)CCCN(C)C)C2)c2cc(C3CC3)c(-c3c(C)c(F)cc4[nH]ncc34)c(OCc3ccc(-c4cn([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](CO)c5ccc(-n6cncn6)cc5)C(C)C)nn4)cc3)c2n1	C62H72FN13O9	KRAS	P01116	VHL	WO-2024261256-A1
TPD-KP2OGI	WO2024261256A1_42	.	CO[C@@H](C)COc1cc(OC2CN(C(=O)C3CN(C)C3)C2)c2cc(C3CC3)c(-c3c(C)c(F)cc4[nH]ncc34)c(OCc3ccc(-c4cn([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](CO)c5ccc(-n6cncn6)cc5)C(C)C)nn4)cc3)c2n1	C61H68FN13O9	KRAS	P01116	VHL	WO-2024261256-A1
TPD-92RP3M	WO2024261256A1_43	.	CO[C@@H](C)COc1cc(OC2CN(C(=O)NCCN(C)C)C2)c2cc(C3CC3)c(-c3c(C)c(F)cc4[nH]ncc34)c(OCc3ccc(-c4cn([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](CO)c5ccc(-c6scnc6C)cc5)C(C)C)nn4)cc3)c2n1	C63H73FN12O9S	KRAS	P01116	VHL	WO-2024261256-A1
TPD-08529Z	WO2025011655A1_nan	.	CC1=NC(N2CCC(=O)NC2=O)=C2C=CC=C(C3=CN=C(C4CCN(C[C@H]5CC[C@@H](N6C=C(NC(=O)C7=C8N=C(N9CCOCC9)C=CN8N=C7)C(C(F)F)=N6)CC5)CC4)C=C3)N12	C44H49F2N13O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-SPV7AH	WO2025011655A1_TM-003	.	CC(=O)NC(=O)N(C)C1=C2C=CC=C(C3=CN=C(OC4CCN(C[C@H]5CC[C@@H](N6C=C(NC(=O)C7=C8N=C(N9CCOCC9)C=CN8N=C7)C(C(F)F)=N6)CC5)CC4)C=C3)N2C(C)=N1	C44H51F2N13O5	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-O4GY6U	WO2025011655A1_TM-004	.	CC1=NC(N2CCC(=O)NC2=O)=C2C=CC=C(C3=CN(C4CCN(C[C@H]5CC[C@@H](N6C=C(NC(=O)C7=C8N=C(N9CCO[C@H](C)C9)C=CN8N=C7)C(C(F)F)=N6)CC5)CC4)N=C3)N12	C43H50F2N14O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-NAF40P	WO2025011655A1_TM-005	.	CC1=NC(N2CCC(=O)NC2=O)=C2C=CC=C(C3=CN(C4CCN(C[C@H]5CC[C@H](N6C=C(NC(=O)C7=C8N=C(N9CCO[C@@H](C)C9)C=CN8N=C7)C(C(F)F)=N6)CC5)CC4)N=C3)N12	C43H50F2N14O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-X5ZPFX	WO2025011655A1_TM-006	.	CC1=NC(N2CCC(=O)NC2=O)=C2C=CC=C(C3=CN(C4CCN(C[C@H]5CC[C@H](N6C=C(NC(=O)C7=C8N=C(N9CCCOCC9)C=CN8N=C7)C(C(F)F)=N6)CC5)CC4)N=C3)N12	C43H50F2N14O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-RLN7ZR	WO2025011655A1_TM-007	.	CC1=NC(N2CCC(=O)NC2=O)=C2C=CC=C(C3=CN(C4CCN(C[C@H]5CC[C@@H](N6C=C(NC(=O)C7C=NN8C=CC(N9CCOC%10(CC%10)C9)=NC78)C(C(F)F)=N6)CC5)CC4)N=C3)N12	C44H52F2N14O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-046W87	WO2025011655A1_TM-008	.	COC1CCN(C2=NC3=C(C(=O)NC4=CN([C@H]5CC[C@@H](CN6CCC(N7C=C(C8=CC=CC9=C(N%10CCC(=O)NC%10=O)N=C(C)N89)C=N7)CC6)CC5)N=C4C(F)F)C=NN3C=C2)CC1	C44H52F2N14O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-VR05IQ	WO2025011655A1_TM-009	.	CC1=NC(N2CCC(=O)NC2=O)=C2C=CC=C(C3=CN(C4CCN(C[C@H]5CC[C@@H](N6C=C(NC(=O)C7=C8N=C(N9CCOC[C@@H]9C)C=CN8N=C7)C(C(F)F)=N6)CC5)CC4)N=C3)N12	C43H50F2N14O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-XG1YIM	WO2025011655A1_TM-010	.	CC1=NC(N2CCC(=O)NC2=O)=C2C=CC=C(C3=CN(C4CCN(C[C@H]5CC[C@H](N6C=C(NC(=O)C7=C8N=C(N9CCOC[C@H]9C)C=CN8N=C7)C(C(F)F)=N6)CC5)CC4)N=C3)N12	C43H50F2N14O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-BK74VX	WO2025011655A1_TM-011	.	CC1=NC(N2CCC(=O)NC2=O)=C2C=CC=C(C3=CN(C4CCN(C[C@H]5CC[C@@H](N6C=C(NC(=O)C7=C8N=C(N9CCC%10(COC%10)C9)C=CN8N=C7)C(C(F)F)=N6)CC5)CC4)N=C3)N12	C44H50F2N14O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-L2OFQX	WO2025011655A1_TM-012	.	CC1=NC(N2CCC(=O)NC2=O)=C2C=CC=C(C3=CN(C4CCN(C[C@H]5CC[C@H](N6C=C(NC(=O)C7=C8N=C(N9CC%10(COC%10)C9)C=CN8N=C7)C(C(F)F)=N6)CC5)CC4)N=C3)N12	C43H48F2N14O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-MFN738	WO2025011655A1_TM-013	.	CC1=NC(N2CCC(=O)NC2=O)=C2C=CC=C(C3=CN(C4CCN(C[C@H]5CC[C@H](N6C=C(NC(=O)C7=C8N=C(N9CC%10COCC%10C9)C=CN8N=C7)C(C(F)F)=N6)CC5)CC4)N=C3)N12	C44H50F2N14O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-V0ECYH	WO2025011655A1_TM-014	.	CC1=C(N2CCC(=O)NC2=O)N2C=CC(C3=CN(C4CCN(C[C@H]5CC[C@@H](N6C=C(NC(=O)C7=C8N=C(N9CCOCC9)C=CN8N=C7)C(C(F)F)=N6)CC5)CC4)N=C3)=CC2=N1	C42H48F2N14O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-6UY427	WO2025011655A1_TM-015	.	CC1=CC=C(N2CCC(=O)NC2=O)C2=NC=C(C3=CN(C4CCN(C[C@H]5CC[C@@H](N6C=C(NC(=O)C7=C8N=C(N9CCOCC9)C=CN8N=C7)C(C(F)F)=N6)CC5)CC4)N=C3)N12	C42H48F2N14O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-I9YDX8	WO2025011655A1_TM-016	.	O=C1CCN(C2=CC=CN3C(C4=CN(C5CCN(C[C@H]6CC[C@@H](N7C=C(NC(=O)C8=C9N=C(N%10CCOCC%10)C=CN9N=C8)C(C(F)F)=N7)CC6)CC5)N=C4)=CN=C23)C(=O)N1	C41H46F2N14O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-0SEXUT	WO2025011655A1_TM-017	.	CC1=C(C2=CN(C3CCN(C[C@H]4CC[C@H](N5C=C(NC(=O)C6=C7N=C(N8CCOCC8)C=CN7N=C6)C(C(F)F)=N5)CC4)CC3)N=C2)N2C=CC=C(N3CCC(=O)NC3=O)C2=N1	C42H48F2N14O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-2QXKZL	WO2025011655A1_TM-018	.	CC1=NN2C=C(C3=CN(C4CCN(C[C@H]5CC[C@@H](N6C=C(NC(=O)C7=C8N=C(N9CCOCC9)C=CN8N=C7)C(C(F)F)=N6)CC5)CC4)C=C3)C=CC2=C1N1CCC(=O)NC1=O	C43H49F2N13O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-MBD87A	WO2025011655A1_TM-019	.	CC1=NN2C(C3=CN(C4CCN(C[C@H]5CC[C@@H](N6C=C(NC(=O)C7=C8N=C(N9CCOCC9)C=CN8N=C7)C(C(F)F)=N6)CC5)CC4)N=C3)=CC=CC2=C1N1CCC(=O)NC1=O	C42H48F2N14O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-UGXML3	WO2025011655A1_TM-020	.	CC1=C(N2CCC(=O)NC2=O)N=C2C=C(C3=CN(C(C)CCN(C)C[C@H]4CC[C@H](N5C=C(NC(=O)C6=C7N=C(N8CCOCC8)C=CN7N=C6)C(C(F)F)=N5)CC4)N=C3)C=CN21	C42H50F2N14O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-M6FBS8	WO2025011655A1_TM-021	.	CC1=C(N2CCC(=O)NC2=O)N=C2C=CC(C3=CN(C4CCN(C[C@H]5CC[C@@H](N6C=C(NC(=O)C7=C8N=C(N9CCOCC9)C=CN8N=C7)C(C(F)F)=N6)CC5)CC4)N=C3)=CN21	C42H48F2N14O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-YUBTGJ	WO2025011655A1_TM-022	.	CC1=C2C=C(C3=CN(C(C)CCN(C)C[C@H]4CC[C@H](N5C=C(NC(=O)C6=C7N=C(N8CCOCC8)C=CN7N=C6)C(C(F)F)=N5)CC4)N=C3)C=CN2N=C1N1CCC(=O)NC1=O	C42H50F2N14O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-2EZY5W	WO2025011655A1_TM-023	.	CC1=C2C=CC(C3=CN(C4CCN(C[C@H]5CC[C@@H](N6C=C(NC(=O)C7=C8N=C(N9CCOCC9)C=CN8N=C7)C(C(F)F)=N6)CC5)CC4)N=C3)=CN2N=C1N1CCC(=O)NC1=O	C42H48F2N14O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-CSBYJU	WO2025011655A1_TM-024	.	CC1=NC(N2CCC(=O)NC2=O)=C2C=CC=C(C#CCOC3CCN(C[C@H]4CC[C@@H](N5C=C(NC(=O)C6=C7N=C(N8CCOCC8)C=CN7N=C6)C(C(F)F)=N5)CC4)CC3)N12	C42H48F2N12O5	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-3KEBGL	WO2025011655A1_TM-029	.	COC1=CC2=NN([C@H]3CC[C@H](CN4CCN(C5=CC=CC6=C5C(C)=NN6C5CCC(=O)NC5=O)CC4)CC3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C39H42F3N9O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-WLCDQA	WO2025011655A1_TM-030	.	COC1=CC2=NN([C@H]3CC[C@@H](CN4CCN(C5=CC=CC6=C5C(C)=NN6C5CCC(=O)NC5=O)CC4)CC3)C=C2C=C1NC(=O)C1=C2N=CC=CN2N=C1	C39H43N11O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-2Q8TYV	WO2025011655A1_TM-031	.	COC1=CC2=NN([C@H]3CC[C@@H](CN4CCN(C5=CC=CC6=C5C(C)=NN6C5CCC(=O)NC5=O)CC4)CC3)C=C2C=C1NC(=O)C1=C2N=C(C)C=CN2N=C1	C40H45N11O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-QX62S1	WO2025011655A1_TM-032	.	COC1=CC2=NN([C@H]3CC[C@@H](CN4CCN(C5=CC=CC6=C5C(C)=NN6C5CCC(=O)NC5=O)CC4)CC3)C=C2C=C1NC(=O)C1=NC(C)=CC=C1	C39H45N9O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-8Y12EI	WO2025011655A1_TM-033	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CCN(C[C@H]3CC[C@@H](N4C=C5C=C(NC(=O)C6=C7N=CC=CN7N=C6)C(N6CCOCC6)=CC5=N4)CC3)CC1)=CC=C2	C42H48N12O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-G94VJ2	WO2025011655A1_TM-034	.	COC1=CC2=NN([C@H]3CC[C@H](CN4CC5CN(C6=CC=CC7=C6N(C)N=C7C6CCC(=O)NC6=O)CC5C4)CC3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C41H44F3N9O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-2348GJ	WO2025011655A1_TM-035	.	COC1=CC2=NN([C@H]3CC[C@@H](CN4CC5CN(C6=CC=CC7=C6C(C)=NN7C6CCC(=O)NC6=O)CC5C4)CC3)C=C2C=C1NC(=O)C1=NC(C)=CC=C1	C41H47N9O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-WS7Z8D	WO2025011655A1_TM-036	.	COC1=CC2=NN([C@H]3CC[C@H](CN4CC5CN(C6=CC=CC7=C6C(C)=NN7C6CCC(=O)NC6=O)CC5C4)CC3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C41H44F3N9O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-ATJNBA	WO2025011655A1_TM-037	.	COC1=CC2=NN([C@H]3CC[C@H](CN4CC5CN(C6=CC=CC7=C6C(C)=NN7C6CCC(=O)NC6=O)CC5C4)CC3)C=C2C=C1NC(=O)C1=C2N=CC=CN2N=C1	C41H45N11O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-8WUUNQ	WO2025011655A1_TM-038	.	COC1=CC2=NN([C@H]3CC[C@@H](CN4CC5CN(C6=CC=CC7=C6C(C)=NN7C6CCC(=O)NC6=O)CC5C4)CC3)C=C2C=C1NC(=O)C1=C2N=C(C)C=CN2N=C1	C42H47N11O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-FTV28H	WO2025011655A1_TM-039	.	COC1=CC2=NN([C@H]3CC[C@H](CN4CC5CN(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)N=C7C)CC5C4)CC3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C41H44F3N9O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-EKS3NO	WO2025011655A1_TM-040	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C=C(N1CC3CN(C[C@H]4CC[C@H](N5C=C6C=C(NC(=O)C7=C8N=CC=CN8N=C7)C(N7CCOCC7)=CC6=N5)CC4)CC3C1)C=C2	C44H50N12O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-TXLQQZ	WO2025011655A1_TM-041	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CC3(CCN(C[C@H]4CC[C@@H](N5C=C6C=C(NC(=O)C7=C8N=CC=CN8N=C7)C(N7CCOCC7)=CC6=N5)CC4)CC3)C1)=CC=C2	C45H52N12O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-W538RZ	WO2025011655A1_TM-042	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CCC3(CC1)CN(C[C@H]1CC[C@@H](N4C=C5C=C(NC(=O)C6=C7N=CC=CN7N=C6)C(N6CCOCC6)=CC5=N4)CC1)C3)=CC=C2	C45H52N12O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-DGXS4U	WO2025011655A1_TM-043	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1C[C@H]3CC[C@@H]1CN3C[C@H]1CC[C@H](N3C=C4C=C(NC(=O)C5=C6N=CC=CN6N=C5)C(N5CCOCC5)=CC4=N3)CC1)=CC=C2	C44H50N12O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-R165UL	WO2025011655A1_TM-044	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1C[C@@H]3C[C@H]1CN3CC1CCC(N3C=C4C=C(NC(=O)C5=C6N=CC=CN6N=C5)C(N5CCOCC5)=CC4=N3)CC1)=CC=C2	C43H48N12O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-6NHSPG	WO2025011655A1_TM-045	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CCN(C[C@H]3CC[C@H](N4C=C5C=C(NC(=O)C6=C7N=CC=CN7N=C6)C(N6C[C@@H]7C[C@H]6CO7)=CC5=N4)CC3)CC1)=CC=C2	C43H48N12O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-MRQ82M	WO2025011655A1_TM-046	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CC3CN(C[C@H]4CC[C@H](N5C=C6C=C(NC(=O)C7=C8N=CC=CN8N=C7)C(N7C[C@H]8C[C@@H]7CO8)=CC6=N5)CC4)CC3C1)=CC=C2	C45H50N12O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-R74T1S	WO2025011655A1_TM-047	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CCN(C[C@H]3CC[C@H](N4C=C5C=C(NC(=O)C6=C7N=CC=CN7N=C6)C(N6CCOC7(CC7)C6)=CC5=N4)CC3)CC1)=CC=C2	C44H50N12O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-9IB0OO	WO2025011655A1_TM-048	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CC3CN(C[C@H]4CC[C@H](N5C=C6C=C(NC(=O)C7=C8N=CC=CN8N=C7)C(N7CCOC8(CC8)C7)=CC6=N5)CC4)CC3C1)=CC=C2	C46H52N12O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-UR7TN8	WO2025011655A1_TM-049	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CCN(C[C@H]3CC[C@H](N4C=C5C=C(NC(=O)C6=C7N=CC=CN7N=C6)C(C(F)F)=CC5=N4)CC3)CC1)=CC=C2	C39H41F2N11O3	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-YEXZX0	WO2025011655A1_TM-050	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CC3CN(C[C@H]4CC[C@H](N5C=C6C=C(NC(=O)C7=C8N=CC=CN8N=C7)C(C(F)F)=CC6=N5)CC4)CC3C1)=CC=C2	C41H43F2N11O3	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-3BQ6XL	WO2025011655A1_TM-051	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CCC(CN3CCC(N4C=C5C=C(NC(=O)C6=C7N=CC=CN7N=C6)C(N6CCOCC6)=CC5=N4)CC3)CC1)=CC=C2	C42H48N12O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-SVCOVL	WO2025011655A1_TM-052	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CCN(CC3CCC(N4C=C5C=C(NC(=O)C6=C7N=CC=CN7N=C6)C(N6CCO[C@@H](C)C6)=CC5=N4)CC3)CC1)=CC=C2	C43H50N12O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-WHHO2W	WO2025011655A1_TM-053	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CC3CN(C[C@H]4CC[C@@H](N5C=C6C=C(NC(=O)C7=C8N=CC=CN8N=C7)C(N7CCO[C@@H](C)C7)=CC6=N5)CC4)CC3C1)=CC=C2	C45H52N12O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-T2PUF4	WO2025011655A1_TM-054	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CCN(CC3CCC(N4C=C5C=C(NC(=O)C6=C7N=CC=CN7N=C6)C(N6CCO[C@H](C)C6)=CC5=N4)CC3)CC1)=CC=C2	C43H50N12O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-2PV4CM	WO2025011655A1_TM-055	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CC3CN(C[C@H]4CC[C@@H](N5C=C6C=C(NC(=O)C7=C8N=CC=CN8N=C7)C(N7CCO[C@H](C)C7)=CC6=N5)CC4)CC3C1)=CC=C2	C45H52N12O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-GH8CPN	WO2025011655A1_TM-056	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(OC1CCN(C[C@H]3CC[C@H](N4C=C5C=C(NC(=O)C6=C7N=CC=CN7N=C6)C(N6CCOCC6)=CC5=N4)CC3)CC1)=CC=C2	C43H49N11O5	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-GEMWQS	WO2025011655A1_TM-057	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CC3CN(C[C@H]4CC[C@H](N5C=C6C=C(NC(=O)C7=C8N=CC=CN8N=C7)C(N7CCOCC7)=CC6=N5)CC4)CC3C1)=CC=C2	C44H50N12O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-19ZITK	WO2025011655A1_TM-058	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CCN(C[C@H]3CC[C@@H](N4CC5=C(C=C(N6CCOCC6)C(NC(=O)C6=C7N=CC=CN7N=C6)=C5)C4=O)CC3)CC1)=CC=C2	C43H49N11O5	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-D0A68Y	WO2025011655A1_TM-059	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CC3CN(C[C@H]4CC[C@@H](N5CC6=C(C=C(N7CCOCC7)C(NC(=O)C7=C8N=CC=CN8N=C7)=C6)C5=O)CC4)CC3C1)=CC=C2	C45H51N11O5	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-3CQWSP	WO2025011655A1_TM-060	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(OC1CCN(C[C@H]3CC[C@H](N4CC5=C(C=C(N6CCOCC6)C(NC(=O)C6=C7N=CC=CN7N=C6)=C5)C4=O)CC3)CC1)=CC=C2	C44H50N10O6	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-Y34F2I	WO2025011655A1_TM-061	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CCN(C[C@H]3CC[C@H](N4C=C5C=C(NC(=O)C6=C7N=CC=CN7N=C6)C(N6CC7C[C@@H]6CO7)=CC5=N4)CC3)CC1)=CC=C2	C43H48N12O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-K990H2	WO2025011655A1_TM-063	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CCN(C[C@H]3CC[C@H](N4CC5=C(C=C(N6CCO[C@H](C)C6)C(NC(=O)C6=C7N=CC=CN7N=C6)=C5)C4=O)CC3)CC1)=CC=C2	C44H51N11O5	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-B5BVVU	WO2025011655A1_TM-064	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CCN(C[C@H]3CC[C@@H](N4CC5=C(C=C(N6CCCOCC6)C(NC(=O)C6=C7N=CC=CN7N=C6)=C5)C4=O)CC3)CC1)=CC=C2	C44H51N11O5	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-W5NIUP	WO2025011655A1_TM-065	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CCN(C[C@H]3CC[C@H](N4CC5=C(C=C(N(C)C)C(NC(=O)C6=C7N=CC=CN7N=C6)=C5)C4=O)CC3)CC1)=CC=C2	C41H47N11O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-VYCSWX	WO2025011655A1_TM-066	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CCC(CN3CCC(N4CC5=C(C=C(N(C)C)C(NC(=O)C6=C7N=CC=CN7N=C6)=C5)C4=O)CC3)CC1)=CC=C2	C41H47N11O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-JN1Y3A	WO2025011655A1_TM-067	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CCC(CN3CCC(N4CC5=C(C=C(N6CCOCC6)C(NC(=O)C6=C7N=CC=CN7N=C6)=C5)C4=O)CC3)CC1)=CC=C2	C43H49N11O5	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-M5KHGW	WO2025011655A1_TM-068	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CCC(CN3CCC(N4CC5=C(C=C(N6CCCOCC6)C(NC(=O)C6=C7N=CC=CN7N=C6)=C5)C4=O)CC3)CC1)=CC=C2	C44H51N11O5	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-UXD03D	WO2025011655A1_TM-069	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CCC(CN3CCC(N4CC5=C(C=C(N6CCO[C@H](C)C6)C(NC(=O)C6=C7N=CC=CN7N=C6)=C5)C4=O)CC3)CC1)=CC=C2	C44H51N11O5	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-V7YNNJ	WO2025011655A1_TM-070	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CCN(C[C@H]3CC[C@@H](N4C=C5C=C(NC(=O)C6=C7N=CC=CN7N=C6)C(N(C)C)=CC5=N4)CC3)CC1)=CC=C2	C40H46N12O3	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-5YWC2W	WO2025011655A1_TM-071	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CCC(CN3CCC(N4C=C5C=C(NC(=O)C6=C7N=CC=CN7N=C6)C(N(C)C)=CC5=N4)CC3)CC1)=CC=C2	C40H46N12O3	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-Y9QP05	WO2025011655A1_TM-072	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CCC(CN3CCC(N4C=C5C=C(NC(=O)C6=C7N=CC=CN7N=C6)C(N6CCO[C@H](C)C6)=CC5=N4)CC3)CC1)=CC=C2	C43H50N12O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-XIM2VL	WO2025011655A1_TM-073	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CCN(C[C@H]3CC[C@H](N4C=C5C=C(NC(=O)C6=C7N=CC=CN7N=C6)C(N6CCOC[C@H]6C)=CC5=N4)CC3)CC1)=CC=C2	C43H50N12O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-SKWY4P	WO2025011655A1_TM-074	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CCN(C[C@H]3CC[C@@H](N4C=C5C=C(NC(=O)C6=C7N=CC=CN7N=C6)C(N6CCOC[C@@H]6C)=CC5=N4)CC3)CC1)=CC=C2	C43H50N12O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-00GKH5	WO2025011655A1_TM-075	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CC[C@@H](CN3CCC(N4CC5=C(C=C(N6CCOCC6)C(NC(=O)C6=C7N=CC=CN7N=C6)=C5)C4=O)CC3)C1)=CC=C2	C42H47N11O5	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-9VNSKA	WO2025011655A1_TM-076	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CC[C@H](CN3CCC(N4CC5=C(C=C(N6CCOCC6)C(NC(=O)C6=C7N=CC=CN7N=C6)=C5)C4=O)CC3)C1)=CC=C2	C42H47N11O5	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-W9XUYX	WO2025011655A1_TM-077	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CC[C@@H](CN3CCC(N4C=C5C=C(NC(=O)C6=C7N=CC=CN7N=C6)C(N6CCOCC6)=CC5=N4)CC3)C1)=CC=C2	C41H46N12O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-LYCMCS	WO2025011655A1_TM-078	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CC[C@H](CN3CCC(N4C=C5C=C(NC(=O)C6=C7N=CC=CN7N=C6)C(N6CCOCC6)=CC5=N4)CC3)C1)=CC=C2	C41H46N12O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-N7RB6E	WO2025011655A1_TM-079	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CCN(C[C@H]3CC[C@@H](N4C=C5C=C(NC(=O)C6=C7N=CC=CN7N=C6)C(N6CCCOCC6)=CC5=N4)CC3)CC1)=CC=C2	C43H50N12O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-TDIJSL	WO2025011655A1_TM-080	.	CC1=NN(C2CCC(=O)NC2=O)C2=CC=CC(N3CC[C@H](CN4CCC(N5CC6=C(C=C(N(C)C)C(NC(=O)C7=C8N=CC=CN8N=C7)=C6)C5=O)CC4)C3)=C21	C40H45N11O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-8I1GFN	WO2025011655A1_TM-081	.	CC1=NN(C2CCC(=O)NC2=O)C2=CC=CC(N3CC[C@@H](CN4CCC(N5CC6=C(C=C(N(C)C)C(NC(=O)C7=C8N=CC=CN8N=C7)=C6)C5=O)CC4)C3)=C21	C40H45N11O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-EBIN3A	WO2025011655A1_TM-082	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CCC(CN3CCC(N4C=C5C=C(NC(=O)C6=C7N=CC=CN7N=C6)C(N6CCCOCC6)=CC5=N4)CC3)CC1)=CC=C2	C43H50N12O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-PBNXXN	WO2025011655A1_TM-083	.	CC1=NN(C2CCC(=O)NC2=O)C2=CC=CC(N3CCN(CCN4CCC(N5C=C6C=C(NC(=O)C7=C8N=CC=CN8N=C7)C(N(C)C)=CC6=N5)CC4)CC3)=C21	C40H47N13O3	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-6NZTZZ	WO2025011655A1_TM-084	.	CC1=NN(C2CCC(=O)NC2=O)C2=CC=CC(N3CCN(CCN4CCC(N5C=C6C=C(NC(=O)C7=C8N=CC=CN8N=C7)C(N7CCOCC7)=CC6=N5)CC4)CC3)=C21	C42H49N13O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-EJHS1V	WO2025011655A1_TM-085	.	CCC(CCN(C)CC1CCN(C2=C(F)C=CC3=C2C(C)=NN3C2CCC(=O)NC2=O)CC1)N1CC2=C(C=C(N(C)C)C(NC(=O)C3=C4N=CC=CN4N=C3)=C2)C1=O	C42H50FN11O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-GWLJ4H	WO2025011655A1_TM-086	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CCC(CN3CCC(N4CC5=C(C=C(N(C)C)C(NC(=O)C6=C7N=CC=CN7N=C6)=C5)C4=O)CC3)CC1)=CC(F)=C2	C41H46FN11O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-D420XJ	WO2025011655A1_TM-087	.	CN(C)C1=CC2=C(C=C1NC(=O)C1=C3N=CC=CN3N=C1)CN(C1CCN(CC3CCN(C4=CC=CC5=C4C(C4CC4)=NN5C4CCC(=O)NC4=O)CC3)CC1)C2=O	C43H49N11O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-SGVBIS	WO2025011655A1_TM-088	.	CCC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CCC(CN3CCC(N4CC5=C(C=C(N(C)C)C(NC(=O)C6=C7N=CC=CN7N=C6)=C5)C4=O)CC3)CC1)=CC=C2	C42H49N11O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-J59GF6	WO2025011655A1_TM-089	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CCC(CN3CCC(N4CC5=C(C=C(N(C)C)C(NC(=O)C6=C7N=CC=CN7N=C6)=C5)C4=O)CC3)CC1)=C(Cl)C=C2	C41H46ClN11O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-X8J3BU	WO2025011655A1_TM-090	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CCC(CN3CCC(N4CC5=C(C=C(N(C)C)C(NC(=O)C6=C7N=CC=CN7N=C6)=C5)C4=O)CC3)CC1)=CC(Cl)=C2	C41H46ClN11O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-CHY21D	WO2025011655A1_TM-091	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CC[C@@H](CN3CCC(N4C=C5C=C(NC(=O)C6=C7N=CC=CN7N=C6)C(N(C)C)=CC5=N4)CC3)C1)=CC=C2	C39H44N12O3	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-17GLWD	WO2025011655A1_TM-092	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CC[C@H](CN3CCC(N4C=C5C=C(NC(=O)C6=C7N=CC=CN7N=C6)C(N(C)C)=CC5=N4)CC3)C1)=CC=C2	C39H44N12O3	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-2M0NTL	WO2025011655A1_TM-093	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CCC(CN3CCC(N4C=C5C=C(NC(=O)C6=C7N=CC=CN7N=C6)C(N(C)C)=CC5=N4)CC3)CC1)=C(F)C=C2	C40H45FN12O3	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-VVTMJQ	WO2025011655A1_TM-094	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CCC(CN3CCC(N4C=C5C=C(NC(=O)C6=C7N=CC=CN7N=C6)C(N(C)C)=CC5=N4)CC3)CC1)=CC(F)=C2	C40H45FN12O3	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-8XR8IT	WO2025011655A1_TM-095	.	CCC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CCC(CN3CCC(N4C=C5C=C(NC(=O)C6=C7N=CC=CN7N=C6)C(N(C)C)=CC5=N4)CC3)CC1)=CC=C2	C41H48N12O3	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-UQRP5K	WO2025011655A1_TM-096	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CCCN(C[C@H]3CC[C@H](N4C=C5C=C(NC(=O)C6=C7N=CC=CN7N=C6)C(N(C)C)=CC5=N4)CC3)CC1)=CC=C2	C41H48N12O3	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-QV50PJ	WO2025011655A1_TM-097	.	CN(C)C1=CC2=NN([C@H]3CC[C@H](CN4CCN(C5=CC=CC6=C5N(C)N=C6C5CCC(=O)NC5=O)CC4)CC3)C=C2C=C1NC(=O)C1=C2N=CC=CN2N=C1	C40H46N12O3	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-RH9J0Y	WO2025011655A1_TM-098	.	CN(C)C1=CC2=NN([C@H]3CC[C@H](CN4CCN(C5=CC=CC6=C5N(C)N=C6N5CCC(=O)NC5=O)CC4)CC3)C=C2C=C1NC(=O)C1=C2N=CC=CN2N=C1	C39H45N13O3	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-N2HQNL	WO2025011655A1_TM-099	.	[2H]C([2H])([2H])N(C1=CC2=NN([C@H]3CC[C@H](CN4CCN(C5=CC=CC6=C5C(C)=NN6C5CCC(=O)NC5=O)CC4)CC3)C=C2C=C1NC(=O)C1=C2N=CC=CN2N=C1)C([2H])([2H])[2H]	C40H46N12O3	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-KJ1OW8	WO2025011655A1_TM-100	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CC3C(CN4CCC(N5C=C6C=C(NC(=O)C7=C8N=CC=CN8N=C7)C(N(C)C)=CC6=N5)CC4)C3C1)=CC=C2	C40H44N12O3	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-KRVGZU	WO2025011655A1_TM-101	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CCC3(CC1)CN(C[C@H]1CC[C@@H](N4C=C5C=C(NC(=O)C6=C7N=CC=CN7N=C6)C(N(C)C)=CC5=N4)CC1)C3)=CC=C2	C43H50N12O3	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-TW5C1L	WO2025011655A1_TM-102	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CC3CN(C[C@H]4CC[C@H](N5C=C6C=C(NC(=O)C7=C8N=CC=CN8N=C7)C(N(C)C)=CC6=N5)CC4)CC3C1)=CC=C2	C42H48N12O3	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-TUP599	WO2025011655A1_TM-103	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CCN(C[C@H]3CC[C@@H](N4C=C5C=C(NC(=O)C6=C7N=CC=CN7N=C6)C(N(C)C)=CC5=N4)CC3)CC1)=NC=C2	C39H45N13O3	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-06F77E	WO2025011655A1_TM-104	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CCC(CN3CCC(N4C=C5C=C(NC(=O)C6=C7N=CC=CN7N=C6)C(N(C)C)=CC5=N4)CC3)CC1)=NC=C2	C39H45N13O3	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-W5R6AC	WO2025011655A1_TM-105	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CCN(C[C@H]3CC[C@H](N4C=C5C=C(NC(=O)C6=C7N=CC=CN7N=C6)C(N(C)C)=CC5=N4)CC3)CC1)=CN=C2	C39H45N13O3	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-0GU8CZ	WO2025011655A1_TM-106	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CCC(CN3CCC(N4C=C5C=C(NC(=O)C6=C7N=CC=CN7N=C6)C(N(C)C)=CC5=N4)CC3)CC1)=CN=C2	C39H45N13O3	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-D6TX2E	WO2025011655A1_TM-107	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CCN(C[C@H]3CC[C@@H](N4C=C5C=C(NC(=O)C6=C7N=CC=CN7N=C6)C(N(C)C)=CC5=N4)CC3)CC1)=CC=N2	C39H45N13O3	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-LZPNVU	WO2025011655A1_TM-108	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CCC(CN3CCC(N4C=C5C=C(NC(=O)C6=C7N=CC=CN7N=C6)C(N(C)C)=CC5=N4)CC3)CC1)=CC=N2	C39H45N13O3	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-CV55FH	WO2025011655A1_TM-109	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CCN(C[C@H]3CC[C@H](N4C=C5C=C(NC(=O)C6=C7N=CC=CN7N=C6)C(N6CCO[C@H](C)C6)=CC5=N4)CC3)CC1)=CN=C2	C42H49N13O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-REUJ8R	WO2025011655A1_TM-110	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CCN(C[C@H]3CC[C@H](N4C=C5C=C(NC(=O)C6=C7N=CC=CN7N=C6)C(N6CCOCC6)=CC5=N4)CC3)CC1)=CN=C2	C41H47N13O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-HP2DZP	WO2025011655A1_TM-111	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CCC3(CC1)CN(C[C@H]1CC[C@@H](N4C=C5C=C(NC(=O)C6=C7N=CC=CN7N=C6)C(N6CCO[C@H](C)C6)=CC5=N4)CC1)C3)=CC=C2	C46H54N12O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-J3JKK1	WO2025011655A1_TM-112	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CC3CN(C[C@H]4CC[C@@H](N5C=C6C=C(NC(=O)C7=C8N=CC=CN8N=C7)C(N7CCOC[C@@H]7C)=CC6=N5)CC4)CC3C1)=CC=C2	C45H52N12O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-1S40DV	WO2025011655A1_TM-113	.	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CCC3(CC1)CN(C[C@H]1CC[C@@H](N4C=C5C=C(NC(=O)C6=C7N=CC=CN7N=C6)C(N(C)C)=CC5=N4)CC1)C3)=NC=C2	C42H49N13O3	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-9UEK4R	WO2025011655A1_TM-114	.	CC1=NN(C2CCC(=O)NC2=O)C2=NC=CC(N3CCC4(CC3)CN(C[C@H]3CC[C@H](N5C=C6C=C(NC(=O)C7=C8N=CC=CN8N=C7)C(N(C)C)=CC6=N5)CC3)C4)=C12	C42H49N13O3	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-65OQ7J	WO2025011655A1_TM-116	.	COC1=CC2=NN([C@H]3CC[C@H](CN4CCC(C5=CC6=NC(C)=C(N7CCC(=O)NC7=O)N6C=C5)CC4)CC3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C39H42F3N9O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-468CPH	WO2025011655A1_TM-117	.	COC1=CC2=NN([C@H]3CC[C@H](CN4CCC(C5=CN=C6C(N7CCC(=O)NC7=O)=CC=C(C)N56)CC4)CC3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C39H42F3N9O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-X8FS50	WO2025011655A1_TM-118	.	COC1=CC2=NN([C@H]3CC[C@H](CN4CCC(C5=CN=C6C(N7CCC(=O)NC7=O)=CC=CN56)CC4)CC3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C38H40F3N9O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-7979JM	WO2025011655A1_TM-119	.	COC1=CC2=NN([C@H]3CC[C@H](CN4CCC(C5=C(C)N=C6C(N7CCC(=O)NC7=O)=CC=CN65)CC4)CC3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C39H42F3N9O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-JCKGUR	WO2025011655A1_TM-120	.	COC1=CC2=NN([C@H]3CC[C@@H](CN4CCC(C5=CN6N=C(C)C(N7CCC(=O)NC7=O)=C6C=C5)CC4)CC3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C39H42F3N9O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-0S46D2	WO2025011655A1_TM-121	.	COC1=CC2=NN([C@H]3CC[C@@H](CN4CCC(C5=CC=CC6=C(N7CCC(=O)NC7=O)C(C)=NN56)CC4)CC3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C39H42F3N9O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-070PRU	WO2025011655A1_TM-122	.	COC1=CC2=NN([C@H]3CC[C@H](CN4CCC(C5=CC6=NC(N7CCC(=O)NC7=O)=C(C)N6C=C5)CC4)CC3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C39H42F3N9O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-SPZNKX	WO2025011655A1_TM-123	.	COC1=CC2=NN([C@H]3CC[C@@H](CN4CCC(C5=CN6C(=NC(N7CCC(=O)NC7=O)=C6C)C=C5)CC4)CC3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C39H42F3N9O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-4S5PLC	WO2025011655A1_TM-124	.	COC1=CC2=NN([C@H]3CC[C@@H](CN4CCC(C5=CC6=C(C)C(N7CCC(=O)NC7=O)=NN6C=C5)CC4)CC3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C39H42F3N9O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-4UYHQO	WO2025011655A1_TM-125	.	COC1=CC2=NN([C@H]3CC[C@H](CN4CCC(C5=CN6N=C(N7CCC(=O)NC7=O)C(C)=C6C=C5)CC4)CC3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C39H42F3N9O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-A1SK2V	WO2025011655A1_TM-126	.	COC1=CC2=NN([C@H]3CC[C@H](CN4CCC(C5=CC=CC6=C(N7CCC(=O)NC7=O)N=C(C)N56)CC4)CC3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C39H42F3N9O4	IRAK4	Q9NWZ3	CRBN	WO-2025011655-A1
TPD-OKXESZ	WO2025026283A1_1	.	COC1(C#Cc2cc(-c3ccccc3O)nnc2N)CCC(N2CCC3(CCc4cc5c(cc4O3)CN(C3CCC(=O)NC3=O)C5=O)CC2)CC1	C39H42N6O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-5AKSAB	WO2025026283A1_2	.	COC1(C#Cc2cc(-c3ccccc3O)nnc2N)CCC(N2CC3(CCc4cc5c(cc4O3)C(=O)N(C3CCC(=O)NC3=O)C5)C2)CC1	C37H38N6O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-J5JUR0	WO2025026283A1_3	.	COC1(C#Cc2cc(-c3ccccc3O)nnc2NI)CCC(N2CC3(CCc4cc5c(cc4O3)CN(C3CCC(=O)NC3=O)C5=O)C2)CC1	C37H37IN6O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-FGB9UM	WO2025026283A1_4	.	COC1(C#CC2C=C(c3ccccc3O)N=NC2N)CCC(N2CCC3(CC2)COc2cc4c(cc2C3)C(=O)N(C2CCC(=O)NC2=O)C4=O)CC1	C39H42N6O7	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-JDDXWD	SCHEMBL31380500	3-[1'-[4-[2-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]ethynyl]-4-methoxycyclohexyl]-9-oxospiro[4,7-dihydro-2H-pyrano[2,3-e]isoindole-3,4'-piperidine]-8-yl]piperidine-2,6-dione	COC1(C#Cc2cc(-c3ccccc3O)nnc2N)CCC(N2CCC3(CC2)COc2c(ccc4c2C(=O)N(C2CCC(=O)NC2=O)C4)C3)CC1	C39H42N6O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-0NU070	WO2025026283A1_6	.	Nc1nnc(-c2ccccc2O)cc1C#CC1CCC2(CC1)CC(N1CCC3(CCc4cc5c(cc4O3)CN(C3CCC(=O)NC3=O)C5=O)CC1)C2	C41H44N6O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-U9GY7E	WO2025026283A1_7	.	Nc1nnc(-c2ccccc2O)cc1C#CC1CCC2(CC1)CC(N1CCC3(CC1)COc1cc4c(cc1O3)CN(C1CCC(=O)NC1=O)C4=O)C2	C40H42N6O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-7SN0DF	WO2025026283A1_8	.	Nc1nnc(-c2ccccc2O)cc1C#CC1CCC2(CC1)CC(N1CC3(CCc4cc5c(cc4O3)CC(C3CCC(=O)NC3=O)C5=O)C1)C2	C40H41N5O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-0Y8KR7	WO2025026283A1_9	.	Nc1nnc(-c2ccccc2O)cc1C#CC1CCC2(CC1)CC(N1CC3(CCc4cc5c(cc4O3)C(=O)N(C3CCC(=O)NC3=O)C5)C1)C2	C39H40N6O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-A64OHO	WO2025026283A1_10	.	Nc1nnc(-c2ccccc2O)cc1C#CC1CCC2(CC1)CC(N1CCC(O)(CCc3ccc4c(c3)CN(C3CCC(=O)NC3=O)C4O)CC1)C2	C41H48N6O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-A2TYAE	WO2025026283A1_11	.	Nc1nnc(-c2ccccc2O)cc1C#CC1CCC2(CC1)CC(N1CC3(CCc4cc5c(cc4O3)C(=O)N(C3CCC(=O)NC3=O)C5=O)C1)C2	C39H38N6O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-DRUUO3	WO2025026283A1_12	.	Nc1nnc(-c2ccccc2O)cc1C#CC1CCC2(CC1)CC(N1CCC3(CC1)COc1cc4c(cc13)C(=O)N(C1CCC(=O)NC1=O)C4=O)C2	C40H40N6O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-6OKGQ9	WO2025026283A1_13	.	Nc1nnc(-c2ccccc2O)cc1C#CC1CCC2(CC1)CC(N1CCC3(CC1)COc1c3ccc3c1C(=O)N(C1CCC(=O)NC1=O)C3=O)C2	C40H40N6O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-QI30KD	WO2025026283A1_14	.	Nc1nnc(-c2ccccc2O)cc1C#CC1CCC2(CC1)CC(N1CCN(c3cc4c(cc3F)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC1)C2	C38H38FN7O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-T5EDXK	SCHEMBL31380551	3-[6-[4-[7-[2-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]ethynyl]spiro[3.5]nonan-2-yl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	Nc1nnc(-c2ccccc2O)cc1C#CC1CCC2(CC1)CC(N1CCN(c3ccc4c(c3)CN(C3CCC(=O)NC3=O)C4=O)CC1)C2	C38H41N7O4	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-KMVZVL	WO2025026283A1_16	.	Nc1nnc(-c2ccccc2O)cc1C#CC1CCC2(CC1)CC(N1CCC3(CCc4ccc5c(c4O3)CN(C3CCC(=O)NC3=O)C5=O)CC1)C2	C41H44N6O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-TNKD0N	WO2025026283A1_17	.	Nc1nnc(-c2ccccc2O)cc1C#CC1CCC2(CC1)CC(N1CCC3(CC1)COc1c(ccc4c1C(=O)N(C1CCC(=O)NC1=O)C4)C3)C2	C41H44N6O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-Q9OMXA	WO2025026283A1_18	.	Nc1nnc(-c2ccccc2O)cc1C#CC1CCC2(CC1)CC(N1CCC3(CCc4cc5c(cc4O3)C(=O)N(C3CCC(=O)NC3=O)C5=O)CC1)C2	C41H42N6O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-DLW0G4	WO2025026283A1_19	.	NC1=NNC(c2ccccc2O)C=C1C#CC1CCC2(CC1)CC(N1CCC3(CC1)COc1cc4c(cc1C3)C(=O)N(C1CCC(=O)NC1=O)C4=O)C2	C41H44N6O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-2TKEGI	WO2025026283A1_20	.	Nc1nnc(-c2ccccc2O)cc1C#CC1CCC2(CC1)CC(N1CCC3(CC1)Cc1cc4c(cc1O3)C(=O)N(C1CCC(=O)NC1=O)C4=O)C2	C40H40N6O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-6FZOWI	WO2025026283A1_21	.	Nc1nnc(-c2ccccc2O)cc1C#CC1CCC2(CC1)CC(N1CC3(CCc4ccc5c(c4O3)C(=O)N(C3CCC(=O)NC3=O)C5=O)C1)C2	C39H38N6O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-40LPXS	SCHEMBL31380499	5-[4-[2-[2-[3-Amino-6-(2-hydroxyphenyl)pyridazin-4-yl]ethynyl]spiro[3.5]nonan-7-yl]piperazin-1-yl]-2-(2,6-dioxopiperidin-3-yl)-6-fluoroisoindole-1,3-dione	Nc1nnc(-c2ccccc2O)cc1C#CC1CC2(CCC(N3CCN(c4cc5c(cc4F)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)C1	C38H38FN7O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-RFX2WS	WO2025026283A1_23	.	Nc1nnc(-c2ccccc2O)cc1C#CC1CC2(CCC(N3CC4(CCc5cc6c(cc5O4)C(=O)N(C4CCC(=O)NC4=O)C6)C3)CC2)C1	C39H40N6O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-SBSVOD	WO2025026283A1_24	.	Nc1nnc(-c2ccccc2O)cc1C#CC1CC2(CCC(N3CCC4(CCc5cc6c(cc5O4)CN(C4CCC(=O)NC4=O)C6=O)CC3)CC2)C1	C41H44N6O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-7UQSZV	SCHEMBL31380527	1'-[2-[2-[3-Amino-6-(2-hydroxyphenyl)pyridazin-4-yl]ethynyl]spiro[3.5]nonan-7-yl]-7-(2,6-dioxopiperidin-3-yl)spiro[3,4-dihydropyrano[3,2-f]isoindole-2,3'-azetidine]-6,8-dione	Nc1nnc(-c2ccccc2O)cc1C#CC1CC2(CCC(N3CC4(CCc5cc6c(cc5O4)C(=O)N(C4CCC(=O)NC4=O)C6=O)C3)CC2)C1	C39H38N6O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-VSQD8B	WO2025026283A1_26	.	Nc1nnc(-c2ccccc2O)cc1C#CC1CC2(CCC(N3CCC4(CCc5cc6c(cc5O4)C(=O)N(C4CCC(=O)NC4=O)C6)CC3)CC2)C1	C41H44N6O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-3DCRPL	WO2025026283A1_27	.	Nc1nnc(-c2ccccc2O)cc1C#CC1CC2(CCC(N3CCC4(CC3)COc3cc5c(cc3O4)CN(C3CCC(=O)NC3=O)C5=O)CC2)C1	C40H42N6O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-YJZ24E	WO2025026283A1_28	.	Nc1nnc(-c2ccccc2O)cc1C#CC1CC2(CCC(N3CC4(CCc5cc6c(cc5O4)CN(C4CCC(=O)NC4=O)C6=O)C3)CC2)C1	C39H40N6O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-FC822N	SCHEMBL31380539	3-[6-[4-[2-[2-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]ethynyl]spiro[3.5]nonan-7-yl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	Nc1nnc(-c2ccccc2O)cc1C#CC1CC2(CCC(N3CCN(c4ccc5c(c4)CN(C4CCC(=O)NC4=O)C5=O)CC3)CC2)C1	C38H41N7O4	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-WWL4KM	WO2025026283A1_31	.	Nc1nnc(-c2ccccc2O)cc1C#CC1CC2(C1)CC(N1CCC3(CCc4cc5c(cc4O3)CN(C3CCC(=O)NC3=O)C5=O)CC1)C2	C39H40N6O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-8EEHJN	WO2025026283A1_32	.	Nc1nnc(-c2ccccc2O)cc1C#CC1CC2(C1)CC(N1CCC3(CC1)COc1cc4c(cc1O3)CN(C1CCC(=O)NC1=O)C4=O)C2	C38H38N6O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-6O6401	WO2025026283A1_33	.	Nc1nnc(-c2ccccc2O)cc1C#CC1CC2(C1)CC(N1CCC3(CCc4cc5c(cc4O3)C(=O)N(C3CCC(=O)NC3=O)C5)CC1)C2	C39H40N6O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-3XAK3V	WO2025026283A1_34	.	Nc1nnc(-c2ccccc2O)cc1C#CC1CC2(C1)CC(N1CC3(CCc4cc5c(cc4O3)C(=O)N(C3CCC(=O)NC3=O)C5)C1)C2	C37H36N6O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-IT2G2R	WO2025026283A1_35	.	Nc1nnc(-c2ccccc2O)cc1C#CC1CC2(C1)CC(N1CCC3(CCc4ccc5c(c4O3)CN(C3CCC(=O)NC3=O)C5=O)CC1)C2	C39H40N6O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-ZHRCBB	SCHEMBL31380555	1'-[6-[2-[3-Amino-6-(2-hydroxyphenyl)pyridazin-4-yl]ethynyl]spiro[3.3]heptan-2-yl]-7-(2,6-dioxopiperidin-3-yl)spiro[3,4-dihydropyrano[3,2-f]isoindole-2,3'-azetidine]-6,8-dione	Nc1nnc(-c2ccccc2O)cc1C#CC1CC2(C1)CC(N1CC3(CCc4cc5c(cc4O3)C(=O)N(C3CCC(=O)NC3=O)C5=O)C1)C2	C37H34N6O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-77OB5N	WO2025026283A1_37	.	Nc1nnc(-c2ccccc2O)cc1C#CC1CC2(C1)CC(N1CCC3(CC1)COc1cc4c(cc13)C(=O)N(C1CCC(=O)NC1=O)C4=O)C2	C38H36N6O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-FIA5CW	WO2025026283A1_38	.	Nc1nnc(-c2ccccc2O)cc1C#CC1CC2(C1)CC(N1CCC3(CCc4cc5c(cc4O3)C(=O)N(C3CCC(=O)NC3=O)C5=O)CC1)C2	C39H38N6O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-M1ES4W	SCHEMBL31380542	1'-[6-[2-[3-Amino-6-(2-hydroxyphenyl)pyridazin-4-yl]ethynyl]spiro[3.3]heptan-2-yl]-7-(2,6-dioxopiperidin-3-yl)spiro[2,4-dihydropyrano[3,2-f]isoindole-3,4'-piperidine]-6,8-dione	Nc1nnc(-c2ccccc2O)cc1C#CC1CC2(C1)CC(N1CCC3(CC1)COc1cc4c(cc1C3)C(=O)N(C1CCC(=O)NC1=O)C4=O)C2	C39H38N6O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-VSXH84	WO2025026283A1_42	.	Nc1nnc(-c2ccccc2O)cc1C#CC1CC2(C1)CC(N1CCC3(CC1)COc1c(ccc4c1C(=O)N(C1CCC(=O)NC1=O)C4)C3)C2	C39H40N6O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-2S5I99	WO2025026283A1_43	.	Nc1nnc(-c2ccccc2O)cc1C#CC1CC2(C1)CC(N1CCC3(CC1)COc1c3ccc3c1CN(C1CCC(=O)NC1=O)C3=O)C2	C38H38N6O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-GRXDI4	SCHEMBL31380508	1'-[6-[2-[3-Amino-6-(2-hydroxyphenyl)pyridazin-4-yl]ethynyl]spiro[3.3]heptan-2-yl]-8-(2,6-dioxopiperidin-3-yl)spiro[3,4-dihydropyrano[2,3-e]isoindole-2,3'-azetidine]-7,9-dione	Nc1nnc(-c2ccccc2O)cc1C#CC1CC2(C1)CC(N1CC3(CCc4ccc5c(c4O3)C(=O)N(C3CCC(=O)NC3=O)C5=O)C1)C2	C37H34N6O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-D65THD	WO2025026283A1_45	.	Nc1nnc(C2C=CC=CC2O)cc1C#C[C@H]1CC[C@@H](CN2CCC3(CCc4cc5c(cc4O3)C(=O)N(C3CCC(=O)NC3=O)C5=O)CC2)CC1	C39H42N6O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-WLJSRY	WO2025026283A1_46	.	Nc1nnc(-c2ccccc2O)cc1C#C[C@H]1CC[C@@H](CN2CCC3(CCc4cc5c(cc4O3)CN(C3CCC(=O)NC3=O)C5=O)CC2)CC1	C39H42N6O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-1UUJLU	WO2025026283A1_47	.	Nc1nnc(-c2ccccc2O)cc1C#C[C@H]1CC[C@@H](CN2CCC3(CCc4cc5c(cc4O3)C(=O)N(C3CCC(=O)NC3=O)C5)CC2)CC1	C39H42N6O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-MRAHYX	WO2025026283A1_48	.	Nc1nnc(-c2ccccc2O)cc1C#C[C@H]1CC[C@@H](CN2CC3(CCc4cc5c(cc4O3)C(=O)N(C3CCC(=O)NC3=O)C5)C2)CC1	C37H38N6O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-BEA5IX	WO2025026283A1_49	.	Nc1nnc(-c2ccccc2O)cc1C#C[C@H]1CC[C@@H](CN2CCC3(CC2)COc2cc4c(cc2O3)CN(C2CCC(=O)NC2=O)C4=O)CC1	C38H40N6O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-AKPAXK	WO2025026283A1_50	.	Nc1nnc(-c2ccccc2O)cc1C#C[C@H]1CC[C@@H](CN2CC3(CCc4cc5c(cc4O3)C(=O)N(C3CCC(=O)NC3=O)C5=O)C2)CC1	C37H36N6O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-TS6MW0	SCHEMBL31380520	3-[1'-[[4-[2-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]ethynyl]cyclohexyl]methyl]-6-oxospiro[4,8-dihydro-3H-pyrano[3,2-f]isoindole-2,3'-azetidine]-7-yl]piperidine-2,6-dione; SCHEMBL31380522	Nc1nnc(-c2ccccc2O)cc1C#C[C@H]1CC[C@@H](CN2CC3(CCc4cc5c(cc4O3)CN(C3CCC(=O)NC3=O)C5=O)C2)CC1	C37H38N6O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-W1SGBA	WO2025026283A1_52	.	Nc1nnc(C2C=CC=CC2O)cc1C#C[C@H]1CC[C@@H](CN2CCC3(CC2)COc2cc4c(cc2C3)C(=O)N(C2CCC(=O)NC2=O)C4=O)CC1	C39H42N6O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-YSHHM5	WO2025026283A1_53	.	Nc1nnc(-c2ccccc2O)cc1C#C[C@H]1CC[C@@H](CN2CCC3(CC2)COc2cc4c(cc23)C(=O)N(C2CCC(=O)NC2=O)C4=O)CC1	C38H38N6O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-JUY1MS	SCHEMBL31380498	3-[6-[4-[[4-[2-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]ethynyl]cyclohexyl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	Nc1nnc(-c2ccccc2O)cc1C#C[C@H]1CC[C@@H](CN2CCN(c3ccc4c(c3)CN(C3CCC(=O)NC3=O)C4=O)CC2)CC1	C36H39N7O4	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-6MCFVN	WO2025026283A1_55	.	Nc1nnc(-c2ccccc2O)cc1C#C[C@H]1CC[C@@H](CN2CCN(c3cc4c(cc3F)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)CC1	C36H36FN7O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-64S1QR	WO2025026283A1_56	.	Nc1nnc(-c2ccccc2O)cc1C#C[C@H]1CC[C@@H](CN2CCC3(CC2)COc2c3ccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)CC1	C38H38N6O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-AK0AOW	SCHEMBL31380496	1'-[[4-[2-[3-Amino-6-(2-hydroxyphenyl)pyridazin-4-yl]ethynyl]cyclohexyl]methyl]-8-(2,6-dioxopiperidin-3-yl)spiro[3,4-dihydropyrano[2,3-e]isoindole-2,4'-piperidine]-7,9-dione	Nc1nnc(-c2ccccc2O)cc1C#C[C@H]1CC[C@@H](CN2CCC3(CCc4ccc5c(c4O3)C(=O)N(C3CCC(=O)NC3=O)C5=O)CC2)CC1	C39H40N6O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-MF9PU5	WO2025026283A1_58	.	Nc1nnc(-c2ccccc2O)cc1C#C[C@H]1CC[C@@H](CN2CCC3(CC2)COc2c(ccc4c2C(=O)N(C2CCC(=O)NC2=O)C4)C3)CC1	C39H42N6O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-GYJWZK	WO2025026283A1_59	.	Nc1nnc(-c2ccccc2O)cc1C#C[C@H]1CC[C@@H](CN2CCC3(CC2)COc2c3ccc3c2CN(C2CCC(=O)NC2=O)C3=O)CC1	C38H40N6O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-5LS9RX	WO2025026283A1_60	.	Nc1nnc(-c2ccccc2O)cc1C#C[C@H]1CC[C@@H](CN2CCC3(CC2)COc2ccc4c(c23)C(=O)N(C2CCC(=O)NC2=O)C4=O)CC1	C38H38N6O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-TOPIRH	WO2025026283A1_62	.	Nc1nnc(-c2ccccc2O)cc1C#CC1CCC2(CC1)CC(N1CCC3(CC1)COc1c3ccc3c1CN(C1CCC(=O)NC1=O)C3=O)C2	C40H42N6O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-GFD46O	SCHEMBL31380515	1'-[7-[2-[3-Amino-6-(2-hydroxyphenyl)pyridazin-4-yl]ethynyl]spiro[3.5]nonan-2-yl]-8-(2,6-dioxopiperidin-3-yl)spiro[3,4-dihydropyrano[2,3-e]isoindole-2,4'-piperidine]-7,9-dione	Nc1nnc(-c2ccccc2O)cc1C#CC1CCC2(CC1)CC(N1CCC3(CCc4ccc5c(c4O3)C(=O)N(C3CCC(=O)NC3=O)C5=O)CC1)C2	C41H42N6O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-TFSCVL	SCHEMBL31380579	3-[1'-[7-[2-[3-Amino-6-(2-hydroxyphenyl)pyridazin-4-yl]ethynyl]spiro[3.5]nonan-2-yl]-7-oxospiro[2,5-dihydrofuro[2,3-f]isoindole-3,4'-piperidine]-6-yl]piperidine-2,6-dione	Nc1nnc(-c2ccccc2O)cc1C#CC1CCC2(CC1)CC(N1CCC3(CC1)COc1cc4c(cc13)CN(C1CCC(=O)NC1=O)C4=O)C2	C40H42N6O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-3R7MVI	SCHEMBL31380486	3-[1'-[7-[2-[3-Amino-6-(2-hydroxyphenyl)pyridazin-4-yl]ethynyl]spiro[3.5]nonan-2-yl]-5-oxospiro[2,7-dihydrofuro[3,2-f]isoindole-3,4'-piperidine]-6-yl]piperidine-2,6-dione	Nc1nnc(-c2ccccc2O)cc1C#CC1CCC2(CC1)CC(N1CCC3(CC1)COc1cc4c(cc13)C(=O)N(C1CCC(=O)NC1=O)C4)C2	C40H42N6O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-6ZF9V6	SCHEMBL31380492	1'-[6-[2-[3-Amino-6-(2-hydroxyphenyl)pyridazin-4-yl]ethynyl]spiro[3.3]heptane-2-carbonyl]-7-(2,6-dioxopiperidin-3-yl)spiro[3,4-dihydropyrano[3,2-f]isoindole-2,4'-piperidine]-6,8-dione	Nc1nnc(-c2ccccc2O)cc1C#CC1CC2(C1)CC(C(=O)N1CCC3(CCc4cc5c(cc4O3)C(=O)N(C3CCC(=O)NC3=O)C5=O)CC1)C2	C40H38N6O7	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-YNEBZL	WO2025026283A1_88	.	CN(CC1(C)CCc2cc3c(cc2O1)CN(C1CCC(=O)NC1=O)C3=O)C[C@H]1CC[C@H](C#Cc2cc(-c3ccccc3O)nnc2N)CC1	C38H42N6O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-58J23D	WO2025026283A1_89	.	Nc1nnc(-c2ccccc2O)cc1C#C[C@H]1CC[C@H](CN2CC3(CCc4cc5c(cc4O3)C(=O)N(C3CCC(=O)NC3=O)C5=O)C2)CC1	C37H36N6O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-AOI9JT	WO2025026283A1_90	.	Nc1nnc(-c2ccccc2O)cc1C#C[C@H]1CC[C@H](CN2CC3(CCc4cc5c(cc4O3)C(=O)N(C3CCC(=O)NC3=O)C5)C2)CC1	C37H38N6O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-8QWX5Y	SCHEMBL31380576	1'-[4-[2-[3-Amino-6-(2-hydroxyphenyl)pyridazin-4-yl]ethynyl]-4-methoxycyclohexyl]-7-(2,6-dioxopiperidin-3-yl)spiro[3,4-dihydropyrano[3,2-f]isoindole-2,3'-azetidine]-6,8-dione	COC1(C#Cc2cc(-c3ccccc3O)nnc2N)CCC(N2CC3(CCc4cc5c(cc4O3)C(=O)N(C3CCC(=O)NC3=O)C5=O)C2)CC1	C37H36N6O7	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-7RQ6LB	WO2025026283A1_93	.	Nc1nnc(-c2ccccc2O)cc1C#C[C@H]1CC[C@H](C(=O)N2CCC3(CC2)COc2c3ccc3c2CN(C2CCC(=O)NC2=O)C3=O)CC1	C38H38N6O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-QOLYNJ	WO2025026283A1_94	.	Nc1nnc(-c2ccccc2O)cc1C#C[C@H]1CC[C@H](C(=O)N2CCC3(CCc4cc5c(cc4O3)CN(C3CCC(=O)NC3=O)C5=O)CC2)CC1	C39H40N6O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-4TNMBP	WO2025026283A1_95	.	Nc1nnc(-c2ccccc2O)cc1C#CC1CCC(N2CCC3(CCc4ccc5c(c4O3)CN(C3CCC(=O)NC3=O)C5=O)CC2)CC1	C38H40N6O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-SR5GP0	WO2025026283A1_96	.	Nc1nnc(-c2ccccc2O)cc1C#CC1CCC(N2CCC3(CC2)COc2c3ccc3c2CN(C2CCC(=O)NC2=O)C3=O)CC1	C37H38N6O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-8O3HTT	WO2025026283A1_98	.	Nc1nnc(-c2ccccc2O)cc1C#CC1CCN(C[C@H]2CC[C@H](C(=O)N3CCC4(CCc5cc6c(cc5O4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)CC2)CC1	C45H49N7O7	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-Z6VLMP	WO2025026283A1_102	.	Nc1nnc(-c2ccccc2O)cc1N1CCC(C(=O)N2CCC3(CCc4cc5c(cc4O3)C(=O)N(C3CCC(=O)NC3=O)C5=O)CC2)CC1	C36H37N7O7	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-MXNMTH	SCHEMBL31380478	1'-[[4-[2-[3-Amino-6-(2-hydroxyphenyl)pyridazin-4-yl]ethynyl]cyclohexyl]methyl]-7-(2,6-dioxopiperidin-3-yl)spiro[3,4-dihydropyrano[3,2-f]isoindole-2,4'-piperidine]-6,8-dione	Nc1nnc(-c2ccccc2O)cc1C#C[C@H]1CC[C@H](CN2CCC3(CCc4cc5c(cc4O3)C(=O)N(C3CCC(=O)NC3=O)C5=O)CC2)CC1	C39H40N6O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-7G16LU	SCHEMBL31380479	1'-[[4-[2-[3-Amino-6-(2-hydroxyphenyl)pyridazin-4-yl]ethynyl]cyclohexyl]methyl]-7-(2,6-dioxopiperidin-3-yl)spiro[2,4-dihydropyrano[3,2-f]isoindole-3,4'-piperidine]-6,8-dione	Nc1nnc(-c2ccccc2O)cc1C#C[C@H]1CC[C@H](CN2CCC3(CC2)COc2cc4c(cc2C3)C(=O)N(C2CCC(=O)NC2=O)C4=O)CC1	C39H40N6O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-165SZR	WO2025026283A1_105	.	Nc1nnc(-c2ccccc2O)cc1C#C[C@H]1CC[C@H](CN2CCC3(CC2)COc2cc4c(cc2O3)CN(C2CCC(=O)NC2=O)C4=O)CC1	C38H40N6O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-8ZNJVW	WO2025026283A1_106	.	Nc1nnc(-c2ccccc2O)cc1C#C[C@H]1CC[C@H](CN2CCC3(CC2)COc2cc4c(cc23)C(=O)N(C2CCC(=O)NC2=O)C4=O)CC1	C38H38N6O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-88CTIS	WO2025026283A1_107	.	Nc1nnc(-c2ccccc2O)cc1C#C[C@H]1CC[C@H](CN2CCC3(CCc4cc5c(cc4O3)CN(C3CCC(=O)NC3=O)C5=O)CC2)CC1	C39H42N6O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-XSVMZH	WO2025026283A1_108	.	COC1(C#Cc2cc(-c3ccccc3O)nnc2N)CCC(N2CCC3(CCc4ccc5c(c4O3)CN(C3CCC(=O)NC3=O)C5=O)CC2)CC1	C39H42N6O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-4Y7PAA	SCHEMBL31380495	3-[1'-[4-[2-[3-Amino-6-(2-hydroxyphenyl)pyridazin-4-yl]ethynyl]-4-methoxycyclohexyl]-6-oxospiro[2,8-dihydrofuro[2,3-e]isoindole-3,4'-piperidine]-7-yl]piperidine-2,6-dione	COC1(C#Cc2cc(-c3ccccc3O)nnc2N)CCC(N2CCC3(CC2)COc2c3ccc3c2CN(C2CCC(=O)NC2=O)C3=O)CC1	C38H40N6O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-MCVRZX	SCHEMBL31380553	3-[1'-[4-[4-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]piperazin-1-yl]cyclohexyl]-8-oxospiro[4,6-dihydro-3H-pyrano[2,3-f]isoindole-2,3'-azetidine]-7-yl]piperidine-2,6-dione	Nc1nnc(-c2ccccc2O)cc1N1CCN(C2CCC(N3CC4(CCc5cc6c(cc5O4)C(=O)N(C4CCC(=O)NC4=O)C6)C3)CC2)CC1	C38H44N8O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-HT6BAY	WO2025026283A1_111	.	Nc1nnc(-c2ccccc2O)cc1N1CCN(C2CCC(N3CCC4(CCc5ccc6c(c5O4)CN(C4CCC(=O)NC4=O)C6=O)CC3)CC2)CC1	C40H48N8O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-E5AKDL	WO2025026283A1_112	.	Nc1nnc(-c2ccccc2O)cc1N1CCN(C2CCC(N3CCC4(CC3)COc3c4ccc4c3CN(C3CCC(=O)NC3=O)C4=O)CC2)CC1	C39H46N8O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-XZMGKU	WO2025026283A1_113	.	Nc1nnc(-c2ccccc2O)cc1C#Cc1ccc(N2CCC(N3CC4(CCc5cc6c(cc5O4)C(=O)N(C4CCC(=O)NC4=O)C6)C3)CC2)cc1	C41H39N7O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-RHD9RC	WO2025026283A1_114	.	Nc1nnc(-c2ccccc2O)cc1C#Cc1ccc(N2CCC(CN3CC4(CCc5cc6c(cc5O4)C(=O)N(C4CCC(=O)NC4=O)C6)C3)CC2)cc1	C42H41N7O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-TVU28C	WO2025026283A1_123	.	Nc1nnc(-c2ccccc2O)cc1-c1cnn(CC2CCC(C(=O)N3CCC4(CC3)COc3c4ccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)c1	C40H40N8O7	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-QV3ANV	WO2025026283A1_124	.	Nc1nnc(-c2ccccc2O)cc1-c1cnn(C[C@H]2CC[C@H](C(=O)N3CC4(CCc5cc6c(cc5O4)C(=O)N(C4CCC(=O)NC4=O)C6=O)C3)CC2)c1	C39H38N8O7	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-EQRLRZ	SCHEMBL31380554	3-[1'-[4-[[4-[3-Amino-6-(2-hydroxyphenyl)pyridazin-4-yl]pyrazol-1-yl]methyl]cyclohexanecarbonyl]-6-oxospiro[2,8-dihydrofuro[2,3-e]isoindole-3,4'-piperidine]-7-yl]piperidine-2,6-dione	Nc1nnc(-c2ccccc2O)cc1-c1cnn(C[C@H]2CC[C@H](C(=O)N3CCC4(CC3)COc3c4ccc4c3CN(C3CCC(=O)NC3=O)C4=O)CC2)c1	C40H42N8O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-HHJM2B	WO2025026283A1_126	.	Nc1nnc(-c2ccccc2O)cc1-c1cnn(C[C@H]2CC[C@H](CN3CC4(CCc5cc6c(cc5O4)C(=O)N(C4CCC(=O)NC4=O)C6=O)C3)CC2)c1	C39H40N8O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-FLN5VT	SCHEMBL31380525	3-[1'-[[4-[[4-[3-Amino-6-(2-hydroxyphenyl)pyridazin-4-yl]pyrazol-1-yl]methyl]cyclohexyl]methyl]-6-oxospiro[2,8-dihydrofuro[2,3-e]isoindole-3,4'-piperidine]-7-yl]piperidine-2,6-dione	Nc1nnc(-c2ccccc2O)cc1-c1cnn(C[C@H]2CC[C@H](CN3CCC4(CC3)COc3c4ccc4c3CN(C3CCC(=O)NC3=O)C4=O)CC2)c1	C40H44N8O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-L9A9O3	WO2025026283A1_128	.	Nc1nnc(-c2ccccc2O)cc1-c1cnn(C[C@H]2CC[C@H](CN3CCC4(CC3)COc3c4ccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)c1	C40H42N8O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-Y22GSG	SCHEMBL31380510	1'-[1-[3-amino-6-(2-hydroxyphenyl)pyridazin-4-yl]azetidin-3-yl]-7-(2,6-dioxopiperidin-3-yl)spiro[2H-furo[2,3-e]isoindole-3,4'-piperidine]-6,8-dione	Nc1nnc(-c2ccccc2O)cc1N1CC(N2CCC3(CC2)COc2c3ccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)C1	C32H31N7O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-ZADTRR	SCHEMBL31380511	3-[1'-[1-[3-Amino-6-(2-hydroxyphenyl)pyridazin-4-yl]azetidin-3-yl]-6-oxospiro[2,8-dihydrofuro[2,3-e]isoindole-3,4'-piperidine]-7-yl]piperidine-2,6-dione	Nc1nnc(-c2ccccc2O)cc1N1CC(N2CCC3(CC2)COc2c3ccc3c2CN(C2CCC(=O)NC2=O)C3=O)C1	C32H33N7O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-J31ZG8	WO2025026283A1_131	.	Nc1nnc(-c2ccccc2O)cc1-c1cnn([C@H]2CC[C@H](C(=O)N3CCC4(CC3)COc3c4ccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)c1	C39H38N8O7	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-FNTD9F	WO2025026283A1_132	.	Nc1nnc(-c2ccccc2O)cc1-c1cnn([C@H]2CC[C@H](C(=O)N3CC4(CCc5cc6c(cc5O4)C(=O)N(C4CCC(=O)NC4=O)C6=O)C3)CC2)c1	C38H36N8O7	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-51CXJR	WO2025026283A1_133	.	Nc1nnc(-c2ccccc2O)cc1-c1cnn(C2CCC(C(=O)N3CCC4(CC3)COc3c4ccc4c3CN(C3CCC(=O)NC3=O)C4=O)CC2)c1	C39H40N8O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-4FVQ1Y	WO2025026283A1_134	.	Nc1nnc(-c2ccccc2O)cc1-c1cnn([C@H]2CC[C@H](C(=O)N3CCC(N4CC5(CCc6cc7c(cc6O5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C4)CC3)CC2)c1	C43H45N9O7	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-FTEODZ	WO2025026283A1_135	.	Nc1nnc(-c2ccccc2O)cc1-c1cnn([C@H]2CC[C@H](C(=O)N3CCC(N4CCC5(CC4)COc4c5ccc5c4CN(C4CCC(=O)NC4=O)C5=O)CC3)CC2)c1	C44H49N9O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-4GXN53	WO2025026283A1_136	.	Nc1nnc(-c2ccccc2O)cc1-c1cnn([C@H]2CC[C@H](CN3CC4(CCc5cc6c(cc5O4)C(=O)N(C4CCC(=O)NC4=O)C6=O)C3)CC2)c1	C38H38N8O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-E77XGQ	WO2025026283A1_137	.	Nc1nnc(-c2ccccc2O)cc1-c1cnn([C@H]2CC[C@H](CN3CCC4(CC3)COc3c4ccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)c1	C39H40N8O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-ONC807	WO2025026283A1_138	.	Nc1nnc(-c2ccccc2O)cc1-c1cnn([C@H]2CC[C@H](CN3CCC4(CC3)COc3c4ccc4c3CN(C3CCC(=O)NC3=O)C4=O)CC2)c1	C39H42N8O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-2L1IKC	SCHEMBL31380544	3-[1'-[4-[[7-[4-[3-Amino-6-(2-hydroxyphenyl)pyridazin-4-yl]pyrazol-1-yl]-2-azaspiro[3.5]nonan-2-yl]methyl]cyclohexanecarbonyl]-6-oxospiro[2,8-dihydrofuro[2,3-e]isoindole-3,4'-piperidine]-7-yl]piperidine-2,6-dione	Nc1nnc(-c2ccccc2O)cc1-c1cnn(C2CCC3(CC2)CN(C[C@H]2CC[C@H](C(=O)N4CCC5(CC4)COc4c5ccc5c4CN(C4CCC(=O)NC4=O)C5=O)CC2)C3)c1	C48H55N9O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-Z8ZLH6	SCHEMBL31380582	3-[1'-[2-[4-[3-Amino-6-(2-hydroxyphenyl)pyridazin-4-yl]pyrazol-1-yl]acetyl]-6-oxospiro[2,8-dihydrofuro[2,3-e]isoindole-3,4'-piperidine]-7-yl]piperidine-2,6-dione	Nc1nnc(-c2ccccc2O)cc1-c1cnn(CC(=O)N2CCC3(CC2)COc2c3ccc3c2CN(C2CCC(=O)NC2=O)C3=O)c1	C34H32N8O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-3XH4SK	SCHEMBL31380517	3-[1'-[3-[4-[3-Amino-6-(2-hydroxyphenyl)pyridazin-4-yl]pyrazol-1-yl]cyclobutanecarbonyl]-6-oxospiro[2,8-dihydrofuro[2,3-e]isoindole-3,4'-piperidine]-7-yl]piperidine-2,6-dione	Nc1nnc(-c2ccccc2O)cc1-c1cnn([C@H]2C[C@H](C(=O)N3CCC4(CC3)COc3c4ccc4c3CN(C3CCC(=O)NC3=O)C4=O)C2)c1	C37H36N8O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-NV4ZVS	SCHEMBL31380521	3-[1'-[1-[3-[4-[3-Amino-6-(2-hydroxyphenyl)pyridazin-4-yl]pyrazol-1-yl]cyclobutanecarbonyl]piperidin-4-yl]-6-oxospiro[2,8-dihydrofuro[2,3-e]isoindole-3,4'-piperidine]-7-yl]piperidine-2,6-dione	Nc1nnc(-c2ccccc2O)cc1-c1cnn([C@H]2C[C@H](C(=O)N3CCC(N4CCC5(CC4)COc4c5ccc5c4CN(C4CCC(=O)NC4=O)C5=O)CC3)C2)c1	C42H45N9O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-0KB661	WO2025026283A1_143	.	Nc1nnc(-c2ccccc2O)cc1-c1cnn(C2CCC3(CC2)CN(C2CCC(C(=O)N4CCC5(CC4)COc4c5ccc5c4CN(C4CCC(=O)NC4=O)C5=O)CC2)C3)c1	C47H53N9O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-YPGL86	WO2025026283A1_144	.	Nc1nnc(-c2ccccc2O)cc1-c1cnn(C2CCC3(CC2)CN(C2CCC(C(=O)N4CCC(N5CCC6(CC5)COc5c6ccc6c5CN(C5CCC(=O)NC5=O)C6=O)CC4)CC2)C3)c1	C52H62N10O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-XON49B	WO2025026283A1_145	.	Nc1nnc(-c2ccccc2O)cc1-c1ccnc(N2CCC(N3CCC4(CC3)COc3c4ccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)c1	C39H38N8O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-WNN83S	WO2025026283A1_146	.	Nc1nnc(-c2ccccc2O)cc1-c1ccnc(N2CCC(N3CC4(CCc5cc6c(cc5O4)C(=O)N(C4CCC(=O)NC4=O)C6=O)C3)CC2)c1	C38H36N8O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-PGH3WM	SCHEMBL31380533	3-[1'-[1-[4-[3-Amino-6-(2-hydroxyphenyl)pyridazin-4-yl]pyridin-2-yl]piperidin-4-yl]-6-oxospiro[2,8-dihydrofuro[2,3-e]isoindole-3,4'-piperidine]-7-yl]piperidine-2,6-dione	Nc1nnc(-c2ccccc2O)cc1-c1ccnc(N2CCC(N3CCC4(CC3)COc3c4ccc4c3CN(C3CCC(=O)NC3=O)C4=O)CC2)c1	C39H40N8O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-GA7QAJ	WO2025026283A1_148	.	Nc1nnc(-c2ccccc2O)cc1-c1cccc(N2CCC(N3CCC4(CC3)COc3c4ccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)n1	C39H38N8O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-XF0ND0	WO2025026283A1_149	.	Nc1nnc(-c2ccccc2O)cc1-c1cccc(N2CCC(N3CC4(CCc5cc6c(cc5O4)C(=O)N(C4CCC(=O)NC4=O)C6=O)C3)CC2)n1	C38H36N8O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-JAJ8H8	SCHEMBL31380562	3-[1'-[1-[6-[3-Amino-6-(2-hydroxyphenyl)pyridazin-4-yl]pyridin-2-yl]piperidin-4-yl]-6-oxospiro[2,8-dihydrofuro[2,3-e]isoindole-3,4'-piperidine]-7-yl]piperidine-2,6-dione	Nc1nnc(-c2ccccc2O)cc1-c1cccc(N2CCC(N3CCC4(CC3)COc3c4ccc4c3CN(C3CCC(=O)NC3=O)C4=O)CC2)n1	C39H40N8O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-MFR2Y3	WO2025026283A1_151	.	Nc1nnc(-c2ccccc2O)cc1-c1ccc(N2CCC(N3CC4(CCc5cc6c(cc5O4)C(=O)N(C4CCC(=O)NC4=O)C6=O)C3)CC2)nc1	C38H36N8O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-EAQSJ8	WO2025026283A1_152	.	Nc1nnc(-c2ccccc2O)cc1-c1ccc(N2CCC(N3CCC4(CC3)COc3c4ccc4c3CN(C3CCC(=O)NC3=O)C4=O)CC2)nc1	C39H40N8O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-MI2ZR1	WO2025026283A1_154	.	CCOC1(C#Cc2cc(-c3ccccc3O)nnc2N)CCC(N2CCC3(CC2)COc2cc4c(cc2C3)C(=O)N(C2CCC(=O)NC2=O)C4=O)CC1	C40H42N6O7	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-OB5NUO	WO2025026283A1_155	.	Nc1nnc(-c2ccccc2O)cc1N1CCC(N2CCC3(CC2)COc2c3ccc3c2C(=O)N(C2CCC(=O)NC2=O)C3=O)CC1	C34H35N7O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-BMA48G	WO2025026283A1_156	.	Nc1nnc(-c2ccccc2O)cc1N1CCC(N2CCC3(CC2)COc2c3ccc3c2CN(C2CCC(=O)NC2=O)C3=O)CC1	C34H37N7O5	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-LN184V	WO2025026283A1_157	.	Nc1nnc(-c2ccccc2O)cc1N1CCC(N2CC3(CCc4cc5c(cc4O3)C(=O)N(C3CCC(=O)NC3=O)C5=O)C2)CC1	C33H33N7O6	SMARCA2;SMARCA4	P51531/P51532	CRBN	WO-2025026283-A1
TPD-LK8GJE	SCHEMBL31379763	N-[[4-[[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]amino]methyl]phenyl]methyl]-2-[(3S)-1-[2-[3-fluoro-5-hydroxy-4-(1,1,4-trioxo-1,2,5-thiadiazolidin-2-yl)phenyl]ethyl]pyrrolidin-3-yl]acetamide	O=C(C[C@@H]1CCN(CCc2cc(O)c(N3CC(=O)NS3(=O)=O)c(F)c2)C1)NCc1ccc(CNc2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)cc1	C37H38FN7O9S	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2025030006-A2
TPD-XF382G	WO2025030006A2_2	.	O=C(C[C@@H]1CCN(CCc2cc(O)c(N3CC(=O)NS3(=O)=O)c(F)c2)C1)NCCCCCCNc1ccc2c(c1)C(=O)N(C1CCC(=O)NC1=O)C2=O	C35H42FN7O9S	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2025030006-A2
TPD-SMK7E5	WO2025030006A2_3	.	O=C(C[C@@H]1CCN(CCc2cc(O)c(N3CC(=O)NS3(=O)=O)c(F)c2)C1)NCCCCCCCCNc1ccc2c(c1)C(=O)N(C1CCC(=O)NC1=O)C2=O	C37H46FN7O9S	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2025030006-A2
TPD-XNZP2Q	WO2025030006A2_4	.	O=C(C[C@@H]1CCN(CCc2cc(O)c(N3CC(=O)NS3(=O)=O)c(F)c2)C1)NCCCCCCCCCCNc1ccc2c(c1)C(=O)N(C1CCC(=O)NC1=O)C2=O	C39H50FN7O9S	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2025030006-A2
TPD-SNWXR8	WO2025030006A2_5	.	O=C(C[C@@H]1CCN(CCc2cc(O)c(N3CC(=O)NS3(=O)=O)c(F)c2)C1)NCc1cccc(CNc2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3=O)c1	C37H38FN7O9S	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2025030006-A2
TPD-ZZMSJK	WO2025030006A2_6	.	O=C(C[C@@H]1CCN(CCc2cc(O)c(N3CC(=O)NS3(=O)=O)c(F)c2)C1)NCCCCNc1ccc2c(c1)C(=O)N(C1CCC(=O)NC1=O)C2=O	C33H38FN7O9S	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2025030006-A2
TPD-OELVJN	WO2025030006A2_7	.	O=C(C[C@@H]1CCN(CCc2cc(O)c(N3CC(=O)NS3(=O)=O)c(F)c2)C1)NCCNc1ccc2c(c1)C(=O)N(C1CCC(=O)NC1=O)C2=O	C31H34FN7O9S	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2025030006-A2
TPD-YTOFJP	WO2025030006A2_8	.	O=C(C[C@@H]1CCN(CCc2cc(O)c(N3CC(=O)NS3(=O)=O)c(F)c2)C1)NCCNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O	C31H34FN7O9S	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2025030006-A2
TPD-TKMQV8	WO2025030006A2_9	.	O=C(C[C@@H]1CCN(CCc2cc(O)c(N3CC(=O)NS3(=O)=O)c(F)c2)C1)NCC#Cc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O	C32H31FN6O9S	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2025030006-A2
TPD-GVNOAA	WO2025030006A2_10	.	O=C1CCC(c2ccc(NC(=O)C[C@@H]3CCN(CCc4cc(O)c(N5CC(=O)NS5(=O)=O)c(F)c4)C3)cc2)C(=O)N1	C27H30FN5O7S	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2025030006-A2
TPD-X1TLHO	WO2025030006A2_11	.	O=C1CCC(N2C(=O)c3cccc(NC(=O)C[C@@H]4CCN(CCc5cc(O)c(N6CC(=O)NS6(=O)=O)c(F)c5)C4)c3C2=O)C(=O)N1	C29H29FN6O9S	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2025030006-A2
TPD-JHFJML	WO2025030006A2_12	.	O=C1CCC(N2Cc3c(NC(=O)C[C@@H]4CCN(CCc5cc(O)c(N6CC(=O)NS6(=O)=O)c(F)c5)C4)cccc3C2=O)C(=O)N1	C29H31FN6O8S	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2025030006-A2
TPD-29K6DC	WO2025030006A2_13	.	O=C1CCC(N2C(=O)c3ccc(NCC[C@@H]4CCN(CCc5cc(O)c(N6CC(=O)NS6(=O)=O)c(F)c5)C4)cc3C2=O)C(=O)N1	C29H31FN6O8S	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2025030006-A2
TPD-D89IN4	WO2025030006A2_14	.	O=C1CCC(N2Cc3c(NCC[C@@H]4CCN(CCc5cc(O)c(N6CC(=O)NS6(=O)=O)c(F)c5)C4)cccc3C2=O)C(=O)N1	C29H33FN6O7S	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2025030006-A2
TPD-48F7OB	WO2025030006A2_15	.	O=C1CCC(c2ccc(NCC[C@@H]3CCN(CCc4cc(O)c(N5CC(=O)NS5(=O)=O)c(F)c4)C3)cc2)C(=O)N1	C27H32FN5O6S	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2025030006-A2
TPD-K6J1AT	WO2025030006A2_16	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)Cc2ccc(CNC(=O)C[C@@H]3CCN(CCc4cc(O)c(N5CC(=O)NS5(=O)=O)c(F)c4)C3)cc2)C(C)(C)C)cc1	C48H59FN8O9S2	PTPN1;PTPN2	P18031/P17706	VHL	WO-2025030006-A2
TPD-WWLSI9	WO2025030006A2_17	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCNC(=O)C[C@@H]2CCN(CCc3cc(O)c(N4CC(=O)NS4(=O)=O)c(F)c3)C2)C(C)(C)C)cc1	C45H61FN8O9S2	PTPN1;PTPN2	P18031/P17706	VHL	WO-2025030006-A2
TPD-HO8YMZ	WO2025030006A2_18	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCCNC(=O)C[C@@H]2CCN(CCc3cc(O)c(N4CC(=O)NS4(=O)=O)c(F)c3)C2)C(C)(C)C)cc1	C47H65FN8O9S2	PTPN1;PTPN2	P18031/P17706	VHL	WO-2025030006-A2
TPD-EGVTJ9	WO2025030006A2_19	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCCCCNC(=O)C[C@@H]2CCN(CCc3cc(O)c(N4CC(=O)NS4(=O)=O)c(F)c3)C2)C(C)(C)C)cc1	C49H69FN8O9S2	PTPN1;PTPN2	P18031/P17706	VHL	WO-2025030006-A2
TPD-N6561N	WO2025030006A2_20	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)Cc2cccc(CNC(=O)C[C@@H]3CCN(CCc4cc(O)c(N5CC(=O)NS5(=O)=O)c(F)c4)C3)c2)C(C)(C)C)cc1	C48H59FN8O9S2	PTPN1;PTPN2	P18031/P17706	VHL	WO-2025030006-A2
TPD-6XAHXI	WO2025030006A2_21	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCNC(=O)C[C@@H]2CCN(CCc3cc(O)c(N4CC(=O)NS4(=O)=O)c(F)c3)C2)C(C)(C)C)cc1	C43H57FN8O9S2	PTPN1;PTPN2	P18031/P17706	VHL	WO-2025030006-A2
TPD-SWSKEN	WO2025030006A2_22	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)C[C@@H]2CCN(CCc3cc(O)c(N4CC(=O)NS4(=O)=O)c(F)c3)C2)C(C)(C)C)cc1	C39H50FN7O8S2	PTPN1;PTPN2	P18031/P17706	VHL	WO-2025030006-A2
TPD-5P1GOR	WO2025030006A2_23	.	O=C(C[C@@H]1CCN(CCc2cc(O)c(N3CC(=O)NS3(=O)=O)c(F)c2)C1)NCCCCCCNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O	C35H42FN7O9S	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2025030006-A2
TPD-9CRPUN	WO2025030006A2_24	.	O=C(C[C@@H]1CCN(CCc2cc(O)c(N3CC(=O)NS3(=O)=O)c(F)c2)C1)NCCCCNc1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2=O	C33H38FN7O9S	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2025030006-A2
TPD-VAOOU0	WO2025030006A2_25	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCN2CCc3cc(O)c(N4CC(=O)NS4(=O)=O)c(F)c3CC2)C(C)(C)C)cc1	C41H54FN7O8S2	PTPN1;PTPN2	P18031/P17706	VHL	WO-2025030006-A2
TPD-M2F6CY	WO2025030006A2_26	.	Cc1ncsc1-c1ccc([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](NC(=O)CCCCCCCCCN2CCc3cc(O)c(N4CC(=O)NS4(=O)=O)c(F)c3CC2)C(C)(C)C)cc1	C45H62FN7O8S2	PTPN1;PTPN2	P18031/P17706	VHL	WO-2025030006-A2
TPD-UUAPCB	WO2025030006A2_27	.	O=C1CCC(N2C(=O)c3ccc(NCCCCCCCCCCN4CCc5cc(O)c(N6CC(=O)NS6(=O)=O)c(F)c5CC4)cc3C2=O)C(=O)N1	C35H43FN6O8S	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2025030006-A2
TPD-RB28MW	WO2025030006A2_28	.	O=C1CCC(N2C(=O)c3ccc(NCCCCCCN4CCc5cc(O)c(N6CC(=O)NS6(=O)=O)c(F)c5CC4)cc3C2=O)C(=O)N1	C31H35FN6O8S	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2025030006-A2
TPD-JKXVSH	WO2025031294A1_1	.	NC1=NC=CC(C2=NC(C(=O)NC3=CC4=C(C=C3Cl)OC3(CCN(CCOCCOCCNC5=CC=CC6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC3)C4)=CO2)=C1	C40H41ClN8O9	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-Y2C869	WO2025031294A1_2	.	NC1=NC=CC(C2=NC(C(=O)NC3=CC4=C(C=C3Cl)OC3(CCN(CCOCCOCCOCCNC5=CC=CC6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC3)C4)=CO2)=C1	C42H45ClN8O10	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-HCEZBA	WO2025031294A1_3	.	NC1=NC=CC(C2=NC(C(=O)NC3=CC4=C(C=C3Cl)OC3(CCN(CCOCCOCCOCCOCCNC5=CC=CC6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC3)C4)=CO2)=C1	C44H49ClN8O11	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-01L2AW	WO2025031294A1_4	.	NC1=NC=CC(C2=NC(C(=O)NC3=CC4=C(C=C3Cl)OC3(CCN(CCOCCOCCOC5=CC=CC6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC3)C4)=CO2)=C1	C40H40ClN7O10	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-AJUSCE	WO2025031294A1_5	.	NC1=NC=CC(C2=NC(C(=O)NC3=CC4=C(C=C3Cl)OC3(CCN(CCOCCOCCOCCOC5=CC=CC6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC3)C4)=CO2)=C1	C42H44ClN7O11	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-B2F9T7	WO2025031294A1_6	.	NC1=NC=CC(C2=NC(C(=O)NC3=CC4=C(C=C3C3=CC=NC=C3)OC3(CCN(CCOCCOCCOCCNC5=CC=CC6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC3)C4)=CO2)=C1	C47H49N9O10	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-0XOGPL	WO2025031294A1_7	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCOCCOCCOCCN3CCC4(CC3)CC3=C(C=C(Cl)C(NC(=O)C5=COC(C6=CC(N)=NC=C6)=N5)=C3)O4)C(C)(C)C)C=C2)SC=N1	C53H66ClN9O10S	IRAK4	Q9NWZ3	VHL	WO-2025031294-A1
TPD-969IZZ	WO2025031294A1_8	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCOCCOCCN3CCC4(CC3)CC3=C(C=C(Cl)C(NC(=O)C5=COC(C6=CC(N)=NC=C6)=N5)=C3)O4)C(C)(C)C)C=C2)SC=N1	C51H62ClN9O9S	IRAK4	Q9NWZ3	VHL	WO-2025031294-A1
TPD-KK0QYQ	WO2025031294A1_9	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCOCCN3CCC4(CC3)CC3=C(C=C(Cl)C(NC(=O)C5=COC(C6=CC(N)=NC=C6)=N5)=C3)O4)C(C)(C)C)C=C2)SC=N1	C49H58ClN9O8S	IRAK4	Q9NWZ3	VHL	WO-2025031294-A1
TPD-POQ82O	WO2025031294A1_10	.	NC1=NC=CC(C2=NC(C(=O)NC3=CC4=C(C=C3Cl)OC3(CCN(CCOCCOC5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC3)C4)=CO2)=C1	C38H36ClN7O9	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-VIAZVW	WO2025031294A1_11	.	O=C1CCC(N2C(=O)C3=CC=C(OCCOCCOCCN4CCC5(CC4)CC4=C(C=C(Cl)C(NC(=O)C6=C7N=CC=CN7N=C6)=C4)O5)C=C3C2=O)C(=O)N1	C38H38ClN7O9	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-VBV4BC	WO2025031294A1_12	.	O=C1CCC(N2C(=O)C3=CC=C(OCCOCCOCCN4CCC5(CC4)CC4=C(C=C(Cl)C(NC(=O)C6=COC(C7=CC=NC=C7)=N6)=C4)O5)C=C3C2=O)C(=O)N1	C40H39ClN6O10	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-SF4PZK	WO2025031294A1_13	.	O=C1CCC(N2C(=O)C3=CC=C(OCCOCCOCCN4CCC5(CC4)CC4=C(C=C(Cl)C(NC(=O)C6=NC(C(F)(F)F)=CC=C6)=C4)O5)C=C3C2=O)C(=O)N1	C38H37ClF3N5O9	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-O5LDGP	WO2025031294A1_14	.	O=C1CCC(N2C(=O)C3=CC=C(OCCOCCOCCN4CCC5(CC4)CC4=C(C=C(Cl)C(NC(=O)C6=NC(Cl)=CC=C6)=C4)O5)C=C3C2=O)C(=O)N1	C37H37Cl2N5O9	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-WHLUK4	WO2025031294A1_15	.	O=C1CCC(N2C(=O)C3=CC=C(OCCOCCOCCN4CCC5(CC4)CC4=C(C=C(Cl)C(NC(=O)C6=NC=CC=C6)=C4)O5)C=C3C2=O)C(=O)N1	C37H38ClN5O9	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-812J6O	WO2025031294A1_16	.	NC(=O)C(CCC=O)N1C(=O)C2=CC=C(N3CCC(CCCN4CCC5(CC4)CC4=C(C=C(Cl)C(NC(=O)C6=COC(C7=CC(N)=NC=C7)=N6)=C4)O5)CC3)C=C2C1=O	C42H45ClN8O7	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-2I95SX	WO2025031294A1_17	.	NC1=NC=CC(C2=NC(C(=O)NC3=CC4=C(C=C3Cl)OC3(CCN(C5CCN(CC6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)CC5)CC3)C4)=CO2)=C1	C45H48ClN9O7	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-QXKMTG	WO2025031294A1_18	.	NC1=NC=CC(C2=NC(C(=O)NC3=CC4=C(C=C3Cl)OC3(CCN(CC5CCN(CC6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)CC5)CC3)C4)=CO2)=C1	C46H50ClN9O7	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-I0CREN	WO2025031294A1_19	.	NC1=NC=CC(C2=NC(C(=O)NC3=CC4=C(C=C3Cl)OC3(CCN(CCC5CCN(CC6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)CC5)CC3)C4)=CO2)=C1	C47H52ClN9O7	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-7HCT6Z	WO2025031294A1_20	.	O=C1CCC(N2C(=O)C3=CC=C(N4CCC(CCCN5CCC6(CC5)CC5=C(C=C(Cl)C(NC(=O)C7=COC(C8=CC=NC=C8)=N7)=C5)O6)CC4)C=C3C2=O)C(=O)N1	C42H42ClN7O7	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-F9GE21	WO2025031294A1_21	.	O=C1CCC(N2C(=O)C3=CC=C(N4CCC(CN5CCC(N6CCC7(CC6)CC6=C(C=C(Cl)C(NC(=O)C8=COC(C9=CC=NC=C9)=N8)=C6)O7)CC5)CC4)C=C3C2=O)C(=O)N1	C45H47ClN8O7	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-TEG77B	WO2025031294A1_22	.	O=C1CCC(N2C(=O)C3=CC=C(N4CCC(CN5CCC(CN6CCC7(CC6)CC6=C(C=C(Cl)C(NC(=O)C8=COC(C9=CC=NC=C9)=N8)=C6)O7)CC5)CC4)C=C3C2=O)C(=O)N1	C46H49ClN8O7	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-RT9CEF	WO2025031294A1_23	.	O=C1CCC(N2C(=O)C3=CC=C(N4CCC(CN5CCC(CCN6CCC7(CC6)CC6C=C(NC(=O)C8=COC(C9=CC=NC=C9)=N8)C(Cl)=CC6O7)CC5)CC4)C=C3C2=O)C(=O)N1	C47H53ClN8O7	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-9DCR6E	WO2025031294A1_24	.	O=C1CCC(N2C(=O)C3=CC=C(OCC(F)(F)CNC(=O)C4CCC(N5CCC6(CC5)CC5=C(C=C(Cl)C(NC(=O)C7=COC(C8=CC=NC=C8)=N7)=C5)O6)CC4)C=C3C2=O)C(=O)N1	C44H42ClF2N7O9	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-TU0HUH	WO2025031294A1_25	.	O=C1CCC(N2C(=O)C3=CC=C(OCC(CNC(=O)C4CCC(N5CCC6(CC5)CC5=C(C=C(Cl)C(NC(=O)C7=COC(C8=CC=NC=C8)=N7)=C5)O6)CC4)C(F)(F)F)C=C3C2=O)C(=O)N1	C45H43ClF3N7O9	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-1L08OX	WO2025031294A1_26	.	COC(CNC(=O)C1CCC(N2CCC3(CC2)CC2=C(C=C(Cl)C(NC(=O)C4=COC(C5=CC=NC=C5)=N4)=C2)O3)CC1)COC1=CC=C2C(=O)N(C3CCC(=O)NC3=O)C(=O)C2=C1	C45H46ClN7O10	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-P8QX6H	WO2025031294A1_27	.	CN(C)C(CNC(=O)C1CCC(N2CCC3(CC2)CC2=C(C=C(Cl)C(NC(=O)C4=COC(C5=CC=NC=C5)=N4)=C2)O3)CC1)COC1=CC=C2C(=O)N(C3CCC(=O)NC3=O)C(=O)C2=C1	C46H49ClN8O9	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-6OAG8I	WO2025031294A1_28	.	O=C1CCC(N2C(=O)C3=CC=C(OCCN4C=C(CCN5CCC6(CC5)CC5=C(C=C(Cl)C(NC(=O)C7=COC(C8=CC=NC=C8)=N7)=C5)O6)N=N4)C=C3C2=O)C(=O)N1	C40H36ClN9O8	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-2UMNDI	WO2025031294A1_29	.	O=C1CCC(N2C(=O)C3=CC=C(OCCC4=CC=C(CCN5CCC6(CC5)CC5=C(C=C(Cl)C(NC(=O)C7=COC(C8=CC=NC=C8)=N7)=C5)O6)C=C4)C=C3C2=O)C(=O)N1	C44H39ClN6O8	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-8GJJDI	WO2025031294A1_30	.	O=C1CCC(N2C(=O)C3=CC=C(OCC4CC5(CCN(CC(=O)N6CCC7(CC6)CC6=C(C=C(Cl)C(NC(=O)C8=COC(C9=CC=NC=C9)=N8)=C6)O7)CC5)C4)C=C3C2=O)C(=O)N1	C45H44ClN7O9	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-BFPHKL	WO2025031294A1_31	.	CC(C)(C1CN(C2=CC=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=C2)C1)N1CCC(CN2CCC3(CC2)CC2=C(C=C(Cl)C(NC(=O)C4=COC(C5=CC=NC=C5)=N4)=C2)O3)CC1	C46H49ClN8O7	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-JGMKV1	WO2025031294A1_32	.	O=C1CCC(N2C(=O)C3=CC=C(OCC(=O)N4CCC(O)(CC(=O)N5CCC6(CC5)CC5=C(C=C(Cl)C(NC(=O)C7=COC(C8=CC=NC=C8)=N7)=C5)O6)CC4)C=C3C2=O)C(=O)N1	C43H40ClN7O11	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-RC7CBQ	WO2025031294A1_33	.	COC1=C2C(=O)N(C3CCC(=O)NC3=O)CC2=CC(N2CCC(CN3CCC(CN4CCC5(CC4)CC4=C(C=C(Cl)C(NC(=O)C6=COC(C7=CC=NC=C7)=N6)=C4)O5)CC3)CC2)=C1	C47H53ClN8O7	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-UQ5DDG	WO2025031294A1_34	.	O=C1CCC(N2CC3=CC(N4CCC(CN5CCC(CN6CCC7(CC6)CC6=C(C=C(Cl)C(NC(=O)C8=COC(C9=CC=NC=C9)=N8)=C6)O7)CC5)CC4)=C(C(F)(F)F)C=C3C2=O)C(=O)N1	C47H50ClF3N8O6	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-TSORFC	WO2025031294A1_35	.	O=C1CCC(N2C(=O)C3=CC(F)=C(N4CCC(CN5CCC(CN6CCC7(CC6)CC6=C(C=C(Cl)C(NC(=O)C8=COC(C9=CC=NC=C9)=N8)=C6)O7)CC5)CC4)C=C3C2=O)C(=O)N1	C46H48ClFN8O7	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-4JYESZ	WO2025031294A1_36	.	NC1=NC=CC(C2=NC(C(=O)NC3=CC4=C(C=C3Cl)OC3(CCN(CCOCCOCCOC5=CC=C(NC6CCC(=O)NC6=O)C=C5F)CC3)C4)=CO2)=C1	C38H41ClFN7O8	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-0O42JM	WO2025031294A1_37	.	CN(C1=CC=C(OCCOCCOCCN2CCC3(CC2)CC2=C(C=C(Cl)C(NC(=O)C4=COC(C5=CC(N)=NC=C5)=N4)=C2)O3)C(F)=C1)C1CCC(=O)NC1=O	C39H43ClFN7O8	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-BMVE0U	WO2025031294A1_38	.	NC1=NC=CC(C2=NC(C(=O)NC3=CC4=C(C=C3Cl)OC3(CCN(CCOCCOCCOC5=CC=C(NC6CCC(=O)NC6=O)C=C5C(F)(F)F)CC3)C4)=CO2)=C1	C39H41ClF3N7O8	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-CT3SJI	WO2025031294A1_39	.	NC1=NC=CC(C2=NC(C(=O)NC3=CC4=C(C=C3Cl)OC3(CCN(CC5CCN(CC6CCN(C7=NC=C(NC8CCC(=O)NC8=O)C=C7)CC6)CC5)CC3)C4)=CO2)=C1	C43H51ClN10O5	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-5HT2HX	WO2025031294A1_40	.	NC1=NC=CC(C2=NC(C(=O)NC3=CC4=C(C=C3Cl)OC3(CCN(CCOCCOCCOC5=CC=C(C(=O)NC6CCC(=O)NC6=O)C(F)=C5)CC3)C4)=CO2)=C1	C39H41ClFN7O9	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-9O3PX1	WO2025031294A1_41	.	CN(C(=O)C1=C(F)C=C(N2CCC(CN3CCC(CN4CCC5(CC4)CC4=C(C=C(Cl)C(NC(=O)C6=COC(C7=CC=NC=C7)=N6)=C4)O5)CC3)CC2)C=C1)C1CCC(=O)NC1=O	C46H52ClFN8O6	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-LH7ROJ	WO2025031294A1_42	.	O=C1CCC(NC(=O)C2=CN=C(N3CCC(CN4CCC(CN5CCC6(CC5)CC5=C(C=C(Cl)C(NC(=O)C7=COC(C8=CC=NC=C8)=N7)=C5)O6)CC4)CC3)C=C2)C(=O)N1	C44H50ClN9O6	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-KEMELB	WO2025031294A1_43	.	COC1=CC(N2CCC(CN3CCC(CN4CCC5(CC4)CC4=C(C=C(Cl)C(NC(=O)C6=COC(C7=CC=NC=C7)=N6)=C4)O5)CC3)CC2)=CC=C1C(=O)NC1CCC(=O)NC1=O	C46H53ClN8O7	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-NG9ZYW	WO2025031294A1_44	.	NC1=NC=CC(C2=NC(C(=O)NC3=CC4=C(C=C3Cl)OC3(CCN(CCOCCOCCOC5=CC=C(N6CCC(=O)NC6=O)C=C5)CC3)C4)=CO2)=C1	C37H40ClN7O8	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-L4EPF9	WO2025031294A1_45	.	O=C1CCN(C2=CC=C(N3CCC(CN4CCC(CN5CCC6(CC5)CC5=C(C=C(Cl)C(NC(=O)C7=COC(C8=CC=NC=C8)=N7)=C5)O6)CC4)CC3)C(F)=C2)C(=O)N1	C43H48ClFN8O5	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-3ZOGUL	WO2025031294A1_46	.	NC1=NC=CC(C2=NC(C(=O)NC3=CC4=C(C=C3Cl)OC3(CCN(CCOCCOCCOC5=CC=C(C6CCC(=O)NC6=O)C=C5)CC3)C4)=CO2)=C1	C38H41ClN6O8	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-X9LZKN	WO2025031294A1_47	.	CN1N=C(N2CCC(=O)NC2=O)C2=C1C=C(OCCOCCOCCN1CCC3(CC1)CC1=C(C=C(Cl)C(NC(=O)C4=COC(C5=CC(N)=NC=C5)=N4)=C1)O3)C(F)=C2	C39H41ClFN9O8	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-JKB2N7	WO2025031294A1_48	.	CN1N=C(N2CCC(=O)NC2=O)C2=C1C(C(F)(F)F)=C(OCCOCCOCCN1CCC3(CC1)CC1=C(C=C(Cl)C(NC(=O)C4=COC(C5=CC(N)=NC=C5)=N4)=C1)O3)C=C2	C40H41ClF3N9O8	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-WBAXGN	WO2025031294A1_49	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=C1C=C(OCCOCCOCCN1CCC3(CC1)CC1=C(C=C(Cl)C(NC(=O)C4=COC(C5=CC(N)=NC=C5)=N4)=C1)O3)C=C2	C40H43ClN8O9	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-807PO7	WO2025031294A1_50	.	COC1=CC=C2C(=C1C1CCN(CC3CCN(CCC(=O)N4CCC5(CC4)CC4=C(C=C(Cl)C(NC(=O)C6=COC(C7=CC=NC=C7)=N6)=C4)O5)CC3)CC1)N(C)C(=O)N2C1CCC(=O)NC1=O	C49H56ClN9O8	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-3D2AWV	WO2025031294A1_51	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(F)C(C3CCN(CC4CCN(CCC(=O)N5CCC6(CC5)CC5=C(C=C(Cl)C(NC(=O)C7=COC(C8=CC=NC=C8)=N7)=C5)O6)CC4)CC3)=C21	C48H53ClFN9O7	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-BVME2A	WO2025031294A1_52	.	COC1=CC2=C(C=C1NC(=O)C1=COC(C3=CC(N)=NC=C3)=N1)CC1(CCN(CCOCCOCCOC3=CC=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)CC1)O2	C41H43N7O11	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-0AABHY	WO2025031294A1_53	.	CC(C)OC1=CC2=C(C=C1NC(=O)C1=COC(C3=CC(N)=NC=C3)=N1)CC1(CCN(CCOCCOCCOC3=CC=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)CC1)O2	C43H47N7O11	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-2R2F0Y	WO2025031294A1_54	.	NC1=NC=CC(C2=NC(C(=O)NC3=CC4=C(C=C3OCCO)OC3(CCN(CCOCCOCCOC5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC3)C4)=CO2)=C1	C42H45N7O12	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-32OV2R	WO2025031294A1_55	.	NC1=NC=CC(C2=NC(C(=O)NC3=CC4=C(C=C3OCC(F)F)OC3(CCN(CCOCCOCCOC5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC3)C4)=CO2)=C1	C42H43F2N7O11	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-CFTSUC	WO2025031294A1_56	.	NC1=NC=CC(C2=NC(C(=O)NC3=CC4=C(C=C3OC3CC3)OC3(CCN(CCOCCOCCOC5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC3)C4)=CO2)=C1	C43H45N7O11	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-NEVUWB	WO2025031294A1_57	.	NC1=NC=CC(C2=NC(C(=O)NC3=CC4=C(C=C3OCC3CC3)OC3(CCN(CCOCCOCCOC5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC3)C4)=CO2)=C1	C44H47N7O11	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-ZNQU2H	WO2025031294A1_58	.	CN1CC(OC2=CC3=C(C=C2NC(=O)C2=COC(C4=CC(N)=NC=C4)=N2)CC2(CCN(CCOCCOCCOC4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC2)O3)C1	C44H48N8O11	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-V084YP	WO2025031294A1_59	.	CN1C=C(OC2=CC3=C(C=C2NC(=O)C2=COC(C4=CC(N)=NC=C4)=N2)CC2(CCN(CCOCCOCCOC4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC2)O3)C=N1	C44H45N9O11	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-KRBVJ0	WO2025031294A1_60	.	NC1=NC=CC(C2=NC(C(=O)NC3=CC4=C(C=C3OCC3CCOC3)OC3(CCN(CCOCCOCCOC5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC3)C4)=CO2)=C1	C45H49N7O12	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-X18S72	WO2025031294A1_61	.	CN(C)C1=CC2=C(C=C1NC(=O)C1=COC(C3=CC(N)=NC=C3)=N1)CC1(CCN(CCOCCOCCOC3=CC=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)CC1)O2	C42H46N8O10	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-JRETGM	WO2025031294A1_62	.	CC(C)C1=CC2=C(C=C1NC(=O)C1=COC(C3=CC(N)=NC=C3)=N1)CC1(CCN(CCOCCOCCOC3=CC=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)CC1)O2	C43H47N7O10	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-BX1LLH	WO2025031294A1_63	.	NC1=NC=CC(C2=NC(C(=O)NC3=CC4=C(C=C3C3CC3)OC3(CCN(CCOCCOCCOC5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC3)C4)=CO2)=C1	C43H45N7O10	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-TJ3EIW	WO2025031294A1_64	.	N#CC1=CC2=C(C=C1NC(=O)C1=COC(C3=CC(N)=NC=C3)=N1)CC1(CCN(CCOCCOCCOC3=CC=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)CC1)O2	C41H40N8O10	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-JI9DL7	WO2025031294A1_65	.	C#CC1=CC2=C(C=C1NC(=O)C1=COC(C3=CC(N)=NC=C3)=N1)CC1(CCN(CCOCCOCCOC3=CC=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)CC1)O2	C42H41N7O10	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-I0AI7D	WO2025031294A1_66	.	NC1=NC=CC(C2=NC(C(=O)NC3=CC4=C(C=C3C3=CC=C(F)C=C3)OC3(CCN(CCOCCOCCOC5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC3)C4)=CO2)=C1	C46H44FN7O10	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-XIU8U1	WO2025031294A1_67	.	NC1=NC=CC(C2=NC(C(=O)NC3=CC4=C(C=C3N3CCOCC3)OC3(CCN(CCOCCOCCOC5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC3)C4)=CO2)=C1	C44H48N8O11	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-NGSAOR	WO2025031294A1_68	.	NC1=NC=CC(C2=NC(C(=O)NC3=CC4=C(C=C3N3CCC(CO)CC3)OC3(CCN(CCOCCOCCOC5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC3)C4)=CO2)=C1	C46H52N8O11	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-4NW8EG	WO2025031294A1_69	.	NC1=NC=CC(C2=NC(C(=O)NC3=CC4=C(C=C3N3CCC(CC(F)F)CC3)OC3(CCN(CCOCCOCCOC5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC3)C4)=CO2)=C1	C47H52F2N8O10	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-WIKUSI	WO2025031294A1_70	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=CC(C#CCOC3CCN(CC(=O)N4CCC5(CC4)CC4=C(C=C(Cl)C(NC(=O)C6=COC(C7=CC(N)=NC=C7)=N6)=C4)O5)CC3)=C21	C44H44ClN9O8	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-13IEQU	WO2025031294A1_71	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=CC(C#CCOC3CCN(CC(=O)N4CCC5(CC4)CC4=C(C=C(Cl)C(NC(=O)C6=COC(C7=CC=NC=C7)=N6)=C4)O5)CC3)=C21	C44H43ClN8O8	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-RYS0IT	WO2025031294A1_72	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=CC(C#CCOC3CCN(CCC(=O)N4CCC5(CC4)CC4=C(C=C(Cl)C(NC(=O)C6=COC(C7=CC(N)=NC=C7)=N6)=C4)O5)CC3)=C21	C45H46ClN9O8	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-W8L0RB	WO2025031294A1_73	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=CC(C#CCOC3CCN(CCC(=O)N4CCC5(CC4)CC4=C(C=C(Cl)C(NC(=O)C6=COC(C7=CC=NC=C7)=N6)=C4)O5)CC3)=C21	C45H45ClN8O8	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-3SAWG2	WO2025031294A1_74	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=CC(C#CCOC3CCN(CCCC(=O)N4CCC5(CC4)CC4=C(C=C(Cl)C(NC(=O)C6=COC(C7=CC(N)=NC=C7)=N6)=C4)O5)CC3)=C21	C46H48ClN9O8	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-6LEQOI	WO2025031294A1_75	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=CC(C#CCOC3CCN(CCCC(=O)N4CCC5(CC4)CC4=C(C=C(Cl)C(NC(=O)C6=COC(C7=CC=NC=C7)=N6)=C4)O5)CC3)=C21	C46H47ClN8O8	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-PX42YS	WO2025031294A1_76	.	NC1=NC=CC(C2=NC(C(=O)NC3=CC4=C(C=C3Cl)OC3(CCN(C(=O)CN5CCN(CC(=O)NC6=C7ON=C(C8CCC(=O)NC8=O)C7=CC=C6)CC5)CC3)C4)=CO2)=C1	C41H41ClN10O8	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-2NHGJ7	WO2025031294A1_77	.	O=C1CCC(C2=NOC3=C(NC(=O)CN4CCN(CC(=O)N5CCC6(CC5)CC5=C(C=C(Cl)C(NC(=O)C7=COC(C8=CC=NC=C8)=N7)=C5)O6)CC4)C=CC=C23)C(=O)N1	C41H40ClN9O8	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-CYM4W4	WO2025031294A1_78	.	NC1=NC=CC(C2=NC(C(=O)NC3=CC4=C(C=C3Cl)OC3(CCN(C(=O)CCN5CCN(CC(=O)NC6=C7ON=C(C8CCC(=O)NC8=O)C7=CC=C6)CC5)CC3)C4)=CO2)=C1	C42H43ClN10O8	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-5MET5U	WO2025031294A1_79	.	O=C1CCC(C2=NOC3=C(NC(=O)CN4CCN(CCC(=O)N5CCC6(CC5)CC5=C(C=C(Cl)C(NC(=O)C7=COC(C8=CC=NC=C8)=N7)=C5)O6)CC4)C=CC=C23)C(=O)N1	C42H42ClN9O8	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-TKMKRV	WO2025031294A1_80	.	NC1=NC=CC(C2=NC(C(=O)NC3=CC4=C(C=C3Cl)OC3(CCN(C(=O)CCCN5CCN(CC(=O)NC6=C7ON=C(C8CCC(=O)NC8=O)C7=CC=C6)CC5)CC3)C4)=CO2)=C1	C43H45ClN10O8	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-76JCDD	WO2025031294A1_81	.	O=C1CCC(C2=NOC3=C(NC(=O)CN4CCN(CCCC(=O)N5CCC6(CC5)CC5=C(C=C(Cl)C(NC(=O)C7=COC(C8=CC=NC=C8)=N7)=C5)O6)CC4)C=CC=C23)C(=O)N1	C43H44ClN9O8	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-TU3H71	WO2025031294A1_82	.	NC1=NC=CC(C2=NC(C(=O)NC3=CC4=C(C=C3Cl)OC3(CCN(C(=O)CCCCN5CCN(CC(=O)NC6=C7ON=C(C8CCC(=O)NC8=O)C7=CC=C6)CC5)CC3)C4)=CO2)=C1	C44H47ClN10O8	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-BN8FDJ	WO2025031294A1_83	.	O=C1CCC(C2=NOC3=C(NC(=O)CN4CCN(CCCCC(=O)N5CCC6(CC5)CC5=C(C=C(Cl)C(NC(=O)C7=COC(C8=CC=NC=C8)=N7)=C5)O6)CC4)C=CC=C23)C(=O)N1	C44H46ClN9O8	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-ZZQZCP	WO2025031294A1_84	.	CC(C)OC1=NC2=C(C=C1C(=O)NC1=NC(C3=CN(C)N=C3)=CC=C1)CC1(CCN(CCOCCOCCOC3=CC=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)CC1)O2	C43H48N8O10	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-OIST1F	WO2025031294A1_85	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3(F)CC3)C(C)(C)SCCOCCOCCN3CCC4(CC3)CC3=C(C=C(Cl)C(NC(=O)C5=COC(C6=CC(N)=NC=C6)=N5)=C3)O4)C=C2)SC=N1	C52H61ClFN9O9S2	IRAK4	Q9NWZ3	VHL	WO-2025031294-A1
TPD-OKH6DL	WO2025031294A1_86	.	CC1(C)CN(CCOCCOCCOC2=CC=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=C2)CC(F)(F)C12CC1=C(C=C(Cl)C(NC(=O)C3=COC(C4=CC(N)=NC=C4)=N3)=C1)O2	C42H42ClF2N7O10	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-I1VZ4K	WO2025031294A1_87	.	NC1=NC=CC(C2=NC(C(=O)NC3=CC4=C(C=C3OCC(F)F)OC3(CCN(CC5CCN(CC6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)CC5)CC3)C4)=CO2)=C1	C48H53F2N9O8	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-S89RHJ	WO2025031294A1_88	.	NC1=NC=CC(C2=NC(C(=O)NC3=CC4=C(C=C3OCC(F)F)OC3(CCN(CC5CCN(CC6CN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)C6)CC5)CC3)C4)=CO2)=C1	C46H49F2N9O8	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-LTR09R	WO2025031294A1_89	.	NC1=NC=CC(C2=NC(C(=O)NC3=CC4=C(C=C3OCC(F)F)OC3(CCN(CC5CN(CC6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)C5)CC3)C4)=CO2)=C1	C46H49F2N9O8	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-CNV9OG	WO2025031294A1_90	.	NC1=NC=CC(C2=NC(C(=O)NC3=CC4=C(C=C3OCC(F)F)OC3(CCN(C5CN(CC6CCN(C7=C(F)C=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)C5)CC3)C4)=CO2)=C1	C45H46F3N9O8	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-DE5QQJ	WO2025031294A1_91	.	NC1=NC=CC(C2=NC(C(=O)NC3=CC4=C(C=C3OCC(F)F)OC3(CCN(C5CCN(CC6CN(C7=C(F)C=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)C6)CC5)CC3)C4)=CO2)=C1	C45H46F3N9O8	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-958L22	WO2025031294A1_92	.	NC1=NC=CC(C2=NC(C(=O)NC3=CC4=C(C=C3OCC(F)F)OC3(CCN(C5CCN(C6CCN(C7=C(F)C=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)CC5)CC3)C4)=CO2)=C1	C46H48F3N9O8	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-RGAWJ8	WO2025031294A1_93	.	NC1=NC=CC(C2=NC(C(=O)NC3=CC4=C(C=C3OCC(F)F)OC3(CCN(C(=O)CN5CCN(C6=C(F)C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)CC3)C4)=CO2)=C1	C42H40F3N9O9	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-STGW77	WO2025031294A1_94	.	NC1=NC=CC(C2=NC(C(=O)NC3=CC4=C(C=C3OCC(F)F)OC3(CCN(C(=O)C5CCN(CC6CN(C7=C(F)C=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)C6)CC5)CC3)C4)=CO2)=C1	C46H46F3N9O9	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-XD5ZLF	WO2025031294A1_95	.	NC1=NC=CC(C2=NC(C(=O)NC3=CC4=C(C=C3OCC(F)F)OC3(CCN(C5CN(CC6CCN(C7=CC=C(C(=O)NC8CCC(=O)NC8=O)C(F)=C7)CC6)C5)CC3)C4)=CO2)=C1	C44H48F3N9O7	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-SDSP13	WO2025031294A1_96	.	NC1=NC=CC(C2=NC(C(=O)NC3=CC4=C(C=C3OCC(F)F)OC3(CCN(C5CN(CC6CCN(C7=C(F)C=C(NC8CCC(=O)NC8=O)C=C7)CC6)C5)CC3)C4)=CO2)=C1	C43H48F3N9O6	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-D3WVTP	WO2025031294A1_97	.	NC1=NC=CC(C2=NC(C(=O)NC3=CC4=C(C=C3OCC(F)F)OC3(CCN(C5CN(CC6CCN(C7=CC=C(N8CCC(=O)NC8=O)C=C7)CC6)C5)CC3)C4)=CO2)=C1	C42H47F2N9O6	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-PZ88EL	WO2025031294A1_98	.	CN1N=C(C2CCC(=O)NC2=O)C2=CC=CC(C#CCOC3CCN(CCN4CCC5(CC4)CC4=C(C=C(OCC(F)F)C(NC(=O)C6=COC(C7=CC(N)=NC=C7)=N6)=C4)O5)CC3)=C21	C46H49F2N9O7	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-DDAQPX	WO2025031294A1_99	.	CN1N=C(C2CCC(=O)NC2=O)C2=CC=CC(C#CCOC3CCN(CC(=O)N4CCC5(CC4)CC4=C(C=C(OCC(F)F)C(NC(=O)C6=COC(C7=CC(N)=NC=C7)=N6)=C4)O5)CC3)=C21	C46H47F2N9O8	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-9GVRZU	WO2025031294A1_100	.	CC(C)OC1=CC2=C(C=C1NC(=O)C1=C3N=CC=CN3N=C1)CC1(CCN(CCN3CCC(OCC#CC4=C5C(=CC=C4)C(C4CCC(=O)NC4=O)=NN5C)CC3)CC1)O2	C45H51N9O6	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-DUQRBZ	WO2025031294A1_101	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=CC(C#CCOC3CCN(CC(=O)N4CCC5(CC4)CC4=C(C=C(OCC(F)F)C(NC(=O)C6=COC(C7=CC(N)=NC=C7)=N6)=C4)O5)CC3)=C21	C46H47F2N9O9	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-JRFH5Q	WO2025031294A1_102	.	O=C1CCC(N2C(=O)C3=CC=C(OCCOCCOCCN4CCC5(CC4)CC4=C(C=C(OCC(F)F)C(NC(=O)C6=COC(C7=CC(C(F)F)=NC=C7)=N6)=C4)O5)C=C3C2=O)C(=O)N1	C43H42F4N6O11	IRAK4	Q9NWZ3	CRBN	WO-2025031294-A1
TPD-3GQL86	WO2025031482A1_1	.	CC(C)(O)C1=C(F)C2=NC(C3CCN(CC4CCN(C5=C(F)C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)=CN2C=C1NC(=O)C1=CC=CC(C2CC2(F)F)=N1	C43H44F4N8O6	IRAK4	Q9NWZ3	CRBN	WO-2025031482-A1
TPD-29OEQ9	WO2025031482A1_11	.	CC(C)(O)C1=C(F)C2=NC(C3CCN(S(=O)(=O)C4CCN(C5=C(F)C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)=CN2C=C1NC(=O)C1=CC=CC(C2CC2(F)F)=N1	C42H42F4N8O8S	IRAK4	Q9NWZ3	CRBN	WO-2025031482-A1
TPD-YGEWCI	WO2025031482A1_12	.	CC(C)(O)C1=C(F)C2=NC(C3CCN(CC4(O)CN(C5=C(F)C=C6C(=O)N(C7CCC(=O)NC7=O)CC6=C5)C4)CC3)=CN2C=C1NC(=O)C1=CC=CC(C2CC2(F)F)=N1	C41H42F4N8O6	IRAK4	Q9NWZ3	CRBN	WO-2025031482-A1
TPD-ZYMNF9	WO2025031482A1_13	.	CC(C)(O)C1=C(F)C2=NC(C3CCN(CC(=O)N4CCN(C5=C(F)C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)=CN2C=C1NC(=O)C1=CC=CC(C2CC2(F)F)=N1	C43H43F4N9O7	IRAK4	Q9NWZ3	CRBN	WO-2025031482-A1
TPD-KA36BU	WO2025031482A1_14	.	CC(C)(O)C1=C(F)C2=NC(C3CCN(C(=O)CN4CCN(C5=C(F)C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)=CN2C=C1NC(=O)C1=CC=CC(C2CC2(F)F)=N1	C43H43F4N9O7	IRAK4	Q9NWZ3	CRBN	WO-2025031482-A1
TPD-ERMM4B	WO2025031482A1_2-P1	.	CC(C)(O)C1=C(F)C2=NC(C3CCN(CC4CN(C5=C(F)C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)=CN2C=C1NC(=O)C1=CC=CC(C2CC2(F)F)=N1	C41H40F4N8O6	IRAK4	Q9NWZ3	CRBN	WO-2025031482-A1
TPD-NGD16J	WO2025031482A1_2-P2	.	CC(C)(O)C1=C(F)C2=NC(C3CCN(CC4CN(C5=C(F)C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)=CN2C=C1NC(=O)C1=CC=CC([C@@H]2CC2(F)F)=N1	C41H40F4N8O6	IRAK4	Q9NWZ3	CRBN	WO-2025031482-A1
TPD-IU9YH8	WO2025031482A1_3	.	C[C@@H](O)C1=C(F)C2=NC(C3CCN(CC4(F)CN(C5=C(F)C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)=CN2C=C1NC(=O)C1=CC=CC(C2CC2(F)F)=N1	C40H37F5N8O6	IRAK4	Q9NWZ3	CRBN	WO-2025031482-A1
TPD-QV4XXQ	WO2025031482A1_4	.	CC(C)(O)C1=C(F)C2=NC(C3CCN(C4CN(C5CN(C6=CC(F)=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)C4)CC3)CN2C=C1NC(=O)C1=CC=CC(C2CC2(F)F)=N1	C43H45F4N9O6	IRAK4	Q9NWZ3	CRBN	WO-2025031482-A1
TPD-00MPTM	WO2025031482A1_5	.	CC(C1CN(C2=C(F)C=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=C2)C1)N1CCC(C2=CN3C=C(NC(=O)C4=CC=CC(C5CC5(F)F)=N4)C(C(C)(C)O)=C(F)C3=N2)CC1	C42H42F4N8O6	IRAK4	Q9NWZ3	CRBN	WO-2025031482-A1
TPD-FYIGDO	WO2025031482A1_6	.	CC(C)(O)C1=C(F)C2=NC(C3CCN(CC4(O)CN(C5=C(F)C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)=CN2C=C1NC(=O)C1=CC=CC(C2CC2(F)F)=N1	C41H40F4N8O7	IRAK4	Q9NWZ3	CRBN	WO-2025031482-A1
TPD-H6QX8G	WO2025031482A1_7	.	CNC(=O)CN1C(=O)C2=CC(F)=C(N3CC(CO)(CN4CCC(C5=CN6C=C(NC(=O)C7=CC=CC(C8CC8(F)F)=N7)C(C(C)(C)O)=CC6=N5)CC4)C3)C=C2C1=O	C40H43F3N8O6	IRAK4	Q9NWZ3	CRBN	WO-2025031482-A1
TPD-LN9N7U	WO2025031482A1_8	.	CC(C)(O)C1=C(F)C2=NC(C3CCN(CC4(O)CN(C5=C(F)C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)=CN2C=C1NC(=O)C1=CC=C(F)C(C2CC2(F)F)=N1	C41H39F5N8O7	IRAK4	Q9NWZ3	CRBN	WO-2025031482-A1
TPD-428D4G	WO2025031482A1_9	.	CC(C)(O)C1=C(F)C2=NC(C3CCN(C(=O)C4CN(C5=C(F)C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)CC3)=CN2C=C1NC(=O)C1=CC=CC(C2CC2(F)F)=N1	C41H38F4N8O7	IRAK4	Q9NWZ3	CRBN	WO-2025031482-A1
TPD-ZTABWI	WO2025036119A1_A13D-1	.	O=C1CCN(C2=CC=C(N3CC(N4CCN(CC#CC5=CC(F)=C(OCCCC6=CC=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=C(C=CC=C%10)S9)=C8C7)N=C6C(=O)O)C=C5)CC4)C3)C=C2)C(=O)N1	C52H50FN9O6S	BCL2L1	Q07817	CRBN	WO-2025036119-A1
TPD-6P7GWS	WO2025036119A1_A13D-2	.	O=C1CCN(C2=CC=C(N3CC(CN4CCN(CC#CC5=CC(F)=C(OCCCC6=CC=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=C(C=CC=C%10)S9)=C8C7)N=C6C(=O)O)C=C5)CC4)C3)C=C2)C(=O)N1	C53H52FN9O6S	BCL2L1	Q07817	VHL	WO-2025036119-A1
TPD-HLCFC8	WO2025036119A1_A13D-6-PF3	.	O=C1CCC(N2C(=O)C3=C(C2=O)C(NC2CC2OCCOCCOCCOCCN2CCN(CC#CC4=CC(F)=C(OCCCC5=CC=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)N=C5C(=O)O)C=C4)CC2)=CC=C3)C(=O)N1	C63H66FN9O12S	BCL2L1	Q07817	CRBN	WO-2025036119-A1
TPD-DHMDJX	WO2025036119A1_A13D-6	.	O=C1CCN(C2=CC=C(N3CCN(C4CCN(CC#CC5=CC(F)=C(OCCCC6=CC=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=C(C=CC=C%10)S9)=C8C7)N=C6C(=O)O)C=C5)CC4)CC3)C=C2)C(=O)N1	C54H54FN9O6S	BCL2L1	Q07817	CRBN	WO-2025036119-A1
TPD-F62O02	WO2025036119A1_AF_3	.	O=C1CCC(N2C(=O)C3=CC=CC(NCCOCCOCCOCCNC(=O)C4=NC(N5CCC6=CC=CC(C(=O)NC7=NC8=C(C=CC=C8)S7)=C6C5)=CC=C4CCCOC4=C(F)C=C(C#CCN5CCNCC5)C=C4)=C3C2=O)C(=O)N1	C60H63FN10O10S	BCL2L1	Q07817	CRBN	WO-2025036119-A1
TPD-QLNZC6	WO2025036119A1_AF_4	.	O=C1CCC(N2C(=O)C3=C(C2=O)C(NCCOCCOCCOCCOCCNC(=O)C2=NC(N4CCC5=CC=CC(C(=O)NC6=NC7C=CC=CC7S6)=C5C4)=CC=C2CCCOC2=C(F)C=C(C#CCN4CCNCC4)C=C2)=CC=C3)C(=O)N1	C62H69FN10O11S	BCL2L1	Q07817	CRBN	WO-2025036119-A1
TPD-BNX8J4	WO2025036119A1_APF-1	.	CC1=C(C2=CC=C(N3CCC4=CC=CC(C(=O)NC5=NC6=C(C=CC=C6)S5)=C4C3)N=C2C(=O)NCCN2C=C(COCCOCCOCCNC3=CC=CC4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)N=N2)C=NN1CC12CC3CC(CC(C3)C1)C2	C62H67N13O9S	BCL2L1	Q07817	CRBN	WO-2025036119-A1
TPD-N0D7JY	WO2025036119A1_APF-3	.	[2H]C1=C([2H])C([2H])=C2SC(NC(=O)C3=CC=CC4=C3CN(C3=NC(C(=O)O)=C(C5=C(C)N(CC67CC8CC(CC(C8)C6)C7)N=C5)C=C3)CC4)=NC2=C1[2H]	C38H38N6O3S	BCL2L1	Q07817	CRBN	WO-2025036119-A1
TPD-CDZ9E6	WO2025036119A1_APF-4	.	[2H]C1([2H])C2=C(C(=O)NC3=NC4=C(C=CC=C4)S3)C=CC=C2C([2H])([2H])C([2H])([2H])N1C1=NC(C(=O)O)=C(C2=C(C)N(CC34CC5CC(CC(C5)C3)C4)N=C2)C=C1	C38H38N6O3S	BCL2L1	Q07817	CRBN	WO-2025036119-A1
TPD-9WAM64	WO2025036119A1_APH1	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3CCC(CN4CCN(CC#CC5=CC=C(OCCCC6=CC=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=C(C=CC=C%10)S9)=C8C7)N=C6C(=O)O)C(F)=C5)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C68H77FN10O7S2	BCL2L1	Q07817	VHL	WO-2025036119-A1
TPD-SAH814	WO2025036119A1_APH10	.	CC1=NOC([C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](CC(=O)NCCN2CCN(CC#CC3=CC=C(OCCCC4=CC=C(N5CCC6=CC=CC(C(=O)NC7=NC8=C(C=CC=C8)S7)=C6C5)N=C4C(=O)O)C(F)=C3)CC2)C2=CC=C(Cl)C=C2)C(C)C)=C1	C64H68ClFN10O9S	BCL2L1	Q07817	VHL	WO-2025036119-A1
TPD-BHHRE8	WO2025036119A1_APH101	.	CC1=NOC([C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](CC(=O)N2CCN(CC3CCN(CC#CC4=CC=C(OCCCC5=CC=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)N=C5C(=O)O)C(F)=C4)CC3)CC2)C2=CC=C(Cl)C=C2)C(C)C)=C1	C68H74ClFN10O9S	BCL2L1	Q07817	VHL	WO-2025036119-A1
TPD-B5LLMU	WO2025036119A1_APH102	.	CC1=NOC([C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](CC(=O)N2CCC(C(=O)N3CCN(CC#CC4=CC=C(OCCCC5=CC=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)N=C5C(=O)O)C(F)=C4)CC3)CC2)C2=CC=C(Cl)C=C2)C(C)C)=C1	C68H72ClFN10O10S	BCL2L1	Q07817	VHL	WO-2025036119-A1
TPD-NHD9XK	WO2025036119A1_APH103	.	CC1=NOC([C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](CC(=O)N2CCC3(CCN(CC#CC4=CC=C(OCCCC5=CC=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)N=C5C(=O)O)C(F)=C4)CC3)CC2)C2=CC=C(Cl)C=C2)C(C)C)=C1	C67H71ClFN9O9S	BCL2L1	Q07817	VHL	WO-2025036119-A1
TPD-Y96EF1	WO2025036119A1_APH104	.	CN[C@@H](C)C(=O)N[C@H](C(=O)N1CCC[C@H]1C1=NC(C(=O)C2=CC=CC(OCCN3CCC(CN4CCN(CC#CC5=CC=C(OCCCC6=CC=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=C(C=CC=C%10)S9)=C8C7)N=C6C(=O)O)C(F)=C5)CC4)CC3)=C2)=CS1)C1CCCCC1	C73H84FN11O8S2	BCL2L1	Q07817	VHL	WO-2025036119-A1
TPD-PDS42H	WO2025036119A1_APH105	.	CC1=NOC([C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](CC(=O)N2CCC3CCN(CC3)CCN(CC#CC3=CC=C(OCCCC4=CC=C(N5CCC6=CC=CC(C(=O)NC7=NC8=C(C=CC=C8)S7)=C6C5)N=C4C(=O)O)C(F)=C3)CC2)C2=CC=C(Cl)C=C2)C(C)C)=C1	C69H76ClFN10O9S	BCL2L1	Q07817	VHL	WO-2025036119-A1
TPD-P6KBPX	WO2025036119A1_APH106	.	CC(C)(C)[C@H](NC(=O)C1(F)CC1)C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](CC(=O)N1CCC(CCN2CCN(CC#CC3=CC=C(OCCCC4=CC=C(N5CCC6=CC=CC(C(=O)NC7=NC8=C(C=CC=C8)S7)=C6C5)N=C4C(=O)O)C(F)=C3)CC2)CC1)C1=CC=C(Cl)C=C1	C70H79ClF2N10O9S	BCL2L1	Q07817	VHL	WO-2025036119-A1
TPD-4DZWQ4	WO2025036119A1_APH11	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN(C)CC#CC3=CC(F)=C(OCCCC4=CC=C(N5CCC6=CC=CC(C(=O)NC7=NC8=C(C=CC=C8)S7)=C6C5)N=C4C(=O)O)C=C3)C(C)(C)C)C=C2)SC=N1	C61H64FN9O8S2	BCL2L1	Q07817	VHL	WO-2025036119-A1
TPD-H725U4	WO2025036119A1_APH12	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C#CC(=O)CCN(C)CC#CC3=CC(F)=C(OCCCC4=CC=C(N5CCC6=CC=CC(C(=O)NC7=NC8=C(C=CC=C8)S7)=C6C5)N=C4C(=O)O)C=C3)C(C)(C)C)C=C2)SC=N1	C64H65FN8O8S2	BCL2L1	Q07817	VHL	WO-2025036119-A1
TPD-W1UO3H	WO2025036119A1_APH14	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCN3CCC(CN4CCN(CC#CC5=CC=C(OCCCC6=CC=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=C(C=CC=C%10)S9)=C8C7)N=C6C(=O)O)C(F)=C5)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C71H82FN11O8S2	BCL2L1	Q07817	VHL	WO-2025036119-A1
TPD-WVIDVV	WO2025036119A1_APH15	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@H]3C[C@H](O)CN3C(=O)[C@@H](NC(=O)CCCN(C)CC#CC3=CC(F)=C(OCCCC4=CC=C(N5CCC6=CC=CC(C(=O)NC7=NC8=C(C=CC=C8)S7)=C6C5)N=C4C(=O)O)C=C3)C(C)(C)C)C=C2)SC=N1	C63H68FN9O8S2	BCL2L1	Q07817	VHL	WO-2025036119-A1
TPD-PIKHYW	WO2025036119A1_APH17	.	CC1=C(C2=CC=C([C@@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCC#CC3=CC=C(OCCCC4=CC=C(N5CCC6=CC=CC(C(=O)NC7=NC8=C(C=CC=C8)S7)=C6C5)N=C4C(=O)O)C(F)=C3)C(C)(C)C)C=C2)SC=N1	C61H63FN8O8S2	BCL2L1	Q07817	VHL	WO-2025036119-A1
TPD-LUIA2H	WO2025036119A1_APH18	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCC#CC3=CC=C(OCCCC4=CC=C(N5CCC6=CC=CC(C(=O)NC7=NC8=C(C=CC=C8)S7)=C6C5)N=C4C(=O)O)C(F)=C3)C(C)(C)C)C=C2)SC=N1	C62H65FN8O8S2	BCL2L1	Q07817	VHL	WO-2025036119-A1
TPD-D0TPGY	WO2025036119A1_APH19	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCC#CC3=CC=C(OCCCC4=CC=C(N5CCC6=CC=CC(C(=O)NC7=NC8=C(C=CC=C8)S7)=C6C5)N=C4C(=O)O)C(F)=C3)C(C)(C)C)C=C2)SC=N1	C63H67FN8O8S2	BCL2L1	Q07817	VHL	WO-2025036119-A1
TPD-I9IKWR	WO2025036119A1_APH20	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCC#CC3=CC=C(OCCCC4=CC=C(N5CCC6=CC=CC(C(=O)NC7=NC8=C(C=CC=C8)S7)=C6C5)N=C4C(=O)O)C(F)=C3)C(C)(C)C)C=C2)SC=N1	C64H69FN8O8S2	BCL2L1	Q07817	VHL	WO-2025036119-A1
TPD-8JK03Z	WO2025036119A1_APH21	.	CC(C)CC(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](CC(=O)N1CC(CN2CCN(CC#CC3=CC=C(OCCCC4=CC=C(N5CCC6=CC=CC(C(=O)NC7=NC8=C(C=CC=C8)S7)=C6C5)N=C4C(=O)O)C(F)=C3)CC2)C1)C1=CC=C(Cl)C=C1	C62H67ClFN9O8S	BCL2L1	Q07817	VHL	WO-2025036119-A1
TPD-OUOC2T	WO2025036119A1_APH3	.	CC1=C(C2=CC=C([C@H](CC(=O)N3CCC(N4CCN(CC#CC5=CC=C(OCCCC6=CC=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=C(C=CC=C%10)S9)=C8C7)N=C6C(=O)O)C(F)=C5)CC4)CC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)CC(C)C)C=C2)SC=N1	C67H73FN10O8S2	BCL2L1	Q07817	VHL	WO-2025036119-A1
TPD-6O7IYK	WO2025036119A1_APH4	.	CC1=NOC([C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](CC(=O)N2CCC(CN3CCN(CC#CC4=CC=C(OCCCC5=CC=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)N=C5C(=O)O)C(F)=C4)CC3)CC2)C2=CC=C(C3=C(C)N=CS3)C=C2)C(C)C)=C1	C72H78FN11O9S2	BCL2L1	Q07817	VHL	WO-2025036119-A1
TPD-8OYDF4	WO2025036119A1_APH5	.	CC1=NOC([C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](CC(=O)N2CCC(N3CCN(CC#CC4=CC=C(OCCCC5=CC=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)N=C5C(=O)O)C(F)=C4)CC3)CC2)C2=CC=CC=C2)C(C)C)=C1	C67H73FN10O9S	BCL2L1	Q07817	VHL	WO-2025036119-A1
TPD-T6QRFT	WO2025036119A1_APH7	.	CC1=NOC([C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](CC(=O)N2CCC(CN3CCN(CC#CC4=CC(F)=C(OCCCC5=CC=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)N=C5C(=O)O)C=C4)CC3)CC2)C2=CC=CC=C2)C(C)C)=C1	C68H75FN10O9S	BCL2L1	Q07817	VHL	WO-2025036119-A1
TPD-GKUG9E	WO2025036119A1_APH8	.	CC1=NOC([C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](CC(=O)N2CCC(CN3CCN(CC#CC4=CC=C(OCCCC5=CC=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)N=C5C(=O)O)C(F)=C4)CC3)CC2)C2=CC=C(Cl)C=C2)C(C)C)=C1	C68H74ClFN10O9S	BCL2L1	Q07817	VHL	WO-2025036119-A1
TPD-ZZAWHA	WO2025036119A1_APH9	.	CC1=NOC([C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](CC(=O)N2CCN(CC#CC3=CC=C(OCCCC4=CC=C(N5CCC6=CC=CC(C(=O)NC7=NC8=C(C=CC=C8)S7)=C6C5)N=C4C(=O)O)C(F)=C3)CC2)C2=CC=C(Cl)C=C2)C(C)C)=C1	C62H63ClFN9O9S	BCL2L1	Q07817	VHL	WO-2025036119-A1
TPD-V7KBZD	SCHEMBL26611024	2-[5-[1-(1-adamantylmethyl)-5-methylpyrazol-4-yl]-6-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethylcarbamoyl]pyridin-2-yl]-N-(1,3-benzothiazol-2-yl)-3,4-dihydro-1H-isoquinoline-8-carboxamide	CC1=C(C2=CC=C(N3CCC4=CC=CC(C(=O)NC5=NC6=C(C=CC=C6)S5)=C4C3)N=C2C(=O)NCCOCCOCCOCCNC2=CC=CC3=C2C(=O)N(C2CCC(=O)NC2=O)C3=O)C=NN1CC12CC3CC(CC(C3)C1)C2	C59H64N10O9S	BCL2L1	Q07817	CRBN	WO-2025036119-A1
TPD-ER203B	WO2025036119A1_APL-2	.	CC1=C(C2=CC=C(N3CCC4=CC=CC(C(=O)NC5=NC6=C(C=CC=C6)S5)=C4C3)N=C2C(=O)NCCOCCOCCOCCOCCNC2=CC=CC3=C2C(=O)N(C2CCC(=O)NC2=O)C3=O)C=NN1CC12CC3CC(CC(C3)C1)C2	C61H68N10O10S	BCL2L1	Q07817	CRBN	WO-2025036119-A1
TPD-ZXU4V2	WO2025036119A1_APL-3	.	CC1=C(C2=CC=C(N3CCC4=CC=CC(C(=O)NC5=NC6=C(C=CC=C6)S5)=C4C3)N=C2C(=O)OCCOCCOCCNC2=CC=CC3=C2C(=O)N(C2CCC(=O)NC2=O)C3=O)C=NN1CC12CC3CC(CC(C3)C1)C2	C57H59N9O9S	BCL2L1	Q07817	CRBN	WO-2025036119-A1
TPD-OZ4H47	WO2025036119A1_APL-4	.	CC1=C(C2=CC=C(N3CCC4=CC=CC(C(=O)NC5=NC6=C(C=CC=C6)S5)=C4C3)N=C2C(=O)NCCN2C=C(COCCNC3=CC=CC4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)N=N2)C=NN1CC12CC3CC(CC(C3)C1)C2	C58H59N13O7S	BCL2L1	Q07817	CRBN	WO-2025036119-A1
TPD-88JNJT	WO2025036119A1_APL-5	.	CC1=C(C2=CC=C(N3CCC4=CC=CC(C(=O)NC5=NC6=C(C=CC=C6)S5)=C4C3)N=C2C(=O)NCCN2C=C(COCCOCCNC3=CC=CC4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)N=N2)C=NN1CC12CC3CC(CC(C3)C1)C2	C60H63N13O8S	BCL2L1	Q07817	CRBN	WO-2025036119-A1
TPD-T542EH	WO2025036119A1_APL-6	.	O=C1CCC(N2C(=O)C3=C(C2=O)C(NCCOCCOCCOCCN2CCN(CC#CC4=CC(F)=C(OCCCC5=CC=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)N=C5C(=O)O)C=C4)CC2)=CC=C3)C(=O)N1	C60H62FN9O11S	BCL2L1	Q07817	CRBN	WO-2025036119-A1
TPD-1EM555	WO2025036119A1_APQ10-1	.	O=C1CCN(C2=CC=C(N3CCN(CC#CC4=CC(F)=C(OCCCC5=CC=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)N=C5C(=O)O)C=C4)CC3)C=C2F)C(=O)N1	C49H44F2N8O6S	BCL2L1	Q07817	CRBN	WO-2025036119-A1
TPD-IWN9XS	WO2025036119A1_APQ10-2	.	COC1=C(N2CCC(=O)NC2=O)C=CC(N2CCN(CC#CC3=CC=C(OCCCC4=CC=C(N5CCC6=CC=CC(C(=O)NC7=NC8=C(C=CC=C8)S7)=C6C5)N=C4C(=O)O)C(F)=C3)CC2)=C1	C50H47FN8O7S	BCL2L1	Q07817	CRBN	WO-2025036119-A1
TPD-XURNEW	WO2025036119A1_APQ10-3	.	O=C1CCN(C2=CC(F)=C(N3CCN(CC#CC4=CC(F)=C(OCCCC5=CC=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)N=C5C(=O)O)C=C4)CC3)C(F)=C2)C(=O)N1	C49H43F3N8O6S	BCL2L1	Q07817	CRBN	WO-2025036119-A1
TPD-XGM7BT	WO2025036119A1_APQ10	.	CS(=O)(=O)NC(=O)C1=NC(N2CCC3=CC=CC(C(=O)NC4=NC5=C(C=CC=C5)S4)=C3C2)=CC=C1CCCOC1=CC=C(C#CCN2CCN(CC3CCN(C4=CC=C(N5CCC(=O)NC5=O)C=C4)CC3)CC2)C=C1F	C56H59FN10O7S2	BCL2L1	Q07817	CRBN	WO-2025036119-A1
TPD-QB15OI	WO2025036119A1_APQ11	.	O=C1CCN(C2=CC=C(N3CCC(CN4CCN(CC#CC5=CC(F)=C(OCCCC6=CC=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=C(C=CC=C%10)S9)=C8C7)N=C6C(=O)O)C=C5)CC4)CC3)C=C2F)C(=O)N1	C55H55F2N9O6S	BCL2L1	Q07817	CRBN	WO-2025036119-A1
TPD-RRQ13V	WO2025036119A1_APQ5a	.	O=C1CCN(C2=CC=C(N3CCN(CC4CCN(CC#CC5=CC(F)=C(OCCCC6=CC=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=C(C=CC=C%10)S9)=C8C7)N=C6C(=O)O)C=C5)CC4)CC3)C=C2)C(=O)N1	C55H56FN9O6S	BCL2L1	Q07817	CRBN	WO-2025036119-A1
TPD-QED4FK	WO2025036119A1_APQ5b	.	O=C1CCN(C2=CC=C(OCCN3CCC(CN4CCN(CC#CC5=CC(F)=C(OCCCC6=CC=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=C(C=CC=C%10)S9)=C8C7)N=C6C(=O)O)C=C5)CC4)CC3)C=C2)C(=O)N1	C57H60FN9O7S	BCL2L1	Q07817	CRBN	WO-2025036119-A1
TPD-L0I1TR	WO2025036119A1_APQ6a	.	O=C1CCN(C2=CC=C(N3CCN(CC#CC4=CC(F)=C(OCCCC5=CC=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)N=C5C(=O)O)C=C4)CC3)C=C2)C(=O)N1	C49H45FN8O6S	BCL2L1	Q07817	CRBN	WO-2025036119-A1
TPD-3XGKYR	WO2025036119A1_APQ6b	.	O=C1CCN(C2=CC=C(N3CCC(CN4CCN(CC#CC5=CC(F)=C(OCCCC6=CC=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=C(C=CC=C%10)S9)=C8C7)N=C6C(=O)O)C=C5)CC4)CC3)C=C2)C(=O)N1	C55H56FN9O6S	BCL2L1	Q07817	CRBN	WO-2025036119-A1
TPD-SS8S4V	WO2025036119A1_APQ7a	.	O=C1CCC(N2N=NC3=CC=C(C#CCN4CCC(CN5CCN(CC#CC6=CC(F)=C(OCCCC7=CC=C(N8CCC9=CC=CC(C(=O)NC%10=NC%11=C(C=CC=C%11)S%10)=C9C8)N=C7C(=O)O)C=C6)CC5)CC4)C=C3C2=O)C(=O)N1	C60H58FN11O7S	BCL2L1	Q07817	CRBN	WO-2025036119-A1
TPD-3WZK23	WO2025036119A1_APQ7b	.	COC(=O)C1=NC(N2CCC3=CC=CC(C(=O)NC4=NC5=C(C=CC=C5)S4)=C3C2)=CC=C1CCCOC1=C(F)C=C(C#CCN2CCN(C3=CC=C(N4CCC(=O)NC4=O)C=C3)CC2)C=C1	C50H47FN8O6S	BCL2L1	Q07817	CRBN	WO-2025036119-A1
TPD-SEH2SV	WO2025036119A1_APQ8	.	CS(=O)(=O)NC(=O)C1=NC(N2CCC3=CC=CC(C(=O)NC4=NC5C=CC=CC5S4)=C3C2)=CC=C1CCCOC1=C(F)C=C(C#CCN2CCN(C3=CC=C(N4CCC(=O)NC4=O)C=C3)CC2)C=C1	C50H50FN9O7S2	BCL2L1	Q07817	CRBN	WO-2025036119-A1
TPD-YNC4TM	WO2025036119A1_APQ9-1	.	O=C1CCC(N2C(=O)C3=C(C2=O)C(NCCN2CCC(CN4CCN(CC#CC5=CC(F)=C(OCCCC6=CCC(N7CCC8=CC=CC(C(=O)NC9=NC%10C=CC=CC%10S9)=C8C7)N=C6C(=O)O)C=C5)CC4)CC2)=CC=C3)C(=O)N1	C60H65FN10O8S	BCL2L1	Q07817	CRBN	WO-2025036119-A1
TPD-RFEV2Y	WO2025036119A1_APQ9-2	.	O=C1CCN(C2=CC=C(N3CCN(CC#CC4=CC(F)=C(OCCCC5=CC=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)N=C5C(=O)O)C=C4)CC3)C(F)=C2)C(=O)N1	C49H44F2N8O6S	BCL2L1	Q07817	CRBN	WO-2025036119-A1
TPD-G4I5C5	WO2025036119A1_APQ9	.	CC(C)COC(=O)C1=NC(N2CCC3=CC=CC(C(=O)NC4=NC5=C(C=CC=C5)S4)=C3C2)=CC=C1CCCOC1=CC=C(C#CCN2CCN(CC3CCN(C4=CC=C(N5CCC(=O)NC5=O)C=C4)CC3)CC2)C=C1F	C59H64FN9O6S	BCL2L1	Q07817	CRBN	WO-2025036119-A1
TPD-KTFQLC	WO2025036119A1_APQ901	.	O=C1CCN(C2=C(F)C=C(N3CCN(CC#CC4=CC(F)=C(OCCCC5=CC=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)N=C5C(=O)O)C=C4)CC3)C(F)=C2)C(=O)N1	C49H43F3N8O6S	BCL2L1	Q07817	CRBN	WO-2025036119-A1
TPD-YOLCHO	WO2025036119A1_APQ902	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCN(CC#CC4=CC(F)=C(OCCCC5=CC=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)N=C5C(=O)O)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C64H69FN10O8S2	BCL2L1	Q07817	VHL	WO-2025036119-A1
TPD-8PI0GR	WO2025036119A1_APQ902a	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCN3CCN(CC#CC4=CC=C(OCCCC5=CC=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)N=C5C(=O)O)C(F)=C4)CC3)C(C)(C)C)C=C2)SC=N1	C66H73FN10O9S2	BCL2L1	Q07817	VHL	WO-2025036119-A1
TPD-2SRK9R	WO2025036119A1_APQ903	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCC(=O)N3CCN(CC#CC4=CC(F)=C(OCCCC5=CC=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)N=C5C(=O)O)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C68H75FN10O11S2	BCL2L1	Q07817	VHL	WO-2025036119-A1
TPD-S8WR0S	WO2025036119A1_APQ904	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3CCC(N4CCN(CC#CC5=CC(F)=C(OCCCC6=CC=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=C(C=CC=C%10)S9)=C8C7)N=C6C(=O)O)C=C5)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C67H75FN10O7S2	BCL2L1	Q07817	VHL	WO-2025036119-A1
TPD-OYIWBG	WO2025036119A1_APQ_2	.	CN[C@@H](C)C(=O)N[C@H](C)C(=O)N1CCC[C@H]1C1=NC(C(=O)C2=CC=CC(OCCOCCOCCOCCN3CCN(CC#CC4=CC(F)=C(OCCC5=CC=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)N=C5C(=O)O)C=C4)CC3)=C2)=CS1	C67H75FN10O11S2	BCL2L1	Q07817	VHL	WO-2025036119-A1
TPD-0VECQE	SCHEMBL26611554	2-[5-[1-(1-adamantylmethyl)-5-methylpyrazol-4-yl]-6-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethylcarbamoyl]pyridin-2-yl]-N-(1,3-benzothiazol-2-yl)-3,4-dihydro-1H-isoquinoline-8-carboxamide	CC1=C(C2=CC=C(N3CCC4=CC=CC(C(=O)NC5=NC6=C(C=CC=C6)S5)=C4C3)N=C2C(=O)NCCOCCNC2=CC=CC3=C2C(=O)N(C2CCC(=O)NC2=O)C3=O)C=NN1CC12CC3CC(CC(C3)C1)C2	C55H56N10O7S	BCL2L1	Q07817	CRBN	WO-2025036119-A1
TPD-T7RLVF	WO2025036119A1_APR1	.	[2H]C1([2H])CC2=CC=CC(C(=O)NC3=NC4=C(C=CC=C4)S3)=C2CN1C1=CC=C(C2=C(C)N(CC34CC5CC(CC(C5)C3)C4)N=C2)C(C(=O)NCCOCCOCCOCCNC2=CC=CC3=C2C(=O)N(C2CCC(=O)NC2=O)C3=O)=N1	C59H64N10O9S	BCL2L1	Q07817	CRBN	WO-2025036119-A1
TPD-JXYT8P	WO2025036119A1_APR2	.	O=C1CCN(C2=CC=C(N3CCN(C(=O)CCN4CCN(CC#CC5=CC(F)=C(OCCCC6=CC=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=C(C=CC=C%10)S9)=C8C7)N=C6C(=O)O)C=C5)CC4)CC3)C=C2)C(=O)N1	C56H57FN10O7S	BCL2L1	Q07817	CRBN	WO-2025036119-A1
TPD-M1N6B6	WO2025036119A1_APR3	.	O=C1CCN(C2=CC=C(N3CCN(C(=O)CCCN4CCN(CC#CC5=CC(F)=C(OCCCC6=CC=C(N7CCC8=CC=CC(C(=O)NC9=NC%10=C(C=CC=C%10)S9)=C8C7)N=C6C(=O)O)C=C5)CC4)CC3)C=C2)C(=O)N1	C57H59FN10O7S	BCL2L1	Q07817	CRBN	WO-2025036119-A1
TPD-8H2YCC	WO2025036119A1_BF_3	.	CN[C@@H](C)C(=O)N[C@H](C(=O)N1CCC[C@H]1C1=NC(C(=O)C2=CC=CC(OCCCCCN3CCN(CC#CC4=CC=C(OCCCC5=CC=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)N=C5C(=O)O)C(F)=C4)CC3)=C2)=CS1)C1CCCCC1	C70H79FN10O8S2	BCL2L1	Q07817	CRBN	WO-2025036119-A1
TPD-VYB2KR	WO2025036119A1_BF_4	.	CN[C@@H](C)C(=O)N[C@H](C(=O)N1CCC[C@H]1C1=NC(C(=O)C2=CC=CC(OCCOCCOCCN3CCN(CC#CC4=CC(F)=C(OCCCC5=CC=C(N6CCC7=CC=CC(C(=O)NC8=NC9=C(C=CC=C9)S8)=C7C6)N=C5C(=O)O)C=C4)CC3)=C2)=CS1)C1CCCCC1	C71H81FN10O10S2	BCL2L1	Q07817	CRBN	WO-2025036119-A1
TPD-P3UNR5	SCHEMBL31383327	N-[2-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperidin-4-yl]-7-(2-hydroxypropan-2-yl)imidazo[1,2-a]pyridin-6-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	CC(C)(O)c1cc2nc(C3CCN(CC4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)cn2cc1NC(=O)c1cccc(C(F)(F)F)n1	C41H43F3N8O6	IRAK4	Q9NWZ3	CRBN	WO-2025039774-A1
TPD-Q0OACW	SCHEMBL31383297	N-[2-[1-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]ethyl]piperidin-4-yl]-7-(2-hydroxypropan-2-yl)imidazo[1,2-a]pyridin-6-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	CC(C)(O)c1cc2nc(C3CCN(CCN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)CC3)cn2cc1NC(=O)c1cccc(C(F)(F)F)n1	C41H46F3N9O5	IRAK4	Q9NWZ3	CRBN	WO-2025039774-A1
TPD-OD9CLQ	WO2025039774A1_11	.	COc1cc2nc(C3CCN(CCN4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)cn2cc1NC(=O)c1cccc(CF)n1	C39H42FN9O6	IRAK4	Q9NWZ3	CRBN	WO-2025039774-A1
TPD-RKMCWG	SCHEMBL31383328	N-[2-[1-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]ethyl]piperidin-4-yl]-7-methoxyimidazo[1,2-a]pyridin-6-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	COc1cc2nc(C3CCN(CCN4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)CC3)cn2cc1NC(=O)c1cccc(C(F)(F)F)n1	C39H42F3N9O5	IRAK4	Q9NWZ3	CRBN	WO-2025039774-A1
TPD-POXXVU	SCHEMBL31383336	N-[2-[1-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-3-oxo-1H-isoindol-5-yl]piperazin-1-yl]ethyl]piperidin-4-yl]-7-(2-hydroxypropan-2-yl)imidazo[1,2-a]pyridin-6-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	CC(C)(O)c1cc2nc(C3CCN(CCN4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6)CC4)CC3)cn2cc1NC(=O)c1cccc(C(F)(F)F)n1	C41H46F3N9O5	IRAK4	Q9NWZ3	CRBN	WO-2025039774-A1
TPD-R08J55	SCHEMBL31383340	N-[2-[1-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-3-oxo-1H-isoindol-5-yl]piperazin-1-yl]ethyl]piperidin-4-yl]-7-methoxyimidazo[1,2-a]pyridin-6-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	COc1cc2nc(C3CCN(CCN4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6)CC4)CC3)cn2cc1NC(=O)c1cccc(C(F)(F)F)n1	C39H42F3N9O5	IRAK4	Q9NWZ3	CRBN	WO-2025039774-A1
TPD-Y2QIQT	SCHEMBL31383254	N-[2-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperidin-4-yl]-7-(2-hydroxypropan-2-yl)imidazo[1,2-a]pyridin-6-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	CC(C)(O)c1cc2nc(C3CCN(CC4CCN(c5cc6c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)cn2cc1NC(=O)c1cccc(C(F)(F)F)n1	C41H42F4N8O6	IRAK4	Q9NWZ3	CRBN	WO-2025039774-A1
TPD-J18RN7	WO2025039774A1_16	.	CC(C)(O)c1cc2nc(C3CCN(CCN4CCC5(CC4)CN(c4ccc6c(c4)C(=O)N(C4CCC(=O)NC4=O)C6=O)C5)CC3)cn2cc1NC(=O)c1cccc(CF)n1	C44H50FN9O6	IRAK4	Q9NWZ3	CRBN	WO-2025039774-A1
TPD-99K1Z0	SCHEMBL31383346	N-[2-[1-[2-[7-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-2,7-diazaspiro[3.5]nonan-2-yl]ethyl]piperidin-4-yl]-7-(2-hydroxypropan-2-yl)imidazo[1,2-a]pyridin-6-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	CC(C)(O)c1cc2nc(C3CCN(CCN4CC5(CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)CC3)cn2cc1NC(=O)c1cccc(C(F)(F)F)n1	C44H48F3N9O6	IRAK4	Q9NWZ3	CRBN	WO-2025039774-A1
TPD-KSCNAH	SCHEMBL31383338	N-[2-[1-[2-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]ethyl]piperidin-4-yl]-7-(2-hydroxypropan-2-yl)imidazo[1,2-a]pyridin-6-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	CC(C)(O)c1cc2nc(C3CCN(CCC4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)cn2cc1NC(=O)c1cccc(C(F)(F)F)n1	C42H45F3N8O6	IRAK4	Q9NWZ3	CRBN	WO-2025039774-A1
TPD-64HK2Z	SCHEMBL31383324	N-[2-[1-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]propyl]piperidin-4-yl]-7-(2-hydroxypropan-2-yl)imidazo[1,2-a]pyridin-6-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	CC(C)(O)c1cc2nc(C3CCN(CCCN4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)cn2cc1NC(=O)c1cccc(C(F)(F)F)n1	C42H46F3N9O6	IRAK4	Q9NWZ3	CRBN	WO-2025039774-A1
TPD-Q0NW5R	SCHEMBL31383318	N-[2-[1-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]-2-oxoethyl]piperidin-4-yl]-7-(2-hydroxypropan-2-yl)imidazo[1,2-a]pyridin-6-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	CC(C)(O)c1cc2nc(C3CCN(CC(=O)N4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)cn2cc1NC(=O)c1cccc(C(F)(F)F)n1	C41H42F3N9O7	IRAK4	Q9NWZ3	CRBN	WO-2025039774-A1
TPD-RO0JRL	SCHEMBL31383323	N-[2-[1-[1-[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]azetidin-3-yl]piperidin-4-yl]-7-(2-hydroxypropan-2-yl)imidazo[1,2-a]pyridin-6-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	CC(C)(O)c1cc2nc(C3CCN(C4CN(C5CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)CC3)cn2cc1NC(=O)c1cccc(C(F)(F)F)n1	C43H46F3N9O6	IRAK4	Q9NWZ3	CRBN	WO-2025039774-A1
TPD-GGARKW	SCHEMBL31383314	N-[2-[1-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-2,6-diazaspiro[3.3]heptan-6-yl]ethyl]piperidin-4-yl]-7-(2-hydroxypropan-2-yl)imidazo[1,2-a]pyridin-6-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	CC(C)(O)c1cc2nc(C3CCN(CCN4CC5(C4)CN(c4ccc6c(c4)C(=O)N(C4CCC(=O)NC4=O)C6=O)C5)CC3)cn2cc1NC(=O)c1cccc(C(F)(F)F)n1	C42H44F3N9O6	IRAK4	Q9NWZ3	CRBN	WO-2025039774-A1
TPD-Q49XZM	SCHEMBL31383343	N-[2-[1-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]ethyl]piperidin-4-yl]-7-(2-hydroxypropan-2-yl)imidazo[1,2-a]pyridin-6-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	CC(C)(O)c1cc2nc(C3CCN(CCN4CCN(c5cc6c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)cn2cc1NC(=O)c1cccc(C(F)(F)F)n1	C41H43F4N9O6	IRAK4	Q9NWZ3	CRBN	WO-2025039774-A1
TPD-WQ7NNG	SCHEMBL31383321	N-[2-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperidin-4-yl]-7-(2-hydroxypropan-2-yl)imidazo[1,2-a]pyridin-6-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	CC(C)(O)c1cc2nc(C3CCN(CC4CCN(c5cc6c(cc5F)C(=O)N(C5CCC(=O)NC5=O)C6)CC4)CC3)cn2cc1NC(=O)c1cccc(C(F)(F)F)n1	C41H44F4N8O5	IRAK4	Q9NWZ3	CRBN	WO-2025039774-A1
TPD-UZHWBB	SCHEMBL31383337	N-[2-[1-[[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-3-azabicyclo[3.1.0]hexan-6-yl]methyl]piperidin-4-yl]-7-(2-hydroxypropan-2-yl)imidazo[1,2-a]pyridin-6-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	CC(C)(O)c1cc2nc(C3CCN(CC4C5CN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC45)CC3)cn2cc1NC(=O)c1cccc(C(F)(F)F)n1	C41H41F3N8O6	IRAK4	Q9NWZ3	CRBN	WO-2025039774-A1
TPD-VQZ43B	SCHEMBL31383330	N-[2-[1-[[1-[2-[(3R)-2,6-dioxopiperidin-3-yl]-6-fluoro-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperidin-4-yl]-7-(2-hydroxypropan-2-yl)imidazo[1,2-a]pyridin-6-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	CC(C)(O)c1cc2nc(C3CCN(CC4CCN(c5cc6c(cc5F)C(=O)N([C@@H]5CCC(=O)NC5=O)C6=O)CC4)CC3)cn2cc1NC(=O)c1cccc(C(F)(F)F)n1	C41H42F4N8O6	IRAK4	Q9NWZ3	CRBN	WO-2025039774-A1
TPD-V51HHY	SCHEMBL31383320	N-[2-[1-[[1-[2-[(3S)-2,6-dioxopiperidin-3-yl]-6-fluoro-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperidin-4-yl]-7-(2-hydroxypropan-2-yl)imidazo[1,2-a]pyridin-6-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	CC(C)(O)c1cc2nc(C3CCN(CC4CCN(c5cc6c(cc5F)C(=O)N([C@H]5CCC(=O)NC5=O)C6=O)CC4)CC3)cn2cc1NC(=O)c1cccc(C(F)(F)F)n1	C41H42F4N8O6	IRAK4	Q9NWZ3	CRBN	WO-2025039774-A1
TPD-E5KVVV	SCHEMBL31383351	N-[2-[1-[3-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]-3-oxopropyl]piperidin-4-yl]-7-(2-hydroxypropan-2-yl)imidazo[1,2-a]pyridin-6-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	CC(C)(O)c1cc2nc(C3CCN(CCC(=O)N4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)cn2cc1NC(=O)c1cccc(C(F)(F)F)n1	C42H44F3N9O7	IRAK4	Q9NWZ3	CRBN	WO-2025039774-A1
TPD-V54OIG	SCHEMBL31383288	N-[2-[1-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]-4-oxobutyl]piperidin-4-yl]-7-(2-hydroxypropan-2-yl)imidazo[1,2-a]pyridin-6-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	CC(C)(O)c1cc2nc(C3CCN(CCCC(=O)N4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)cn2cc1NC(=O)c1cccc(C(F)(F)F)n1	C43H46F3N9O7	IRAK4	Q9NWZ3	CRBN	WO-2025039774-A1
TPD-I23FFL	SCHEMBL31383341	N-[2-[1-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-2,7-diazaspiro[3.5]nonan-7-yl]-2-oxoethyl]piperidin-4-yl]-7-(2-hydroxypropan-2-yl)imidazo[1,2-a]pyridin-6-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	CC(C)(O)c1cc2nc(C3CCN(CC(=O)N4CCC5(CC4)CN(c4ccc6c(c4)C(=O)N(C4CCC(=O)NC4=O)C6=O)C5)CC3)cn2cc1NC(=O)c1cccc(C(F)(F)F)n1	C44H46F3N9O7	IRAK4	Q9NWZ3	CRBN	WO-2025039774-A1
TPD-N1WFEP	SCHEMBL31383352	N-[2-[1-[2-[7-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]-2,7-diazaspiro[3.5]nonan-2-yl]-2-oxoethyl]piperidin-4-yl]-7-(2-hydroxypropan-2-yl)imidazo[1,2-a]pyridin-6-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	CC(C)(O)c1cc2nc(C3CCN(CC(=O)N4CC5(CCN(c6ccc7c(c6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)CC3)cn2cc1NC(=O)c1cccc(C(F)(F)F)n1	C44H46F3N9O7	IRAK4	Q9NWZ3	CRBN	WO-2025039774-A1
TPD-VB4CDZ	SCHEMBL31383310	N-[2-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-4-yl]methyl]piperidin-4-yl]-7-(2-hydroxypropan-2-yl)imidazo[1,2-a]pyridin-6-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	CC(C)(O)c1cc2nc(C3CCN(CC4CCN(c5ccc6c(c5)CN(C5CCC(=O)NC5=O)C6=O)CC4)CC3)cn2cc1NC(=O)c1cccc(C(F)(F)F)n1	C41H45F3N8O5	IRAK4	Q9NWZ3	CRBN	WO-2025039774-A1
TPD-SP5N87	SCHEMBL31383353	N-[2-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperidin-4-yl]-7-methoxyimidazo[1,2-a]pyridin-6-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	COc1cc2nc(C3CCN(CC4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)cn2cc1NC(=O)c1cccc(C(F)(F)F)n1	C39H39F3N8O6	IRAK4	Q9NWZ3	CRBN	WO-2025039774-A1
TPD-WPUL0S	WO2025039774A1_9	.	CC(C)(O)c1cc2nc(C3CCN(CCN4CCN(c5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)cn2cc1NC(=O)c1cccc(CF)n1	C41H46FN9O6	IRAK4	Q9NWZ3	CRBN	WO-2025039774-A1
TPD-PO2GE4	WO2025039774A1_Comparative1	.	CC(C)(O)c1cc2nc(C3CCN(CCOCCCc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)cn2cc1NC(=O)c1cccc(C(F)(F)F)n1	C40H42F3N7O7	IRAK4	Q9NWZ3	CRBN	WO-2025039774-A1
TPD-PB6UAW	WO2025039774A1_Comparative2	.	CC(C)(O)c1cc2nc(C3CCN(CCCCC#Cc4cccc5c4CC(N4CCC(=O)NC4=O)C5=O)CC3)cn2cc1NC(=O)c1cccc(C(F)(F)F)n1	C41H42F3N7O5	IRAK4	Q9NWZ3	CRBN	WO-2025039774-A1
TPD-21G322	WO2025040147A1_1	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCC(CN5CCc6c(ccc7c(C8CCC(=O)NC8=O)noc67)C5)CC4)cc3)C2(C)C)ccc1C#N	C44H50N6O6	AR	P10275	CRBN	WO-2025040147-A1
TPD-421VCT	WO2025040147A1_2	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCC(CN5CCc6c(ccc7c(C8CCC(=O)NC8=O)noc67)C5)CC4)cn3)C2(C)C)ccc1C#N	C43H49N7O6	AR	P10275	CRBN	WO-2025040147-A1
TPD-XB6XKK	WO2025040147A1_3	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCC(CN5CCc6c(ccc7c(C8CCC(=O)NC8=O)noc67)C5)CC4)nc3)C2(C)C)ccc1C#N	C43H49N7O6	AR	P10275	CRBN	WO-2025040147-A1
TPD-WL030A	WO2025040147A1_4	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3cnc(N4CCC(CN5CCc6c(ccc7c(C8CCC(=O)NC8=O)noc67)C5)CC4)nc3)C2(C)C)ccc1C#N	C42H48N8O6	AR	P10275	CRBN	WO-2025040147-A1
TPD-XB6KYR	WO2025040147A1_5	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3cnc(N4CCC(CN5CCc6c(ccc7c(C8CCC(=O)NC8=O)noc67)C5)CC4)cn3)C2(C)C)ccc1C#N	C42H48N8O6	AR	P10275	CRBN	WO-2025040147-A1
TPD-HNNRVB	WO2025040147A1_6	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCC(CN5CCc6c(ccc7c(C8CCC(=O)NC8=O)noc67)C5)CC4)nn3)C2(C)C)ccc1C#N	C42H48N8O6	AR	P10275	CRBN	WO-2025040147-A1
TPD-VU3APV	WO2025040147A1_7	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCN(CC5Cc6ccc7c(C8CCC(=O)NC8=O)noc7c6C5)CC4)cc3)C2(C)C)ccc1C#N	C43H48N6O6	AR	P10275	CRBN	WO-2025040147-A1
TPD-5E6GME	WO2025040147A1_8	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCC(CN5Cc6ccc7c(C8CCC(=O)NC8=O)noc7c6C5)CC4)cc3)C2(C)C)ccc1C#N	C43H48N6O6	AR	P10275	CRBN	WO-2025040147-A1
TPD-SUHOR9	WO2025040147A1_9	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCC(CN5CCc6ccc7c(C8CCC(=O)NC8=O)noc7c6C5)CC4)cc3)C2(C)C)ccc1C#N	C44H50N6O6	AR	P10275	CRBN	WO-2025040147-A1
TPD-ZXCJFU	WO2025040147A1_10	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCC(CN5CCc6ccc7c(C8CCC(=O)NC8=O)noc7c6CC5)CC4)cc3)C2(C)C)ccc1C#N	C45H52N6O6	AR	P10275	CRBN	WO-2025040147-A1
TPD-MT4CJH	WO2025040147A1_11	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCC(CN5Cc6ccc7c(C8CCC(=O)NC8=O)noc7c6C5)CC4)nc3)C2(C)C)ccc1C#N	C42H47N7O6	AR	P10275	CRBN	WO-2025040147-A1
TPD-IN3JCH	WO2025040147A1_12	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCC(CN5CCc6ccc7c(C8CCC(=O)NC8=O)noc7c6C5)CC4)nc3)C2(C)C)ccc1C#N	C43H49N7O6	AR	P10275	CRBN	WO-2025040147-A1
TPD-OS0HLB	WO2025040147A1_13	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCC(CN5CCc6ccc7c(C8CCC(=O)NC8=O)noc7c6CC5)CC4)nc3)C2(C)C)ccc1C#N	C44H51N7O6	AR	P10275	CRBN	WO-2025040147-A1
TPD-R6Q0OA	WO2025040147A1_14	.	CC1(C)[C@H](NC(=O)c2ccc(N3CCN(C[C@H]4Cc5ccc6c(C7CCC(=O)NC7=O)noc6c5C4)CC3)nc2)C(C)(C)[C@H]1Oc1ccc(C#N)c(O)c1	C41H45N7O6	AR	P10275	CRBN	WO-2025040147-A1
TPD-2LBZSR	WO2025040147A1_15	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3cnc(N4CCC(CN5Cc6ccc7c(C8CCC(=O)NC8=O)noc7c6C5)CC4)nc3)C2(C)C)ccc1C#N	C41H46N8O6	AR	P10275	CRBN	WO-2025040147-A1
TPD-MBQJ41	WO2025040147A1_16	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3cnc(N4CCC(CN5CCc6ccc7c(C8CCC(=O)NC8=O)noc7c6C5)CC4)nc3)C2(C)C)ccc1C#N	C42H48N8O6	AR	P10275	CRBN	WO-2025040147-A1
TPD-NAKZGD	WO2025040147A1_17	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3cnc(N4CCC(CN5CCc6ccc7c(C8CCC(=O)NC8=O)noc7c6CC5)CC4)nc3)C2(C)C)ccc1C#N	C43H50N8O6	AR	P10275	CRBN	WO-2025040147-A1
TPD-LK0T6N	WO2025040147A1_18	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3cnc(N4CCN(C[C@H]5Cc6ccc7c(C8CCC(=O)NC8=O)noc7c6C5)CC4)nc3)C2(C)C)ccc1C#N	C41H46N8O6	AR	P10275	CRBN	WO-2025040147-A1
TPD-T02JMX	WO2025040147A1_19	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3cnc(N4CCC(CN5Cc6ccc7c(C8CCC(=O)NC8=O)noc7c6C5)CC4)cn3)C2(C)C)ccc1C#N	C41H46N8O6	AR	P10275	CRBN	WO-2025040147-A1
TPD-XA00XX	WO2025040147A1_20	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3cnc(N4CCC(CN5CCc6ccc7c(C8CCC(=O)NC8=O)noc7c6C5)CC4)cn3)C2(C)C)ccc1C#N	C42H48N8O6	AR	P10275	CRBN	WO-2025040147-A1
TPD-5LGL0N	WO2025040147A1_21	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3cnc(N4CCC(CN5CCc6ccc7c(C8CCC(=O)NC8=O)noc7c6CC5)CC4)cn3)C2(C)C)ccc1C#N	C43H50N8O6	AR	P10275	CRBN	WO-2025040147-A1
TPD-QTHI61	WO2025040147A1_22	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3cnc(N4CCN(C[C@H]5Cc6ccc7c(C8CCC(=O)NC8=O)noc7c6C5)CC4)cn3)C2(C)C)ccc1C#N	C41H46N8O6	AR	P10275	CRBN	WO-2025040147-A1
TPD-HKYE57	WO2025040147A1_23	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCC(CN5Cc6ccc7c(C8CCC(=O)NC8=O)noc7c6C5)CC4)nn3)C2(C)C)ccc1C#N	C41H46N8O6	AR	P10275	CRBN	WO-2025040147-A1
TPD-3ET4EB	WO2025040147A1_24	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCC(CN5CCc6ccc7c(C8CCC(=O)NC8=O)noc7c6C5)CC4)nn3)C2(C)C)ccc1C#N	C42H48N8O6	AR	P10275	CRBN	WO-2025040147-A1
TPD-QM2KEG	WO2025040147A1_25	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCC(CN5CCc6ccc7c(C8CCC(=O)NC8=O)noc7c6CC5)CC4)nn3)C2(C)C)ccc1C#N	C43H50N8O6	AR	P10275	CRBN	WO-2025040147-A1
TPD-9OQC68	WO2025040147A1_26	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCN(C[C@H]5Cc6ccc7c(C8CCC(=O)NC8=O)noc7c6C5)CC4)nn3)C2(C)C)ccc1C#N	C41H46N8O6	AR	P10275	CRBN	WO-2025040147-A1
TPD-JLC2WN	WO2025040147A1_27	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCC(CN5CCc6c(ccc7c(C8CCC(=O)NC8=O)coc67)C5)CC4)nc3)C2(C)C)ccc1C#N	C44H50N6O6	AR	P10275	CRBN	WO-2025040147-A1
TPD-XFRBBE	WO2025040147A1_28	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCC(CN5CCc6ccc7c(N8CCC(=O)NC8=O)coc7c6CC5)CC4)nc3)C2(C)C)ccc1C#N	C44H51N7O6	AR	P10275	CRBN	WO-2025040147-A1
TPD-HI0BMI	WO2025040147A1_30	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CNC(N4CCN(C5Cc6ccc7c(C8CCC(=O)NC8=O)noc7c6C5)CC4)C=C3)C2(C)C)ccc1C#N	C41H47N7O6	AR	P10275	CRBN	WO-2025040147-A1
TPD-O8ZIO8	WO2025040147A1_31	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCN(C5Cc6ccc7c(C8CCC(=O)NC8=O)noc7c6C5)CC4)nc3)C2(C)C)ccc1C#N	C41H45N7O6	AR	P10275	CRBN	WO-2025040147-A1
TPD-BVQ11D	WO2025040147A1_32	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCC(CN5CC6(Cc7ccc8c(C9CCC(=O)NC9=O)noc8c7C6)C5)CC4)nc3)C2(C)C)ccc1C#N	C45H51N7O6	AR	P10275	CRBN	WO-2025040147-A1
TPD-7UNQM9	WO2025040147A1_33	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCC(CN5CCC6(Cc7ccc8c(C9CCC(=O)NC9=O)noc8c7C6)C5)CC4)nc3)C2(C)C)ccc1C#N	C46H53N7O6	AR	P10275	CRBN	WO-2025040147-A1
TPD-LKR0HI	WO2025040147A1_34	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCC(CN5Cc6cc7onc(C8CCC(=O)NC8=O)c7cc6C5)CC4)nc3)C2(C)C)ccc1C#N	C42H47N7O6	AR	P10275	CRBN	WO-2025040147-A1
TPD-SP89B0	WO2025040147A1_35	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCC(CN5Cc6ccc7c(C8CCC(=O)NC8=O)coc7c6C5)CC4)nc3)C2(C)C)ccc1C#N	C43H48N6O6	AR	P10275	CRBN	WO-2025040147-A1
TPD-LK4U7Y	WO2025040147A1_36	.	COc1cc(O[C@H]2C(C)(C)[C@H](NC(=O)c3ccc(N4CCC(CN5Cc6ccc7c(N8CCC(=O)NC8=O)coc7c6C5)CC4)nc3)C2(C)C)ccc1C#N	C42H47N7O6	AR	P10275	CRBN	WO-2025040147-A1
TPD-REXX71	US20240018134A1_1	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C(C)C)C3CC(C4=CC=C(C5=CC(C6=C(O)C=CC=C6)=NN=C5)C=C4)=NO3)C=C2)SC=N1	C41H42N6O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	US-20240018134-A1
TPD-X375XP	SCHEMBL27008085	(2S,4R)-4-hydroxy-1-[(2S)-2-[[2-[4-[4-[6-(2-hydroxyphenyl)pyridazin-4-yl]phenyl]-3,6-dihydro-2H-pyridin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CC=C(C4=CC=C(C5=CC(C6=C(O)C=CC=C6)=NN=C5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C46H51N7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	US-20240018134-A1
TPD-S11FIM	CHEMBL5207758	(2S,4R)-4-hydroxy-1-[(2S)-2-[[2-[4-[4-[6-(2-hydroxyphenyl)pyridazin-4-yl]phenyl]piperidin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL27007957	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCC(C4=CC=C(C5=CC(C6=C(O)C=CC=C6)=NN=C5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C46H53N7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	US-20240018134-A1
TPD-6OY7HE	CHEMBL5203306	(2S,4R)-4-hydroxy-1-[(2S)-2-[[2-[4-[4-[6-(2-hydroxyphenyl)pyridazin-4-yl]phenyl]piperidin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL27007981	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCC(C4=CC=C(C5=CC(C6=C(O)C=CC=C6)=NN=C5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C45H51N7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	US-20240018134-A1
TPD-P7V4J1	US20240018134A1_13	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCC(C4=CC=C(C5=CC(C6=C(O)C=CC(F)C6)=NN=C5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C46H54FN7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	US-20240018134-A1
TPD-E0OC4M	SCHEMBL27007982	(2S,4R)-4-hydroxy-1-[(2S)-2-[2-[4-[4-[6-(2-hydroxyphenyl)pyridazin-4-yl]phenyl]piperidin-1-yl]propanoylamino]-3,3-dimethylbutanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C(C)N3CCC(C4=CC=C(C5=CC(C6=C(O)C=CC=C6)=NN=C5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C47H55N7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	US-20240018134-A1
TPD-ARP80X	SCHEMBL27008008	(2S,4R)-1-[(2S)-2-[[2-[4-[2-fluoro-4-[6-(2-hydroxyphenyl)pyridazin-4-yl]phenyl]piperidin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCC(C4=CC=C(C5=CC(C6=C(O)C=CC=C6)=NN=C5)C=C4F)CC3)C(C)(C)C)C=C2)SC=N1	C46H52FN7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	US-20240018134-A1
TPD-UWH9S3	CHEMBL5189308	N-[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]-1-[4-[6-(2-hydroxyphenyl)pyridazin-4-yl]phenyl]piperidine-4-carboxamide; SCHEMBL27008015	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3CCN(C4=CC=C(C5=CC(C6=C(O)C=CC=C6)=NN=C5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C45H51N7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	US-20240018134-A1
TPD-25FL6L	SCHEMBL27008013	(2S,4R)-4-hydroxy-1-[(2S)-2-[[2-[4-[4-[6-(2-hydroxyphenyl)pyridazin-4-yl]phenyl]cyclohexyl]acetyl]amino]-3,3-dimethylbutanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CC3CCC(C4=CC=C(C5=CC(C6=C(O)C=CC=C6)=NN=C5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C47H54N6O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	US-20240018134-A1
TPD-6RWO11	SCHEMBL27008000	(2S,4R)-4-hydroxy-1-[(2S)-2-[[4-[4-[6-(2-hydroxyphenyl)pyridazin-4-yl]phenyl]cyclohexanecarbonyl]amino]-3,3-dimethylbutanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3CCC(C4=CC=C(C5=CC(C6=C(O)C=CC=C6)=NN=C5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C46H52N6O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	US-20240018134-A1
TPD-HHZ1B2	SCHEMBL27008054	(2S,4R)-4-hydroxy-1-[(2S)-2-[[2-[4-[4-[6-(2-hydroxyphenyl)pyridazin-4-yl]phenoxy]piperidin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCC(OC4=CC=C(C5=CC(C6=C(O)C=CC=C6)=NN=C5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C46H53N7O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	US-20240018134-A1
TPD-IN83OT	CHEMBL5222069	(2S,4R)-4-hydroxy-1-[(2S)-2-[[2-[4-[4-[6-(2-hydroxyphenyl)pyridazin-4-yl]phenyl]piperazin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL25268419	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCN(C4=CC=C(C5=CC(C6=C(O)C=CC=C6)=NN=C5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C45H52N8O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	US-20240018134-A1
TPD-MPTM2R	SCHEMBL27007977	(2S,4R)-4-hydroxy-1-[(2S)-2-[[2-[3-[4-[6-(2-hydroxyphenyl)pyridazin-4-yl]phenyl]piperidin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCCC(C4=CC=C(C5=CC(C6=C(O)C=CC=C6)=NN=C5)C=C4)C3)C(C)(C)C)C=C2)SC=N1	C46H53N7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	US-20240018134-A1
TPD-BAZCVS	SCHEMBL27007973	(2S,4R)-4-hydroxy-1-[(2S)-2-[[2-[3-[4-[6-(2-hydroxyphenyl)pyridazin-4-yl]phenyl]azetidin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CC(C4=CC=C(C5=CC(C6=C(O)C=CC=C6)=NN=C5)C=C4)C3)C(C)(C)C)C=C2)SC=N1	C44H49N7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	US-20240018134-A1
TPD-E8QKQW	SCHEMBL27007944	(2S,4R)-4-hydroxy-1-[(2S)-2-[[2-[3-[4-[6-(2-hydroxyphenyl)pyridazin-4-yl]phenyl]pyrrolidin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCC(C4=CC=C(C5=CC(C6=C(O)C=CC=C6)=NN=C5)C=C4)C3)C(C)(C)C)C=C2)SC=N1	C45H51N7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	US-20240018134-A1
TPD-W9IL8Y	SCHEMBL27007994	(2S,4R)-4-hydroxy-1-[(2S)-2-[[2-[4-[3-[6-(2-hydroxyphenyl)pyridazin-4-yl]phenyl]piperidin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCC(C4=CC(C5=CC(C6=C(O)C=CC=C6)=NN=C5)=CC=C4)CC3)C(C)(C)C)C=C2)SC=N1	C46H53N7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	US-20240018134-A1
TPD-4P4TJ1	SCHEMBL27024886	(2S,4R)-4-hydroxy-1-[(2S)-2-[[2-[8-[4-[6-(2-hydroxyphenyl)pyridazin-4-yl]phenyl]-3,8-diazabicyclo[3.2.1]octan-3-yl]acetyl]amino]-3,3-dimethylbutanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CC4CCC(C3)N4C3=CC=C(C4=CC(C5=C(O)C=CC=C5)=NN=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C47H54N8O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	US-20240018134-A1
TPD-SIMF16	US20240018134A1_25	.	CC1=C(C2=CC=C([C@H](C)OC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3C4CCC3CC(C3=CC=C(C5=CC(C6=C(O)C=CC=C6)=NN=C5)C=C3)C4)C(C)(C)C)C=C2)SC=N1	C48H54N6O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	US-20240018134-A1
TPD-JF0LYS	SCHEMBL27008023	(2S,4R)-1-[(2S)-2-[[2-[4-[2-fluoro-4-[6-(2-hydroxyphenyl)pyridazin-4-yl]phenyl]piperazin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCN(C4=CC=C(C5=CC(C6=C(O)C=CC=C6)=NN=C5)C=C4F)CC3)C(C)(C)C)C=C2)SC=N1	C45H51FN8O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	US-20240018134-A1
TPD-KP11J9	SCHEMBL27007974	(2S,4R)-4-hydroxy-1-[(2S)-2-[[2-[4-[5-[6-(2-hydroxyphenyl)pyridazin-4-yl]pyridin-2-yl]piperidin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCC(C4=CC=C(C5=CC(C6=C(O)C=CC=C6)=NN=C5)C=N4)CC3)C(C)(C)C)C=C2)SC=N1	C45H52N8O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	US-20240018134-A1
TPD-P8IQPG	SCHEMBL27024888	(2S,4R)-4-hydroxy-1-[(2S)-2-[2-[4-[4-[6-(2-hydroxyphenyl)pyridazin-4-yl]phenyl]piperazin-1-yl]propanoylamino]-3,3-dimethylbutanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C(C)N3CCN(C4=CC=C(C5=CC(C6=C(O)C=CC=C6)=NN=C5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C46H54N8O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	US-20240018134-A1
TPD-AMGW8Q	SCHEMBL25226001	(2S,4R)-1-[(2S)-2-[[2-[4-[4-(6-chloropyridazin-4-yl)phenyl]piperazin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCN(C4=CC=C(C5=CC(Cl)=NN=C5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C39H47ClN8O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	US-20240018134-A1
TPD-LRXVYR	SCHEMBL27024890	(2S,4R)-4-hydroxy-1-[(2S)-2-[[2-[6-[4-[6-(2-hydroxyphenyl)pyridazin-4-yl]phenyl]-2-azaspiro[3.3]heptan-2-yl]acetyl]amino]-3,3-dimethylbutanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CC4(CC(C5=CC=C(C6=CC(C7=C(O)C=CC=C7)=NN=C6)C=C5)C4)C3)C(C)(C)C)C=C2)SC=N1	C47H53N7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	US-20240018134-A1
TPD-9CK8L8	SCHEMBL27008037	(2S,4R)-4-hydroxy-1-[(2S)-2-[[2-[4-hydroxy-4-[4-[6-(2-hydroxyphenyl)pyridazin-4-yl]phenyl]piperidin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCC(O)(C4=CC=C(C5=CC(C6=C(O)C=CC=C6)=NN=C5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C46H53N7O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	US-20240018134-A1
TPD-IUXJIW	SCHEMBL27008075	(2S,4R)-4-hydroxy-1-[(2S)-2-[[2-[4-[4-[6-(2-hydroxyphenyl)pyridazin-4-yl]pyrazol-1-yl]piperidin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCC(N4C=C(C5=CC(C6=C(O)C=CC=C6)=NN=C5)C=N4)CC3)C(C)(C)C)C=C2)SC=N1	C43H51N9O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	US-20240018134-A1
TPD-H83SHJ	SCHEMBL27024891	(2S,4R)-4-hydroxy-1-[(2S)-2-[5-[4-[6-(2-hydroxyphenyl)pyridazin-4-yl]phenoxy]pentanoylamino]-3,3-dimethylbutanoyl]-N-[(1S)-1-[4-(1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](NC(=O)CCCCOC1=CC=C(C2=CC(C3=C(O)C=CC=C3)=NN=C2)C=C1)C(C)(C)C)C1=CC=C(C2=CN=CS2)C=C1	C43H48N6O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	US-20240018134-A1
TPD-D9YY60	SCHEMBL25272088	(2S,4R)-4-hydroxy-1-[(2S)-2-[4-[4-[6-(2-hydroxyphenyl)pyridazin-4-yl]phenoxy]butanoylamino]-3,3-dimethylbutanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCOC3=CC=C(C4=CN=NC(C5=C(O)C=CC=C5)=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C43H48N6O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	US-20240018134-A1
TPD-JYZFU4	SCHEMBL25217673	(2S,4R)-4-hydroxy-1-[(2S)-2-[5-[4-[6-(2-hydroxyphenyl)pyridazin-4-yl]anilino]pentanoylamino]-3,3-dimethylbutanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCNC3=CC=C(C4=CC(C5=C(O)C=CC=C5)=NN=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C44H51N7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	US-20240018134-A1
TPD-JLVCS7	SCHEMBL27008042	(2S,4R)-1-[(2S)-2-[[2-[4-[4-[6-[2-(difluoromethyl)phenyl]pyridazin-4-yl]phenyl]piperazin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCN(C4=CC=C(C5=CC(C6=C(C(F)F)C=CC=C6)=NN=C5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C46H52F2N8O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	US-20240018134-A1
TPD-X4175A	SCHEMBL27007988	(2S,4R)-1-[(2S)-3,3-dimethyl-2-[[2-[4-[4-(6-quinolin-8-ylpyridazin-4-yl)phenyl]piperazin-1-yl]acetyl]amino]butanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCN(C4=CC=C(C5=CC(C6=C7N=CC=CC7=CC=C6)=NN=C5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C48H53N9O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	US-20240018134-A1
TPD-SZZVJR	SCHEMBL27008009	(2S,4R)-4-hydroxy-1-[(2S)-2-[[2-[4-[4-[6-(1H-indol-7-yl)pyridazin-4-yl]phenyl]piperazin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCN(C4=CC=C(C5=CC(C6=C7NC=CC7=CC=C6)=NN=C5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C47H53N9O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	US-20240018134-A1
TPD-MUZLV7	SCHEMBL25220727	(2S,4R)-1-[(2S)-2-[[2-[4-[4-[6-(5-fluoro-2-hydroxyphenyl)pyridazin-4-yl]phenyl]piperazin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL30429273	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCN(C4=CC=C(C5=CC(C6=C(O)C=CC(F)=C6)=NN=C5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C45H51FN8O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	US-20240018134-A1
TPD-UUHHZX	SCHEMBL27008033	(2S,4R)-1-[(2S)-2-[[2-[4-[4-[6-(1-benzofuran-7-yl)pyridazin-4-yl]phenyl]piperazin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCN(C4=CC=C(C5=CC(C6=C7OC=CC7=CC=C6)=NN=C5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C47H52N8O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	US-20240018134-A1
TPD-UHOYY0	SCHEMBL27007985	(2S,4R)-4-hydroxy-1-[(2S)-2-[[2-[4-[4-[6-(1H-indazol-7-yl)pyridazin-4-yl]phenyl]piperazin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCN(C4=CC=C(C5=CC(C6=C7NN=CC7=CC=C6)=NN=C5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C46H52N10O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	US-20240018134-A1
TPD-QVPEYG	SCHEMBL25216377	(2S,4R)-4-hydroxy-1-[2-[3-[2-[4-[6-(2-hydroxyphenyl)pyridazin-4-yl]phenoxy]ethoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(OCCOC4=CC=C(C5=CC(C6=C(O)C=CC=C6)=NN=C5)C=C4)=NO3)C(C)C)C=C2)SC=N1	C43H44N6O7S	SMARCA2;SMARCA4	P51531/P51532	VHL	US-20240018134-A1
TPD-HJZ70G	US20240018134A1_43	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C(C)C)C3CC(OCCCNC4=CC=C(C5=CC(C6=C(O)C=CC=C6)=NN=C5)C=C4)=NO3)C=C2)SC=N1	C44H49N7O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	US-20240018134-A1
TPD-A76B0P	SCHEMBL25223425	(2S,4R)-4-hydroxy-1-[2-[3-[2-[4-[6-(2-hydroxyphenyl)pyridazin-4-yl]-N-methylanilino]ethoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	[H]C1=NN=C(C2=C(O)C=CC=C2)C=C1C1=CC=C(N(C)CCOC2=NOC(C(C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](C)C3=CC=C(C4=C(C)N=CS4)C=C3)C(C)C)=C2)C=C1	C44H47N7O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	US-20240018134-A1
TPD-J8XZ7V	orb2695403	(2S,4R)-4-hydroxy-1-[(2S)-2-[[2-[4-[4-[6-(2-hydroxyphenyl)pyridazin-4-yl]anilino]piperidin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; orb2695408; SCHEMBL25263778; 2760247-27-4	[H]C1=NN=C(C2=C(O)C=CC=C2)C=C1C1=CC=C(NC2CCN(CC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](C)C3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)CC2)C=C1	C46H54N8O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	US-20240018134-A1
TPD-1616AB	SCHEMBL25225762	(2S,4R)-4-hydroxy-1-[(2S)-2-[[2-[4-[4-[6-(2-hydroxyphenyl)pyridazin-4-yl]-N-methylanilino]piperidin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCC(N(C)C4=CC=C(C5=CC(C6=C(O)C=CC=C6)=NN=C5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C47H56N8O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	US-20240018134-A1
TPD-XHBYF6	SCHEMBL25226602	(2S,4R)-1-[(2S)-3,3-dimethyl-2-[[2-[4-[4-(6-oxo-1H-pyridazin-4-yl)phenyl]piperazin-1-yl]acetyl]amino]butanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCN(C4=CC=C(C5=CC(O)=NN=C5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C39H48N8O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	US-20240018134-A1
TPD-0UCDXX	US20240018134A1_48	.	CC1=C(C2=CC=C(C(CO)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCN(C4=CC=C(C5=CC(C6=C(O)C=CCC6)=NN=C5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C45H54N8O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	US-20240018134-A1
TPD-L86JFL	SCHEMBL27024907	(4R)-N-[2-(dimethylamino)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]-4-hydroxy-1-[(2S)-2-[[2-[4-[4-[6-(2-hydroxyphenyl)pyridazin-4-yl]phenyl]piperazin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(C(CN(C)C)NC(=O)C3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCN(C4=CC=C(C5=CN=NC(C6=C(O)C=CC=C6)=C5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C47H57N9O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	US-20240018134-A1
TPD-2OFZYH	orb2695461	(2S,4R)-4-hydroxy-1-[(2S)-2-[[2-[4-[5-[6-(2-hydroxyphenyl)pyridazin-4-yl]pyridin-2-yl]piperazin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; CHEMBL5193445; SCHEMBL25221485; 2760246-90-8	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCN(C4=CC=C(C5=CC(C6=C(O)C=CC=C6)=NN=C5)C=N4)CC3)C(C)(C)C)C=C2)SC=N1	C44H51N9O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	US-20240018134-A1
TPD-BTENMB	SCHEMBL25229026	(2S,4R)-4-hydroxy-1-[2-[3-[2-[4-[6-(2-hydroxyphenyl)pyridazin-4-yl]anilino]ethoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(OCCNC4=CC=C(C5=CC(C6=C(O)C=CC=C6)=NN=C5)C=C4)=NO3)C(C)C)C=C2)SC=N1	C43H45N7O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	US-20240018134-A1
TPD-1TU4Y7	CHEMBL5199901	(2S,4R)-4-hydroxy-1-[(2S)-2-[[2-[1-[4-[6-(2-hydroxyphenyl)pyridazin-4-yl]phenyl]piperidin-4-yl]acetyl]amino]-3,3-dimethylbutanoyl]-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL25218790	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CC3CCN(C4=CC=C(C5=CC(C6=C(O)C=CC=C6)=NN=C5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C46H53N7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	US-20240018134-A1
TPD-OPPOM5	SCHEMBL25221305	(2S,4R)-1-[(2S)-2-[[2-[4-[4-[6-(2-fluorophenyl)pyridazin-4-yl]phenyl]piperazin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCN(C4=CC=C(C5=CC(C6=C(F)C=CC=C6)=NN=C5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C45H51FN8O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	US-20240018134-A1
TPD-7E9VX0	US20240018134A1_8	.	CC1=C(C2=CC=C([C@H](C)N[C@H](O)C3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCN3CCN(C4=CC=C(C5=CC(C6=C(O)C=CC=C6)=NN=C5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C46H56N8O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	US-20240018134-A1
TPD-CDOPLA	SCHEMBL25221252	(2S,4R)-1-[(2S)-3,3-dimethyl-2-[[2-[4-[4-[6-(1-methylpyrazol-4-yl)pyridazin-4-yl]phenyl]piperazin-1-yl]acetyl]amino]butanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCN(C4=CC=C(C5=CC(C6=CN(C)N=C6)=NN=C5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C43H52N10O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	US-20240018134-A1
TPD-4P83I6	dBRD4-BD1	dBRD4-BD1; 2839318-19-1; dBRD4(BD1); orb1739974; CHEMBL5200680; GLXC-26325; DA-62706; HY-151593; CS-0617390; 2-((2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindolin-4-yl)oxy)-N-(2-(2-(2-(4-(5-(2-(5-isopropyl-2-methylphenoxy)pyrimidin-4-yl)-4-(4-(trifluoromethyl)phenyl)-1H-imidazol-1-yl)piperidin-1-yl)ethoxy)ethoxy)ethyl)acetamide	CC1=CC=C(C(C)C)C=C1OC1=NC(C2=C(C3=CC=C(C(F)(F)F)C=C3)N=CN2C2CCN(CCOCCOCCNC(=O)COC3=CC=CC4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)=CC=N1	C50H53F3N8O9	BRD4	O60885	CRBN	US-20240051938-A1
TPD-9EHIG9	P13A	(3R,5R)-7-[3-[3-[3-[1-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethyl]triazol-4-yl]propoxy]phenyl]-2-(4-fluorophenyl)-4-(phenylcarbamoyl)-5-propan-2-ylpyrrol-1-yl]-3,5-dihydroxyheptanoic acid; CHEMBL4641349	CC(C)C1=C(C(=O)NC2=CC=CC=C2)C(C2=CC=CC(OCCCC3=CN(CCOCCNC4=CC=CC5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)N=N3)=C2)=C(C2=CC=C(F)C=C2)N1CC[C@@H](O)C[C@@H](O)CC(=O)O	C55H59FN8O11	HMGCR	P04035	CRBN	WO-2019109415-A1
TPD-QFZLAL	P21A	(3R,5R)-7-[3-[3-[5-[1-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethyl]triazol-4-yl]pentoxy]phenyl]-2-(4-fluorophenyl)-4-(phenylcarbamoyl)-5-propan-2-ylpyrrol-1-yl]-3,5-dihydroxyheptanoic acid; CHEMBL4639117	CC(C)C1=C(C(=O)NC2=CC=CC=C2)C(C2=CC=CC(OCCCCCC3=CN(CCOCCOCCOCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)N=N3)=C2)=C(C2=CC=C(F)C=C2)N1CC[C@@H](O)C[C@@H](O)CC(=O)O	C61H71FN8O13	HMGCR	P04035	CRBN	WO-2019109415-A1
TPD-RQMH8I	WO2019109415A1_11	.	CC(C)C1=C(C(=O)NC2=CC=CC=C2)C(C2=CC=CC(OCCCCC3=CN(CCOCCOCCOCCOCCNC4=C5C(=O)N(C6CCC(O)NC6=O)C(=O)C5=CC=C4)N=N3)=C2)C(C2=CC=C(F)C=C2)N1CC[C@@H](O)C[C@@H](O)CC(=O)O	C62H77FN8O14	HMGCR	P04035	CRBN	WO-2019109415-A1
TPD-LKYCPA	P19A1	(3R,5R)-7-[3-[3-[7-[1-[7-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]heptyl]triazol-4-yl]heptoxy]phenyl]-2-(4-fluorophenyl)-4-(phenylcarbamoyl)-5-propan-2-ylpyrrol-1-yl]-3,5-dihydroxyheptanoic acid; CHEMBL4646466	CC(C)C1=C(C(=O)NC2=CC=CC=C2)C(C2=CC=CC(OCCCCCCCC3=CN(CCCCCCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)N=N3)=C2)=C(C2=CC=C(F)C=C2)N1CC[C@@H](O)C[C@@H](O)CC(=O)O	C62H73FN8O10	HMGCR	P04035	CRBN	WO-2019109415-A1
TPD-ZVDNSK	P18A1	(3R,5R)-7-[3-[3-[6-[1-[7-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]heptyl]triazol-4-yl]hexoxy]phenyl]-2-(4-fluorophenyl)-4-(phenylcarbamoyl)-5-propan-2-ylpyrrol-1-yl]-3,5-dihydroxyheptanoic acid; CHEMBL4634883	CC(C)C1=C(C(=O)NC2=CC=CC=C2)C(C2=CC=CC(OCCCCCCC3=CN(CCCCCCCNC4=CC=CC5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)N=N3)=C2)=C(C2=CC=C(F)C=C2)N1CC[C@@H](O)C[C@@H](O)CC(=O)O	C61H71FN8O10	HMGCR	P04035	CRBN	WO-2019109415-A1
TPD-A76TQQ	P17A1	(3R,5R)-7-[3-[3-[5-[1-[7-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]heptyl]triazol-4-yl]pentoxy]phenyl]-2-(4-fluorophenyl)-4-(phenylcarbamoyl)-5-propan-2-ylpyrrol-1-yl]-3,5-dihydroxyheptanoic acid; CHEMBL4639925	CC(C)C1=C(C(=O)NC2=CC=CC=C2)C(C2=CC=CC(OCCCCCC3=CN(CCCCCCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)N=N3)=C2)=C(C2=CC=C(F)C=C2)N1CC[C@@H](O)C[C@@H](O)CC(=O)O	C60H69FN8O10	HMGCR	P04035	CRBN	WO-2019109415-A1
TPD-PCU704	P16A1	(3R,5R)-7-[3-[3-[4-[1-[7-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]heptyl]triazol-4-yl]butoxy]phenyl]-2-(4-fluorophenyl)-4-(phenylcarbamoyl)-5-propan-2-ylpyrrol-1-yl]-3,5-dihydroxyheptanoic acid; CHEMBL4633564	CC(C)C1=C(C(=O)NC2=CC=CC=C2)C(C2=CC=CC(OCCCCC3=CN(CCCCCCCNC4=CC=CC5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)N=N3)=C2)=C(C2=CC=C(F)C=C2)N1CC[C@@H](O)C[C@@H](O)CC(=O)O	C59H67FN8O10	HMGCR	P04035	CRBN	WO-2019109415-A1
TPD-6BOL18	P15A1	(3R,5R)-7-[3-[3-[3-[1-[7-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]heptyl]triazol-4-yl]propoxy]phenyl]-2-(4-fluorophenyl)-4-(phenylcarbamoyl)-5-propan-2-ylpyrrol-1-yl]-3,5-dihydroxyheptanoic acid; CHEMBL4637779	CC(C)C1=C(C(=O)NC2=CC=CC=C2)C(C2=CC=CC(OCCCC3=CN(CCCCCCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)N=N3)=C2)=C(C2=CC=C(F)C=C2)N1CC[C@@H](O)C[C@@H](O)CC(=O)O	C58H65FN8O10	HMGCR	P04035	CRBN	WO-2019109415-A1
TPD-2EXHVT	P14A1	(3R,5R)-7-[3-[3-[3-[1-[6-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]hexyl]triazol-4-yl]propoxy]phenyl]-2-(4-fluorophenyl)-4-(phenylcarbamoyl)-5-propan-2-ylpyrrol-1-yl]-3,5-dihydroxyheptanoic acid; CHEMBL4637083	CC(C)C1=C(C(=O)NC2=CC=CC=C2)C(C2=CC=CC(OCCCC3=CN(CCCCCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)N=N3)=C2)=C(C2=CC=C(F)C=C2)N1CC[C@@H](O)C[C@@H](O)CC(=O)O	C57H63FN8O10	HMGCR	P04035	CRBN	WO-2019109415-A1
TPD-Q1ARZ3	CHEMBL4635561	(3R,5R)-7-[3-[3-[[1-[7-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]heptyl]triazol-4-yl]methoxy]phenyl]-2-(4-fluorophenyl)-4-(phenylcarbamoyl)-5-propan-2-ylpyrrol-1-yl]-3,5-dihydroxyheptanoic acid; PD141348	CC(C)C1=C(C(=O)NC2=CC=CC=C2)C(C2=CC=CC(OCC3=CN(CCCCCCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)N=N3)=C2)=C(C2=CC=C(F)C=C2)N1CC[C@@H](O)C[C@@H](O)CC(=O)O	C56H61FN8O10	HMGCR	P04035	CRBN	WO-2019109415-A1
TPD-366D3A	P16A	(3R,5R)-7-[3-[3-[3-[1-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethyl]triazol-4-yl]propoxy]phenyl]-2-(4-fluorophenyl)-4-(phenylcarbamoyl)-5-propan-2-ylpyrrol-1-yl]-3,5-dihydroxyheptanoic acid; CHEMBL4644182	CC(C)C1=C(C(=O)NC2=CC=CC=C2)C(C2=CC=CC(OCCCC3=CN(CCOCCOCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)N=N3)=C2)=C(C2=CC=C(F)C=C2)N1CC[C@@H](O)C[C@@H](O)CC(=O)O	C57H63FN8O12	HMGCR	P04035	CRBN	WO-2019109415-A1
TPD-LH6GWI	WO2019109415A1_3	.	C=C1CCC(N2C(=O)C3=C(C2=O)C(NCCOCCOCCOCCN2C=C(CCCOC4=CC(C5=C(C6=CC=C(F)C=C6)N(CC[C@@H](O)C[C@@H](O)CC(=O)O)C(C(C)C)=C5C(=O)NC5=CC=CC=C5)=CC=C4)N=N2)=CC=C3)C(=O)N1	C60H69FN8O12	HMGCR	P04035	CRBN	WO-2019109415-A1
TPD-42QSTO	WO2019109415A1_4	.	CC(C)C1=C(C(O)NC2=CC=CC=C2)C(C2=CC=CC(OCCCC3=CN(CCOCCOCCOCCOCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)N=N3)=C2)=C(C2=CC=C(F)C=C2)N1CC[C@@H](O)C[C@@H](O)CC(=O)O	C61H73FN8O14	HMGCR	P04035	CRBN	WO-2019109415-A1
TPD-R6NESI	P14A	(3R,5R)-7-[3-[3-[4-[1-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethyl]triazol-4-yl]butoxy]phenyl]-2-(4-fluorophenyl)-4-(phenylcarbamoyl)-5-propan-2-ylpyrrol-1-yl]-3,5-dihydroxyheptanoic acid; CHEMBL4640295	CC(C)C1=C(C(=O)NC2=CC=CC=C2)C(C2=CC=CC(OCCCCC3=CN(CCOCCNC4=CC=CC5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)N=N3)=C2)=C(C2=CC=C(F)C=C2)N1CC[C@@H](O)C[C@@H](O)CC(=O)O	C56H61FN8O11	HMGCR	P04035	CRBN	WO-2019109415-A1
TPD-X0X21K	P15A	(3R,5R)-7-[3-[3-[5-[1-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethyl]triazol-4-yl]pentoxy]phenyl]-2-(4-fluorophenyl)-4-(phenylcarbamoyl)-5-propan-2-ylpyrrol-1-yl]-3,5-dihydroxyheptanoic acid; CHEMBL4643084	CC(C)C1=C(C(=O)NC2=CC=CC=C2)C(C2=CC=CC(OCCCCCC3=CN(CCOCCNC4=CC=CC5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)N=N3)=C2)=C(C2=CC=C(F)C=C2)N1CC[C@@H](O)C[C@@H](O)CC(=O)O	C57H63FN8O11	HMGCR	P04035	CRBN	WO-2019109415-A1
TPD-FVSIBC	P17A	(3R,5R)-7-[3-[3-[4-[1-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethyl]triazol-4-yl]butoxy]phenyl]-2-(4-fluorophenyl)-4-(phenylcarbamoyl)-5-propan-2-ylpyrrol-1-yl]-3,5-dihydroxyheptanoic acid; CHEMBL4640241	CC(C)C1=C(C(=O)NC2=CC=CC=C2)C(C2=CC=CC(OCCCCC3=CN(CCOCCOCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)N=N3)=C2)=C(C2=CC=C(F)C=C2)N1CC[C@@H](O)C[C@@H](O)CC(=O)O	C58H65FN8O12	HMGCR	P04035	CRBN	WO-2019109415-A1
TPD-8FAYBI	P18A	(3R,5R)-7-[3-[3-[5-[1-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethyl]triazol-4-yl]pentoxy]phenyl]-2-(4-fluorophenyl)-4-(phenylcarbamoyl)-5-propan-2-ylpyrrol-1-yl]-3,5-dihydroxyheptanoic acid; CHEMBL4647320; SCHEMBL23636462	CC(C)C1=C(C(=O)NC2=CC=CC=C2)C(C2=CC=CC(OCCCCCC3=CN(CCOCCOCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)N=N3)=C2)=C(C2=CC=C(F)C=C2)N1CC[C@@H](O)C[C@@H](O)CC(=O)O	C59H67FN8O12	HMGCR	P04035	CRBN	WO-2019109415-A1
TPD-QPCCIG	WO2019109415A1_9	.	CC(C)/C(NCC[C@@H](O)C[C@@H](O)CC(=O)O)=C(C(=O)NC1=CC=CC=C1)/C(=C/C1=CC=C(F)C=C1)C1=CC=CC(OCCCCC2=CN(CCOCCOCCOCCNC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)N=N2)=C1	C60H71FN8O13	HMGCR	P04035	CRBN	WO-2019109415-A1
TPD-1RQNG1	SCHEMBL21401530	1-[2-[3-[2-[2-[2-[2-[2-[[4-[2-[1-(5-fluoro-2-hydroxyphenyl)-2-oxo-2-(1,3-thiazol-2-ylamino)ethyl]-3-oxo-1H-isoindol-5-yl]benzoyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)C3CC(O)CN3C(=O)C(C3=CC(OCCOCCOCCOCCOCCNC(=O)C4=CC=C(C5=CC6=C(C=C5)CN(C(C(=O)NC5=NC=CS5)C5=CC(F)=CC=C5O)C6=O)C=C4)=NO3)C(C)C)C=C2)SC=N1	C60H65FN8O13S2	EGFR	P00533	VHL	WO-2019183523-A1
TPD-16Y1W8	WO2019183523A1_1001a	.	CC1=CC=C(O)C(C(C(=O)NC2=NC=CS2)N2CC3=C(C=C(C4=CCC(C(=O)NCCOCCOCCOCCOCCOC5=NOC(C(C(=O)N6C[C@H](O)C[C@H]6C(=O)NCC6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C5)C=C4)C=C3)C2=O)=C1	C61H70N8O13S2	EGFR	P00533	VHL	WO-2019183523-A1
TPD-N92FPR	WO2019183523A1_1001b	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CC3C(=O)[C@@H](C3=CC(OCCOCCOCCOCCOCCNC(=O)C4=CC=C(C5=CC6=C(C=C5)CN(C(C(=O)NC5=NC=CS5)C5=CC(F)=CC=C5O)C6=O)C=C4)=NO3)C(C)C)C=C2)SC=N1	C61H66FN7O13S2	EGFR	P00533	VHL	WO-2019183523-A1
TPD-QSWGO9	WO2019183523A1_1002	.	CC1=C(C2=CC=C(CNC(=O)C3CC(O)CC3C(=O)C(C3=CC(OCCOCCOCCOCCOCC#CC4=CC5=C(C=C4)CN(C(C(=O)NC4=NC=CS4)C4=CC(F)=CC=C4O)C5=O)=NO3)C(C)C)C=C2)SC=N1	C55H59FN6O12S2	EGFR	P00533	VHL	WO-2019183523-A1
TPD-CVNI0J	SCHEMBL21401379	(2S,4R)-1-[2-[3-[2-[2-[2-[2-[3-[2-[1-(5-fluoro-2-hydroxyphenyl)-2-oxo-2-(1,3-thiazol-2-ylamino)ethyl]-3-oxo-1H-isoindol-5-yl]prop-2-ynoxy]ethoxy]ethoxy]ethoxy]ethoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(OCCOCCOCCOCCOCC#CC4=CC5=C(C=C4)CN(C(C(=O)NC4=NC=CS4)C4=CC(F)=CC=C4O)C5=O)=NO3)C(C)C)C=C2)SC=N1	C54H58FN7O12S2	EGFR	P00533	VHL	WO-2019183523-A1
TPD-L97IBV	WO2019183523A1_1002b	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(OCCOCCOCCOCCOCC#CC4=CC5=C(C=C4)CN(C(C(=O)NC4=NC=CS4)C4=CC(F)=CC=C4O)C5=O)=NO3)C(C)C)C=C2)SC=N1	C54H58FN7O12S2	EGFR	P00533	VHL	WO-2019183523-A1
TPD-DI5RK9	SCHEMBL21401531	1-[2-[[2-[2-[2-[2-[2-[2-[[4-[2-[1-(5-fluoro-2-hydroxyphenyl)-2-oxo-2-(1,3-thiazol-2-ylamino)ethyl]-3-oxo-1H-isoindol-5-yl]benzoyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)C3CC(O)CN3C(=O)C(NC(=O)COCCOCCOCCOCCOCCNC(=O)C3=CC=C(C4=CC5=C(C=C4)CN(C(C(=O)NC4=NC=CS4)C4=CC(F)=CC=C4O)C5=O)C=C3)C(C)(C)C)C=C2)SC=N1	C60H69FN8O13S2	EGFR	P00533	VHL	WO-2019183523-A1
TPD-GLL039	WO2019183523A1_1003a	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CC3C(=O)C(NC(=O)COCCOCCOCCOCCOCCNC(=O)C3=CC=C(C4=CC5=C(C=C4)CN(C(C(=O)NC4=NC=CS4)C4=CC(F)=CC=C4O)C5=O)C=C3)C(C)(C)C)C=C2)SC=N1	C61H70FN7O13S2	EGFR	P00533	VHL	WO-2019183523-A1
TPD-18BZFY	SCHEMBL21401385	(2S,4R)-1-[(2S)-2-[[2-[2-[2-[2-[2-[2-[[4-[2-[1-(5-fluoro-2-hydroxyphenyl)-2-oxo-2-(1,3-thiazol-2-ylamino)ethyl]-3-oxo-1H-isoindol-5-yl]benzoyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCOCCOCCNC(=O)C3=CC=C(C4=CC5=C(C=C4)CN(C(C(=O)NC4=NC=CS4)C4=CC(F)=CC=C4O)C5=O)C=C3)C(C)(C)C)C=C2)SC=N1	C60H69FN8O13S2	EGFR	P00533	VHL	WO-2019183523-A1
TPD-4Y1NAV	WO2021020586A1_1	.	CN/C(C(=O)N1CCN(C(=O)[C@@H](NC(=O)[C@H](C)NC)C2CCCCC2)CC1)=C(/C(=O)N(C)CCOCCOCCOC1=NOC(CN2CCC(OC3=CC=NC4=C3SC=C4)CC2)=C1)C1=CC=C(F)C(F)=C1	C50H67F2N9O9S	IRAK3	Q9Y616	XIAP	WO-2021020586-A1
TPD-XNZY6K	SCHEMBL22944437	(2S)-N-[(1S)-1-cyclohexyl-2-[4-[5,6-difluoro-1-methyl-4-[2-[2-[2-[2-[[5-[(4-thieno[3,2-b]pyridin-7-yloxypiperidin-1-yl)methyl]-1,2-oxazol-3-yl]oxy]ethoxy]ethoxy]ethoxy]ethoxy]indole-2-carbonyl]piperazin-1-yl]-2-oxoethyl]-2-(methylamino)propanamide; SCHEMBL29808644	CN[C@@H](C)C(=O)N[C@H](C(=O)N1CCN(C(=O)C2=CC3=C(C=C(F)C(F)=C3OCCOCCOCCOCCOC3=NOC(CN4CCC(OC5=C6SC=CC6=NC=C5)CC4)=C3)N2C)CC1)C1CCCCC1	C50H66F2N8O10S	IRAK3	Q9Y616	XIAP	WO-2021020586-A1
TPD-WW7V0F	SCHEMBL22944689	(2S)-N-[(1S)-1-cyclohexyl-2-[4-[2-methyl-1-[2-[2-[2-[2-[[5-[(4-thieno[3,2-b]pyridin-7-yloxypiperidin-1-yl)methyl]-1,2-oxazol-3-yl]oxy]ethoxy]ethoxy]ethoxy]ethyl]indole-5-carbonyl]piperazin-1-yl]-2-oxoethyl]-2-(methylamino)propanamide	CN[C@@H](C)C(=O)N[C@H](C(=O)N1CCN(C(=O)C2=CC3=C(C=C2)N(CCOCCOCCOCCOC2=NOC(CN4CCC(OC5=C6SC=CC6=NC=C5)CC4)=C2)C(C)=C3)CC1)C1CCCCC1	C50H68N8O9S	IRAK3	Q9Y616	XIAP	WO-2021020586-A1
TPD-Q2R6QD	SCHEMBL24760038	2-[4-[(2S)-2-cyclohexyl-2-[[(2S)-2-(methylamino)propanoyl]amino]acetyl]piperazine-1-carbonyl]-6-methoxy-1-methyl-N-[2-[2-[2-[4-(4-thieno[3,2-d]pyrimidin-4-yloxypiperidin-1-yl)sulfonylphenoxy]ethoxy]ethoxy]ethyl]indole-3-carboxamide	CN[C@@H](C)C(=O)N[C@H](C(=O)N1CCN(C(=O)C2=C(C(=O)NCCOCCOCCOC3=CC=C(S(=O)(=O)N4CCC(OC5=C6SC=CC6=NC=N5)CC4)C=C3)C3=C(C=C(OC)C=C3)N2C)CC1)C1CCCCC1	C51H67N9O11S2	IRAK3	Q9Y616	XIAP	WO-2021020586-A1
TPD-3TFX9L	SCHEMBL22945080	1-[(2R)-4-(5,6-difluoro-1-methylindole-2-carbonyl)-2-methylpiperazin-1-yl]-2-[(2R,5R)-5-methyl-2-[2-[2-[2-[[5-[(4-thieno[3,2-b]pyridin-7-yloxypiperidin-1-yl)methyl]-1,2-oxazol-3-yl]oxy]ethoxy]ethoxy]ethoxymethyl]piperazin-1-yl]ethanone	C[C@@H]1CN(CC(=O)N2CCN(C(=O)C3=CC4=C(C=C(F)C(F)=C4)N3C)C[C@H]2C)[C@@H](COCCOCCOCCOC2=NOC(CN3CCC(OC4=C5SC=CC5=NC=C4)CC3)=C2)CN1	C45H58F2N8O8S	IRAK3	Q9Y616	XIAP	WO-2021020586-A1
TPD-NS8QQ3	SCHEMBL22945175	(2S)-N-[(1S)-1-cyclohexyl-2-[4-[5,6-difluoro-1-methyl-3-[2-[2-[2-[[5-[(4-thieno[3,2-b]pyridin-7-yloxypiperidin-1-yl)methyl]-1,2-oxazol-3-yl]oxy]ethoxy]ethoxy]ethoxy]indole-2-carbonyl]piperazin-1-yl]-2-oxoethyl]-2-(methylamino)propanamide	CN[C@@H](C)C(=O)N[C@H](C(=O)N1CCN(C(=O)C2=C(OCCOCCOCCOC3=NOC(CN4CCC(OC5=C6SC=CC6=NC=C5)CC4)=C3)C3=C(C=C(F)C(F)=C3)N2C)CC1)C1CCCCC1	C48H62F2N8O9S	IRAK3	Q9Y616	XIAP	WO-2021020586-A1
TPD-ZULU4Q	SCHEMBL22944694	(2S)-N-[(1S)-1-cyclohexyl-2-[4-[5,6-difluoro-1-[2-[methyl-[2-[2-[2-[2-[[5-[(4-thieno[3,2-b]pyridin-7-yloxypiperidin-1-yl)methyl]-1,2-oxazol-3-yl]oxy]ethoxy]ethoxy]ethoxy]ethyl]amino]-2-oxoethyl]indole-2-carbonyl]piperazin-1-yl]-2-oxoethyl]-2-(methylamino)propanamide	CN[C@@H](C)C(=O)N[C@H](C(=O)N1CCN(C(=O)C2=CC3=CC(F)=C(F)C=C3N2CC(=O)N(C)CCOCCOCCOCCOC2=NOC(CN3CCC(OC4=C5SC=CC5=NC=C4)CC3)=C2)CC1)C1CCCCC1	C52H69F2N9O10S	IRAK3	Q9Y616	XIAP	WO-2021020586-A1
TPD-PWH43Y	SCHEMBL22944691	(2S)-N-[(1S)-1-cyclohexyl-2-[4-[5,6-difluoro-1-[2-oxo-2-[(2S)-2-[[5-[(4-thieno[3,2-b]pyridin-7-yloxypiperidin-1-yl)methyl]-1,2-oxazol-3-yl]oxymethyl]pyrrolidin-1-yl]ethyl]indole-2-carbonyl]piperazin-1-yl]-2-oxoethyl]-2-(methylamino)propanamide	CN[C@@H](C)C(=O)N[C@H](C(=O)N1CCN(C(=O)C2=CC3=CC(F)=C(F)C=C3N2CC(=O)N2CCC[C@H]2COC2=NOC(CN3CCC(OC4=C5SC=CC5=NC=C4)CC3)=C2)CC1)C1CCCCC1	C48H59F2N9O7S	IRAK3	Q9Y616	XIAP	WO-2021020586-A1
TPD-M0TW1V	SCHEMBL22945178	(2S)-N-[(1S)-1-cyclohexyl-2-[4-[5-fluoro-1-[2-oxo-2-[(2S)-2-[[5-[(4-thieno[3,2-b]pyridin-7-yloxypiperidin-1-yl)methyl]-1,2-oxazol-3-yl]oxymethyl]pyrrolidin-1-yl]ethyl]indole-2-carbonyl]piperazin-1-yl]-2-oxoethyl]-2-(methylamino)propanamide	CN[C@@H](C)C(=O)N[C@H](C(=O)N1CCN(C(=O)C2=CC3=C(C=CC(F)=C3)N2CC(=O)N2CCC[C@H]2COC2=NOC(CN3CCC(OC4=CC=NC5=C4SC=C5)CC3)=C2)CC1)C1CCCCC1	C48H60FN9O7S	IRAK3	Q9Y616	XIAP	WO-2021020586-A1
TPD-BBZ6DQ	SCHEMBL24760042	(2S)-N-[1-cyclohexyl-2-[(3S)-4-[5,6-difluoro-1-[2-oxo-2-[(2S)-2-[[5-[(4-thieno[3,2-b]pyridin-7-yloxypiperidin-1-yl)methyl]-1,2-oxazol-3-yl]oxymethyl]pyrrolidin-1-yl]ethyl]indole-2-carbonyl]-3-methylpiperazin-1-yl]-2-oxoethyl]-2-(methylamino)propanamide	CN[C@@H](C)C(=O)NC(C(=O)N1CCN(C(=O)C2=CC3=CC(F)=C(F)C=C3N2CC(=O)N2CCC[C@H]2COC2=NOC(CN3CCC(OC4=C5SC=CC5=NC=C4)CC3)=C2)[C@@H](C)C1)C1CCCCC1	C49H61F2N9O7S	IRAK3	Q9Y616	XIAP	WO-2021020586-A1
TPD-OPLZS9	SCHEMBL22947340	(2S)-N-[(1S)-1-cyclohexyl-2-[(3S)-4-[5-fluoro-1-[2-oxo-2-[(2S)-2-[[5-[(4-thieno[3,2-b]pyridin-7-yloxypiperidin-1-yl)methyl]-1,2-oxazol-3-yl]oxymethyl]pyrrolidin-1-yl]ethyl]indole-2-carbonyl]-3-methylpiperazin-1-yl]-2-oxoethyl]-2-(methylamino)propanamide	CN[C@@H](C)C(=O)N[C@H](C(=O)N1CCN(C(=O)C2=CC3=CC(F)=CC=C3N2CC(=O)N2CCC[C@H]2COC2=NOC(CN3CCC(OC4=C5SC=CC5=NC=C4)CC3)=C2)[C@@H](C)C1)C1CCCCC1	C49H62FN9O7S	IRAK3	Q9Y616	XIAP	WO-2021020586-A1
TPD-20PEC2	SCHEMBL23276189	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[5-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]pent-4-ynyl]piperidin-3-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCCN(CCCC#CC6=CC=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C63H65ClN10O10S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-OHHCGP	SCHEMBL23276702	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]acetyl]piperidin-4-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC=C(NCC5CCN(C(=O)CNC6=CC=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C([N+](=O)[O-])=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C60H62ClN11O11S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-D8KZ79	WO2021078301A1_SIAIS230149	.	C[N+](=O)C1=C(NCC2CCN(C(=O)CCNC3=CC=CC4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)C=CC(S(=O)(=O)NC(=O)C2=CC=C(N3CCN(CC4=C(C5=CC=C(Cl)C=C5)CC(C)(C)CC4)CC3)C=C2OC2=CN=C3NC=CC3=C2)=C1	C62H67ClN11O10S+	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-GEIPQ3	SCHEMBL23276061	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]butanoyl]piperidin-4-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCN(C(=O)CCCNC6=CC=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C62H66ClN11O11S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-UPN4CQ	SCHEMBL23276618	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[5-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]pentanoyl]piperidin-4-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCN(C(=O)CCCCNC6=CC=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C63H68ClN11O11S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-2YE7UA	SCHEMBL23276025	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[6-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]hexanoyl]piperidin-4-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCN(C(=O)CCCCCNC6=CC=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C64H70ClN11O11S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-P7Z1EM	SCHEMBL23275972	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[7-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]heptanoyl]piperidin-4-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCN(C(=O)CCCCCCNC6=CC=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C65H72ClN11O11S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-ANT864	SCHEMBL23276279	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]sulfanylpropanoyl]piperidin-4-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCN(C(=O)CCSC6=CC=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C61H63ClN10O11S2	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-785LZY	SCHEMBL23275943	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[5-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]sulfanylpentanoyl]piperidin-4-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCN(C(=O)CCCCSC6=CC=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C63H67ClN10O11S2	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-0A49OY	SCHEMBL23276545	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[7-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]sulfanylheptanoyl]piperidin-4-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCN(C(=O)CCCCCCSC6=CC=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C65H71ClN10O11S2	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-DCTCLH	SCHEMBL23276852	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]sulfanyl]acetyl]piperidin-4-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCN(C(=O)CSC6=CC=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)CC5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C60H63ClN10O10S2	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-DHHATX	SCHEMBL23276287	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[4-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]sulfanyl]butanoyl]piperidin-4-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCN(C(=O)CCCSC6=CC=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)CC5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C62H67ClN10O10S2	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-7SIMSW	SCHEMBL23276308	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[6-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]sulfanyl]hexanoyl]piperidin-4-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCN(C(=O)CCCCCSC6=CC=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)CC5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C64H71ClN10O10S2	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-9F4X72	SCHEMBL23276264	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]sulfanylethoxy]acetyl]piperidin-4-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCN(C(=O)COCCSC6=CC=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C62H65ClN10O12S2	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-OCXD5W	WO2021078301A1_SIAIS230166	.	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([NH2+][O-])=C(NCC5CCN(C(=O)COCCOCCOCCSC6=CC=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C66H75ClN10O13S2	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-UJKKT0	SCHEMBL23276536	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[2-[2-[2-[2-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]sulfanylethoxy]ethoxy]ethoxy]ethoxy]ethoxy]acetyl]piperidin-4-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCN(C(=O)COCCOCCOCCOCCOCCSC6=CC=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C70H81ClN10O16S2	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-ECKW52	SCHEMBL23276225	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]sulfanyl]ethoxy]ethoxy]acetyl]piperidin-4-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCN(C(=O)COCCOCCSC6=CC=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)CC5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C64H71ClN10O12S2	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-VMBZVR	SCHEMBL23276074	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[2-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]sulfanyl]ethoxy]ethoxy]ethoxy]ethoxy]acetyl]piperidin-4-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCN(C(=O)COCCOCCOCCOCCSC6=CC=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)CC5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C68H79ClN10O14S2	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-OAXU7F	SCHEMBL23276587	(2S,4R)-1-[(2S)-2-[[4-[4-[[4-[[4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzoyl]sulfamoyl]-2-nitroanilino]methyl]piperidin-1-yl]-4-oxobutanoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL23276590	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCC(=O)N3CCC(CNC4=C([N+](=O)[O-])C=C(S(=O)(=O)NC(=O)C5=CC=C(N6CCN(CC7=C(C8=CC=C(Cl)C=C8)CC(C)(C)CC7)CC6)C=C5OC5=CN=C6NC=CC6=C5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C71H83ClN12O11S2	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-7EJYIG	WO2021078301A1_SIAIS230171	.	CC1=C(C2=CC=C(CNC(=O)C3C[C@@H](O)CN3C(=O)C(NC(=O)CCCCC(=O)N3CCC(CNC4=C([N+](=O)[O-])C=C(S(=O)(=O)NC(=O)C5=CC=C(N6CCN(CC7=C(C8=CC=C(Cl)C=C8)CC(C)(C)CC7)CC6)C=C5OC5=CN=C6NC=CC6=C5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C73H87ClN12O11S2	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-33JSKF	WO2021078301A1_SIAIS230172	.	CC1=C(C2=CC=C(CNC(=O)C3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCC(=O)N3CCC(CNC4=C([N+](=O)[O-])C=C(S(=O)(=O)NC(=O)C5=CC=C(N6CCN(CC7=C(C8=CC=C(Cl)C=C8)CC(C)(C)CC7)CC6)C=C5OC5=CN=C6NC=CC6=C5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C75H91ClN12O11S2	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-R81BER	WO2021078301A1_SIAIS230173	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(NC(=O)CCCCCCCCC(=O)N3CCC(CNC4=C([N+](=O)[O-])C=C(S(=O)(=O)NC(=O)C5CC=C(N6CCN(CC7=C(C8=CC=C(Cl)C=C8)CC(C)(C)CC7)CC6)C=C5OC5=CN=C6NC=CC6=C5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C77H97ClN12O11S2	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-8B9PWS	WO2021078301A1_SIAIS255044	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]acetyl]piperidin-4-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC=C(NCC5CCN(C(=O)CNC6=CC=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)CC5)C([N+](=O)[O-])=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C60H64ClN11O10S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-LQFJ8R	SCHEMBL28553982	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[3-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]propanoyl]piperidin-4-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCN(C(=O)CCNC6=CC=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)CC5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C61H66ClN11O10S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-0JNOGY	SCHEMBL23277038	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[4-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]butanoyl]piperidin-4-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCN(C(=O)CCCNC6=CC=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)CC5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C62H68ClN11O10S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-XYROVN	WO2021078301A1_SIAIS255047	.	CC1(C)CCC(CN2CCN(C3=CC=C(C(O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCN(C(=O)CCCCNC6=CC=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)CC5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C63H72ClN11O10S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-DQIG80	SCHEMBL28911802	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[6-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]hexanoyl]piperidin-4-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCN(C(=O)CCCCCNC6=CC=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)CC5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C64H72ClN11O10S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-AP4304	WO2021078301A1_SIAIS255049	.	CC1(C)CCC(CN2CCN(C3=CC=C(C(O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCN(C(=O)CCCCCCNC6=CC=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)CC5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C65H76ClN11O10S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-MJTGYP	SCHEMBL23276379	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[5-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]pent-4-ynyl]piperidin-4-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCN(CCCC#CC6=CC=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)CC5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C63H67ClN10O9S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-Y0B1QV	SCHEMBL23276180	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[6-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]hex-5-ynyl]piperidin-4-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCN(CCCCC#CC6=CC=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)CC5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C64H69ClN10O9S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-ATG0Z2	SCHEMBL23276153	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]butyl]piperidin-4-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCN(CCCCC6=CC=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)CC5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C62H69ClN10O9S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-TXE2D2	SCHEMBL23276270	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]butyl]piperidin-3-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCCN(CCCCC6=CC=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)C5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C62H69ClN10O9S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-J3MT5J	SCHEMBL23276461	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[5-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]pent-4-ynyl]piperidin-3-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCCN(CCCC#CC6=CC=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)C5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C63H67ClN10O9S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-CYBQQF	SCHEMBL23276620	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[6-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]hex-5-ynyl]piperidin-3-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCCN(CCCCC#CC6=CC=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)C5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C64H69ClN10O9S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-D7MY1T	SCHEMBL23276296	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[3-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]propanoyl]piperidin-3-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCCN(C(=O)CCNC6=CC=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C61H64ClN11O11S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-NB23GR	SCHEMBL23275987	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]butanoyl]piperidin-3-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCCN(C(=O)CCCNC6=CC=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C62H66ClN11O11S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-7L0MBM	SCHEMBL23276610	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[6-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]hexanoyl]piperidin-3-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCCN(C(=O)CCCCCNC6=CC=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C64H70ClN11O11S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-HVW6DC	SCHEMBL23276754	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[7-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]heptanoyl]piperidin-3-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCCN(C(=O)CCCCCCNC6=CC=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C65H72ClN11O11S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-9RM4FS	SCHEMBL23276259	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[8-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]octanoyl]piperidin-3-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCCN(C(=O)CCCCCCCNC6=CC=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C66H74ClN11O11S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-9QYQ9A	SCHEMBL23276544	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]acetyl]piperidin-3-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCCN(C(=O)CNC6=CC=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C60H62ClN11O11S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-HRYK0E	SCHEMBL23276364	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]sulfanylacetyl]piperidin-3-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCCN(C(=O)CSC6=CC=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C60H61ClN10O11S2	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-IIY79V	SCHEMBL23276615	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]sulfanylpropanoyl]piperidin-3-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCCN(C(=O)CCSC6=CC=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C61H63ClN10O11S2	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-8OI40M	SCHEMBL23276516	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]sulfanylbutanoyl]piperidin-3-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCCN(C(=O)CCCSC6=CC=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C62H65ClN10O11S2	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-5QL6D2	SCHEMBL23276137	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[5-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]sulfanylpentanoyl]piperidin-3-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCCN(C(=O)CCCCSC6=CC=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C63H67ClN10O11S2	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-UQG2WK	SCHEMBL23276213	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[6-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]sulfanylhexanoyl]piperidin-3-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCCN(C(=O)CCCCCSC6=CC=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C64H69ClN10O11S2	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-MMPMEX	SCHEMBL23276777	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[7-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]sulfanylheptanoyl]piperidin-3-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCCN(C(=O)CCCCCCSC6=CC=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C65H71ClN10O11S2	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-D0SXJ8	WO2021078301A1_SIAIS255151	.	C=C1C2=C(CN1C1CCC(=O)NC1=O)C(SCC(=O)N1CCCC(CNC3=C([N+](=O)[O-])C=C(S(=O)(=O)NC(=O)C4=CC=C(N5CCN(CC6=C(C7=CC=C(Cl)C=C7)CC(C)(C)CC6)CC5)C=C4OC4=CN=C5NC=CC5=C4)C=C3)C1)=CC=C2	C61H65ClN10O9S2	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-R8V1J5	SCHEMBL23276571	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[3-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]sulfanyl]propanoyl]piperidin-3-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCCN(C(=O)CCSC6=CC=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)C5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C61H65ClN10O10S2	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-L3XE41	SCHEMBL23276679	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[4-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]sulfanyl]butanoyl]piperidin-3-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCCN(C(=O)CCCSC6=CC=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)C5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C62H67ClN10O10S2	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-NLWX60	SCHEMBL23276540	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[5-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]sulfanyl]pentanoyl]piperidin-3-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCCN(C(=O)CCCCSC6=CC=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)C5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C63H69ClN10O10S2	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-1IROYG	SCHEMBL23276588	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[6-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]sulfanyl]hexanoyl]piperidin-3-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCCN(C(=O)CCCCCSC6=CC=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)C5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C64H71ClN10O10S2	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-DG3YB1	WO2021078301A1_SIAIS255156	.	C[N+](=O)C1=C(NCC2CCCN(C(=O)CCCCCCSC3=CC=CC4=C3CN(C3CCC(=O)NC3=O)C4=O)C2)C=CC(S(=O)(=O)NC(=O)C2=CC=C(N3CCN(CC4=C(C5=CC=C(Cl)C=C5)CC(C)(C)CC4)CC3)C=C2OC2=CN=C3NC=CC3=C2)=C1	C66H76ClN10O9S2+	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-6ELUPM	WO2021078301A1_SIAIS255157	.	C[N+](=O)C1=C(NCC2CCCN(C(=O)CNC3=CC=CC4=C3CN(C3CCC(=O)NC3=O)C4=O)C2)C=CC(S(=O)(=O)NC(=O)C2=CC=C(N3CCN(CC4=C(C5=CC=C(Cl)C=C5)CC(C)(C)CC4)CC3)C=C2OC2=CN=C3NC=CC3=C2)=C1	C61H67ClN11O9S+	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-3EPVEQ	SCHEMBL28554450	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[4-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]butanoyl]piperidin-3-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCCN(C(=O)CCCNC6=CC=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)C5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C62H68ClN11O10S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-4G71EN	SCHEMBL28565018	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[5-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]pentanoyl]piperidin-3-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCCN(C(=O)CCCCNC6=CC=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)C5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C63H70ClN11O10S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-FQAZER	SCHEMBL28560175	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[6-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]hexanoyl]piperidin-3-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCCN(C(=O)CCCCCNC6=CC=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)C5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C64H72ClN11O10S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-8K9Z76	SCHEMBL28560644	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[7-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]heptanoyl]piperidin-3-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCCN(C(=O)CCCCCCNC6=CC=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)C5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C65H74ClN11O10S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-LP9URC	SCHEMBL23276187	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[3-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]propanoyl]piperidin-3-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCCN(C(=O)CCC6=CC=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)C5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C61H65ClN10O10S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-UFQUOC	SCHEMBL23276194	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[3-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]propyl]piperidin-4-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCN(CCCNC6=CC=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C61H66ClN11O10S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-RH3C3L	SCHEMBL23276372	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[5-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]pentyl]piperidin-4-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCN(CCCCCNC6=CC=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C63H70ClN11O10S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-9G8VVS	SCHEMBL23276534	4-[4-[[2-(4-chlorophenyl)-6-[[1-[3-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]propanoyl]azetidin-3-yl]methoxy]phenyl]methyl]piperazin-1-yl]-N-[3-nitro-4-(oxan-4-ylmethylamino)phenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	O=C1CCC(N2C(=O)C3=CC=CC(NCCC(=O)N4CC(COC5=CC=CC(C6=CC=C(Cl)C=C6)=C5CN5CCN(C6=CC=C(C(=O)NS(=O)(=O)C7=CC=C(NCC8CCOCC8)C([N+](=O)[O-])=C7)C(OC7=CN=C8NC=CC8=C7)=C6)CC5)C4)=C3C2=O)C(=O)N1	C63H62ClN11O13S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-KGLX6U	SCHEMBL23276531	4-[4-[[2-(4-chlorophenyl)-6-[[1-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]butanoyl]azetidin-3-yl]methoxy]phenyl]methyl]piperazin-1-yl]-N-[3-nitro-4-(oxan-4-ylmethylamino)phenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	O=C1CCC(N2C(=O)C3=CC=CC(NCCCC(=O)N4CC(COC5=CC=CC(C6=CC=C(Cl)C=C6)=C5CN5CCN(C6=CC=C(C(=O)NS(=O)(=O)C7=CC=C(NCC8CCOCC8)C([N+](=O)[O-])=C7)C(OC7=CN=C8NC=CC8=C7)=C6)CC5)C4)=C3C2=O)C(=O)N1	C64H64ClN11O13S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-L6THRV	SCHEMBL23276646	4-[4-[[2-(4-chlorophenyl)-6-[[1-[5-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]pentanoyl]azetidin-3-yl]methoxy]phenyl]methyl]piperazin-1-yl]-N-[3-nitro-4-(oxan-4-ylmethylamino)phenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	O=C1CCC(N2C(=O)C3=CC=CC(NCCCCC(=O)N4CC(COC5=CC=CC(C6=CC=C(Cl)C=C6)=C5CN5CCN(C6=CC=C(C(=O)NS(=O)(=O)C7=CC=C(NCC8CCOCC8)C([N+](=O)[O-])=C7)C(OC7=CN=C8NC=CC8=C7)=C6)CC5)C4)=C3C2=O)C(=O)N1	C65H66ClN11O13S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-XEDO6U	SCHEMBL23276301	4-[4-[[2-(4-chlorophenyl)-6-[[1-[6-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]hexanoyl]azetidin-3-yl]methoxy]phenyl]methyl]piperazin-1-yl]-N-[3-nitro-4-(oxan-4-ylmethylamino)phenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	O=C1CCC(N2C(=O)C3=CC=CC(NCCCCCC(=O)N4CC(COC5=CC=CC(C6=CC=C(Cl)C=C6)=C5CN5CCN(C6=CC=C(C(=O)NS(=O)(=O)C7=CC=C(NCC8CCOCC8)C([N+](=O)[O-])=C7)C(OC7=CN=C8NC=CC8=C7)=C6)CC5)C4)=C3C2=O)C(=O)N1	C66H68ClN11O13S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-4069HQ	SCHEMBL23276662	4-[4-[[2-(4-chlorophenyl)-6-[[1-[7-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]heptanoyl]azetidin-3-yl]methoxy]phenyl]methyl]piperazin-1-yl]-N-[3-nitro-4-(oxan-4-ylmethylamino)phenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide; SCHEMBL23298730	O=C1CCC(N2C(=O)C3=CC=CC(NCCCCCCC(=O)N4CC(COC5=CC=CC(C6=CC=C(Cl)C=C6)=C5CN5CCN(C6=CC=C(C(=O)NS(=O)(=O)C7=CC=C(NCC8CCOCC8)C([N+](=O)[O-])=C7)C(OC7=CN=C8NC=CC8=C7)=C6)CC5)C4)=C3C2=O)C(=O)N1	C67H70ClN11O13S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-56MD5V	SCHEMBL23276964	4-[4-[[2-(4-chlorophenyl)-6-[[1-[5-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]pent-4-ynyl]azetidin-3-yl]methoxy]phenyl]methyl]piperazin-1-yl]-N-[3-nitro-4-(oxan-4-ylmethylamino)phenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	O=C1CCC(N2CC3=C(C#CCCCN4CC(COC5=CC=CC(C6=CC=C(Cl)C=C6)=C5CN5CCN(C6=CC=C(C(=O)NS(=O)(=O)C7=CC=C(NCC8CCOCC8)C([N+](=O)[O-])=C7)C(OC7=CN=C8NC=CC8=C7)=C6)CC5)C4)C=CC=C3C2=O)C(=O)N1	C65H65ClN10O11S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-PPXO1W	SCHEMBL23276638	4-[4-[[2-(4-chlorophenyl)-6-[[1-[6-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]hex-5-ynyl]azetidin-3-yl]methoxy]phenyl]methyl]piperazin-1-yl]-N-[3-nitro-4-(oxan-4-ylmethylamino)phenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	O=C1CCC(N2CC3=C(C#CCCCCN4CC(COC5=CC=CC(C6=CC=C(Cl)C=C6)=C5CN5CCN(C6=CC=C(C(=O)NS(=O)(=O)C7=CC=C(NCC8CCOCC8)C([N+](=O)[O-])=C7)C(OC7=CN=C8NC=CC8=C7)=C6)CC5)C4)C=CC=C3C2=O)C(=O)N1	C66H67ClN10O11S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-TS3Q3P	SCHEMBL23276569	4-[4-[[2-(4-chlorophenyl)-6-[[1-[8-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]oct-7-ynyl]azetidin-3-yl]methoxy]phenyl]methyl]piperazin-1-yl]-N-[3-nitro-4-(oxan-4-ylmethylamino)phenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	O=C1CCC(N2CC3=C(C#CCCCCCCN4CC(COC5=CC=CC(C6=CC=C(Cl)C=C6)=C5CN5CCN(C6=CC=C(C(=O)NS(=O)(=O)C7=CC=C(NCC8CCOCC8)C([N+](=O)[O-])=C7)C(OC7=CN=C8NC=CC8=C7)=C6)CC5)C4)C=CC=C3C2=O)C(=O)N1	C68H71ClN10O11S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-RRLCEN	SCHEMBL23276586	4-[4-[[2-(4-chlorophenyl)-6-[[1-[9-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]non-8-ynyl]azetidin-3-yl]methoxy]phenyl]methyl]piperazin-1-yl]-N-[3-nitro-4-(oxan-4-ylmethylamino)phenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	O=C1CCC(N2CC3=C(C#CCCCCCCCN4CC(COC5=CC=CC(C6=CC=C(Cl)C=C6)=C5CN5CCN(C6=CC=C(C(=O)NS(=O)(=O)C7=CC=C(NCC8CCOCC8)C([N+](=O)[O-])=C7)C(OC7=CN=C8NC=CC8=C7)=C6)CC5)C4)C=CC=C3C2=O)C(=O)N1	C69H73ClN10O11S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-3V4IK5	SCHEMBL23275974	4-[4-[[2-(4-chlorophenyl)-6-[[1-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]acetyl]azetidin-3-yl]methoxy]phenyl]methyl]piperazin-1-yl]-N-[3-nitro-4-(oxan-4-ylmethylamino)phenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	O=C1CCC(N2C(=O)C3=CC=CC(NCC(=O)N4CC(COC5=CC=CC(C6=CC=C(Cl)C=C6)=C5CN5CCN(C6=CC=C(C(=O)NS(=O)(=O)C7=CC=C(NCC8CCOCC8)C([N+](=O)[O-])=C7)C(OC7=CN=C8NC=CC8=C7)=C6)CC5)C4)=C3C2=O)C(=O)N1	C62H60ClN11O13S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-5CGA8W	SCHEMBL23276473	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[8-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]oct-7-ynyl]piperidin-4-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCN(CCCCCCC#CC6=CC=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)CC5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C66H73ClN10O9S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-IJYBJF	SCHEMBL23276391	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[9-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]non-8-ynyl]piperidin-4-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCN(CCCCCCCC#CC6=CC=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)CC5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C67H75ClN10O9S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-UFEJSZ	SCHEMBL23276447	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[8-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]oct-7-ynyl]piperidin-3-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCCN(CCCCCCC#CC6=CC=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)C5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C66H73ClN10O9S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-F7PN3J	WO2021078301A1_SIAIS268181	.	CC1(C)CCC(CN2CCN(C3=CC=C(C(O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCCN(CCCCCCCC#CC6=CC=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)C5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C67H77ClN10O9S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-QOUY5L	SCHEMBL28565258	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethyl]triazol-4-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5=CN(CCNC6=CC=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7=O)N=N5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C57H56ClN13O10S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-2PJ9SY	SCHEMBL28912361	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[3-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]propyl]triazol-4-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5=CN(CCCNC6=CC=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7=O)N=N5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C58H58ClN13O10S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-9FSK8R	SCHEMBL28553535	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[5-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]pentyl]triazol-4-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5=CN(CCCCCNC6=CC=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7=O)N=N5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C60H62ClN13O10S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-W7VM8N	SCHEMBL23276521	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[7-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]hept-6-ynyl]piperidin-4-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCN(CCCCCC#CC6=CC=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)CC5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C65H71ClN10O9S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-KWRPP7	SCHEMBL23276432	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[7-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]hept-6-ynyl]piperidin-3-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCCN(CCCCCC#CC6=CC=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)C5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C65H71ClN10O9S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-ABTN6W	SCHEMBL23276526	4-[4-[[2-(4-chlorophenyl)-6-[[1-[7-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]hept-6-ynyl]azetidin-3-yl]methoxy]phenyl]methyl]piperazin-1-yl]-N-[3-nitro-4-(oxan-4-ylmethylamino)phenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	O=C1CCC(N2CC3=C(C#CCCCCCN4CC(COC5=CC=CC(C6=CC=C(Cl)C=C6)=C5CN5CCN(C6=CC=C(C(=O)NS(=O)(=O)C7=CC=C(NCC8CCOCC8)C([N+](=O)[O-])=C7)C(OC7=CN=C8NC=CC8=C7)=C6)CC5)C4)C=CC=C3C2=O)C(=O)N1	C67H69ClN10O11S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-D7MXYV	SCHEMBL23276107	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[5-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]pent-4-ynyl]piperidin-4-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCN(CCCC#CC6=CC=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C63H65ClN10O10S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-8AXJCX	SCHEMBL23276086	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[6-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]hex-5-ynyl]piperidin-4-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCN(CCCCC#CC6=CC=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C64H67ClN10O10S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-OYFPPT	SCHEMBL23276016	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[7-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]hept-6-ynyl]piperidin-4-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCN(CCCCCC#CC6=CC=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C65H69ClN10O10S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-QO7KY5	SCHEMBL23276547	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[8-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oct-7-ynyl]piperidin-4-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCN(CCCCCCC#CC6=CC=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C66H71ClN10O10S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-ZZB1OQ	WO2021078301A1_SIAIS292034	.	C=C(NS(=O)(=O)C1=CC([N+](=O)[O-])=C(NCC2CCN(CCCCCCCC#CC3=CC=CC4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)C=C1)C1=CC=C(N2CCN(CC3=C(C4=CC=C(Cl)C=C4)CC(C)(C)CC3)CC2)C=C1OC1=CN=C2NC=CC2=C1	C68H75ClN10O9S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-1XYWYB	SCHEMBL23275977	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[6-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]hex-5-ynyl]piperidin-3-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCCN(CCCCC#CC6=CC=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C64H67ClN10O10S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-WPU4BR	SCHEMBL23276678	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[7-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]hept-6-ynyl]piperidin-3-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCCN(CCCCCC#CC6=CC=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C65H69ClN10O10S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-TWTW05	SCHEMBL23276141	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[8-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oct-7-ynyl]piperidin-3-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCCN(CCCCCCC#CC6=CC=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C66H71ClN10O10S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-O9CAXJ	SCHEMBL23276318	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[9-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]non-8-ynyl]piperidin-3-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCCN(CCCCCCCC#CC6=CC=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C67H73ClN10O10S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-XMFJBQ	SCHEMBL23276309	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[6-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]hexyl]triazol-4-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5=CN(CCCCCCNC6=CC=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7=O)N=N5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C61H64ClN13O10S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-UR74NE	SCHEMBL23276769	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[5-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]pent-4-ynyl]triazol-4-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5=CN(CCCC#CC6=CC=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)N=N5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C60H59ClN12O9S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-2HGZKO	WO2021078301A1_SIAIS292042	.	C=C1C2=C(CN1C1CCC(=O)NC1=O)C(C#CCCCCN1C=C(CNC3=C([N+](=O)[O-])C=C(S(=O)(=O)NC(=O)C4=CC=C(N5CCN(CC6=C(C7=CC=C(Cl)C=C7)CC(C)(C)CC6)CC5)C=C4OC4=CN=C5NC=CC5=C4)C=C3)N=N1)=CC=C2	C62H63ClN12O8S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-BNOHRQ	SCHEMBL23276542	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[7-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]hept-6-ynyl]triazol-4-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5=CN(CCCCCC#CC6=CC=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)N=N5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C62H63ClN12O9S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-GHX71D	WO2021078301A1_SIAIS292044	.	CC1(C)CCC(CN2CCN(C3=CC=C(C(O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5=CN(CCCCCCC#CC6=CC=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)N=N5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C63H67ClN12O9S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-926WKD	SCHEMBL23276561	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[9-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]non-8-ynyl]triazol-4-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5=CN(CCCCCCCC#CC6=CC=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)N=N5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C64H67ClN12O9S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-E4AILE	WO2021078301A1_SIAIS292113	.	CC(CCNCCCC#CC1=CC2=C(C=C1)C(=O)N(C1CCC(=O)NC1=O)C2)CNC1=C([N+](=O)[O-])C=C(S(=O)(=O)NC(=O)C2=CC=C(N3CCN(CC4=C(C5=CC=C(Cl)C=C5)CC(C)(C)CC4)CC3)C=C2OC2=CN=C3NC=CC3=C2)C=C1	C62H67ClN10O9S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-G0GWNI	SCHEMBL23276282	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[6-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]hex-5-ynyl]piperidin-4-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCN(CCCCC#CC6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)CC5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C64H69ClN10O9S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-W237CE	SCHEMBL23276706	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[5-[2-(2,6-dioxopiperidin-3-yl)-3-oxo-1H-isoindol-4-yl]pent-4-ynyl]piperidin-4-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCN(CCCC#CC6=CC=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7)CC5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C63H67ClN10O9S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-L97W0I	SCHEMBL23276007	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[6-[2-(2,6-dioxopiperidin-3-yl)-3-oxo-1H-isoindol-4-yl]hex-5-ynyl]piperidin-4-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCN(CCCCC#CC6=CC=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7)CC5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C64H69ClN10O9S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-ART1I0	SCHEMBL23276078	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[[1-[5-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]pent-4-ynyl]triazol-4-yl]methyl]piperidin-4-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCN(CC6=CN(CCCC#CC7=CC=CC8=C7CN(C7CCC(=O)NC7=O)C8=O)N=N6)CC5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C66H70ClN13O9S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-GQ9YGE	SCHEMBL23276035	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[1-[5-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]pent-4-ynyl]piperidin-4-yl]piperidin-4-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCN(C6CCN(CCCC#CC7=CC=CC8=C7CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C68H76ClN11O9S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-GOMF9G	WO2021078301A1_SIAIS346015	.	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCN(C6CCN(CCCCC#CC7=CC=CC8=C7CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)C=C4)C(OC4=CN=C5NCCC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C69H80ClN11O9S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-2Y55R2	SCHEMBL23276388	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[1-[7-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]hept-6-ynyl]piperidin-4-yl]piperidin-4-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCN(C6CCN(CCCCCC#CC7=CC=CC8=C7CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C70H80ClN11O9S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-4DO8TC	SCHEMBL23276361	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[1-[8-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]oct-7-ynyl]piperidin-4-yl]piperidin-4-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCN(C6CCN(CCCCCCC#CC7=CC=CC8=C7CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C71H82ClN11O9S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-10A7QG	SCHEMBL23275936	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[1-[9-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]non-8-ynyl]piperidin-4-yl]piperidin-4-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCN(C6CCN(CCCCCCCC#CC7=CC=CC8=C7CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C72H84ClN11O9S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-M43WNR	WO2021078301A1_SIAIS361001	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCN3CCC(CNC4=C([N+](=O)[O-])C=C(S(=O)(=O)NC(=O)C5=CC=C(N6CCN(CC7=C(C8=CC=C(Cl)C=C8)CC(C)(C)CC7)CC6)C=C5OC5=CN=C6NC=CC6=C5)C=C4)CC3)C(C)(C)C)C=C2)SCN1	C72H89ClN12O10S2	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-SMLE4C	SCHEMBL23276478	(2S,4R)-1-[(2S)-2-[6-[4-[[4-[[4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzoyl]sulfamoyl]-2-nitroanilino]methyl]piperidin-1-yl]hexanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL23276480	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCN3CCC(CNC4=C([N+](=O)[O-])C=C(S(=O)(=O)NC(=O)C5=CC=C(N6CCN(CC7=C(C8=CC=C(Cl)C=C8)CC(C)(C)CC7)CC6)C=C5OC5=CN=C6NC=CC6=C5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C73H89ClN12O10S2	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-63G6KF	SCHEMBL23276456	(2S,4R)-1-[(2S)-2-[7-[4-[[4-[[4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzoyl]sulfamoyl]-2-nitroanilino]methyl]piperidin-1-yl]heptanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL23276458	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCN3CCC(CNC4=C([N+](=O)[O-])C=C(S(=O)(=O)NC(=O)C5=CC=C(N6CCN(CC7=C(C8=CC=C(Cl)C=C8)CC(C)(C)CC7)CC6)C=C5OC5=CN=C6NC=CC6=C5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C74H91ClN12O10S2	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-2F0247	WO2021078301A1_SIAIS361006	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCN3CCC(CNC4=C([N+](=O)[O-])C=C(S(=O)(=O)NC(=O)C5=CC=C(N6CCN(CC7=C(C8=CC=C(Cl)C=C8)CC(C)(C)CC7)CC6)C=C5OC5=CNC6NC=CC6=C5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C75H95ClN12O10S2	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-2Q54GE	SCHEMBL23276674	(2S,4R)-1-[(2S)-2-[9-[4-[[4-[[4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzoyl]sulfamoyl]-2-nitroanilino]methyl]piperidin-1-yl]nonanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL23276676	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCCN3CCC(CNC4=C([N+](=O)[O-])C=C(S(=O)(=O)NC(=O)C5=CC=C(N6CCN(CC7=C(C8=CC=C(Cl)C=C8)CC(C)(C)CC7)CC6)C=C5OC5=CN=C6NC=CC6=C5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C76H95ClN12O10S2	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-94W7AR	SCHEMBL23276519	(2S,4R)-1-[(2S)-2-[10-[4-[[4-[[4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzoyl]sulfamoyl]-2-nitroanilino]methyl]piperidin-1-yl]decanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL23276522	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCCCN3CCC(CNC4=C([N+](=O)[O-])C=C(S(=O)(=O)NC(=O)C5=CC=C(N6CCN(CC7=C(C8=CC=C(Cl)C=C8)CC(C)(C)CC7)CC6)C=C5OC5=CN=C6NC=CC6=C5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C77H97ClN12O10S2	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-WI47A7	SCHEMBL28555117	(2S,4R)-1-[(2S)-2-[11-[4-[[4-[[4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzoyl]sulfamoyl]-2-nitroanilino]methyl]piperidin-1-yl]undecanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCCCCN3CCC(CNC4=C([N+](=O)[O-])C=C(S(=O)(=O)NC(=O)C5=CC=C(N6CCN(CC7=C(C8=CC=C(Cl)C=C8)CC(C)(C)CC7)CC6)C=C5OC5=CN=C6NC=CC6=C5)C=C4)CC3)C(C)(C)C)C=C2)SC=N1	C78H99ClN12O10S2	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-5K3WAM	SCHEMBL23276664	(2S,4R)-1-[(2S)-2-[5-[3-[[4-[[4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzoyl]sulfamoyl]-2-nitroanilino]methyl]piperidin-1-yl]pentanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL23276668	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCN3CCCC(CNC4=C([N+](=O)[O-])C=C(S(=O)(=O)NC(=O)C5=CC=C(N6CCN(CC7=C(C8=CC=C(Cl)C=C8)CC(C)(C)CC7)CC6)C=C5OC5=CN=C6NC=CC6=C5)C=C4)C3)C(C)(C)C)C=C2)SC=N1	C72H87ClN12O10S2	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-RMKT61	WO2021078301A1_SIAIS361011	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](C)CN3C(=O)[C@@H](NC(=O)CCCCCN3CCCC(CNC4=C([N+](=O)[O-])C=C(S(=O)(=O)NC(O)C5=CC=C(N6CCN(CC7=C(C8=CC=C(Cl)C=C8)CC(C)(C)CC7)CC6)C=C5OC5=CN=C6NC=CC6=C5)C=C4)C3)C(C)(C)C)C=C2)SC=N1	C74H93ClN12O9S2	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-VYXCRJ	SCHEMBL23276725	(2S,4R)-1-[(2S)-2-[7-[3-[[4-[[4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzoyl]sulfamoyl]-2-nitroanilino]methyl]piperidin-1-yl]heptanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL23276729	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCN3CCCC(CNC4=C([N+](=O)[O-])C=C(S(=O)(=O)NC(=O)C5=CC=C(N6CCN(CC7=C(C8=CC=C(Cl)C=C8)CC(C)(C)CC7)CC6)C=C5OC5=CN=C6NC=CC6=C5)C=C4)C3)C(C)(C)C)C=C2)SC=N1	C74H91ClN12O10S2	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-E59IKG	SCHEMBL23276400	(2S,4R)-1-[(2S)-2-[8-[3-[[4-[[4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzoyl]sulfamoyl]-2-nitroanilino]methyl]piperidin-1-yl]octanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL23276404	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCN3CCCC(CNC4=C([N+](=O)[O-])C=C(S(=O)(=O)NC(=O)C5=CC=C(N6CCN(CC7=C(C8=CC=C(Cl)C=C8)CC(C)(C)CC7)CC6)C=C5OC5=CN=C6NC=CC6=C5)C=C4)C3)C(C)(C)C)C=C2)SC=N1	C75H93ClN12O10S2	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-5T9JHF	SCHEMBL23276449	(2S,4R)-1-[(2S)-2-[9-[3-[[4-[[4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzoyl]sulfamoyl]-2-nitroanilino]methyl]piperidin-1-yl]nonanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL23276450	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCCN3CCCC(CNC4=C([N+](=O)[O-])C=C(S(=O)(=O)NC(=O)C5=CC=C(N6CCN(CC7=C(C8=CC=C(Cl)C=C8)CC(C)(C)CC7)CC6)C=C5OC5=CN=C6NC=CC6=C5)C=C4)C3)C(C)(C)C)C=C2)SC=N1	C76H95ClN12O10S2	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-PGBDJS	SCHEMBL23276828	(2S,4R)-1-[(2S)-2-[10-[3-[[4-[[4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzoyl]sulfamoyl]-2-nitroanilino]methyl]piperidin-1-yl]decanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL23276832	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCCCN3CCCC(CNC4=C([N+](=O)[O-])C=C(S(=O)(=O)NC(=O)C5=CC=C(N6CCN(CC7=C(C8=CC=C(Cl)C=C8)CC(C)(C)CC7)CC6)C=C5OC5=CN=C6NC=CC6=C5)C=C4)C3)C(C)(C)C)C=C2)SC=N1	C77H97ClN12O10S2	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-08UP96	SCHEMBL28560481	(2S,4R)-1-[(2S)-2-[11-[3-[[4-[[4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzoyl]sulfamoyl]-2-nitroanilino]methyl]piperidin-1-yl]undecanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCCCCN3CCCC(CNC4=C([N+](=O)[O-])C=C(S(=O)(=O)NC(=O)C5=CC=C(N6CCN(CC7=C(C8=CC=C(Cl)C=C8)CC(C)(C)CC7)CC6)C=C5OC5=CN=C6NC=CC6=C5)C=C4)C3)C(C)(C)C)C=C2)SC=N1	C78H99ClN12O10S2	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-ZUOE7X	SCHEMBL23276551	(2S,4R)-1-[(2S)-2-[5-[4-[4-[[4-[[4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzoyl]sulfamoyl]-2-nitroanilino]methyl]piperidin-1-yl]piperidin-1-yl]pentanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCN3CCC(N4CCC(CNC5=C([N+](=O)[O-])C=C(S(=O)(=O)NC(=O)C6=CC=C(N7CCN(CC8=C(C9=CC=C(Cl)C=C9)CC(C)(C)CC8)CC7)C=C6OC6=CN=C7NC=CC7=C6)C=C5)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C77H96ClN13O10S2	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-W7U1VE	SCHEMBL23276704	(2S,4R)-1-[(2S)-2-[6-[4-[4-[[4-[[4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzoyl]sulfamoyl]-2-nitroanilino]methyl]piperidin-1-yl]piperidin-1-yl]hexanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCN3CCC(N4CCC(CNC5=C([N+](=O)[O-])C=C(S(=O)(=O)NC(=O)C6=CC=C(N7CCN(CC8=C(C9=CC=C(Cl)C=C9)CC(C)(C)CC8)CC7)C=C6OC6=CN=C7NC=CC7=C6)C=C5)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C78H98ClN13O10S2	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-D36OU6	SCHEMBL23276517	(2S,4R)-1-[(2S)-2-[7-[4-[4-[[4-[[4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzoyl]sulfamoyl]-2-nitroanilino]methyl]piperidin-1-yl]piperidin-1-yl]heptanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCN3CCC(N4CCC(CNC5=C([N+](=O)[O-])C=C(S(=O)(=O)NC(=O)C6=CC=C(N7CCN(CC8=C(C9=CC=C(Cl)C=C9)CC(C)(C)CC8)CC7)C=C6OC6=CN=C7NC=CC7=C6)C=C5)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C79H100ClN13O10S2	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-VA33XR	SCHEMBL28553844	(2S,4R)-1-[(2S)-2-[8-[4-[4-[[4-[[4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzoyl]sulfamoyl]-2-nitroanilino]methyl]piperidin-1-yl]piperidin-1-yl]octanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCN3CCC(N4CCC(CNC5=C([N+](=O)[O-])C=C(S(=O)(=O)NC(=O)C6=CC=C(N7CCN(CC8=C(C9=CC=C(Cl)C=C9)CC(C)(C)CC8)CC7)C=C6OC6=CN=C7NC=CC7=C6)C=C5)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C80H102ClN13O10S2	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-TX1SMP	WO2021078301A1_SIAIS361022	.	C/C=C(\C=C/CCNC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](NC(=O)CCCCCCCCN1CCC(N2CCC(CNC3=C([N+](=O)[O-])C=C(S(=O)(=O)NC(O)C4=CC=C(N5CCN(CC6=C(C7=CC=C(Cl)C=C7)CC(C)(C)CC6)CC5)C=C4OC4=CN=C5NC=CC5=C4)C=C3)CC2)CC1)C(C)(C)C)C1=C(C)N=CS1	C81H110ClN13O10S2	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-X5VYLQ	WO2021078301A1_SIAIS361023	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(O)[C@@H](NC(=O)CCCCCCCCCN3CCC(N4CCC(CNC5=C([N+](=O)[O-])C=C(S(=O)(=O)NC(=O)C6=CC=C(N7CCN(CC8=C(C9=CC=C(Cl)C=C9)CC(C)(C)CC8)CC7)C=C6OC6=CN=C7NC=CC7=C6)C=C5)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C82H108ClN13O10S2	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-JENVEN	WO2021078301A1_SIAIS361024	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCCCCN3CCC(N4CCC(CNC5=C([N+](=O)[O-])C=C(S(=O)(=O)NC(=O)C6=CC=C(N7CCN(CC8=C(C9=CC=C(Cl)C=C9)CC(C)(C)CC8)CC7)C=C6OC6=CN=C7NC=CC7=C6)C=C5)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C83H108ClN13O10S2	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-E0O87B	SCHEMBL23276756	4-[4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[(2R)-4-[4-[5-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]pent-4-ynyl]piperazin-1-yl]-1-phenylsulfanylbutan-2-yl]amino]-3-(trifluoromethylsulfonyl)phenyl]sulfonylbenzamide	CC1(C)CCC(C2=CC=C(Cl)C=C2)=C(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC=C(N[C@H](CCN5CCN(CCCC#CC6=CC=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)CC5)CSC5=CC=CC=C5)C(S(=O)(=O)C(F)(F)F)=C4)C=C3)CC2)C1	C65H72ClF3N8O8S3	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-EJJSHO	SCHEMBL23276619	4-[4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[(2R)-4-[4-[6-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]hex-5-ynyl]piperazin-1-yl]-1-phenylsulfanylbutan-2-yl]amino]-3-(trifluoromethylsulfonyl)phenyl]sulfonylbenzamide	CC1(C)CCC(C2=CC=C(Cl)C=C2)=C(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC=C(N[C@H](CCN5CCN(CCCCC#CC6=CC=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)CC5)CSC5=CC=CC=C5)C(S(=O)(=O)C(F)(F)F)=C4)C=C3)CC2)C1	C66H74ClF3N8O8S3	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-4E0ESJ	SCHEMBL23276835	4-[4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[(2R)-4-[4-[7-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]hept-6-ynyl]piperazin-1-yl]-1-phenylsulfanylbutan-2-yl]amino]-3-(trifluoromethylsulfonyl)phenyl]sulfonylbenzamide; SCHEMBL23276841	CC1(C)CCC(C2=CC=C(Cl)C=C2)=C(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC=C(N[C@H](CCN5CCN(CCCCCC#CC6=CC=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)CC5)CSC5=CC=CC=C5)C(S(=O)(=O)C(F)(F)F)=C4)C=C3)CC2)C1	C67H76ClF3N8O8S3	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-AZ6ES4	SCHEMBL23276433	4-[4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[(2R)-4-[4-[8-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]oct-7-ynyl]piperazin-1-yl]-1-phenylsulfanylbutan-2-yl]amino]-3-(trifluoromethylsulfonyl)phenyl]sulfonylbenzamide; SCHEMBL23276436	CC1(C)CCC(C2=CC=C(Cl)C=C2)=C(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC=C(N[C@H](CCN5CCN(CCCCCCC#CC6=CC=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)CC5)CSC5=CC=CC=C5)C(S(=O)(=O)C(F)(F)F)=C4)C=C3)CC2)C1	C68H78ClF3N8O8S3	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-836LHW	SCHEMBL23276239	4-[4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[(2R)-4-[4-[9-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]non-8-ynyl]piperazin-1-yl]-1-phenylsulfanylbutan-2-yl]amino]-3-(trifluoromethylsulfonyl)phenyl]sulfonylbenzamide; SCHEMBL23276241	CC1(C)CCC(C2=CC=C(Cl)C=C2)=C(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC=C(N[C@H](CCN5CCN(CCCCCCCC#CC6=CC=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)CC5)CSC5=CC=CC=C5)C(S(=O)(=O)C(F)(F)F)=C4)C=C3)CC2)C1	C69H80ClF3N8O8S3	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-LL0QKK	WO2021078301A1_SIAIS361048	4-[4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[(2R)-4-[4-[5-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]pent-4-ynyl]piperazin-1-yl]-1-phenylsulfanylbutan-2-yl]amino]-3-(trifluoromethylsulfonyl)phenyl]sulfonylbenzamide	CC1(C)CCC(C2=CC=C(Cl)C=C2)=C(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC=C(N[C@H](CCN5CCN(CCCC#CC6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)CC5)CSC5=CC=CC=C5)C(S(=O)(=O)C(F)(F)F)=C4)C=C3)CC2)C1	C65H72ClF3N8O8S3	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-12TDLD	SCHEMBL23276713	4-[4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[(2R)-4-[4-[6-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]hex-5-ynyl]piperazin-1-yl]-1-phenylsulfanylbutan-2-yl]amino]-3-(trifluoromethylsulfonyl)phenyl]sulfonylbenzamide	CC1(C)CCC(C2=CC=C(Cl)C=C2)=C(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC=C(N[C@H](CCN5CCN(CCCCC#CC6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)CC5)CSC5=CC=CC=C5)C(S(=O)(=O)C(F)(F)F)=C4)C=C3)CC2)C1	C66H74ClF3N8O8S3	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-VTZ41U	SCHEMBL23276585	(2S,4R)-1-[(2S)-2-[10-[4-[4-[[4-[[4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzoyl]sulfamoyl]-2-nitroanilino]methyl]piperidin-1-yl]piperidin-1-yl]decylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NCCCCCCCCCCN3CCC(N4CCC(CNC5=C([N+](=O)[O-])C=C(S(=O)(=O)NC(=O)C6=CC=C(N7CCN(CC8=C(C9=CC=C(Cl)C=C9)CC(C)(C)CC8)CC7)C=C6OC6=CN=C7NC=CC7=C6)C=C5)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C82H108ClN13O9S2	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-6WKT8F	WO2021078301A1_SIAIS363008	.	CC1=C(C2=CC=C(CNC(=O)C3C[C@@H](O)CN3C(=O)[C@@H](NCCCCCCCCCN3CCC(N4CCC(CNC5=C([N+](=O)[O-])C=C(S(=O)(=O)NC(=O)C6=CC=C(N7CCN(CC8=C(C9=CC=C(Cl)C=C9)CC(C)(C)CC8)CC7)C=C6OC6=CN=C7NC=CC7=C6)C=C5)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C81H106ClN13O9S2	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-32JLQS	WO2021078301A1_SIAIS363009	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(NCCOCCOCCN3CCC(N4CCC(CNC5=C([N+](=O)[O-])C=C(S(=O)(=O)NC(=O)C6=CC=C(N7CCN(CC8=C(C9=CC=C(Cl)C=C9)CC(C)(C)CC8)CC7)C=C6OC6=CN=C7NC=CC7=C6)C=C5)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C78H100ClN13O11S2	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-G3Z9AX	SCHEMBL23277029	4-[4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[(2R)-4-[4-[3-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]prop-2-ynyl]piperazin-1-yl]-1-phenylsulfanylbutan-2-yl]amino]-3-(trifluoromethylsulfonyl)phenyl]sulfonylbenzamide	CC1(C)CCC(C2=CC=C(Cl)C=C2)=C(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC=C(N[C@H](CCN5CCN(CC#CC6=CC=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)CC5)CSC5=CC=CC=C5)C(S(=O)(=O)C(F)(F)F)=C4)C=C3)CC2)C1	C63H68ClF3N8O8S3	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-TE83GD	SCHEMBL23275903	4-[4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[(2R)-4-[4-[3-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]sulfanyl]propyl]piperazin-1-yl]-1-phenylsulfanylbutan-2-yl]amino]-3-(trifluoromethylsulfonyl)phenyl]sulfonylbenzamide	CC1(C)CCC(C2=CC=C(Cl)C=C2)=C(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC=C(N[C@H](CCN5CCN(CCCSC6=CC=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)CC5)CSC5=CC=CC=C5)C(S(=O)(=O)C(F)(F)F)=C4)C=C3)CC2)C1	C63H72ClF3N8O8S4	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-53GILF	SCHEMBL23275957	4-[4-[[2-(4-chlorophenyl)-5,5-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[(2R)-4-[4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]sulfanyl]butyl]piperazin-1-yl]-1-phenylsulfanylbutan-2-yl]amino]-3-(trifluoromethylsulfonyl)phenyl]sulfonylbenzamide; SCHEMBL23275959	CC1(C)CCC(C2=CC=C(Cl)C=C2)=C(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC=C(N[C@H](CCN5CCN(CCCCSC6=CC=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)CC5)CSC5=CC=CC=C5)C(S(=O)(=O)C(F)(F)F)=C4)C=C3)CC2)C1	C64H74ClF3N8O8S4	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-QMG05B	WO2021078301A1_SIAIS363023	.	CC1(C)CCC(C2=CC=C(Cl)C=C2)=C(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC=C(N[C@H](CCN5CCN(CCCCCSC6=CC=CC7=C6CN(C6CCC(=O)NC6=O)C7O)CC5)CSC5=CC=CC=C5)C(S(=O)(=O)C(F)(F)F)=C4)C=C3)CC2)C1	C65H78ClF3N8O8S4	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-1UZVML	SCHEMBL23276848	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[1-[3-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]sulfanyl]propyl]piperidin-4-yl]piperidin-4-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCN(C6CCN(CCCSC7=CC=CC8=C7CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C66H76ClN11O9S2	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-UJL2DY	SCHEMBL23276814	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[1-[4-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]sulfanyl]butyl]piperidin-4-yl]piperidin-4-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCN(C6CCN(CCCCSC7=CC=CC8=C7CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C67H78ClN11O9S2	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-D71ELO	SCHEMBL23276075	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[1-[5-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]sulfanyl]pentyl]piperidin-4-yl]piperidin-4-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCN(C6CCN(CCCCCSC7=CC=CC8=C7CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C68H80ClN11O9S2	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-78DO0N	WO2021078301A1_SIAIS363046	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NCCCCCCN3CCN(CCC(CSC4=CC=CC=C4)NC4=CC=C(S(=O)(=O)NC(=O)C5=CC=C(N6CCN(CC7=C(C8=CC=C(Cl)C=C8)CCC(C)(C)C7)CC6)C=C5)C=C4S(=O)(=O)C(F)(F)F)CC3)C(C)(C)C)C=C2)SC=N1	C75H96ClF3N10O8S4	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-3DNV9I	WO2021078301A1_SIAIS363047	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NCCCCCCN3CCC(N4CCC(CNC5=C([N+](=O)[O-])C=C(S(=O)(=O)NC(=O)C6=CC=C(N7CCN(CC8=C(C9=CC=C(Cl)C=C9)CC(C)(C)CC8)CC7)C=C6OC6=CN=C7NC=CC7=C6)C=C5)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C78H100ClN13O9S2	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-HZ5SD6	WO2021078301A1_SIAIS363048	.	CC1=C(C2=CC=C(CNC(=O)C3C[C@@H](O)CN3C(=O)[C@@H](NCCCCCCCN3CCC(N4CCC(CNC5=C([N+](=O)[O-])C=C(S(=O)(=O)NC(=O)C6=CC=C(N7CCN(CC8=C(C9=CC=C(Cl)C=C9)CC(C)(C)CC8)CC7)C=C6OC6=CN=C7NC=CC7=C6)C=C5)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C79H102ClN13O9S2	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-YP99DY	SCHEMBL23276581	(2S,4R)-1-[(2S)-2-[8-[4-[4-[[4-[[4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzoyl]sulfamoyl]-2-nitroanilino]methyl]piperidin-1-yl]piperidin-1-yl]octylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NCCCCCCCCN3CCC(N4CCC(CNC5=C([N+](=O)[O-])C=C(S(=O)(=O)NC(=O)C6=CC=C(N7CCN(CC8=C(C9=CC=C(Cl)C=C9)CC(C)(C)CC8)CC7)C=C6OC6=CN=C7NC=CC7=C6)C=C5)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C80H104ClN13O9S2	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-URL0CU	SCHEMBL28560249	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[1-[3-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]propyl]piperidin-4-yl]piperidin-4-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCN(C6CCN(CCCNC7=CC=CC8=C7C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C66H75ClN12O10S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-S11UYX	SCHEMBL28549274	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[1-[5-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]pentyl]piperidin-4-yl]piperidin-4-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCN(C6CCN(CCCCCNC7=CC=CC8=C7C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C68H79ClN12O10S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-SXTM31	SCHEMBL28550052	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[1-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]butyl]piperidin-4-yl]piperidin-4-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCN(C6CCN(CCCCC7=CC=CC8=C7CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C67H78ClN11O9S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-TDBGSM	WO2021078301A1_SIAIS364019	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NCCCCCCCN3CCN(CC[C@H](CSC4=CC=CC=C4)NC4=CC=C(S(=O)(=O)NC(O)C5=CC=C(N6CCN(CC7=C(C8=CC=C(Cl)C=C8)CCC(C)(C)C7)CC6)C=C5)C=C4S(=O)(=O)C(F)(F)F)CC3)C(C)C)C=C2)SC=N1	C75H98ClF3N10O8S4	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-PXJ3JN	WO2021078301A1_SIAIS364020	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NCCOCCOCCOCCN3CCC(N4CCC(CNC5=C([N+](=O)[O-])C=C(S(=O)(=O)NC(O)C6=CC=C(N7CCN(CC8=C(C9=CC=C(Cl)C=C9)CC(C)(C)CC8)CC7)C=C6OC6=CN=C7NC=CC7=C6)C=C5)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C80H106ClN13O12S2	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-11FBF6	WO2021078301A1_SIAIS364021	.	CC1=C(C2=CC=C(CNC(=O)C3C[C@@H](O)CN3C(=O)[C@@H](NCCOCCOCCOCCOCCN3CCC(N4CCC(CNC5=C([N+](=O)[O-])C=C(S(=O)(=O)NC(=O)C6=CC=C(N7CCN(CC8=C(C9=CC=C(Cl)C=C9)CC(C)(C)CC8)CC7)C=C6OC6=CN=C7NC=CC7=C6)C=C5)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C82H108ClN13O13S2	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-QDWTHY	WO2021078301A1_SIAIS364022	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NCCOCCOCCOCCOCCOCCN3CCC(N4CCC(CNC5=C([N+](=O)[O-])C=C(S(=O)(=O)NC(=O)C6=CC=C(N7CCN(CC8=C(C9=CC=C(Cl)C=C9)CC(C)(C)CC8)CC7)C=C6OC6=CN=C7NC=CC7=C6)C=C5)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C84H112ClN13O14S2	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-TG0XG6	SCHEMBL28552327	4-[4-[[2-(4-chlorophenyl)-4,4-dimethylcyclohexen-1-yl]methyl]piperazin-1-yl]-N-[4-[[1-[1-[5-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]pent-4-ynoyl]piperidin-4-yl]piperidin-4-yl]methylamino]-3-nitrophenyl]sulfonyl-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzamide	CC1(C)CCC(CN2CCN(C3=CC=C(C(=O)NS(=O)(=O)C4=CC([N+](=O)[O-])=C(NCC5CCN(C6CCN(C(=O)CCC#CC7=CC=CC8=C7CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)C=C4)C(OC4=CN=C5NC=CC5=C4)=C3)CC2)=C(C2=CC=C(Cl)C=C2)C1	C68H74ClN11O10S	BCL-2;MCL-1	P10415/Q07820	CRBN	WO-2021078301-A1
TPD-RR8KXQ	SCHEMBL23660845	3-[4-[4-[5-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenoxy]pentyl]piperazin-1-yl]-8-oxo-6H-[1,3]dioxolo[4,5-e]isoindol-7-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C2=O)C2=C(OCO2)C(N2CCN(CCCCCOC4=CC=C([C@@H]5C6=CC=C(O)C=C6CC[C@@H]5C5=CC=CC=C5)C=C4)CC2)=C3)C(=O)N1	C45H48N4O7	ERα	P03372	CRBN	WO-2021143822-A1
TPD-U31E9Q	SCHEMBL23660909	3-[4-[4-[[1-[3,5-difluoro-4-[(1R,3R)-2-(2-fluoro-2-methylpropyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-8-oxo-6H-[1,3]dioxolo[4,5-e]isoindol-7-yl]piperidine-2,6-dione	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(N3CCC(CN4CCN(C5=CC6=C(C(=O)N(C7CCC(=O)NC7=O)C6)C6=C5OCO6)CC4)CC3)C=C2F)N1CC(C)(C)F	C46H52F3N7O5	ERα	P03372	CRBN	WO-2021143822-A1
TPD-F8U15J	PROTAC ER|A Y537S degrader-1	PROTAC ER; A Y537S degrader-1; 2667598-05-0; orb1982998; SCHEMBL23660868; HY-145071; CS-0343060; 3-[4-[4-[[1-[4-[(1R,2S)-6-hydroxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-8-oxo-6H-[1,3]dioxolo[4,5-e]isoindol-7-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C2=O)C2=C(OCO2)C(N2CCN(CC4CCN(C5=CC=C([C@@H]6C7=C(C=C(O)C=C7)CC[C@@H]6C6=CC=CC=C6)C=C5)CC4)CC2)=C3)C(=O)N1	C46H49N5O6	ERα	P03372	CRBN	WO-2021143822-A1
TPD-Z2NC2O	SCHEMBL23660910	3-[4-[4-[[1-[5-[[2-(4-fluorophenyl)-6-hydroxy-1-benzothiophen-3-yl]oxy]pyridin-2-yl]piperidin-4-yl]methyl]piperazin-1-yl]-8-oxo-6H-[1,3]dioxolo[4,5-e]isoindol-7-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C2=O)C2=C(OCO2)C(N2CCN(CC4CCN(C5=CC=C(OC6=C(C7=CC=C(F)C=C7)SC7=C6C=CC(O)=C7)C=N5)CC4)CC2)=C3)C(=O)N1	C43H41FN6O7S	ERα	P03372	CRBN	WO-2021143822-A1
TPD-IW13MX	SCHEMBL23660842	3-[4-[7-[3,5-difluoro-4-[(1R,3R)-2-(2-fluoro-2-methylpropyl)-3-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indol-1-yl]phenoxy]heptyl]-7-oxo-3,9-dihydro-2H-pyrrolo[3,4-h][1,4]benzoxazin-8-yl]piperidine-2,6-dione	C[C@@H]1CC2=C(NC3=C2C=CC=C3)[C@@H](C2=C(F)C=C(OCCCCCCCN3CCOC4=C3C=CC3=C4CN(C4CCC(=O)NC4=O)C3=O)C=C2F)N1CC(C)(C)F	C44H50F3N5O5	ERα	P03372	CRBN	WO-2021143822-A1
TPD-0XK3PD	CHEMBL5076514	N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-5-[4-[[4-[10-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxydecyl]piperazin-1-yl]methyl]phenyl]-3-[ethyl(oxan-4-yl)amino]-2-methylbenzamide; SCHEMBL24072462; BDBM50582392; PD155640	CCN(C1=CC(C2=CC=C(CN3CCN(CCCCCCCCCCOC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C57H73N7O8	EZH2	Q15910	CRBN	WO-2021238007-A1
TPD-R3RIPH	CHEMBL5085241	N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-5-[4-[[4-[11-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyundecyl]piperazin-1-yl]methyl]phenyl]-3-[ethyl(oxan-4-yl)amino]-2-methylbenzamide; SCHEMBL24072841; BDBM50582393; PD155639	CCN(C1=CC(C2=CC=C(CN3CCN(CCCCCCCCCCCOC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C58H75N7O8	EZH2	Q15910	CRBN	WO-2021238007-A1
TPD-5GQZCR	WO2021238007A1_E12	.	CCN(C1=CC(C2=CC=C(CN3CCN(CCCCCCCCCCCCOC4=C5C(=CC=C4)C(=O)N(C4CCC(=O)NC4=O)C5O)CC3)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C59H79N7O8	EZH2	Q15910	CRBN	WO-2021238007-A1
TPD-O799OH	CHEMBL5085953	N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-5-[4-[[4-[5-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxypentyl]piperazin-1-yl]methyl]phenyl]-3-[ethyl(oxan-4-yl)amino]-2-methylbenzamide; SCHEMBL23342557; BDBM50582387; PD155645	CCN(C1=CC(C2=CC=C(CN3CCN(CCCCCOC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C52H63N7O8	EZH2	Q15910	CRBN	WO-2021238007-A1
TPD-0B86B3	CHEMBL5090885	N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-5-[4-[[4-[6-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyhexyl]piperazin-1-yl]methyl]phenyl]-3-[ethyl(oxan-4-yl)amino]-2-methylbenzamide; SCHEMBL24071945; BDBM50582388; PD155644	CCN(C1=CC(C2=CC=C(CN3CCN(CCCCCCOC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C53H65N7O8	EZH2	Q15910	CRBN	WO-2021238007-A1
TPD-9470CY	PROTAC EZH2 Degrader-1	PROTAC EZH2 Degrader-1; 2641601-67-2; CHEMBL5089835; orb1982793; SCHEMBL23343057; SCHEMBL29943222; EX-A7166; BDBM50582389; BP-42270; DA-77145; MS-31755; HY-147525; H43107; EN300-44827606; N-[(4,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)methyl]-4'-{[4-(7-{[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]oxy}heptyl)piperazin-1-yl]methyl}-5-[ethyl(oxan-4-yl)amino]-4-methyl-[1,1'-biphenyl]-3-carboxamide	CCN(C1=CC(C2=CC=C(CN3CCN(CCCCCCCOC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C54H67N7O8	EZH2	Q15910	CRBN	WO-2021238007-A1
TPD-OS9OCU	WO2021238007A1_E8	.	C=C1C2=CC=CC(OCCCCCCCCN3CCN(CC4=CC=C(C5=CC(C(=O)NCC6=C(C)C=C(C)NC6=O)=C(C)C(N(CC)C6CCOCC6)=C5)C=C4)CC3)=C2C(=O)N1C1CCC(=O)NC1=O	C56H71N7O7	EZH2	Q15910	CRBN	WO-2021238007-A1
TPD-ICN6BG	CHEMBL5073227	N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-5-[4-[[4-[9-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxynonyl]piperazin-1-yl]methyl]phenyl]-3-[ethyl(oxan-4-yl)amino]-2-methylbenzamide; SCHEMBL24071953; BDBM50582391; PD155641	CCN(C1=CC(C2=CC=C(CN3CCN(CCCCCCCCCOC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C56H71N7O8	EZH2	Q15910	CRBN	WO-2021238007-A1
TPD-1VK6C1	CHEMBL5070010	1-[(2S)-butan-2-yl]-N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-6-[6-[4-[10-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxydecyl]piperazin-1-yl]pyridin-3-yl]-3-methylindole-4-carboxamide; SCHEMBL24072792; BDBM50582383; PD155651	CC[C@H](C)N1C=C(C)C2=C1C=C(C1=CC=C(N3CCN(CCCCCCCCCCOC4=CC=CC5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)N=C1)C=C2C(=O)NCC1=C(C)C=C(C)NC1=O	C54H66N8O7	EZH2	Q15910	CRBN	WO-2021238007-A1
TPD-7MKTKO	CHEMBL5090331	1-[(2S)-butan-2-yl]-N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-6-[6-[4-[11-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyundecyl]piperazin-1-yl]pyridin-3-yl]-3-methylindole-4-carboxamide; SCHEMBL24072780; BDBM50582384; PD155649	CC[C@H](C)N1C=C(C)C2=C1C=C(C1=CC=C(N3CCN(CCCCCCCCCCCOC4=CC=CC5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)N=C1)C=C2C(=O)NCC1=C(C)C=C(C)NC1=O	C55H68N8O7	EZH2	Q15910	CRBN	WO-2021238007-A1
TPD-OIKYFZ	CHEMBL5086887	1-[(2S)-butan-2-yl]-N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-6-[6-[4-[12-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxydodecyl]piperazin-1-yl]pyridin-3-yl]-3-methylindole-4-carboxamide; SCHEMBL24072852; BDBM50582385; PD155647	CC[C@H](C)N1C=C(C)C2=C1C=C(C1=CC=C(N3CCN(CCCCCCCCCCCCOC4=CC=CC5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)N=C1)C=C2C(=O)NCC1=C(C)C=C(C)NC1=O	C56H70N8O7	EZH2	Q15910	CRBN	WO-2021238007-A1
TPD-EUFS8A	CHEMBL5076965	1-[(2S)-butan-2-yl]-N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-6-[6-[4-[5-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxypentyl]piperazin-1-yl]pyridin-3-yl]-3-methylindole-4-carboxamide; SCHEMBL24072864; BDBM50582378; PD155661	CC[C@H](C)N1C=C(C)C2=C1C=C(C1=CC=C(N3CCN(CCCCCOC4=CC=CC5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)N=C1)C=C2C(=O)NCC1=C(C)C=C(C)NC1=O	C49H56N8O7	EZH2	Q15910	CRBN	WO-2021238007-A1
TPD-W7NS69	CHEMBL5091654	1-[(2S)-butan-2-yl]-N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-6-[6-[4-[6-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyhexyl]piperazin-1-yl]pyridin-3-yl]-3-methylindole-4-carboxamide; SCHEMBL24072452; BDBM50582379; PD155659	CC[C@H](C)N1C=C(C)C2=C1C=C(C1=CC=C(N3CCN(CCCCCCOC4=CC=CC5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)N=C1)C=C2C(=O)NCC1=C(C)C=C(C)NC1=O	C50H58N8O7	EZH2	Q15910	CRBN	WO-2021238007-A1
TPD-K780NP	WO2021238007A1_G7	.	CC[C@H](C)N1C=C(C)C2C(C(=O)NCC3=C(C)C=C(C)NC3=O)=CC(C3=CC=C(N4CCN(CCCCCCCOC5=CC=CC6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)N=C3)=CC21	C51H62N8O7	EZH2	Q15910	CRBN	WO-2021238007-A1
TPD-GVD626	CHEMBL5088302	1-[(2S)-butan-2-yl]-N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-6-[6-[4-[8-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyoctyl]piperazin-1-yl]pyridin-3-yl]-3-methylindole-4-carboxamide; SCHEMBL24072454; BDBM50582381; PD155655	CC[C@H](C)N1C=C(C)C2=C1C=C(C1=CC=C(N3CCN(CCCCCCCCOC4=CC=CC5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)N=C1)C=C2C(=O)NCC1=C(C)C=C(C)NC1=O	C52H62N8O7	EZH2	Q15910	CRBN	WO-2021238007-A1
TPD-IP4LFE	CHEMBL5085848	1-[(2S)-butan-2-yl]-N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-6-[6-[4-[9-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxynonyl]piperazin-1-yl]pyridin-3-yl]-3-methylindole-4-carboxamide; SCHEMBL24072441; BDBM50582382; PD155653	CC[C@H](C)N1C=C(C)C2=C1C=C(C1=CC=C(N3CCN(CCCCCCCCCOC4=CC=CC5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)N=C1)C=C2C(=O)NCC1=C(C)C=C(C)NC1=O	C53H64N8O7	EZH2	Q15910	CRBN	WO-2021238007-A1
TPD-LDM170	SCHEMBL24071955	N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-5-[4-[[4-[7-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]sulfanylheptyl]piperazin-1-yl]methyl]phenyl]-3-[ethyl(oxan-4-yl)amino]-2-methylbenzamide	CCN(C1=CC(C2=CC=C(CN3CCN(CCCCCCCSC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C54H67N7O7S	EZH2	Q15910	CRBN	WO-2021238007-A1
TPD-YU97FX	SCHEMBL24071958	1-[(2S)-butan-2-yl]-N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-6-[6-[4-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]sulfanylbutyl]piperazin-1-yl]pyridin-3-yl]-3-methylindole-4-carboxamide	CC[C@H](C)N1C=C(C)C2=C1C=C(C1=CC=C(N3CCN(CCCCSC4=CC=CC5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)N=C1)C=C2C(=O)NCC1=C(C)C=C(C)NC1=O	C48H54N8O6S	EZH2	Q15910	CRBN	WO-2021238007-A1
TPD-KMVWK2	SCHEMBL24071959	1-[(2S)-butan-2-yl]-N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-6-[6-[4-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]butanoyl]piperazin-1-yl]pyridin-3-yl]-3-methylindole-4-carboxamide	CC[C@H](C)N1C=C(C)C2=C1C=C(C1=CC=C(N3CCN(C(=O)CCCNC4=CC=CC5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)N=C1)C=C2C(=O)NCC1=C(C)C=C(C)NC1=O	C48H53N9O7	EZH2	Q15910	CRBN	WO-2021238007-A1
TPD-L1UN2R	SCHEMBL24072787	5-[6-[4-[10-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxydecyl]piperazin-1-yl]pyridin-3-yl]-3-[ethyl(oxan-4-yl)amino]-2-methyl-N-[(1-methyl-3-oxo-5,6,7,8-tetrahydro-2H-isoquinolin-4-yl)methyl]benzamide	CCN(C1=CC(C2=CC=C(N3CCN(CCCCCCCCCCOC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)N=C2)=CC(C(=O)NCC2=C3CCCCC3=C(C)NC2=O)=C1C)C1CCOCC1	C58H74N8O8	EZH2	Q15910	CRBN	WO-2021238007-A1
TPD-GX0E8Y	WO2021238007A1_S11	.	CCC(CC)N(CC)C1=CC(C2=CC=C(N3CCN(CCCCCCCCCCCOC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CCC4)CC3)N=C2)=CC(C(=O)NCC2=C3CCCCC3=C(C)NC2=O)=C1C	C59H80N8O7	EZH2	Q15910	CRBN	WO-2021238007-A1
TPD-PZXBPU	SCHEMBL24072463	5-[6-[4-[6-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyhexyl]piperazin-1-yl]pyridin-3-yl]-3-[ethyl(oxan-4-yl)amino]-2-methyl-N-[(1-methyl-3-oxo-5,6,7,8-tetrahydro-2H-isoquinolin-4-yl)methyl]benzamide	CCN(C1=CC(C2=CC=C(N3CCN(CCCCCCOC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)N=C2)=CC(C(=O)NCC2=C3CCCCC3=C(C)NC2=O)=C1C)C1CCOCC1	C54H66N8O8	EZH2	Q15910	CRBN	WO-2021238007-A1
TPD-84QB4V	SCHEMBL24071954	5-[6-[4-[7-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyheptyl]piperazin-1-yl]pyridin-3-yl]-3-[ethyl(oxan-4-yl)amino]-2-methyl-N-[(1-methyl-3-oxo-5,6,7,8-tetrahydro-2H-isoquinolin-4-yl)methyl]benzamide	CCN(C1=CC(C2=CC=C(N3CCN(CCCCCCCOC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)N=C2)=CC(C(=O)NCC2=C3CCCCC3=C(C)NC2=O)=C1C)C1CCOCC1	C55H68N8O8	EZH2	Q15910	CRBN	WO-2021238007-A1
TPD-E5QKNE	SCHEMBL24072851	5-[6-[4-[8-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyoctyl]piperazin-1-yl]pyridin-3-yl]-3-[ethyl(oxan-4-yl)amino]-2-methyl-N-[(1-methyl-3-oxo-5,6,7,8-tetrahydro-2H-isoquinolin-4-yl)methyl]benzamide	CCN(C1=CC(C2=CC=C(N3CCN(CCCCCCCCOC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)N=C2)=CC(C(=O)NCC2=C3CCCCC3=C(C)NC2=O)=C1C)C1CCOCC1	C56H70N8O8	EZH2	Q15910	CRBN	WO-2021238007-A1
TPD-DSFSQJ	SCHEMBL24072796	5-[6-[4-[9-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxynonyl]piperazin-1-yl]pyridin-3-yl]-3-[ethyl(oxan-4-yl)amino]-2-methyl-N-[(1-methyl-3-oxo-5,6,7,8-tetrahydro-2H-isoquinolin-4-yl)methyl]benzamide	CCN(C1=CC(C2=CC=C(N3CCN(CCCCCCCCCOC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)N=C2)=CC(C(=O)NCC2=C3CCCCC3=C(C)NC2=O)=C1C)C1CCOCC1	C57H72N8O8	EZH2	Q15910	CRBN	WO-2021238007-A1
TPD-79W76N	WO2022031772A1_BRD-E2+8305	.	[H][C@@]1(CC(=O)NCCNC(=O)C2=CC=CC(B3OC4=C(O3)C(C(=O)N[C@@H](C(=O)N3C[C@H](O)C[C@H]3C(O)NCC3=CC=C(C5=C(C)N=CS5)C=C3)C(C)(C)C)=CC=C4)=C2)N=C(C2=CC=C(Cl)C=C2)C2=CC(OC)=CC=C2N2C(C)=NN=C21	C58H60BClN10O9S	BRD4	O60885	VHL	WO-2022031772-A1
TPD-5DBAJI	WO2022031772A1_BRD-E20+8305	.	[H][C@@]1(CC(=O)NCC)N=C(C2=CC=C(Cl)C=C2)C2=CC(OCCCCC(=O)NC3=CC(B4OC5=C(O4)C(C(=O)N[C@@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)NCC4=CC=C(C6=C(C)N=CS6)C=C4)C(C)(C)C)=CC=C5)=CC=C3)=CC=C2N2C(C)=NN=C21	C61H64BClN10O9S	BRD4	O60885	VHL	WO-2022031772-A1
TPD-GR6MYA	WO2022031772A1_BRD-E21+8047	.	[H][C@@]1(CC(=O)NCC)N=C(C2=CC=C(Cl)C=C2)C2=CC(OCCNC(=O)C3=CC=CC(B4OC5=CC=CC(C(=O)NCC6=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)=C5O4)=C3)=CC=C2N2C(C)=NN=C21	C51H43BClN9O10	BRD4	O60885	CRBN	WO-2022031772-A1
TPD-C23G09	WO2022031772A1_BRD-E30+8047	.	[H][C@@]1(CC(=O)NCCNC(=O)/C=C/C2=CC(B3OC4=CC=CC(C(=O)NCC5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)=C4O3)=CC=C2)N=C(C2=CC=C(Cl)C=C2)C2=C(C=CC(OC)=C2)N2C(C)=NN=C21	C52H43BClN9O10	BRD4	O60885	CRBN	WO-2022031772-A1
TPD-WMEAEV	WO2022031772A1_BRD-E4+8046	.	[H][C@@]1(CC(=O)NCCCNC(=O)C2=CC=CC(B3OC4=C(C=C(C(=O)NCC5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)C=C4)O3)=C2)N=C(C2=CC=C(Cl)C=C2)C2=CC(OC)=CC=C2N2C(C)=NN=C21	C51H43BClN9O10	BRD4	O60885	CRBN	WO-2022031772-A1
TPD-IHTS06	WO2022031772A1_BRD-E50+8305	.	[H][C@](C)(CC(=O)NCC)C1=NN=C(C)N1C1=C(C(=N)C2=CC=C(Cl)C=C2)C=C(B2OC3=C(O2)C(C(=O)N[C@@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(C4=C(C)N=CS4)C=C2)C(C)(C)C)=CC=C3)C=C1	C51H55BClN9O7S	BRD4	O60885	VHL	WO-2022031772-A1
TPD-O74EFJ	WO2022031772A1_BRD-E72+8047	.	CCNC(=O)C[C@@H]1N=C(C2=CC=C(Cl)C=C2)C2=C(C=CC(C3=CC=CC(B4OC5=CC=CC(C(=O)NCC6=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)=C5O4)=C3)=C2)N2C(C)=NN=C12	C48H38BClN8O8	BRD4	O60885	CRBN	WO-2022031772-A1
TPD-19Y3L9	WO2022031772A1_BRD-E79+8047	.	CCNC(=O)C[C@@H]1N=C(C2=CC=C(Cl)C=C2)C2C=C(OCCCCCCNC(=O)C3=CC=C(B4OC5=CC=CC(C(=O)NCC6=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)=C5O4)C=C3)C=CC2N2C(C)=NN=C12	C55H53BClN9O10	BRD4	O60885	CRBN	WO-2022031772-A1
TPD-LSICRT	WO2022031772A1_BRD-E9+8305	.	[H][C@@]1(CC(=O)NCC2=CC=C(B3OC4=C(O3)C(C(=O)N[C@@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCC3=CC=C(C5=C(C)N=CS5)C=C3)C(C)(C)C)=CC=C4)C=C2)N=C(C2=CC=C(Cl)C=C2)C2=CC(OC)=CC=C2N2C(C)=NN=C21	C56H55BClN9O8S	BRD4	O60885	VHL	WO-2022031772-A1
TPD-0HJLMP	WO2022031772A1_BRD-N10+8049	.	[H][C@@]1(CC(=O)NCCC2=CC=C3OB(C4=CC=CC(C(=O)NCC5=CC=CC6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)=C4)OC3=C2)N=C(C2=CC=C(Cl)C=C2)C2=CC(OC)=CC=C2N2C(C)=NN=C21	C49H40BClN8O9	BRD4	O60885	CRBN	WO-2022031772-A1
TPD-6NXY45	WO2022031772A1_BRD-N2+8049	.	[H][C@@]1(CC(=O)NCCNC(O)C2=C3OB(C4=CC=CC(C(=O)NCC5=CC=CC6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)=C4)OC3=CC=C2)N=C(C2=CC=C(Cl)C=C2)C2=CC(OC)=CC=C2N2C(C)=NN=C21	C50H43BClN9O10	BRD4	O60885	CRBN	WO-2022031772-A1
TPD-Y1AXE0	WO2022031772A1_BRD-N25+8049	.	[H][C@@]1(CC(=O)NCC)N=C(C2=CC=C(Cl)C=C2)C2=CC(OCCNC(=O)C3=CC=CC4=C3OB(C3=CC=CC(C(=O)NCC5=CC=CC6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)=C3)O4)=CC=C2N2C(C)=NN=C21	C51H43BClN9O10	BRD4	O60885	CRBN	WO-2022031772-A1
TPD-Q6IZG9	WO2022031772A1_BRD-N25+8310	.	[H]C1(C2=CC=C(Cl)C=C2)N=C(C2=C(OC(C)C)C=C(OC)C=C2)N(C(=O)N2CCN(CCNC(=O)C3=CC=C(B4OC5=C(O4)C(C(=O)NCCOC4=CC=C6C(=C4)C(C4=CC=C(Cl)C=C4)=N[C@@]([H])(CC(=O)NCC)C4=NN=C(C)N64)=CC=C5)C=C3)C(=O)C2)[C@]1([H])C1=CC=C(Cl)C=C1	C69H65BCl3N11O10	BRD4	O60885	MDM2	WO-2022031772-A1
TPD-GUUN5U	WO2022031772A1_BRD-N67+8048	.	CCNC(=O)C[C@@H]1N=C(C2=CC=C(Cl)C=C2)C2=C(C=CC(C3=CC4=CC5=C(C=C4C=C3)OB(C3=CC=C(C(=O)NC4=CC=CC6=C4C(=O)N(C4CCC(=O)NC4=O)C6=O)C=C3)O5)=C2)N2C(C)=NN=C12	C51H38BClN8O8	BRD4	O60885	CRBN	WO-2022031772-A1
TPD-ZA5SJB	WO2022031772A1_BRD-N8+8049	.	[H][C@@]1(CC(=O)NCCCCCNC(=O)C2=CC=CC3=C2OB(C2=CC=CC(C(=O)NCC4=CC=CC5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)=C2)O3)N=C(C2=CC=C(Cl)C=C2)C2=CC(OC)=CC=C2N2C(C)=NN=C21	C53H47BClN9O10	BRD4	O60885	CRBN	WO-2022031772-A1
TPD-CNGYCK	SCHEMBL26957040	3-[6-[4-[5-[4-(2-hydroxy-6-phenyl-8,9-dihydro-7H-benzo[7]annulen-5-yl)phenoxy]pentyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(N4CCN(CCCCCOC5=CC=C(C6=C(C7=CC=CC=C7)CCCC7=C6C=CC(O)=C7)C=C5)CC4)=C3)C2=O)C(=O)N1	C45H48N4O5	ERα	P03372	CRBN	WO-2022166879-A1
TPD-31VGSA	WO2022166879A1_10	(3S)-3-[6-[4-[[1-[4-(8-methoxy-4-phenyl-2,3-dihydro-1-benzoxepin-5-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	COC1=CC2=C(C=C1)C(C1=CC=C(N3CCC(CN4CCN(C5=CC=C6C(=O)N([C@H]7CCC(=O)NC7=O)CC6=C5)CC4)CC3)C=C1)=C(C1=CC=CC=C1)CCO2	C46H49N5O5	ERα	P03372	CRBN	WO-2022166879-A1
TPD-B46EVC	WO2022166879A1_11	.	CC1=CC=C(C2=C(C3=CC=C(N4CCC(CN5CCN(C6=CC=C7C(=O)N([C@H]8CCC(=O)NC8=O)CC7C6)CC5)CC4)C=C3)C3=C(C=C(O)C=C3)CCC2)C=C1	C47H53N5O4	ERα	P03372	CRBN	WO-2022166879-A1
TPD-5IRJIL	SCHEMBL30724083	5-[4-[4-[[4-[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]phenyl]-6-phenyl-8,9-dihydro-7H-benzo[7]annulene-2-carboxylic acid	O=C1CC[C@H](N2CC3=CC(N4CCN(CC5CCN(C6=CC=C(C7=C(C8=CC=CC=C8)CCCC8=C7C=CC(C(=O)O)=C8)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C47H49N5O5	ERα	P03372	CRBN	WO-2022166879-A1
TPD-I19EB7	WO2022166879A1_13	.	O=C1CC[C@H](N2CC3=CC(N4CCN(CCC5CCN(C6=CC7=C(C=C6)C6=C(CCCC8=CC(C(=O)O)=CC=C86)C6=CC=CC=C67)CC5)CC4)=CC=C3C2=O)C(=O)N1	C48H49N5O5	ERα	P03372	CRBN	WO-2022166879-A1
TPD-70YS1K	SCHEMBL30724021	(3S)-3-[6-[4-[[1-[4-(2-hydroxy-6-phenyl-8,9-dihydro-7H-benzo[7]annulen-5-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CC[C@H](N2CC3=CC(N4CCN(CC5CCN(C6=CC=C(C7=C(C8=CC=CC=C8)CCCC8=C7C=CC(O)=C8)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C46H49N5O4	ERα	P03372	CRBN	WO-2022166879-A1
TPD-QCTHRY	SCHEMBL26957078	3-[6-[4-[[1-[4-[2-hydroxy-6-[6-(trifluoromethyl)pyridin-3-yl]-8,9-dihydro-7H-benzo[7]annulen-5-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=CC(N4CCN(CC5CCN(C6=CC=C(C7=C(C8=CC=C(C(F)(F)F)N=C8)CCCC8=C7C=CC(O)=C8)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C46H47F3N6O4	ERα	P03372	CRBN	WO-2022166879-A1
TPD-7YTJVW	WO2022166879A1_16	.	CC1=NC=C2C(=C1)C1=C(C=CC(N3CCC(CN4CCN(C5=CC=C6C(=O)N([C@H]7CCC(=O)NC7=O)CC6=C5)CC4)CC3)=C1)C1=C2CCCC2=C1C=CC(O)=C2	C46H48N6O4	ERα	P03372	CRBN	WO-2022166879-A1
TPD-GNVYBR	SCHEMBL26957195	(3S)-3-[6-[4-[[1-[4-[6-(6-cyclopropylpyridin-3-yl)-2-hydroxy-8,9-dihydro-7H-benzo[7]annulen-5-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CC[C@H](N2CC3=CC(N4CCN(CC5CCN(C6=CC=C(C7=C(C8=CN=C(C9CC9)C=C8)CCCC8=C7C=CC(O)=C8)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C48H52N6O4	ERα	P03372	CRBN	WO-2022166879-A1
TPD-GE6MI3	WO2022166879A1_18	(3S)-3-[6-[4-[[1-[4-[6-(1,3-dimethylpyrazol-4-yl)-2-hydroxy-8,9-dihydro-7H-benzo[7]annulen-5-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CC1=NN(C)C=C1C1=C(C2=CC=C(N3CCC(CN4CCN(C5=CC=C6C(=O)N([C@H]7CCC(=O)NC7=O)CC6=C5)CC4)CC3)C=C2)C2=C(C=C(O)C=C2)CCC1	C45H51N7O4	ERα	P03372	CRBN	WO-2022166879-A1
TPD-8YB27W	WO2022166879A1_19	(3S)-3-[6-[4-[[1-[4-[6-(6-fluoropyridin-3-yl)-2-hydroxy-8,9-dihydro-7H-benzo[7]annulen-5-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CC[C@H](N2CC3=CC(N4CCN(CC5CCN(C6=CC=C(C7=C(C8=CN=C(F)C=C8)CCCC8=C7C=CC(O)=C8)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C45H47FN6O4	ERα	P03372	CRBN	WO-2022166879-A1
TPD-9IJJV7	SCHEMBL26957039	3-[6-[4-[[1-[4-(2-hydroxy-6-phenyl-8,9-dihydro-7H-benzo[7]annulen-5-yl)phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30723789	O=C1CCC(N2CC3=CC(N4CCN(CC5CCN(C6=CC=C(C7=C(C8=CC=CC=C8)CCCC8=C7C=CC(O)=C8)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C46H49N5O4	ERα	P03372	CRBN	WO-2022166879-A1
TPD-VKA3GJ	WO2022166879A1_20	.	O=C1CC[C@H](N2CC3=CC(N4CCN(CC5CCN(C6=CC7=C(C=C6)C6=C(CCCC8=C6C=CC(O)=C8)C6=CC=NC=C67)CC5)CC4)=CC=C3C2=O)C(=O)N1	C45H46N6O4	ERα	P03372	CRBN	WO-2022166879-A1
TPD-8ORWF9	WO2022166879A1_21	.	O=C1CC[C@H](N2CC3=CC(N4CCN(CC5CCN(C6=CC7=C(C=C6)C6=C(CCCC8=C6C=CC(O)=C8)C6=CN=CC=C67)CC5)CC4)=CC=C3C2=O)C(=O)N1	C45H46N6O4	ERα	P03372	CRBN	WO-2022166879-A1
TPD-RU2770	WO2022166879A1_22	.	CC1=NC(C)=C2C(=C1)C1=C(C=CC(N3CCC(CN4CCN(C5=CC=C6C(=O)N([C@H]7CCC(=O)NC7=O)CC6=C5)CC4)CC3)=C1)C1=C2CCCC2=C1C=CC(O)=C2	C47H50N6O4	ERα	P03372	CRBN	WO-2022166879-A1
TPD-6ZXNZI	WO2022166879A1_23	(3S)-3-[6-[4-[[1-[4-[2-hydroxy-6-[6-(2-hydroxypropan-2-yl)pyridin-3-yl]-8,9-dihydro-7H-benzo[7]annulen-5-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CC(C)(O)C1=NC=C(C2=C(C3=CC=C(N4CCC(CN5CCN(C6=CC=C7C(=O)N([C@H]8CCC(=O)NC8=O)CC7=C6)CC5)CC4)C=C3)C3=C(C=C(O)C=C3)CCC2)C=C1	C48H54N6O5	ERα	P03372	CRBN	WO-2022166879-A1
TPD-DULKUD	SCHEMBL26957246	(3S)-3-[6-[4-[[1-[4-[6-[4-(difluoromethoxy)phenyl]-2-hydroxy-8,9-dihydro-7H-benzo[7]annulen-5-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CC[C@H](N2CC3=CC(N4CCN(CC5CCN(C6=CC=C(C7=C(C8=CC=C(OC(F)F)C=C8)CCCC8=C7C=CC(O)=C8)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C47H49F2N5O5	ERα	P03372	CRBN	WO-2022166879-A1
TPD-AJTWCD	SCHEMBL26957251	(3S)-3-[6-[4-[[1-[4-[2-hydroxy-6-[4-(trifluoromethoxy)phenyl]-8,9-dihydro-7H-benzo[7]annulen-5-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CC[C@H](N2CC3=CC(N4CCN(CC5CCN(C6=CC=C(C7=C(C8=CC=C(OC(F)(F)F)C=C8)CCCC8=C7C=CC(O)=C8)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C47H48F3N5O5	ERα	P03372	CRBN	WO-2022166879-A1
TPD-X3E33C	WO2022166879A1_26	.	O=C1CC[C@H](N2CC3=CC(N4CCN(CC5CCN(C6=CC7=C(C=C6)C6=C(CCCC8=C6C=CC(O)=C8)C6=CC=C(OC8CC8)C=C67)CC5)CC4)=CC=C3C2=O)C(=O)N1	C49H51N5O5	ERα	P03372	CRBN	WO-2022166879-A1
TPD-R0ORL9	WO2022166879A1_3	.	O=C1CCC(N2CC3=C(C=CC(N4CCN(CC5CCN(C6=CC=C(C7=C(C8=CC=C(Cl)C=C8Cl)CCCC8=CC(C(=O)O)=CC=C87)C=C6)CC5)CC4)=C3)C2=O)C(=O)N=N1	C47H46Cl2N6O5	ERα	P03372	CRBN	WO-2022166879-A1
TPD-PR5X4F	SCHEMBL26957132	(3S)-3-[6-[4-[2-[1-[4-(2-hydroxy-6-phenyl-8,9-dihydro-7H-benzo[7]annulen-5-yl)phenyl]piperidin-4-yl]ethyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CC[C@H](N2CC3=CC(N4CCN(CCC5CCN(C6=CC=C(C7=C(C8=CC=CC=C8)CCCC8=C7C=CC(O)=C8)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C47H51N5O4	ERα	P03372	CRBN	WO-2022166879-A1
TPD-Y2KT71	SCHEMBL26957167	(3S)-3-[6-[4-[[1-[4-[2-hydroxy-6-(4-methylphenyl)-8,9-dihydro-7H-benzo[7]annulen-5-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CC1=CC=C(C2=C(C3=CC=C(N4CCC(CN5CCN(C6=CC=C7C(=O)N([C@H]8CCC(=O)NC8=O)CC7=C6)CC5)CC4)C=C3)C3=C(C=C(O)C=C3)CCC2)C=C1	C47H51N5O4	ERα	P03372	CRBN	WO-2022166879-A1
TPD-RZKDC2	WO2022166879A1_6	(3S)-3-[6-[4-[[1-[4-[6-(4-fluorophenyl)-2-hydroxy-8,9-dihydro-7H-benzo[7]annulen-5-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CC[C@H](N2CC3=CC(N4CCN(CC5CCN(C6=CC=C(C7=C(C8=CC=C(F)C=C8)CCCC8=C7C=CC(O)=C8)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C46H48FN5O4	ERα	P03372	CRBN	WO-2022166879-A1
TPD-2T11L1	WO2022166879A1_7	.	COC1=CC2=C(C=C1)C1=C(CCC2)C2=CC=CC=C2C2=C1C=CC(N1CCC(CN3CCN(C4=CC=C5C(=O)N([C@H]6CCC(=O)NC6=O)CC5=C4)CC3)CC1)=C2	C47H49N5O4	ERα	P03372	CRBN	WO-2022166879-A1
TPD-IS022T	WO2022166879A1_8	(3S)-3-[6-[4-[[1-[4-[6-(4-fluorophenyl)-2-methoxy-8,9-dihydro-7H-benzo[7]annulen-5-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	COC1=CC2=C(C=C1)C(C1=CC=C(N3CCC(CN4CCN(C5=CC=C6C(=O)N([C@H]7CCC(=O)NC7=O)CC6=C5)CC4)CC3)C=C1)=C(C1=CC=C(F)C=C1)CCC2	C47H50FN5O4	ERα	P03372	CRBN	WO-2022166879-A1
TPD-RLVYIQ	SCHEMBL26957157	(3S)-3-[6-[4-[[1-[4-[2-hydroxy-6-(4-hydroxyphenyl)-8,9-dihydro-7H-benzo[7]annulen-5-yl]phenyl]piperidin-4-yl]methyl]piperazin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30724029	O=C1CC[C@H](N2CC3=CC(N4CCN(CC5CCN(C6=CC=C(C7=C(C8=CC=C(O)C=C8)CCCC8=C7C=CC(O)=C8)C=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C46H49N5O5	ERα	P03372	CRBN	WO-2022166879-A1
TPD-E0EHUD	WO2022228556A1_1	3-[7-[3-[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-ethoxy-2-ethylphenyl]piperidin-4-yl]piperazine-1-carbonyl]azetidin-1-yl]-1-methylindazol-3-yl]piperidine-2,6-dione	CCOC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)C=C(CC)C(N2CCC(N3CCN(C(=O)C4CN(C5=CC=CC6=C5N(C)N=C6C5CCC(=O)NC5=O)C4)CC3)CC2)=C1	C55H66BrN12O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-CUUD5W	WO2022228556A1_10	3-[4-[2-[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-ethoxy-2-ethylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2,6-difluorophenyl]piperidine-2,6-dione	CCOC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)C=C(CC)C(N2CCC(N3CCN(CCC4=CC(F)=C(C5CCC(=O)NC5=O)C(F)=C4)CC3)CC2)=C1	C51H61BrF2N9O4P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-74US9T	WO2022228556A1_100	3-[4'-[2-[4-[1-[4-[[5-Bromo-4-[[2-methyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-ethoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2'-oxospiro[cyclopropane-1,3'-indole]-1'-yl]piperidine-2,6-dione	CCOC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(C)C=C4)=N2)C=C(C)C(N2CCC(N3CCN(CCC4=CC=CC5=C4C4(CC4)C(=O)N5C4CCC(=O)NC4=O)CC3)CC2)=C1	C53H62BrN10O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-ODEF7H	WO2022228556A1_101	3-[4-[2-[4-[1-[4-[[5-Bromo-4-[[2-methyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-ethoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2,6-difluorophenyl]piperidine-2,6-dione	CCOC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(C)C=C4)=N2)C=C(C)C(N2CCC(N3CCN(CCC4=CC(F)=C(C5CCC(=O)NC5=O)C(F)=C4)CC3)CC2)=C1	C49H57BrF2N9O4P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-28VVEP	WO2022228556A1_102	3-[4-[3-[4-[1-[4-[[5-Bromo-4-[[2-methyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-ethoxy-2-methylphenyl]piperidin-4-yl]piperazine-1-carbonyl]azetidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCOC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(C)C=C4)=N2)C=C(C)C(N2CCC(N3CCN(C(=O)C4CN(C5=CC(F)=C(C6CCC(=O)NC6=O)C(F)=C5)C4)CC3)CC2)=C1	C51H58BrF2N10O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-2KPPEQ	WO2022228556A1_103	3-[4-[(3R)-3-[4-[1-[4-[[5-bromo-4-[[2-methyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-ethoxy-2-methylphenyl]piperidin-4-yl]piperazine-1-carbonyl]pyrrolidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCOC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(C)C=C4)=N2)C=C(C)C(N2CCC(N3CCN(C(=O)[C@@H]4CCN(C5=CC(F)=C(C6CCC(=O)NC6=O)C(F)=C5)C4)CC3)CC2)=C1	C52H60BrF2N10O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-93FDW3	WO2022228556A1_104	3-[4-[(4R)-4-[4-[1-[4-[[5-bromo-4-[[2-methyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-ethoxy-2-methylphenyl]piperidin-4-yl]piperazine-1-carbonyl]-3,3-dimethylpyrrolidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCOC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(C)C=C4)=N2)C=C(C)C(N2CCC(N3CCN(C(=O)[C@H]4CN(C5=CC(F)=C(C6CCC(=O)NC6=O)C(F)=C5)CC4(C)C)CC3)CC2)=C1	C54H64BrF2N10O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-DMRS6J	WO2022228556A1_105	3-[4-[(3R)-3-[4-[1-[4-[[5-bromo-4-[[2-ethyl-8-fluoro-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazine-1-carbonyl]pyrrolidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(N=C(CC)C=C4)C(F)=C3)=N2)=C(OC)C=C1N1CCC(N2CCN(C(=O)[C@@H]3CCN(C4=CC(F)=C(C5CCC(=O)NC5=O)C(F)=C4)C3)CC2)CC1	C53H61BrF3N10O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-87NCAD	WO2022228556A1_106	3-[4-[(3R)-3-[4-[1-[4-[[5-bromo-4-[[2-methyl-5-(1-oxo-1lambda5-phosphetan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazine-1-carbonyl]pyrrolidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCC4)C4=C(C=C3)N=C(C)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(C(=O)[C@@H]3CCN(C4=CC(F)=C(C5CCC(=O)NC5=O)C(F)=C4)C3)CC2)CC1	C51H58BrF2N10O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-36WE7O	WO2022228556A1_107	3-[4-[(3R)-3-[4-[1-[4-[[5-bromo-4-[[2-methyl-5-(1-methyl-4-oxo-1,4lambda5-azaphosphinan-4-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazine-1-carbonyl]pyrrolidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCN(C)CC4)C4=C(C=C3)N=C(C)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(C(=O)[C@@H]3CCN(C4=CC(F)=C(C5CCC(=O)NC5=O)C(F)=C4)C3)CC2)CC1	C53H63BrF2N11O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-ENSWRS	WO2022228556A1_108	3-[4-[(3R)-3-[4-[1-[4-[[5-bromo-4-[[3-fluoro-2-methyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazine-1-carbonyl]pyrrolidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(C)C(F)=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(C(=O)[C@@H]3CCN(C4=CC(F)=C(C5CCC(=O)NC5=O)C(F)=C4)C3)CC2)CC1	C52H59BrF3N10O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-8C63HV	WO2022228556A1_109	.	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=CC=C4)N=C3)N2)=C(OC)C=C1N1CCC(N2CCN(C(=O)[C@@H]3CCN(C4=CC(F)=C(C5CCC(=O)NC5=O)C(F)=C4)C3)CC2)CC1	C51H60BrF2N10O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-8B8YWV	WO2022228556A1_11	3-[4-[3-[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-ethoxy-2-ethylphenyl]piperidin-4-yl]piperazine-1-carbonyl]azetidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCOC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)C=C(CC)C(N2CCC(N3CCN(C(=O)C4CN(C5=CC(F)=C(C6CCC(=O)NC6=O)C(F)=C5)C4)CC3)CC2)=C1	C53H62BrF2N10O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-AGF3R3	WO2022228556A1_110	3-[4-[(3R)-3-[4-[1-[4-[[5-bromo-4-[[7-fluoro-4-(1-oxo-1lambda5-phospholan-1-yl)quinolin-3-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazine-1-carbonyl]pyrrolidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C(F)C=C4)N=C3)=N2)=C(OC)C=C1N1CCC(N2CCN(C(=O)[C@@H]3CCN(C4=CC(F)=C(C5CCC(=O)NC5=O)C(F)=C4)C3)CC2)CC1	C51H57BrF3N10O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-A22L5A	WO2022228556A1_111	.	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C=CC=C3)N2)=C(OC)C=C1N1CCC(N2CCN(C(=O)[C@@H]3CCN(C4=CC(F)=C(C5CCC(=O)NC5=O)C(F)=C4)C3)CC2)CC1	C48H59BrF2N9O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-N67V8U	WO2022228556A1_112	3-[4-[(3R)-3-[4-[1-[4-[[5-bromo-4-[[2-methyl-1-oxo-5-(1-oxo-1lambda5-phospholan-1-yl)phthalazin-6-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazine-1-carbonyl]pyrrolidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)C(=O)N(C)N=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(C(=O)[C@@H]3CCN(C4=CC(F)=C(C5CCC(=O)NC5=O)C(F)=C4)C3)CC2)CC1	C51H59BrF2N11O6P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-CCT9L7	WO2022228556A1_113	3-[4-[(3R)-3-[4-[1-[4-[[5-bromo-4-[[2-cyclopropyl-1-oxo-5-(1-oxo-1lambda5-phospholan-1-yl)phthalazin-6-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazine-1-carbonyl]pyrrolidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)C(=O)N(C3CC3)N=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(C(=O)[C@@H]3CCN(C4=CC(F)=C(C5CCC(=O)NC5=O)C(F)=C4)C3)CC2)CC1	C53H61BrF2N11O6P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-SW92A1	WO2022228556A1_114	3-[4-[(3R)-3-[4-[1-[2-ethyl-5-methoxy-4-[[6-methyl-4-[[2-methyl-4-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazine-1-carbonyl]pyrrolidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC3=C(C=C(C)N3)C(NC3=CC4=C(C=C3)N=C(C)C=C4P3(=O)CCCC3)=N2)=C(OC)C=C1N1CCC(N2CCN(C(=O)[C@@H]3CCN(C4=CC(F)=C(C5CCC(=O)NC5=O)C(F)=C4)C3)CC2)CC1	C55H64F2N11O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-N5ACLI	WO2022228556A1_115	3-[4-[(3R)-3-[4-[1-[4-[[5-chloro-4-[[2-methyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazine-1-carbonyl]pyrrolidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC3=C(C(Cl)=CN3)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(C)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(C(=O)[C@@H]3CCN(C4=CC(F)=C(C5CCC(=O)NC5=O)C(F)=C4)C3)CC2)CC1	C54H61ClF2N11O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-MYT6MH	WO2022228556A1_116	3-[4-[(3R)-3-[4-[1-[2-ethyl-5-methoxy-4-[[4-[[2-methyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazine-1-carbonyl]pyrrolidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC3=C(C=CN3)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(C)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(C(=O)[C@@H]3CCN(C4=CC(F)=C(C5CCC(=O)NC5=O)C(F)=C4)C3)CC2)CC1	C54H62F2N11O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-4MX460	WO2022228556A1_117	3-[4-[(3R)-3-[4-[1-[2-ethyl-4-[[4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]-5-methoxyphenyl]piperidin-4-yl]piperazine-1-carbonyl]pyrrolidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC3=C(C=CN3)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(C(=O)[C@@H]3CCN(C4=CC(F)=C(C5CCC(=O)NC5=O)C(F)=C4)C3)CC2)CC1	C55H64F2N11O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-TMH4RD	WO2022228556A1_118	3-[4-[(3R)-3-[4-[1-[2-ethyl-5-methoxy-4-[[4-[[4-(1-oxo-1lambda5-phospholan-1-yl)quinolin-3-yl]amino]-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]phenyl]piperidin-4-yl]piperazine-1-carbonyl]pyrrolidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC3=C(C=CN3)C(NC3=C(P4(=O)CCCC4)C4=C(C=CC=C4)N=C3)=N2)=C(OC)C=C1N1CCC(N2CCN(C(=O)[C@@H]3CCN(C4=CC(F)=C(C5CCC(=O)NC5=O)C(F)=C4)C3)CC2)CC1	C53H60F2N11O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-XL2BYK	WO2022228556A1_119	3-[4-[(3R)-3-[4-[1-[4-[[5-bromo-4-[[4-(1-oxo-1lambda5-phospholan-1-yl)pyridin-3-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazine-1-carbonyl]pyrrolidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C=CN=C3)=N2)=C(OC)C=C1N1CCC(N2CCN(C(=O)[C@@H]3CCN(C4=CC(F)=C(C5CCC(=O)NC5=O)C(F)=C4)C3)CC2)CC1	C47H56BrF2N10O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-KHYO3C	WO2022228556A1_12	3-[4-[(3R)-3-[4-[1-[4-[[5-bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-ethoxy-2-ethylphenyl]piperidin-4-yl]piperazine-1-carbonyl]pyrrolidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCOC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)C=C(CC)C(N2CCC(N3CCN(C(=O)[C@@H]4CCN(C5=CC(F)=C(C6CCC(=O)NC6=O)C(F)=C5)C4)CC3)CC2)=C1	C54H64BrF2N10O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-U6UJY3	WO2022228556A1_120	3-[7-[2-[4-[1-[4-[[5-bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]ethoxy]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(CCOC3=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)CC2)CC1	C52H62BrN10O6P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-Z049AM	WO2022228556A1_121	3-[7-[2-[4-[1-[4-[[5-bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]ethyl-methylamino]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(CCN(C)C3=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)CC2)CC1	C53H65BrN11O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-5P5KWL	WO2022228556A1_122	3-[6-[(3R)-3-[4-[1-[4-[[5-bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazine-1-carbonyl]pyrrolidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(C(=O)[C@@H]3CCN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5)C3)CC2)CC1	C55H65BrN11O6P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-MC1YAR	WO2022228556A1_123	3-[6-[(3S)-3-[[4-[1-[4-[[5-bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]methyl]pyrrolidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(C[C@@H]3CCN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5)C3)CC2)CC1	C55H67BrN11O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-N6PMPP	WO2022228556A1_124	.	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(C(=O)C3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)C3)CC2)CC1	C55H63BrN11O7P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-KGSFEP	WO2022228556A1_125	5-[3-[3-[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]propyl]azetidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(CCCC3CN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)CC2)CC1	C56H67BrN11O6P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-U6Z1UN	WO2022228556A1_126	5-[3-[[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]methyl]azetidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(CC3CN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)CC2)CC1	C54H63BrN11O6P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-0KG3MH	WO2022228556A1_127	5-[3-[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazine-1-carbonyl]azetidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(C(=O)C3CN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)CC2)CC1	C54H61BrN11O7P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-JK2QDZ	WO2022228556A1_128	3-[5-[3-[[4-[1-[4-[[5-bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]methyl]azetidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(CC3CN(C4=CC=C5CN(C6CCC(=O)NC6=O)C(=O)C5=C4)C3)CC2)CC1	C54H65BrN11O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-0EF4W4	WO2022228556A1_129	3-[4-[3-[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]cyclobutyl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(C3CC(C4=CC(F)=C(C5CCC(=O)NC5=O)C(F)=C4)C3)CC2)CC1	C52H61BrF2N9O4P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-LEXAVN	WO2022228556A1_13	.	CCOC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)C=C(CC)C(N2CCC(N3CCN(C(=O)C4CN(C5=CC(F)=C(C6CCC(=O)NC6=O)C(F)=C5)CC4(C)C)CC3)CC2)=C1	C56H68BrF2N10O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-3SBVUW	WO2022228556A1_130	3-[4-[[3-[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazine-1-carbonyl]cyclobutyl]-methylamino]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(C(=O)[C@H]3C[C@H](N(C)C4=CC(F)=C(C5CCC(=O)NC5=O)C(F)=C4)C3)CC2)CC1	C54H64BrF2N10O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-I49673	WO2022228556A1_131	3-[4-[3-[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazine-1-carbonyl]cyclobutyl]oxyphenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(C(=O)C3CC(OC4=CC=C(C5CCC(=O)NC5=O)C=C4)C3)CC2)CC1	C53H63BrN9O6P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-8ZBYDP	WO2022228556A1_132	3-[3-[3-[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazine-1-carbonyl]azetidin-1-yl]phenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(C(=O)C3CN(C4=CC(C5CCC(=O)NC5=O)=CC=C4)C3)CC2)CC1	C52H62BrN10O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-5SL405	WO2022228556A1_133	.	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(C)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(CCC3=CC=C(C4(F)CCC(=O)NC4=O)C=C3)CC2)CC1	C49H58BrFN9O4P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-ZXPD54	WO2022228556A1_134	3-[4-[[2-[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]-2-oxoethyl]amino]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(C(=O)CNC3=CC(F)=C(C4CCC(=O)NC4=O)C(F)=C3)CC2)CC1	C50H58BrF2N10O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-14GXP8	WO2022228556A1_136	3-[4-[2-[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]anilino]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(CCC3=CC=C(NC4CCC(=O)NC4=O)C=C3)CC2)CC1	C50H62BrN10O4P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-IVL9J1	WO2022228556A1_137	3-[4-[2-[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]phenoxy]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(CCC3=CC=C(OC4CCC(=O)NC4=O)C=C3)CC2)CC1	C50H61BrN9O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-H6OC5S	WO2022228556A1_138	3-[4-[2-[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]phenyl]-3-methylpiperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(CCC3=CC=C(C4(C)CCC(=O)NC4=O)C=C3)CC2)CC1	C51H63BrN9O4P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-VE805O	WO2022228556A1_14	3-[7-[3-[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazine-1-carbonyl]azetidin-1-yl]-1-methylindazol-3-yl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(C(=O)C3CN(C4=CC=CC5=C4N(C)N=C5C4CCC(=O)NC4=O)C3)CC2)CC1	C54H64BrN12O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-48LIBM	WO2022228556A1_140	3-[4-[4-[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazine-1-carbonyl]piperidin-1-yl]-2,6-difluoroanilino]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(C(=O)C3CCN(C4=CC(F)=C(NC5CCC(=O)NC5=O)C(F)=C4)CC3)CC2)CC1	C54H65BrF2N11O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-0WAWUE	WO2022228556A1_141	1-[4-[2-[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]phenyl]-1,3-diazinane-2,4-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(CCC3=CC=C(N4CCC(=O)NC4=O)C=C3)CC2)CC1	C49H60BrN10O4P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-8SJZ02	WO2022228556A1_142	3-[4-[[4-[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazine-1-carbonyl]-1-bicyclo[2.2.1]heptanyl]amino]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(C(=O)C34CCC(NC5=CC(F)=C(C6CCC(=O)NC6=O)C(F)=C5)(CC3)C4)CC2)CC1	C56H66BrF2N10O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-I7VT5X	SCHEMBL27207137	3-[4-[(3R)-3-[4-[1-[4-[[5-bromo-4-[[2-methyl-5-(1-oxo-2,5-dihydro-1lambda5-phosphol-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazine-1-carbonyl]pyrrolidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=CC=C4N=C(C)C=CC4=C3P3(=O)CC=CC3)=N2)=C(OC)C=C1N1CCC(N2CCN(C(=O)[C@@H]3CCN(C4=CC(F)=C(C5CCC(=O)NC5=O)C(F)=C4)C3)CC2)CC1	C52H58BrF2N10O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-E1SZQQ	SCHEMBL27207018	3-[4-[2-[4-[1-[4-[[5-Bromo-4-[[2-methyl-5-(1-oxo-2,5-dihydro-1lambda5-phosphol-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=CC=C4N=C(C)C=CC4=C3P3(=O)CC=CC3)=N2)=C(OC)C=C1N1CCC(N2CCN(CCC3=CC(F)=C(C4CCC(=O)NC4=O)C(F)=C3)CC2)CC1	C49H55BrF2N9O4P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-4CXND8	SCHEMBL27206964	3-[6-[2-[4-[1-[4-[[5-Bromo-4-[[2-methyl-5-(1-oxo-2,5-dihydro-1lambda5-phosphol-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2-oxo-1,3-benzoxazol-3-yl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=CC=C4N=C(C)C=CC4=C3P3(=O)CC=CC3)=N2)=C(OC)C=C1N1CCC(N2CCN(CCC3=CC=C4C(=C3)OC(=O)N4C3CCC(=O)NC3=O)CC2)CC1	C50H56BrN10O6P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-Q46BLT	SCHEMBL27206996	3-[4-[3-[4-[1-[4-[[5-Bromo-4-[[2-methyl-5-(1-oxo-2,5-dihydro-1lambda5-phosphol-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazine-1-carbonyl]azetidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CC=CC4)C4=C(C=C3)N=C(C)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(C(=O)C3CN(C4=CC(F)=C(C5CCC(=O)NC5=O)C(F)=C4)C3)CC2)CC1	C51H56BrF2N10O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-6TRJ7H	SCHEMBL27207075	3-[4-[2-[4-[1-[4-[[5-Bromo-4-[2-(1-oxo-1lambda5-phospholan-1-yl)anilino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C=CC=C3)=N2)=C(OC)C=C1N1CCC(N2CCN(CCC3=CC(F)=C(C4CCC(=O)NC4=O)C(F)=C3)CC2)CC1	C45H54BrF2N8O4P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-75CWPV	SCHEMBL27207419	3-[4-[3-[4-[1-[4-[[5-Bromo-4-[2-(1-oxo-1lambda5-phospholan-1-yl)anilino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazine-1-carbonyl]azetidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C=CC=C3)=N2)=C(OC)C=C1N1CCC(N2CCN(C(=O)C3CN(C4=CC(F)=C(C5CCC(=O)NC5=O)C(F)=C4)C3)CC2)CC1	C47H55BrF2N9O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-DTVAMU	WO2022228556A1_149	3-[4-[2-[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-3-methyl-2-oxo-1,3-benzoxazol-7-yl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(CCC3=CC=C(C4CCC(=O)NC4=O)C4=C3N(C)C(=O)O4)CC2)CC1	C52H62BrN10O6P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-TH25HM	WO2022228556A1_15	3-[4-[2-[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-3-cyclopropyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(CCC3=CC=CC4=C3N(C3CC3)C(=O)N4C3CCC(=O)NC3=O)CC2)CC1	C54H65BrN11O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-IUO0FD	WO2022228556A1_150	3-[7-[2-[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-1,3-dimethyl-2-oxobenzimidazol-4-yl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(CCC3=CC=C(C4CCC(=O)NC4=O)C4=C3N(C)C(=O)N4C)CC2)CC1	C53H65BrN11O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-VSLXN6	WO2022228556A1_151	3-[7-[2-[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-1-methylindazol-4-yl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(CCC3=CC=C(C4CCC(=O)NC4=O)C4=C3N(C)N=C4)CC2)CC1	C52H63BrN11O4P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-EY7IBG	WO2022228556A1_152	3-[4-[2-[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-1-methylindazol-7-yl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(CCC3=CC=C(C4CCC(=O)NC4=O)C4=C3C=NN4C)CC2)CC1	C52H63BrN11O4P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-CWHLTG	WO2022228556A1_153	.	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(CCC3=CC=C(C4CCC(=O)NC4=O)C4C3OC(=O)N4C)CC2)CC1	C52H64BrN10O6P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-DN3JS7	WO2022228556A1_154	3-[6-[2-[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-2-cyclopropyl-5-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2-oxo-1,3-benzoxazol-3-yl]piperidine-2,6-dione	CCC1=NC2=C(C=C1)C(P1(=O)CCCC1)=C(NC1=NC(NC3=C(OC)C=C(N4CCC(N5CCN(CCC6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)O7)CC5)CC4)C(C4CC4)=C3)=NC=C1Br)C=C2	C52H60BrN10O6P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-8AC45M	WO2022228556A1_155	3-[6-[2-[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-(trifluoromethoxy)phenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2-oxo-1,3-benzoxazol-3-yl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)=C(OC(F)(F)F)C=C1N1CCC(N2CCN(CCC3=CC4=C(C=C3)N(C3CCC(=O)NC3=O)C(=O)O4)CC2)CC1	C51H57BrF3N10O6P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-TADDGH	WO2022228556A1_156	3-[4-[2-[(2S)-4-[1-[4-[[5-bromo-4-[[2-ethyl-8-fluoro-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-cyclopropyloxy-2-ethylphenyl]piperidin-4-yl]-2-(hydroxymethyl)piperazin-1-yl]ethyl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(N=C(CC)C=C4)C(F)=C3)=N2)=C(OC2CC2)C=C1N1CCC(N2CCN(CCC3=CC(F)=C(C4CCC(=O)NC4=O)C(F)=C3)[C@H](CO)C2)CC1	C53H62BrF3N9O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-VHK8TU	WO2022228556A1_157	.	CCC1=CC(NC2=NC=C(Br)C(NC3=CC=C4N=C(C)C=CC4=C3P3(=O)CCC3)N2)=C(OC)C=C1N1CCC(N2CCN(CCC3=C4C(=CC=C3)N(C3CCC(=O)NC3=O)C(=O)N4CC)CC2)CC1	C51H63BrN11O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-LOTSC6	WO2022228556A1_158	3-[6-[2-[4-[1-[4-[[5-Bromo-4-[[2-methyl-5-(1-oxo-1lambda5-phosphetan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-5-fluoro-2-oxo-1,3-benzoxazol-3-yl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=CC=C4N=C(C)C=CC4=C3P3(=O)CCC3)=N2)=C(OC)C=C1N1CCC(N2CCN(CCC3=C(F)C=C4C(=C3)OC(=O)N4C3CCC(=O)NC3=O)CC2)CC1	C49H55BrFN10O6P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-82IYNT	WO2022228556A1_16	3-[4-[2-[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(CCC3=CC=CC4=C3N(C)C(=O)N4C3CCC(=O)NC3=O)CC2)CC1	C52H63BrN11O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-5AGISW	WO2022228556A1_17	3-[4-[2-[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-3-ethyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(CCC3=CC=CC4=C3N(CC)C(=O)N4C3CCC(=O)NC3=O)CC2)CC1	C53H65BrN11O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-IF9JEN	WO2022228556A1_18	3-[7-[2-[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2-oxo-1,3-benzoxazol-3-yl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(CCC3=CC=CC4=C3OC(=O)N4C3CCC(=O)NC3=O)CC2)CC1	C51H60BrN10O6P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-DS7Z8O	WO2022228556A1_19	3-[6-[2-[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2-oxo-1,3-benzoxazol-3-yl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(CCC3=CC4=C(C=C3)N(C3CCC(=O)NC3=O)C(=O)O4)CC2)CC1	C51H60BrN10O6P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-KXT5HU	WO2022228556A1_2	3-[4-[2-[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-ethoxy-2-ethylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-3-cyclopropyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	CCOC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)C=C(CC)C(N2CCC(N3CCN(CCC4=CC=CC5=C4N(C4CC4)C(=O)N5C4CCC(=O)NC4=O)CC3)CC2)=C1	C55H67BrN11O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-I5RWGF	WO2022228556A1_20	3-[5-[2-[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-3,3-dimethyl-2-oxoindol-1-yl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(CCC3=CC4=C(C=C3)N(C3CCC(=O)NC3=O)C(=O)C4(C)C)CC2)CC1	C54H66BrN10O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-WP4YUR	WO2022228556A1_21	3-[4-[2-[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-3,3-dimethyl-2-oxoindol-1-yl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(CCC3=CC=CC4=C3C(C)(C)C(=O)N4C3CCC(=O)NC3=O)CC2)CC1	C54H66BrN10O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-XN8BJ6	WO2022228556A1_22	3-[4'-[2-[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2'-oxospiro[cyclopropane-1,3'-indole]-1'-yl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(CCC3=CC=CC4=C3C3(CC3)C(=O)N4C3CCC(=O)NC3=O)CC2)CC1	C54H64BrN10O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-4H19GA	WO2022228556A1_23	3-[4-[2-[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(CCC3=CC(F)=C(C4CCC(=O)NC4=O)C(F)=C3)CC2)CC1	C50H59BrF2N9O4P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-QIOPLM	WO2022228556A1_24	3-[4-[3-[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazine-1-carbonyl]azetidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(C(=O)C3CN(C4=CC(F)=C(C5CCC(=O)NC5=O)C(F)=C4)C3)CC2)CC1	C52H60BrF2N10O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-PA9T0H	WO2022228556A1_25	.	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)=C(OC)C=C1C1CCC(N2CCN(C(=O)C3CCN(C4=CC(F)=C(C5CCC(=O)NC5=O)C(F)=C4)C3)CC2)CC1	C54H63BrF2N9O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-C58R6T	WO2022228556A1_26	3-[4-[(4R)-4-[4-[1-[4-[[5-bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazine-1-carbonyl]-3,3-dimethylpyrrolidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(C(=O)[C@H]3CN(C4=CC(F)=C(C5CCC(=O)NC5=O)C(F)=C4)CC3(C)C)CC2)CC1	C55H66BrF2N10O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-C43CHX	WO2022228556A1_27	3-[7-[3-[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazine-1-carbonyl]azetidin-1-yl]-1-methylindazol-3-yl]piperidine-2,6-dione	CCC1=NC2=C(C=C1)C(P1(=O)CCCC1)=C(NC1=NC(NC3=C(OC)C=C(N4CCC(N5CCN(C(=O)C6CN(C7=CC=CC8=C7N(C)N=C8C7CCC(=O)NC7=O)C6)CC5)CC4)C(C)=C3)=NC=C1Br)C=C2	C53H62BrN12O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-T9SW0A	WO2022228556A1_28	3-[4-[2-[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-3-ethyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	CCC1=NC2=C(C=C1)C(P1(=O)CCCC1)=C(NC1=NC(NC3=C(OC)C=C(N4CCC(N5CCN(CCC6=CC=CC7=C6N(CC)C(=O)N7C6CCC(=O)NC6=O)CC5)CC4)C(C)=C3)=NC=C1Br)C=C2	C52H63BrN11O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-UDQPHO	WO2022228556A1_29	3-[4-[2-[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	CCC1=NC2=C(C=C1)C(P1(=O)CCCC1)=C(NC1=NC(NC3=C(OC)C=C(N4CCC(N5CCN(CCC6=CC=CC7=C6N(C)C(=O)N7C6CCC(=O)NC6=O)CC5)CC4)C(C)=C3)=NC=C1Br)C=C2	C51H61BrN11O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-P8QFTJ	WO2022228556A1_3	3-[4-[2-[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-ethoxy-2-ethylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	CCOC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)C=C(CC)C(N2CCC(N3CCN(CCC4=CC=CC5=C4N(C)C(=O)N5C4CCC(=O)NC4=O)CC3)CC2)=C1	C53H65BrN11O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-O61TZQ	WO2022228556A1_31	3-[7-[2-[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2-oxo-1,3-benzoxazol-3-yl]piperidine-2,6-dione	CCC1=NC2=C(C=C1)C(P1(=O)CCCC1)=C(NC1=NC(NC3=C(OC)C=C(N4CCC(N5CCN(CCC6=CC=CC7=C6OC(=O)N7C6CCC(=O)NC6=O)CC5)CC4)C(C)=C3)=NC=C1Br)C=C2	C50H58BrN10O6P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-FB8YA4	WO2022228556A1_32	3-[6-[2-[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2-oxo-1,3-benzoxazol-3-yl]piperidine-2,6-dione	CCC1=NC2=C(C=C1)C(P1(=O)CCCC1)=C(NC1=NC(NC3=C(OC)C=C(N4CCC(N5CCN(CCC6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)O7)CC5)CC4)C(C)=C3)=NC=C1Br)C=C2	C50H58BrN10O6P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-XQF2G7	WO2022228556A1_33	3-[5-[2-[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-3,3-dimethyl-2-oxoindol-1-yl]piperidine-2,6-dione	CCC1=NC2=C(C=C1)C(P1(=O)CCCC1)=C(NC1=NC(NC3=C(OC)C=C(N4CCC(N5CCN(CCC6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)C7(C)C)CC5)CC4)C(C)=C3)=NC=C1Br)C=C2	C53H64BrN10O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-L8MNJD	WO2022228556A1_34	3-[4-[2-[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-3,3-dimethyl-2-oxoindol-1-yl]piperidine-2,6-dione	CCC1=NC2=C(C=C1)C(P1(=O)CCCC1)=C(NC1=NC(NC3=C(OC)C=C(N4CCC(N5CCN(CCC6=CC=CC7=C6C(C)(C)C(=O)N7C6CCC(=O)NC6=O)CC5)CC4)C(C)=C3)=NC=C1Br)C=C2	C53H64BrN10O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-UHDC3M	WO2022228556A1_35	3-[4'-[2-[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2'-oxospiro[cyclopropane-1,3'-indole]-1'-yl]piperidine-2,6-dione	CCC1=NC2=C(C=C1)C(P1(=O)CCCC1)=C(NC1=NC(NC3=C(OC)C=C(N4CCC(N5CCN(CCC6=CC=CC7=C6C6(CC6)C(=O)N7C6CCC(=O)NC6=O)CC5)CC4)C(C)=C3)=NC=C1Br)C=C2	C53H62BrN10O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-O636OM	WO2022228556A1_36	.	CCC1=NC2=C(C=C1)C(P1(=O)CCCC1)=C(NC1=NC(NC3=C(OC)C=C(N4CCC(N5CCN(CCC6=CC(C)=C(C7CCC(=O)NC7=O)C(F)=C6)CC5)CC4)C(C)=C3)=NC=C1Br)C=C2	C50H60BrFN9O4P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-OOZN0C	WO2022228556A1_37	3-[4-[3-[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazine-1-carbonyl]azetidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=NC2=C(C=C1)C(P1(=O)CCCC1)=C(NC1=NC(NC3=C(OC)C=C(N4CCC(N5CCN(C(=O)C6CN(C7=CC(F)=C(C8CCC(=O)NC8=O)C(F)=C7)C6)CC5)CC4)C(C)=C3)=NC=C1Br)C=C2	C51H58BrF2N10O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-680RER	WO2022228556A1_38	.	CCC1=NC2=C(C=C1)C(P1(=O)CCCC1)=C(NC1NC(NC3=C(OC)C=C(N4CCC(N5CCN(C(=O)[C@@H]6CCN(C7=CC(F)=C(C8CCC(=O)NC8=O)C(F)=C7)C6)CC5)CC4)C(C)=C3)=NC=C1Br)C=C2	C52H62BrF2N10O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-XJFPKA	WO2022228556A1_39	3-[4-[(4R)-4-[4-[1-[4-[[5-bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazine-1-carbonyl]-3,3-dimethylpyrrolidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=NC2=C(C=C1)C(P1(=O)CCCC1)=C(NC1=NC(NC3=C(OC)C=C(N4CCC(N5CCN(C(=O)[C@H]6CN(C7=CC(F)=C(C8CCC(=O)NC8=O)C(F)=C7)CC6(C)C)CC5)CC4)C(C)=C3)=NC=C1Br)C=C2	C54H64BrF2N10O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-78VGRU	WO2022228556A1_4	3-[4-[2-[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-ethoxy-2-ethylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-3-ethyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	CCOC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)C=C(CC)C(N2CCC(N3CCN(CCC4=CC=CC5=C4N(CC)C(=O)N5C4CCC(=O)NC4=O)CC3)CC2)=C1	C54H67BrN11O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-CS84XF	WO2022228556A1_40	3-[7-[3-[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-ethoxy-2-methylphenyl]piperidin-4-yl]piperazine-1-carbonyl]azetidin-1-yl]-1-methylindazol-3-yl]piperidine-2,6-dione	CCOC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)C=C(C)C(N2CCC(N3CCN(C(=O)C4CN(C5=CC=CC6=C5N(C)N=C6C5CCC(=O)NC5=O)C4)CC3)CC2)=C1	C54H64BrN12O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-Y6GXTQ	WO2022228556A1_41	3-[4-[2-[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-ethoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-3-cyclopropyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	CCOC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)C=C(C)C(N2CCC(N3CCN(CCC4=CC=CC5=C4N(C4CC4)C(=O)N5C4CCC(=O)NC4=O)CC3)CC2)=C1	C54H65BrN11O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-ZDFC5T	WO2022228556A1_42	3-[4-[2-[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-ethoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	CCOC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)C=C(C)C(N2CCC(N3CCN(CCC4=CC=CC5=C4N(C)C(=O)N5C4CCC(=O)NC4=O)CC3)CC2)=C1	C52H63BrN11O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-9GTUEB	WO2022228556A1_43	3-[4-[2-[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-ethoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-3-ethyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	CCOC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)C=C(C)C(N2CCC(N3CCN(CCC4=CC=CC5=C4N(CC)C(=O)N5C4CCC(=O)NC4=O)CC3)CC2)=C1	C53H65BrN11O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-OR9ZXG	WO2022228556A1_44	3-[7-[2-[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-ethoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2-oxo-1,3-benzoxazol-3-yl]piperidine-2,6-dione	CCOC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)C=C(C)C(N2CCC(N3CCN(CCC4=CC=CC5=C4OC(=O)N5C4CCC(=O)NC4=O)CC3)CC2)=C1	C51H60BrN10O6P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-26NRY1	WO2022228556A1_45	3-[6-[2-[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-ethoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2-oxo-1,3-benzoxazol-3-yl]piperidine-2,6-dione	CCOC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)C=C(C)C(N2CCC(N3CCN(CCC4=CC5=C(C=C4)N(C4CCC(=O)NC4=O)C(=O)O5)CC3)CC2)=C1	C51H60BrN10O6P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-5TC3OR	WO2022228556A1_46	3-[5-[2-[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-ethoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-3,3-dimethyl-2-oxoindol-1-yl]piperidine-2,6-dione	CCOC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)C=C(C)C(N2CCC(N3CCN(CCC4=CC5=C(C=C4)N(C4CCC(=O)NC4=O)C(=O)C5(C)C)CC3)CC2)=C1	C54H66BrN10O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-ZL6XWZ	WO2022228556A1_47	3-[4-[2-[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-ethoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-3,3-dimethyl-2-oxoindol-1-yl]piperidine-2,6-dione	CCOC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)C=C(C)C(N2CCC(N3CCN(CCC4=CC=CC5=C4C(C)(C)C(=O)N5C4CCC(=O)NC4=O)CC3)CC2)=C1	C54H66BrN10O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-NOB8J7	WO2022228556A1_48	3-[4'-[2-[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-ethoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2'-oxospiro[cyclopropane-1,3'-indole]-1'-yl]piperidine-2,6-dione	CCOC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)C=C(C)C(N2CCC(N3CCN(CCC4=CC=CC5=C4C4(CC4)C(=O)N5C4CCC(=O)NC4=O)CC3)CC2)=C1	C54H64BrN10O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-O9V6NJ	WO2022228556A1_49	3-[4-[2-[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-ethoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2,6-difluorophenyl]piperidine-2,6-dione	CCOC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)C=C(C)C(N2CCC(N3CCN(CCC4=CC(F)=C(C5CCC(=O)NC5=O)C(F)=C4)CC3)CC2)=C1	C50H59BrF2N9O4P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-K4ZUQA	WO2022228556A1_5	3-[7-[2-[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-ethoxy-2-ethylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2-oxo-1,3-benzoxazol-3-yl]piperidine-2,6-dione	CCOC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)C=C(CC)C(N2CCC(N3CCN(CCC4=CC=CC5=C4OC(=O)N5C4CCC(=O)NC4=O)CC3)CC2)=C1	C52H62BrN10O6P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-XT2NAG	WO2022228556A1_51	3-[4-[(3R)-3-[4-[1-[4-[[5-bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-ethoxy-2-methylphenyl]piperidin-4-yl]piperazine-1-carbonyl]pyrrolidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCOC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)C=C(C)C(N2CCC(N3CCN(C(=O)[C@@H]4CCN(C5=CC(F)=C(C6CCC(=O)NC6=O)C(F)=C5)C4)CC3)CC2)=C1	C53H62BrF2N10O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-SW3MDR	WO2022228556A1_52	3-[4-[(4R)-4-[4-[1-[4-[[5-bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-ethoxy-2-methylphenyl]piperidin-4-yl]piperazine-1-carbonyl]-3,3-dimethylpyrrolidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCOC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)C=C(C)C(N2CCC(N3CCN(C(=O)[C@H]4CN(C5=CC(F)=C(C6CCC(=O)NC6=O)C(F)=C5)CC4(C)C)CC3)CC2)=C1	C55H66BrF2N10O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-PCJ0JI	WO2022228556A1_53	3-[7-[3-[4-[1-[4-[[5-Bromo-4-[[2-methyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-ethoxy-2-ethylphenyl]piperidin-4-yl]piperazine-1-carbonyl]azetidin-1-yl]-1-methylindazol-3-yl]piperidine-2,6-dione	CCOC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(C)C=C4)=N2)C=C(CC)C(N2CCC(N3CCN(C(=O)C4CN(C5=CC=CC6=C5N(C)N=C6C5CCC(=O)NC5=O)C4)CC3)CC2)=C1	C54H64BrN12O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-SAJIPE	WO2022228556A1_54	.	CCOC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(C)C=C4)N2)C=C(CC)C(N2CCC(N3CCN(CCC4=CC=CC5=C4N(C4CC4)C(=O)N5C4CCC(=O)NC4=O)CC3)CC2)=C1	C54H67BrN11O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-ZAMQMV	WO2022228556A1_55	3-[4-[2-[4-[1-[4-[[5-Bromo-4-[[2-methyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-ethoxy-2-ethylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	CCOC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(C)C=C4)=N2)C=C(CC)C(N2CCC(N3CCN(CCC4=CC=CC5=C4N(C)C(=O)N5C4CCC(=O)NC4=O)CC3)CC2)=C1	C52H63BrN11O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-FR4LT3	WO2022228556A1_56	3-[4-[2-[4-[1-[4-[[5-Bromo-4-[[2-methyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-3-ethyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(C)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(CCC3=CC=CC4=C3N(CC)C(=O)N4C3CCC(=O)NC3=O)CC2)CC1	C52H63BrN11O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-8RJZSF	WO2022228556A1_57	3-[7-[2-[4-[1-[4-[[5-Bromo-4-[[2-methyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-ethoxy-2-ethylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2-oxo-1,3-benzoxazol-3-yl]piperidine-2,6-dione	CCOC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(C)C=C4)=N2)C=C(CC)C(N2CCC(N3CCN(CCC4=CC=CC5=C4OC(=O)N5C4CCC(=O)NC4=O)CC3)CC2)=C1	C51H60BrN10O6P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-K1OE90	WO2022228556A1_58	.	CCOC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(C)C=C4)=N2)C=C(CC)C(N2CCC(N3CCN(CCC4=CC5=C(C=C4)N(C4CCC(=O)NC4=O)C(=O)O5)C3)CC2)=C1	C50H58BrN10O6P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-L56I1I	WO2022228556A1_59	3-[5-[2-[4-[1-[4-[[5-Bromo-4-[[2-methyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-ethoxy-2-ethylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-3,3-dimethyl-2-oxoindol-1-yl]piperidine-2,6-dione	CCOC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(C)C=C4)=N2)C=C(CC)C(N2CCC(N3CCN(CCC4=CC5=C(C=C4)N(C4CCC(=O)NC4=O)C(=O)C5(C)C)CC3)CC2)=C1	C54H66BrN10O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-WQRX9B	WO2022228556A1_6	3-[6-[2-[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-ethoxy-2-ethylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2-oxo-1,3-benzoxazol-3-yl]piperidine-2,6-dione	CCOC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)C=C(CC)C(N2CCC(N3CCN(CCC4=CC5=C(C=C4)N(C4CCC(=O)NC4=O)C(=O)O5)CC3)CC2)=C1	C52H62BrN10O6P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-6T3XAH	WO2022228556A1_60	3-[4-[2-[4-[1-[4-[[5-Bromo-4-[[2-methyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-ethoxy-2-ethylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-3,3-dimethyl-2-oxoindol-1-yl]piperidine-2,6-dione	CCOC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(C)C=C4)=N2)C=C(CC)C(N2CCC(N3CCN(CCC4=CC=CC5=C4C(C)(C)C(=O)N5C4CCC(=O)NC4=O)CC3)CC2)=C1	C54H66BrN10O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-WZ4BYH	WO2022228556A1_61	3-[4'-[2-[4-[1-[4-[[5-Bromo-4-[[2-methyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-ethoxy-2-ethylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2'-oxospiro[cyclopropane-1,3'-indole]-1'-yl]piperidine-2,6-dione	CCOC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(C)C=C4)=N2)C=C(CC)C(N2CCC(N3CCN(CCC4=CC=CC5=C4C4(CC4)C(=O)N5C4CCC(=O)NC4=O)CC3)CC2)=C1	C54H64BrN10O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-PZNHO9	SCHEMBL27207052	3-[4-[2-[4-[1-[4-[[5-Bromo-4-[[2-methyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-ethoxy-2-ethylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2,6-difluorophenyl]piperidine-2,6-dione	CCOC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(C)C=C4)=N2)C=C(CC)C(N2CCC(N3CCN(CCC4=CC(F)=C(C5CCC(=O)NC5=O)C(F)=C4)CC3)CC2)=C1	C50H59BrF2N9O4P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-B49FQX	WO2022228556A1_63	3-[4-[3-[4-[1-[4-[[5-Bromo-4-[[2-methyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-ethoxy-2-ethylphenyl]piperidin-4-yl]piperazine-1-carbonyl]azetidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCOC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(C)C=C4)=N2)C=C(CC)C(N2CCC(N3CCN(C(=O)C4CN(C5=CC(F)=C(C6CCC(=O)NC6=O)C(F)=C5)C4)CC3)CC2)=C1	C52H60BrF2N10O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-QXC5U5	WO2022228556A1_64	3-[4-[(3R)-3-[4-[1-[4-[[5-bromo-4-[[2-methyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-ethoxy-2-ethylphenyl]piperidin-4-yl]piperazine-1-carbonyl]pyrrolidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCOC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(C)C=C4)=N2)C=C(CC)C(N2CCC(N3CCN(C(=O)[C@@H]4CCN(C5=CC(F)=C(C6CCC(=O)NC6=O)C(F)=C5)C4)CC3)CC2)=C1	C53H62BrF2N10O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-786YMH	WO2022228556A1_65	3-[4-[(4R)-4-[4-[1-[4-[[5-bromo-4-[[2-methyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-ethoxy-2-ethylphenyl]piperidin-4-yl]piperazine-1-carbonyl]-3,3-dimethylpyrrolidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCOC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(C)C=C4)=N2)C=C(CC)C(N2CCC(N3CCN(C(=O)[C@H]4CN(C5=CC(F)=C(C6CCC(=O)NC6=O)C(F)=C5)CC4(C)C)CC3)CC2)=C1	C55H66BrF2N10O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-Q0FSDD	WO2022228556A1_66	3-[7-[3-[4-[1-[4-[[5-Bromo-4-[[2-methyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazine-1-carbonyl]azetidin-1-yl]-1-methylindazol-3-yl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(C)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(C(=O)C3CN(C4=CC=CC5=C4N(C)N=C5C4CCC(=O)NC4=O)C3)CC2)CC1	C53H62BrN12O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-2TEM5C	WO2022228556A1_67	3-[4-[2-[4-[1-[4-[[5-Bromo-4-[[2-methyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-3-cyclopropyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(C)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(CCC3=CC=CC4=C3N(C3CC3)C(=O)N4C3CCC(=O)NC3=O)CC2)CC1	C53H63BrN11O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-XZOANX	SCHEMBL27207377	3-[4-[2-[4-[1-[4-[[5-Bromo-4-[[2-methyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(C)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(CCC3=CC=CC4=C3N(C)C(=O)N4C3CCC(=O)NC3=O)CC2)CC1	C51H61BrN11O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-IOXSG0	WO2022228556A1_7	3-[5-[2-[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-ethoxy-2-ethylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-3,3-dimethyl-2-oxoindol-1-yl]piperidine-2,6-dione	CCOC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)C=C(CC)C(N2CCC(N3CCN(CCC4=CC5=C(C=C4)N(C4CCC(=O)NC4=O)C(=O)C5(C)C)CC3)CC2)=C1	C55H68BrN10O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-RYPIXI	WO2022228556A1_70	3-[7-[2-[4-[1-[4-[[5-Bromo-4-[[2-methyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2-oxo-1,3-benzoxazol-3-yl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(C)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(CCC3=CC=CC4=C3OC(=O)N4C3CCC(=O)NC3=O)CC2)CC1	C50H58BrN10O6P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-0K8ZT8	SCHEMBL27207024	3-[6-[2-[4-[1-[4-[[5-Bromo-4-[[2-methyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2-oxo-1,3-benzoxazol-3-yl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(C)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(CCC3=CC4=C(C=C3)N(C3CCC(=O)NC3=O)C(=O)O4)CC2)CC1	C50H58BrN10O6P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-7UQ11P	WO2022228556A1_72	3-[5-[2-[4-[1-[4-[[5-Bromo-4-[[2-methyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-3,3-dimethyl-2-oxoindol-1-yl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(C)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(CCC3=CC4=C(C=C3)N(C3CCC(=O)NC3=O)C(=O)C4(C)C)CC2)CC1	C53H64BrN10O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-2GM59K	SCHEMBL27207284	3-[4-[2-[4-[1-[4-[[5-Bromo-4-[[2-methyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-3,3-dimethyl-2-oxoindol-1-yl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(C)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(CCC3=CC=CC4=C3C(C)(C)C(=O)N4C3CCC(=O)NC3=O)CC2)CC1	C53H64BrN10O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-T594UR	WO2022228556A1_74	3-[4'-[2-[4-[1-[4-[[5-Bromo-4-[[2-methyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2'-oxospiro[cyclopropane-1,3'-indole]-1'-yl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(C)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(CCC3=CC=CC4=C3C3(CC3)C(=O)N4C3CCC(=O)NC3=O)CC2)CC1	C53H62BrN10O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-OZTGOH	SCHEMBL27207160	3-[4-[2-[4-[1-[4-[[5-Bromo-4-[[2-methyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(C)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(CCC3=CC(F)=C(C4CCC(=O)NC4=O)C(F)=C3)CC2)CC1	C49H57BrF2N9O4P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-RU80F8	SCHEMBL27207258	3-[4-[3-[4-[1-[4-[[5-Bromo-4-[[2-methyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazine-1-carbonyl]azetidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(C)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(C(=O)C3CN(C4=CC(F)=C(C5CCC(=O)NC5=O)C(F)=C4)C3)CC2)CC1	C51H58BrF2N10O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-V4APH8	SCHEMBL27207450	3-[4-[(3R)-3-[4-[1-[4-[[5-bromo-4-[[2-methyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazine-1-carbonyl]pyrrolidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(C)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(C(=O)[C@@H]3CCN(C4=CC(F)=C(C5CCC(=O)NC5=O)C(F)=C4)C3)CC2)CC1	C52H60BrF2N10O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-KKPM9X	WO2022228556A1_78	3-[4-[(4R)-4-[4-[1-[4-[[5-bromo-4-[[2-methyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazine-1-carbonyl]-3,3-dimethylpyrrolidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(C)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(C(=O)[C@H]3CN(C4=CC(F)=C(C5CCC(=O)NC5=O)C(F)=C4)CC3(C)C)CC2)CC1	C54H64BrF2N10O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-ZPCHEI	WO2022228556A1_79	3-[7-[3-[4-[1-[4-[[5-Bromo-4-[[2-methyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazine-1-carbonyl]azetidin-1-yl]-1-methylindazol-3-yl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(C)C=C4)=N2)C=C(C)C(N2CCC(N3CCN(C(=O)C4CN(C5=CC=CC6=C5N(C)N=C6C5CCC(=O)NC5=O)C4)CC3)CC2)=C1	C52H60BrN12O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-6YK6DB	WO2022228556A1_8	3-[4-[2-[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-ethoxy-2-ethylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-3,3-dimethyl-2-oxoindol-1-yl]piperidine-2,6-dione	CCOC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)C=C(CC)C(N2CCC(N3CCN(CCC4=CC=CC5=C4C(C)(C)C(=O)N5C4CCC(=O)NC4=O)CC3)CC2)=C1	C55H68BrN10O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-O0HSV1	WO2022228556A1_80	3-[4-[2-[4-[1-[4-[[5-Bromo-4-[[2-methyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-3-cyclopropyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(C)C=C4)=N2)C=C(C)C(N2CCC(N3CCN(CCC4=CC=CC5=C4N(C4CC4)C(=O)N5C4CCC(=O)NC4=O)CC3)CC2)=C1	C52H61BrN11O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-O4K1TH	WO2022228556A1_81	3-[4-[2-[4-[1-[4-[[5-Bromo-4-[[2-methyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(C)C=C4)=N2)C=C(C)C(N2CCC(N3CCN(CCC4=CC=CC5=C4N(C)C(=O)N5C4CCC(=O)NC4=O)CC3)CC2)=C1	C50H59BrN11O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-9VB911	WO2022228556A1_82	3-[4-[2-[4-[1-[4-[[5-Bromo-4-[[2-methyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-3-ethyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	CCN1C(=O)N(C2CCC(=O)NC2=O)C2=C1C(CCN1CCN(C3CCN(C4=CC(OC)=C(NC5=NC=C(Br)C(NC6=C(P7(=O)CCCC7)C7=C(C=C6)N=C(C)C=C7)=N5)C=C4C)CC3)CC1)=CC=C2	C51H61BrN11O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-QPA1KT	WO2022228556A1_83	3-[7-[2-[4-[1-[4-[[5-Bromo-4-[[2-methyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2-oxo-1,3-benzoxazol-3-yl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(C)C=C4)=N2)C=C(C)C(N2CCC(N3CCN(CCC4=CC=CC5=C4OC(=O)N5C4CCC(=O)NC4=O)CC3)CC2)=C1	C49H56BrN10O6P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-0LVU4I	WO2022228556A1_84	3-[6-[2-[4-[1-[4-[[5-Bromo-4-[[2-methyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2-oxo-1,3-benzoxazol-3-yl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(C)C=C4)=N2)C=C(C)C(N2CCC(N3CCN(CCC4=CC5=C(C=C4)N(C4CCC(=O)NC4=O)C(=O)O5)CC3)CC2)=C1	C49H56BrN10O6P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-6TUVKV	WO2022228556A1_85	3-[5-[2-[4-[1-[4-[[5-Bromo-4-[[2-methyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-3,3-dimethyl-2-oxoindol-1-yl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(C)C=C4)=N2)C=C(C)C(N2CCC(N3CCN(CCC4=CC5=C(C=C4)N(C4CCC(=O)NC4=O)C(=O)C5(C)C)CC3)CC2)=C1	C52H62BrN10O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-VII2AT	WO2022228556A1_86	3-[4-[2-[4-[1-[4-[[5-Bromo-4-[[2-methyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-3,3-dimethyl-2-oxoindol-1-yl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(C)C=C4)=N2)C=C(C)C(N2CCC(N3CCN(CCC4=CC=CC5=C4C(C)(C)C(=O)N5C4CCC(=O)NC4=O)CC3)CC2)=C1	C52H62BrN10O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-DC35JW	WO2022228556A1_87	3-[4'-[2-[4-[1-[4-[[5-Bromo-4-[[2-methyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2'-oxospiro[cyclopropane-1,3'-indole]-1'-yl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(C)C=C4)=N2)C=C(C)C(N2CCC(N3CCN(CCC4=CC=CC5=C4C4(CC4)C(=O)N5C4CCC(=O)NC4=O)CC3)CC2)=C1	C52H60BrN10O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-WCCD9O	WO2022228556A1_88	3-[4-[2-[4-[1-[4-[[5-Bromo-4-[[2-methyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2,6-difluorophenyl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(C)C=C4)=N2)C=C(C)C(N2CCC(N3CCN(CCC4=CC(F)=C(C5CCC(=O)NC5=O)C(F)=C4)CC3)CC2)=C1	C48H55BrF2N9O4P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-8UX7JW	WO2022228556A1_89	3-[4-[3-[4-[1-[4-[[5-Bromo-4-[[2-methyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazine-1-carbonyl]azetidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(C)C=C4)=N2)C=C(C)C(N2CCC(N3CCN(C(=O)C4CN(C5=CC(F)=C(C6CCC(=O)NC6=O)C(F)=C5)C4)CC3)CC2)=C1	C50H56BrF2N10O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-C8BIUV	WO2022228556A1_9	3-[4'-[2-[4-[1-[4-[[5-Bromo-4-[[2-ethyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-ethoxy-2-ethylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2'-oxospiro[cyclopropane-1,3'-indole]-1'-yl]piperidine-2,6-dione	CCOC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(CC)C=C4)=N2)C=C(CC)C(N2CCC(N3CCN(CCC4=CC=CC5=C4C4(CC4)C(=O)N5C4CCC(=O)NC4=O)CC3)CC2)=C1	C55H66BrN10O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-G7VFB6	WO2022228556A1_90	3-[4-[(3R)-3-[4-[1-[4-[[5-bromo-4-[[2-methyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazine-1-carbonyl]pyrrolidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(C)C=C4)=N2)C=C(C)C(N2CCC(N3CCN(C(=O)[C@@H]4CCN(C5=CC(F)=C(C6CCC(=O)NC6=O)C(F)=C5)C4)CC3)CC2)=C1	C51H58BrF2N10O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-3W2OSH	WO2022228556A1_91	3-[4-[(4R)-4-[4-[1-[4-[[5-bromo-4-[[2-methyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazine-1-carbonyl]-3,3-dimethylpyrrolidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(C)C=C4)=N2)C=C(C)C(N2CCC(N3CCN(C(=O)[C@H]4CN(C5=CC(F)=C(C6CCC(=O)NC6=O)C(F)=C5)CC4(C)C)CC3)CC2)=C1	C53H62BrF2N10O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-KPW5AE	WO2022228556A1_92	.	CCOC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(C)C=C4)N2)C=C(C)C(N2CCC(N3CCN(C(=O)C4CN(C5=CC=CC6=C5N(C)N=C6C5CCC(=O)NC5=O)C4)CC3)CC2)=C1	C53H64BrN12O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-JOW9GO	WO2022228556A1_93	3-[4-[2-[4-[1-[4-[[5-Bromo-4-[[2-methyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-ethoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-3-cyclopropyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	CCOC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(C)C=C4)=N2)C=C(C)C(N2CCC(N3CCN(CCC4=CC=CC5=C4N(C4CC4)C(=O)N5C4CCC(=O)NC4=O)CC3)CC2)=C1	C53H63BrN11O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-0T2AVT	WO2022228556A1_94	3-[4-[2-[4-[1-[4-[[5-Bromo-4-[[2-methyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-ethoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	CCOC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(C)C=C4)=N2)C=C(C)C(N2CCC(N3CCN(CCC4=CC=CC5=C4N(C)C(=O)N5C4CCC(=O)NC4=O)CC3)CC2)=C1	C51H61BrN11O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-5XU73Z	WO2022228556A1_95	3-[4-[2-[4-[1-[4-[[5-Bromo-4-[[2-methyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-ethoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-3-ethyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	CCOC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(C)C=C4)=N2)C=C(C)C(N2CCC(N3CCN(CCC4=CC=CC5=C4N(CC)C(=O)N5C4CCC(=O)NC4=O)CC3)CC2)=C1	C52H63BrN11O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-O5H22X	WO2022228556A1_96	3-[7-[2-[4-[1-[4-[[5-Bromo-4-[[2-methyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-ethoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2-oxo-1,3-benzoxazol-3-yl]piperidine-2,6-dione	CCOC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(C)C=C4)=N2)C=C(C)C(N2CCC(N3CCN(CCC4=CC=CC5=C4OC(=O)N5C4CCC(=O)NC4=O)CC3)CC2)=C1	C50H58BrN10O6P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-SW3Z0N	WO2022228556A1_97	3-[6-[2-[4-[1-[4-[[5-Bromo-4-[[2-methyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-ethoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-2-oxo-1,3-benzoxazol-3-yl]piperidine-2,6-dione	CCOC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(C)C=C4)=N2)C=C(C)C(N2CCC(N3CCN(CCC4=CC5=C(C=C4)N(C4CCC(=O)NC4=O)C(=O)O5)CC3)CC2)=C1	C50H58BrN10O6P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-7Z20HT	WO2022228556A1_98	3-[5-[2-[4-[1-[4-[[5-Bromo-4-[[2-methyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-ethoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-3,3-dimethyl-2-oxoindol-1-yl]piperidine-2,6-dione	CCOC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(C)C=C4)=N2)C=C(C)C(N2CCC(N3CCN(CCC4=CC5=C(C=C4)N(C4CCC(=O)NC4=O)C(=O)C5(C)C)CC3)CC2)=C1	C53H64BrN10O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-WSEEC6	WO2022228556A1_99	3-[4-[2-[4-[1-[4-[[5-Bromo-4-[[2-methyl-5-(1-oxo-1lambda5-phospholan-1-yl)quinolin-6-yl]amino]pyrimidin-2-yl]amino]-5-ethoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]ethyl]-3,3-dimethyl-2-oxoindol-1-yl]piperidine-2,6-dione	CCOC1=C(NC2=NC=C(Br)C(NC3=C(P4(=O)CCCC4)C4=C(C=C3)N=C(C)C=C4)=N2)C=C(C)C(N2CCC(N3CCN(CCC4=CC=CC5=C4C(C)(C)C(=O)N5C4CCC(=O)NC4=O)CC3)CC2)=C1	C53H64BrN10O5P	EGFR	P00533	CRBN	WO-2022228556-A1
TPD-B8SZAR	SCHEMBL30273908	3-(Carboxymethoxy)-4-chloro-5-[3-[[1-[[3-[6-[4-[[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]methyl]triazol-1-yl]hexanoylamino]phenyl]methylsulfonyl]piperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	O=C(O)COC1=C(C(=O)O)SC(C2=CC(NC3CCN(S(=O)(=O)CC4=CC(NC(=O)CCCCCN5C=C(CNC6=CC=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7=O)N=N5)=CC=C4)CC3)=CC=C2)=C1Cl	C47H48ClN9O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-7F2Q3H	WO2023019166A1_10	.	O=C(O)COC1=C(C(=O)O)SC(C2=CC(NC3CCN(S(=O)(=O)CC4=CC(NC(=O)CCCCCCNC(=O)COC5=C6CN(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)CC=C4)CC3)=CC=C2)=C1Cl	C47H53ClN6O13S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-IPUAA8	WO2023019166A1_100	.	C=C1C2=CC=CC(OCC(=O)N3CC4CC(C(=O)NC5=CC=CC(CS(=O)(=O)N6CC[C@H](NC7=CC=CC(C8=C(Cl)C(OCC(=O)O)=C(C(=O)O)S8)=C7)CC6(C)C)=C5)CC4C3)=C2CN1C1CCC(=O)NC1=O	C51H55ClN6O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-FSHAMS	SCHEMBL25036901	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[(1S,5R)-3-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]oxy]acetyl]-3-azabicyclo[3.1.0]hexane-6-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid; SCHEMBL30273997	[H][C@@]12CN(C(=O)COC3=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)C[C@]1([H])[C@H]2C(=O)NC1=CC=CC(CS(=O)(=O)N2CC[C@H](NC3=CC=CC(C4=C(Cl)C(OCC(=O)O)=C(C(=O)O)S4)=C3)CC2(C)C)=C1	C48H49ClN6O13S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-COY0XE	SCHEMBL25036722	3-(Carboxymethoxy)-4-chloro-5-[3-[[1-[[3-[[7-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]-2,7-diazaspiro[3.5]nonane-2-carbonyl]amino]phenyl]methylsulfonyl]piperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid; SCHEMBL30273903	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(N3CCC4(CC3)CN(C(=O)NC3=CC=CC(CS(=O)(=O)N5CCC(NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC5)=C3)C4)C=C21	C46H49ClN8O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-QV7G4Z	SCHEMBL25034863	3-(Carboxymethoxy)-4-chloro-5-[3-[1-[[3-[[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidine-1-carbonyl]amino]phenyl]methylsulfonyl]piperidin-4-yl]oxyphenyl]thiophene-2-carboxylic acid	CN1C(=O)N(C2CCC(=O)NC2=O)C2=C1C=C(C1CCN(C(=O)NC3=CC=CC(CS(=O)(=O)N4CCC(OC5=CC=CC(C6=C(Cl)C(OCC(=O)O)=C(C(=O)O)S6)=C5)CC4)=C3)CC1)C=C2	C44H45ClN6O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-G8JW1B	SCHEMBL25036267	3-(Carboxymethoxy)-4-chloro-5-[3-[[1-[[3-[[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidine-1-carbonyl]amino]-4-fluorophenyl]methylsulfonyl]piperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid; SCHEMBL30273610	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(C3CCN(C(=O)NC4=C(F)C=CC(CS(=O)(=O)N5CCC(NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC5)=C4)CC3)C=C21	C44H45ClFN7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-FSGAAA	SCHEMBL30273568	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[2-[1-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidin-4-yl]oxyacetyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(N3CCC(OCC(=O)NC4=CC=CC(CS(=O)(=O)N5CC[C@H](NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC5(C)C)=C4)CC3)C=C21	C47H52ClN7O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-ZNY9FU	SCHEMBL25036707	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[3-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]azetidine-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid; SCHEMBL30273708	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(C3CN(C(=O)NC4=CC=CC(CS(=O)(=O)N5CC[C@H](NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC5(C)C)=C4)C3)C=C21	C44H46ClN7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-58V79E	WO2023019166A1_107	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2CC=C(N3CC(OCC(=O)NC4=CC=CC(CS(=O)(=O)N5CC[C@H](NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC5(C)C)=C4)C3)C=C21	C45H50ClN7O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-T53LKM	WO2023019166A1_108	.	CC1(C)CC(NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)C2CN(C(=O)CNC3=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)C2)=C(F)C=C1	C46H47ClFN7O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-V55QLX	WO2023019166A1_109	.	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NCC2CN(C(=O)CNC3=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)C2)=C(F)C=C1	C46H51ClFN7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-ZOHIGC	SCHEMBL25036374	3-(carboxymethoxy)-4-chloro-5-[3-[[1-[[3-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]oxy]acetyl]amino]phenyl]methylsulfonyl]piperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	O=C(O)COC1=C(C(=O)O)SC(C2=CC(NC3CCN(S(=O)(=O)CC4=CC(NC(=O)COC5=C6CN(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)=CC=C4)CC3)=CC=C2)=C1Cl	C40H38ClN5O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-DPXOQR	SCHEMBL30273571	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[(1S,5R)-3-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]acetyl]-3-azabicyclo[3.1.0]hexane-6-carbonyl]amino]-4-fluorophenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	[H][C@@]12CN(C(=O)CNC3=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)C[C@]1([H])[C@H]2C(=O)NC1=C(F)C=CC(CS(=O)(=O)N2CC[C@H](NC3=CC=CC(C4=C(Cl)C(OCC(=O)O)=C(C(=O)O)S4)=C3)CC2(C)C)=C1	C48H49ClFN7O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-4B5QAM	WO2023019166A1_111	.	[H][C@@]12CN(C(=O)CNC3=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)C[C@]1([H])[C@H]2C(=O)NC1=C(F)C=CC(CS(=O)(=O)N2CCC(NC3=CC=CC(C4=C(CI)C(OCC(=O)O)=C(C(=O)O)S4)=C3)CC2(C)C)=C1	C49H51FIN7O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-KPXGSI	SCHEMBL25036182	3-(Carboxymethoxy)-4-chloro-5-[3-[[1-[[3-[[1-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidine-4-carbonyl]amino]phenyl]methylsulfonyl]piperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid; SCHEMBL30273639	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(N3CCC(C(=O)NC4=CC=CC(CS(=O)(=O)N5CCC(NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC5)=C4)CC3)C=C21	C44H46ClN7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-XDIOMU	SCHEMBL25036179	3-(Carboxymethoxy)-4-chloro-5-[3-[[1-[[3-[[2-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]-2,7-diazaspiro[3.5]nonane-7-carbonyl]amino]phenyl]methylsulfonyl]piperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid; SCHEMBL30273738	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(N3CC4(CCN(C(=O)NC5=CC=CC(CS(=O)(=O)N6CCC(NC7=CC=CC(C8=C(Cl)C(OCC(=O)O)=C(C(=O)O)S8)=C7)CC6)=C5)CC4)C3)C=C21	C46H49ClN8O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-18JPBZ	SCHEMBL25036181	3-(Carboxymethoxy)-4-chloro-5-[3-[[1-[[3-[[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidine-1-carbonyl]amino]-4-fluorophenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid; SCHEMBL30273681	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(C3CCN(C(=O)NC4=C(F)C=CC(CS(=O)(=O)N5CCC(NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC5(C)C)=C4)CC3)C=C21	C46H49ClFN7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-9JSBKN	SCHEMBL25034723	3-(Carboxymethoxy)-4-chloro-5-[3-[[1-[[3-[[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidine-1-carbonyl]amino]-2-fluorophenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid; SCHEMBL30273730	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(C3CCN(C(=O)NC4=CC=CC(CS(=O)(=O)N5CCC(NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC5(C)C)=C4F)CC3)C=C21	C46H49ClFN7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-2O602B	SCHEMBL30274111	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[3-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]oxyazetidine-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(OC3CN(C(=O)NC4=CC=CC(CS(=O)(=O)N5CC[C@H](NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC5(C)C)=C4)C3)C=C21	C44H46ClN7O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-KA5J0V	SCHEMBL25034727	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[1-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidin-4-yl]oxycarbonylamino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid; SCHEMBL30273790	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(N3CCC(OC(=O)NC4=CC=CC(CS(=O)(=O)N5CC[C@H](NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC5(C)C)=C4)CC3)C=C21	C46H50ClN7O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-ART7J8	WO2023019166A1_118	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(OC3CCN(C(=O)NC4=CC=CC(CS(=O)(=O)N5CC[C@H](NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)C6)CC5(C)C)=C4)CC3)C=C21	C46H52ClN7O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-1GHAH7	SCHEMBL25034730	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidine-1-carbonyl]amino]-4-fluorophenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid; SCHEMBL30274103	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(C3CCN(C(=O)NC4=C(F)C=CC(CS(=O)(=O)N5CC[C@H](NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC5(C)C)=C4)CC3)C=C21	C46H49ClFN7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-MJGZMZ	SCHEMBL30274145	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[6-[4-[[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]methyl]triazol-1-yl]hexanoylamino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC1(C)C[C@@H](NC2=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=CC=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)CCCCCN2C=C(CNC3=CC=CC4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)N=N2)=CC=C1	C49H52ClN9O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-HCCHK2	SCHEMBL25036519	3-(carboxymethoxy)-4-chloro-5-[3-[[(4R)-1-[[3-[[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidine-1-carbonyl]amino]-4-fluorophenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid; SCHEMBL30273996	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(C3CCN(C(=O)NC4=C(F)C=CC(CS(=O)(=O)N5CC[C@@H](NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC5(C)C)=C4)CC3)C=C21	C46H49ClFN7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-S9193P	SCHEMBL25036332	3-(Carboxymethoxy)-4-chloro-5-[3-[[1-[[3-[[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidine-1-carbonyl]amino]phenyl]methylsulfonyl]piperidin-4-yl]amino]-4-fluorophenyl]thiophene-2-carboxylic acid	CN1C(=O)N(C2CCC(=O)NC2=O)C2=C1C=C(C1CCN(C(=O)NC3=CC=CC(CS(=O)(=O)N4CCC(NC5=C(F)C=CC(C6=C(Cl)C(OCC(=O)O)=C(C(=O)O)S6)=C5)CC4)=C3)CC1)C=C2	C44H45ClFN7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-S7FPKJ	WO2023019166A1_122	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CCC(N3CCC(C(=O)NC4=CC=CC(CS(=O)(=O)N5CC[C@H](NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC5(C)C)=C4)CC3)C=C21	C46H52ClN7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-AB7NGJ	WO2023019166A1_123	.	CC1=C(C2=C(F)C(NC3CCN(S(=O)(=O)CC4=CC(NC(=O)N5CCC(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC5)=CC=C4)CC3)=CC=C2)SC(C(=O)O)=C1OCC(=O)O	C45H48FN7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-YDPLEA	SCHEMBL30273827	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[4-[3-(2,6-dioxopiperidin-3-yl)-2-oxobenzimidazol-1-yl]piperidine-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)N2CCC(N3C(=O)N(C4CCC(=O)NC4=O)C4=C3C=CC=C4)CC2)=CC=C1	C45H48ClN7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-FFLPC2	SCHEMBL25036522	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidine-1-carbonyl]amino]-2-fluorophenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid; SCHEMBL30273725	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(C3CCN(C(=O)NC4=CC=CC(CS(=O)(=O)N5CC[C@H](NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC5(C)C)=C4F)CC3)C=C21	C46H49ClFN7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-V8VFBJ	SCHEMBL30274056	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[4-[1-(2,6-dioxopiperidin-3-yl)-2-oxobenzo[cd]indol-6-yl]piperidine-1-carbonyl]amino]-4-fluorophenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)N2CCC(C3=CC=C4C5=C(C=CC=C35)C(=O)N4C3CCC(=O)NC3=O)CC2)=C(F)C=C1	C49H48ClFN6O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-1Y697Q	SCHEMBL25036734	3-(carboxymethoxy)-4-chloro-5-[3-[[(4R)-1-[[3-[[4-[1-(2,6-dioxopiperidin-3-yl)-2-oxobenzo[cd]indol-6-yl]piperidine-1-carbonyl]amino]-4-fluorophenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC1(C)C[C@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)N2CCC(C3=CC=C4C5=C(C=CC=C35)C(=O)N4C3CCC(=O)NC3=O)CC2)=C(F)C=C1	C49H48ClFN6O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-2YAFRR	SCHEMBL25036728	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[4-[1-(2,6-dioxopiperidin-3-yl)-2-oxobenzo[cd]indol-6-yl]piperidine-1-carbonyl]amino]-2-fluorophenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=C(F)C(NC(=O)N2CCC(C3=CC=C4C5=C(C=CC=C35)C(=O)N4C3CCC(=O)NC3=O)CC2)=CC=C1	C49H48ClFN6O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-ICWSCX	SCHEMBL30273860	3-(carboxymethoxy)-4-chloro-5-[3-[[(4R)-1-[[3-[[4-[1-(2,6-dioxopiperidin-3-yl)-2-oxobenzo[cd]indol-6-yl]piperidine-1-carbonyl]amino]-2-fluorophenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC1(C)C[C@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=C(F)C(NC(=O)N2CCC(C3=CC=C4C5=C(C=CC=C35)C(=O)N4C3CCC(=O)NC3=O)CC2)=CC=C1	C49H48ClFN6O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-5OG2V9	WO2023019166A1_13	.	CC1(C)C[C@@H](NC2=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=CC=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)CCN2C=C(CNC3=CC=CC4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)N=N2)=CC=C1	C46H46ClN9O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-ISWBMQ	SCHEMBL30274173	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[2-[4-[3-(2,6-dioxopiperidin-3-yl)-2-oxobenzimidazol-1-yl]piperidin-1-yl]acetyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)CN2CCC(N3C(=O)N(C4CCC(=O)NC4=O)C4=C3C=CC=C4)CC2)=CC=C1	C46H50ClN7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-WS5XOD	SCHEMBL25036729	3-(carboxymethoxy)-4-chloro-5-[3-[[(4R)-1-[[3-[[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidine-1-carbonyl]amino]-2-fluorophenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid; SCHEMBL30273518	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(C3CCN(C(=O)NC4=CC=CC(CS(=O)(=O)N5CC[C@@H](NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC5(C)C)=C4F)CC3)C=C21	C46H49ClFN7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-BSOC53	SCHEMBL25036733	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidine-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]-4-fluorophenyl]thiophene-2-carboxylic acid	CN1C(=O)N(C2CCC(=O)NC2=O)C2=C1C=C(C1CCN(C(=O)NC3=CC=CC(CS(=O)(=O)N4CC[C@H](NC5=C(F)C=CC(C6=C(Cl)C(OCC(=O)O)=C(C(=O)O)S6)=C5)CC4(C)C)=C3)CC1)C=C2	C46H49ClFN7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-QVPWON	SCHEMBL30274097	3-(carboxymethoxy)-4-chloro-5-[3-[[(4R)-1-[[3-[[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidine-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]-4-fluorophenyl]thiophene-2-carboxylic acid	CN1C(=O)N(C2CCC(=O)NC2=O)C2=C1C=C(C1CCN(C(=O)NC3=CC=CC(CS(=O)(=O)N4CC[C@@H](NC5=C(F)C=CC(C6=C(Cl)C(OCC(=O)O)=C(C(=O)O)S6)=C5)CC4(C)C)=C3)CC1)C=C2	C46H49ClFN7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-ZUG0G1	WO2023019166A1_134	.	CC1=C(C2=C(F)C(N[C@H]3CCN(S(=O)(=O)CC4=CC(NC(=O)N5CCC(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC5)=CC=C4)C(C)(C)C3)=CC=C2)SC(C(=O)O)=C1OCC(=O)O	C47H52FN7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-VD2F3H	SCHEMBL30273835	3-(carboxymethoxy)-4-chloro-5-[3-[[(4R)-1-[[3-[[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidine-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]-2-fluorophenyl]thiophene-2-carboxylic acid	CN1C(=O)N(C2CCC(=O)NC2=O)C2=C1C=C(C1CCN(C(=O)NC3=CC=CC(CS(=O)(=O)N4CC[C@@H](NC5=CC=CC(C6=C(Cl)C(OCC(=O)O)=C(C(=O)O)S6)=C5F)CC4(C)C)=C3)CC1)C=C2	C46H49ClFN7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-KEHVGZ	SCHEMBL30273728	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[1-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]azetidin-3-yl]oxycarbonylamino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(N3CC(OC(=O)NC4=CC=CC(CS(=O)(=O)N5CC[C@H](NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC5(C)C)=C4)C3)C=C21	C44H46ClN7O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-MNP6WP	WO2023019166A1_137	.	CC(C)N1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(C3CCN(C(=O)NC4=CC=CC(CS(=O)(=O)N5CCC(NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC5(C)C)=C4)CC3)C=C21	C48H54ClN7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-Q6RAZX	WO2023019166A1_138	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C([C@H]3CC[C@H](C(=O)NC4=CC=CC(CS(=O)(=O)N5CC[C@H](NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC5(C)C)=C4)CC3)C=C21	C47H51ClN6O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-HLEJFR	WO2023019166A1_139	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C([C@H]3CC[C@@H](C(=O)NC4=CC=CC(CS(=O)(=O)N5CC[C@H](NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC5(C)C)=C4)CC3)C=C21	C47H51ClN6O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-WMT28W	SCHEMBL30274197	3-(carboxymethoxy)-4-chloro-5-[3-[[(4R)-1-[[3-[3-[4-[[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]methyl]triazol-1-yl]propanoylamino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC1(C)C[C@H](NC2=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=CC=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)CCN2C=C(CNC3=CC=CC4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)N=N2)=CC=C1	C46H46ClN9O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-L90HKM	WO2023019166A1_140	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=C1C=C(N1CC3(CN(C(=O)NC4=CC=CC(CS(=O)(=O)N5CCC(NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC5(C)C)=C4)C3)C1)C=C2	C46H49ClN8O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-8LGZGO	SCHEMBL30274137	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[8-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]-2,8-diazaspiro[3.5]nonane-2-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CN1C(=O)N(C2CCC(=O)NC2=O)C2=C1C=C(N1CCCC3(CN(C(=O)NC4=CC=CC(CS(=O)(=O)N5CC[C@H](NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC5(C)C)=C4)C3)C1)C=C2	C48H53ClN8O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-GG0OCS	WO2023019166A1_142	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=C1C=C(N1CCC(N3CCN(C4C=C(CS(=O)(=O)N5CCC(NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC5)C=CC4)C3=O)CC1)C=C2	C46H51ClN8O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-3ZC6KU	SCHEMBL25036685	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[4-[3-(2,6-dioxopiperidin-3-yl)-1-methylindazol-6-yl]piperidine-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid; SCHEMBL30273985	CN1N=C(C2CCC(=O)NC2=O)C2=C1C=C(C1CCN(C(=O)NC3=CC=CC(CS(=O)(=O)N4CC[C@H](NC5=CC=CC(C6=C(Cl)C(OCC(=O)O)=C(C(=O)O)S6)=C5)CC4(C)C)=C3)CC1)C=C2	C46H50ClN7O10S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-C4NCLA	SCHEMBL30273858	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[4-[[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]amino]benzoyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(NC3=CC=C(C(=O)NC4=CC=CC(CS(=O)(=O)N5CC[C@H](NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC5(C)C)=C4)C=C3)C=C21	C47H46ClN7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-137929	SCHEMBL30273557	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]phenyl]carbamoylamino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(C3=CC=C(NC(=O)NC4=CC=CC(CS(=O)(=O)N5CC[C@H](NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC5(C)C)=C4)C=C3)C=C21	C47H46ClN7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-6Y8EDL	WO2023019166A1_146	.	CC1(C)CC(NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2F)CCN1S(=O)(=O)CC1=CC(NC(=O)C2CN(C(=O)CNC3=C4CN(C5CCC(=O)NC5=O)CC4=CC=C3)C2)=C(F)C=C1	C46H48ClF2N7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-9L0TYI	WO2023019166A1_147	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=C1C=C(C1CCN(C(=O)NC3=CC=CC(CS(=O)(=O)N4CC[C@H](NC5=CC=CC(C6=C(Cl)C(OCC(=O)O)=C(C(=O)O)S6)=C5)CC4(C)C)=C3)CC1(C)F)C=C2	C47H51ClFN7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-XSCBWH	SCHEMBL25037042	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[1-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]acetyl]azetidine-3-carbonyl]amino]-4-fluorophenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]-2-fluorophenyl]thiophene-2-carboxylic acid	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2F)CCN1S(=O)(=O)CC1=CC(NC(=O)C2CN(C(=O)CNC3=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)C2)=C(F)C=C1	C46H46ClF2N7O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-O144IK	SCHEMBL25036369	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[1-[2-[[2-[(3R)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-4-yl]amino]acetyl]azetidine-3-carbonyl]amino]-4-fluorophenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]-2-fluorophenyl]thiophene-2-carboxylic acid	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2F)CCN1S(=O)(=O)CC1=CC(NC(=O)C2CN(C(=O)CNC3=C4CN([C@@H]5CCC(=O)NC5=O)C(=O)C4=CC=C3)C2)=C(F)C=C1	C46H46ClF2N7O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-DM3PPT	SCHEMBL30274161	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[1-[2-[[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-4-yl]amino]acetyl]azetidine-3-carbonyl]amino]-4-fluorophenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]-2-fluorophenyl]thiophene-2-carboxylic acid	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2F)CCN1S(=O)(=O)CC1=CC(NC(=O)C2CN(C(=O)CNC3=C4CN([C@H]5CCC(=O)NC5=O)C(=O)C4=CC=C3)C2)=C(F)C=C1	C46H46ClF2N7O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-ZHSS0U	SCHEMBL25036371	3-(carboxymethoxy)-4-chloro-5-[3-[[(4R)-1-[[3-[[1-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]acetyl]azetidine-3-carbonyl]amino]-4-fluorophenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]-2-fluorophenyl]thiophene-2-carboxylic acid	CC1(C)C[C@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2F)CCN1S(=O)(=O)CC1=CC(NC(=O)C2CN(C(=O)CNC3=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)C2)=C(F)C=C1	C46H46ClF2N7O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-G5WGO5	SCHEMBL30273793	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[3-[2-[4-[[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]methyl]triazol-1-yl]ethoxy]propanoylamino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC1(C)C[C@@H](NC2=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=CC=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)CCOCCN2C=C(CNC3=CC=CC4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)N=N2)=CC=C1	C48H50ClN9O13S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-SLF65U	SCHEMBL30273907	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[4-[1'-(2,6-dioxopiperidin-3-yl)-2'-oxospiro[cyclopropane-1,3'-indole]-5'-yl]piperidine-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)N2CCC(C3=CC4=C(C=C3)N(C3CCC(=O)NC3=O)C(=O)C43CC3)CC2)=CC=C1	C48H51ClN6O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-ES1NJR	SCHEMBL30274175	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-4-yl]oxypiperidine-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=CC(OC3CCN(C(=O)NC4=CC=CC(CS(=O)(=O)N5CC[C@H](NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC5(C)C)=C4)CC3)=C21	C46H50ClN7O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-8OC2T1	WO2023019166A1_152	.	C=S(=O)(CC1=CC(NC(=O)N2CCC(C3=CC=C4C(=C3F)N(C)C(=O)N4C3CCC(=O)NC3=O)CC2)=CC=C1)N1CC[C@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CC1(C)C	C47H51ClFN7O10S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-YY3QBQ	SCHEMBL25036547	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[4-[1-(2,6-dioxopiperidin-3-yl)-6-fluoro-3-methyl-2-oxobenzimidazol-5-yl]piperidine-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid; SCHEMBL30273541	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC(F)=C(C3CCN(C(=O)NC4=CC=CC(CS(=O)(=O)N5CC[C@H](NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC5(C)C)=C4)CC3)C=C21	C46H49ClFN7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-ZQGRGW	WO2023019166A1_154	.	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)N2CCC(C3=CCC4C(=C3)N(C3CC3)C(=O)N4C3CCC(=O)NC3=O)CC2)=CC=C1	C48H54ClN7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-W4DIMT	SCHEMBL25036933	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[4-[1-(2,6-dioxopiperidin-3-yl)-2-oxo-3-(2,2,2-trifluoroethyl)benzimidazol-5-yl]piperidine-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid; SCHEMBL30273716	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)N2CCC(C3=CC=C4C(=C3)N(CC(F)(F)F)C(=O)N4C3CCC(=O)NC3=O)CC2)=CC=C1	C47H49ClF3N7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-09N5K3	SCHEMBL25036939	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[3-[1-(2,6-dioxopiperidin-3-yl)-2-oxobenzo[cd]indol-6-yl]propylcarbamoylamino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid; SCHEMBL30274015	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)NCCCC2=CC=C3C4=C2C=CC=C4C(=O)N3C2CCC(=O)NC2=O)=CC=C1	C47H47ClN6O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-1JZS7M	SCHEMBL25036934	3-(Carboxymethoxy)-4-chloro-5-[3-[[1-[[3-[3-[3-(2,6-dioxopiperidin-3-yl)-1-methylindazol-6-yl]propanoylamino]phenyl]methylsulfonyl]piperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CN1N=C(C2CCC(=O)NC2=O)C2=CC=C(CCC(=O)NC3=CC=CC(CS(=O)(=O)N4CCC(NC5=CC=CC(C6=C(Cl)C(OCC(=O)O)=C(C(=O)O)S6)=C5)CC4)=C3)C=C21	C41H41ClN6O10S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-6R7W3K	WO2023019166A1_158	.	CC1(C)CC(NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)N2CCC(CC3=C4C=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=C54)C=C3)CC2)=CC=C1	C50H51ClN6O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-IGJCWM	SCHEMBL25036387	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[4-[1-(2,6-dioxopiperidin-3-yl)-3-(oxan-4-yl)-2-oxobenzimidazol-5-yl]piperidine-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid; SCHEMBL30273583	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)N2CCC(C3=CC=C4C(=C3)N(C3CCOCC3)C(=O)N4C3CCC(=O)NC3=O)CC2)=CC=C1	C50H56ClN7O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-WHILSA	WO2023019166A1_16	.	CC1=C(C2=CC(NC3CCN(S(=O)(=O)CC4=CC=CC(NC(=O)C5CCN(C(=O)CNC6=CC=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)=C4)CC3)=CC=C2)SC(C(=O)O)=C1OCC(=O)O	C47H49N7O13S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-ON825G	SCHEMBL25036390	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[4-[1-(2,6-dioxopiperidin-3-yl)-3-(2-methoxyethyl)-2-oxobenzimidazol-5-yl]piperidine-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	COCCN1C(=O)N(C2CCC(=O)NC2=O)C2=C1C=C(C1CCN(C(=O)NC3=CC=CC(CS(=O)(=O)N4CC[C@H](NC5=CC=CC(C6=C(Cl)C(OCC(=O)O)=C(C(=O)O)S6)=C5)CC4(C)C)=C3)CC1)C=C2	C48H54ClN7O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-2W5WXD	WO2023019166A1_161	.	CC1=C(C2=CC(N[C@H]3CCN(S(=O)(=O)CC4=CC(NC(=O)N5CCC(C6=CC=C7C8=C(C=CC=C68)C(=O)N7C6CCC(=O)NC6=O)CC5)=CC=C4F)C(C)(C)C3)=CC=C2)SC(C(=O)O)=C1OCC(=O)O	C50H51FN6O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-A62SN6	SCHEMBL30274081	3-(carboxymethoxy)-4-chloro-5-[3-[[(4R)-1-[[5-[[4-[1-(2,6-dioxopiperidin-3-yl)-2-oxobenzo[cd]indol-6-yl]piperidine-1-carbonyl]amino]-2-fluorophenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC1(C)C[C@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)N2CCC(C3=CC=C4C5=C(C=CC=C35)C(=O)N4C3CCC(=O)NC3=O)CC2)=CC=C1F	C49H48ClFN6O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-4T0KB0	SCHEMBL30273560	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[4-[1-(2,6-dioxopiperidin-3-yl)-2-oxobenzo[cd]indol-6-yl]-1,4-diazepane-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)N2CCCN(C3=CC=C4C5=C(C=CC=C35)C(=O)N4C3CCC(=O)NC3=O)CC2)=CC=C1	C49H50ClN7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-F5D9QE	SCHEMBL30274057	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[4-[1-(2,6-dioxopiperidin-3-yl)-2-oxobenzo[cd]indol-5-yl]-1,4-diazepane-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC=CC(NC(=O)N2CCCN(C3=C4C=CC=C5C4=C(C=C3)C(=O)N5C3CCC(=O)NC3=O)CC2)=C1	C49H50ClN7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-MQSJFU	WO2023019166A1_165	.	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)[C@H]2CC[C@H](C3=CC=C4C5=C(C=CC=C53)C(=O)N4C3CCC(=O)NC3=O)CC2)=CC=C1	C50H50ClN5O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-9O3JM8	WO2023019166A1_166	.	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)[C@H]2CC[C@@H](C3=CC=C4C5=C(C=CC=C53)C(=O)N4C3CCC(=O)NC3=O)CC2)=CC=C1	C50H50ClN5O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-HH9M6F	SCHEMBL30273845	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[4-[1-(2,6-dioxopiperidin-3-yl)-2-oxobenzo[cd]indol-6-yl]piperidine-1-carbonyl]amino]-4-fluorophenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]-2-fluorophenyl]thiophene-2-carboxylic acid	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2F)CCN1S(=O)(=O)CC1=CC(NC(=O)N2CCC(C3=CC=C4C5=C(C=CC=C35)C(=O)N4C3CCC(=O)NC3=O)CC2)=C(F)C=C1	C49H47ClF2N6O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-UT548M	SCHEMBL25036388	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[(4R)-4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]-3,3-difluoropiperidine-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid; SCHEMBL30274138	CN1C(=O)N(C2CCC(=O)NC2=O)C2=C1C=C([C@H]1CCN(C(=O)NC3=CC=CC(CS(=O)(=O)N4CC[C@H](NC5=CC(C6=C(Cl)C(OCC(=O)O)=C(C(=O)O)S6)=CC=C5)CC4(C)C)=C3)CC1(F)F)C=C2	C46H48ClF2N7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-L4N329	SCHEMBL25036688	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]-3,3-difluoropiperidine-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CN1C(=O)N(C2CCC(=O)NC2=O)C2=C1C=C(C1CCN(C(=O)NC3=CC=CC(CS(=O)(=O)N4CC[C@H](NC5=CC=CC(C6=C(Cl)C(OCC(=O)O)=C(C(=O)O)S6)=C5)CC4(C)C)=C3)CC1(F)F)C=C2	C46H48ClF2N7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-A1WA5M	WO2023019166A1_169a	.	CN1C(=O)N([C@@H]2CCC(=O)NC2=O)C2=C1C=C([C@@H]1CCN(C(=O)NC3=CC=CC(CS(=O)(=O)N4CCC(NC5=CC=CC(C6=C(Cl)C(OCC(=O)O)=C(C(=O)O)S6)=C5)CC4(C)C)=C3)CC1(F)F)C=C2	C46H48ClF2N7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-NLC7L6	WO2023019166A1_169b	.	CN1C(=O)N([C@H]2CCC(=O)NC2=O)C2=C1C=C([C@@H]1CCN(C(=O)NC3=CC=CC(CS(=O)(=O)N4CCC(NC5=CC=CC(C6=C(Cl)C(OCC(=O)O)=C(C(=O)O)S6)=C5)CC4(C)C)=C3)CC1(F)F)C=C2	C46H48ClF2N7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-EMX95S	SCHEMBL30273658	3-(Carboxymethoxy)-4-chloro-5-[3-[[1-[[3-[3-[4-[[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]methyl]triazol-1-yl]propanoylamino]phenyl]methylsulfonyl]piperidin-4-yl]-methylamino]phenyl]thiophene-2-carboxylic acid	CN(C1=CC=CC(C2=C(Cl)C(OCC(=O)O)=C(C(=O)O)S2)=C1)C1CCN(S(=O)(=O)CC2=CC(NC(=O)CCN3C=C(CNC4=CC=CC5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)N=N3)=CC=C2)CC1	C45H44ClN9O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-OSYUPD	SCHEMBL30273670	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]-3-fluoropiperidine-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(C3CCN(C(=O)NC4=CC=CC(CS(=O)(=O)N5CC[C@H](NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC5(C)C)=C4)CC3F)C=C21	C46H49ClFN7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-HWOIQ9	SCHEMBL30273497	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[(3R,4R)-4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]-3-fluoropiperidine-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C([C@H]3CCN(C(=O)NC4=CC=CC(CS(=O)(=O)N5CC[C@H](NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC5(C)C)=C4)C[C@@H]3F)C=C21	C46H49ClFN7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-7A044H	WO2023019166A1_172	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(C3CCN(C(=O)NC4=CC=CC(CS(=O)(=O)N5CC[C@H](NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC5(C)C)=C4)C[C@H]3F)C=C21	C46H49ClFN7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-70ZKXM	SCHEMBL25034739	3-(Carboxymethoxy)-4-chloro-5-[3-[[1-[[3-[[4-[1-(2,6-dioxopiperidin-3-yl)-2-oxobenzo[cd]indol-6-yl]piperidine-1-carbonyl]amino]phenyl]methylsulfonyl]piperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	O=C(O)COC1=C(C(=O)O)SC(C2=CC(NC3CCN(S(=O)(=O)CC4=CC(NC(=O)N5CCC(C6=CC=C7C8=C(C=CC=C68)C(=O)N7C6CCC(=O)NC6=O)CC5)=CC=C4)CC3)=CC=C2)=C1Cl	C47H45ClN6O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-OKRNUL	SCHEMBL25037026	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[2-[1-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidin-4-yl]ethylcarbamoylamino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid; SCHEMBL30273811	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(N3CCC(CCNC(=O)NC4=CC(CS(=O)(=O)N5CC[C@H](NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC5(C)C)=CC=C4)CC3)C=C21	C48H55ClN8O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-Z3SHBJ	SCHEMBL30273643	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[4-[[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]methyl]piperidine-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CN1C(=O)N(C2CCC(=O)NC2=O)C2=C1C=C(CC1CCN(C(=O)NC3=CC=CC(CS(=O)(=O)N4CC[C@H](NC5=CC=CC(C6=C(Cl)C(OCC(=O)O)=C(C(=O)O)S6)=C5)CC4(C)C)=C3)CC1)C=C2	C47H52ClN7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-41BYAJ	SCHEMBL30274095	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[2-[4-[1-(2,6-dioxopiperidin-3-yl)-2-oxo-3-propan-2-ylbenzimidazol-5-yl]-3,3-difluoropiperidin-1-yl]acetyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC(C)N1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(C3CCN(CC(=O)NC4=CC=CC(CS(=O)(=O)N5CC[C@H](NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC5(C)C)=C4)CC3(F)F)C=C21	C49H54ClF2N7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-SCI395	SCHEMBL25036694	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[3-[1-(2,6-dioxopiperidin-3-yl)-2-oxobenzo[cd]indol-5-yl]propylcarbamoylamino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid; SCHEMBL30274100	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)NCCCC2=CC=C3C(=O)N(C4CCC(=O)NC4=O)C4=CC=CC2=C34)=CC=C1	C47H47ClN6O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-E1RZ7T	WO2023019166A1_178	.	CC1=C(C2=CC(N[C@H]3CCN(S(=O)(=O)CC4=CC(NC(=O)CC5=CC(F)=C(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)C=C5)=CC=C4)C(C)(C)C3)=CC=C2)SC(C(=O)O)=C1OCC(=O)O	C49H49FN6O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-FUPRJE	WO2023019166A1_179	.	CC1C[C@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)CC2(O)CCN(C3=CC4=C(C=C3)N(C3CCC(=O)NC3=O)C(=O)N4C)CC2)=CC=C1	C46H50ClN7O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-YUIXU6	SCHEMBL30273967	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[7-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]acetyl]amino]heptanoylamino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)CCCCCCNC(=O)CNC2=C3CN(C4CCC(=O)NC4=O)C(=O)C3=CC=C2)=CC=C1	C49H56ClN7O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-Q3Y6SG	SCHEMBL25036011	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[4-[1-(2,6-dioxopiperidin-3-yl)-2-oxobenzo[cd]indol-6-yl]-3,3-difluoropiperidine-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)N2CCC(C3=CC=C4C5=C(C=CC=C35)C(=O)N4C3CCC(=O)NC3=O)C(F)(F)C2)=CC=C1	C49H47ClF2N6O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-8TB958	SCHEMBL30273659	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[4-[1-(2,6-dioxopiperidin-3-yl)-2-oxo-3-propan-2-ylbenzimidazol-5-yl]-3,3-difluoropiperidine-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC(C)N1C(=O)N(C2CCC(=O)NC2=O)C2=C1C=C(C1CCN(C(=O)NC3=CC=CC(CS(=O)(=O)N4CC[C@H](NC5=CC=CC(C6=C(Cl)C(OCC(=O)O)=C(C(=O)O)S6)=C5)CC4(C)C)=C3)CC1(F)F)C=C2	C48H52ClF2N7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-SRLII6	SCHEMBL25036013	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[4-[3-(2,6-dioxopiperidin-3-yl)-1-methylindazol-6-yl]-3,3-difluoropiperidine-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid; SCHEMBL30274012	CN1N=C(C2CCC(=O)NC2=O)C2=C1C=C(C1CCN(C(=O)NC3=CC=CC(CS(=O)(=O)N4CC[C@H](NC5=CC=CC(C6=C(Cl)C(OCC(=O)O)=C(C(=O)O)S6)=C5)CC4(C)C)=C3)CC1(F)F)C=C2	C46H48ClF2N7O10S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-RJKROT	SCHEMBL25034713	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[2-[1-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]-4-hydroxypiperidin-4-yl]acetyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid; SCHEMBL30273632	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(N3CCC(O)(CC(=O)NC4=CC=CC(CS(=O)(=O)N5CC[C@H](NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC5(C)C)=C4)CC3)C=C21	C47H52ClN7O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-E7SFLZ	SCHEMBL25034717	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[2-[3-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]azetidin-1-yl]acetyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid; SCHEMBL30273607	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(C3CN(CC(=O)NC4=CC=CC(CS(=O)(=O)N5CC[C@H](NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC5(C)C)=C4)C3)C=C21	C45H48ClN7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-1FHHTV	SCHEMBL25034714	3-(carboxymethoxy)-4-chloro-5-[3-[[(4R)-1-[[3-[[4-[3-(2,6-dioxopiperidin-3-yl)-1-methylindazol-6-yl]-3,3-difluoropiperidine-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CN1N=C(C2CCC(=O)NC2=O)C2=CC=C(C3CCN(C(=O)NC4=CC=CC(CS(=O)(=O)N5CC[C@@H](NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC5(C)C)=C4)CC3(F)F)C=C21	C46H48ClF2N7O10S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-IEE0PG	SCHEMBL25034716	5-[3-[[(4S)-1-[[3-[[4-[3-tert-butyl-1-(2,6-dioxopiperidin-3-yl)-2-oxobenzimidazol-5-yl]piperidine-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]-3-(carboxymethoxy)-4-chlorothiophene-2-carboxylic acid; SCHEMBL30273481	CC(C)(C)N1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(C3CCN(C(=O)NC4=CC=CC(CS(=O)(=O)N5CC[C@H](NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC5(C)C)=C4)CC3)C=C21	C49H56ClN7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-CEQAWJ	SCHEMBL30274071	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[4-[1-[(3R)-2,6-dioxopiperidin-3-yl]-2-oxobenzo[cd]indol-6-yl]piperidine-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC1(C)C[C@@H](NC2=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=CC=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)N2CCC(C3=CC=C4C5=C(C=CC=C35)C(=O)N4[C@@H]3CCC(=O)NC3=O)CC2)=CC=C1	C49H49ClN6O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-BYS91D	PROTAC PTPN2 degrader-2	PROTAC PTPN2 degrader-2; 2912307-38-9; orb2278156; SCHEMBL25036361; EX-A9144; HY-153938; CS-0867624	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)N2CCC(C3=CC=C4C5=C(C=CC=C35)C(=O)N4[C@H]3CCC(=O)NC3=O)CC2)=CC=C1	C49H49ClN6O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-ONHU5V	SCHEMBL30273774	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[2-[[1-[1-(2,6-dioxopiperidin-3-yl)-2-oxobenzo[cd]indol-6-yl]piperidin-4-yl]amino]ethylamino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC=CC(NCCNC2CCN(C3=CC=C4C5=C(C=CC=C35)C(=O)N4C3CCC(=O)NC3=O)CC2)=C1	C50H54ClN7O10S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-DDAL6U	SCHEMBL30273775	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[3-[1-[1-(2,6-dioxopiperidin-3-yl)-2-oxobenzo[cd]indol-6-yl]piperidin-4-yl]-2-oxoimidazolidin-1-yl]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC=CC(N2CCN(C3CCN(C4=CC=C5C6=C(C=CC=C46)C(=O)N5C4CCC(=O)NC4=O)CC3)C2=O)=C1	C51H52ClN7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-WLY8HA	SCHEMBL25036167	3-(carboxymethoxy)-4-chloro-5-[3-[[1-[[3-[3-[2-[2-[3-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]propoxy]ethoxy]ethoxy]propanoylamino]phenyl]methylsulfonyl]piperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid; SCHEMBL30273925	O=C(O)COC1=C(C(=O)O)SC(C2=CC(NC3CCN(S(=O)(=O)CC4=CC(NC(=O)CCOCCOCCOCCCC5=CC=C6C(=O)N(C7CCC(=O)NC7=O)CC6=C5)=CC=C4)CC3)=CC=C2)=C1Cl	C48H54ClN5O14S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-L08282	SCHEMBL25034719	3-(carboxymethoxy)-4-chloro-5-[3-[[(7S)-4-[[3-[[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidine-1-carbonyl]amino]phenyl]methylsulfonyl]-4-azaspiro[2.5]octan-7-yl]amino]phenyl]thiophene-2-carboxylic acid; SCHEMBL30273722	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(C3CCN(C(=O)NC4=CC=CC(CS(=O)(=O)N5CC[C@H](NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC56CC6)=C4)CC3)C=C21	C46H48ClN7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-FMSLYZ	WO2023019166A1_191	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=C1C=C(NC1=CC=CC(CC(=O)NC3=CC=CC(CS(=O)(=O)C4CC[C@H](NC5=CC=CC(C6=C(Cl)C(OCC(=O)O)=C(C(=O)O)S6)=C5)CC4(C)C)=C3)=C1)C=C2	C49H49ClN6O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-KSH4D2	WO2023019166A1_192	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=C1C=C(C1=CC=CC(CC(=O)NC3=CC=CC(CS(=O)(=O)N4CCC(NC5=CC=CC(C6=C(Cl)C(OCC(=O)O)=C(C(=O)O)S6)=C5)CC4)=C3)=C1)C=C2	C46H43ClN6O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-HJ8EEV	SCHEMBL30273743	3-(carboxymethoxy)-4-chloro-5-[3-[[(4R)-1-[[3-[[4-[3-(2,6-dioxopiperidin-3-yl)pyrazolo[1,5-a]pyridin-6-yl]piperidine-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC1(C)C[C@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)N2CCC(C3=CN4N=CC(C5CCC(=O)NC5=O)=C4C=C3)CC2)=CC=C1	C45H48ClN7O10S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-ZD6MUO	WO2023019166A1_194	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=C1C=C(C1=CN(CC(=O)NC3=CC=CC(CS(=O)(=O)N4CC[C@H]([Ni]C5=CC=CC(C6=C(Cl)C(OCC(=O)O)=C(C(=O)O)S6)=C5)CC4(C)C)=C3)N=C1)C=C2	C45H44ClN7NiO11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-V6ASJP	SCHEMBL30274199	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[4-[9-(2,6-dioxopiperidin-3-yl)pyrido[2,3-b]indol-6-yl]piperidine-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)N2CCC(C3=CC4=C(C=C3)N(C3CCC(=O)NC3=O)C3=C4C=CC=N3)CC2)=CC=C1	C49H50ClN7O10S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-5RT5RJ	SCHEMBL25036737	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[4-[1-(2,6-dioxopiperidin-3-yl)indol-5-yl]piperidine-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)N2CCC(C3=CC4=C(C=C3)N(C3CCC(=O)NC3=O)C=C4)CC2)=CC=C1	C46H49ClN6O10S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-OL0PJD	WO2023019166A1_197	.	C=C1N(C)C2=C(C=CC(N3CCC(NCCNC4=CC=CC(CS(=O)(=O)N5CC[C@H](NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC5(C)C)=C4)CC3)=C2)N1C1CCC(=O)NC1=O	C48H57ClN8O9S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-QEZ7B5	SCHEMBL30273712	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[3-[1-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidin-4-yl]-2-oxoimidazolidin-1-yl]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CN1C(=O)N(C2CCC(=O)NC2=O)C2=C1C=C(N1CCC(N3CCN(C4=CC=CC(CS(=O)(=O)N5CC[C@H](NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC5(C)C)=C4)C3=O)CC1)C=C2	C48H53ClN8O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-6QW0FL	SCHEMBL25036511	3-(Carboxymethoxy)-4-chloro-5-[3-[[1-[[3-[3-[4-[[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]methyl]triazol-1-yl]propanoylamino]phenyl]methylsulfonyl]piperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	O=C(O)COC1=C(C(=O)O)SC(C2=CC(NC3CCN(S(=O)(=O)CC4=CC(NC(=O)CCN5C=C(CNC6=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)N=N5)=CC=C4)CC3)=CC=C2)=C1Cl	C44H42ClN9O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-GYB3ZV	SCHEMBL25036290	3-(Carboxymethoxy)-4-chloro-5-[3-[[1-[[3-[3-[2-[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]propoxy]ethoxy]propanoylamino]phenyl]methylsulfonyl]piperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	O=C(O)COC1=C(C(=O)O)SC(C2=CC(NC3CCN(S(=O)(=O)CC4=CC(NC(=O)CCOCCOCCCC5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)=CC=C4)CC3)=CC=C2)=C1Cl	C46H48ClN5O14S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-9D8LB2	SCHEMBL25036738	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[4-[3-(2,6-dioxopiperidin-3-yl)-1-ethylindazol-6-yl]-3,3-difluoropiperidine-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CCN1N=C(C2CCC(=O)NC2=O)C2=CC=C(C3CCN(C(=O)NC4=CC=CC(CS(=O)(=O)N5CC[C@H](NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC5(C)C)=C4)CC3(F)F)C=C21	C47H50ClF2N7O10S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-RDETNU	SCHEMBL30273458	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[2-[3-[1-(2,6-dioxopiperidin-3-yl)-2-oxobenzo[cd]indol-6-yl]propylamino]ethylamino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NCCNCCCC2=CC=C3C4=C2C=CC=C4C(=O)N3C2CCC(=O)NC2=O)=CC=C1	C48H51ClN6O10S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-I0YABU	SCHEMBL30273931	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[3-[3-[1-(2,6-dioxopiperidin-3-yl)-2-oxobenzo[cd]indol-6-yl]propyl]-2-oxoimidazolidin-1-yl]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(N2CCN(CCCC3=CC=C4C5=C3C=CC=C5C(=O)N4C3CCC(=O)NC3=O)C2=O)=CC=C1	C49H49ClN6O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-BIHXQU	SCHEMBL25036486	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[3-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidine-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CN1C(=O)N(C2CCC(=O)NC2=O)C2=C1C=C(C1CCCN(C(=O)NC3=CC=CC(CS(=O)(=O)N4CC[C@H](NC5=CC=CC(C6=C(Cl)C(OCC(=O)O)=C(C(=O)O)S6)=C5)CC4(C)C)=C3)C1)C=C2	C46H50ClN7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-PKZRRI	SCHEMBL30273885	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[2-[4-[1-(2,6-dioxopiperidin-3-yl)-2-oxo-3-propan-2-ylbenzimidazol-5-yl]piperidin-1-yl]acetyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC(C)N1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(C3CCN(CC(=O)NC4=CC=CC(CS(=O)(=O)N5CC[C@H](NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC5(C)C)=C4)CC3)C=C21	C49H56ClN7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-17G75I	SCHEMBL25036391	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[4-[1-(2,6-dioxopiperidin-3-yl)-2-oxobenzo[cd]indol-5-yl]piperidine-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid; SCHEMBL30274119	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)N2CCC(C3=C4C=CC=C5C4=C(C=C3)C(=O)N5C3CCC(=O)NC3=O)CC2)=CC=C1	C49H49ClN6O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-QM2C7C	SCHEMBL30273530	3-(carboxymethoxy)-4-chloro-5-[3-[[(4R)-1-[[3-[[4-[1-(2,6-dioxopiperidin-3-yl)-3-(oxetan-3-yl)-2-oxobenzimidazol-5-yl]piperidine-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC1(C)C[C@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)N2CCC(C3=CC4=C(C=C3)N(C3CCC(=O)NC3=O)C(=O)N4C3COC3)CC2)=CC=C1	C48H52ClN7O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-5FIJ63	SCHEMBL30273565	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[4-[4-chloro-1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidine-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(C3CCN(C(=O)NC4=CC(CS(=O)(=O)N5CC[C@H](NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC5(C)C)=CC=C4)CC3)C(Cl)=C21	C46H49Cl2N7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-4CKTDI	SCHEMBL25036396	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[4-[1-(2,6-dioxopiperidin-3-yl)-2-methylindol-5-yl]piperidine-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC1=CC2=C(C=CC(C3CCN(C(=O)NC4=CC=CC(CS(=O)(=O)N5CC[C@H](NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC5(C)C)=C4)CC3)=C2)N1C1CCC(=O)NC1=O	C47H51ClN6O10S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-UHZY0K	SCHEMBL25036398	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[(3R)-4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]-3-methylpiperazine-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	C[C@@H]1CN(C(=O)NC2=CC=CC(CS(=O)(=O)N3CC[C@H](NC4=CC=CC(C5=C(Cl)C(OCC(=O)O)=C(C(=O)O)S5)=C4)CC3(C)C)=C2)CCN1C1=CC2=C(C=C1)N(C1CCC(=O)NC1=O)C(=O)N2C	C46H51ClN8O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-WMEGS1	SCHEMBL25036168	3-(carboxymethoxy)-4-chloro-5-[3-[[1-[[3-[6-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]acetyl]amino]hexanoylamino]phenyl]methylsulfonyl]piperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	O=C(O)COC1=C(C(=O)O)SC(C2=CC(NC3CCN(S(=O)(=O)CC4=CC(NC(=O)CCCCCNC(=O)CNC5=C6CN(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)=CC=C4)CC3)=CC=C2)=C1Cl	C46H50ClN7O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-T6IDX9	SCHEMBL25036690	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[(3S)-4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]-3-methylpiperazine-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	C[C@H]1CN(C(=O)NC2=CC=CC(CS(=O)(=O)N3CC[C@H](NC4=CC=CC(C5=C(Cl)C(OCC(=O)O)=C(C(=O)O)S5)=C4)CC3(C)C)=C2)CCN1C1=CC2=C(C=C1)N(C1CCC(=O)NC1=O)C(=O)N2C	C46H51ClN8O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-MTP4L7	SCHEMBL30274124	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[4-[1-(2,6-dioxopiperidin-3-yl)-3-methylindol-5-yl]piperidine-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC1=CN(C2CCC(=O)NC2=O)C2=C1C=C(C1CCN(C(=O)NC3=CC=CC(CS(=O)(=O)N4CC[C@H](NC5=CC=CC(C6=C(Cl)C(OCC(=O)O)=C(C(=O)O)S6)=C5)CC4(C)C)=C3)CC1)C=C2	C47H51ClN6O10S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-LY3URD	SCHEMBL25036698	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[3-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]-4-fluoropiperidine-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid; SCHEMBL30274167	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(C3CN(C(=O)NC4=CC=CC(CS(=O)(=O)N5CC[C@H](NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC5(C)C)=C4)CCC3F)C=C21	C46H49ClFN7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-EOVUPN	WO2023019166A1_213	.	CC1=C(C2=CC(N[C@H]3CCN(S(=O)(=O)CC4=CC(NC(=O)N5CC[C@@H](F)[C@H](C6=CC=C7C(=C6)N(C)C(=O)N7C6CCC(=O)NC6=O)C5)=CC=C4)C(C)(C)C3)=CC=C2)SC(C(=O)O)=C1OCC(=O)O	C47H52FN7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-ERWAIP	SCHEMBL25036474	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[(3S,4S)-3-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]-4-fluoropiperidine-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid; SCHEMBL30273669	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C([C@H]3CN(C(=O)NC4=CC=CC(CS(=O)(=O)N5CC[C@H](NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC5(C)C)=C4)CC[C@@H]3F)C=C21	C46H49ClFN7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-9EBNQV	SCHEMBL30274083	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[3-[1-(2,6-dioxopiperidin-3-yl)-2-oxobenzo[cd]indol-4-yl]propylcarbamoylamino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)NCCCC2=CC3=C4C(=C2)C(=O)N(C2CCC(=O)NC2=O)C4=CC=C3)=CC=C1	C47H47ClN6O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-INDC9R	SCHEMBL25036472	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[1-[1-(2,6-dioxopiperidin-3-yl)-2-oxobenzo[cd]indol-5-yl]piperidine-4-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid; SCHEMBL30274036	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)C2CCN(C3=C4C=CC=C5C4=C(C=C3)C(=O)N5C3CCC(=O)NC3=O)CC2)=CC=C1	C49H49ClN6O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-R135S1	SCHEMBL25036475	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[1-[1-(2,6-dioxopiperidin-3-yl)-2-oxobenzo[cd]indol-6-yl]piperidine-4-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)C2CCN(C3=CC=C4C5=C(C=CC=C35)C(=O)N4C3CCC(=O)NC3=O)CC2)=CC=C1	C49H49ClN6O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-W5DJT3	SCHEMBL25036517	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[4-[9-(2,6-dioxopiperidin-3-yl)pyrido[2,3-b]indol-3-yl]piperidine-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)N2CCC(C3=CC4=C(N=C3)N(C3CCC(=O)NC3=O)C3=CC=CC=C34)CC2)=CC=C1	C49H50ClN7O10S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-XI6ZO1	SCHEMBL30273803	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[2-[1-[1-(2,6-dioxopiperidin-3-yl)-2-oxobenzo[cd]indol-6-yl]piperidin-4-yl]ethylcarbamoylamino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)NCCC2CCN(C3=CC=C4C5=C(C=CC=C35)C(=O)N4C3CCC(=O)NC3=O)CC2)=CC=C1	C51H54ClN7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-2LOXI5	SCHEMBL25036897	3-(carboxymethoxy)-4-chloro-5-[3-[[1-[[3-[5-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]acetyl]amino]pentanoylamino]phenyl]methylsulfonyl]piperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	O=C(O)COC1=C(C(=O)O)SC(C2=CC(NC3CCN(S(=O)(=O)CC4=CC(NC(=O)CCCCNC(=O)CNC5=C6CN(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)=CC=C4)CC3)=CC=C2)=C1Cl	C45H48ClN7O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-O0BFRL	SCHEMBL25036518	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[4-[[1-(2,6-dioxopiperidin-3-yl)-2-oxobenzo[cd]indol-6-yl]methylamino]-4-oxobutanoyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)CCC(=O)NCC2=CC=C3C4=C(C=CC=C24)C(=O)N3C2CCC(=O)NC2=O)=CC=C1	C48H47ClN6O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-9JD924	SCHEMBL30273764	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[4-[[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]methyl]piperazine-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CN1C(=O)N(C2CCC(=O)NC2=O)C2=C1C=C(CN1CCN(C(=O)NC3=CC=CC(CS(=O)(=O)N4CC[C@H](NC5=CC=CC(C6=C(Cl)C(OCC(=O)O)=C(C(=O)O)S6)=C5)CC4(C)C)=C3)CC1)C=C2	C46H51ClN8O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-7T140J	WO2023019166A1_222	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=C1C1CCCN(C3CCN(C(=O)NC4=CC=CC(CS(=O)(=O)N5CC[C@H](NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC5(C)C)=C4)CC3)C1C=C2	C49H57ClN8O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-EW7Q8V	SCHEMBL25034743	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[(4S)-4-[1-(2,6-dioxopiperidin-3-yl)-2-oxobenzo[cd]indol-5-yl]azepane-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid; SCHEMBL30274195	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)N2CCC[C@H](C3=C4C=CC=C5C4=C(C=C3)C(=O)N5C3CCC(=O)NC3=O)CC2)=CC=C1	C50H51ClN6O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-IJFKF6	SCHEMBL30274074	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[(4R)-4-[1-(2,6-dioxopiperidin-3-yl)-2-oxobenzo[cd]indol-5-yl]azepane-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)N2CCC[C@@H](C3=C4C=CC=C5C4=C(C=C3)C(=O)N5C3CCC(=O)NC3=O)CC2)=CC=C1	C50H51ClN6O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-EY7WRP	WO2023019166A1_225	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=C1C=C(C1CCN(C(=O)NC3=CC=CC(CS(=O)(=O)N4CCC(OC5=CC=CC(C6=C(Cl)C(OCC(=O)O)=C(C(=O)O)S6)=C5)CC4(C)C)=C3)CC1)C=C2	C46H49ClN6O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-LPEMGH	SCHEMBL25036663	3-(carboxymethoxy)-4-chloro-5-[3-[(4R)-1-[[3-[[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidine-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]oxyphenyl]thiophene-2-carboxylic acid	CN1C(=O)N(C2CCC(=O)NC2=O)C2=C1C=C(C1CCN(C(=O)NC3=CC=CC(CS(=O)(=O)N4CC[C@@H](OC5=CC=CC(C6=C(Cl)C(OCC(=O)O)=C(C(=O)O)S6)=C5)CC4(C)C)=C3)CC1)C=C2	C46H49ClN6O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-NYY8JI	SCHEMBL30273753	3-(carboxymethoxy)-4-chloro-5-[3-[(4R)-1-[[3-[[4-[1-(2,6-dioxopiperidin-3-yl)-2-oxobenzo[cd]indol-6-yl]piperidine-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]oxyphenyl]thiophene-2-carboxylic acid	CC1(C)C[C@H](OC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)N2CCC(C3=C4C=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=C54)C=C3)CC2)=CC=C1	C49H48ClN5O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-3SP5NG	SCHEMBL25034926	3-(carboxymethoxy)-4-chloro-5-[3-[(4S)-1-[[3-[[4-[1-(2,6-dioxopiperidin-3-yl)-2-oxobenzo[cd]indol-6-yl]piperidine-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]oxyphenyl]thiophene-2-carboxylic acid	CC1(C)C[C@@H](OC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)N2CCC(C3=C4C=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=C54)C=C3)CC2)=CC=C1	C49H48ClN5O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-C8SEZK	SCHEMBL25036732	3-(carboxymethoxy)-4-chloro-5-[3-[[(7S)-4-[[3-[[4-[1-(2,6-dioxopiperidin-3-yl)-2-oxobenzo[cd]indol-6-yl]piperidine-1-carbonyl]amino]phenyl]methylsulfonyl]-4-azaspiro[2.5]octan-7-yl]amino]phenyl]thiophene-2-carboxylic acid	O=C(O)COC1=C(C(=O)O)SC(C2=CC(N[C@H]3CCN(S(=O)(=O)CC4=CC(NC(=O)N5CCC(C6=CC=C7C8=C(C=CC=C68)C(=O)N7C6CCC(=O)NC6=O)CC5)=CC=C4)C4(CC4)C3)=CC=C2)=C1Cl	C49H47ClN6O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-RFMLOC	SCHEMBL25036898	3-(Carboxymethoxy)-4-chloro-5-[3-[[1-[[3-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]amino]acetyl]amino]phenyl]methylsulfonyl]piperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid; SCHEMBL30273994	O=C(O)COC1=C(C(=O)O)SC(C2=CC(NC3CCN(S(=O)(=O)CC4=CC(NC(=O)CNC5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)=CC=C4)CC3)=CC=C2)=C1Cl	C40H37ClN6O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-NSCB14	SCHEMBL30273841	3-(carboxymethoxy)-4-chloro-5-[3-[[(7R)-4-[[3-[[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidine-1-carbonyl]amino]phenyl]methylsulfonyl]-4-azaspiro[2.5]octan-7-yl]amino]phenyl]thiophene-2-carboxylic acid	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(C3CCN(C(=O)NC4=CC=CC(CS(=O)(=O)N5CC[C@@H](NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC56CC6)=C4)CC3)C=C21	C46H48ClN7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-LBXPHG	SCHEMBL25036719	3-(carboxymethoxy)-4-chloro-5-[3-[[(7R)-4-[[3-[[4-[1-(2,6-dioxopiperidin-3-yl)-2-oxobenzo[cd]indol-6-yl]piperidine-1-carbonyl]amino]phenyl]methylsulfonyl]-4-azaspiro[2.5]octan-7-yl]amino]phenyl]thiophene-2-carboxylic acid	O=C(O)COC1=C(C(=O)O)SC(C2=CC(N[C@@H]3CCN(S(=O)(=O)CC4=CC(NC(=O)N5CCC(C6=CC=C7C8=C(C=CC=C68)C(=O)N7C6CCC(=O)NC6=O)CC5)=CC=C4)C4(CC4)C3)=CC=C2)=C1Cl	C49H47ClN6O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-CHSW5C	SCHEMBL25036726	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[2-[1-[1-(2,6-dioxopiperidin-3-yl)-3-methylindol-5-yl]piperidin-4-yl]ethylcarbamoylamino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC1=CN(C2CCC(=O)NC2=O)C2=C1C=C(N1CCC(CCNC(=O)NC3=CC=CC(CS(=O)(=O)N4CC[C@H](NC5=CC=CC(C6=C(Cl)C(OCC(=O)O)=C(C(=O)O)S6)=C5)CC4(C)C)=C3)CC1)C=C2	C49H56ClN7O10S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-XZAVMH	SCHEMBL30273586	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[4-[1-(2,6-dioxopiperidin-3-yl)-3-methylindazol-5-yl]piperidine-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC1=NN(C2CCC(=O)NC2=O)C2=CC=C(C3CCN(C(=O)NC4=CC=CC(CS(=O)(=O)N5CC[C@H](NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC5(C)C)=C4)CC3)C=C21	C46H50ClN7O10S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-5I7TEW	SCHEMBL30273707	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[4-[1-[(3S)-2,6-dioxopiperidin-3-yl]-3-methyl-2-oxobenzimidazol-5-yl]piperidine-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	[H][C@]1(N2C(=O)N(C)C3=CC(C4CCN(C(=O)NC5=CC=CC(CS(=O)(=O)N6CC[C@H](NC7=CC=CC(C8=C(Cl)C(OCC(=O)O)=C(C(=O)O)S8)=C7)CC6(C)C)=C5)CC4)=CC=C32)CCC(=O)NC1=O	C46H50ClN7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-HHHDQE	SCHEMBL25036196	(5P)-3-(carboxymethoxy)-4-chloro-5-(3-{[(4S)-1-({3-[(4-{1-[(3R)-2,6-dioxopiperidin-3-yl]-3-methyl-2-oxo-2,3-dihydro-1H-benzimidazol-5-yl}piperidine-1-carbonyl)amino]phenyl}methanesulfonyl)-2,2-dimethylpiperidin-4-yl]amino}phenyl)thiophene-2-carboxylic acid; SCHEMBL30273950; (5P)-3-(carboxymethoxy)-4-chloro-5-(3-{[(4S)-1-({3-[(4-{1-[(3R)-2,6-dioxopiperidin-3-yl]-3-methyl-2-oxo-2,3-dihydro-1H-benzimidazol-5-yl}piperidine-1-carbonyl)amino]phenyl}methanesulfonyl)-2,2-dimethylpiperidin-4-yl]amino}phenyl)thiophene-2-carboxylic acid; WO8	[H][C@@]1(N2C(=O)N(C)C3=CC(C4CCN(C(=O)NC5=CC=CC(CS(=O)(=O)N6CC[C@H](NC7=CC=CC(C8=C(Cl)C(OCC(=O)O)=C(C(=O)O)S8)=C7)CC6(C)C)=C5)CC4)=CC=C32)CCC(=O)NC1=O	C46H50ClN7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-JN5MYH	SCHEMBL25036191	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[2-[4-[[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]methyl]phenyl]acetyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CN1C(=O)N(C2CCC(=O)NC2=O)C2=C1C=C(CC1=CC=C(CC(=O)NC3=CC=CC(CS(=O)(=O)N4CC[C@H](NC5=CC=CC(C6=C(Cl)C(OCC(=O)O)=C(C(=O)O)S6)=C5)CC4(C)C)=C3)C=C1)C=C2	C49H49ClN6O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-STM0VL	SCHEMBL30273601	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[2-[2-[1-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidin-4-yl]ethylamino]ethylamino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(N3CCC(CCNCCNC4=CC(CS(=O)(=O)N5CC[C@H](NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC5(C)C)=CC=C4)CC3)C=C21	C49H59ClN8O10S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-TB0WZ6	SCHEMBL25036199	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[3-[2-[1-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidin-4-yl]ethyl]-2-oxoimidazolidin-1-yl]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid; SCHEMBL30273634	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(N3CCC(CCN4CCN(C5=CC(CS(=O)(=O)N6CC[C@H](NC7=CC=CC(C8=C(Cl)C(OCC(=O)O)=C(C(=O)O)S8)=C7)CC6(C)C)=CC=C5)C4=O)CC3)C=C21	C50H57ClN8O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-4MQHB1	SCHEMBL30273768	3-(Carboxymethoxy)-4-chloro-5-[3-[[1-[[3-[3-[2-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]amino]acetyl]amino]ethoxy]propanoylamino]phenyl]methylsulfonyl]piperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	O=C(O)COC1=C(C(=O)O)SC(C2=CC(NC3CCN(S(=O)(=O)CC4=CC(NC(=O)CCOCCNC(=O)CNC5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)=CC=C4)CC3)=CC=C2)=C1Cl	C45H46ClN7O14S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-74J0MR	SCHEMBL30273655	3-(carboxymethoxy)-4-chloro-5-[3-[[1-[[3-[7-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]amino]acetyl]amino]heptanoylamino]phenyl]methylsulfonyl]piperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	O=C(O)COC1=C(C(=O)O)SC(C2=CC(NC3CCN(S(=O)(=O)CC4=CC(NC(=O)CCCCCCNC(=O)CNC5=CC=C6C(=O)N(C7CCC(=O)NC7=O)CC6=C5)=CC=C4)CC3)=CC=C2)=C1Cl	C47H52ClN7O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-UX6LWI	WO2023019166A1_26	.	CC(NC1=C2CN(C3CCC(=O)NC3=O)C(=O)C2=CC=C1)C(=O)NCCCCCCC(=O)NC1=CC=CC(CS(=O)(=O)N2CCC(NC3=CC=CC(C4=C(Cl)C(OCC(=O)O)C(C(=O)O)S4)=C3)CC2)=C1	C48H56ClN7O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-4IA6XG	SCHEMBL25034836	3-(Carboxymethoxy)-4-chloro-5-[3-[[1-[[3-[3-[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]propoxy]propanoylamino]phenyl]methylsulfonyl]piperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	O=C(O)COC1=C(C(=O)O)SC(C2=CC(NC3CCN(S(=O)(=O)CC4=CC(NC(=O)CCOCCCC5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)=CC=C4)CC3)=CC=C2)=C1Cl	C44H44ClN5O13S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-P065AH	SCHEMBL25036865	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[4-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]acetyl]amino]butanoylamino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)CCCNC(=O)CNC2=C3CN(C4CCC(=O)NC4=O)C(=O)C3=CC=C2)=CC=C1	C46H50ClN7O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-W0FNEU	SCHEMBL30274107	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]oxy]acetyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)COC2=C3CN(C4CCC(=O)NC4=O)C(=O)C3=CC=C2)=CC=C1	C42H42ClN5O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-T0AVFB	SCHEMBL30273726	3-(Carboxymethoxy)-4-chloro-5-[3-[[1-[[3-[3-[2-[2-[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]propoxy]ethoxy]ethoxy]propanoylamino]phenyl]methylsulfonyl]piperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	O=C(O)COC1=C(C(=O)O)SC(C2=CC(NC3CCN(S(=O)(=O)CC4=CC(NC(=O)CCOCCOCCOCCCC5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)=CC=C4)CC3)=CC=C2)=C1Cl	C48H52ClN5O15S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-X3M1X5	SCHEMBL30273877	3-(carboxymethoxy)-4-chloro-5-[3-[[1-[[3-[7-[[2-[[2-(2,6-dioxopiperidin-3-yl)-3-oxo-1H-isoindol-4-yl]amino]acetyl]amino]heptanoylamino]phenyl]methylsulfonyl]piperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	O=C(O)COC1=C(C(=O)O)SC(C2=CC(NC3CCN(S(=O)(=O)CC4=CC(NC(=O)CCCCCCNC(=O)CNC5=C6C(=O)N(C7CCC(=O)NC7=O)CC6=CC=C5)=CC=C4)CC3)=CC=C2)=C1Cl	C47H52ClN7O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-VRBYC3	SCHEMBL25036280	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[1-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]acetyl]piperidine-4-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid; SCHEMBL30273809	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC=CC(NC(=O)C2CCN(C(=O)CNC3=CC=CC4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)=C1	C48H50ClN7O13S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-J8648I	SCHEMBL25036680	3-(carboxymethoxy)-4-chloro-5-[3-[[1-[[3-[6-[4-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]piperidin-1-yl]hexanoylamino]phenyl]methylsulfonyl]piperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	O=C(O)COC1=C(C(=O)O)SC(C2=CC(NC3CCN(S(=O)(=O)CC4=CC(NC(=O)CCCCCN5CCC(NC6=C7CN(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)CC5)=CC=C4)CC3)=CC=C2)=C1Cl	C49H56ClN7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-0UPCXH	SCHEMBL25034682	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]amino]acetyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid; SCHEMBL30274147	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)CNC2=CC=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=C2)=CC=C1	C42H41ClN6O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-ZFTTMI	SCHEMBL25034680	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[3-[2-[2-[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]propoxy]ethoxy]ethoxy]propanoylamino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)CCOCCOCCOCCCC2=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=CC=C2)=CC=C1	C50H56ClN5O15S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-1CMPKV	SCHEMBL25034685	3-(carboxymethoxy)-4-chloro-5-[3-[[1-[[3-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]amino]acetyl]amino]phenyl]methylsulfonyl]piperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid; SCHEMBL30273754	O=C(O)COC1=C(C(=O)O)SC(C2=CC(NC3CCN(S(=O)(=O)CC4=CC(NC(=O)CNC5=CC=C6C(=O)N(C7CCC(=O)NC7=O)CC6=C5)=CC=C4)CC3)=CC=C2)=C1Cl	C40H39ClN6O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-F0BGIC	SCHEMBL25034683	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]amino]acetyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid; SCHEMBL30273880	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)CNC2=CC=C3C(=O)N(C4CCC(=O)NC4=O)CC3=C2)=CC=C1	C42H43ClN6O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-0EGT0K	SCHEMBL25034681	3-(carboxymethoxy)-4-chloro-5-[3-[[1-[[3-[3-[4-[[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]methyl]pyrazol-1-yl]propanoylamino]phenyl]methylsulfonyl]piperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	O=C(O)COC1=C(C(=O)O)SC(C2=CC(NC3CCN(S(=O)(=O)CC4=CC(NC(=O)CCN5C=C(CNC6=C7CN(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)C=N5)=CC=C4)CC3)=CC=C2)=C1Cl	C45H45ClN8O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-UD2L70	SCHEMBL30273859	3-(carboxymethoxy)-4-chloro-5-[3-[[1-[2-[3-[7-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]amino]acetyl]amino]heptanoylamino]phenyl]propan-2-ylsulfonyl]piperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC(C)(C1=CC(NC(=O)CCCCCCNC(=O)CNC2=CC=C3C(=O)N(C4CCC(=O)NC4=O)CC3=C2)=CC=C1)S(=O)(=O)N1CCC(NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CC1	C49H56ClN7O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-3ZJIQO	SCHEMBL25036512	3-(Carboxymethoxy)-4-chloro-5-[3-[[1-[[3-[7-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]acetyl]amino]heptanoylamino]phenyl]methylsulfonyl]piperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	O=C(O)COC1=C(C(=O)O)SC(C2=CC(NC3CCN(S(=O)(=O)CC4=CC(NC(=O)CCCCCCNC(=O)CNC5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)=CC=C4)CC3)=CC=C2)=C1Cl	C47H50ClN7O13S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-MXS40K	SCHEMBL25036699	3-(carboxymethoxy)-4-chloro-5-[3-[[1-[2-[3-[7-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]acetyl]amino]heptanoylamino]phenyl]propan-2-ylsulfonyl]piperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC(C)(C1=CC(NC(=O)CCCCCCNC(=O)CNC2=C3CN(C4CCC(=O)NC4=O)C(=O)C3=CC=C2)=CC=C1)S(=O)(=O)N1CCC(NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CC1	C49H56ClN7O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-D567J9	SCHEMBL30273752	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[1-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]amino]acetyl]piperidine-4-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC=CC(NC(=O)C2CCN(C(=O)CNC3=CC=C4C(=O)N(C5CCC(=O)NC5=O)CC4=C3)CC2)=C1	C48H52ClN7O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-4RHPN0	SCHEMBL30273686	3-(Carboxymethoxy)-4-chloro-5-[3-[[1-[[3-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]amino]acetyl]amino]phenyl]-phenylmethyl]sulfonylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	O=C(O)COC1=C(C(=O)O)SC(C2=CC(NC3CCN(S(=O)(=O)C(C4=CC=CC=C4)C4=CC(NC(=O)CNC5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)=CC=C4)CC3)=CC=C2)=C1Cl	C46H41ClN6O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-076F2J	SCHEMBL30273796	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[1-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]amino]acetyl]piperidine-4-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)C2CCN(C(=O)CNC3=CC=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)CC2)=CC=C1	C48H50ClN7O13S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-88E657	WO2023019166A1_44	.	O=C(O)COC1=C(C(=O)O)SC(C2=CC(NC3CCN(S(=O)(=O)CC4=CC(NC(=O)C5CN(C(=O)CNC6=C7CN(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)C5)=CC=C4)CC3)=CC=C2)=C1Cl	C44H44ClN7O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-G15U13	SCHEMBL25036691	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[1-[2-[[2-[(3R)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-4-yl]amino]acetyl]azetidine-3-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)C2CN(C(=O)CNC3=C4CN([C@@H]5CCC(=O)NC5=O)C(=O)C4=CC=C3)C2)=CC=C1	C46H48ClN7O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-YLPTMF	SCHEMBL30273969	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[1-[2-[[2-[(3S)-2,6-dioxopiperidin-3-yl]-1-oxo-3H-isoindol-4-yl]amino]acetyl]azetidine-3-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)C2CN(C(=O)CNC3=C4CN([C@H]5CCC(=O)NC5=O)C(=O)C4=CC=C3)C2)=CC=C1	C46H48ClN7O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-JMGIFW	SCHEMBL25036682	3-(carboxymethoxy)-4-chloro-5-[3-[[1-[[3-[[2-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]piperidin-1-yl]acetyl]amino]phenyl]methylsulfonyl]piperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid; SCHEMBL30273717	O=C(O)COC1=C(C(=O)O)SC(C2=CC(NC3CCN(S(=O)(=O)CC4=CC(NC(=O)CN5CCC(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)CC5)=CC=C4)CC3)=CC=C2)=C1Cl	C45H47ClN6O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-PK0W5H	SCHEMBL25036684	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[3-[4-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]piperidin-1-yl]propanoylamino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)CCN2CCC(NC3=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)CC2)=CC=C1	C48H54ClN7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-BWWHOQ	SCHEMBL25036262	3-(carboxymethoxy)-4-chloro-5-[3-[[1-[[3-[3-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]propanoylamino]phenyl]methylsulfonyl]piperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid; SCHEMBL30274073	O=C(O)COC1=C(C(=O)O)SC(C2=CC(NC3CCN(S(=O)(=O)CC4=CC(NC(=O)CCC5=CC=C6C(=O)N(C7CCC(=O)NC7=O)CC6=C5)=CC=C4)CC3)=CC=C2)=C1Cl	C41H40ClN5O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-EDCT40	SCHEMBL25036358	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[1-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]acetyl]piperidine-4-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)C2CCN(C(=O)CNC3=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)CC2)=CC=C1	C48H52ClN7O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-9V0L8P	SCHEMBL25036357	3-(Carboxymethoxy)-4-chloro-5-[3-[[1-[[3-[3-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]propanoylamino]phenyl]methylsulfonyl]piperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid; SCHEMBL30274058	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(CCC(=O)NC3=CC=CC(CS(=O)(=O)N4CCC(NC5=CC=CC(C6=C(Cl)C(OCC(=O)O)=C(C(=O)O)S6)=C5)CC4)=C3)C=C21	C41H41ClN6O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-O3F0DV	WO2023019166A1_5	.	CC1=C(C2=CC(NC3CCN(S(=O)(=O)CC4=CC(NC(=O)CCOCCOCCNC(=O)COC5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)=CC=C4)CC3)=CC=C2)SC(C(=O)O)=C1OCC(=O)O	C48H52N6O16S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-EHCX2K	SCHEMBL30273942	3-(carboxymethoxy)-4-chloro-5-[3-[[1-[[3-[3-[4-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]piperidin-1-yl]propanoylamino]phenyl]methylsulfonyl]piperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	O=C(O)COC1=C(C(=O)O)SC(C2=CC(NC3CCN(S(=O)(=O)CC4=CC(NC(=O)CCN5CCC(NC6=C7CN(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)CC5)=CC=C4)CC3)=CC=C2)=C1Cl	C46H50ClN7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-DF6F8F	SCHEMBL25036089	3-(Carboxymethoxy)-4-chloro-5-[3-[[1-[[3-[[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidine-1-carbonyl]amino]phenyl]methylsulfonyl]piperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid; SCHEMBL30273595	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(C3CCN(C(=O)NC4=CC=CC(CS(=O)(=O)N5CCC(NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC5)=C4)CC3)C=C21	C44H46ClN7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-89M5GA	SCHEMBL25036847	3-(Carboxymethoxy)-4-chloro-5-[3-[[1-[[3-[[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-4-yl]piperidine-1-carbonyl]amino]phenyl]methylsulfonyl]piperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid; SCHEMBL30274151	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=CC(C3CCN(C(=O)NC4=CC=CC(CS(=O)(=O)N5CCC(NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC5)=C4)CC3)=C21	C44H46ClN7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-HTMI30	WO2023019166A1_53	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=CC(CCC(=O)NC3=CC=CC(CS(=O)(=O)N4CCC(NC5=CC=CC(C6=C(Cl)C(OCC(=O)O)=C(C(=O)O)S6)=C5)CC4)=C3)C21	C41H43ClN6O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-MDBTLB	SCHEMBL25036115	3-(Carboxymethoxy)-4-chloro-5-[3-[[1-[[3-[[2-[4-[3-(2,6-dioxopiperidin-3-yl)indazol-1-yl]piperidin-1-yl]acetyl]amino]phenyl]methylsulfonyl]piperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	O=C(O)COC1=C(C(=O)O)SC(C2=CC(NC3CCN(S(=O)(=O)CC4=CC(NC(=O)CN5CCC(N6N=C(C7CCC(=O)NC7=O)C7=CC=CC=C76)CC5)=CC=C4)CC3)=CC=C2)=C1Cl	C44H46ClN7O10S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-2UQSV7	SCHEMBL25036099	3-(Carboxymethoxy)-4-chloro-5-[3-[[1-[[3-[[2-[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidin-1-yl]acetyl]amino]phenyl]methylsulfonyl]piperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid; SCHEMBL30273922	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(C3CCN(CC(=O)NC4=CC=CC(CS(=O)(=O)N5CCC(NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC5)=C4)CC3)C=C21	C45H48ClN7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-IA7Z3O	SCHEMBL30273514	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[3-[4-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]oxy]piperidin-1-yl]propanoylamino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)CCN2CCC(OC3=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)CC2)=CC=C1	C48H53ClN6O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-MD8N64	SCHEMBL25036652	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[1-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-5-yl]amino]acetyl]azetidine-3-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid; SCHEMBL30273540	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)C2CN(C(=O)CNC3=CC=C4C(=O)N(C5CCC(=O)NC5=O)CC4=C3)C2)=CC=C1	C46H48ClN7O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-1JX74Q	SCHEMBL25036654	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[1-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyacetyl]piperidine-4-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)C2CCN(C(=O)COC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)CC2)=CC=C1	C48H49ClN6O14S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-LORK6Z	SCHEMBL30274158	3-(carboxymethoxy)-4-chloro-5-[3-[[1-[[3-[[4-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]piperidine-1-carbonyl]amino]phenyl]methylsulfonyl]piperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	O=C(O)COC1=C(C(=O)O)SC(C2=CC=CC(NC3CCN(S(=O)(=O)CC4=CC(NC(=O)N5CCC(NC6=C7CN(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)CC5)=CC=C4)CC3)=C2)=C1Cl	C44H46ClN7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-2MYQF4	SCHEMBL30273792	3-(Carboxymethoxy)-4-chloro-5-[3-[[1-[[3-[7-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]-methylamino]acetyl]amino]heptanoylamino]phenyl]methylsulfonyl]piperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CN(CC(=O)NCCCCCCC(=O)NC1=CC=CC(CS(=O)(=O)N2CCC(NC3=CC=CC(C4=C(Cl)C(OCC(=O)O)=C(C(=O)O)S4)=C3)CC2)=C1)C1=C2C(=O)N(C3CCC(=O)NC3=O)C(=O)C2=CC=C1	C48H52ClN7O13S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-KIQMTM	SCHEMBL30273932	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidine-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(C3CCN(C(=O)NC4=CC=CC(CS(=O)(=O)N5CC[C@H](NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC5(C)C)=C4)CC3)C=C21	C46H50ClN7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-09NNUI	SCHEMBL25036890	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[1-[3-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]propanoyl]piperidine-4-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)C2CCN(C(=O)CCC3=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)CC2)=CC=C1	C49H53ClN6O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-9EY9PO	SCHEMBL25036631	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[4-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]acetyl]piperazine-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)N2CCN(C(=O)CNC3=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)CC2)=CC=C1	C47H51ClN8O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-97PXVK	WO2023019166A1_63	.	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)C2CCN(C(=O)COC3C=CC=C4C(=O)N(C5CCC(=O)NC5=O)CC43)CC2)=CC=C1	C48H53ClN6O13S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-7WREQP	SCHEMBL30273502	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[4-[3-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]propanoyl]piperazine-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)N2CCN(C(=O)CCC3=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)CC2)=CC=C1	C48H52ClN7O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-29TMU3	SCHEMBL25036634	3-(carboxymethoxy)-4-chloro-5-[3-[[1-[[3-[[4-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]oxy]piperidine-1-carbonyl]amino]phenyl]methylsulfonyl]piperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	O=C(O)COC1=C(C(=O)O)SC(C2=CC(NC3CCN(S(=O)(=O)CC4=CC(NC(=O)N5CCC(OC6=C7CN(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)CC5)=CC=C4)CC3)=CC=C2)=C1Cl	C44H45ClN6O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-B1T3O3	WO2023019166A1_66	.	CN(C(=O)C1CCN(C(=O)CNC2=C3CN(C4CCC(=O)NC4=O)C(=O)C3=CC=C2)CC1)C1=CC=CC(CS(=O)(=O)N2CCC(NC3=CC=CC(C4=C(Cl)C(OCC(=O)O)=C(C(=O)O)S4)=C3)CC2(C)C)=C1	C49H54ClN7O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-KKRBDC	SCHEMBL30273973	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[1-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]acetyl]piperidine-4-carbonyl]-methylamino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CN(C(=O)C1CCN(C(=O)CNC2=C3CN(C4CCC(=O)NC4=O)C(=O)C3=CC=C2)CC1)C1=CC=CC(CS(=O)(=O)N2CC[C@H](NC3=CC=CC(C4=C(Cl)C(OCC(=O)O)=C(C(=O)O)S4)=C3)CC2(C)C)=C1	C49H54ClN7O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-9LUXCO	WO2023019166A1_68	.	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(CC(=O)N2CCC(C3=CC=C4C(=C3)OC(=O)N4C3CCC(=O)NC3=O)CC2)=CC=C1	C46H48ClN5O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-FSPKTI	SCHEMBL25036479	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[2-[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidin-1-yl]acetyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid; SCHEMBL30273534	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(C3CCN(CC(=O)NC4=CC=CC(CS(=O)(=O)N5CC[C@H](NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC5(C)C)=C4)CC3)C=C21	C47H52ClN7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-FQI1I0	WO2023019166A1_7	.	CC(CCNS(=O)(=O)CC1=CC(NC(=O)CCCCCCNC(=O)CNC2=C3CN(C4CCC(=O)NC4=O)C(=O)C3=CC=C2)=CC=C1)NC1=CC=CC(C2=C(Cl)C(OCC(=O)O)=C(C(=O)O)S2)=C1	C46H52ClN7O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-7VDXJG	WO2023019166A1_70	.	CC1=C(C2=CC(N[C@H]3CCN(S(=O)(=O)CC4=CC(NC(=O)CN5CCC(C6=CC=C7C(=C6)OC(=O)N7C6CCC(=O)NC6=O)CC5)=CC=C4)C(C)(C)C3)=CC=C2)SC(C(=O)O)=C1OCC(=O)O	C47H52N6O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-4ZGK7B	SCHEMBL25036478	3-(carboxymethoxy)-4-chloro-5-[3-[[1-[[3-[3-[4-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]piperidin-1-yl]propanoyl-methylamino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CN(C(=O)CCN1CCC(NC2=C3CN(C4CCC(=O)NC4=O)C(=O)C3=CC=C2)CC1)C1=CC=CC(CS(=O)(=O)N2CCC(NC3=CC=CC(C4=C(Cl)C(OCC(=O)O)=C(C(=O)O)S4)=C3)CC2(C)C)=C1	C49H56ClN7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-HX5SYW	SCHEMBL25036480	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[4-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]oxy]piperidine-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)N2CCC(OC3=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)CC2)=CC=C1	C46H49ClN6O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-ULGFED	SCHEMBL25036477	3-(carboxymethoxy)-4-chloro-5-[3-[[1-[[3-[[1-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]acetyl]piperidine-4-carbonyl]amino]-2-fluorophenyl]methylsulfonyl]piperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	O=C(O)COC1=C(C(=O)O)SC(C2=CC(NC3CCN(S(=O)(=O)CC4=C(F)C(NC(=O)C5CCN(C(=O)CNC6=C7CN(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)CC5)=CC=C4)CC3)=CC=C2)=C1Cl	C46H47ClFN7O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-TQ8U3C	SCHEMBL30273603	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[1-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]oxy]acetyl]azetidine-3-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC1(C)C[C@@H](NC2=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=CC=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)C2CN(C(=O)COC3=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)C2)=CC=C1	C46H47ClN6O13S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-147HEP	SCHEMBL25036674	3-(carboxymethoxy)-4-chloro-5-[3-[[1-[[3-[[1-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]acetyl]azetidine-3-carbonyl]amino]-2-fluorophenyl]methylsulfonyl]piperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	O=C(O)COC1=C(C(=O)O)SC(C2=CC(NC3CCN(S(=O)(=O)CC4=C(F)C(NC(=O)C5CN(C(=O)CNC6=C7CN(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)C5)=CC=C4)CC3)=CC=C2)=C1Cl	C44H43ClFN7O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-HYLS35	WO2023019166A1_76	.	CC1=C(C2=CC(N[C@H]3CCN(S(=O)(=O)CC4=CC(NC(=O)N5CCC(OC6=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)CC5)=CC=C4)C(C)(C)C3)=CC=C2)SC(C(=O)O)=C1OCC(=O)O	C47H52N6O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-BTXR8E	WO2023019166A1_77	.	CC1=C(C2=CC(NC3CCN(S(=O)(=O)CC4=CC(NC(=O)C5CCN(C(=O)CNC6=C7CN(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)CC5)=C(F)C=C4)CC3)=CC=C2)SC(C(=O)O)=C1OCC(=O)O	C47H50FN7O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-JDPVGM	SCHEMBL25034784	3-(carboxymethoxy)-4-chloro-5-[3-[[1-[[3-[[1-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]acetyl]azetidine-3-carbonyl]amino]-4-fluorophenyl]methylsulfonyl]piperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	O=C(O)COC1=C(C(=O)O)SC(C2=CC(NC3CCN(S(=O)(=O)CC4=CC(NC(=O)C5CN(C(=O)CNC6=C7CN(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)C5)=C(F)C=C4)CC3)=CC=C2)=C1Cl	C44H43ClFN7O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-SYQPWX	SCHEMBL25036717	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[3-[[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]amino]azetidine-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid; SCHEMBL30273815	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(NC3CN(C(=O)NC4=CC=CC(CS(=O)(=O)N5CC[C@H](NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC5(C)C)=C4)C3)C=C21	C44H47ClN8O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-L163QZ	SCHEMBL30273825	3-(Carboxymethoxy)-4-chloro-5-[3-[[1-[[3-[3-[2-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyethoxy]ethoxy]ethoxy]propanoylamino]phenyl]methylsulfonyl]piperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	O=C(O)COC1=C(C(=O)O)SC(C2=CC(NC3CCN(S(=O)(=O)CC4=CC(NC(=O)CCOCCOCCOCCOC5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)=CC=C4)CC3)=CC=C2)=C1Cl	C47H50ClN5O16S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-M9I6ZI	SCHEMBL25036720	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperazine-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid; SCHEMBL30274021	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(N3CCN(C(=O)NC4=CC=CC(CS(=O)(=O)N5CC[C@H](NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC5(C)C)=C4)CC3)C=C21	C45H49ClN8O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-2S9DK2	SCHEMBL25036724	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[4-[[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]amino]piperidine-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid; SCHEMBL30273628	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(NC3CCN(C(=O)NC4=CC=CC(CS(=O)(=O)N5CC[C@H](NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC5(C)C)=C4)CC3)C=C21	C46H51ClN8O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-XNMN1M	SCHEMBL25036718	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[4-[1-(2,6-dioxopiperidin-3-yl)-2-oxobenzo[cd]indol-6-yl]piperidine-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)N2CCC(C3=CC=C4C5=C(C=CC=C35)C(=O)N4C3CCC(=O)NC3=O)CC2)=CC=C1	C49H49ClN6O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-VZXBJA	SCHEMBL30273818	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[2-[4-[1-(2,6-dioxopiperidin-3-yl)-2-oxobenzo[cd]indol-6-yl]piperidin-1-yl]acetyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)CN2CCC(C3=CC=C4C5=C(C=CC=C35)C(=O)N4C3CCC(=O)NC3=O)CC2)=CC=C1	C50H51ClN6O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-2AVZ5E	SCHEMBL30273772	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[4-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]methylcarbamoyl]piperidine-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)N2CCC(C(=O)NCC3=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)CC2)=CC=C1	C48H52ClN7O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-Z9094H	WO2023019166A1_85	.	CC1(C)C[C@@H](CC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)OC2CCN(C(=O)CNC3=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)CC2)=CC=C1	C49H53ClN6O13S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-CZXXLW	SCHEMBL25036855	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[4-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]carbamoyl]cyclohexanecarbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid; SCHEMBL30273465	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)C2CCC(C(=O)NC3=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)CC2)=CC=C1	C48H51ClN6O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-J3VN9X	WO2023019166A1_87	.	CC(C)N1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(C3CCN(C(=O)NC4=CC=CC(CS(=O)(=O)N5CC[C@H](NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC5(C)C)C4)CC3)C=C21	C48H56ClN7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-UQEVRP	WO2023019166A1_87a	.	CC(C)N1C(=O)N([C@@H]2CCC(=O)NC2=O)C2=CC=C(C3CCN(C(=O)NC4=CC=CC(CS(=O)(=O)N5CCC(NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC5(C)C)=C4)CC3)C=C21	C48H54ClN7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-SLVPWB	WO2023019166A1_87b	.	CC(C)N1C(=O)N([C@H]2CCC(=O)NC2=O)C2=CC=C(C3CCN(C(=O)NC4=CC=CC(CS(=O)(=O)N5CCC(NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC5(C)C)=C4)CC3)C=C21	C48H54ClN7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-8XPI7H	WO2023019166A1_88	.	CCN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(C3CCN(C(=O)NC4=CC=CC(CS(=O)(=O)C5CC[C@H](NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC5(C)C)=C4)CC3)C=C21	C48H53ClN6O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-8MA6ZJ	SCHEMBL30274132	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[3-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]methylcarbamoyl]azetidine-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)N2CC(C(=O)NCC3=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)C2)=CC=C1	C46H48ClN7O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-4C95YD	SCHEMBL25036867	3-(carboxymethoxy)-4-chloro-5-[3-[[1-[[3-[3-[2-[2-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]oxy]acetyl]amino]ethoxy]ethoxy]propanoylamino]phenyl]methylsulfonyl]piperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	O=C(O)COC1=C(C(=O)O)SC(C2=CC(NC3CCN(S(=O)(=O)CC4=CC(NC(=O)CCOCCOCCNC(=O)COC5=C6CN(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)=CC=C4)CC3)=CC=C2)=C1Cl	C47H51ClN6O15S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-TU9SKS	SCHEMBL30274187	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[2-[1-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]acetyl]piperidin-4-yl]oxyacetyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)COC2CCN(C(=O)CNC3=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)CC2)=CC=C1	C49H54ClN7O13S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-PTU7DA	WO2023019166A1_91	.	CC1=C(C2=CC(N[C@H]3CCN(S(=O)(=O)CC4=CC(NC(=O)NCC#CC5=CC=C6C(=C5)N(C)C(=O)N6C5CCC(=O)NC5=O)=CC=C4)C(C)(C)C3)=CC=C2)SC(C(=O)O)=C1OCC(=O)O	C45H47N7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-265XXE	SCHEMBL30274148	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[2-[1-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]acetyl]azetidin-3-yl]oxyacetyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)COC2CN(C(=O)CNC3=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)C2)=CC=C1	C47H50ClN7O13S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-2NFA2W	SCHEMBL25036793	3-(carboxymethoxy)-4-chloro-5-[3-[[1-[[3-[[1-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]oxy]acetyl]azetidine-3-carbonyl]amino]-4-fluorophenyl]methylsulfonyl]piperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	O=C(O)COC1=C(C(=O)O)SC(C2=CC(NC3CCN(S(=O)(=O)CC4=CC(NC(=O)C5CN(C(=O)COC6=C7CN(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)C5)=C(F)C=C4)CC3)=CC=C2)=C1Cl	C44H42ClFN6O13S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-EN00YM	SCHEMBL25036791	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[4-[1-(2,6-dioxopiperidin-3-yl)-2,3-dihydroindol-5-yl]piperidine-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid; SCHEMBL30273849	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)N2CCC(C3=CC=C4C(=C3)CCN4C3CCC(=O)NC3=O)CC2)=CC=C1	C46H51ClN6O10S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-FLWQ24	SCHEMBL30273893	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[4-[1-(2,6-dioxopiperidin-3-yl)-2-methyl-2,3-dihydroindol-5-yl]piperidine-1-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	CC1CC2=CC(C3CCN(C(=O)NC4=CC=CC(CS(=O)(=O)N5CC[C@H](NC6=CC=CC(C7=C(Cl)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC5(C)C)=C4)CC3)=CC=C2N1C1CCC(=O)NC1=O	C47H53ClN6O10S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-OES2JI	WO2023019166A1_96	.	CC1(C)C[C@@H](NC2=CC=CC(C3=C(CI)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)OC2CN(C(=O)CNC3=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)C2)=CC=C1	C47H50IN7O13S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-6WJXSH	WO2023019166A1_97	.	CC1(C)C[C@@H](NC2=CC=CC(C3=C(Cl)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)C2CC3CN(C(=O)CNC4=C5CN(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3C2)=CC=C1	C50H54ClN7O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-CWF8PK	SCHEMBL30273492	3-(carboxymethoxy)-4-chloro-5-[3-[[(4S)-1-[[3-[[(1R,5S)-3-[2-[[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]amino]acetyl]-3-azabicyclo[3.1.0]hexane-6-carbonyl]amino]phenyl]methylsulfonyl]-2,2-dimethylpiperidin-4-yl]amino]phenyl]thiophene-2-carboxylic acid	[H][C@@]12CN(C(=O)CNC3=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)C[C@]1([H])[C@H]2C(=O)NC1=CC=CC(CS(=O)(=O)N2CC[C@H](NC3=CC=CC(C4=C(Cl)C(OCC(=O)O)=C(C(=O)O)S4)=C3)CC2(C)C)=C1	C48H50ClN7O12S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-0ZRJZL	WO2023019166A1_99	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(C3CCN(C(=O)NC4=CC=CC(CS(=O)(=O)N5CCC(NC6=CC=CC(C7=C(CI)C(OCC(=O)O)=C(C(=O)O)S7)=C6)CC5)=C4F)CC3)C=C21	C45H47FIN7O11S2	PTPN1;PTPN2	P18031/P17706	CRBN	WO-2023019166-A1
TPD-2J1ECP	CHEMBL5417088	(2S,4R)-1-[2-[3-[3-[(3S)-4-[4-[5-[(4S)-2-amino-3-cyano-4-methyl-6,7-dihydro-5H-1-benzothiophen-4-yl]-1,2,4-oxadiazol-3-yl]pyrimidin-2-yl]-3-methyl-1,4-diazepan-1-yl]propoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(OCCCN4CCCN(C5=NC=CC(C6=NOC([C@@]7(C)CCCC8=C7C(C#N)=C(N)S8)=N6)=N5)[C@@H](C)C4)=NO3)C(C)C)C=C2)SC=N1	C49H58N12O6S2	KRAS	P01116	VHL	WO-2023099620-A1
TPD-P5H06P	WO2023099620A1_I-10	.	CC1=C(C2=C(C)N=CS2)C=CC(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)C(C2=CC(OCCCCN3CCCN(C4=NC=CC(C5=NOC([C@@]6(C)CCCC7=C6C(C#N)=C(N)S7)=N5)=N4)[C@@H](C)C3)=NN2)C(C)C)=C1	C51H63N13O5S2	KRAS	P01116	VHL	WO-2023099620-A1
TPD-BELA0D	WO2023099620A1_I-11	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(OCCCCN4CCN(C5=NC(C6=NOC([C@@]7(C)CCCC8=C7C(C#N)=C(N)S8)=N6)=CC=N5)[C@@H](C)C4)=NO3)C(C)C)C=C2)SC=N1	C49H58N12O6S2	KRAS	P01116	VHL	WO-2023099620-A1
TPD-WLMI1K	WO2023099620A1_I-12	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(OCCCCN4CCCN(C5=NC=CC(C6=NSC([C@@]7(C)CCCC8=C7C(C#N)=C(N)S8)=C6)=N5)[C@@H](C)C4)=NO3)C(C)C)C=C2)SC=N1	C51H61N11O5S3	KRAS	P01116	VHL	WO-2023099620-A1
TPD-HZGGRJ	WO2023099620A1_I-13	.	CC1=C(C2=C(C)N=CS2)C=C(F)C(CNC(=O)C2C[C@@H](O)CN2C(=O)C(C2=CC(OCCCCN3CCCN(C4=NC=CC(C5=COC([C@@]6(C)CCCC7=C6C(C#N)=C(N)S7)=N5)=N4)[C@@H](C)C3)=NO2)C(C)C)=C1	C52H62FN11O6S2	KRAS	P01116	VHL	WO-2023099620-A1
TPD-UZQAL3	WO2023099620A1_I-14	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(OCCOCCN4CCCN(C5=NC=CC(C6=NOC([C@@]7(C)CCCC8=C7C(C#N)=C(N)S8)=N6)=N5)[C@@H](C)C4)=NO3)C(C)C)C=C2)SC=N1	C50H60N12O7S2	KRAS	P01116	VHL	WO-2023099620-A1
TPD-X1VR58	WO2023099620A1_I-15	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(OC/C=C/CN4CCCN(C5=NC=CC(C6=NOC([C@@]7(C)CCCC8=C7C(C#N)=C(N)S8)=NNN6)=N5)[C@@H](C)C4)=NO3)C(C)C)C=C2)SC=N1	C50H60N14O6S2	KRAS	P01116	VHL	WO-2023099620-A1
TPD-EKCB4R	WO2023099620A1_I-16	.	CC(C)C(C(=O)N1CC(O)C[C@H]1C(=O)NCC1=CC=C(C#N)C=C1)C1=CC(OCCCCN2CCCN(C3=NC=CC(C4=NOC([C@@]5(C)CCCC6=C5C(C#N)=C(N)S6)=N4)=N3)[C@@H](C)C2)=NO1	C47H56N12O6S	KRAS	P01116	VHL	WO-2023099620-A1
TPD-T2R7TQ	CHEMBL5416223	(2S,4R)-1-[2-[3-[4-[(3S)-4-[4-[5-[(4S)-2-amino-3-cyano-4-methyl-6,7-dihydro-5H-1-benzothiophen-4-yl]-1,2,4-oxadiazol-3-yl]pyrimidin-2-yl]-3-methyl-1,4-diazepan-1-yl]butoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[[4-(1,2,4-triazol-1-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC(C)C(C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(N2C=NC=N2)C=C1)C1=CC(OCCCCN2CCCN(C3=NC(C4=NOC([C@@]5(C)CCCC6=C5C(C#N)=C(N)S6)=N4)=CC=N3)[C@@H](C)C2)=NO1	C48H58N14O6S	KRAS	P01116	VHL	WO-2023099620-A1
TPD-4B1JO7	WO2023099620A1_I-18	.	CC(C)C(C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C#N)C(Cl)=C1)C1=CC(OCCCCN2CCCN(C3=NC=CC(C4=NOC([C@@]5(C)CCCC6=C5C(C#N)=C(N)S6)=N4)=N3)[C@@H](C)C2)=NO1	C47H55ClN12O6S	KRAS	P01116	VHL	WO-2023099620-A1
TPD-6JC975	CHEMBL5407519	(2S,4R)-1-[2-[3-[4-[(3S)-4-[4-[5-[(4S)-2-amino-3-cyano-4-methyl-6,7-dihydro-5H-1-benzothiophen-4-yl]-1,2,4-oxadiazol-3-yl]pyrimidin-2-yl]-3-methyl-1,4-diazepan-1-yl]butoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(4-imidazol-1-ylphenyl)methyl]pyrrolidine-2-carboxamide	CC(C)C(C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(N2C=CN=C2)C=C1)C1=CC(OCCCCN2CCCN(C3=NC(C4=NOC([C@@]5(C)CCCC6=C5C(C#N)=C(N)S6)=N4)=CC=N3)[C@@H](C)C2)=NO1	C49H59N13O6S	KRAS	P01116	VHL	WO-2023099620-A1
TPD-30IX01	WO2023099620A1_I-2	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(OCCN4CCCN(C5=NC=CC(C6=NOC([C@@]7(C)CCCC8=C7C(C#N)=C(N)S8)=N6)=N5)[C@@H](C)C4)=NO3)C(C)C)C=C2)SC=N1	C48H56N12O6S2	KRAS	P01116	VHL	WO-2023099620-A1
TPD-EJ4X6G	WO2023099620A1_I-20	.	CC(C)C(C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(Cl)C=C1)C1=CC(OCCCCN2CCCN(C3=NC(C4=NOC([C@@]5(C)CCCC6=C5C(C#N)=C(N)S6)=N4)=CC=N3)[C@@H](C)C2)=NO1	C46H56ClN11O6S	KRAS	P01116	VHL	WO-2023099620-A1
TPD-819E8O	WO2023099620A1_I-21	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(OCCCN4CCCN(C5=NC(C6=NOC([C@@]7(C)CCCC8=C7C(C#N)=C(N)S8)=N6)=NC=C5)[C@@H](C)C4)=NO3)C(C)C)C=C2)SC=N1	C49H58N12O6S2	KRAS	P01116	VHL	WO-2023099620-A1
TPD-DJVQCN	WO2023099620A1_I-22	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(OCCCCN4CCCN(C5=NC(C6=NOC([C@@]7(C)CCCC8=C7C(C#N)=C(N)S8)=N6)=NC=C5)[C@@H](C)C4)=NO3)C(C)C)C=C2)SC=N1	C50H60N12O6S2	KRAS	P01116	VHL	WO-2023099620-A1
TPD-HKY2QP	WO2023099620A1_I-23	.	CC(C)C1=CC=C(CNC(=O)[C@@H]2C[C@@H](O)CN2C(=O)C(C2=CC(OCCCCN3CCCN(C4=NC(C5=NOC([C@@]6(C)CCCC7=C6C(C#N)=C(N)S7)=N5)=CC=N4)[C@@H](C)C3)=NO2)C(C)C)C=C1	C49H63N11O6S	KRAS	P01116	VHL	WO-2023099620-A1
TPD-C77WJF	WO2023099620A1_I-24	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3=CC(OCCCN4CCCN(C5=NC=CC(C6=NOC([C@@]7(C)CCCC8=C7C(C#N)=C(N)S8)=N6)=N5)[C@@H](C)C4)NO3)C(C)C)C=C2)SC=N1	C49H60N12O6S2	KRAS	P01116	VHL	WO-2023099620-A1
TPD-KZRFU9	WO2023099620A1_I-26	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3=CC(OCCCCN4CCCN(C5=NC=CC(C6=NOC([C@@]7(C)CCCC8=C7C(C#N)=C(N)S8)=N6)=N5)[C@@H](C)C4)=NO3)C(C)C)C=C2)SC=N1	C50H60N12O6S2	KRAS	P01116	VHL	WO-2023099620-A1
TPD-3MA0QB	WO2023099620A1_I-27	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3CC(=O)CN3C(=O)[C@@H](C3=CC(OCCCCN4CCCN(C5=NC=CC(C6=NOC([C@@]7(C)CCCC8=C7C(C#N)=C(N)S8)=N6)=N5)[C@@H](C)C4)=NO3)C(C)C)C=C2)SC=N1	C50H58N12O6S2	KRAS	P01116	VHL	WO-2023099620-A1
TPD-XSH5MM	WO2023099620A1_I-28	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C(C)C)N3C=C(OCCCCN4CCCN(C5=NC(C6=NOC([C@@]7(C)CCCC8=C7C(C#N)=C(N)S8)=N6)=CC=N5)CC4)N=N3)C=C2)SC=N1	C49H60N14O5S2	KRAS	P01116	VHL	WO-2023099620-A1
TPD-40N4SM	ACBI3	(2S,4R)-1-[(2S)-2-[4-[4-[(3S)-4-[4-[5-[(4S)-2-azanyl-3-cyano-4-methyl-6,7-dihydro-5H-1-benzothiophen-4-yl]-1,2,4-oxadiazol-3-yl]pyrimidin-2-yl]-3-methyl-1,4-diazepan-1-yl]butoxy]-1,2,3-triazol-1-yl]-3-methyl-butanoyl]-N-[(1R)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]-2-oxidanyl-ethyl]-4-oxidanyl-pyrrolidine-2-carboxamide; 2938169-76-5; (2S,4R)-1-[(2S)-2-[4-[4-[(3S)-4-[4-[5-[(4S)-2-azanyl-3-cyano-4-methyl-6,7-dihydro-5H-1-benzothiophen-4-yl]-1,2,4-oxadiazol-3-yl]pyrimidin-2-yl]-3-methyl-1,4-diazepan-1-yl]butoxy]-1,2,3-triazol-1-yl]-3-methyl-butanoyl]-N-[(1R)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]-2-oxidanyl-ethyl]-4-oxidanyl-pyrrolidine-2-carboxamide; Wyl; orb2567120; EX-A8406; DA-50120; HY-157228; CS-0907910; H42640; (2S,4R)-1-((S)-2-(4-(4-((S)-4-(4-(5-((S)-2-Amino-3-cyano-4-methyl-4,5,6,7-tetrahydrobenzo[b]thiophen-4-yl)-1,2,4-oxadiazol-3-yl)pyrimidin-2-yl)-3-methyl-1,4-diazepan-1-yl)butoxy)-1H-1,2,3-triazol-1-yl)-3-methylbutanoyl)-4-hydroxy-N-((R)-2-hydroxy-1-(4-(4-methylthiazol-5-yl)phenyl)ethyl)pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CO)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C(OCCCCN4CCCN(C5=NC(C6=NOC([C@@]7(C)CCCC8=C7C(C#N)=C(N)S8)=N6)=CC=N5)[C@@H](C)C4)N=N3)C=C2)SC=N1	C50H62N14O6S2	KRAS	P01116	VHL	WO-2023099620-A1
TPD-8GXTKL	CHEMBL5404045	(2S,4R)-1-[2-[3-[4-[(3S)-4-[4-[5-[(4S)-2-amino-3-cyano-4-methyl-6,7-dihydro-5H-1-benzothiophen-4-yl]-1,2,4-oxadiazol-3-yl]pyrimidin-2-yl]-3-methyl-1,4-diazepan-1-yl]butoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(OCCCCN4CCCN(C5=NC=CC(C6=NOC([C@@]7(C)CCCC8=C7C(C#N)=C(N)S8)=N6)=N5)[C@@H](C)C4)=NO3)C(C)C)C=C2)SC=N1	C50H60N12O6S2	KRAS	P01116	VHL	WO-2023099620-A1
TPD-16NFX6	CHEMBL5415108	(2S,4R)-1-[(2S)-2-[4-[4-[(3S)-4-[4-[5-[(4S)-2-amino-3-cyano-4-methyl-6,7-dihydro-5H-1-benzothiophen-4-yl]-1,2,4-oxadiazol-3-yl]pyrimidin-2-yl]-3-methyl-1,4-diazepan-1-yl]pentoxy]triazol-1-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1R)-2-hydroxy-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CO)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C(OCCCC(C)N4CCCN(C5=NC(C6=NOC([C@@]7(C)CCCC8=C7C(C#N)=C(N)S8)=N6)=CC=N5)[C@@H](C)C4)N=N3)C=C2)SC=N1	C51H64N14O6S2	KRAS	P01116	VHL	WO-2023099620-A1
TPD-EQ6OQ8	WO2023099620A1_I-31	(2S,4R)-1-[(2S)-2-[4-[5-[(3S)-4-[4-[5-[(4S)-2-amino-3-cyano-4-methyl-6,7-dihydro-5H-1-benzothiophen-4-yl]-1,2,4-oxadiazol-3-yl]pyrimidin-2-yl]-3-methyl-1,4-diazepan-1-yl]pentan-2-yloxy]triazol-1-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1R)-2-hydroxy-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CO)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C(OC(C)CCCN4CCCN(C5=NC(C6=NOC([C@@]7(C)CCCC8=C7C(C#N)=C(N)S8)=N6)=CC=N5)[C@@H](C)C4)N=N3)C=C2)SC=N1	C51H64N14O6S2	KRAS	P01116	VHL	WO-2023099620-A1
TPD-KT8VRR	WO2023099620A1_I-32	.	CC1=C(C2=CC=C([C@H](CO)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C(C)C)N3C=C(OCCCCN4C[C@H](C)N(C5=NC=CC(C6=NOC([C@@]7(C)CCCC8=C7C(C#N)=C(N)S8)=N6)=N5)CCC4(C)C)N=N3)C=C2)SC=N1	C52H66N14O6S2	KRAS	P01116	VHL	WO-2023099620-A1
TPD-EVAAP7	SCHEMBL25597935	(2R)-2-[[(2S,4R)-1-[2-[4-[4-[(3S)-4-[4-[5-[(4S)-2-amino-3-cyano-4-methyl-6,7-dihydro-5H-1-benzothiophen-4-yl]-1,2,4-oxadiazol-3-yl]pyrimidin-2-yl]-3-methyl-1,4-diazepan-1-yl]butoxy]triazol-1-yl]-3-methylbutanoyl]-4-hydroxypyrrolidine-2-carbonyl]amino]-2-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]acetic acid	CC1=C(C2=CC=C([C@@H](NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C(C)C)N3C=C(OCCCCN4CCCN(C5=NC(C6=NOC([C@@]7(C)CCCC8=C7C(C#N)=C(N)S8)=N6)=CC=N5)[C@@H](C)C4)N=N3)C(=O)O)C=C2)SC=N1	C50H60N14O7S2	KRAS	P01116	VHL	WO-2023099620-A1
TPD-Q716HS	WO2023099620A1_I-34	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C(C)C)N3C=C(CCCCCN4CCCN(C5=NC=CC(C6=NOC([C@@]7(C)CCCC8=C7C(C#N)=C(N)S8)=N6)=N5)[C@@H](C)C4)N=N3)C=C2)SC=N1	C50H62N14O4S2	KRAS	P01116	VHL	WO-2023099620-A1
TPD-SA9D5J	WO2023099620A1_I-35	.	CC1=C(C2=CC=C([C@@H](NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C(C)C)N3C=C(OCCCCN4CCCN(C5=NC(C6=NOC([C@@]7(C)CCCC8=C7C(C#N)=C(N)S8)=N6)=CC=N5)[C@@H](C)C4)N=N3)[C@H](C)O)C=C2)SC=N1	C51H64N14O6S2	KRAS	P01116	VHL	WO-2023099620-A1
TPD-CHERSW	WO2023099620A1_I-36	.	CC1=C(C2=CC=C([C@@H](NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C(C)C)N3C=C(OCCCN4CCCN(C5=NC(C6=NOC([C@@]7(C)CCCC8=C7C(C#N)=C(N)S8)=N6)=CC=N5)[C@@H](C)C4)N=N3)[C@H](O)C(C)C)C=C2)SC=N1	C52H66N14O6S2	KRAS	P01116	VHL	WO-2023099620-A1
TPD-9QHK8V	WO2023099620A1_I-37	.	CC1=C(C2=CC=C([C@@H](NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C(C)C)N3C=C(OCCCCN4CCCN(C5=NC(C6=NOC([C@@]7(C)CCCC8=C7C(C#N)=C(N)S8)=N6)=CC=N5)[C@@H](C)C4)N=N3)[C@H](O)C(C)C)C=C2)SC=N1	C53H68N14O6S2	KRAS	P01116	VHL	WO-2023099620-A1
TPD-KPGTNY	WO2023099620A1_I-38	.	CC1=C(C2=CC=C([C@H](CCO)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C(OCCCCN4CCCN(C5=NC=CC(C6=NOC([C@@]7(C)CCCC8=C7C(C#N)=C(N)S8)=N6)=N5)[C@@H](C)C4)N=N3)C=C2)SC=N1	C51H64N14O6S2	KRAS	P01116	VHL	WO-2023099620-A1
TPD-X92V2L	WO2023099620A1_I-39	.	CC1=C(C2=CC=C([C@H](CCOP(=O)(O)O)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C(OCCCCN4CCCN(C5=NC=CC(C6=NOC([C@@]7(C)CCCC8=C7C(C#N)=C(N)S8)=N6)=N5)[C@@H](C)C4)N=N3)C=C2)SC=N1	C51H65N14O9PS2	KRAS	P01116	VHL	WO-2023099620-A1
TPD-1QRNMV	CHEMBL5411939	(2S,4R)-1-[2-[3-[4-[(3S)-4-[4-[5-[(4S)-2-amino-3-cyano-4-methyl-6,7-dihydro-5H-1-benzothiophen-4-yl]-1,2-oxazol-3-yl]pyrimidin-2-yl]-3-methyl-1,4-diazepan-1-yl]butoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(OCCCCN4CCCN(C5=NC=CC(C6=NOC([C@@]7(C)CCCC8=C7C(C#N)=C(N)S8)=C6)=N5)[C@@H](C)C4)=NO3)C(C)C)C=C2)SC=N1	C51H61N11O6S2	KRAS	P01116	VHL	WO-2023099620-A1
TPD-73PBO9	WO2023099620A1_I-40	.	CC1=C(C2=CC=C([C@@H](NC(=O)[C@@H]3CC(=O)CN3C(=O)[C@@H](C(C)C)N3C=C(OCCCCN4CCCN(C5=NC(C6=NOC([C@@]7(C)CCCC8=C7C(C#N)=C(N)S8)=N6)=CC=N5)[C@@H](C)C4)N=N3)[C@H](C)O)C=C2)SC=N1	C51H62N14O6S2	KRAS	P01116	VHL	WO-2023099620-A1
TPD-JGGKOK	WO2023099620A1_I-41	.	CC1=C(C2=CC=C([C@@H](NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C(OCCCCN4CCCN(C5=NC(C6=NOC([C@@]7(C)CCCC8=C7C(C#N)=C(N)S8)=N6)=CC=N5)[C@@H](C)C4)N=N3)[C@H](C)O)C=C2)SC=N1	C51H64N14O6S2	KRAS	P01116	VHL	WO-2023099620-A1
TPD-LNJP22	SCHEMBL25597844	(2S,4R)-1-[(2R)-2-[4-[3-[(3S)-4-[4-[5-[(4S)-2-amino-3-cyano-4-methyl-6,7-dihydro-5H-1-benzothiophen-4-yl]-1,2,4-oxadiazol-3-yl]pyrimidin-2-yl]-3-methyl-1,4-diazepan-1-yl]propoxy]triazol-1-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1R,2R)-2-hydroxy-3-methyl-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]butyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@@H](NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C(C)C)N3C=C(OCCCN4CCCN(C5=NC(C6=NOC([C@@]7(C)CCCC8=C7C(C#N)=C(N)S8)=N6)=CC=N5)[C@@H](C)C4)N=N3)[C@H](O)C(C)C)C=C2)SC=N1	C52H66N14O6S2	KRAS	P01116	VHL	WO-2023099620-A1
TPD-EU6UJ2	SCHEMBL25598008	(2S,4R)-1-[(2S)-2-[4-[3-[(3S)-4-[4-[5-[(4S)-2-amino-3-cyano-4-methyl-6,7-dihydro-5H-1-benzothiophen-4-yl]-1,2,4-oxadiazol-3-yl]pyrimidin-2-yl]-3-methyl-1,4-diazepan-1-yl]propoxy]triazol-1-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1R,2R)-2-hydroxy-3-methyl-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]butyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@@H](NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C(OCCCN4CCCN(C5=NC(C6=NOC([C@@]7(C)CCCC8=C7C(C#N)=C(N)S8)=N6)=CC=N5)[C@@H](C)C4)N=N3)[C@H](O)C(C)C)C=C2)SC=N1	C52H66N14O6S2	KRAS	P01116	VHL	WO-2023099620-A1
TPD-GFKEW0	WO2023099620A1_I-44	.	CC1=C(C2=CC=C([C@@H](NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C(C)C)N3C=C(OCCCCN4CCCN(C5=NC(C6=NOC([C@@]7(C)CCCC8=C7C(C#N)=C(N)S8)=N6)=CC=N5)[C@@H](C)C4)N=N3)[C@H](O)C(C)C)C=C2)SC=N1	C53H68N14O6S2	KRAS	P01116	VHL	WO-2023099620-A1
TPD-R1H3QX	WO2023099620A1_I-45	.	CC1=C(C2=CC=C([C@@H](NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C(OCCCCN4CCCN(C5=NC(C6=NOC([C@@]7(C)CCCC8=C7C(C#N)=C(N)S8)=N6)=CC=N5)[C@@H](C)C4)N=N3)[C@H](O)C(C)C)C=C2)SC=N1	C53H68N14O6S2	KRAS	P01116	VHL	WO-2023099620-A1
TPD-MJOZM4	WO2023099620A1_I-47	(2S,4R)-1-[(2S)-2-[6-[(3S)-4-[4-[5-[(4S)-2-azanyl-3-cyano-4-methyl-6,7-dihydro-5H-1-benzothiophen-4-yl]-1,2,4-oxadiazol-3-yl]pyrimidin-2-yl]-3-methyl-1,4-diazepan-1-yl]hexanoylamino]-3,3-dimethyl-butanoyl]-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-4-oxidanyl-pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCN3CCCN(C4=NC=CC(C5=NOC([C@@]6(C)CCCC7=C6C(C#N)=C(N)S7)=N5)=N4)[C@@H](C)C3)C(C)(C)C)C=C2)SC=N1	C50H64N12O5S2	KRAS	P01116	VHL	WO-2023099620-A1
TPD-2G09L6	SCHEMBL25598263	(2S,4R)-1-[(2S)-2-[[2-[3-[(3S)-4-[4-[5-[(4S)-2-amino-3-cyano-4-methyl-6,7-dihydro-5H-1-benzothiophen-4-yl]-1,2,4-oxadiazol-3-yl]pyrimidin-2-yl]-3-methyl-1,4-diazepan-1-yl]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCN3CCCN(C4=NC=CC(C5=NOC([C@@]6(C)CCCC7=C6C(C#N)=C(N)S7)=N5)=N4)[C@@H](C)C3)C(C)(C)C)C=C2)SC=N1	C49H62N12O6S2	KRAS	P01116	VHL	WO-2023099620-A1
TPD-BT893B	CHEMBL5397269	(2S,4R)-1-[2-[3-[4-[(3S)-4-[4-[5-[(4S)-2-amino-3-cyano-4-methyl-6,7-dihydro-5H-1-benzothiophen-4-yl]-1,2,4-oxadiazol-3-yl]pyrimidin-2-yl]-3-methyl-1,4-diazepan-1-yl]butoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-N-[[3-fluoro-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-4-hydroxypyrrolidine-2-carboxamide	CC1=C(C2=C(F)C=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(OCCCCN4CCCN(C5=NC=CC(C6=NOC([C@@]7(C)CCCC8=C7C(C#N)=C(N)S8)=N6)=N5)[C@@H](C)C4)=NO3)C(C)C)C=C2)SC=N1	C50H59FN12O6S2	KRAS	P01116	VHL	WO-2023099620-A1
TPD-J1IO3B	CHEMBL5403628	(2S,4R)-1-[2-[3-[4-[(3S)-4-[4-[3-[(4S)-2-amino-3-cyano-4-methyl-6,7-dihydro-5H-1-benzothiophen-4-yl]-1,2-oxazol-5-yl]pyrimidin-2-yl]-3-methyl-1,4-diazepan-1-yl]butoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(OCCCCN4CCCN(C5=NC=CC(C6=CC([C@@]7(C)CCCC8=C7C(C#N)=C(N)S8)=NO6)=N5)[C@@H](C)C4)=NO3)C(C)C)C=C2)SC=N1	C51H61N11O6S2	KRAS	P01116	VHL	WO-2023099620-A1
TPD-NHGJUG	WO2023099620A1_I-7	.	CC(C)C(C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(Br)C=C1)C1=CC(OCCCCN2CCCN(C3=NC=CC(C4=NOC([C@@]5(C)CCCC6=C5C(C#N)=C(N)S6)=N4)=N3)[C@@H](C)C2)=NO1	C46H56BrN11O6S	KRAS	P01116	VHL	WO-2023099620-A1
TPD-T10E0S	WO2023099620A1_I-8	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(OCCCCCN4CCCN(C5=NC=CC(C6=NOC([C@@]7(C)CCCC8=C7C(C#N)=C(N)S8)=N6)=N5)[C@@H](C)C4)=NO3)C(C)C)C=C2)SC=N1	C51H62N12O6S2	KRAS	P01116	VHL	WO-2023099620-A1
TPD-TTK8MX	WO2023099620A1_I-9	.	CC(C)C(C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=C(CO)N=CS2)C=C1)C1=CC(OCCCCN2CCCN(C3=NC(C4=NOC([C@@]5(C)CCCC6=C5C(C#N)=C(N)S6)=N4)=CC=N3)[C@@H](C)C2)=NO1	C50H60N12O7S2	KRAS	P01116	VHL	WO-2023099620-A1
TPD-AKPYY2	SCHEMBL25871544	N-[6-bromo-2-[4-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethylamino]-4-oxobutyl]-1-oxo-3H-isoindol-5-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	O=C(CCCN1CC2=C(C=C(Br)C(NC(=O)C3=CC=CC(C(F)(F)F)=N3)=C2)C1=O)NCCOCCOCCNC1=C2C(=O)N(C3CCC(=O)NC3=O)C(=O)C2=CC=C1	C38H37BrF3N7O9	IRAK4	Q9NWZ3	CRBN	WO-2023116920-A1
TPD-328QS2	SCHEMBL25871049	N-[2-[2-[3-[2-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]butylamino]-2-oxoethyl]-2-oxoimidazolidin-1-yl]ethyl]-6-(2-hydroxypropan-2-yl)indazol-5-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	CC(C)(O)C1=CC2=NN(CCN3CCN(CC(=O)NCCCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C3=O)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C41H43F3N10O8	IRAK4	Q9NWZ3	CRBN	WO-2023116920-A1
TPD-YDVJP8	SCHEMBL25871051	N-[2-[2-[3-[2-[9-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-oxoethyl]-2-oxoimidazolidin-1-yl]ethyl]-6-(2-hydroxypropan-2-yl)indazol-5-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	CC(C)(O)C1=CC2=NN(CCN3CCN(CC(=O)N4CCC5(CC4)CCN(C4=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C4)CC5)C3=O)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C46H49F3N10O8	IRAK4	Q9NWZ3	CRBN	WO-2023116920-A1
TPD-2CNLKR	SCHEMBL25871052	N-[2-[2-[3-[2-[7-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]-2,7-diazaspiro[3.5]nonan-2-yl]-2-oxoethyl]-2-oxoimidazolidin-1-yl]ethyl]-6-(2-hydroxypropan-2-yl)indazol-5-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	CC(C)(O)C1=CC2=NN(CCN3CCN(CC(=O)N4CC5(CCN(C6=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)CC5)C4)C3=O)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C44H45F3N10O8	IRAK4	Q9NWZ3	CRBN	WO-2023116920-A1
TPD-S9PXUB	SCHEMBL25871053	N-[2-[2-[3-[2-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperidin-4-yl]amino]-2-oxoethyl]-2-oxoimidazolidin-1-yl]ethyl]-6-(2-hydroxypropan-2-yl)indazol-5-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	CC(C)(O)C1=CC2=NN(CCN3CCN(CC(=O)NC4CCN(C5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)CC4)C3=O)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C42H43F3N10O8	IRAK4	Q9NWZ3	CRBN	WO-2023116920-A1
TPD-JHFZQ3	SCHEMBL25871054	N-[2-[2-[3-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperazin-1-yl]-2-oxoethyl]-2-oxoimidazolidin-1-yl]ethyl]-6-(2-hydroxypropan-2-yl)indazol-5-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	CC(C)(O)C1=CC2=NN(CCN3CCN(CC(=O)N4CCN(C5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)CC4)C3=O)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C41H41F3N10O8	IRAK4	Q9NWZ3	CRBN	WO-2023116920-A1
TPD-2MUCZE	SCHEMBL25871056	N-[2-[2-[3-[2-[2-[2-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]ethylamino]-2-oxoethyl]-2-oxoimidazolidin-1-yl]ethyl]-6-(2-hydroxypropan-2-yl)indazol-5-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCNC(=O)CN3CCN(CCN4C=C5C=C(NC(=O)C6=CC=CC(C(F)(F)F)=N6)C(C(C)(C)O)=CC5=N4)C3=O)C(C)(C)C)C=C2)SC=N1	C51H62F3N11O9S	IRAK4	Q9NWZ3	VHL	WO-2023116920-A1
TPD-E6X0UQ	SCHEMBL25876935	N-[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]-7-[2-[3-[2-[6-(2-hydroxypropan-2-yl)-5-[[6-(trifluoromethyl)pyridine-2-carbonyl]amino]indazol-2-yl]ethyl]-2-oxoimidazolidin-1-yl]acetyl]-7-azaspiro[3.5]nonane-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3CC4(CCN(C(=O)CN5CCN(CCN6C=C7C=C(NC(=O)C8=CC=CC(C(F)(F)F)=N8)C(C(C)(C)O)=CC7=N6)C5=O)CC4)C3)C(C)(C)C)C=C2)SC=N1	C56H68F3N11O8S	IRAK4	Q9NWZ3	VHL	WO-2023116920-A1
TPD-XTHJT0	SCHEMBL25871119	N-[(2S)-1-[(4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]-3-[2-[3-[2-[6-(2-hydroxypropan-2-yl)-5-[[6-(trifluoromethyl)pyridine-2-carbonyl]amino]indazol-2-yl]ethyl]-2-oxoimidazolidin-1-yl]acetyl]-3-azaspiro[5.5]undecane-9-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)C3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3CCC4(CC3)CCN(C(=O)CN3CCN(CCN5C=C6C=C(NC(=O)C7=CC=CC(C(F)(F)F)=N7)C(C(C)(C)O)=CC6=N5)C3=O)CC4)C(C)(C)C)C=C2)SC=N1	C58H72F3N11O8S	IRAK4	Q9NWZ3	VHL	WO-2023116920-A1
TPD-O8L9Y6	SCHEMBL25871120	N-[2-[2-[3-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]-2,7-diazaspiro[3.5]nonan-7-yl]-2-oxoethyl]-2-oxoimidazolidin-1-yl]ethyl]-6-methoxyindazol-5-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	COC1=CC2=NN(CCN3CCN(CC(=O)N4CCC5(CC4)CN(C4=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C4)C5)C3=O)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C42H41F3N10O8	IRAK4	Q9NWZ3	CRBN	WO-2023116920-A1
TPD-9KR0KL	WO2023116920A1_19	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CC3CC4(C3)CN(C(=O)CN3CCN(CCN5C=C6C=C(NC(=O)C7=CC=CC(C(F)(F)F)=N7)C(C(C)(C)O)=CC6=N5)C3=O)C4)C(C)(C)C)C=C2)SC=N1	C55H66F3N11O8S	IRAK4	Q9NWZ3	VHL	WO-2023116920-A1
TPD-8O5AAP	SCHEMBL25871047	N-[2-[2-[3-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethylamino]-2-oxoethyl]-2-oxoimidazolidin-1-yl]ethyl]-6-(2-hydroxypropan-2-yl)indazol-5-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	CC(C)(O)C1=CC2=NN(CCN3CCN(CC(=O)NCCOCCOCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C3=O)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C43H47F3N10O10	IRAK4	Q9NWZ3	CRBN	WO-2023116920-A1
TPD-SVXOAJ	SCHEMBL25871121	N-[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]-7-[2-[3-[2-[6-methoxy-5-[[6-(trifluoromethyl)pyridine-2-carbonyl]amino]indazol-2-yl]ethyl]-2-oxoimidazolidin-1-yl]acetyl]-7-azaspiro[3.5]nonane-2-carboxamide	COC1=CC2=NN(CCN3CCN(CC(=O)N4CCC5(CC4)CC(C(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)N[C@@H](C)C4=CC=C(C6=C(C)N=CS6)C=C4)C(C)(C)C)C5)C3=O)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C54H64F3N11O8S	IRAK4	Q9NWZ3	VHL	WO-2023116920-A1
TPD-PRMP6Z	SCHEMBL25871122	N-[(2S)-1-[(4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]-3-[2-[3-[2-[6-methoxy-5-[[6-(trifluoromethyl)pyridine-2-carbonyl]amino]indazol-2-yl]ethyl]-2-oxoimidazolidin-1-yl]acetyl]-3-azaspiro[5.5]undecane-9-carboxamide	COC1=CC2=NN(CCN3CCN(CC(=O)N4CCC5(CCC(C(=O)N[C@H](C(=O)N6C[C@H](O)CC6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)(C)C)CC5)CC4)C3=O)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C56H68F3N11O8S	IRAK4	Q9NWZ3	VHL	WO-2023116920-A1
TPD-AMTH2A	WO2023116920A1_22	.	COC1=CC2=NN(CCN3CCN(CC(=O)N4CC5(CC(CC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)(C)C)C5)C4)C3=O)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C53H62F3N11O8S	IRAK4	Q9NWZ3	VHL	WO-2023116920-A1
TPD-EPG2RT	SCHEMBL25871124	N-[2-[2-[3-[2-[9-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-oxoethyl]-2-oxoimidazolidin-1-yl]ethyl]-6-methoxyindazol-5-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	COC1=CC2=NN(CCN3CCN(CC(=O)N4CCC5(CC4)CCN(C4=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C4)CC5)C3=O)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C44H45F3N10O8	IRAK4	Q9NWZ3	CRBN	WO-2023116920-A1
TPD-0PHJ5U	SCHEMBL25871550	N-[2-[2-[9-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-oxoethyl]-6-methoxy-1-oxo-3H-isoindol-5-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	COC1=CC2=C(C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1)CN(CC(=O)N1CCC3(CC1)CCN(C1=CC=CC4=C1C(=O)N(C1CCC(=O)NC1=O)C4=O)CC3)C2=O	C40H38F3N7O8	IRAK4	Q9NWZ3	CRBN	WO-2023116920-A1
TPD-Y0GDG9	SCHEMBL25871552	N-[2-[4-[9-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]-3,9-diazaspiro[5.5]undecan-3-yl]-3,3-dimethyl-4-oxobutyl]-6-methoxy-1-oxo-3H-isoindol-5-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	COC1=CC2=C(C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1)CN(CCC(C)(C)C(=O)N1CCC3(CC1)CCN(C1=CC=CC4=C1C(=O)N(C1CCC(=O)NC1=O)C4=O)CC3)C2=O	C44H46F3N7O8	IRAK4	Q9NWZ3	CRBN	WO-2023116920-A1
TPD-A2XR7N	SCHEMBL25871555	N-[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]-3-[4-[5-methoxy-3-oxo-6-[[6-(trifluoromethyl)pyridine-2-carbonyl]amino]-1H-isoindol-2-yl]-2,2-dimethylbutanoyl]-3-azaspiro[5.5]undecane-9-carboxamide	COC1=CC2=C(C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1)CN(CCC(C)(C)C(=O)N1CCC3(CCC(C(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)N[C@@H](C)C4=CC=C(C5=C(C)N=CS5)C=C4)C(C)(C)C)CC3)CC1)C2=O	C56H69F3N8O8S	IRAK4	Q9NWZ3	VHL	WO-2023116920-A1
TPD-XYMDK2	WO2023116920A1_27	.	COC1=CC2=C(C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1)CN(CCC(C)(C)C(=O)N1CC3(CC(CC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)N[C@@H](C)C4=CC=C(C5=C(C)N=CS5)C=C4)C(C)(C)C)C3)C1)C2=O	C53H63F3N8O8S	IRAK4	Q9NWZ3	VHL	WO-2023116920-A1
TPD-CBIJ5I	WO2023116920A1_28	.	COC1=CC2=NN(CCN3CCN(CC(=O)N4CCC5(CC4)CC(N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)N[C@@H](C)C4=CC=C(C6=C(C)N=CS6)C=C4)C(C)(C)C)C5)C3=O)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C53H64F3N11O7S	IRAK4	Q9NWZ3	VHL	WO-2023116920-A1
TPD-7S4T7M	WO2023116920A1_29	.	COC1=CC2=NN(CCN3CCN(CC(=O)N4CCC5(CCC(C(=O)N[C@H](C(=O)N6C[C@H](C)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)(C)C)CC5)CC4)CC3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C58H74F3N11O6S	IRAK4	Q9NWZ3	VHL	WO-2023116920-A1
TPD-S02VAK	SCHEMBL25871547	N-[6-bromo-2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethyl]-1-oxo-3H-isoindol-5-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	O=C1CCC(N2C(=O)C3=CC=CC(NCCOCCOCCN4CC5=C(C=C(Br)C(NC(=O)C6=CC=CC(C(F)(F)F)=N6)=C5)C4=O)=C3C2=O)C(=O)N1	C34H30BrF3N6O8	IRAK4	Q9NWZ3	CRBN	WO-2023116920-A1
TPD-96O8B4	SCHEMBL25870980	N-[2-[2-[4-[2-[9-[5-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]pyrimidin-2-yl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-oxoethyl]piperazin-1-yl]ethyl]-6-methoxyindazol-5-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	COC1=CC2=NN(CCN3CCN(CC(=O)N4CCC5(CC4)CCN(C4=NC=C(NC6=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)C=N4)CC5)CC3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C49H52F3N13O7	IRAK4	Q9NWZ3	CRBN	WO-2023116920-A1
TPD-2S938C	WO2023116920A1_31	.	COC1=CC2=NN(CCN3CCN(CC(=O)N4CC5(CC(CC(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)(C)C)C5)C4)CC3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C54H66F3N11O7S	IRAK4	Q9NWZ3	VHL	WO-2023116920-A1
TPD-UGHDF1	WO2023116920A1_32	.	COC1=C(NC(=O)C2=NC(C(F)(F)F)=CC=C2)C=C2CN(CCC(C)(C)C(=O)N3CCC4(CC3)CCN(C3=NC=C(C(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=C(C)N=CS6)C=C5)C(C)(C)C)C=N3)CC4)C(=O)C2=C1	C59H70F3N11O8S	IRAK4	Q9NWZ3	VHL	WO-2023116920-A1
TPD-EC6SFF	SCHEMBL25871688	N-[2-[4-[9-[5-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]pyrimidin-2-yl]-3,9-diazaspiro[5.5]undecan-3-yl]-3,3-dimethyl-4-oxobutyl]-6-methoxy-1-oxo-3H-isoindol-5-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	COC1=C(NC(=O)C2=NC(C(F)(F)F)=CC=C2)C=C2CN(CCC(C)(C)C(=O)N3CCC4(CC3)CCN(C3=NC=C(NC5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)C=N3)CC4)C(=O)C2=C1	C48H49F3N10O8	IRAK4	Q9NWZ3	CRBN	WO-2023116920-A1
TPD-VG2U9Z	SCHEMBL25870982	N-[2-[2-[4-[5-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]pyrimidin-2-yl]piperazin-1-yl]ethyl]-6-methoxyindazol-5-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	COC1=CC2=NN(CCN3CCN(C4=NC=C(NC5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)C=N4)CC3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C38H34F3N11O6	IRAK4	Q9NWZ3	CRBN	WO-2023116920-A1
TPD-8NODV6	WO2023116920A1_35	N-[2-[2-[3-[2-[9-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-3-azaspiro[5.5]undecan-3-yl]-2-oxoethyl]-2-oxoimidazolidin-1-yl]ethyl]-6-methoxyindazol-5-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	COC1=CC2=NN(CCN3CCN(CC(=O)N4CCC5(CCC(N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)(C)C)CC5)CC4)C3=O)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C55H68F3N11O7S	IRAK4	Q9NWZ3	VHL	WO-2023116920-A1
TPD-L49HCJ	SCHEMBL25877271	N-[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]-5-[3-[4-[5-methoxy-3-oxo-6-[[6-(trifluoromethyl)pyridine-2-carbonyl]amino]-1H-isoindol-2-yl]-2,2-dimethylbutanoyl]-3,9-diazaspiro[5.5]undecan-9-yl]pyrimidine-2-carboxamide	COC1=C(NC(=O)C2=NC(C(F)(F)F)=CC=C2)C=C2CN(CCC(C)(C)C(=O)N3CCC4(CC3)CCN(C3=CN=C(C(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=C(C)N=CS6)C=C5)C(C)(C)C)N=C3)CC4)C(=O)C2=C1	C59H70F3N11O8S	IRAK4	Q9NWZ3	VHL	WO-2023116920-A1
TPD-5P98UR	SCHEMBL25871044	N-[2-[2-[4-[3-[5-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]pyrimidin-2-yl]-3-azaspiro[5.5]undecane-9-carbonyl]piperazin-1-yl]ethyl]-6-methoxyindazol-5-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	COC1=CC2=NN(CCN3CCN(C(=O)C4CCC5(CC4)CCN(C4=NC=C(NC6=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)C=N4)CC5)CC3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C49H51F3N12O7	IRAK4	Q9NWZ3	CRBN	WO-2023116920-A1
TPD-QTAMIB	SCHEMBL25871126	N-[2-[2-[4-[2-[9-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-oxoethyl]piperazin-1-yl]ethyl]-6-methoxyindazol-5-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	COC1=CC2=NN(CCN3CCN(CC(=O)N4CCC5(CC4)CCN(C4=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C4)CC5)CC3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C45H49F3N10O7	IRAK4	Q9NWZ3	CRBN	WO-2023116920-A1
TPD-3ZTG0J	SCHEMBL25871192	N-[2-[2-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperazin-1-yl]ethyl]-6-methoxyindazol-5-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	COC1=CC2=NN(CCN3CCN(C4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C34H31F3N8O6	IRAK4	Q9NWZ3	CRBN	WO-2023116920-A1
TPD-O818NQ	SCHEMBL25871549	N-[6-bromo-2-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethyl]-1-oxo-3H-isoindol-5-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	O=C1CCC(N2C(=O)C3=CC=CC(NCCOCCOCCOCCN4CC5=C(C=C(Br)C(NC(=O)C6=CC=CC(C(F)(F)F)=N6)=C5)C4=O)=C3C2=O)C(=O)N1	C36H34BrF3N6O9	IRAK4	Q9NWZ3	CRBN	WO-2023116920-A1
TPD-PSQP57	SCHEMBL25877018	N-[2-[2-[4-[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]-3-azaspiro[5.5]undecan-9-yl]piperazin-1-yl]ethyl]-6-methoxyindazol-5-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	COC1=CC2=NN(CCN3CCN(C4CCC5(CC4)CCN(C4=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C4)CC5)CC3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C44H48F3N9O6	IRAK4	Q9NWZ3	CRBN	WO-2023116920-A1
TPD-BMCW1S	SCHEMBL25871690	N-[2-[4-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]piperidin-4-yl]amino]-3,3-dimethyl-4-oxobutyl]-6-methoxy-1-oxo-3H-isoindol-5-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	COC1=CC2=C(C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1)CN(CCC(C)(C)C(=O)NC1CCN(C3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)CC1)C2=O	C40H40F3N7O8	IRAK4	Q9NWZ3	CRBN	WO-2023116920-A1
TPD-E1TEHT	WO2023116920A1_42	.	COC1=CC2=NN(CCN3CCN(C(=O)C4CCC5(CC4)CCN(C4=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C4)CC5)CC3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C45H48F3N9O7	IRAK4	Q9NWZ3	CRBN	WO-2023116920-A1
TPD-ZFCAN7	WO2023116920A1_43	.	COC1=CC2=C(C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1)CN(CCN1CCN(CC(=O)N3CCC4(CCC(C(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=C(C)N=CS6)C=C5)C(C)(C)C)CC4)CC3)CC1)C2=O	C58H73F3N10O8S	IRAK4	Q9NWZ3	VHL	WO-2023116920-A1
TPD-LJUDKQ	SCHEMBL25871693	N-[2-[2-[4-[2-[9-[[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-3-azaspiro[5.5]undecan-3-yl]-2-oxoethyl]piperazin-1-yl]ethyl]-6-methoxy-1-oxo-3H-isoindol-5-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	COC1=CC2=C(C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1)CN(CCN1CCN(CC(=O)N3CCC4(CCC(N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=C(C)N=CS6)C=C5)C(C)(C)C)CC4)CC3)CC1)C2=O	C57H73F3N10O7S	IRAK4	Q9NWZ3	VHL	WO-2023116920-A1
TPD-1NFDIW	SCHEMBL25871198	N-[2-[2-[(3R)-4-[2-[9-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-oxoethyl]-3-methylpiperazin-1-yl]ethyl]-6-methoxyindazol-5-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	COC1=CC2=NN(CCN3CCN(CC(=O)N4CCC5(CC4)CCN(C4=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C4)CC5)[C@H](C)C3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C46H51F3N10O7	IRAK4	Q9NWZ3	CRBN	WO-2023116920-A1
TPD-P0LQT5	WO2023116920A1_46	.	COC1=CC2=NN(CCN3CCN(CC(=O)N4CCC5(CC4)CCN(C4=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C4)CC5)[C@@H](C)C3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C46H51F3N10O7	IRAK4	Q9NWZ3	CRBN	WO-2023116920-A1
TPD-BT9IZ8	SCHEMBL25871203	N-[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]-3-[2-[(2S)-4-[2-[6-methoxy-5-[[6-(trifluoromethyl)pyridine-2-carbonyl]amino]indazol-2-yl]ethyl]-2-methylpiperazin-1-yl]acetyl]-3-azaspiro[5.5]undecane-9-carboxamide	COC1=CC2=NN(CCN3CCN(CC(=O)N4CCC5(CCC(C(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)(C)C)CC5)CC4)[C@@H](C)C3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C58H74F3N11O7S	IRAK4	Q9NWZ3	VHL	WO-2023116920-A1
TPD-QYST72	SCHEMBL25871204	N-[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]-3-[2-[(2R)-4-[2-[6-methoxy-5-[[6-(trifluoromethyl)pyridine-2-carbonyl]amino]indazol-2-yl]ethyl]-2-methylpiperazin-1-yl]acetyl]-3-azaspiro[5.5]undecane-9-carboxamide	COC1=CC2=NN(CCN3CCN(CC(=O)N4CCC5(CCC(C(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)(C)C)CC5)CC4)[C@H](C)C3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C58H74F3N11O7S	IRAK4	Q9NWZ3	VHL	WO-2023116920-A1
TPD-TFX855	WO2023116920A1_49	.	COC1=CC2=C(C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1)CN(CCN1CCN(CC(=O)N3CC4(CC(N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=C(C)N=CS6)C=C5)C(C)(C)C)C4)C3)CC1)C2=O	C53H65F3N10O7S	IRAK4	Q9NWZ3	VHL	WO-2023116920-A1
TPD-TFM39W	SCHEMBL25871048	N-[2-[2-[3-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]-2,7-diazaspiro[3.5]nonan-7-yl]-2-oxoethyl]-2-oxoimidazolidin-1-yl]ethyl]-6-(2-hydroxypropan-2-yl)indazol-5-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	CC(C)(O)C1=CC2=NN(CCN3CCN(CC(=O)N4CCC5(CC4)CN(C4=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C4)C5)C3=O)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C44H45F3N10O8	IRAK4	Q9NWZ3	CRBN	WO-2023116920-A1
TPD-WK5SOF	WO2023116920A1_50	.	CC(C)(O)C1=CC2=NN(CCN3CCN(CC(=O)N4CCC5(CC4)CCN(C4=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C4)CC5)CC3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C47H53F3N10O7	IRAK4	Q9NWZ3	CRBN	WO-2023116920-A1
TPD-PRTHTP	WO2023116920A1_51	.	CC1CN(C(=O)C2=NC(C(F)(F)F)=CC=C2)C2=CC3=CN(CC(=O)N4CCN(CC(=O)N5CCC6(CC5)CCN(C5=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C5)CC6)CC4)N=C3C=C2O1	C47H49F3N10O8	IRAK4	Q9NWZ3	CRBN	WO-2023116920-A1
TPD-UEFPK4	WO2023116920A1_52	.	COC1=CC2=C(C=C1NC(=O)C1C=CC=C(C(F)(F)F)N1)CN(CCN1CCN(CC(=O)N3CC4(CC(CC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=C(C)N=CS6)C=C5)C(C)(C)C)C4)C3)CC1)C2=O	C55H69F3N10O8S	IRAK4	Q9NWZ3	VHL	WO-2023116920-A1
TPD-HQ1BPN	SCHEMBL25871276	N-[2-[2-[3-[2-[9-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-oxoethyl]-3,8-diazabicyclo[3.2.1]octan-8-yl]ethyl]-6-methoxyindazol-5-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	COC1=CC2=NN(CCN3C4CCC3CN(CC(=O)N3CCC5(CC3)CCN(C3=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C3)CC5)C4)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C47H51F3N10O7	IRAK4	Q9NWZ3	CRBN	WO-2023116920-A1
TPD-SWX2LS	SCHEMBL25877083	N-[2-[2-[8-[2-[9-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-oxoethyl]-3,8-diazabicyclo[3.2.1]octan-3-yl]ethyl]-6-methoxyindazol-5-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	COC1=CC2=NN(CCN3CC4CCC(C3)N4CC(=O)N3CCC4(CC3)CCN(C3=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C3)CC4)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C47H51F3N10O7	IRAK4	Q9NWZ3	CRBN	WO-2023116920-A1
TPD-7UJWXM	SCHEMBL25871277	N-[2-[2-[4-[2-[9-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-oxoethyl]piperazin-1-yl]ethyl]-6-methoxyindazol-5-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	COC1=CC2=NN(CCN3CCN(CC(=O)N4CCC5(CC4)CCN(C4=C(F)C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C4)CC5)CC3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C45H48F4N10O7	IRAK4	Q9NWZ3	CRBN	WO-2023116920-A1
TPD-CW4ONT	WO2023116920A1_56	.	COC1=CC2=NN(CCN3CCN(CC(=O)N4CCC5(CCC(OC6=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)CC5)CC4)CC3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C46H50F3N9O8	IRAK4	Q9NWZ3	CRBN	WO-2023116920-A1
TPD-VV6WHI	WO2023116920A1_57	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3CCC4(CC3)CCN(C(=O)CN3CCN(CCN5C=C6C=C(NC(=O)C7=NC(C(F)(F)F)=CC=C7)C(OC(C)C)=CC6=N5)CC3)CC4)C(C)(C)C)C=C2)SC=N1	C59H76F3N11O7S	IRAK4	Q9NWZ3	VHL	WO-2023116920-A1
TPD-Z5KS7P	SCHEMBL25871814	N-[2-[2-[4-[2-[9-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-oxoethyl]piperazin-1-yl]ethyl]-6-methoxy-1-oxo-3H-isoindol-5-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	COC1=CC2=C(C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1)CN(CCN1CCN(CC(=O)N3CCC4(CC3)CCN(C3=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C3)CC4)CC1)C2=O	C46H50F3N9O8	IRAK4	Q9NWZ3	CRBN	WO-2023116920-A1
TPD-1AQSVN	SCHEMBL25871816	N-[2-[4-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]-2,7-diazaspiro[3.5]nonan-7-yl]-3,3-dimethyl-4-oxobutyl]-6-methoxy-1-oxo-3H-isoindol-5-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	COC1=CC2=C(C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1)CN(CCC(C)(C)C(=O)N1CCC3(CC1)CN(C1=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C1)C3)C2=O	C42H42F3N7O8	IRAK4	Q9NWZ3	CRBN	WO-2023116920-A1
TPD-YTNSLC	WO2023116920A1_60	.	CC(C)OC1=CC2=NN(CCN3CCN(CC(=O)N4CC5(C4)CN(C4=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C4)C5)CC3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C43H45F3N10O7	IRAK4	Q9NWZ3	CRBN	WO-2023116920-A1
TPD-K2NYGM	WO2023116920A1_61	.	COC1=CC2=NN(CCN3CCN(CC(=O)N4CC5(C4)CN(C4=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C4)C5)CC3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C41H41F3N10O7	IRAK4	Q9NWZ3	CRBN	WO-2023116920-A1
TPD-BV3RFM	SCHEMBL25871323	N-[2-[2-[4-[2-[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]-2,7-diazaspiro[3.5]nonan-7-yl]-2-oxoethyl]piperazin-1-yl]ethyl]-6-methoxyindazol-5-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	COC1=CC2=NN(CCN3CCN(CC(=O)N4CCC5(CC4)CN(C4=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C4)C5)CC3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C43H45F3N10O7	IRAK4	Q9NWZ3	CRBN	WO-2023116920-A1
TPD-FC6ZSO	WO2023116920A1_63	.	CC(C)(O)C1=CC2=NN(CCN3CCN(CC(=O)N4CC5(C4)CN(C4=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C4)C5)CC3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C43H45F3N10O7	IRAK4	Q9NWZ3	CRBN	WO-2023116920-A1
TPD-XMLTQR	WO2023116920A1_64	.	COC1=CC2=C(C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1)CN(CCC(C)(C)C(=O)N1CC3(C1)CN(C1=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C1)C3)C2=O	C40H38F3N7O8	IRAK4	Q9NWZ3	CRBN	WO-2023116920-A1
TPD-2EM4E7	SCHEMBL25871325	N-[2-[2-[4-[3-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]prop-2-ynoxy]piperidin-1-yl]ethyl]-6-methoxyindazol-5-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	COC1=CC2=NN(CCN3CCC(OCC#CC4=CC=CC5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C38H34F3N7O7	IRAK4	Q9NWZ3	CRBN	WO-2023116920-A1
TPD-DOT3DO	SCHEMBL25871326	N-[2-[2-[1-[2-[9-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-oxoethyl]piperidin-4-yl]ethyl]-6-methoxyindazol-5-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	COC1=CC2=NN(CCC3CCN(CC(=O)N4CCC5(CC4)CCN(C4=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C4)CC5)CC3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C46H50F3N9O7	IRAK4	Q9NWZ3	CRBN	WO-2023116920-A1
TPD-V4HQEE	SCHEMBL25871327	N-[2-[3-[1-[2-[9-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-oxoethyl]piperidin-4-yl]prop-2-ynyl]-6-methoxyindazol-5-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	COC1=CC2=NN(CC#CC3CCN(CC(=O)N4CCC5(CC4)CCN(C4=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C4)CC5)CC3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C47H48F3N9O7	IRAK4	Q9NWZ3	CRBN	WO-2023116920-A1
TPD-4XSW5L	SCHEMBL25871329	N-[(2S)-1-[(2S,4R)-4-hydroxy-2-[[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]-3-[2-[4-[2-[6-methoxy-5-[[6-(trifluoromethyl)pyridine-2-carbonyl]amino]indazol-2-yl]ethyl]piperidin-1-yl]acetyl]-3-azaspiro[5.5]undecane-9-carboxamide	COC1=CC2=NN(CCC3CCN(CC(=O)N4CCC5(CCC(C(=O)N[C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)(C)C)CC5)CC4)CC3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C58H73F3N10O7S	IRAK4	Q9NWZ3	VHL	WO-2023116920-A1
TPD-GSKRKV	WO2023116920A1_69	.	COC1=CC2=NN(CCN3CCN(C4=CC=C(OCC#CC5=CC=CC6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)C=C4)CC3)C=C2C=C1NC(=O)C1=CC=CC(C(F)(F)F)=N1	C43H37F3N8O7	IRAK4	Q9NWZ3	CRBN	WO-2023116920-A1
TPD-02FIE7	WO2023116920A1_70	.	COC1=CC2=NN(CCC3CCN(CC(=O)N4CC5(CC(CC(=O)N[C@H](C(=O)N6C[C@H](O)CC6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)(C)C)C5)C4)CC3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C55H67F3N10O7S	IRAK4	Q9NWZ3	VHL	WO-2023116920-A1
TPD-HD7KCF	SCHEMBL25871441	N-[2-[2-[4-[2-[9-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-oxoethyl]piperidin-1-yl]ethyl]-6-methoxyindazol-5-yl]-6-(trifluoromethyl)pyridine-2-carboxamide	COC1=CC2=NN(CCN3CCC(CC(=O)N4CCC5(CC4)CCN(C4=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C4)CC5)CC3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C46H50F3N9O7	IRAK4	Q9NWZ3	CRBN	WO-2023116920-A1
TPD-XTKFMD	WO2023116920A1_72	.	COC1=CC2=NN(CCN3CCC(CC(=O)N4CC5(C4)CN(C4=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C4)C5)CC3)C=C2C=C1NC(=O)C1=NC(C(F)(F)F)=CC=C1	C42H42F3N9O7	IRAK4	Q9NWZ3	CRBN	WO-2023116920-A1
TPD-LCP841	WO2023116920A1_73	.	O=C1CCC(N2C(=O)C3=CC=CC(N4CCC5(CCN(C(=O)CN6CCN(CCN7C=C8C=C(NC(=O)C9=NC(C(F)(F)F)=CC=C9)C(OC(F)(F)F)=CC8=N7)CC6)CC5)CC4)=C3C2=O)C(=O)N1	C45H46F6N10O7	IRAK4	Q9NWZ3	CRBN	WO-2023116920-A1
TPD-CDC4PW	WO2023119677A1_1	(2S,4R)-1-[(2S)-2-[[4-[[6-cyclopropyl-4-[(1S,4S)-2,5-diazabicyclo[2.2.1]heptan-2-yl]-7-(6-fluoro-5-methyl-1H-indazol-4-yl)-2-(oxan-4-yloxy)quinazolin-8-yl]oxymethyl]benzoyl]amino]-3-methylbutanoyl]-4-hydroxy-N-[1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]cyclopropyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(C3(NC(=O)[C@@H]4C[C@@H](O)CN4C(=O)[C@@H](NC(=O)C4=CC=C(COC5=C(C6=C(C)C(F)=CC7=C6C=NN7)C(C6CC6)=CC6=C5N=C(OC5CCOCC5)N=C6N5C[C@@H]6C[C@H]5CN6)C=C4)C(C)C)CC3)C=C2)SC=N1	C60H65FN10O7S	KRAS	P01116	VHL	WO-2023119677-A1
TPD-2ZMHVA	WO2023119677A1_10	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C(C4=CC=C(COC5=C(C6=C(C)C(F)=CC7=C6C=NN7)C(C6CC6)=CC6=C5N=C(OC5CCOCC5)N=C6N5C[C@@H]6C[C@H]5CN6)C=C4)N=N3)C=C2)SC=N1	C59H63FN12O6S	KRAS	P01116	VHL	WO-2023119677-A1
TPD-H4H1YO	WO2023119677A1_11	.	CC1=C(C2=CC=C([C@H](CO)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C(C)C)N3C=C(C4=CC=C(COC5=C(C6=C(C)C(F)=CC7=C6C=NN7)C(C6CC6)=CC6=C5N=C(OC5CCOCC5)N=C6N5C[C@@H]6C[C@H]5CN6)C=C4)C=N3)C=C2)SC=N1	C61H66FN11O7S	KRAS	P01116	VHL	WO-2023119677-A1
TPD-R3YED6	WO2023119677A1_12	.	CC1=C(C2=C(OCC3=CC=C(C4=CN([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](CO)C5=CC=C(Br)C=C5)C(C)C)N=N4)C=C3)C3=C(C=C2C2CC2)C(N2C[C@@H]4C[C@H]2CN4)=NC(OC2CCOCC2)=N3)C2=C(C=C1F)NN=C2	C56H61BrFN11O7	KRAS	P01116	VHL	WO-2023119677-A1
TPD-VLYMHQ	WO2023119677A1_13	.	CC1=C(C2=C(OCC3=CC=C(C4=CN([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](CO)C5=CC=C(F)C=C5)C(C)C)N=N4)C=C3)C3=C(C=C2C2CC2)C(N2C[C@@H]4C[C@H]2CN4)=NC(OC2CCOCC2)=N3)C2=C(C=C1F)NN=C2	C56H61F2N11O7	KRAS	P01116	VHL	WO-2023119677-A1
TPD-HXBXE0	WO2023119677A1_14	.	CC1=C(C2=C(OCC3=CC=C(C4=CN([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](CO)C5=CC=CC=C5)C(C)C)N=N4)C=C3)C3=C(C=C2C2CC2)C(N2C[C@@H]4C[C@H]2CN4)=NC(OC2CCOCC2)=N3)C2=C(C=C1F)NN=C2	C56H62FN11O7	KRAS	P01116	VHL	WO-2023119677-A1
TPD-FE72Z9	WO2023119677A1_15	.	CC1=C(C2=CC=C([C@H](CO)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C(C4=CC=C(COC5=C6N=C(OC7CCOCC7)N=C(N7C[C@@H]8C[C@H]7CN8)C6=CC(C6CC6)=C5C5=CC(O)=CC(F)=C5C)C=C4)N=N3)C=C2)SC=N1	C59H65FN10O8S	KRAS	P01116	VHL	WO-2023119677-A1
TPD-YUSG1X	WO2023119677A1_16	.	CC1=C(C2=CC=C(C(NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C(C4=CC=C(COC5=C(C6=C(C)C(F)=CC7=C6C=NN7)C(C6CC6)=CC6=C5N=C(OC5CCOCC5)N=C6N5C[C@@H]6C[C@H]5CN6)C=C4)N=N3)C(F)F)C=C2)SC=N1	C60H63F3N12O6S	KRAS	P01116	VHL	WO-2023119677-A1
TPD-Y98TTY	WO2023119677A1_17	.	CC1=C(C2=CC=C([C@H](CF)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C(C4=CC=C(COC5=C(C6=C(C)C(F)=CC7=C6C=NN7)C(C6CC6)=CC6=C5N=C(OC5CCOCC5)NC6N5C[C@@H]6C[C@H]5CN6)C=C4)N=N3)C=C2)SC=N1	C60H66F2N12O6S	KRAS	P01116	VHL	WO-2023119677-A1
TPD-XO3MT1	SCHEMBL29859964	(2S,4R)-1-[(2S)-2-[4-[4-[[6-cyclopropyl-4-[(1S,4S)-2,5-diazabicyclo[2.2.1]heptan-2-yl]-7-(6-fluoro-5-methyl-1H-indazol-4-yl)-2-(oxan-4-yloxy)quinazolin-8-yl]oxymethyl]phenyl]triazol-1-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1R)-2-hydroxy-1-[4-[4-(hydroxymethyl)-1,3-thiazol-5-yl]phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=C(OCC3=CC=C(C4=CN([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](CO)C5=CC=C(C6=C(CO)N=CS6)C=C5)C(C)C)N=N4)C=C3)C3=C(C=C2C2CC2)C(N2C[C@@H]4C[C@H]2CN4)=NC(OC2CCOCC2)=N3)C2=C(C=C1F)NN=C2	C60H65FN12O8S	KRAS	P01116	VHL	WO-2023119677-A1
TPD-F3HQIS	WO2023119677A1_19	.	CC1=C(C2=CC=C([C@H](CN(C)C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C(C4=CC=C(COC5=C(C6=C7C=NNC7=CC(F)=C6C)C(C6CC6)=CC6=C(N7C[C@@H]8C[C@H]7CN8)N=C(OC7CCOCC7)N=C65)C=C4)N=N3)C=C2)SC=N1	C62H70FN13O6S	KRAS	P01116	VHL	WO-2023119677-A1
TPD-H4P0SW	WO2023119677A1_2	.	CC1=C(C2=CC=C(C3(NC(=O)C4C[C@@H](O)CN4C(=O)[C@@H](NC(=O)C4=NC=C(COC5=C(C6=C(C)C(F)=CC7=C6C=NN7)C(C6CC6)=CC6=C5N=C(OC5CCOCC5)N=C6N5C[C@@H]6C[C@H]5CN6)C=C4)C(C)C)CC3)C=C2)SC=N1	C59H64FN11O7S	KRAS	P01116	VHL	WO-2023119677-A1
TPD-D3RPQ7	WO2023119677A1_20	.	CC1=C(C2=C(OCC3=CC=C(/C(=C/N(C)[C@H](C(=O)N4C[C@H](O)CC4C(=O)N[C@@H](CO)C4=CC=C(N5CCOC5=O)C=C4)C(C)C)N=N)C=C3)C3=C(C=C2C2CC2)C(N2C[C@@H]4C[C@H]2CN4)=NC(OC2CCOCC2)=N3)C2=C(C=C1F)NN=C2	C60H69FN12O9	KRAS	P01116	VHL	WO-2023119677-A1
TPD-2AHVTI	SCHEMBL26963168	(2S,4R)-1-[(2S)-2-[4-[4-[[6-cyclopropyl-4-[(1S,4S)-2,5-diazabicyclo[2.2.1]heptan-2-yl]-2-[1-(2,2-difluoroethyl)piperidin-4-yl]oxy-7-(6-fluoro-5-methyl-1H-indazol-4-yl)quinazolin-8-yl]oxymethyl]phenyl]triazol-1-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1R)-2-hydroxy-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL29860048	CC1=C(C2=CC=C([C@H](CO)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C(C4=CC=C(COC5=C6N=C(OC7CCN(CC(F)F)CC7)N=C(N7C[C@@H]8C[C@H]7CN8)C6=CC(C6CC6)=C5C5=C(C)C(F)=CC6=C5C=NN6)C=C4)N=N3)C=C2)SC=N1	C62H68F3N13O6S	KRAS	P01116	VHL	WO-2023119677-A1
TPD-8CEMGT	SCHEMBL26963152	(2S,4R)-1-[(2S)-2-[4-[4-[[6-cyclopropyl-4-[(1S,4S)-2,5-diazabicyclo[2.2.1]heptan-2-yl]-7-(6-fluoro-5-methyl-1H-indazol-4-yl)-2-(oxan-4-yloxy)quinazolin-8-yl]oxymethyl]phenyl]triazol-1-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1R)-2-hydroxy-1-[4-(2-methylpyrazol-3-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL29859893	CC1=C(F)C=C2NN=CC2=C1C1=C(OCC2=CC=C(C3=CN([C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)N[C@@H](CO)C4=CC=C(C5=CC=NN5C)C=C4)C(C)C)N=N3)C=C2)C2=NC(OC3CCOCC3)=NC(N3C[C@@H]4C[C@H]3CN4)=C2C=C1C1CC1	C60H66FN13O7	KRAS	P01116	VHL	WO-2023119677-A1
TPD-Q4A25Q	WO2023119677A1_24	.	CC1=C(C2=CC=C([C@H](CO)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C(C4=CC=C(COC5=C6N=C(OC7CCN(C8COC8)CC7)N=C(N7C[C@@H]8C[C@H]7CN8)C6=CC(C6CC6)=C5C5=C(C)C(F)=CC6=C5C=NN6)C=C4)N=N3)C=C2)SC=N1	C63H70FN13O7S	KRAS	P01116	VHL	WO-2023119677-A1
TPD-JMIPR9	WO2023119677A1_25	.	CCC1=CC=NC=C1OC1=NC2=C(OCC3=CC=C(C4=CN([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](CO)C5=CC=C(C6=C(C)N=CS6)C=C5)C(C)C)N=N4)C=C3)C(C3=C(C)C(F)=CC4=C3C=NN4)=C(C3CC3)C=C2C(N2C[C@@H]3C[C@H]2CN3)=N1	C62H64FN13O6S	KRAS	P01116	VHL	WO-2023119677-A1
TPD-YBMOOR	WO2023119677A1_26	.	CCN1N=CC=C1C1=CC=C([C@H](CO)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](C(C)C)N2C=NC(C3=CC=C(COC4=C(C5=C(C)C(F)=CC6=C5C=NN6)C(C5CC5)=CC5=C4N=C(OC4CCOCC4)N=C5N4C[C@@H]5C[C@H]4CN5)C=C3)=C2)C=C1	C62H69FN12O7	KRAS	P01116	VHL	WO-2023119677-A1
TPD-S2NTJ4	WO2023119677A1_27	.	CC1=C(C2=CC=C([C@H](CO)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C(C4=CC=C(COC5=C(C6=C(C)C(F)=CC7=C6C=NN7)C(C6CC6)=CC6=C5N=C(OC5COC5)N=C6N5C[C@@H]6C[C@H]5CN6)C=C4)N=N3)C=C2)SC=N1	C58H61FN12O7S	KRAS	P01116	VHL	WO-2023119677-A1
TPD-M1R6IF	WO2023119677A1_28	.	CC1=C(C2=CC=C([C@H](CO)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C(C4=CC=C(COC5=C(C6=C(C)C(F)=CC7=C6C=NN7)C(C6CC6)=CC6=C5N=C(O[C@@H]5CCOC5)N=C6N5C[C@@H]6C[C@H]5CN6)C=C4)N=N3)C=C2)SC=N1	C59H63FN12O7S	KRAS	P01116	VHL	WO-2023119677-A1
TPD-5V5D7X	WO2023119677A1_29	.	CC1=C(C2=CC=C([C@H](CO)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C(C4=CC=C(COC5=C(C6=C(C)C(F)=CC7=C6C=NN7)C(C6CC6)=CC6=C5N=C(O[C@H]5CCOC5)N=C6N5C[C@@H]6C[C@H]5CN6)C=C4)N=N3)C=C2)SC=N1	C59H63FN12O7S	KRAS	P01116	VHL	WO-2023119677-A1
TPD-2S4IEO	WO2023119677A1_3	(2S,4R)-1-[(2S)-2-[[4-[[6-cyclopropyl-4-[(1S,4S)-2,5-diazabicyclo[2.2.1]heptan-2-yl]-7-(6-fluoro-5-methyl-1H-indazol-4-yl)-2-(oxan-4-yloxy)quinazolin-8-yl]oxymethyl]benzoyl]amino]-3-methylbutanoyl]-4-hydroxy-N-[(1R)-2-hydroxy-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CO)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3=CC=C(COC4=C(C5=C(C)C(F)=CC6=C5C=NN6)C(C5CC5)=CC5=C4N=C(OC4CCOCC4)N=C5N4C[C@@H]5C[C@H]4CN5)C=C3)C(C)C)C=C2)SC=N1	C59H65FN10O8S	KRAS	P01116	VHL	WO-2023119677-A1
TPD-Z8845T	WO2023119677A1_4	.	CC1=C(C2=CC=C([C@H](CO)NC(=O)C3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3CC4=C(C=CC(COC5=C(C6=C(C)C(F)=CC7=C6C=NN7)C(C6CC6)=CC6=C5N=C(OC5CCOCC5)N=C6N5C[C@@H]6C[C@H]5CN6)=C4)C3=O)C=C2)SC=N1	C60H65FN10O8S	KRAS	P01116	VHL	WO-2023119677-A1
TPD-C1633M	WO2023119677A1_5	.	CCOC1=NC2=C(C=C(C3CC3)C(C3=C(C)C(F)=CC4=C3C=NN4)=C2OCC2=CC=C(C(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](CO)C3=CC=C(C4=C(C)N=CS4)C=C3)C(C)C)C=C2)C(N2C[C@@H]3C[C@H]2CN3)=N1	C56H61FN10O7S	KRAS	P01116	VHL	WO-2023119677-A1
TPD-JP5NYO	WO2023119677A1_6	.	CC1=C(C2=CC=C(C3(NC(=O)C4C[C@@H](O)CN4C(=O)C(C(C)C)N4C=C(C5=CC=C(COC6=C(C7=C(C)C(F)=CC8=C7C=NN8)C(C7CC7)=CC7=C6N=C(OC6CCOCC6)N=C7N6C[C@@H]7C[C@H]6CN7)C=C5)N=N4)CC3)C=C2)SC=N1	C61H65FN12O6S	KRAS	P01116	VHL	WO-2023119677-A1
TPD-GQZTKK	KRAS G12D inhibitor 17	KRAS G12D inhibitor 17; Setidegrasib; 2821793-99-9; setidegrasib [INN]; 3NQ4ME292X; orb1982739; SCHEMBL26963151; SCHEMBL29860092; EX-A11454; DA-54678; HY-148273; CS-0618100; EN300-44826014; (2S,4R)-1-[(2S)-2-(4-{4-[({6-cyclopropyl-4-[(1S,4S)-2,5-diazabicyclo[2.2.1]heptan-2-yl]-7-(6-fluoro-5-methyl-1H-indazol-4-yl)-2-(oxan-4-yloxy)quinazolin-8-yl}oxy)methyl]phenyl}-1H-1,2,3-triazol-1-yl)-3-methylbutanoyl]-4-hydroxy-N-[(1R)-2-hydroxy-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; (2S,4R)-1-[(2S)-2-[4-[4-[[6-cyclopropyl-4-[(1S,4S)-2,5-diazabicyclo[2.2.1]heptan-2-yl]-7-(6-fluoro-5-methyl-1H-indazol-4-yl)-2-(oxan-4-yloxy)quinazolin-8-yl]oxymethyl]phenyl]triazol-1-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1R)-2-hydroxy-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; 2-Pyrrolidinecarboxamide, 1-[(2S)-2-[4-[4-[[[6-cyclopropyl-4-(1S,4S)-2,5-diazabicyclo[2.2.1]hept-2-yl-7-(6-fluoro-5-methyl-1H-indazol-4-yl)-2-[(tetrahydro-2H-pyran-4-yl)oxy]-8-quinazolinyl]oxy]methyl]phenyl]-1H-1,2,3-triazol-1-yl]-3-methyl-1-oxobutyl]-4-hydroxy-N-[(1R)-2-hydroxy-1-[4-(4-methyl-5-thiazolyl)phenyl]ethyl]-, (2S,4R)-	CC1=C(C2=CC=C([C@H](CO)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C(C4=CC=C(COC5=C(C6=C(C)C(F)=CC7=C6C=NN7)C(C6CC6)=CC6=C5N=C(OC5CCOCC5)N=C6N5C[C@@H]6C[C@H]5CN6)C=C4)N=N3)C=C2)SC=N1	C60H65FN12O7S	KRAS	P01116	VHL	WO-2023119677-A1
TPD-JKHE43	WO2023119677A1_9	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)C3C=C(C4=CC=C(COC5=C(C6=C(C)C(F)=CC7=C6C=NN7)C(C6CC6)=CC6=C5N=C(OC5CCOCC5)N=C6N5C[C@@H]6C[C@H]5CN6)C=C4)N=N3)C=C2)SC=N1	C61H66FN11O6S	KRAS	P01116	VHL	WO-2023119677-A1
TPD-HUF9L7	SCHEMBL31143458	(3R)-3-[4-[4-[3-[4-[[5-bromo-4-[(5-dimethylphosphoryl-3-fluoro-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]piperidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(C)C(F)=C4)=N2)=C(OC)C=C1N1CCC2(CC1)CCN(C1CCN(C3=CC(F)=C([C@H]4CCC(=O)NC4=O)C(F)=C3)CC1)CC2	C50H58BrF3N9O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-N0LWA9	WO2023138607A1_10	(3R)-3-[4-[4-[4-[1-[4-[[5-bromo-4-[(5-dimethylphosphoryl-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]piperidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(C)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(C3CCN(C4=CC(F)=C([C@H]5CCC(=O)NC5=O)C(F)=C4)CC3)CC2)CC1	C50H60BrF2N10O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-RCZ6W2	WO2023138607A1_101	(3R)-3-[4-[3-[[3-[4-[[5-bromo-4-[(5-dimethylphosphoryl-2-ethylquinazolin-6-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]methyl]azetidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=NC2=C(C=N1)C(P(C)(C)=O)=C(NC1=NC(NC3=C(OC)C=C(N4CCC5(CCN(CC6CN(C7=CC(F)=C([C@H]8CCC(=O)NC8=O)C(F)=C7)C6)CC5)CC4)C(C)=C3)=NC=C1Br)C=C2	C48H56BrF2N10O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-87UQ4E	WO2023138607A1_102	(3R)-3-[4-[4-[3-[4-[[5-bromo-4-[(5-dimethylphosphoryl-2-ethylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]piperidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=NC2=C(C=C1)C(P(C)(C)=O)=C(NC1=NC(NC3=C(OC)C=C(N4CCC5(CC4)CCN(C4CCN(C6=CC(F)=C([C@H]7CCC(=O)NC7=O)C(F)=C6)CC4)CC5)C(C)=C3)=NC=C1Br)C=C2	C50H59BrF2N9O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-EBS66F	WO2023138607A1_103	(3R)-3-[4-[2-[3-[4-[[5-bromo-4-[(5-dimethylphosphoryl-2-ethylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]ethylamino]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=NC2=C(C=C1)C(P(C)(C)=O)=C(NC1=NC(NC3=C(OC)C=C(N4CCC5(CCN(CCNC6=CC(F)=C([C@H]7CCC(=O)NC7=O)C(F)=C6)CC5)CC4)C(C)=C3)=NC=C1Br)C=C2	C47H55BrF2N9O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-C725HM	WO2023138607A1_104	(3R)-3-[4-[2-[3-[4-[[5-bromo-4-[(5-dimethylphosphoryl-2-ethylquinazolin-6-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]ethylamino]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=NC2=C(C=N1)C(P(C)(C)=O)=C(NC1=NC(NC3=C(OC)C=C(N4CCC5(CCN(CCNC6=CC(F)=C([C@H]7CCC(=O)NC7=O)C(F)=C6)CC5)CC4)C(C)=C3)=NC=C1Br)C=C2	C46H54BrF2N10O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-YODJ9K	WO2023138607A1_105	.	CCC1=NC2=C(C=C1)C(P(C)(C)=O)=C(NC1NC(NC3=C(OC)C=C(N4CCC5(CCN(CCCC6=C7C(=CC=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC5)CC4)C(C)=C3)=NC=C1Br)C=C2	C50H62BrN10O5P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-7PJMVV	WO2023138607A1_106	3-[4-[3-[3-[4-[[5-Bromo-4-[(5-dimethylphosphoryl-2-ethylquinazolin-6-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]propyl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	CCC1=NC2=C(C=N1)C(P(C)(C)=O)=C(NC1=NC(NC3=C(OC)C=C(N4CCC5(CCN(CCCC6=C7C(=CC=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC5)CC4)C(C)=C3)=NC=C1Br)C=C2	C49H59BrN11O5P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-P96KFI	WO2023138607A1_107	.	COC1=C(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(C)C=C4)=N2)C=C(C)C(N2CCC3(CCN(CCC4=C5C(=CC=C4)N(C4CCC(=O)NC4=O)C(=O)N5C)CC3)CC2)=C1	C48H56BrN10O5P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-K66J7Q	WO2023138607A1_108	3-[4-[2-[3-[4-[[5-Bromo-4-[(5-dimethylphosphoryl-2-ethylquinazolin-6-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]ethyl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	CCC1=NC2=C(C=N1)C(P(C)(C)=O)=C(NC1=NC(NC3=C(OC)C=C(N4CCC5(CCN(CCC6=C7C(=CC=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC5)CC4)C(C)=C3)=NC=C1Br)C=C2	C48H57BrN11O5P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-S98D58	WO2023138607A1_109	(3R)-3-[4-[3-[[2-[4-[[5-chloro-4-[(5-dimethylphosphoryl-2-ethylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]-2,6-diazaspiro[3.3]heptan-6-yl]methyl]azetidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=NC2=CC=C(NC3=NC(NC4=C(OC)C=C(N5CC6(CN(CC7CN(C8=CC(F)=C([C@H]9CCC(=O)NC9=O)C(F)=C8)C7)C6)C5)C(C)=C4)=NC=C3Cl)C(P(C)(C)=O)=C2C=C1	C45H49ClF2N9O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-QAC1BF	SCHEMBL31143302	(3R)-3-[4-[4-[1-[1-[4-[[5-bromo-4-[(5-dimethylphosphoryl-2-ethylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperidin-4-yl]piperazin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=NC2=CC=C(NC3=NC(NC4=CC(CC)=C(N5CCC(N6CCC(N7CCN(C8=CC(F)=C([C@H]9CCC(=O)NC9=O)C(F)=C8)CC7)CC6)CC5)C=C4OC)=NC=C3Br)C(P(C)(C)=O)=C2C=C1	C51H62BrF2N10O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-U0T9TG	WO2023138607A1_110	(3R)-3-[4-[3-[[2-[4-[[5-chloro-4-[(5-dimethylphosphoryl-2-ethylquinazolin-6-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]-2,6-diazaspiro[3.3]heptan-6-yl]methyl]azetidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=NC2=CC=C(NC3=NC(NC4=C(OC)C=C(N5CC6(CN(CC7CN(C8=CC(F)=C([C@H]9CCC(=O)NC9=O)C(F)=C8)C7)C6)C5)C(C)=C4)=NC=C3Cl)C(P(C)(C)=O)=C2C=N1	C44H48ClF2N10O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-R6T49D	WO2023138607A1_111	(3R)-3-[4-[4-[2-[4-[[5-chloro-4-[(5-dimethylphosphoryl-3-fluoro-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]-2,6-diazaspiro[3.3]heptan-6-yl]piperidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=CC=C4N=C(C)C(F)=CC4=C3P(C)(C)=O)=N2)C=C(C)C(N2CC3(C2)CN(C2CCN(C4=CC(F)=C([C@H]5CCC(=O)NC5=O)C(F)=C4)CC2)C3)=C1	C45H48ClF3N9O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-61WJA1	WO2023138607A1_112	(3R)-3-[4-[4-[2-[4-[[5-chloro-4-[(5-dimethylphosphoryl-2-ethylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]-2,6-diazaspiro[3.3]heptan-6-yl]piperidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=NC2=CC=C(NC3=NC(NC4=C(OC)C=C(N5CC6(C5)CN(C5CCN(C7=CC(F)=C([C@H]8CCC(=O)NC8=O)C(F)=C7)CC5)C6)C(C)=C4)=NC=C3Cl)C(P(C)(C)=O)=C2C=C1	C46H51ClF2N9O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-QB3VVL	WO2023138607A1_113	3-[4-[3-[2-[4-[[5-Chloro-4-[(5-dimethylphosphoryl-3-fluoro-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]-2,6-diazaspiro[3.3]heptan-6-yl]propyl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=CC=C4N=C(C)C(F)=CC4=C3P(C)(C)=O)=N2)C=C(C)C(N2CC3(CN(CCCC4=C5C(=CC=C4)N(C4CCC(=O)NC4=O)C(=O)N5C)C3)C2)=C1	C45H49ClFN10O5P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-5PRH81	WO2023138607A1_114	3-[4-[3-[2-[4-[[5-Chloro-4-[(5-dimethylphosphoryl-2-ethylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]-2,6-diazaspiro[3.3]heptan-6-yl]propyl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	CCC1=NC2=CC=C(NC3=NC(NC4=C(OC)C=C(N5CC6(CN(CCCC7=C8C(=CC=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)C6)C5)C(C)=C4)=NC=C3Cl)C(P(C)(C)=O)=C2C=C1	C46H52ClN10O5P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-DN269C	WO2023138607A1_115	.	CCC1N=CC2=C(P(C)(C)=O)C(NC3=NC(NC4=C(OC)C=C(N5CC6(C5)CN(C5CCN(C7=CC(F)=C([C@H]8CCC(=O)NC8=O)C(F)=C7)CC5)C6)C(C)=C4)=NC=C3Cl)=CC=C2N1	C45H52ClF2N10O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-UDSSFY	WO2023138607A1_116	(3R)-3-[4-[4-[2-[4-[[5-chloro-4-[(5-dimethylphosphoryl-2-methylquinazolin-6-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]-2,6-diazaspiro[3.3]heptan-6-yl]piperidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=CC=C4N=C(C)N=CC4=C3P(C)(C)=O)=N2)C=C(C)C(N2CC3(C2)CN(C2CCN(C4=CC(F)=C([C@H]5CCC(=O)NC5=O)C(F)=C4)CC2)C3)=C1	C44H48ClF2N10O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-F4OZ7O	WO2023138607A1_117	3-[4-[2-[2-[4-[[5-Chloro-4-[(5-dimethylphosphoryl-3-fluoro-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]-2,6-diazaspiro[3.3]heptan-6-yl]ethyl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=CC=C4N=C(C)C(F)=CC4=C3P(C)(C)=O)=N2)C=C(C)C(N2CC3(CN(CCC4=C5C(=CC=C4)N(C4CCC(=O)NC4=O)C(=O)N5C)C3)C2)=C1	C44H47ClFN10O5P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-MF3BG9	WO2023138607A1_118	3-[4-[2-[2-[4-[[5-Chloro-4-[(5-dimethylphosphoryl-2-ethylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]-2,6-diazaspiro[3.3]heptan-6-yl]ethyl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	CCC1=NC2=CC=C(NC3=NC(NC4=C(OC)C=C(N5CC6(CN(CCC7=C8C(=CC=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)C6)C5)C(C)=C4)=NC=C3Cl)C(P(C)(C)=O)=C2C=C1	C45H50ClN10O5P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-CXDR90	WO2023138607A1_119	3-[4-[4-[2-[4-[[5-Chloro-4-[(5-dimethylphosphoryl-3-fluoro-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]-2,6-diazaspiro[3.3]heptan-6-yl]piperidin-1-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=CC=C4N=C(C)C(F)=CC4=C3P(C)(C)=O)=N2)C=C(C)C(N2CC3(C2)CN(C2CCN(C4=C5C(=CC=C4)N(C4CCC(=O)NC4=O)C(=O)N5C)CC2)C3)=C1	C47H52ClFN11O5P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-6WA3AJ	SCHEMBL31143280	(3R)-3-[4-[4-[1-[1-[4-[[5-chloro-4-[(5-dimethylphosphoryl-3-fluoro-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperidin-4-yl]piperazin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Cl)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(C)C(F)=C4)=N2)=C(OC)C=C1N1CCC(N2CCC(N3CCN(C4=CC(F)=C([C@H]5CCC(=O)NC5=O)C(F)=C4)CC3)CC2)CC1	C50H59ClF3N10O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-KQOA8M	WO2023138607A1_120	3-[4-[4-[2-[4-[[5-Chloro-4-[(5-dimethylphosphoryl-2-ethylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]-2,6-diazaspiro[3.3]heptan-6-yl]piperidin-1-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	CCC1=NC2=CC=C(NC3=NC(NC4=C(OC)C=C(N5CC6(C5)CN(C5CCN(C7=C8C(=CC=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)CC5)C6)C(C)=C4)=NC=C3Cl)C(P(C)(C)=O)=C2C=C1	C48H55ClN11O5P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-VVUWF9	WO2023138607A1_121	(3R)-3-[4-[4-[3-[4-[[5-bromo-4-[(5-dimethylphosphoryl-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]piperidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=C(N2CCC3(CC2)CCN(C2CCN(C4=CC(F)=C([C@H]5CCC(=O)NC5=O)C(F)=C4)CC2)CC3)C=C(OC)C(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(C)C=C4)=N2)=C1	C50H59BrF2N9O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-076EBP	SCHEMBL31143313	(3R)-3-[4-[4-[3-[4-[[5-bromo-4-[(5-dimethylphosphoryl-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]piperidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	COC1=CC(N2CCC3(CC2)CCN(C2CCN(C4=CC(F)=C([C@H]5CCC(=O)NC5=O)C(F)=C4)CC2)CC3)=C(C)C=C1NC1=NC=C(Br)C(NC2=C(P(C)(C)=O)C3=C(C=C2)N=C(C)C=C3)=N1	C49H57BrF2N9O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-GVDB04	WO2023138607A1_123	(3R)-3-[4-[4-[3-[4-[[5-chloro-4-[(5-dimethylphosphoryl-2-ethylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]piperidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=NC2=C(C=C1)C(P(C)(C)=O)=C(NC1=NC(NC3=CC(C)=C(N4CCC5(CC4)CCN(C4CCN(C6=CC(F)=C([C@H]7CCC(=O)NC7=O)C(F)=C6)CC4)CC5)C=C3OC)=NC=C1Cl)C=C2	C50H59ClF2N9O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-9O4S67	WO2023138607A1_125	(3R)-3-[4-[4-[3-[4-[[5-bromo-4-[(5-dimethylphosphoryl-2-ethylquinazolin-6-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]piperidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=NC2=C(C=N1)C(P(C)(C)=O)=C(NC1=NC(NC3=CC(C)=C(N4CCC5(CC4)CCN(C4CCN(C6=CC(F)=C([C@H]7CCC(=O)NC7=O)C(F)=C6)CC4)CC5)C=C3OC)=NC=C1Br)C=C2	C49H58BrF2N10O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-6UASYA	WO2023138607A1_126	3-[4-[4-[3-[4-[[5-Bromo-4-[(5-dimethylphosphoryl-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]piperidin-1-yl]-2-fluorophenyl]piperidine-2,6-dione	COC1=CC(N2CCC3(CC2)CCN(C2CCN(C4=CC=C(C5CCC(=O)NC5=O)C(F)=C4)CC2)CC3)=C(C)C=C1NC1=NC=C(Br)C(NC2=C(P(C)(C)=O)C3=C(C=C2)N=C(C)C=C3)=N1	C49H58BrFN9O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-L1T21D	WO2023138607A1_127	3-[4-[4-[3-[4-[[5-Bromo-4-[(5-dimethylphosphoryl-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]piperidin-1-yl]phenyl]piperidine-2,6-dione	COC1=CC(N2CCC3(CC2)CCN(C2CCN(C4=CC=C(C5CCC(=O)NC5=O)C=C4)CC2)CC3)=C(C)C=C1NC1=NC=C(Br)C(NC2=C(P(C)(C)=O)C3=C(C=C2)N=C(C)C=C3)=N1	C49H59BrN9O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-HK2PFF	WO2023138607A1_128	3-[4-[4-[3-[4-[[5-Bromo-4-[(5-dimethylphosphoryl-2-ethylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]piperidin-1-yl]phenyl]piperidine-2,6-dione	CCC1=NC2=C(C=C1)C(P(C)(C)=O)=C(NC1=NC(NC3=CC(C)=C(N4CCC5(CC4)CCN(C4CCN(C6=CC=C(C7CCC(=O)NC7=O)C=C6)CC4)CC5)C=C3OC)=NC=C1Br)C=C2	C50H61BrN9O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-ASTH12	WO2023138607A1_129	3-[4-[4-[2-[4-[[5-Bromo-4-[(5-dimethylphosphoryl-3-fluoro-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]-2,6-diazaspiro[3.3]heptan-6-yl]piperidin-1-yl]-2-fluorophenyl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Br)C(NC3=CC=C4N=C(C)C(F)=CC4=C3P(C)(C)=O)=N2)C=C(C)C(N2CC3(C2)CN(C2CCN(C4=CC=C(C5CCC(=O)NC5=O)C(F)=C4)CC2)C3)=C1	C45H49BrF2N9O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-PBXINV	WO2023138607A1_13	.	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(CC)NC4)=N2)=C(OC)C=C1N1CCC(N2CC(N3CCC(C4=CC(F)=C([C@H]5CCC(=O)NC5=O)C(F)=C4)CC3)C2)CC1	C49H60BrF2N10O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-AZVDED	WO2023138607A1_130	3-[4-[4-[2-[4-[[5-Chloro-4-[(5-dimethylphosphoryl-3-fluoro-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]-2,6-diazaspiro[3.3]heptan-6-yl]piperidin-1-yl]phenyl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Cl)C(NC3=CC=C4N=C(C)C(F)=CC4=C3P(C)(C)=O)=N2)C=C(C)C(N2CC3(C2)CN(C2CCN(C4=CC=C(C5CCC(=O)NC5=O)C=C4)CC2)C3)=C1	C45H50ClFN9O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-423AXH	WO2023138607A1_131	3-[4-[4-[2-[4-[[5-Chloro-4-[(5-dimethylphosphoryl-2-ethylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]-2,6-diazaspiro[3.3]heptan-6-yl]piperidin-1-yl]phenyl]piperidine-2,6-dione	CCC1=NC2=CC=C(NC3=NC(NC4=C(OC)C=C(N5CC6(C5)CN(C5CCN(C7=CC=C(C8CCC(=O)NC8=O)C=C7)CC5)C6)C(C)=C4)=NC=C3Cl)C(P(C)(C)=O)=C2C=C1	C46H53ClN9O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-T02Z8E	WO2023138607A1_132	.	COC1=CC(N2CCC3(CCN(CC4CCN(C5=CC=C(C6CCC(=O)NC6=O)C(F)=C5)CC4)CC3)CC2)=C(C)C=C1NC1=NC=C(Br)C(NC2=C(P(C)(C)=O)C3=C(C=C2)NC(C)C(F)=C3)=N1	C50H61BrF2N9O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-HUJROW	WO2023138607A1_133	3-[4-[4-[[3-[4-[[5-Bromo-4-[(5-dimethylphosphoryl-3-fluoro-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]methyl]piperidin-1-yl]phenyl]piperidine-2,6-dione	COC1=CC(N2CCC3(CCN(CC4CCN(C5=CC=C(C6CCC(=O)NC6=O)C=C5)CC4)CC3)CC2)=C(C)C=C1NC1=NC=C(Br)C(NC2=C(P(C)(C)=O)C3=C(C=C2)N=C(C)C(F)=C3)=N1	C50H60BrFN9O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-TPILKV	WO2023138607A1_134	3-[4-[4-[[3-[4-[[5-Bromo-4-[(5-dimethylphosphoryl-2-ethylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]methyl]piperidin-1-yl]-2-fluorophenyl]piperidine-2,6-dione	CCC1=NC2=C(C=C1)C(P(C)(C)=O)=C(NC1=NC(NC3=CC(C)=C(N4CCC5(CCN(CC6CCN(C7=CC=C(C8CCC(=O)NC8=O)C(F)=C7)CC6)CC5)CC4)C=C3OC)=NC=C1Br)C=C2	C51H62BrFN9O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-0152HI	WO2023138607A1_135	3-[4-[4-[[3-[4-[[5-Bromo-4-[(5-dimethylphosphoryl-2-ethylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]methyl]piperidin-1-yl]phenyl]piperidine-2,6-dione	CCC1=NC2=C(C=C1)C(P(C)(C)=O)=C(NC1=NC(NC3=CC(C)=C(N4CCC5(CCN(CC6CCN(C7=CC=C(C8CCC(=O)NC8=O)C=C7)CC6)CC5)CC4)C=C3OC)=NC=C1Br)C=C2	C51H63BrN9O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-MZJPKG	WO2023138607A1_136	3-[4-[3-[[3-[4-[[5-Bromo-4-[(5-dimethylphosphoryl-3-fluoro-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]methyl]azetidin-1-yl]-2-fluorophenyl]piperidine-2,6-dione	COC1=CC(N2CCC3(CCN(CC4CN(C5=CC=C(C6CCC(=O)NC6=O)C(F)=C5)C4)CC3)CC2)=C(C)C=C1NC1=NC=C(Br)C(NC2=C(P(C)(C)=O)C3=C(C=C2)N=C(C)C(F)=C3)=N1	C48H55BrF2N9O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-YQ7SOF	WO2023138607A1_137	3-[4-[3-[[3-[4-[[5-Bromo-4-[(5-dimethylphosphoryl-3-fluoro-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]methyl]azetidin-1-yl]phenyl]piperidine-2,6-dione	COC1=CC(N2CCC3(CCN(CC4CN(C5=CC=C(C6CCC(=O)NC6=O)C=C5)C4)CC3)CC2)=C(C)C=C1NC1=NC=C(Br)C(NC2=C(P(C)(C)=O)C3=C(C=C2)N=C(C)C(F)=C3)=N1	C48H56BrFN9O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-C5PJYV	WO2023138607A1_138	3-[4-[3-[[3-[4-[[5-Bromo-4-[(5-dimethylphosphoryl-2-ethylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]methyl]azetidin-1-yl]-2-fluorophenyl]piperidine-2,6-dione	CCC1=NC2=C(C=C1)C(P(C)(C)=O)=C(NC1=NC(NC3=CC(C)=C(N4CCC5(CCN(CC6CN(C7=CC=C(C8CCC(=O)NC8=O)C(F)=C7)C6)CC5)CC4)C=C3OC)=NC=C1Br)C=C2	C49H58BrFN9O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-94PYBM	WO2023138607A1_139	3-[4-[3-[[3-[4-[[5-Bromo-4-[(5-dimethylphosphoryl-2-ethylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]methyl]azetidin-1-yl]phenyl]piperidine-2,6-dione	CCC1=NC2=C(C=C1)C(P(C)(C)=O)=C(NC1=NC(NC3=CC(C)=C(N4CCC5(CCN(CC6CN(C7=CC=C(C8CCC(=O)NC8=O)C=C7)C6)CC5)CC4)C=C3OC)=NC=C1Br)C=C2	C49H59BrN9O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-5GK1B2	WO2023138607A1_14	.	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(CC)C=C4)=N2)=C(OC)C=C1N1CCC(N2CC(N3CCC(C4=CC(F)=C(C5CCC(=O)NC5=O)C(F)=C4)CC3)C2)CC1	C50H59BrF2N9O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-AZYT42	WO2023138607A1_140	(3R)-3-[4-[4-[3-[4-[[5-bromo-4-[(5-dimethylphosphoryl-2-ethyl-8-fluoroquinolin-6-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]piperidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=NC2=C(C=C1)C(P(C)(C)=O)=C(NC1=NC(NC3=C(OC)C=C(N4CCC5(CC4)CCN(C4CCN(C6=CC(F)=C([C@H]7CCC(=O)NC7=O)C(F)=C6)CC4)CC5)C(C)=C3)=NC=C1Br)C=C2F	C50H58BrF3N9O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-2SMSPO	WO2023138607A1_141	(3R)-3-[4-[2-[3-[4-[[5-bromo-4-[(5-dimethylphosphoryl-2-ethyl-8-fluoroquinolin-6-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]ethyl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=NC2=C(C=C1)C(P(C)(C)=O)=C(NC1=NC(NC3=C(OC)C=C(N4CCC5(CCN(CCC6=CC(F)=C([C@H]7CCC(=O)NC7=O)C(F)=C6)CC5)CC4)C(C)=C3)=NC=C1Br)C=C2F	C47H53BrF3N8O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-JCZI4N	WO2023138607A1_142	(3R)-3-[4-[4-[4-[1-[4-[[5-bromo-4-[(5-dimethylphosphoryl-2-ethylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]piperidin-4-yl]piperazin-1-yl]piperidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=NC2=C(C=C1)C(P(C)(C)=O)=C(NC1=NC(NC3=CC(C)=C(N4CCC(N5CCN(C6CCN(C7=CC(F)=C([C@H]8CCC(=O)NC8=O)C(F)=C7)CC6)CC5)CC4)C=C3OC)=NC=C1Br)C=C2	C50H60BrF2N10O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-SBQ2OG	WO2023138607A1_15	.	CCOC1=C(NC2=NC=C(Cl)C(N/C(C)=C(/C3=C(C)N=C(C)C(F)=C3)P(C)(C)=O)=N2)C=C(CC)C(N2CCC(N3CC(N4CCC(C5=CC(F)=C(C6CCC(=O)NC6=O)C(F)=C5)CC4)C3)CC2)=C1	C50H62ClF3N9O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-ZQG57U	WO2023138607A1_16	.	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(C)C(F)=C4)=N2)=C(OC)C=C1N1CCC(N2CC(N3CCN(C4=CC(F)=C(C5CCC(=O)NC5=O)C(F)=C4)CC3)C2)CC1	C48H55BrF3N10O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-AF6SOV	WO2023138607A1_17	.	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(C)C(F)=C4)=N2)=C(OC)C=C1N1CCC(N2CCC3(CCN(C4=CC(F)=C(C5CCC(=O)NC5=O)C(F)=C4)C3)C2)CC1	C48H54BrF3N9O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-773KH3	WO2023138607A1_18	.	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4C=C(F)C(C)=NC4C=C3)=N2)=C(OC)C=C1N1CCC(N2CC3(CCN(C4=CC(F)=C([C@H]5CCC(=O)NC5=O)C(F)=C4)CC3)C2)CC1	C48H56BrF3N9O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-EU1I2K	WO2023138607A1_19	.	CCOC1=CC(N2CCC(N3CCC4(CC3)CN(C3=CC(F)=C([C@H]5CCC(=O)NC5=O)C(F)=C3)C4)CC2)=C(CC)C=C1NC1=NC=C(Br)C(NC2=C(P(C)(C)=O)C3=C(C=C2)N=C(CC)NC3)=N1	C49H60BrF2N10O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-2BUKFR	SCHEMBL31143488	(3R)-3-[4-[4-[3-[4-[[5-chloro-4-[(5-dimethylphosphoryl-3-fluoro-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]piperidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Cl)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(C)C(F)=C4)=N2)=C(OC)C=C1N1CCC2(CC1)CCN(C1CCN(C3=CC(F)=C([C@H]4CCC(=O)NC4=O)C(F)=C3)CC1)CC2	C50H58ClF3N9O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-Q5UUKR	SCHEMBL31143340	(3R)-3-[4-[2-[1-[4-[[5-bromo-4-[(5-dimethylphosphoryl-2-ethylquinazolin-6-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]-2,7-diazaspiro[3.5]nonan-7-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(CC)N=C4)=N2)=C(OC)C=C1N1CCC(N2CC3(CCN(C4=CC(F)=C([C@H]5CCC(=O)NC5=O)C(F)=C4)CC3)C2)CC1	C48H56BrF2N10O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-LGMWA7	WO2023138607A1_21	.	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(C)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(C3CN(C4=C5C(=CC=C4)N(C4CCC(=O)NC4=O)C(=O)N5C)C3)CC2)CC1	C50H60BrN12O5P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-1ZBVUD	SCHEMBL31143461	3-[4-[3-[4-[1-[4-[[5-Bromo-4-[(5-dimethylphosphoryl-3-fluoro-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]azetidin-1-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(C)C(F)=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(C3CN(C4=C5C(=CC=C4)N(C4CCC(=O)NC4=O)C(=O)N5C)C3)CC2)CC1	C50H59BrFN12O5P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-JIDXLL	WO2023138607A1_23	.	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(C)N=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(C3CN(C4=C5C(=CC=C4)N(C4CCC(=O)NC4=O)C(=O)N5C)C3)CC2)CC1	C49H59BrN13O5P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-5KKMPW	SCHEMBL31143506	(3S)-3-[4-[3-[4-[1-[4-[[5-bromo-4-[(5-dimethylphosphoryl-3-fluoro-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazine-1-carbonyl]azetidin-1-yl]-7-fluoro-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(C)C(F)=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(C(=O)C3CN(C4=C5C(=C(F)C=C4)N([C@H]4CCC(=O)NC4=O)C(=O)N5C)C3)CC2)CC1	C51H58BrF2N12O6P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-SCIAJZ	SCHEMBL31143446	3-[4-[6-[1-[4-[[5-Bromo-4-[(5-dimethylphosphoryl-2-ethylquinazolin-6-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]-2,6-diazaspiro[3.3]heptan-2-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(CC)N=C4)=N2)=C(OC)C=C1N1CCC(N2CC3(CN(C4=C5C(=CC=C4)N(C4CCC(=O)NC4=O)C(=O)N5C)C3)C2)CC1	C48H56BrN12O5P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-K1K20K	SCHEMBL31143445	3-[4-[6-[1-[4-[[5-Bromo-4-[(5-dimethylphosphoryl-3-fluoro-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]-2,6-diazaspiro[3.3]heptan-2-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(C)C(F)=C4)=N2)=C(OC)C=C1N1CCC(N2CC3(CN(C4=C5C(=CC=C4)N(C4CCC(=O)NC4=O)C(=O)N5C)C3)C2)CC1	C48H54BrFN11O5P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-PAUSGW	SCHEMBL31143295	(3R)-3-[4-[6-[1-[4-[[5-bromo-4-[(5-dimethylphosphoryl-2-ethylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]-2,6-diazaspiro[3.3]heptan-2-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(CC)C=C4)=N2)=C(OC)C=C1N1CCC(N2CC3(CN(C4=CC(F)=C([C@H]5CCC(=O)NC5=O)C(F)=C4)C3)C2)CC1	C47H53BrF2N9O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-JOAMFM	SCHEMBL31143293	3-[4-[3-[3-[4-[[5-Bromo-4-[(5-dimethylphosphoryl-3-fluoro-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]propyl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(C)C(F)=C4)=N2)=C(OC)C=C1N1CCC2(CCN(CCCC3=C4C(=CC=C3)N(C3CCC(=O)NC3=O)C(=O)N4C)CC2)CC1	C50H59BrFN10O5P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-46475N	WO2023138607A1_29	.	CCC1=CC(NC2=NC=C(Br)C(NC3=C(CP(C)(C)=O)C4=C(C=C3)N=C(C)C(F)=C4)=N2)=C(OC)C=C1N1CCC2(CCN(C(=O)CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)CC1	C53H65BrFN10O5P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-TO36EI	WO2023138607A1_3	.	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(C)N=C4)N2)=C(OC)C=C1N1CCC2(CC1)CCN(C1CCN(C3=CC(F)=C([C@H]4CCC(=O)NC4=O)C(F)=C3)CC1)CC2	C49H60BrF2N10O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-0Y19MM	SCHEMBL31143365	(3R)-3-[4-[1-[1-[1-[4-[[5-bromo-4-[(5-dimethylphosphoryl-2-ethylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperidin-4-yl]azetidin-3-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(CC)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCC(N3CC(C4=CC(F)=C([C@H]5CCC(=O)NC5=O)C(F)=C4)C3)CC2)CC1	C50H59BrF2N9O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-7WTUHP	WO2023138607A1_31	3-[4-[2-[1-[4-[[5-Bromo-4-[(5-dimethylphosphoryl-2-ethylquinazolin-6-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]-2,7-diazaspiro[3.5]nonan-7-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(CC)N=C4)=N2)=C(OC)C=C1N1CCC(N2CC3(CCN(C4=C5C(=CC=C4)N(C4CCC(=O)NC4=O)C(=O)N5C)CC3)C2)CC1	C50H60BrN12O5P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-OCHPM6	WO2023138607A1_32	3-[4-[2-[1-[4-[[5-Chloro-4-[(5-dimethylphosphoryl-3-fluoro-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-5-ethoxy-2-ethylphenyl]piperidin-4-yl]-2,7-diazaspiro[3.5]nonan-7-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	CCOC1=CC(N2CCC(N3CC4(CCN(C5=C6C(=CC=C5)N(C5CCC(=O)NC5=O)C(=O)N6C)CC4)C3)CC2)=C(CC)C=C1NC1=NC=C(Cl)C(NC2=CC=C3N=C(C)C(F)=CC3=C2P(C)(C)=O)=N1	C51H60ClFN11O5P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-KEUL18	SCHEMBL31143311	3-[7-[3-[[3-[4-[[5-bromo-4-[(5-dimethylphosphoryl-3-fluoro-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]methyl]azetidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(C)C(F)=C4)=N2)=C(OC)C=C1N1CCC2(CCN(CC3CN(C4=C5CN(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C3)CC2)CC1	C51H59BrFN10O5P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-BM6EVQ	SCHEMBL31143344	3-[7-[2-[3-[4-[[5-bromo-4-[(5-dimethylphosphoryl-3-fluoro-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]ethyl-methylamino]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(C)C(F)=C4)=N2)=C(OC)C=C1N1CCC2(CCN(CCN(C)C3=CC=CC4=C3CN(C3CCC(=O)NC3=O)C4=O)CC2)CC1	C50H59BrFN10O5P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-VU1L1I	WO2023138607A1_35	.	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(C)N=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(CC3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)CC5=C4)CC3)CC2)CC1	C52H64BrN12O5P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-XNI98F	SCHEMBL31143274	(3R)-3-[4-[4-[3-[4-[[5-bromo-4-[(5-dimethylphosphorylquinoxalin-6-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]piperidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=CC=N4)=N2)C=C(C)C(N2CCC3(CC2)CCN(C2CCN(C4=CC(F)=C([C@H]5CCC(=O)NC5=O)C(F)=C4)CC2)CC3)=C1	C47H54BrF2N10O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-8VBSCN	SCHEMBL31143301	(3R)-3-[4-[4-[3-[4-[[5-bromo-4-[(5-dimethylphosphoryl-3-fluoro-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]piperidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(C)C(F)=C4)=N2)C=C(C)C(N2CCC3(CC2)CCN(C2CCN(C4=CC(F)=C([C@H]5CCC(=O)NC5=O)C(F)=C4)CC2)CC3)=C1	C49H56BrF3N9O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-0A81TJ	SCHEMBL31143269	(3R)-3-[4-[3-[3-[4-[[5-bromo-4-[(5-dimethylphosphoryl-3-fluoro-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]azetidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(C)C(F)=C4)=N2)=C(OC)C=C1N1CCC2(CC1)CCN(C1CN(C3=CC(F)=C([C@H]4CCC(=O)NC4=O)C(F)=C3)C1)CC2	C48H54BrF3N9O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-F8PAMT	SCHEMBL31143334	(3R)-3-[4-[3-[[3-[4-[[5-bromo-4-[(5-dimethylphosphoryl-3-fluoro-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]methyl]azetidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(C)C(F)=C4)=N2)=C(OC)C=C1N1CCC2(CCN(CC3CN(C4=CC(F)=C([C@H]5CCC(=O)NC5=O)C(F)=C4)C3)CC2)CC1	C49H56BrF3N9O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-FZ7I5H	SCHEMBL31143317	(3R)-3-[4-[9-[1-[4-[[5-bromo-4-[(5-dimethylphosphoryl-2-ethylquinazolin-6-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]-3,9-diazaspiro[5.5]undecan-3-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(CC)N=C4)=N2)=C(OC)C=C1N1CCC(N2CCC3(CCN(C4=CC(F)=C([C@H]5CCC(=O)NC5=O)C(F)=C4)CC3)CC2)CC1	C50H60BrF2N10O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-3Q5WNW	SCHEMBL31143289	(3R)-3-[4-[2-[3-[4-[[5-bromo-4-[(5-dimethylphosphoryl-2-ethylquinazolin-6-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]ethyl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(CC)N=C4)=N2)=C(OC)C=C1N1CCC2(CCN(CCC3=CC(F)=C([C@H]4CCC(=O)NC4=O)C(F)=C3)CC2)CC1	C47H55BrF2N9O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-DUQC0Y	SCHEMBL31143478	(3R)-3-[4-[2-[3-[4-[[5-chloro-4-[(5-dimethylphosphoryl-3-fluoro-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]ethyl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Cl)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(C)C(F)=C4)=N2)=C(OC)C=C1N1CCC2(CCN(CCC3=CC(F)=C([C@H]4CCC(=O)NC4=O)C(F)=C3)CC2)CC1	C47H53ClF3N8O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-NPH9G6	SCHEMBL31143268	(3R)-3-[4-[2-[3-[4-[[5-chloro-4-[(5-dimethylphosphoryl-2-ethylquinazolin-6-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]ethyl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=NC2=C(C=N1)C(P(C)(C)=O)=C(NC1=NC(NC3=CC(C)=C(N4CCC5(CCN(CCC6=CC(F)=C([C@H]7CCC(=O)NC7=O)C(F)=C6)CC5)CC4)C=C3OC)=NC=C1Cl)C=C2	C46H53ClF2N9O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-ITKNLI	WO2023138607A1_43	.	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(C)C(F)=C4)=N2)=C(OC)C=C1N1CCC2(CCN(CCNC3=CC(F)C([C@H]4CCC(=O)NC4=O)C(F)=C3)CC2)CC1	C47H56BrF3N9O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-UR731I	SCHEMBL31143325	(3R)-3-[4-[2-[3-[4-[[5-bromo-4-[(5-dimethylphosphoryl-3-fluoro-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]ethyl-methylamino]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(C)C(F)=C4)=N2)=C(OC)C=C1N1CCC2(CCN(CCN(C)C3=CC(F)=C([C@H]4CCC(=O)NC4=O)C(F)=C3)CC2)CC1	C48H56BrF3N9O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-P39KUZ	SCHEMBL31143326	4-[4-[[3-[4-[[5-Bromo-4-[(5-dimethylphosphoryl-3-fluoro-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]methyl]piperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(C)C(F)=C4)=N2)=C(OC)C=C1N1CCC2(CCN(CC3CCN(C4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)CC2)CC1	C53H61BrFN10O6P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-YDNCYO	SCHEMBL31143477	5-[4-[[3-[4-[[5-Bromo-4-[(5-dimethylphosphoryl-3-fluoro-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]methyl]piperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(C)C(F)=C4)=N2)=C(OC)C=C1N1CCC2(CCN(CC3CCN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)CC1	C53H61BrFN10O6P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-WREUO1	SCHEMBL31143391	5-[4-[[3-[4-[[5-Bromo-4-[(5-dimethylphosphoryl-3-fluoro-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]methyl]piperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)-6-fluoroisoindole-1,3-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(C)C(F)=C4)=N2)=C(OC)C=C1N1CCC2(CCN(CC3CCN(C4=C(F)C=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)CC1	C53H60BrF2N10O6P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-3NI5R6	SCHEMBL31143306	3-[6-[4-[[3-[4-[[5-bromo-4-[(5-dimethylphosphoryl-3-fluoro-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(C)C(F)=C4)=N2)=C(OC)C=C1N1CCC2(CCN(CC3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)CC5=C4)CC3)CC2)CC1	C53H63BrFN10O5P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-EEP5V5	SCHEMBL31143328	5-[(3S)-3-[[3-[4-[[5-bromo-4-[(5-dimethylphosphoryl-3-fluoro-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]methyl]pyrrolidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(C)C(F)=C4)=N2)=C(OC)C=C1N1CCC2(CCN(C[C@@H]3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)C3)CC2)CC1	C52H59BrFN10O6P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-S8QBLY	WO2023138607A1_5	.	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(C)C(F)=C4)=N2)=C(OC)C=C1N1CCC2(CC1)CCN(C1CC(C3=CC(F)=C([C@H]4CCC(=O)NC4=O)C(F)C3)C1)CC2	C49H57BrF3N8O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-5M5K6M	SCHEMBL31143297	3-[4-[4-[3-[4-[[5-Bromo-4-[(5-dimethylphosphoryl-3-fluoro-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]piperidin-1-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(C)C(F)=C4)=N2)=C(OC)C=C1N1CCC2(CC1)CCN(C1CCN(C3=C4C(=CC=C3)N(C3CCC(=O)NC3=O)C(=O)N4C)CC1)CC2	C52H62BrFN11O5P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-4EPSJ9	SCHEMBL31143314	3-[4-[4-[3-[4-[[5-Bromo-4-[(5-dimethylphosphoryl-3-fluoro-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]piperidin-1-yl]-3,3-dimethyl-2-oxoindol-1-yl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(C)C(F)=C4)=N2)=C(OC)C=C1N1CCC2(CC1)CCN(C1CCN(C3=C4C(=CC=C3)N(C3CCC(=O)NC3=O)C(=O)C4(C)C)CC1)CC2	C54H65BrFN10O5P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-73GX9T	SCHEMBL25310575	(3R)-3-[4-[4-[4-[1-[4-[[5-chloro-4-[(5-dimethylphosphoryl-3-fluoro-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-5-ethoxy-2-ethylphenyl]piperidin-4-yl]piperazin-1-yl]piperidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione; SCHEMBL31143521	CCOC1=C(NC2=NC=C(Cl)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(C)C(F)=C4)=N2)C=C(CC)C(N2CCC(N3CCN(C4CCN(C5=CC(F)=C([C@H]6CCC(=O)NC6=O)C(F)=C5)CC4)CC3)CC2)=C1	C51H61ClF3N10O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-AXC1YT	WO2023138607A1_55	.	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(CC)NC4)=N2)=C(OC)C=C1N1CCC(N2CC(CN3CCC(C4=CC(F)=C([C@H]5CCC(=O)NC5=O)C(F)=C4)CC3)C2)CC1	C50H62BrF2N10O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-5RKC9O	SCHEMBL25309688	(3R)-3-[4-[1-[[1-[1-[4-[[5-bromo-4-[(5-dimethylphosphoryl-3-fluoro-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]azetidin-3-yl]methyl]piperidin-4-yl]-2,6-difluorophenyl]piperidine-2,6-dione; SCHEMBL31143501	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(C)C(F)=C4)=N2)=C(OC)C=C1N1CCC(N2CC(CN3CCC(C4=CC(F)=C([C@H]5CCC(=O)NC5=O)C(F)=C4)CC3)C2)CC1	C50H58BrF3N9O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-EEGKQB	WO2023138607A1_57	.	CCOC1=C(NC2=NC=C(Cl)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(C)C(F)=C4)=N2)C=C(CC)C(N2CCC(N3CCC4(CC3)CN(C3=CC(F)=C(C5CCC(=O)NC5=O)C(F)=C3)C4)CC2)=C1	C49H56ClF3N9O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-O2B9DV	SCHEMBL31143349	(3R)-3-[4-[2-[1-[4-[[5-bromo-4-[(5-dimethylphosphoryl-2-ethylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]-2,7-diazaspiro[3.5]nonan-7-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(CC)C=C4)=N2)=C(OC)C=C1N1CCC(N2CC3(CCN(C4=CC(F)=C([C@H]5CCC(=O)NC5=O)C(F)=C4)CC3)C2)CC1	C49H57BrF2N9O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-QOOYY9	SCHEMBL31143331	(3R)-3-[4-[2-[1-[4-[[5-chloro-4-[(5-dimethylphosphoryl-3-fluoro-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-5-ethoxy-2-ethylphenyl]piperidin-4-yl]-2,7-diazaspiro[3.5]nonan-7-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCOC1=CC(N2CCC(N3CC4(CCN(C5=CC(F)=C([C@H]6CCC(=O)NC6=O)C(F)=C5)CC4)C3)CC2)=C(CC)C=C1NC1=NC=C(Cl)C(NC2=CC=C3N=C(C)C(F)=CC3=C2P(C)(C)=O)=N1	C49H56ClF3N9O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-X7KLXB	WO2023138607A1_6	.	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(C)C(F)=C4)=N2)=C(O)C=C1N1CCC2(CCN(CCC3=CC(F)=C([C@H]4CCC(=O)NC4=O)C(F)=C3)CC2)CC1	C46H51BrF3N8O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-GFNEEU	WO2023138607A1_60	(3R)-3-[4-[6-[1-[4-[[5-bromo-4-[(5-dimethylphosphoryl-3-fluoro-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]-2,6-diazaspiro[3.3]heptan-2-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(C)C(F)=C4)=N2)=C(OC)C=C1N1CCC(N2CC3(CN(C4=CC(F)=C([C@H]5CCC(=O)NC5=O)C(F)=C4)C3)C2)CC1	C46H50BrF3N9O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-QB9UWQ	SCHEMBL31143315	(3R)-3-[4-[4-[2-[4-[[5-chloro-4-[(5-dimethylphosphoryl-3-fluoro-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]-2,6-diazaspiro[3.3]heptan-6-yl]piperidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Cl)C(NC3=CC=C4N=C(C)C(F)=CC4=C3P(C)(C)=O)=N2)=C(OC)C=C1N1CC2(C1)CN(C1CCN(C3=CC(F)=C([C@H]4CCC(=O)NC4=O)C(F)=C3)CC1)C2	C46H50ClF3N9O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-N6C94V	SCHEMBL31143450	(3R)-3-[4-[4-[7-[4-[[5-bromo-4-[(5-dimethylphosphoryl-3-fluoro-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]-2,7-diazaspiro[3.5]nonan-2-yl]piperidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(C)C(F)=C4)=N2)=C(OC)C=C1N1CCC2(CC1)CN(C1CCN(C3=CC(F)=C([C@H]4CCC(=O)NC4=O)C(F)=C3)CC1)C2	C48H54BrF3N9O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-JVN64J	SCHEMBL31143377	3-[4-[1-[1-[1-[4-[[5-Bromo-4-[(5-dimethylphosphoryl-2-ethylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperidin-4-yl]azetidin-3-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(CC)C=C4)=N2)=C(OC)C=C1N1CCC(N2CCC(N3CC(C4=C5C(=CC=C4)N(C4CCC(=O)NC4=O)C(=O)N5C)C3)CC2)CC1	C52H63BrN11O5P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-KSWUWI	SCHEMBL31143498	(3R)-3-[4-[4-[2-[4-[[5-bromo-4-[(5-dimethylphosphoryl-3-fluoro-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]-2,6-diazaspiro[3.3]heptan-6-yl]piperidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=CC=C4N=C(C)C(F)=CC4=C3P(C)(C)=O)=N2)=C(OC)C=C1N1CC2(C1)CN(C1CCN(C3=CC(F)=C([C@H]4CCC(=O)NC4=O)C(F)=C3)CC1)C2	C46H50BrF3N9O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-ZY0DID	SCHEMBL31143288	(3R)-3-[4-[4-[2-[4-[[5-bromo-4-[(5-dimethylphosphoryl-3-fluoro-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]-2,6-diazaspiro[3.3]heptan-6-yl]piperidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Br)C(NC3=CC=C4N=C(C)C(F)=CC4=C3P(C)(C)=O)=N2)C=C(C)C(N2CC3(C2)CN(C2CCN(C4=CC(F)=C([C@H]5CCC(=O)NC5=O)C(F)=C4)CC2)C3)=C1	C45H48BrF3N9O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-JCS9MP	SCHEMBL31143278	(3R)-3-[4-[4-[3-[4-[[5-bromo-4-[(5-dimethylphosphoryl-2-methylquinazolin-6-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]piperidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(C)N=C4)=N2)C=C(C)C(N2CCC3(CC2)CCN(C2CCN(C4=CC(F)=C([C@H]5CCC(=O)NC5=O)C(F)=C4)CC2)CC3)=C1	C48H56BrF2N10O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-400NHF	WO2023138607A1_68	3-[4-[2-[3-[4-[[5-Bromo-4-[(5-dimethylphosphoryl-2-ethylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]ethyl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	CCC1=NC2=C(C=C1)C(P(C)(C)=O)=C(NC1=NC(NC3=C(OC)C=C(N4CCC5(CCN(CCC6=C7C(=CC=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC5)CC4)C(C)=C3)=NC=C1Br)C=C2	C49H58BrN10O5P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-M93NGC	WO2023138607A1_69	3-[6-[4-[[3-[4-[[5-bromo-4-[(5-dimethylphosphoryl-3-fluoro-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	COC1=C(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(C)C(F)=C4)=N2)C=C(C)C(N2CCC3(CCN(CC4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)CC6=C5)CC4)CC3)CC2)=C1	C52H61BrFN10O5P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-FWA4HD	SCHEMBL31143489	(3R)-3-[4-[3-[4-[1-[4-[[5-bromo-4-[(5-dimethylphosphoryl-2-ethylquinazolin-6-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]azetidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(CC)N=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(C3CN(C4=CC(F)=C([C@H]5CCC(=O)NC5=O)C(F)=C4)C3)CC2)CC1	C48H57BrF2N11O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-WV357G	WO2023138607A1_71	3-[6-[4-[[3-[4-[[5-bromo-4-[(5-dimethylphosphoryl-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CCC1=C(N2CCC3(CCN(CC4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)CC6=C5)CC4)CC3)CC2)C=C(OC)C(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(C)C=C4)=N2)=C1	C53H64BrN10O5P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-4QBZI2	SCHEMBL31143504	3-[6-[4-[[3-[4-[[5-bromo-4-[(5-dimethylphosphoryl-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	COC1=CC(N2CCC3(CCN(CC4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)CC6=C5)CC4)CC3)CC2)=C(C)C=C1NC1=NC=C(Br)C(NC2=C(P(C)(C)=O)C3=C(C=C2)N=C(C)C=C3)=N1	C52H62BrN10O5P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-1PCUYL	WO2023138607A1_73	.	COC1=C(NC2=NC=C(C)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(C)C=C4)=N2)C=C(C)C(N2CCC3(CC2)CCN(C2CCN(C4=CC(F)=C([C@H]5CCC(=O)NC5=O)C(F)=C4)CC2)CC3)=C1	C50H60F2N9O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-MYI76N	WO2023138607A1_74	3-[6-[4-[[2-[4-[[5-chloro-4-[(5-dimethylphosphoryl-3-fluoro-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]-2,6-diazaspiro[3.3]heptan-6-yl]methyl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Cl)C(NC3=CC=C4N=C(C)C(F)=CC4=C3P(C)(C)=O)=N2)=C(OC)C=C1N1CC2(CN(CC3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)CC5=C4)CC3)C2)C1	C49H55ClFN10O5P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-CWVL50	WO2023138607A1_75	(3R)-3-[4-[(3R)-3-[[2-[4-[[5-chloro-4-[(5-dimethylphosphoryl-3-fluoro-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]-2,6-diazaspiro[3.3]heptan-6-yl]methyl]pyrrolidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Cl)C(NC3=CC=C4N=C(C)C(F)=CC4=C3P(C)(C)=O)=N2)=C(OC)C=C1N1CC2(CN(C[C@H]3CCN(C4=CC(F)=C([C@H]5CCC(=O)NC5=O)C(F)=C4)C3)C2)C1	C46H50ClF3N9O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-GBISJ3	WO2023138607A1_76	(3R)-3-[4-[(3S)-3-[[2-[4-[[5-chloro-4-[(5-dimethylphosphoryl-3-fluoro-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]-2,6-diazaspiro[3.3]heptan-6-yl]methyl]pyrrolidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Cl)C(NC3=CC=C4N=C(C)C(F)=CC4=C3P(C)(C)=O)=N2)=C(OC)C=C1N1CC2(CN(C[C@@H]3CCN(C4=CC(F)=C([C@H]5CCC(=O)NC5=O)C(F)=C4)C3)C2)C1	C46H50ClF3N9O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-9RA3GW	WO2023138607A1_77	(3R)-3-[4-[4-[[2-[4-[[5-chloro-4-[(5-dimethylphosphoryl-3-fluoro-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]-2,6-diazaspiro[3.3]heptan-6-yl]methyl]piperidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Cl)C(NC3=CC=C4N=C(C)C(F)=CC4=C3P(C)(C)=O)=N2)=C(OC)C=C1N1CC2(CN(CC3CCN(C4=CC(F)=C([C@H]5CCC(=O)NC5=O)C(F)=C4)CC3)C2)C1	C47H52ClF3N9O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-QX885O	WO2023138607A1_78	(3R)-3-[4-[3-[[2-[4-[[5-chloro-4-[(5-dimethylphosphoryl-3-fluoro-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]-2,6-diazaspiro[3.3]heptan-6-yl]methyl]azetidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Cl)C(NC3=CC=C4N=C(C)C(F)=CC4=C3P(C)(C)=O)=N2)=C(OC)C=C1N1CC2(CN(CC3CN(C4=CC(F)=C([C@H]5CCC(=O)NC5=O)C(F)=C4)C3)C2)C1	C45H48ClF3N9O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-055UZP	SCHEMBL31143440	(3R)-3-[4-[4-[[3-[4-[[5-bromo-4-[(5-dimethylphosphoryl-3-fluoro-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]methyl]piperidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(C)C(F)=C4)=N2)=C(OC)C=C1N1CCC2(CCN(CC3CCN(C4=CC(F)=C([C@H]5CCC(=O)NC5=O)C(F)=C4)CC3)CC2)CC1	C51H60BrF3N9O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-GTHZTM	SCHEMBL31143525	(3R)-3-[4-[3-[4-[1-[4-[[5-bromo-4-[(5-dimethylphosphoryl-3-fluoro-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]azetidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(C)C(F)=C4)=N2)=C(OC)C=C1N1CCC(N2CCN(C3CN(C4=CC(F)=C([C@H]5CCC(=O)NC5=O)C(F)=C4)C3)CC2)CC1	C48H55BrF3N10O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-AOY50A	WO2023138607A1_80	(3R)-3-[4-[(3R)-3-[[3-[4-[[5-bromo-4-[(5-dimethylphosphoryl-3-fluoro-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]methyl]pyrrolidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(C)C(F)=C4)=N2)=C(OC)C=C1N1CCC2(CCN(C[C@H]3CCN(C4=CC(F)=C([C@H]5CCC(=O)NC5=O)C(F)=C4)C3)CC2)CC1	C50H58BrF3N9O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-GVXBBK	WO2023138607A1_81	(3R)-3-[4-[(3S)-3-[[3-[4-[[5-bromo-4-[(5-dimethylphosphoryl-3-fluoro-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]methyl]pyrrolidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(C)C(F)=C4)=N2)=C(OC)C=C1N1CCC2(CCN(C[C@@H]3CCN(C4=CC(F)=C([C@H]5CCC(=O)NC5=O)C(F)=C4)C3)CC2)CC1	C50H58BrF3N9O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-8KYKAE	SCHEMBL31143279	(3S)-3-[4-[3-[3-[4-[[5-bromo-4-[(5-dimethylphosphoryl-3-fluoro-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]propyl]-7-fluoro-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(C)C(F)=C4)=N2)=C(OC)C=C1N1CCC2(CCN(CCCC3=C4C(=C(F)C=C3)N([C@H]3CCC(=O)NC3=O)C(=O)N4C)CC2)CC1	C50H58BrF2N10O5P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-DYHIBR	WO2023138607A1_84	3-[4-[4-[3-[4-[[5-Bromo-4-[(5-dimethylphosphoryl-2-ethylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]piperidin-1-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	CCC1=NC2=C(C=C1)C(P(C)(C)=O)=C(NC1=NC(NC3=C(OC)C=C(N4CCC5(CC4)CCN(C4CCN(C6=C7C(=CC=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC4)CC5)C(C)=C3)=NC=C1Br)C=C2	C52H63BrN11O5P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-ATRXS0	SCHEMBL31143367	3-[7-[2-[3-[4-[[5-Bromo-4-[(5-dimethylphosphoryl-3-fluoro-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]ethyl]-2-oxo-1,3-benzoxazol-3-yl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(C)C(F)=C4)=N2)=C(OC)C=C1N1CCC2(CCN(CCC3=C4OC(=O)N(C5CCC(=O)NC5=O)C4=CC=C3)CC2)CC1	C48H54BrFN9O6P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-3HYCSO	SCHEMBL31143396	3-[4'-[2-[3-[4-[[5-Bromo-4-[(5-dimethylphosphoryl-3-fluoro-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]ethyl]-2'-oxospiro[cyclopropane-1,3'-indole]-1'-yl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(C)C(F)=C4)=N2)=C(OC)C=C1N1CCC2(CCN(CCC3=C4C(=CC=C3)N(C3CCC(=O)NC3=O)C(=O)C43CC3)CC2)CC1	C51H58BrFN9O5P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-GBYD9O	SCHEMBL31143281	3-[6-[4-[3-[4-[[5-bromo-4-[(5-dimethylphosphoryl-3-fluoro-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]piperidin-1-yl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(C)C(F)=C4)=N2)=C(OC)C=C1N1CCC2(CC1)CCN(C1CCN(C3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4)CC1)CC2	C52H61BrFN10O5P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-HHX96Y	WO2023138607A1_88	3-[6-[3-[3-[4-[[5-bromo-4-[(5-dimethylphosphoryl-3-fluoro-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]propyl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(C)C(F)=C4)=N2)=C(OC)C=C1N1CCC2(CCN(CCCC3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4)CC2)CC1	C50H58BrFN9O5P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-0NWHJ2	WO2023138607A1_89	3-[4-[3-[[3-[4-[[5-Bromo-4-[(5-dimethylphosphoryl-3-fluoro-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]methyl]azetidin-1-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(C)C(F)=C4)=N2)=C(OC)C=C1N1CCC2(CCN(CC3CN(C4=C5C(=CC=C4)N(C4CCC(=O)NC4=O)C(=O)N5C)C3)CC2)CC1	C51H60BrFN11O5P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-NY9P64	SCHEMBL31143497	(3R)-3-[4-[(3S)-3-[4-[1-[4-[[5-bromo-4-[(5-dimethylphosphoryl-2-ethylquinazolin-6-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]piperidin-4-yl]piperazin-1-yl]pyrrolidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(CC)N=C4)=N2)=C(OC)C=C1N1CCC(N2CCN([C@H]3CCN(C4=CC(F)=C([C@H]5CCC(=O)NC5=O)C(F)=C4)C3)CC2)CC1	C49H59BrF2N11O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-IRVBN2	SCHEMBL31143312	3-[6-[2-[3-[4-[[5-bromo-4-[(5-dimethylphosphoryl-3-fluoro-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]ethyl-methylamino]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(C)C(F)=C4)=N2)=C(OC)C=C1N1CCC2(CCN(CCN(C)C3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4)CC2)CC1	C50H59BrFN10O5P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-3MQF3U	SCHEMBL31143320	5-[4-[3-[4-[[5-Bromo-4-[(5-dimethylphosphoryl-3-fluoro-2-methylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-2-ethyl-5-methoxyphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]piperidin-1-yl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CCC1=CC(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C4=C(C=C3)N=C(C)C(F)=C4)=N2)=C(OC)C=C1N1CCC2(CC1)CCN(C1CCN(C3=CC=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)CC1)CC2	C52H59BrFN10O6P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-LFXX0V	WO2023138607A1_93	(3R)-3-[4-[3-[[3-[4-[[5-bromo-4-[(5-dimethylphosphoryl-2-ethylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]methyl]azetidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=NC2=C(C=C1)C(P(C)(C)=O)=C(NC1=NC(NC3=C(OC)C=C(N4CCC5(CCN(CC6CN(C7=CC(F)=C([C@H]8CCC(=O)NC8=O)C(F)=C7)C6)CC5)CC4)C(C)=C3)=NC=C1Br)C=C2	C49H57BrF2N9O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-UVATZ3	WO2023138607A1_94	3-[4-[4-[3-[4-[[5-Bromo-4-[(5-dimethylphosphoryl-2-ethylquinolin-6-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]piperidin-1-yl]-7-fluoro-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	CCC1=NC2=C(C=C1)C(P(C)(C)=O)=C(NC1=NC(NC3=C(OC)C=C(N4CCC5(CC4)CCN(C4CCN(C6=C7C(=C(F)C=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC4)CC5)C(C)=C3)=NC=C1Br)C=C2	C52H62BrFN11O5P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-TJZX49	WO2023138607A1_95	3-[4-[4-[3-[4-[[5-Bromo-4-[(5-dimethylphosphoryl-2-ethylquinazolin-6-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]piperidin-1-yl]-7-fluoro-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	CCC1=NC2=C(C=N1)C(P(C)(C)=O)=C(NC1=NC(NC3=C(OC)C=C(N4CCC5(CC4)CCN(C4CCN(C6=C7C(=C(F)C=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC4)CC5)C(C)=C3)=NC=C1Br)C=C2	C51H61BrFN12O5P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-Z21P98	WO2023138607A1_97	3-[4-[4-[3-[4-[[5-Bromo-4-[(5-dimethylphosphoryl-2-ethylquinazolin-6-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]piperidin-1-yl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione	CCC1=NC2=C(C=N1)C(P(C)(C)=O)=C(NC1=NC(NC3=C(OC)C=C(N4CCC5(CC4)CCN(C4CCN(C6=C7C(=CC=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC4)CC5)C(C)=C3)=NC=C1Br)C=C2	C51H62BrN12O5P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-G7R7EU	WO2023138607A1_98	.	CCC1=NC2=C(C=C1)C(P(C)(C)=O)=C(NC1=NC(NC3=C(OC)CC(N4CCC5(CCN(CC6CCN(C7=CC(F)=C([C@H]8CCC(=O)NC8=O)C(F)=C7)CC6)CC5)CC4)C(C)=C3)=NC=C1Br)C=C2	C51H63BrF2N9O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-HNPHUI	WO2023138607A1_99	(3R)-3-[4-[4-[[3-[4-[[5-bromo-4-[(5-dimethylphosphoryl-2-ethylquinazolin-6-yl)amino]pyrimidin-2-yl]amino]-5-methoxy-2-methylphenyl]-3,9-diazaspiro[5.5]undecan-9-yl]methyl]piperidin-1-yl]-2,6-difluorophenyl]piperidine-2,6-dione	CCC1=NC2=C(C=N1)C(P(C)(C)=O)=C(NC1=NC(NC3=C(OC)C=C(N4CCC5(CCN(CC6CCN(C7=CC(F)=C([C@H]8CCC(=O)NC8=O)C(F)=C7)CC6)CC5)CC4)C(C)=C3)=NC=C1Br)C=C2	C50H60BrF2N10O4P	EGFR	P00533	CRBN	WO-2023138607-A1
TPD-5ID0OS	WO2023143249A1_1	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(Cl)=CN=C2OCCNC(=O)CCCCCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)C=NC2=CC(Cl)=NN21	C47H59Cl2N11O8S	MALT1	Q9UDY8	VHL	WO-2023143249-A1
TPD-K7IQH0	WO2023143249A1_10	(2S,4R)-1-[(2S)-2-[7-[2-[3-[[2-chloro-7-[(1S)-1-methoxyethyl]pyrazolo[1,5-a]pyrimidin-6-yl]carbamoylamino]-6-(triazol-2-yl)pyridin-2-yl]oxyethylamino]heptanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide	CO[C@@H](C)C1=C(NC(=O)NC2=CC=C(N3N=CC=N3)N=C2OCCNCCCCCCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)C=NC2=CC(Cl)=NN21	C48H61ClN14O7S	MALT1	Q9UDY8	VHL	WO-2023143249-A1
TPD-6PV3CM	SCHEMBL25336944	(2R,4S)-1-[(2S)-2-[7-[2-[5-chloro-3-[[2-chloro-7-[(1S)-1-methoxyethyl]pyrazolo[1,5-a]pyrimidin-6-yl]carbamoylamino]pyridin-2-yl]oxyethylamino]heptanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; SCHEMBL30606748	CO[C@@H](C)C1=C(NC(=O)NC2=CC(Cl)=CN=C2OCCNCCCCCCC(=O)N[C@H](C(=O)N2C[C@@H](O)C[C@@H]2C(=O)NCC2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)C=NC2=CC(Cl)=NN21	C46H59Cl2N11O7S	MALT1	Q9UDY8	VHL	WO-2023143249-A1
TPD-434K5D	WO2023143249A1_12	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCNCCOC3=NC=C(Cl)C=C3NC(=O)NC3=C(C(C)O)N4N=C(Cl)C=C4NC3)C(C)(C)C)C=C2)SC=N1	C43H55Cl2N11O7S	MALT1	Q9UDY8	VHL	WO-2023143249-A1
TPD-JT50OL	WO2023143249A1_13	.	COC(C)C1=C(NC(=O)NC2=CC(Cl)=CN=C2OCCNCCCCCC(=O)N[C@H](C(=O)N2C[C@H](O)CC2C(=O)NCC2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)C=NC2=CC(Cl)=NN21	C45H57Cl2N11O7S	MALT1	Q9UDY8	VHL	WO-2023143249-A1
TPD-2XXZ6L	WO2023143249A1_14	.	COC(C)C1=C(NC(=O)NC2=CC(Cl)=CN=C2OCCNCCCCCCC(=O)N[C@H](C(=O)N2C[C@H](O)CC2C(=O)NCC2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)CNC2=CC(Cl)=NN21	C46H61Cl2N11O7S	MALT1	Q9UDY8	VHL	WO-2023143249-A1
TPD-Y4G5S4	WO2023143249A1_15	.	COC(C)C1=C(NC(=O)NC2=CC(Cl)=CN=C2OCCNCCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)C=NC2=CC(Cl)=NN21	C42H51Cl2N11O7S	MALT1	Q9UDY8	VHL	WO-2023143249-A1
TPD-0XI1ZL	WO2023143249A1_16	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3CC4(CC(C(=O)NCCOC5=NC=C(Cl)C=C5NC(=O)NC5=C([C@H](C)O)N6N=C(Cl)C=C6N=C5)C4)C3)C(C)(C)C)C=C2)SC=N1	C47H55Cl2N11O8S	MALT1	Q9UDY8	VHL	WO-2023143249-A1
TPD-BWKUKX	WO2023143249A1_17	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(Cl)=CN=C2OCCNC(=O)CCOCCOCCNC2=CC=CC3=C2N(C)C(=O)N3C2CCC(=O)NC2=O)C=NC2=CC(Cl)=NN21	C37H43Cl2N11O9	MALT1	Q9UDY8	VHL	WO-2023143249-A1
TPD-H9PH87	WO2023143249A1_18	.	CO[C@@H](C)C1=C(NC(=O)NC2=C(OCCNC(=O)CCN3CCC(CNC4=CC=CC5=C4N(C)C(=O)N5C4CCC(=O)NC4=O)CC3)N=CC(Cl)=C2)C=NC2=CC(Cl)=NN21	C39H46Cl2N12O7	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-W8WT0M	SCHEMBL25337220	1-[5-chloro-2-[2-[4-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]butylamino]ethoxy]pyridin-3-yl]-3-[2-chloro-7-[(1S)-1-methoxyethyl]pyrazolo[1,5-a]pyrimidin-6-yl]urea; SCHEMBL30606705	CO[C@@H](C)C1=C(NC(=O)NC2=CC(Cl)=CN=C2OCCNCCCCNC2=CC=CC3=C2C(=O)N(C2CCC(=O)NC2=O)C3=O)C=NC2=CC(Cl)=NN21	C34H36Cl2N10O7	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-FE5540	WO2023143249A1_2	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(C(F)(F)F)=CN=C2OCCNC(=O)CCCCCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)C=NC2=CC(Cl)=NN21	C48H59ClF3N11O8S	MALT1	Q9UDY8	VHL	WO-2023143249-A1
TPD-7ZBFBA	WO2023143249A1_20	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(Cl)=CN=C2OCCNCCCCCCCNC2=CC=CC3=C2C(=O)N(C2CCC(=O)NC2=O)C3=O)CNC2=CC(Cl)=NN21	C37H44Cl2N10O7	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-T0NS4O	SCHEMBL25337561	1-[5-chloro-2-[2-[5-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]pentylamino]ethoxy]pyridin-3-yl]-3-[2-chloro-7-[(1S)-1-methoxyethyl]pyrazolo[1,5-a]pyrimidin-6-yl]urea; SCHEMBL30606681	CO[C@@H](C)C1=C(NC(=O)NC2=CC(Cl)=CN=C2OCCNCCCCCNC2=CC=CC3=C2C(=O)N(C2CCC(=O)NC2=O)C3=O)C=NC2=CC(Cl)=NN21	C35H38Cl2N10O7	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-D5TIXD	WO2023143249A1_22	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(Cl)=CN=C2OCCNC(=O)CCCCCCNC2=CC=CC3=C2C(=O)N(C2CCC(=O)NC2=O)C3=O)C=NC2=CC(Cl)=NN21	C37H40Cl2N10O8	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-R5VFEV	WO2023143249A1_23	.	COC(C)C1=C(NC(=O)NC2=CC(Cl)=C(N3N=CC=N3)N=C2OCCNC(=O)CCCCCCCCNC2=CC=CC3=C2C(=O)N(C2CCC(=O)NC2=O)C3=O)C=NC2=CC(Cl)=NN21	C41H45Cl2N13O8	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-3DP3FQ	SCHEMBL25337509	N-[2-[5-chloro-3-[[2-chloro-7-(1-methoxyethyl)pyrazolo[1,5-a]pyrimidin-6-yl]carbamoylamino]-6-(triazol-2-yl)pyridin-2-yl]oxyethyl]-3-[4-[3-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]propoxy]piperidin-1-yl]propanamide; SCHEMBL30606739	COC(C)C1=C(NC(=O)NC2=CC(Cl)=C(N3N=CC=N3)N=C2OCCNC(=O)CCN2CCC(OCCCNC3=CC=CC4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)C=NC2=CC(Cl)=NN21	C43H48Cl2N14O9	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-1VKH8F	SCHEMBL25337111	N-[2-[5-chloro-3-[[2-chloro-7-(1-methoxyethyl)pyrazolo[1,5-a]pyrimidin-6-yl]carbamoylamino]-6-(triazol-2-yl)pyridin-2-yl]oxyethyl]-3-[3-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]propyl-methylamino]propanamide; SCHEMBL30606720	COC(C)C1=C(NC(=O)NC2=CC(Cl)=C(N3N=CC=N3)N=C2OCCNC(=O)CCN(C)CCCOCCNC2=CC=CC3=C2C(=O)N(C2CCC(=O)NC2=O)C3=O)C=NC2=CC(Cl)=NN21	C41H46Cl2N14O9	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-PE0ZRX	WO2023143249A1_26	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(Cl)=CN=C2OCCNCCCCCCC#CC2=CC=CC3=C2CN(C2CCC(=O)NC2=O)C3=O)C=NC2=CC(Cl)=NN21	C38H41Cl2N9O6	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-ULGMZ7	WO2023143249A1_27	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(Cl)=CN=C2OCCNCCCC#CC2=C3CN(C4CCC(=O)NC4=O)C(=O)C3=CC=C2)C=NC2=CC(Cl)=NN21	C35H35Cl2N9O6	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-HGJJV3	SCHEMBL25336987	1-[5-chloro-2-[2-[[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]cyclohexyl]amino]ethoxy]pyridin-3-yl]-3-[2-chloro-7-[(1S)-1-methoxyethyl]pyrazolo[1,5-a]pyrimidin-6-yl]urea; SCHEMBL30606701	CO[C@@H](C)C1=C(NC(=O)NC2=CC(Cl)=CN=C2OCCNC2CCC(CN3CCN(C4=C(F)C=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)C=NC2=CC(Cl)=NN21	C41H46Cl2FN11O7	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-BB7R7H	WO2023143249A1_29	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(Cl)=CN=C2OCCNC2CCN(C3CN(C4=CC5=C(C=C4F)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)CC2)C=NC2=CC(Cl)=NN21	C38H40Cl2FN11O7	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-Y2A5X7	WO2023143249A1_3	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(Cl)=CN=C2OCC(=O)NCCCCCCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)C=NC2=CC(Cl)NN21	C47H61Cl2N11O8S	MALT1	Q9UDY8	VHL	WO-2023143249-A1
TPD-TRQHBL	WO2023143249A1_30	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(Cl)=CN=C2OCCNC(=O)C2CCN(C3CN(C4=CC5=C(C=C4F)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)CC2)C=NC2=CC(Cl)=NN21	C39H40Cl2FN11O8	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-48SQY0	WO2023143249A1_31	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(C(F)(F)F)=CN=C2OCCNC(=O)C2CCN(C3CN(C4=CC5=C(C=C4F)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)CC2)C=NC2=CC(Cl)=NN21	C40H40ClF4N11O8	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-TME2JT	WO2023143249A1_32	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(Cl)=CN=C2OCCNC(=O)C2CCC(N3CCN(C4=C(F)C=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)C=NC2=CC(Cl)=NN21	C41H44Cl2FN11O8	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-V5UZKL	WO2023143249A1_33	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(C(F)(F)F)=CN=C2OCCNC(=O)C2CCC(N3CCN(C4=C(F)C=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)C=NC2=CC(Cl)=NN21	C42H44ClF4N11O8	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-XGJT4X	WO2023143249A1_34	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(C(F)(F)F)=CN=C2OCCN(C)C(=O)C2CCN(C3CN(C4=CC5=C(C=C4F)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)CC2)C=NC2=CC(Cl)=NN21	C41H42ClF4N11O8	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-5CT9IK	WO2023143249A1_35	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(Cl)=CN=C2OCCNCC#CC2=CC=CC3=C2N(C)C(=O)N3C2CCC(=O)NC2=O)C=NC2=CC(Cl)=NN21	C33H32Cl2N10O6	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-H6PSVZ	WO2023143249A1_36	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(C(F)(F)F)=CN=C2OCCNC(=O)CC2CCN(C3=CC4=C(C=C3F)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)C=NC2=CC(Cl)=NN21	C38H37ClF4N10O8	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-V5UX00	WO2023143249A1_37	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(C(F)(F)F)=CN=C2OCCNCCC2CCN(C3=CC4=C(C=C3F)C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)C=NC2=CC(Cl)=NN21	C38H39ClF4N10O7	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-P3O0QY	WO2023143249A1_38	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(Cl)=CN=C2OCCNCCN2CCC3(CC2)CC(NC2=C(F)C=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C2)C3)C=NC2=CC(Cl)=NN21	C40H44Cl2FN11O7	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-WRV2VN	WO2023143249A1_39	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(C(F)(F)F)=CN=C2OCCNC(=O)CN2CCC3(CC2)CC(NC2=C(F)C=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C2)C3)C=NC2=CC(Cl)=NN21	C41H42ClF4N11O8	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-MJMO02	WO2023143249A1_4	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(Cl)=CN=C2OCCNC(=O)CCCCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)C=NC2=CC(Cl)=NN21	C46H57Cl2N11O8S	MALT1	Q9UDY8	VHL	WO-2023143249-A1
TPD-5IG0R8	WO2023143249A1_40	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(Cl)=CN=C2OCCCN2CCC3(CC2)CC(NC2=C(F)C=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C2)C3)C=NC2=CC(Cl)=NN21	C39H41Cl2FN10O7	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-G8UTHL	WO2023143249A1_41	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(C(F)(F)F)=CN=C2OCCN2CCC(CN3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)C=NC2=CC(Cl)=NN21	C41H45ClF3N11O7	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-K4IN8A	SCHEMBL25338079	1-[5-chloro-2-[2-[[4-[4-[2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindol-5-yl]piperazin-1-yl]cyclohexyl]amino]ethoxy]pyridin-3-yl]-3-[2-chloro-7-[(1S)-1-methoxyethyl]pyrazolo[1,5-a]pyrimidin-6-yl]urea; SCHEMBL30606723	CO[C@@H](C)C1=C(NC(=O)NC2=CC(Cl)=CN=C2OCCNC2CCC(N3CCN(C4=C(F)C=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)C=NC2=CC(Cl)=NN21	C40H44Cl2FN11O7	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-HT5IPB	WO2023143249A1_43	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(C(F)(F)F)=CNC2OCCNC2CCC(CN3CCN(C4=C(F)C=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)C=NC2=CC(Cl)=NN21	C42H48ClF4N11O7	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-64A5MR	WO2023143249A1_44	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(Cl)=CN=C2OCCNC2CCN(CC3CCN(C4=CC5=C(C=C4F)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)C=NC2=CC(Cl)=NN21	C41H46Cl2FN11O7	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-9CVNKK	WO2023143249A1_45	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(Cl)=CN=C2OCCNC(=O)CCN2CCN(C3=CC=CC4=C3N(C)C(=O)N4C3CCC(=O)NC3=O)CC2)C=NC2=CC(Cl)=NN21	C37H42Cl2N12O7	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-DPQAIJ	WO2023143249A1_46	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(Cl)=CN=C2OCCNC2CCC(C(=O)N3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)CC5=C4)CC3)CC2)C=NC2=CC(Cl)=NN21	C41H47Cl2N11O7	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-GD6YZW	WO2023143249A1_47	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(C(F)(F)F)=CN=C2OCCNC2CCC(C3=CC=C(NC4CCC(=O)NC4=O)C=C3)CC2)C=NC2=CC(Cl)=NN21	C35H39ClF3N9O5	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-UJAUSI	WO2023143249A1_48	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(C(F)(F)F)=CN=C2OCCNC(=O)C2CCC(CNC3=CC=C(C4CCC(=O)NC4=O)C=C3)CC2)C=NC2=CC(Cl)=NN21	C37H41ClF3N9O6	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-10CYVM	WO2023143249A1_49	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(C(F)(F)F)=CN=C2OCCN2CCC(CN3CCN(C4=CC=CC5=C4N(C)C(=O)N5C4CCC(=O)NC4=O)CC3)CC2)C=NC2=CC(Cl)=NN21	C41H48ClF3N12O6	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-T4RO0K	SCHEMBL25336621	(2S,4R)-1-[(2S)-2-[7-[2-[5-chloro-3-[[2-chloro-7-[(1S)-1-methoxyethyl]pyrazolo[1,5-a]pyrimidin-6-yl]carbamoylamino]pyridin-2-yl]oxyethylamino]heptanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL30606730	CO[C@@H](C)C1=C(NC(=O)NC2=CC(Cl)=CN=C2OCCNCCCCCCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)C=NC2=CC(Cl)=NN21	C47H61Cl2N11O7S	MALT1	Q9UDY8	VHL	WO-2023143249-A1
TPD-X93GAH	WO2023143249A1_50	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(C(F)(F)F)=CN=C2OCCN2CCC3(CC2)CC(NC2=CC=CC4=C2N(C)C(=O)N4C2CCC(=O)NC2=O)C3)CNC2=CC(Cl)=NN21	C39H45ClF3N11O6	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-RR2EFF	WO2023143249A1_51	.	CO[C@@H](C)C1=C(CC(=O)NC2=CC(C(F)(F)F)=CN=C2OCCN2CCC(CN3CCN(C4=C(F)C=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)C=NC2=CC(Cl)=NN21	C40H47ClF4N10O5	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-DOX86Y	WO2023143249A1_52	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(C(F)(F)F)=CN=C2OCCC2CCN(CC3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)C=NC2=CC(Cl)=NN21	C42H46ClF3N10O7	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-MKNRZA	WO2023143249A1_53	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(C(F)(F)F)=CN=C2OCCN2CCC(CN3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)C[C@H]3C)CC2)C=NC2=CC(Cl)=NN21	C42H47ClF3N11O7	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-H9QDGU	WO2023143249A1_54	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(C(F)(F)F)=CN=C2OCCNCCC2CCN(C3=CC=CC4=C3N(C)C(=O)N4C3CCC(=O)NC3=O)CC2)C=NC2=CC(Cl)=NN21	C38H43ClF3N11O6	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-JZ6RCW	WO2023143249A1_55	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(C(F)(F)F)=CN=C2OCCN2CCC(N3CCN(CC4=CC=C5C(=C4)N(C)C(=O)N5C4CCC(=O)NC4=O)CC3)CC2)C=NC2=CC(Cl)=NN21	C41H48ClF3N12O6	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-W3QUTA	WO2023143249A1_56	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(C(F)(F)F)=CN=C2OCCN2CCC(CN3CC4(C3)CN(C3=CC=CC5=C3N(C)C(=O)N5C3CCC(=O)NC3=O)C4)CC2)C=NC2=CC(Cl)=NN21	C42H48ClF3N12O6	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-667A2P	WO2023143249A1_57	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(C(F)(F)F)=CN=C2OCCN2CCN(CC3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)C=NC2=CC(Cl)=NN21	C41H45ClF3N11O7	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-J4HGS3	WO2023143249A1_58	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(C(F)(F)F)=CN=C2OCCN2CCC(CN3CCC(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)C=NC2=CC(Cl)=NN21	C42H46ClF3N10O7	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-RHBY63	WO2023143249A1_59	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(C(F)(F)F)=CN=C2OCCN2CCC(CN3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)CC5=C4)CC3)CC2)C=NC2=CC(Cl)=NN21	C41H47ClF3N11O6	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-YCJUI0	WO2023143249A1_6	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(Cl)=C(N3N=CC=N3)N=C2OCCNCCCCCCC(=O)N[C@H](C(=O)N2C[C@H](O)CC2C(=O)N[C@@H](C)C2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)C=NC2=CC(Cl)=NN21	C49H62Cl2N14O7S	MALT1	Q9UDY8	VHL	WO-2023143249-A1
TPD-NOQIQP	WO2023143249A1_60	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(C(F)(F)F)=CN=C2OCCN2CCC(NC3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)C=NC2=CC(Cl)=NN21	C41H45ClF3N11O7	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-272QXB	WO2023143249A1_61	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(C(F)(F)F)=CN=C2OCCN2CCC(CN3CCN(C4=CC=C5CN(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)C=NC2=CC(Cl)=NN21	C41H47ClF3N11O6	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-8Z4HPC	WO2023143249A1_62	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(C(F)(F)F)=CN=C2OCCNCCN2CCC3(CC2)CN(C2=CC=CC4=C2N(C)C(=O)N4C2CCC(=O)NC2=O)C3)C=NC2=CC(Cl)=NN21	C40H46ClF3N12O6	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-PZE3SH	WO2023143249A1_63	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(C(F)(F)F)=CN=C2OC2CC3(C2)CN(CCC2CCN(C4=C(F)C=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC2)C3)CNC2=CC(Cl)=NN21	C42H45ClF4N10O7	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-2045I7	WO2023143249A1_64	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(C(F)(F)F)=CN=C2OCCN2CCC(CN3CCC4(CC3)CCN(C3=CC=CC5=C3N(C)C(=O)N5C3CCC(=O)NC3=O)CC4)CC2)C=NC2=CC(Cl)=NN21	C46H56ClF3N12O6	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-H4CVAJ	WO2023143249A1_65	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(Cl)=CN=C2OCCN2CCC(CN3CCC4(CC3)CCN(C3=CC=CC5=C3N(C)C(=O)N5C3CCC(=O)NC3=O)CC4)CC2)C=NC2=CC(Cl)=NN21	C45H56Cl2N12O6	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-FTF9VB	WO2023143249A1_66	.	COC1=C(NC2CC3(CCN(CCOC4=NC=C(C(F)(F)F)C=C4NC(=O)NC4=C([C@H](C)OC)N5N=C(Cl)C=C5N=C4)CC3)C2)C2=C(C=C1)N(C1CCC(=O)NC1=O)C(=O)N2C	C40H45ClF3N11O7	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-N5WWJM	WO2023143249A1_67	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(C(F)(F)F)=CN=C2OCCN2CCC3(CC2)CC(NC2=C(F)C=CC4=C2N(C)C(=O)N4C2CCC(=O)NC2=O)C3)C=NC2=CC(Cl)=NN21	C39H42ClF4N11O6	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-A6C9YK	WO2023143249A1_68	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(C(F)(F)F)=CN=C2OCCN2CCC3(CC2)CC(NC2=CC=CC4=C2C(C)(C)C(=O)N4C2CCC(=O)NC2=O)C3)C=NC2=CC(Cl)=NN21	C41H46ClF3N10O6	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-WQJ0J5	WO2023143249A1_69	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(C(F)(F)F)=CN=C2OCCN2CC3(CC(CCNC4=CC=CC5=C4N(C)C(=O)N5C4CCC(=O)NC4=O)C3)C2)C=NC2=CC(Cl)=NN21	C39H43ClF3N11O6	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-GQWYPW	WO2023143249A1_7	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(Cl)=CN=C2OCCNCCCCCCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)C=NC2=CC(Cl)=NN21	C46H59Cl2N11O7S	MALT1	Q9UDY8	VHL	WO-2023143249-A1
TPD-E2NO3H	WO2023143249A1_70	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(C(F)(F)F)=CN=C2OCCN2CC3(CC(NC4=CC=CC5=C4N(C)C(=O)N5C4CCC(=O)NC4=O)C3)C2)C=NC2=CC(Cl)=NN21	C37H39ClF3N11O6	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-8Y1NPW	WO2023143249A1_71	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(C(F)(F)F)=CN=C2OCCC2CCN(CC3CCN(C4=CC=CC5=C4N(C)C(=O)N5C4CCC(=O)NC4=O)CC3)CC2)C=NC2=CC(Cl)=NN21	C42H49ClF3N11O6	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-JXG6KD	SCHEMBL25336261	1-[2-chloro-7-[(1S)-1-methoxyethyl]pyrazolo[1,5-a]pyrimidin-6-yl]-3-[2-[2-[1-[[1-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperidin-4-yl]methyl]piperidin-4-yl]oxyethoxy]-5-(trifluoromethyl)pyridin-3-yl]urea	CO[C@@H](C)C1=C(NC(=O)NC2=CC(C(F)(F)F)=CN=C2OCCOC2CCN(CC3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)C=NC2=CC(Cl)=NN21	C42H46ClF3N10O8	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-Z7642A	WO2023143249A1_73	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(C(F)(F)F)=CN=C2OCCN2CCC(CN3CCN(C4=CC(F)=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)C=NC2=CC(Cl)=NN21	C39H46ClF4N11O5	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-I7PE4Y	WO2023143249A1_74	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(C(F)(F)F)=CN=C2OCCN2CCC(CN3CCC(C4=CC=C(NC5CCC(=O)NC5=O)C=C4)CC3)CC2)C=NC2=CC(Cl)=NN21	C40H48ClF3N10O5	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-Z3X81G	WO2023143249A1_75	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(C(F)(F)F)=CN=C2OCCN2CCC(CN3CCN(C4=CC=C(NC5CCC(=O)NC5=O)C=N4)CC3)CC2)C=NC2=CC(Cl)=NN21	C38H46ClF3N12O5	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-D654QT	WO2023143249A1_76	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(C(F)(F)F)=CN=C2OCCN2CCC(CN3CCC(C4=CC=CC5=C4N(C)C(=O)N5C4CCC(=O)NC4=O)CC3)CC2)C=NC2=CC(Cl)=NN21	C42H49ClF3N11O6	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-M4RJRP	WO2023143249A1_77	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(C(F)(F)F)=CN=C2OCCN2CCC(N(C)C3CCN(C4=CC=CC5=C4N(C)C(=O)N5C4CCC(=O)NC4=O)CC3)CC2)C=NC2=CC(Cl)=NN21	C42H50ClF3N12O6	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-F90WFN	SCHEMBL25337845	1-[2-chloro-7-[(1S)-1-methoxyethyl]pyrazolo[1,5-a]pyrimidin-6-yl]-3-[2-[2-[4-[[4-[4-(2,6-dioxopiperidin-3-yl)-2-fluorophenyl]piperazin-1-yl]methyl]piperidin-1-yl]ethoxy]-5-(trifluoromethyl)pyridin-3-yl]urea	CO[C@@H](C)C1=C(NC(=O)NC2=CC(C(F)(F)F)=CN=C2OCCN2CCC(CN3CCN(C4=CC=C(C5CCC(=O)NC5=O)C=C4F)CC3)CC2)C=NC2=CC(Cl)=NN21	C39H45ClF4N10O5	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-GC223H	SCHEMBL25336577	11-chloro-N-[2-[2-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]piperazin-1-yl]methyl]piperidin-1-yl]ethoxy]-5-(trifluoromethyl)pyridin-3-yl]-3-methyl-3-(trifluoromethyl)-1,5,8,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),7,9,11-tetraene-5-carboxamide	CC1(C(F)(F)F)CN(C(=O)NC2=CC(C(F)(F)F)=CN=C2OCCN2CCC(CN3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)C2=C1N1N=C(Cl)C=C1N=C2	C42H42ClF6N11O6	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-DJ27TQ	WO2023143249A1_8	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(Cl)=CN=C2OCCNC(=O)CCCCCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)C=NC2=CC(Cl)=NN21	C46H57Cl2N11O8S	MALT1	Q9UDY8	VHL	WO-2023143249-A1
TPD-IG9CYA	WO2023143249A1_80	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(C(F)(F)F)=CN=C2OCCNC(=O)CCCCCC(=O)N[C@H](C(=O)N2C[C@H](O)CC2C(=O)N[C@@H](CO)C2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)C=NC2=CC(Cl)=NN21	C48H59ClF3N11O9S	MALT1	Q9UDY8	VHL	WO-2023143249-A1
TPD-8YUS1U	SCHEMBL25335215	(2S,4R)-N-[[2-[2-[1-[2-[3-[[2-chloro-7-[(1S)-1-methoxyethyl]pyrazolo[1,5-a]pyrimidin-6-yl]carbamoylamino]-5-(trifluoromethyl)pyridin-2-yl]oxyethyl]piperidin-4-yl]ethoxy]-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-1-[(2S)-2-[(1-fluorocyclopropanecarbonyl)amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide; SCHEMBL30606708	CO[C@@H](C)C1=C(NC(=O)NC2=CC(C(F)(F)F)=CN=C2OCCN2CCC(CCOC3=C(CNC(=O)[C@@H]4C[C@@H](O)CN4C(=O)[C@@H](NC(=O)C4(F)CC4)C(C)(C)C)C=CC(C4=C(C)N=CS4)=C3)CC2)C=NC2=CC(Cl)=NN21	C51H62ClF4N11O8S	MALT1	Q9UDY8	VHL	WO-2023143249-A1
TPD-V4OF6S	WO2023143249A1_82	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(C(F)(F)F)=CN=C2OCCN2CCC(COC3=C(CNC(=O)[C@@H]4C[C@@H](O)CN4C(=O)[C@@H](NC(=O)C4(F)CC4)C(C)(C)C)C=CC(C4=C(C)N=CS4)=C3)CC2)C=NC2=CC(Cl)=NN21	C50H60ClF4N11O8S	MALT1	Q9UDY8	VHL	WO-2023143249-A1
TPD-B8BL4N	WO2023143249A1_83	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(C(F)(F)F)=CN=C2OCCN2CCC(CNC(=O)C[C@H](NC(=O)C3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3(F)CC3)C(C)(C)C)C3=CC=C(C4=C(C)N=CS4)C=C3)CC2)C=NC2=CC(Cl)=NN21	C52H63ClF4N12O8S	MALT1	Q9UDY8	VHL	WO-2023143249-A1
TPD-0K7IF9	WO2023143249A1_84	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(C(F)(F)F)=CN=C2OCCN2CCN(C(=O)C[C@H](NC(=O)C3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3(F)CC3)C(C)(C)C)C3=CC=C(C4=C(C)N=CS4)C=C3)CC2)C=NC2=CC(Cl)=NN21	C50H59ClF4N12O8S	MALT1	Q9UDY8	VHL	WO-2023143249-A1
TPD-SWWJ2Z	WO2023143249A1_85	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(C(F)(F)F)=CN=C2OCCN2CCC3(CCC(NC4=CC=CC5=C4N(C)C(=O)N5C4CCC(=O)NC4=O)CC3)CC2)C=NC2=CC(Cl)=NN21	C41H47ClF3N11O6	MALT1	Q9UDY8	CRBN	WO-2023143249-A1
TPD-A5PBX1	WO2023143249A1_9	.	CO[C@@H](C)C1=C(NC(=O)NC2=CC(Cl)=CN=C2OCCNCCCCCCCC(=O)N[C@H](C(=O)N2C[C@H](O)CC2C(=O)NCC2=CC=C(C3=C(C)N=CS3)C=C2)C(C)(C)C)CNC2=CC(Cl)=NN21	C47H63Cl2N11O7S	MALT1	Q9UDY8	VHL	WO-2023143249-A1
TPD-3QBIFP	SCHEMBL30810427	2-(2,6-Dioxopiperidin-3-yl)-5-fluoro-6-[4-[[3-[4-[[4-[1-(2,2,2-trifluoroethyl)pyrazol-4-yl]-5-(trifluoromethyl)pyrimidin-2-yl]amino]piperidin-1-yl]sulfonylphenyl]methyl]piperazin-1-yl]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC(F)=C(N4CCN(CC5=CC=CC(S(=O)(=O)N6CCC(NC7=NC(C8=CN(CC(F)(F)F)N=C8)=C(C(F)(F)F)C=N7)CC6)=C5)CC4)C=C3C2=O)C(=O)N1	C39H37F7N10O6S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-PPZ2GE	WO2023249970A1_10	.	O=C1CCC(N2C(=O)C3=CC(F)=C(N4CCN(CC5=CC=CC(S(=O)(=O)N6CCC(NC7=NC(C8=CN(C9CCOCC9)N=C8)=C(C(F)(F)F)C=N7)CC6)=C5)CC4)C=C3C2=O)C(=O)N1	C42H44F4N10O7S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-JPW9J0	SCHEMBL30810301	3-[4-[1-[[3-[4-[[4-[1-(2,2,2-Trifluoroethyl)pyrazol-4-yl]-5-(trifluoromethyl)pyrimidin-2-yl]amino]piperidin-1-yl]sulfonylphenyl]methyl]piperidin-4-yl]anilino]piperidine-2,6-dione	O=C1CCC(NC2=CC=C(C3CCN(CC4=CC=CC(S(=O)(=O)N5CCC(NC6=NC(C7=CN(CC(F)(F)F)N=C7)=C(C(F)(F)F)C=N6)CC5)=C4)CC3)C=C2)C(=O)N1	C38H41F6N9O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-XZK0M1	WO2023249970A1_12	.	O=C1CCC(N2CC3=CC(N4CCC5(CCN(CC6=CC(S(=O)(=O)N7CCC(NC8=NC(C9=CN(CC(F)(F)F)N=C9)=C(C(F)(F)F)C=N8)CC7)=CC=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C44H48F6N10O5S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-91SVXU	WO2023249970A1_13	.	O=C1CCN(C2=CC=C(N3CCN(CC4=CC=CC(S(=O)(=O)N5CCC(NC6=NC(C7=CN(CC(F)(F)F)N=C7)=C(C(F)(F)F)C=N6)CC5)=C4)CC3)C(F)=C2)C(=O)N1	C36H37F7N10O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-C4C1GC	WO2023249970A1_14	3-[3-Fluoro-4-[4-[[3-[4-[[4-[1-(2,2,2-trifluoroethyl)pyrazol-4-yl]-5-(trifluoromethyl)pyrimidin-2-yl]amino]piperidin-1-yl]sulfonylphenyl]methyl]piperazin-1-yl]phenyl]piperidine-2,6-dione	O=C1CCC(C2=CC=C(N3CCN(CC4=CC=CC(S(=O)(=O)N5CCC(NC6=NC(C7=CN(CC(F)(F)F)N=C7)=C(C(F)(F)F)C=N6)CC5)=C4)CC3)C(F)=C2)C(=O)N1	C37H38F7N9O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-MCE3ON	WO2023249970A1_15	.	O=C1CCC(N2CC3=CC(N4CCN(CC5=CC=CC(S(=O)(=O)N6CCC(NC7=NC(C8=CN(CC(F)(F)F)N=C8)=C(C(F)(F)F)C=N7)CC6)=C5)CC4)=C(F)C=C3C2=O)C(=O)N1	C39H39F7N10O5S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-Z5VD1J	WO2023249970A1_16	.	O=C1CCN(C2=CC=C(N3CCN(CC4=CC=CC(S(=O)(=O)N5CCC(NC6=NC(C7=CN(CC(F)(F)F)N=C7)=C(C(F)(F)F)C=N6)CC5)=C4)CC3)C(C(F)(F)F)=C2)C(=O)N1	C37H37F9N10O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-THTQ98	WO2023249970A1_17	2-(2,6-Dioxopiperidin-3-yl)-5-fluoro-6-[4-[[3-[4-[[4-[1-(2,2,2-trifluoroethyl)pyrazol-4-yl]pyrimidin-2-yl]amino]piperidin-1-yl]sulfonylphenyl]methyl]piperazin-1-yl]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC(F)=C(N4CCN(CC5=CC=CC(S(=O)(=O)N6CCC(NC7=NC(C8=CN(CC(F)(F)F)N=C8)=CC=N7)CC6)=C5)CC4)C=C3C2=O)C(=O)N1	C38H38F4N10O6S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-746IYU	WO2023249970A1_18	.	O=C1CCC(C2=CC=C(N3CC4CCC(C3)N4CC3=CC=CC(S(=O)(=O)N4CCC(NC5=NC(C6=CN(CC(F)(F)F)N=C6)=C(C(F)(F)F)C=N5)CC4)=C3)C=C2)C(=O)N1	C39H41F6N9O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-F5FJI4	WO2023249970A1_19	.	O=C1CCC(C2=CC=C(N3CCN(CC4=CC=CC(S(=O)(=O)N5CC[C@H](NC6=NC(C7=CN(CC(F)(F)F)N=C7)=C(C(F)(F)F)C=N6)[C@H](F)C5)=C4)CC3)C=C2)C(=O)N1	C37H38F7N9O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-7Y0J7H	WO2023249970A1_2	.	O=C1CCC(C2=CC=C(N3CCN(CC4=CC=CC(S(=O)(=O)N5CCC(NC6=NC(C7=CN(CC(F)(F)F)N=C7)=C(C(F)(F)F)C=N6)CC5)=C4)CC3)C=C2)C(=O)N1	C37H39F6N9O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-J4K2T2	WO2023249970A1_20	.	CN1C(S(=O)(=O)N2CCC(NC3=NC(C4=CN(CC(F)(F)F)N=C4)=C(C(F)(F)F)C=N3)CC2)=CN=C1CN1CCN(C2=CC=C(C3CCC(=O)NC3=O)C=C2F)CC1	C35H38F7N11O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-3DC7X0	WO2023249970A1_21	1-[6-[1-[[3-[4-[[4-[1-(2,2-Difluoroethyl)pyrazol-4-yl]-5-(trifluoromethyl)pyrimidin-2-yl]amino]piperidin-1-yl]sulfonylphenyl]methyl]piperidin-4-yl]-1-methylindazol-3-yl]-1,3-diazinane-2,4-dione	CN1N=C(N2CCC(=O)NC2=O)C2=C1C=C(C1CCN(CC3=CC=CC(S(=O)(=O)N4CCC(NC5=NC(C6=CN(CC(F)F)N=C6)=C(C(F)(F)F)C=N5)CC4)=C3)CC1)C=C2	C39H42F5N11O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-L9NUXP	WO2023249970A1_23	.	O=C1CCC(C2=CC=C(N3CCN(CC4=CC=CC(S(=O)(=O)N5CCC(NC6=NC(C7=CN(CC(F)(F)F)N=C7)=C(C(F)(F)F)C=N6)CC5)=C4)CC3)C(C(F)(F)F)=C2)C(=O)N1	C38H38F9N9O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-B72HQO	WO2023249970A1_24	.	CC(C)(O)CN1C=C(C2=C(C(F)(F)F)C=NC(NC3CCN(S(=O)(=O)C4=CC(CN5CCN(C6=CC=C(N7CCC(=O)NC7=O)C=C6)CC5)=CC=C4)CC3)=N2)C=N1	C38H45F3N10O5S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-HDH7WO	WO2023249970A1_25	1-[4-[4-[[3-[4-[[4-[1-(2,2,2-Trifluoroethyl)pyrazol-4-yl]-5-(trifluoromethyl)pyrimidin-2-yl]amino]piperidin-1-yl]sulfonylphenyl]methyl]piperazin-1-yl]phenyl]-1,3-diazinane-2,4-dione	O=C1CCN(C2=CC=C(N3CCN(CC4=CC=CC(S(=O)(=O)N5CCC(NC6=NC(C7=CN(CC(F)(F)F)N=C7)=C(C(F)(F)F)C=N6)CC5)=C4)CC3)C=C2)C(=O)N1	C36H38F6N10O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-TN1DKY	WO2023249970A1_26	.	CN1C(S(=O)(=O)N2CCC(NC3=NC(C4=CN(CC(F)(F)F)N=C4)=C(C(F)(F)F)C=N3)CC2)=CN=C1CN1CCN(C2=CC=C(N3CCC(=O)NC3=O)C=C2)CC1	C34H38F6N12O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-OGN1QE	WO2023249970A1_27	.	O=C1CCC(N2CC3=CC(N4CCN(CC5CCN(C6=CC(S(=O)(=O)N7CCC(NC8=NC(C9=CN(CC(F)(F)F)N=C9)=C(C(F)(F)F)C=N8)CC7)=CC=C6)CC5)CC4)=CC=C3C2=O)C(=O)N1	C44H49F6N11O5S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-TXSNOO	WO2023249970A1_28	.	O=C1CCN(C2=CC=C(N3CCN(CC4=CC=CC(S(=O)(=O)N5CC[C@H](NC6=NC(C7=CN(CC(F)(F)F)N=C7)=C(C(F)(F)F)C=N6)[C@H](F)C5)=C4)CC3)C=C2)C(=O)N1	C36H37F7N10O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-1N6MRB	WO2023249970A1_29	.	O=C1CCC(C2=CC(F)=C(N3CCN(CC4=CC=CC(S(=O)(=O)N5CC[C@H](NC6=NC(C7=CN(CC(F)(F)F)N=C7)=C(C(F)(F)F)C=N6)[C@H](F)C5)=C4)CC3)C=C2)C(=O)N1	C37H37F8N9O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-PPJ0Y2	WO2023249970A1_3	3-[3-oxo-6-[1-[[3-[4-[[4-[1-(2,2,2-trifluoroethyl)pyrazol-4-yl]-5-(trifluoromethyl)pyrimidin-2-yl]amino]piperidin-1-yl]sulfonylphenyl]methyl]azetidin-3-yl]-1H-isoindol-2-yl]piperidine-2,6-dione	O=C1CCC(N2CC3=C(C=CC(C4CN(CC5=CC=CC(S(=O)(=O)N6CCC(NC7=NC(C8=CN(CC(F)(F)F)N=C8)=C(C(F)(F)F)C=N7)CC6)=C5)C4)=C3)C2=O)C(=O)N1	C38H37F6N9O5S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-RZZ81J	WO2023249970A1_30	.	CN1C(S(=O)(=O)N2CCC(NC3=NC(C4=CN(CC(F)(F)F)N=C4)=C(C(F)(F)F)C=N3)CC2)=CN=C1CN1CCN(C2=C(F)C=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=C2)CC1	C37H37F7N12O6S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-AATH10	WO2023249970A1_31	.	O=C1CCC(N2C(=O)C3=CC(F)=C(N4CC5(CN(CC6=CC=CC(S(=O)(=O)N7CCC(NC8=NC(C9=CN(CC(F)(F)F)N=C9)=C(C(F)(F)F)C=N8)CC7)=C6)C5)C4)C=C3C2=O)C(=O)N1	C40H37F7N10O6S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-BW3IFK	WO2023249970A1_32	2-(2,6-dioxopiperidin-3-yl)-5-fluoro-6-[4-[[3-[(3R,4S)-3-fluoro-4-[[4-[1-(2,2,2-trifluoroethyl)pyrazol-4-yl]-5-(trifluoromethyl)pyrimidin-2-yl]amino]piperidin-1-yl]sulfonylphenyl]methyl]piperazin-1-yl]isoindole-1,3-dione	O=C1CCC(N2C(=O)C3=CC(F)=C(N4CCN(CC5=CC=CC(S(=O)(=O)N6CC[C@H](NC7=NC(C8=CN(CC(F)(F)F)N=C8)=C(C(F)(F)F)C=N7)[C@H](F)C6)=C5)CC4)C=C3C2=O)C(=O)N1	C39H36F8N10O6S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-SLYIW8	WO2023249970A1_33	.	CN1C=C(C2=C(C(F)(F)F)C=NC(NC3CCN(S(=O)(=O)C4=CC(CN5CCC(C6=CC7=C(C=C6)C(N6CCC(=O)NC6=O)=NN7C)CC5)=CC=C4)CC3)=N2)C=N1	C38H42F3N11O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-ANAA8D	WO2023249970A1_34	1-[1-methyl-6-[1-[[3-[(3R,4S)-3-methyl-4-[[4-[1-(2,2,2-trifluoroethyl)pyrazol-4-yl]-5-(trifluoromethyl)pyrimidin-2-yl]amino]piperidin-1-yl]sulfonylphenyl]methyl]piperidin-4-yl]indazol-3-yl]-1,3-diazinane-2,4-dione	C[C@@H]1CN(S(=O)(=O)C2=CC(CN3CCC(C4=CC5=C(C=C4)C(N4CCC(=O)NC4=O)=NN5C)CC3)=CC=C2)CC[C@@H]1NC1=NC(C2=CN(CC(F)(F)F)N=C2)=C(C(F)(F)F)C=N1	C40H43F6N11O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-CQDOVV	WO2023249970A1_35	.	CC1=CN(C2=C(C(F)(F)F)C=NC(NC3CCN(S(=O)(=O)C4=CC(CN5CCC(C6=CC7=C(C=C6)C(N6CCC(=O)NC6=O)=NN7C)CC5)=CC=C4)CC3)=N2)C=N1	C38H42F3N11O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-7B9WLV	WO2023249970A1_36	3-[4-[1-[[3-[(3R,4S)-3-fluoro-4-[[4-[1-(2,2,2-trifluoroethyl)pyrazol-4-yl]-5-(trifluoromethyl)pyrimidin-2-yl]amino]piperidin-1-yl]sulfonylphenyl]methyl]piperidin-4-yl]anilino]piperidine-2,6-dione	O=C1CCC(NC2=CC=C(C3CCN(CC4=CC=CC(S(=O)(=O)N5CC[C@H](NC6=NC(C7=CN(CC(F)(F)F)N=C7)=C(C(F)(F)F)C=N6)[C@H](F)C5)=C4)CC3)C=C2)C(=O)N1	C38H40F7N9O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-0XQ6Y2	WO2023249970A1_37	.	CN1N=C(N2CCC(=O)NC2=O)C2=C1C=C(C1CCN(CC3=CC=CC(S(=O)(=O)N4CC[C@H](NC5=NC(C6=CN(CC(F)F)N=C6)=C(C(F)(F)F)C=N5)[C@H](F)C4)=C3)CC1)C=C2	C39H41F6N11O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-4HO1AE	WO2023249970A1_38	.	CN1N=C(N2CCC(=O)NC2=O)C2=C1C=C(C1CCN(CC3=C(C(F)(F)F)C=CC(S(=O)(=O)N4CC[C@H](NC5=NC(C6=CN(CC(F)(F)F)N=C6)=C(C(F)(F)F)C=N5)[C@H](F)C4)=C3)CC1)C=C2	C40H39F10N11O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-BRQZ9V	WO2023249970A1_39	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=CC(C#CCOC3CCN(CC4=CC=CC(S(=O)(=O)N5CCC(NC6=NC(C7=CN(CC(F)(F)F)N=C7)=C(C(F)(F)F)C=N6)CC5)=C4)CC3)=C21	C43H44F6N10O6S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-FQXZL3	WO2023249970A1_4	.	CN1N=C(N2CCC(=O)NC2=O)C2=C1C=C(C1CCN(CC3=CC=CC(S(=O)(=O)N4CCC(NC5=NC(C6=CN(CC(F)(F)F)N=C6)=C(C(F)(F)F)C=N5)CC4)=C3)CC1)C=C2	C39H41F6N11O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-451WCE	WO2023249970A1_40	.	CC(C1=CC=CC(S(=O)(=O)N2CC[C@H](NC3=NC(C4=CN(CC(F)(F)F)N=C4)=C(C(F)(F)F)C=N3)[C@H](C)C2)=C1)N1CCC(C2=CC3=C(C=C2)C(N2CCC(=O)NC2=O)=NN3C)CC1	C41H45F6N11O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-6TRV81	WO2023249970A1_41	.	O=C1CCN(C2=CN=C(N3CCN(CC4=CC=CC(S(=O)(=O)N5CCC(NC6=NC(C7=CN(CC(F)(F)F)N=C7)=C(C(F)(F)F)C=N6)CC5)=C4)CC3)C=C2)C(=O)N1	C35H37F6N11O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-8IC3GO	SCHEMBL30810308	1-[1-Methyl-6-[1-[[5-[4-[[4-[1-(2,2,2-trifluoroethyl)pyrazol-4-yl]-5-(trifluoromethyl)pyrimidin-2-yl]amino]piperidin-1-yl]sulfonyl-2-(trifluoromethyl)phenyl]methyl]piperidin-4-yl]indazol-3-yl]-1,3-diazinane-2,4-dione	CN1N=C(N2CCC(=O)NC2=O)C2=C1C=C(C1CCN(CC3=C(C(F)(F)F)C=CC(S(=O)(=O)N4CCC(NC5=NC(C6=CN(CC(F)(F)F)N=C6)=C(C(F)(F)F)C=N5)CC4)=C3)CC1)C=C2	C40H40F9N11O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-VV0QTL	WO2023249970A1_43	.	CN1N=C(N2CCC(=O)NC2=O)C2=C1C=C(C1CCN(CC3=CC=CC(S(=O)(=O)N4CCC(NC5=NC(C6=CN(CC(F)(F)F)N=C6)=C(C(F)(F)F)C=N5)CC4)=C3)CC1(F)F)C=C2	C39H39F8N11O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-M1J0UD	WO2023249970A1_44	.	CN1N=C(N2CCC(=O)NC2=O)C2=CC(F)=C(C3CCN(CC4=CC=CC(S(=O)(=O)N5CCC(NC6=NC(C7=CN(CC(F)(F)F)N=C7)=C(C(F)(F)F)C=N6)CC5)=C4)CC3)C=C21	C39H40F7N11O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-PDE50Q	WO2023249970A1_45	.	O=C1CCC(N2CC3=C(C=CC(N4CCC(CN5CCN(C6=CC=CC(S(=O)(=O)N7CCC(NC8=NC(C9=CN(CCF)N=C9)=C(C(F)(F)F)C=N8)CC7)=C6)CC5)CC4)=C3)C2=O)C(=O)N1	C44H51F4N11O5S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-7KX98V	WO2023249970A1_46	.	O=C1CCN(C2CCN(CC3=CC=CC(S(=O)(=O)N4CCC(NC5=NC(C6=CN(CC(F)(F)F)C=C6)=C(C(F)(F)F)C=N5)CC4)=C3)CC2)C(=O)N1	C32H36F6N8O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-JTRRJ6	SCHEMBL30810341	1-[1-Methyl-6-[1-[2-[3-[4-[[4-[1-(2,2,2-trifluoroethyl)pyrazol-4-yl]-5-(trifluoromethyl)pyrimidin-2-yl]amino]piperidin-1-yl]sulfonylphenyl]ethyl]piperidin-4-yl]indazol-3-yl]-1,3-diazinane-2,4-dione	CN1N=C(N2CCC(=O)NC2=O)C2=C1C=C(C1CCN(CCC3=CC=CC(S(=O)(=O)N4CCC(NC5=NC(C6=CN(CC(F)(F)F)N=C6)=C(C(F)(F)F)C=N5)CC4)=C3)CC1)C=C2	C40H43F6N11O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-CQJ8NT	WO2023249970A1_48	.	CN1N=C(N2CCC(=O)NC2=O)C2=C1C=C(C1CCN(CC3=CC=CC(S[C@H]4CC[C@H](NC5=NC(C6=CN(CC(F)(F)F)NC6)=C(C(F)(F)F)C=N5)CC4)=C3)CC1)C=C2	C40H44F6N10O2S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-KGISKY	WO2023249970A1_49	.	O=C1CCN(C2=C(F)C=C(N3CCN(CC4=CC=CC(S(=O)(=O)N5CCC(NC6=NC(C7=CN(CC(F)(F)F)N=C7)=C(C(F)(F)F)C=N6)CC5)=C4)CC3)C=C2)C(=O)N1	C36H37F7N10O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-E0EKFJ	WO2023249970A1_5	.	CN1C=C(C2=C(C(F)(F)F)C=NC(NC3CCN(S(=O)(=O)C4=CC(CN5CCN(C6=C(F)C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)=CC=C4)CC3)=N2)C=N1	C38H38F4N10O6S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-8VHIH3	SCHEMBL30810399	1-[1-Methyl-6-[1-[[1-[3-[4-[[4-[1-(2,2,2-trifluoroethyl)pyrazol-4-yl]-5-(trifluoromethyl)pyrimidin-2-yl]amino]piperidin-1-yl]sulfonylphenyl]piperidin-4-yl]methyl]piperidin-4-yl]indazol-3-yl]-1,3-diazinane-2,4-dione	CN1N=C(N2CCC(=O)NC2=O)C2=C1C=C(C1CCN(CC3CCN(C4=CC=CC(S(=O)(=O)N5CCC(NC6=NC(C7=CN(CC(F)(F)F)N=C7)=C(C(F)(F)F)C=N6)CC5)=C4)CC3)CC1)C=C2	C44H50F6N12O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-0DIFM4	orb2665085	1-[1-Methyl-6-[1-[[1-[4-[[4-[1-(2,2,2-trifluoroethyl)pyrazol-4-yl]-5-(trifluoromethyl)pyrimidin-2-yl]amino]piperidin-1-yl]sulfonylpiperidin-4-yl]methyl]piperidin-4-yl]indazol-3-yl]-1,3-diazinane-2,4-dione; 3024971-78-3	CN1N=C(N2CCC(=O)NC2=O)C2=C1C=C(C1CCN(CC3CCN(S(=O)(=O)N4CCC(NC5=NC(C6=CN(CC(F)(F)F)N=C6)=C(C(F)(F)F)C=N5)CC4)CC3)CC1)C=C2	C38H46F6N12O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-1DZOI6	SCHEMBL30810492	1-[6-[1-[[3-[(3R,4S)-3-fluoro-4-[[4-[1-(2,2,2-trifluoroethyl)pyrazol-4-yl]-5-(trifluoromethyl)pyrimidin-2-yl]amino]piperidin-1-yl]sulfonylphenyl]methyl]piperidin-4-yl]-1-methylindazol-3-yl]-1,3-diazinane-2,4-dione	CN1N=C(N2CCC(=O)NC2=O)C2=C1C=C(C1CCN(CC3=CC=CC(S(=O)(=O)N4CC[C@H](NC5=NC(C6=CN(CC(F)(F)F)N=C6)=C(C(F)(F)F)C=N5)[C@H](F)C4)=C3)CC1)C=C2	C39H40F7N11O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-UAFCIU	WO2023249970A1_53	.	O=C1CCC(NC2=CC=C(N3CCN(CC4=CC=CC(S(=O)(=O)N5CCC(NC6=NC(C7=CN(CC(F)(F)F)N=C7)=C(C(F)(F)F)C=N6)CC5)=C4)CC3)C=C2)C(=O)N1	C37H40F6N10O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-M3PC3U	WO2023249970A1_54	1-[1-(2,2,2-Trifluoroethyl)-6-[1-[[3-[4-[[4-[1-(2,2,2-trifluoroethyl)pyrazol-4-yl]-5-(trifluoromethyl)pyrimidin-2-yl]amino]piperidin-1-yl]sulfonylphenyl]methyl]piperidin-4-yl]indazol-3-yl]-1,3-diazinane-2,4-dione	O=C1CCN(C2=NN(CC(F)(F)F)C3=C2C=CC(C2CCN(CC4=CC=CC(S(=O)(=O)N5CCC(NC6=NC(C7=CN(CC(F)(F)F)N=C7)=C(C(F)(F)F)C=N6)CC5)=C4)CC2)=C3)C(=O)N1	C40H40F9N11O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-6HD8A6	WO2023249970A1_55	.	CN1N=C(N2CCC(=O)NC2=O)C2=C1C=C(C1CCN(CC3=C(C(F)(F)F)C=CC(S(=O)(=O)N4CCC(NC5=NC(C6=CN(CC(F)(F)F)N=C6)=C(C(F)(F)F)C=N5)CC4)=C3)CC1(F)F)C=C2	C40H38F11N11O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-YLCF3K	WO2023249970A1_56	.	CN1N=C(N2CCC(=O)NC2=O)C2=C1C=C(N1CCN(CC3=CC=CC(S(=O)(=O)N4CC[C@H](NC5=NC(C6=CN(CC(F)(F)F)N=C6)=C(C(F)(F)F)C=N5)[C@H](F)C4)=C3)CC1)C=C2	C38H39F7N12O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-2YM6PE	WO2023249970A1_57	.	CN1N=C(N2CCC(=O)NC2=O)C2=C1C=C(N1CCN(CC3=CC=CC(S(=O)(=O)N4CCC(NC5=NC(C6=CN(CC(F)(F)F)N=C6)=C(C(F)(F)F)C=N5)CC4)=C3)CC1)C=C2	C38H40F6N12O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-EE8Y3Z	SCHEMBL30810450	1-[1-Methyl-6-[1-[[1-[4-[[4-[1-(2,2,2-trifluoroethyl)pyrazol-4-yl]-5-(trifluoromethyl)pyrimidin-2-yl]amino]piperidin-1-yl]sulfonylpiperidin-3-yl]methyl]piperidin-4-yl]indazol-3-yl]-1,3-diazinane-2,4-dione	CN1N=C(N2CCC(=O)NC2=O)C2=C1C=C(C1CCN(CC3CCCN(S(=O)(=O)N4CCC(NC5=NC(C6=CN(CC(F)(F)F)N=C6)=C(C(F)(F)F)C=N5)CC4)C3)CC1)C=C2	C38H46F6N12O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-958GF7	SCHEMBL30810440	1-[6-[1-[[3-[4-[[4-[1-(2-Fluorophenyl)pyrazol-4-yl]-5-(trifluoromethyl)pyrimidin-2-yl]amino]piperidin-1-yl]sulfonylphenyl]methyl]piperidin-4-yl]-1-methylindazol-3-yl]-1,3-diazinane-2,4-dione; SCHEMBL30810443	CN1N=C(N2CCC(=O)NC2=O)C2=C1C=C(C1CCN(CC3=CC=CC(S(=O)(=O)N4CCC(NC5=NC(C6=CN(C7=C(F)C=CC=C7)N=C6)=C(C(F)(F)F)C=N5)CC4)=C3)CC1)C=C2	C43H43F4N11O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-7OS00B	WO2023249970A1_6	.	O=C1CCN(C2=NNC3=C2C=CC(C2CCN(CC4=CC=CC(S(=O)(=O)N5CC[C@H](NC6=CC(C7=CN(CC(F)(F)F)N=C7)=C(C(F)(F)F)C=N6)[C@H](F)C5)=C4)CC2)=C3)C(=O)N1	C39H39F7N10O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-K3Y815	WO2023249970A1_60	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3CCN(CC4=CC=CC(S(=O)(=O)N5CCC(NC6=NC(C7=CN(CC(F)(F)F)N=C7)=C(C(F)(F)F)C=N6)CC5)=C4)CC3)C(C)(C)C)C=C2)SC=N1	C51H61F6N11O6S2	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-BDH1QS	WO2023249970A1_61	.	CN1N=C(N2CCC(=O)NC2=O)C2=C1C=C(C1CCN(CC3=C(F)C=CC(S(=O)(=O)N4CCC(NC5=NC(C6=CN(CC(F)(F)F)N=C6)=C(C(F)(F)F)C=N5)CC4)=C3)CC1)C=C2	C39H40F7N11O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-A2LYTE	WO2023249970A1_62	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CC3CCN(CC4=CC=CC(S(=O)(=O)N5CCC(NC6=NC(C7=CN(CC(F)(F)F)N=C7)=C(C(F)(F)F)C=N6)CC5)=C4)CC3)C(C)(C)C)C=C2)SC=N1	C52H63F6N11O6S2	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-UR0NVP	WO2023249970A1_63	.	O=C1CCC(N2CCN(CC3=CC=CC(S(=O)(=O)N4CCC(NC5=NC(C6=CN(CC(F)(F)F)N=C6)=C(C(F)(F)F)C=N5)CC4)=C3)C3CC32)C(=O)N1	C32H35F6N9O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-JWFCTD	WO2023249970A1_64	.	CN1N=C(N2CCC(=O)NC2=O)C2=C1C(F)=C(C1CCN(CC3=CC=CC(S(=O)(=O)N4CCC(NC5=NC(C6=CN(CC(F)(F)F)N=C6)=C(C(F)(F)F)C=N5)CC4)=C3)CC1)C=C2	C39H40F7N11O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-BQGYPN	WO2023249970A1_65	3-[8-[[3-[4-[[4-[1-(2,2,2-Trifluoroethyl)pyrazol-4-yl]-5-(trifluoromethyl)pyrimidin-2-yl]amino]piperidin-1-yl]sulfonylphenyl]methyl]-3,8-diazabicyclo[3.2.1]octan-3-yl]piperidine-2,6-dione	O=C1CCC(N2CC3CCC(C2)N3CC2=CC=CC(S(=O)(=O)N3CCC(NC4=NC(C5=CN(CC(F)(F)F)N=C5)=C(C(F)(F)F)C=N4)CC3)=C2)C(=O)N1	C33H37F6N9O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-PLZUG5	WO2023249970A1_66	.	CN1N=C(N2CCC(=O)NC2=O)C2=C1C=C(C1CCN(CC3=CC=CC(S(=O)(=O)N4CC[C@H](NC5=NC(C6=CN(CC(F)(F)F)N=C6)=C(C(F)(F)F)C=N5)[C@@H](F)C4)=C3)CC1(C)F)C=C2	C40H41F8N11O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-FMPS3Z	WO2023249970A1_67	.	CN1N=C(N2CCC(=O)NC2=O)C2=C1C=C(N1CCN(CC3CCN(C4=CC=CC(S(=O)(=O)N5CCC(NC6=NC(C7=CN(CC(F)(F)F)N=C7)=C(C(F)(F)F)C=N6)CC5)=C4)CC3)CC1)C=C2	C43H49F6N13O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-KGK1RR	WO2023249970A1_68	.	O=C1CCC(NCC2=CC=CC(S(=O)(=O)N3CCC(NC4=NC(C5=CN(CC(F)(F)F)N=C5)=C(C(F)(F)F)C=N4)CC3)=C2)C(=O)N1	C27H28F6N8O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-F9U578	SCHEMBL30810446	1-[1-Methyl-6-[4-[[1-methyl-5-[4-[[4-[1-(2,2,2-trifluoroethyl)pyrazol-4-yl]-5-(trifluoromethyl)pyrimidin-2-yl]amino]piperidin-1-yl]sulfonylimidazol-2-yl]methyl]piperazin-1-yl]indazol-3-yl]-1,3-diazinane-2,4-dione	CN1N=C(N2CCC(=O)NC2=O)C2=C1C=C(N1CCN(CC3=NC=C(S(=O)(=O)N4CCC(NC5=NC(C6=CN(CC(F)(F)F)N=C6)=C(C(F)(F)F)C=N5)CC4)N3C)CC1)C=C2	C36H40F6N14O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-PFOCMZ	WO2023249970A1_7	.	N#CC1=C(C2=CN(CC(F)(F)F)N=C2)N=C(NC2CCN(S(=O)(=O)C3=CC(CN4CCN(C5=C(F)C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)=CC=C3)CC2)N=C1	C39H37F4N11O6S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-EHKG7R	WO2023249970A1_70	1-[6-[1-[[3-[(3R,4S)-3-fluoro-4-[[4-[1-(2-hydroxy-2-methylpropyl)pyrazol-4-yl]-5-(trifluoromethyl)pyrimidin-2-yl]amino]piperidin-1-yl]sulfonylphenyl]methyl]piperidin-4-yl]-1-methylindazol-3-yl]-1,3-diazinane-2,4-dione	CN1N=C(N2CCC(=O)NC2=O)C2=C1C=C(C1CCN(CC3=CC=CC(S(=O)(=O)N4CC[C@H](NC5=NC(C6=CN(CC(C)(C)O)N=C6)=C(C(F)(F)F)C=N5)[C@H](F)C4)=C3)CC1)C=C2	C41H47F4N11O5S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-QKFWXL	WO2023249970A1_71	.	O=C1CCN(C2=CC=C(N3CCN(CC4=CC=CC(S(=O)(=O)N5CCC(NC6=NC(C7=CN(C8=C(F)C=CC=C8)N=C7)=C(C(F)(F)F)C=N6)CC5)=C4)CC3)C=C2)C(=O)N1	C40H40F4N10O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-7P3H5C	WO2023249970A1_72	.	O=C1CCC(NC2CCN(CC3=CC=CC(S(=O)(=O)N4CCC(NC5=NC(C6=CN(CC(F)(F)F)N=C6)=C(C(F)(F)F)C=N5)CC4)=C3)CC2)C(=O)N1	C32H37F6N9O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-O99WZ9	WO2023249970A1_73	.	CN1N=C(N2CCC(=O)NC2=O)C2=CC(F)=C(N3CCN(CC4=CC=CC(S(=O)(=O)N5CC[C@H](NC6=NC(C7=CC(CC(F)(F)F)N=C7)=C(C(F)(F)F)C=N6)[C@H](F)C5)=C4)CC3)C=C21	C39H39F8N11O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-440115	SCHEMBL30810404	1-[1-Methyl-6-[1-[[3-[4-[[4-[1-(2,2,2-trifluoroethyl)pyrazol-4-yl]-5-(trifluoromethyl)pyrimidin-2-yl]amino]cyclohexyl]sulfonylphenyl]methyl]piperidin-4-yl]indazol-3-yl]-1,3-diazinane-2,4-dione	CN1N=C(N2CCC(=O)NC2=O)C2=C1C=C(C1CCN(CC3=CC=CC(S(=O)(=O)[C@H]4CC[C@H](NC5=NC(C6=CN(CC(F)(F)F)N=C6)=C(C(F)(F)F)C=N5)CC4)=C3)CC1)C=C2	C40H42F6N10O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-XWUTCQ	SCHEMBL30810391	1-[1-Methyl-6-[1-[[3-[4-[[4-(1-methylimidazol-4-yl)-5-(trifluoromethyl)pyrimidin-2-yl]amino]piperidin-1-yl]sulfonylphenyl]methyl]piperidin-4-yl]indazol-3-yl]-1,3-diazinane-2,4-dione	CN1C=NC(C2=C(C(F)(F)F)C=NC(NC3CCN(S(=O)(=O)C4=CC(CN5CCC(C6=CC7=C(C=C6)C(N6CCC(=O)NC6=O)=NN7C)CC5)=CC=C4)CC3)=N2)=C1	C38H42F3N11O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-TYEA3U	WO2023249970A1_76	.	O=C1CCC(N2CCN(CC3=CC=CC(S(=O)(=O)N4CCC(NC5=NC(C6=CN(CC(F)(F)F)N=C6)=C(C(F)(F)F)C=N5)CC4)=C3)CC2)C(=O)N1	C31H35F6N9O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-E8AF8F	WO2023249970A1_77	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3(F)CC3)C(C)(C)SCC3CCN(CC4=CC=CC5=C4C4CC(NC6=NC(C7=CN(CC(F)(F)F)N=C7)=C(C(F)(F)F)C=N6)CCN4S5(=O)=O)CC3)C=C2)SC=N1	C54H62F7N11O6S3	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-6U8J3T	SCHEMBL30810468	1-[1-Methyl-6-[1-[2-methyl-3-[3-[4-[[4-[1-(2,2,2-trifluoroethyl)pyrazol-4-yl]-5-(trifluoromethyl)pyrimidin-2-yl]amino]piperidin-1-yl]sulfonylphenyl]propyl]piperidin-4-yl]indazol-3-yl]-1,3-diazinane-2,4-dione	CC(CC1=CC=CC(S(=O)(=O)N2CCC(NC3=NC(C4=CN(CC(F)(F)F)N=C4)=C(C(F)(F)F)C=N3)CC2)=C1)CN1CCC(C2=CC3=C(C=C2)C(N2CCC(=O)NC2=O)=NN3C)CC1	C42H47F6N11O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-XJCAQU	WO2023249970A1_79	.	CN1CCC(N2C=C(C3=C(C(F)(F)F)C=NC(NC4CCN(S(=O)(=O)C5=CC(CN6CCC(C7=CC8=C(C=C7)C(N7CCC(=O)NC7=O)=NN8C)CC6)=CC=C5)CC4)=N3)C=N2)CC1	C43H51F3N12O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-6QDMFA	WO2023249970A1_8	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=CC(C3CCN(CC4=CC=CC(S(=O)(=O)N5CCC(NC6=NC(C7=CN(CC(F)(F)F)N=C7)=C(C(F)(F)F)C=N6)CC5)=C4)CC3)=C21	C40H42F6N10O5S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-EXW11L	WO2023249970A1_80	1-[1-[[3-[4-[[4-[1-(2,2,2-Trifluoroethyl)pyrazol-4-yl]-5-(trifluoromethyl)pyrimidin-2-yl]amino]piperidin-1-yl]sulfonylphenyl]methyl]piperidin-3-yl]-1,3-diazinane-2,4-dione	O=C1CCN(C2CCCN(CC3=CC=CC(S(=O)(=O)N4CCC(NC5=NC(C6=CN(CC(F)(F)F)N=C6)=C(C(F)(F)F)C=N5)CC4)=C3)C2)C(=O)N1	C31H35F6N9O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-KFRWME	WO2023249970A1_81	1-[1-[[3-[4-[[4-[1-(2,2,2-Trifluoroethyl)pyrazol-4-yl]-5-(trifluoromethyl)pyrimidin-2-yl]amino]piperidin-1-yl]sulfonylphenyl]methyl]pyrrolidin-3-yl]-1,3-diazinane-2,4-dione	O=C1CCN(C2CCN(CC3=CC=CC(S(=O)(=O)N4CCC(NC5=NC(C6=CN(CC(F)(F)F)N=C6)=C(C(F)(F)F)C=N5)CC4)=C3)C2)C(=O)N1	C30H33F6N9O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-2LDUDG	WO2023249970A1_82	.	CN1N=C(N2CCC(=O)NC2=O)C2=C1C=C(N1CC3CC(C1)N3CC1=CC=CC(S(=O)(=O)N3CC[C@H](NC4=NC(C5=CN(CC(F)(F)F)N=C5)=C(C(F)(F)F)C=N4)[C@H](F)C3)=C1)C=C2	C39H39F7N12O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-DS5OMG	SCHEMBL30810464	N-(2,6-dioxopiperidin-3-yl)-4-[[4-[1-(2,2,2-trifluoroethyl)pyrazol-4-yl]-5-(trifluoromethyl)pyrimidin-2-yl]amino]piperidine-1-sulfonamide	O=C1CCC(NS(=O)(=O)N2CCC(NC3=NC(C4=CN(CC(F)(F)F)N=C4)=C(C(F)(F)F)C=N3)CC2)C(=O)N1	C20H22F6N8O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-4F72WU	SCHEMBL30810420	1-[6-[1-[2,2-Difluoro-1-[3-[4-[[4-[1-(2,2,2-trifluoroethyl)pyrazol-4-yl]-5-(trifluoromethyl)pyrimidin-2-yl]amino]piperidin-1-yl]sulfonylphenyl]ethyl]piperidin-4-yl]-1-methylindazol-3-yl]-1,3-diazinane-2,4-dione	CN1N=C(N2CCC(=O)NC2=O)C2=C1C=C(C1CCN(C(C3=CC=CC(S(=O)(=O)N4CCC(NC5=NC(C6=CN(CC(F)(F)F)N=C6)=C(C(F)(F)F)C=N5)CC4)=C3)C(F)F)CC1)C=C2	C40H41F8N11O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-2IK97W	WO2023249970A1_85	.	CN1N=C(N2CCC(=O)NC2=O)C2=C1C=C(N1CC3CCC(C1)N3CC1=CCCC(S(=O)(=O)N3CC[C@H](NC4=NC(C5=CN(CC(F)(F)F)N=C5)=C(C(F)(F)F)C=N4)[C@H](F)C3)=C1)C=C2	C40H43F7N12O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-SSSS72	WO2023249970A1_86	.	CN1N=C(N2CCC(=O)NC2=O)C2=C1C=C(N1CCN(CC3CCN(S(=O)(=O)N4CCC(NC5=NC(C6=CN(CC(F)(F)F)N=C6)=C(C(F)(F)F)C=N5)CC4)CC3)CC1)C=C2	C37H45F6N13O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-FSL5D7	SCHEMBL30810416	1-[1-Methyl-6-[1-[[3-[4-[[4-[1-(2,2,2-trifluoroethyl)pyrazol-4-yl]-5-(trifluoromethyl)pyrimidin-2-yl]amino]piperidin-1-yl]sulfonyl-2-(trifluoromethyl)phenyl]methyl]piperidin-4-yl]indazol-3-yl]-1,3-diazinane-2,4-dione	CN1N=C(N2CCC(=O)NC2=O)C2=C1C=C(C1CCN(CC3=CC=CC(S(=O)(=O)N4CCC(NC5=NC(C6=CN(CC(F)(F)F)N=C6)=C(C(F)(F)F)C=N5)CC4)=C3C(F)(F)F)CC1)C=C2	C40H40F9N11O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-FVGPFY	WO2023249970A1_88	.	CN1N=C(N2CCC(=O)NC2=O)C2=C1C=C(C1CCN(CC3CCN(S(=O)(=O)N4CCC(NC5=NC(C6=CN(CC(F)(F)F)N=C6)=C(C(F)(F)F)C=N5)CC4)C3)CC1)C=C2	C37H44F6N12O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-E8UCPO	SCHEMBL30810356	1-[1-Methyl-6-[1-[[3-[4-[[4-[1-(2,2,2-trifluoroethyl)pyrazol-4-yl]-5-(trifluoromethyl)pyrimidin-2-yl]amino]piperidin-1-yl]sulfonylcyclohexyl]methyl]piperidin-4-yl]indazol-3-yl]-1,3-diazinane-2,4-dione	CN1N=C(N2CCC(=O)NC2=O)C2=C1C=C(C1CCN(CC3CCCC(S(=O)(=O)N4CCC(NC5=NC(C6=CN(CC(F)(F)F)N=C6)=C(C(F)(F)F)C=N5)CC4)C3)CC1)C=C2	C39H47F6N11O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-5WM0ED	WO2023249970A1_9	.	O=C1CCC(N2C(=O)C3=CC(F)=C(N4CCN(CC5=CC=CC(S(=O)(=O)N6CCC(NC7=NC(C8=CN(CC(F)(F)F)N=C8)=C(Cl)C=N7)CC6)=C5)CC4)C=C3C2=O)C(=O)N1	C38H37ClF4N10O6S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-47490Z	SCHEMBL30810388	1-[1-Methyl-6-[1-[2-methyl-2-[3-[4-[[4-[1-(2,2,2-trifluoroethyl)pyrazol-4-yl]-5-(trifluoromethyl)pyrimidin-2-yl]amino]piperidin-1-yl]sulfonylphenyl]propyl]piperidin-4-yl]indazol-3-yl]-1,3-diazinane-2,4-dione	CN1N=C(N2CCC(=O)NC2=O)C2=C1C=C(C1CCN(CC(C)(C)C3=CC=CC(S(=O)(=O)N4CCC(NC5=NC(C6=CN(CC(F)(F)F)N=C6)=C(C(F)(F)F)C=N5)CC4)=C3)CC1)C=C2	C42H47F6N11O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-X2IJCT	WO2023249970A1_91	.	CN1N=C(N2CCC(=O)NC2=O)C2=C1C=C(C1CCN(C(C3=CC=CC(S(=O)(=O)N4CCC(NC5=NC(C6=CN(CC(F)(F)F)N=C6)=C(C(F)(F)F)C=N5)CC4)=C3)C(F)(F)F)CC1)C=C2	C40H40F9N11O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-2QC1UA	WO2023249970A1_92	.	CN1N=C(N2CCC(=O)NC2=O)C2=C1C=C(N1CCC(CN3CCC(S(=O)(=O)N4CCC(NC5=NC(C6=CN(CC(F)(F)F)N=C6)=C(C(F)(F)F)C=N5)CC4)CC3)CC1)C=C2	C38H46F6N12O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-ZMJZHU	SCHEMBL30810483	1-[1-Methyl-6-[1-[1-[3-[4-[[4-[1-(2,2,2-trifluoroethyl)pyrazol-4-yl]-5-(trifluoromethyl)pyrimidin-2-yl]amino]piperidin-1-yl]sulfonylphenyl]propan-2-yl]piperidin-4-yl]indazol-3-yl]-1,3-diazinane-2,4-dione	CC(CC1=CC=CC(S(=O)(=O)N2CCC(NC3=NC(C4=CN(CC(F)(F)F)N=C4)=C(C(F)(F)F)C=N3)CC2)=C1)N1CCC(C2=CC3=C(C=C2)C(N2CCC(=O)NC2=O)=NN3C)CC1	C41H45F6N11O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-TRJXFO	SCHEMBL30810353	1-[1-Methyl-6-[1-[[1-[4-[[4-[1-(2,2,2-trifluoroethyl)pyrazol-4-yl]-5-(trifluoromethyl)pyrimidin-2-yl]amino]cyclohexyl]sulfonylpiperidin-4-yl]methyl]piperidin-4-yl]indazol-3-yl]-1,3-diazinane-2,4-dione	CN1N=C(N2CCC(=O)NC2=O)C2=C1C=C(C1CCN(CC3CCN(S(=O)(=O)[C@H]4CC[C@H](NC5=NC(C6=CN(CC(F)(F)F)N=C6)=C(C(F)(F)F)C=N5)CC4)CC3)CC1)C=C2	C39H47F6N11O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-7SRUJB	SCHEMBL30810397	1-[1-Methyl-6-[1-[2-[3-[4-[[4-[1-(2,2,2-trifluoroethyl)pyrazol-4-yl]-5-(trifluoromethyl)pyrimidin-2-yl]amino]cyclohexyl]sulfonylphenyl]ethyl]piperidin-4-yl]indazol-3-yl]-1,3-diazinane-2,4-dione	CN1N=C(N2CCC(=O)NC2=O)C2=C1C=C(C1CCN(CCC3=CC=CC(S(=O)(=O)[C@H]4CC[C@H](NC5=NC(C6=CN(CC(F)(F)F)N=C6)=C(C(F)(F)F)C=N5)CC4)=C3)CC1)C=C2	C41H44F6N10O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-GJ3FTD	WO2023249970A1_96	.	CC(CC1=CC=CC(S(=O)(=O)N2CCC(NC3=NC(C4=CN(C5=C(F)C=CC=C5)N=C4)=C(C(F)(F)F)C=N3)CC2)=C1)N1CCC(C2=CC3=C(C=C2)C(N2CCC(=O)NC2=O)=NN3C)CC1	C45H47F4N11O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-78G0YG	WO2023249970A1_97	1-[1-Methyl-6-[4-[[4-[4-[[4-[1-(2,2,2-trifluoroethyl)pyrazol-4-yl]-5-(trifluoromethyl)pyrimidin-2-yl]amino]piperidin-1-yl]sulfonylpiperazin-1-yl]methyl]piperidin-1-yl]indazol-3-yl]-1,3-diazinane-2,4-dione	CN1N=C(N2CCC(=O)NC2=O)C2=C1C=C(N1CCC(CN3CCN(S(=O)(=O)N4CCC(NC5=NC(C6=CN(CC(F)(F)F)N=C6)=C(C(F)(F)F)C=N5)CC4)CC3)CC1)C=C2	C37H45F6N13O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-CE1I9B	SCHEMBL30810539	1-[6-[1-[2,2-Dimethyl-3-[3-[4-[[4-[1-(2,2,2-trifluoroethyl)pyrazol-4-yl]-5-(trifluoromethyl)pyrimidin-2-yl]amino]piperidin-1-yl]sulfonylphenyl]propyl]piperidin-4-yl]-1-methylindazol-3-yl]-1,3-diazinane-2,4-dione	CN1N=C(N2CCC(=O)NC2=O)C2=C1C=C(C1CCN(CC(C)(C)CC3=CC=CC(S(=O)(=O)N4CCC(NC5=NC(C6=CN(CC(F)(F)F)N=C6)=C(C(F)(F)F)C=N5)CC4)=C3)CC1)C=C2	C43H49F6N11O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-XB23FZ	WO2023249970A1_99	.	O=C1CCN(C2=NN(CC(F)(F)F)C3=C2C=CC(N2CCN(CC4=CC=CC(S(=O)(=O)N5CCC(NC6=NC(C7=CN(CC(F)(F)F)N=C7)=C(C(F)(F)F)C=N6)CC5)=C4)CC2)=C3)C(=O)N1	C39H39F9N12O4S	CDK2	P24941	CRBN	WO-2023249970-A1
TPD-X34DVP	WO2024019103A1_1	.	CC1=C(C2=C(C3CC3)C=C3C(N4C[C@@H]5C[C@H]4CN5)=NC(OC4CCOCC4)=NC3=C2OCC2=CC=C(C(=O)N3CCN(CC4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)C=C2)C2=C(C=C1F)NN=C2	C55H55FN10O8	KRAS	P01116	CRBN	WO-2024019103-A1
TPD-JWALEN	SCHEMBL27034438	3-[5-[[(3S)-4-[4-[[6-cyclopropyl-4-[(1S,4S)-2,5-diazabicyclo[2.2.1]heptan-2-yl]-7-(6-fluoro-5-methyl-1H-indazol-4-yl)-2-[(2S)-2-methoxypropoxy]quinazolin-8-yl]oxymethyl]benzoyl]-3-methylpiperazin-1-yl]methyl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione; SCHEMBL30798870	CO[C@@H](C)COC1=NC2=C(OCC3=CC=C(C(=O)N4CCN(CC5=CC=C6C(=C5)N(C)C(=O)N6C5CCC(=O)NC5=O)C[C@@H]4C)C=C3)C(C3=C(C)C(F)=CC4=C3C=NN4)=C(C3CC3)C=C2C(N2C[C@@H]3C[C@H]2CN3)=N1	C55H60FN11O7	KRAS	P01116	CRBN	WO-2024019103-A1
TPD-NZTJ0M	WO2024019103A1_11	.	CC1=C(C2=C(C3CC3)C=C3C(N4C[C@@H]5C[C@H]4CN5)=NC(OC4CCOCC4)=NC3=C2OCC2=CC=C(C(=O)N3CCN(CC4=CC=C5C(=N4)N(C)C(=O)N5C4CCC(=O)NC4=O)CC3)C=C2)C2=C(C=C1F)NN=C2	C54H57FN12O7	KRAS	P01116	CRBN	WO-2024019103-A1
TPD-12G339	WO2024019103A1_12	.	CO[C@H](COC1=CC(O[C@H]2CCNC2)=C2C=C(C3CC3)C(C3=C(C)C(F)=CC4=C3C=NN4)=C(OCC3=CC=C(C(=O)N4CCN(CC5=CC6=C(C=C5)N(C5CCC(=O)NC5=O)C(=O)N6C)C[C@@H]4C)C=C3)C2=N1)N=NC#N	C55H57FN12O8	KRAS	P01116	CRBN	WO-2024019103-A1
TPD-F1P50P	WO2024019103A1_13	.	CC1=C(C2=C(C3CC3)C=C3C(N4C[C@@H]5C[C@H]4CN5)=NC(OC4CCOCC4)=NC3=C2OCC2=CC=C(C(=O)N3CCN(CC4=CC5=C(C=C4)C(N4CCC(=O)NC4=O)=NN5C)CC3)C=C2)C2=C(C=C1F)NN=C2	C54H57FN12O6	KRAS	P01116	CRBN	WO-2024019103-A1
TPD-M40UBE	WO2024019103A1_14	.	CC1=C(N2CCC(=O)NC2=O)C=CC(N2CCN(C(=O)C3=CC=C(COC4=C5N=C(OC6CCOCC6)N=C(N6C[C@@H]7C[C@H]6CN7)C5=CC(C5CC5)=C4C4=C(C)C(F)=CC5=C4C=NN5)C=C3)CC2)=N1	C51H54FN11O6	KRAS	P01116	CRBN	WO-2024019103-A1
TPD-W1IAZS	WO2024019103A1_15	.	CC1=C(C2=C(C3CC3)C=C3C(N4C[C@@H]5C[C@H]4CN5)=NC(OC4CCOCC4)=NC3=C2OCC2=CC=C(C(=O)N3CCN(CC4=CC5=C(C=C4)C(N4CCC(=O)NC4=O)=NN5C)C[C@H]3C)C=C2)C2=C(C=C1F)NN=C2	C55H59FN12O6	KRAS	P01116	CRBN	WO-2024019103-A1
TPD-3DWW17	SCHEMBL27034544	1-[6-[[(3S)-4-[4-[[6-cyclopropyl-4-[(1S,4S)-2,5-diazabicyclo[2.2.1]heptan-2-yl]-7-(6-fluoro-5-methyl-1H-indazol-4-yl)-2-(oxan-4-yloxy)quinazolin-8-yl]oxymethyl]benzoyl]-3-methylpiperazin-1-yl]methyl]-1-methylindazol-3-yl]-1,3-diazinane-2,4-dione; SCHEMBL30798817	CC1=C(C2=C(C3CC3)C=C3C(N4C[C@@H]5C[C@H]4CN5)=NC(OC4CCOCC4)=NC3=C2OCC2=CC=C(C(=O)N3CCN(CC4=CC5=C(C=C4)C(N4CCC(=O)NC4=O)=NN5C)C[C@@H]3C)C=C2)C2=C(C=C1F)NN=C2	C55H59FN12O6	KRAS	P01116	CRBN	WO-2024019103-A1
TPD-ZFZMB2	WO2024019103A1_17	.	CC1=NC(OC2CCN(C(=O)C3=CC=C(COC4=C(C5=C(C)C(F)=CC6=C5C=NN6)C(C5CC5)=CC5=C(N6C[C@@H]7C[C@H]6CN7)N=C(OC6CCOCC6)N=C54)C=C3)CC2)=CC=C1N1CCC(=O)NC1=O	C52H55FN10O7	KRAS	P01116	CRBN	WO-2024019103-A1
TPD-0C59HW	WO2024019103A1_18	.	CO[C@@H](C)COC1=NC2=C(OCC3=CC=C(C(=O)N4CCN(CC5=CC6=C(C=C5)N(C5CCC(=O)NC5=O)C(=O)N6C)C[C@@H]4C)C=C3)C(C3=C(C)C(F)=CC4=C3C=NN4)C(C3CC3)C=C2C(N(C)[C@H]2CCNC2)=N1	C55H64FN11O7	KRAS	P01116	CRBN	WO-2024019103-A1
TPD-BG3PAY	WO2024019103A1_19	.	CC1=C(C2=C(OCC3=CC=C(C(=O)N4CCC5(CN(CC6=CC7=C(C=C6)C(N6CCC(=O)NC6=O)=NN7C)C5)C4)C=C3)C3=NC(OC4CCOCC4)=NC(N4C[C@@H]5C[C@H]4CN5)=C3C=C2C2CC2)C2=C(C=C1F)NN=C2	C56H59FN12O6	KRAS	P01116	CRBN	WO-2024019103-A1
TPD-RY0YMZ	WO2024019103A1_2	.	CC1=C(C2=C(C3CC3)C=C3C(N4C[C@@H]5C[C@H]4CN5)=NC(OC4CCOCC4)=NC3=C2OCC2=CC=C(C(=O)N3CCC(CN4CCN(C5=CC6=C(C=C5F)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)C=C2)C2=C(C=C1F)NN=C2	C60H63F2N11O8	KRAS	P01116	CRBN	WO-2024019103-A1
TPD-SRFQ7E	WO2024019103A1_20	.	CC1=C(C2=C(C3CC3)C=C3C(N4C[C@@H]5C[C@H]4CN5)=NC(OC4CCOCC4)=NC3=C2OCC2=CC=C(C(=O)N3CC[C@H](N(C)CC4=CC5=C(C=C4)C(N4CCC(=O)NC4=O)=NN5C)C3)C=C2)C2=C(C=C1F)NN=C2	C55H59FN12O6	KRAS	P01116	CRBN	WO-2024019103-A1
TPD-XH6EBE	WO2024019103A1_21	.	CC1=C(OC2CCN(C(=O)C3=CC=C(COC4=C5N=C(OC6CCOCC6)N=C(N6C[C@@H]7C[C@H]6CN7)C5=CC(C5CC5)=C4C4=C(C)C(F)=CC5=C4C=NN5)C=C3)CC2)N=CC=C1N1CCC(=O)NC1=O	C52H55FN10O7	KRAS	P01116	CRBN	WO-2024019103-A1
TPD-IW6ELQ	WO2024019103A1_22	.	CC1=C(C2=C(C)C(F)=CC3=C2C=NN3)C(OCC2=CC=C(C(=O)N3CCN(CC4=CC5=NN(C)C(N6CCC(=O)NC6=O)=C5C=C4)C[C@@H]3C)C=C2)=C2N=C(OC3CCOCC3)N=C(N3C[C@@H]4C[C@H]3CN4)C2=C1	C53H57FN12O6	KRAS	P01116	CRBN	WO-2024019103-A1
TPD-7RIW5U	WO2024019103A1_23	.	CC1=C(C2=C(C3CC3)C=C3C(N4C[C@@H]5C[C@H]4CN5)=NC(OC4CCOCC4)=NC3=C2OCC2=CC=C(C(=O)N3CCN(CC4=C5C(=CC=C4)C(N4CCC(=O)NC4=O)=NN5C)CC3)C=C2)C2=C(C=C1F)NN=C2	C54H57FN12O6	KRAS	P01116	CRBN	WO-2024019103-A1
TPD-3RN8XA	WO2024019103A1_24	.	CC1=C(C2=C(C3CC3)C=C3C(N4C[C@@H]5C[C@H]4CN5)=NC(OC4CCOCC4)=NC3=C2OCC2=CC=C(C(=O)N3CCN(CC4=NC5=C(C=C4)C(N4CCC(=O)NC4=O)=NN5C)C[C@@H]3C)C=C2)C2=C(C=C1F)NN=C2	C54H58FN13O6	KRAS	P01116	CRBN	WO-2024019103-A1
TPD-C1V3R5	WO2024019103A1_25	.	CC[C@H]1CN(CC2=CC3=C(C=C2)C(N2CCC(=O)NC2=O)=NN3C)CCN1C(=O)C1=CC=C(COC2=C3N=C(OC4CCOCC4)N=C(N4C[C@@H]5C[C@H]4CN5)C3=CC(C3CC3)=C2C2=C(C)C(F)=CC3=C2C=NN3)C=C1	C56H61FN12O6	KRAS	P01116	CRBN	WO-2024019103-A1
TPD-JZ9ZZ6	WO2024019103A1_26	.	CC1=C(C2=C(OCC3=CC=C(C(=O)N4CCN(CC5=C(F)C=C(CN6CCC(=O)NC6=O)C=C5)C[C@@H]4C)C=C3)C3=NC(OC4CCOCC4)=NC(N4C[C@@H]5C[C@H]4CN5)=C3C=C2C2CC2)C2=C(C=C1F)NN=C2	C54H58F2N10O6	KRAS	P01116	CRBN	WO-2024019103-A1
TPD-QFKT6Z	WO2024019103A1_27	.	CC1=C(C2=C(C3CC3)C=C3C(N4C[C@@H]5C[C@H]4CN5)=NC(OC4CCOCC4)=NC3=C2OCC2=CC=C(C(=O)N3CCN(CC4=CC5=C(C=C4)N(C)N=C5N4CCC(=O)NC4=O)C[C@@H]3C)C=C2)C2=C(C=C1F)NN=C2	C55H59FN12O6	KRAS	P01116	CRBN	WO-2024019103-A1
TPD-LFH9TR	WO2024019103A1_28	.	CC1=C(C2=C(C3CC3)C=C3C(N4C[C@@H]5C[C@H]4CN5)=NC(OC4CCOCC4)=NC3=C2OCC2=CC=C(C(=O)N3CCN(CCOC4=CC(N5CCC(=O)NC5=O)=CC=C4)CC3)C=C2)C2=C(C=C1F)NN=C2	C53H57FN10O7	KRAS	P01116	CRBN	WO-2024019103-A1
TPD-UL7NYA	SCHEMBL27034437	3-[5-[[(3S)-4-[4-[[6-cyclopropyl-4-[(1S,4S)-2,5-diazabicyclo[2.2.1]heptan-2-yl]-7-(6-fluoro-5-methyl-1H-indazol-4-yl)-2-[(2S)-2-methoxypropoxy]quinolin-8-yl]oxymethyl]benzoyl]-3-methylpiperazin-1-yl]methyl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione; SCHEMBL30798726	CO[C@@H](C)COC1=CC(N2C[C@@H]3C[C@H]2CN3)=C2C=C(C3CC3)C(C3=C(C)C(F)=CC4=C3C=NN4)=C(OCC3=CC=C(C(=O)N4CCN(CC5=CC6=C(C=C5)N(C5CCC(=O)NC5=O)C(=O)N6C)C[C@@H]4C)C=C3)C2=N1	C56H61FN10O7	KRAS	P01116	CRBN	WO-2024019103-A1
TPD-A1CVJF	WO2024019103A1_3	.	CC1=C(C2=C(C3CC3)C=C3C(N4C[C@@H]5C[C@H]4CN5)=NC(OC4CCOCC4)=NC3=C2OCC2=CC=C(C(=O)N3CCN(CC4=CC=C5C(=C4)OC(=O)N5C4CCC(=O)NC4=O)CC3)C=C2)C2=C(C=C1F)NN=C2	C54H55FN10O8	KRAS	P01116	CRBN	WO-2024019103-A1
TPD-WDJOCW	WO2024019103A1_30	.	CC1=C(C2=C(OCC3=CC=C(C(=O)N4CCC(CNC5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)CC4)C=C3)C3=NC(OC4CCOCC4)=NC(N4C[C@@H]5C[C@H]4CN5)=C3C=C2C2CC2)C2=C(C=C1F)NN=C2	C56H57FN10O8	KRAS	P01116	CRBN	WO-2024019103-A1
TPD-XPH83S	WO2024019103A1_31	.	CC1=C(C2=C(OCC3=CC=C(C(=O)N4CCN(CC5=CC6=C(C=C5)N(C5CCC(=O)NC5=O)C(=O)N6C)C[C@@H]4C)C=C3)C3=NC(OC[C@@H]4CCCO4)=CC(O[C@H]4CCNC4)=C3C=C2C2CC2)C2=C(C=C1F)NN=C2	C56H60FN9O8	KRAS	P01116	CRBN	WO-2024019103-A1
TPD-I9SQZ8	WO2024019103A1_32	.	CC1=C(C2=C(OCC3=CC=C(C(=O)N4CCN(CC5=CC6=C(C=C5)N(C5CCC(=O)NC5=O)C(=O)N6C)C[C@@H]4C)C=C3)C3=NC(OC[C@H]4CCCO4)=CC(O[C@H]4CCNC4)=C3C=C2C2CC2)C2=C(C=C1F)NN=C2	C56H60FN9O8	KRAS	P01116	CRBN	WO-2024019103-A1
TPD-O16JH4	SCHEMBL27034441	3-[6-[[(3S)-4-[4-[[6-cyclopropyl-4-[(1S,4S)-2,5-diazabicyclo[2.2.1]heptan-2-yl]-7-(6-fluoro-5-methyl-1H-indazol-4-yl)-2-(oxan-4-yloxy)quinazolin-8-yl]oxymethyl]benzoyl]-3-methylpiperazin-1-yl]methyl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; SCHEMBL30798729	CC1=C(C2=C(OCC3=CC=C(C(=O)N4CCN(CC5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6)C[C@@H]4C)C=C3)C3=NC(OC4CCOCC4)=NC(N4C[C@@H]5C[C@H]4CN5)=C3C=C2C2CC2)C2=C(C=C1F)NN=C2	C56H59FN10O7	KRAS	P01116	CRBN	WO-2024019103-A1
TPD-ZPZC6K	SCHEMBL27034500	1-[7-[[(3S)-4-[4-[[6-cyclopropyl-4-[(1S,4S)-2,5-diazabicyclo[2.2.1]heptan-2-yl]-7-(6-fluoro-5-methyl-1H-indazol-4-yl)-2-(oxan-4-yloxy)quinazolin-8-yl]oxymethyl]benzoyl]-3-methylpiperazin-1-yl]methyl]imidazo[1,2-a]pyridin-3-yl]-1,3-diazinane-2,4-dione; SCHEMBL30798732	CC1=C(C2=C(OCC3=CC=C(C(=O)N4CCN(CC5=CC6=NC=C(N7CCC(=O)NC7=O)N6C=C5)C[C@@H]4C)C=C3)C3=NC(OC4CCOCC4)=NC(N4C[C@@H]5C[C@H]4CN5)=C3C=C2C2CC2)C2=C(C=C1F)NN=C2	C54H57FN12O6	KRAS	P01116	CRBN	WO-2024019103-A1
TPD-MPTH9D	WO2024019103A1_35	.	CO[C@@H](C)COC1=NC2=C(C=C(C3CC3)C(C3=C(C)C(F)=CC4=C3C=NN4)=C2OCC2=CC=C(C(=O)N3CCN(CC4=CC=C5C(=C4)N(C)C(=O)N5C4CCC(=O)NC4=O)C[C@H]3C)C=C2)C(N(C)[C@@H]2CCNC2)=N1	C55H62FN11O7	KRAS	P01116	CRBN	WO-2024019103-A1
TPD-9VJI38	WO2024019103A1_36	.	CC1=C(C2=C(OCC3=CC=C(C(=O)N4CCN(CC5=CC=C6C(C5)N(C)C(=O)N6C5CCC(=O)NC5=O)C[C@@H]4C)C=C3)C3=C(C=C2C2CC2)C(N2C[C@@H]4C[C@H]2CN4)=NC(O[C@@H]2CCOC2)=N3)C2=C(C=C1F)NN=C2	C55H60FN11O7	KRAS	P01116	CRBN	WO-2024019103-A1
TPD-4IWYZ1	WO2024019103A1_37	.	CC1=C(C2=C(OCC3=CC=C(C(=O)N4CCN(CC5=CC=C6C(=C5)N(C)C(=O)N6C5CCC(=O)NC5=O)C[C@@H]4C)C=C3)C3=C(C=C2C2CC2)C(N2C[C@@H]4C[C@H]2CN4)=NC(OC[C@H]2CCCO2)=N3)C2=C(C=C1F)NN=C2	C56H60FN11O7	KRAS	P01116	CRBN	WO-2024019103-A1
TPD-DQJVHM	WO2024019103A1_38	.	CO[C@H](C)COC1=NC2=C(C=C(C3CC3)C(C3=C(C)C(F)=CC4=C3C=NN4)=C2OCC2=CC=C(C(=O)N3CCN(CC4=CC=C5C(=C4)N(C)C(=O)N5C4CCC(=O)NC4=O)C[C@@H]3C)C=C2)C(N2C[C@@H]3C[C@H]2CN3)=N1	C55H60FN11O7	KRAS	P01116	CRBN	WO-2024019103-A1
TPD-R9GAEE	WO2024019103A1_39	.	CO[C@@H](C)COC1=NC2=C(C=C(C3CC3)C(C3=C(C)C(F)=CC4=C3C=NN4)=C2OCC2=CC=C(C(=O)N3CCN(CC4=CC=C5C(=C4)N(C)C(=O)N5C4CCC(=O)NC4=O)C[C@@H]3C)C=C2)C(O[C@@H]2CCNC2)=N1	C54H59FN10O8	KRAS	P01116	CRBN	WO-2024019103-A1
TPD-O4BXF5	WO2024019103A1_4	.	CC1=C(C2=C(C3CC3)C=C3C(N4C[C@@H]5C[C@H]4CN5)=NC(OC4CCOCC4)=NC3=C2OCC2=CC=C(C(=O)N3C[C@H]4C[C@@H]3CN4CC3=CC=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)C=C2)C2=C(C=C1F)NN=C2	C56H55FN10O8	KRAS	P01116	CRBN	WO-2024019103-A1
TPD-V8Q2YX	WO2024019103A1_40	.	CC1=C(C2=C(OCC3=CC=C(C(=O)N4CCN(CC5=CC=C6C(=C5)N(C)C(=O)N6C5CCC(=O)NC5=O)C[C@@H]4C)C=C3)C3=C(C=C2C2CC2)C(N2C[C@@H]4C[C@H]2CN4)=NC(OC[C@@H]2CCCO2)=N3)C2=C(C=C1F)NN=C2	C56H60FN11O7	KRAS	P01116	CRBN	WO-2024019103-A1
TPD-BYLMQW	WO2024019103A1_41	.	CC1=C(C2=C(OCC3=CC=C(C(=O)N4CCN(CC5=CC=C6C(=C5)N(C)C(=O)N6C5CCC(=O)NC5=O)C[C@@H]4C)C=C3)C3=C(C=C2C2CC2)C(N2C[C@@H]4C[C@H]2CN4)=NC(O[C@H]2CCOC2)=N3)C2=C(C=C1F)NN=C2	C55H58FN11O7	KRAS	P01116	CRBN	WO-2024019103-A1
TPD-MZZ0OC	WO2024019103A1_42	.	CC1=C(C2=C(C3CC3)C=C3C(N4C[C@@H]5C[C@H]4CN5)=NC(OC4CCOCC4)=NC3=C2OCC2=CC=C(C(=O)N3CCN(CCC4=CC5=C(C=C4)N(C)N=C5N4CCC(=O)N=NC4=O)C[C@@H]3C)C=C2)C2=C(C=C1F)NN=C2	C56H60FN13O6	KRAS	P01116	CRBN	WO-2024019103-A1
TPD-MD35ZD	WO2024019103A1_43	.	CO[C@@H](C)COC1=NC2=C(C=C(C3CC3)C(C3=C(C)C(F)=CC4=C3C=NN4)=C2OCC2=CC=C(C(=O)N3CCN(CC4=CC=C5C(=C4)N(C)C(=O)N5C4CCC(=O)NC4=O)C[C@@H]3C)C=C2)C(O[C@H]2CCNC2)=N1	C54H59FN10O8	KRAS	P01116	CRBN	WO-2024019103-A1
TPD-RZNKOH	WO2024019103A1_44	.	CO[C@H](C)COC1=CC(O[C@H]2CCNC2)=C2C=C(C3CC3)C(C3=C(C)C(F)=CC4=C3C=NN4)=C(OCC3=CC=C(C(=O)N4CCN(CC5=CC6=C(C=C5)N(C5CCC(=O)NC5=O)C(=O)N6C)C[C@@H]4C)C=C3)C2=N1	C55H60FN9O8	KRAS	P01116	CRBN	WO-2024019103-A1
TPD-K9VO1N	WO2024019103A1_45	.	CO[C@@H](C)COC1=NC2=C(OCC3=CC=C(C(=O)N4CCN(CC5=CC=C6C(=C5)N(C)C(=O)N6C5CCC(=O)NC5=O)C[C@@H]4C)C=C3)C(C3=C(C)C(F)=CC4=C3C=NN4)=C(C3CC3)C=C2C(N2CCNCC2)=N1	C54H60FN11O7	KRAS	P01116	CRBN	WO-2024019103-A1
TPD-D89CXH	WO2024019103A1_46	.	CC1=C(C2=C(C3CC3)C=C3C(N4C[C@@H]5C[C@H]4CN5)=NC(OC4CCOCC4)=NC3=C2OCC2=CC=C(C(=O)N3CCN(CC4=CC5=C(C=C4)N(C)C(=O)C(N4CCC(=O)NC4=O)=C5)C[C@@H]3C)C=C2)C2=C(C=C1F)NN=C2	C57H60FN11O7	KRAS	P01116	CRBN	WO-2024019103-A1
TPD-2FUFYP	WO2024019103A1_47	.	CC1=C(C2=C(CC3CC3)C=C3C(N4C[C@@H]5C[C@H]4CN5)=NC(OC4CCOCC4)=NC3=C2OCC2=CC=C(C(=O)N3CCN(CC4=CC=C5C(=C4)N(C)C(=O)N5N4CCC(=O)NC4=O)C[C@@H]3C)C=C2)C2=C(C=C1F)NN=C2	C56H61FN12O7	KRAS	P01116	CRBN	WO-2024019103-A1
TPD-D73DCQ	WO2024019103A1_48	.	CC1=C(F)C=C2NN=CC2=C1C1=C(C2CC2)N=C2C(N3C[C@@H]4C[C@H]3CN4)=NC(OC3CCOCC3)=NC2=C1OCC1=CC=C(C(=O)N2CCN(CC3=CC4=C(C=C3)N(C3CCC(=O)NC3=O)C(=O)N4C)C[C@@H]2C)C=C1	C55H59FN12O7	KRAS	P01116	CRBN	WO-2024019103-A1
TPD-5MY85K	SCHEMBL27034571	3-[5-[[(3S)-4-[4-[[6-cyclopropyl-4-[(1S,4S)-2,5-diazabicyclo[2.2.1]heptan-2-yl]-7-(6-fluoro-5-methyl-1H-indazol-4-yl)-2-(oxan-4-yloxy)quinazolin-8-yl]oxymethyl]benzoyl]-3-methylpiperazin-1-yl]methyl]-3-methyl-2-oxobenzimidazol-1-yl]piperidine-2,6-dione; SCHEMBL30798806	CC1=C(C2=C(C3CC3)C=C3C(N4C[C@@H]5C[C@H]4CN5)=NC(OC4CCOCC4)=NC3=C2OCC2=CC=C(C(=O)N3CCN(CC4=CC=C5C(=C4)N(C)C(=O)N5C4CCC(=O)NC4=O)C[C@@H]3C)C=C2)C2=C(C=C1F)NN=C2	C56H60FN11O7	KRAS	P01116	CRBN	WO-2024019103-A1
TPD-7YBUOP	SCHEMBL27034467	5-[[8-[4-[[6-cyclopropyl-4-[(1S,4S)-2,5-diazabicyclo[2.2.1]heptan-2-yl]-7-(6-fluoro-5-methyl-1H-indazol-4-yl)-2-(oxan-4-yloxy)quinazolin-8-yl]oxymethyl]benzoyl]-3,8-diazabicyclo[3.2.1]octan-3-yl]methyl]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione; SCHEMBL30798787	CC1=C(C2=C(C3CC3)C=C3C(N4C[C@@H]5C[C@H]4CN5)=NC(OC4CCOCC4)=NC3=C2OCC2=CC=C(C(=O)N3C4CCC3CN(CC3=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C3)C4)C=C2)C2=C(C=C1F)NN=C2	C57H57FN10O8	KRAS	P01116	CRBN	WO-2024019103-A1
TPD-60GFY6	WO2024019103A1_50	.	CO[C@@H](C)COC1=NC2=C(OCC3=CC=C(C(=O)N4CCN(CC5=CC=C6C(=C5)N(C)C(O)N6C5CCC(=O)NC5=O)C[C@@H]4C)C=C3)C(C3=C(C)C(F)=CC4=C3C=NN4)=C(C3CC3)C=C2C(N2C[C@@H]3C[C@H]2CN3)=N1	C55H62FN11O7	KRAS	P01116	CRBN	WO-2024019103-A1
TPD-5O1VBH	WO2024019103A1_6	.	CC1=C(C2=C(C3CC3)C=C3C(N4C[C@@H]5C[C@H]4CN5)=NC(OC4CCOCC4)=NC3=C2OCC2=CC=C(C(=O)N3CCN(CC4=C5OC(=O)N(C6CCC(=O)NC6=O)C5=CC=C4)CC3)C=C2)C2=C(C=C1F)NN=C2	C54H55FN10O8	KRAS	P01116	CRBN	WO-2024019103-A1
TPD-HO7KL4	WO2024019103A1_7	.	CC1=C(C2=C(C3CC3)C=C3C(N4C[C@@H]5C[C@H]4CN5)=NC(OC4CCOCC4)=NC3=C2OCC2=CC=C(C(=O)N3CCN(CC4=CC=C5C(=C4)N(C)C(=O)N5C4CCC(=O)NC4=O)CC3)C=C2)C2=C(C=C1F)NN=C2	C55H58FN11O7	KRAS	P01116	CRBN	WO-2024019103-A1
TPD-BYRO1N	WO2024019103A1_9	.	CC1=C(C2=C(C3CC3)C=C3C(N4C[C@@H]5C[C@H]4CN5)=NC(OC4CCOCC4)=NC3=C2CCC2=CC=C(C(=O)N3CCN(CC4=CC=C5C(=C4)N(C)C(=O)N5C4CCC(=O)NC4=O)C[C@H]3C)C=C2)C2=C(C=C1F)NN=C2	C57H62FN11O6	KRAS	P01116	CRBN	WO-2024019103-A1
TPD-LW0Z0B	WO2024064316A1_C1	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3CCC(CN4CCC(C5=CC6=C(C=C5)N5C(=NC(=O)C7=C5C=CC=C7Cl)C6(C)C)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C53H64ClN7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064316-A1
TPD-QEPHDY	SCHEMBL30843711	(2S,4R)-1-[(2R)-2-[3-[4-[[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-8-yl)piperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCC(C6=CC=CC7=C6C(C)(C)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C53H61ClN8O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064316-A1
TPD-U9KOYR	SCHEMBL27369596	(2S,4R)-N-[(1S)-6-[4-(4-bromo-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-9-yl)piperidin-1-yl]-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]hexyl]-1-[(2S)-2-[(1-fluorocyclopropanecarbonyl)amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide; SCHEMBL30843560	CC1=C(C2=CC=C([C@H](CCCCCN3CCC(C4=CC5=C(C=C4)N4C(=NC(=O)C6=C4C=CC=C6Br)C5(C)C)CC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3(F)CC3)C(C)(C)C)C=C2)SC=N1	C53H63BrFN7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064316-A1
TPD-ZKZK95	SCHEMBL27369667	(2S,4R)-N-[(1S)-6-[4-(4-bromo-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-9-yl)piperidin-1-yl]-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]hexyl]-1-[(2S)-2-[(1-cyanocyclopropanecarbonyl)amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide; SCHEMBL30843439	CC1=C(C2=CC=C([C@H](CCCCCN3CCC(C4=CC5=C(C=C4)N4C(=NC(=O)C6=C4C=CC=C6Br)C5(C)C)CC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3(C#N)CC3)C(C)(C)C)C=C2)SC=N1	C54H63BrN8O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064316-A1
TPD-BJQAUA	SCHEMBL27369668	(2S,4R)-1-[(2R)-2-[3-[2-[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-9-yl)piperidin-1-yl]ethoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL30843379	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(OCCN4CCC(C5=CC6=C(C=C5)N5C(=NC(=O)C7=C5C=CC=C7Cl)C6(C)C)CC4)=NO3)C(C)C)C=C2)SC=N1	C49H54ClN7O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064316-A1
TPD-X4MHIS	SCHEMBL30843510	(2S,4R)-1-[(2S)-2-[[2-[4-(4-bromo-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-9-yl)piperidin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCC(C4=CC5=C(C=C4)N4C(=NC(=O)C6=C4C=CC=C6Br)C5(C)C)CC3)C(C)(C)C)C=C2)SC=N1	C47H54BrN7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064316-A1
TPD-5F0MN8	SCHEMBL27369670	(2S,4R)-1-[(2S)-2-[[2-[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-9-yl)piperidin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL30843446	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCC(C4=CC5=C(C=C4)N4C(=NC(=O)C6=C4C=CC=C6Cl)C5(C)C)CC3)C(C)(C)C)C=C2)SC=N1	C47H54ClN7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064316-A1
TPD-DBULME	SCHEMBL27369750	(2S,4R)-N-[(1S)-6-[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-9-yl)piperidin-1-yl]-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]hexyl]-1-[(2S)-2-[(1-fluorocyclopropanecarbonyl)amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide; SCHEMBL30843417	CC1=C(C2=CC=C([C@H](CCCCCN3CCC(C4=CC5=C(C=C4)N4C(=NC(=O)C6=C4C=CC=C6Cl)C5(C)C)CC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3(F)CC3)C(C)(C)C)C=C2)SC=N1	C53H63ClFN7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064316-A1
TPD-96DWXE	SCHEMBL30843471	(2S,4R)-1-[2-[3-[[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-9-yl)piperidin-1-yl]methyl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(CN4CCC(C5=CC6=C(C=C5)N5C(=NC(=O)C7=C5C=CC=C7Cl)C6(C)C)CC4)=NO3)C(C)C)C=C2)SC=N1	C48H52ClN7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064316-A1
TPD-Y8VC4C	SCHEMBL30843621	(2S,4R)-1-[(2R)-2-[3-[4-[[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-9-yl)piperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCC(C6=CC7=C(C=C6)N6C(=NC(=O)C8=C6C=CC=C8Cl)C7(C)C)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C53H61ClN8O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064316-A1
TPD-G5XNQ8	WO2024064328A1_A1	.	CC1=C(C2=CC=C([C@H](CCCCN3CCC(C4=CC5=C(C=C4)N4C(=NC(=O)C6=C4C=CC=C6Cl)C54CCCC4)CC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3(F)CC3)C(C)(C)C)C=C2)SCN1	C54H65ClFN7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-P0CZTB	SCHEMBL30843514	(2S,4R)-N-[(1S)-5-[4-(4-chloro-5-oxospiro[indolo[1,2-a]quinazoline-7,4'-oxane]-10-yl)piperidin-1-yl]-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]pentyl]-1-[(2S)-2-[(1-fluorocyclopropanecarbonyl)amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CCCCN3CCC(C4=CC=C5C(=C4)N4C(=NC(=O)C6=C4C=CC=C6Cl)C54CCOCC4)CC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3(F)CC3)C(C)(C)C)C=C2)SC=N1	C54H63ClFN7O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-AQYMUB	SCHEMBL30843595	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4'-chloro-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-2-(oxan-4-yl)acetyl]-4-hydroxy-N-[(1R)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]-2-morpholin-4-ylethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CN3CCOCC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3CCOCC3)N3C=C([C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N3)C=C2)SC=N1	C62H75ClN10O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-3M9J3H	WO2024064328A1_A101	.	CC1=C(C2=CC=C([C@H](CN3CCOCC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3CCOCC3)N3C=C([C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Br)N67)CC5)CC4)N=N3)C=C2)SC=N1	C62H75BrN10O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-DPFGQX	WO2024064328A1_A102	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-10-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-2-(oxan-4-yl)acetyl]-4-hydroxy-N-[(1R)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]-2-morpholin-4-ylethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CN3CCOCC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3CCOCC3)N3C=C([C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)C(C)(C)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N3)C=C2)SC=N1	C59H71ClN10O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-B32QJU	WO2024064328A1_A103	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4'-chloro-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1R)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]-2-morpholin-4-ylethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CN3CCOCC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C([C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N3)C=C2)SC=N1	C60H73ClN10O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-GRBT7W	WO2024064328A1_A104	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-10-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1R)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]-2-morpholin-4-ylethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CN3CCOCC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C([C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)C(C)(C)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N3)C=C2)SC=N1	C57H69ClN10O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-X04ABW	SCHEMBL30843383	(2S,4R)-1-[(2S)-2-[1-[2-[4-(4'-chloro-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]acetyl]piperidin-4-yl]-2-(4-cyclopropyltriazol-1-yl)acetyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3CCN(C(=O)CN4CCC(C5=CC6=C(C=C5)C5(CCCCC5)C5=NC(=O)C7=C(C=CC=C7Cl)N56)CC4)CC3)N3C=C(C4CC4)N=N3)C=C2)SC=N1	C56H63ClN10O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-1NPSSK	SCHEMBL30843413	(2S,4R)-1-[(2S)-2-[1-[4-[4-(4'-chloro-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]butanoyl]piperidin-4-yl]-2-(4-cyclopropyltriazol-1-yl)acetyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3CCN(C(=O)CCCN4CCC(C5=CC6=C(C=C5)C5(CCCCC5)C5=NC(=O)C7=C(C=CC=C7Cl)N56)CC4)CC3)N3C=C(C4CC4)N=N3)C=C2)SC=N1	C58H67ClN10O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-FOLVIC	SCHEMBL30843712	(2S,4R)-1-[(2S)-2-[1-[5-[4-(4'-chloro-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]pentanoyl]piperidin-4-yl]-2-(4-cyclopropyltriazol-1-yl)acetyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3CCN(C(=O)CCCCN4CCC(C5=CC6=C(C=C5)C5(CCCCC5)C5=NC(=O)C7=C(C=CC=C7Cl)N56)CC4)CC3)N3C=C(C4CC4)N=N3)C=C2)SC=N1	C59H69ClN10O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-5N99GX	SCHEMBL30843590	(2S,4R)-1-[(2S)-2-[1-[4-[[4-(4'-chloro-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]cyclohexanecarbonyl]piperidin-4-yl]-2-(4-cyclopropyltriazol-1-yl)acetyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3CCN(C(=O)[C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)CC3)N3C=C(C4CC4)N=N3)C=C2)SC=N1	C62H73ClN10O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-EY9LTF	SCHEMBL30843649	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4'-chloro-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-2-piperidin-4-ylacetyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3CCNCC3)N3C=C(C4CCC(CN5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N3)C=C2)SC=N1	C58H69ClN10O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-DFQJLN	SCHEMBL27395169	(2S,4R)-1-[(2S)-2-[[4-[[4-(4'-chloro-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-9'-yl)piperidin-1-yl]methyl]cyclohexanecarbonyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL30843468	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)[C@H]3CC[C@H](CN4CCC(C5=CC6=C(C=C5)N5C(=NC(=O)C7=C5C=CC=C7Cl)C65CCCCC5)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C56H68ClN7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-HJEZIC	SCHEMBL30843617	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4'-chloro-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-2-(1-methylpiperidin-4-yl)acetyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3CCN(C)CC3)N3C=C([C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N3)C=C2)SC=N1	C59H71ClN10O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-199QXX	WO2024064328A1_A111	.	CC(=O)N1CCC([C@@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=C(C)N=CS3)C=C2)N2C=C([C@H]3CC[C@H](CN4CCC(C5=CC6=C(C=C5)C5(CCCCC5)C5=NC(=O)C7=C(C=CC=C7Cl)N56)CC4)CC3)N=N2)CC1	C60H71ClN10O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-TAKUCF	SCHEMBL30843690	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4'-chloro-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-2-[1-(oxan-4-yl)piperidin-4-yl]acetyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3CCN(C4CCOCC4)CC3)N3C=C([C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N3)C=C2)SC=N1	C63H77ClN10O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-T5ARUR	SCHEMBL30843639	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4'-chloro-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-2-[1-[(2S)-1,4-dioxane-2-carbonyl]piperidin-4-yl]acetyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3CCN(C(=O)[C@@H]4COCCO4)CC3)N3C=C(C4CCC(CN5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N3)C=C2)SC=N1	C63H75ClN10O7S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-MQ0J5I	SCHEMBL30843435	(2S,4R)-N-[(1R)-2-[4-[[4-(4'-bromo-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]triazol-1-yl]-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]-1-[(2S)-2-(4-cyclopropyltriazol-1-yl)-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CN3C=C(CN4CCC(C5=CC6=C(C=C5)C5(CCCCC5)C5=NC(=O)C7=C(C=CC=C7Br)N56)CC4)N=N3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C(C4CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C56H63BrN12O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-OGIW8F	WO2024064328A1_A115	.	CC1=C(C2=CC=C([C@H](CN3C=NC(CN4CCC(C5=CC6=C(C=C5)N5C(=NC(=O)C7=C5C=CC=C7Br)C65CCCCC5)CC4)=C3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C(C4CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C57H64BrN11O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-JEZFXU	SCHEMBL30843519	(2S,4R)-N-[(1R)-2-[[4-[[4-(4'-bromo-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]cyclohexanecarbonyl]amino]-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]-1-[(2S)-2-(4-cyclopropyltriazol-1-yl)-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CNC(=O)[C@H]3CC[C@H](CN4CCC(C5=CC6=C(C=C5)C5(CCCCC5)C5=NC(=O)C7=C(C=CC=C7Br)N56)CC4)CC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C(C4CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C61H73BrN10O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-LGO4C4	SCHEMBL30843483	(2S,4R)-N-[(1R)-2-[[4-[[4-(4'-bromo-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-9'-yl)piperidin-1-yl]methyl]cyclohexanecarbonyl]amino]-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]-1-[(2S)-2-(4-cyclopropyltriazol-1-yl)-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CNC(=O)[C@H]3CC[C@H](CN4CCC(C5=CC6=C(C=C5)N5C(=NC(=O)C7=C5C=CC=C7Br)C65CCCCC5)CC4)CC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C(C4CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C61H73BrN10O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-K5LK8T	WO2024064328A1_A118	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3CCCCC3)N3C=C([C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N3)C=C2)SC=N1	C59H70ClN9O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-HWXUVB	SCHEMBL30843660	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4'-bromo-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-2-cyclohexylacetyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3CCCCC3)N3C=C([C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Br)N67)CC5)CC4)N=N3)C=C2)SC=N1	C59H70BrN9O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-DQ2PB7	SCHEMBL27395244	(2S,4R)-1-[(2S)-2-[[4-[[3-[4-(4'-chloro-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-9'-yl)piperidin-1-yl]azetidin-1-yl]methyl]cyclohexanecarbonyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL30843546	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)[C@H]3CC[C@H](CN4CC(N5CCC(C6=CC7=C(C=C6)N6C(=NC(=O)C8=C6C=CC=C8Cl)C76CCCCC6)CC5)C4)CC3)C(C)(C)C)C=C2)SC=N1	C59H73ClN8O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-13X1B9	SCHEMBL30843402	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4'-chloro-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-2-(oxan-4-yl)acetyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3CCOCC3)N3C=C([C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N3)C=C2)SC=N1	C58H68ClN9O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-G51TWP	SCHEMBL30843725	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4'-bromo-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-2-(oxan-4-yl)acetyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3CCOCC3)N3C=C([C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Br)N67)CC5)CC4)N=N3)C=C2)SC=N1	C58H68BrN9O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-69LPTV	SCHEMBL30843695	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4'-chloro-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-2-cyclohexylacetyl]-4-hydroxy-N-[(1R)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]-2-morpholin-4-ylethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CN3CCOCC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3CCCCC3)N3C=C([C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N3)C=C2)SC=N1	C63H77ClN10O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-924O04	SCHEMBL30843687	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4'-bromo-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-2-cyclohexylacetyl]-4-hydroxy-N-[(1R)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]-2-morpholin-4-ylethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CN3CCOCC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3CCCCC3)N3C=C([C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Br)N67)CC5)CC4)N=N3)C=C2)SC=N1	C63H77BrN10O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-B3TFEK	WO2024064328A1_A124	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3CC=CCC3)N3C=C([C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)C(C)(C)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N3)C=C2)SC=N1	C56H64ClN9O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-SN4STV	SCHEMBL30843702	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-10-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-2-cyclohexylacetyl]-4-hydroxy-N-[(1R)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]-2-morpholin-4-ylethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CN3CCOCC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3CCCCC3)N3C=C([C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)C(C)(C)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N3)C=C2)SC=N1	C60H73ClN10O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-XQGXTZ	SCHEMBL30843566	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4'-chloro-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-2-cyclohexylacetyl]-4-hydroxy-N-[(1R)-2-hydroxy-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CO)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3CCCCC3)N3C=C([C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N3)C=C2)SC=N1	C59H70ClN9O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-WHYLIX	WO2024064328A1_A127	.	CC1=C(C2=CC=C([C@H](CO)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3CCCCC3)N3C=C([C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Br)N67)CC5)CC4)N=N3)C=C2)SC=N1	C59H70BrN9O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-AWNFOP	SCHEMBL30843564	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4'-bromo-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]phenyl]triazol-1-yl]-2-cyclohexylacetyl]-4-hydroxy-N-[(1R)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]-2-morpholin-4-ylethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CN3CCOCC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3CCCCC3)N3C=C(C4=CC=C(CN5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Br)N67)CC5)C=C4)N=N3)C=C2)SC=N1	C63H71BrN10O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-BTM0U8	SCHEMBL30843654	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4'-bromo-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]phenyl]triazol-1-yl]-2-cyclohexylacetyl]-4-hydroxy-N-[(1R)-2-hydroxy-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CO)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3CCCCC3)N3C=C(C4=CC=C(CN5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Br)N67)CC5)C=C4)N=N3)C=C2)SC=N1	C59H64BrN9O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-B2Y44Z	SCHEMBL27395332	(2S,4R)-1-[(2S)-2-[[4-[[4-[4-(4'-chloro-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-9'-yl)piperidin-1-yl]piperidin-1-yl]methyl]cyclohexanecarbonyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL30843643	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)[C@H]3CC[C@H](CN4CCC(N5CCC(C6=CC7=C(C=C6)N6C(=NC(=O)C8=C6C=CC=C8Cl)C76CCCCC6)CC5)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C61H77ClN8O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-92GAVD	SCHEMBL30843641	(2S,4R)-1-[(2S)-2-[4-[4-[[3-(4'-chloro-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)pyrrolidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-2-cyclohexylacetyl]-4-hydroxy-N-[(1R)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]-2-morpholin-4-ylethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CN3CCOCC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3CCCCC3)N3C=C([C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Cl)N67)C5)CC4)N=N3)C=C2)SC=N1	C62H75ClN10O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-QSVK4L	SCHEMBL30843665	(2S,4R)-1-[(2S)-2-[4-[4-[[3-(4'-chloro-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-2-cyclohexylacetyl]-4-hydroxy-N-[(1R)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]-2-morpholin-4-ylethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CN3CCOCC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3CCCCC3)N3C=C([C@H]4CC[C@H](CN5CCCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Cl)N67)C5)CC4)N=N3)C=C2)SC=N1	C63H77ClN10O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-T0HP1D	SCHEMBL30843745	(2S,4R)-1-[(2S)-2-[1-[4-[[4-(4'-bromo-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]cyclohexanecarbonyl]piperidin-4-yl]-2-(4-cyclopropyltriazol-1-yl)acetyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3CCN(C(=O)[C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Br)N67)CC5)CC4)CC3)N3C=C(C4CC4)N=N3)C=C2)SC=N1	C62H73BrN10O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-7UB3BY	WO2024064328A1_A133	.	CC1(C)C2=NC(=O)C3=C(C=CC=C3Cl)N2C2=C1C=CC(C1CCN(C[C@H]3CC[C@H](C4=CN([C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](CN5CCOCC5)C5=CC=C(C6=C(COO)N=CS6)C=C5)C5CCOCC5)N=N4)CC3)CC1)=C2	C59H71ClN10O8S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-DMLSXG	WO2024064328A1_A134	.	O=C1N=C2N(C3=C1C(Cl)=CC=C3)C1=C(C=CC(C3CCN(C[C@H]4CC[C@H](C5=CN([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](CN6CCOCC6)C6=CC=C(C7=C(COO)N=CS7)C=C6)C6CCOCC6)N=N5)CC4)CC3)=C1)C21CCCCC1	C62H75ClN10O8S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-Y14Z4H	SCHEMBL30843411	(2S,4R)-N-[(1R)-2-[4-(4'-bromo-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]-2-oxoethyl]-1-[(2S)-2-(4-cyclopropyltriazol-1-yl)-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@@H](NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C(C4CC4)N=N3)C(C)(C)C)C(=O)N3CCC(C4=CC5=C(C=C4)C4(CCCCC4)C4=NC(=O)C6=C(C=CC=C6Br)N45)CC3)C=C2)SC=N1	C53H58BrN9O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-Z58UKQ	SCHEMBL30843661	(2S,4R)-N-[(1R)-2-[4-[[4-(4'-bromo-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]piperidin-1-yl]-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]-2-oxoethyl]-1-[(2S)-2-(4-cyclopropyltriazol-1-yl)-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@@H](NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C(C4CC4)N=N3)C(C)(C)C)C(=O)N3CCC(CN4CCC(C5=CC6=C(C=C5)C5(CCCCC5)C5=NC(=O)C7=C(C=CC=C7Br)N56)CC4)CC3)C=C2)SC=N1	C59H69BrN10O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-AOZCTD	SCHEMBL30843664	(2S,4R)-N-[(1R)-2-[9-[[4-(4'-bromo-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]-3-azaspiro[5.5]undecan-3-yl]-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]-2-oxoethyl]-1-[(2S)-2-(4-cyclopropyltriazol-1-yl)-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@@H](NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C(C4CC4)N=N3)C(C)(C)C)C(=O)N3CCC4(CCC(CN5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Br)N67)CC5)CC4)CC3)C=C2)SC=N1	C64H77BrN10O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-9AVKXU	SCHEMBL30843692	(2S,4R)-N-[(1R)-2-[4-[4-(4'-bromo-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]piperidin-1-yl]-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]-2-oxoethyl]-1-[(2S)-2-(4-cyclopropyltriazol-1-yl)-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@@H](NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C(C4CC4)N=N3)C(C)(C)C)C(=O)N3CCC(N4CCC(C5=CC6=C(C=C5)C5(CCCCC5)C5=NC(=O)C7=C(C=CC=C7Br)N56)CC4)CC3)C=C2)SC=N1	C58H67BrN10O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-0EPTTT	WO2024064328A1_A139	.	CC1=C(C2=CC=C([C@@H](NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C(C4CC4)N=N3)C(C)(C)C)C(=O)N3CCC4(CCC(N5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Br)N67)CC5)CC4)CC3)C=C2)SC=N1	C63H75BrN10O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-83ZNJX	SCHEMBL30843669	(2S,4R)-1-[(2S)-2-[[4-[[4-(4'-bromo-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-9'-yl)piperidin-1-yl]methyl]cyclohexanecarbonyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)[C@H]3CC[C@H](CN4CCC(C5=CC6=C(C=C5)N5C(=NC(=O)C7=C5C=CC=C7Br)C65CCCCC5)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C56H68BrN7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-GHNSR2	SCHEMBL30843662	(2S,4R)-N-[(1S)-3-[4-(4'-chloro-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]-3-oxopropyl]-1-[(2S)-2-(4-cyclopropyltriazol-1-yl)-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CC(=O)N3CCC(C4=CC5=C(C=C4)C4(CCCCC4)C4=NC(=O)C6=C(C=CC=C6Cl)N45)CC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C(C4CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C54H60ClN9O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-WJDOZG	WO2024064328A1_A141	.	CC1=C(C2=CC=C([C@H](CC(=O)N3CCC(CN4CCC(C5=CC6=C(C=C5)C5(CCCCC5)C5=NC(=O)C7=C(C=CC=C7Br)N56)CC4)CC3)NC(=O)C3C[C@@H](O)CN3C(=O)[C@@H](N3C=C(C4CC4)NN3)C(C)(C)C)C=C2)SC=N1	C60H73BrN10O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-XOC85X	WO2024064328A1_A142	.	CC1=C(C2=CC=C([C@H](CC(=O)N3CCC4(CCC(CN5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Br)N67)CC5)CC4)CC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=NC(C4CC4)=C3)C(C)(C)C)C=C2)SC=N1	C66H80BrN9O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-C4ULOD	WO2024064328A1_A143	(2S,4R)-N-[(1S)-3-[4-[4-(4'-chloro-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]piperidin-1-yl]-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]-3-oxopropyl]-1-[(2S)-2-(4-cyclopropyltriazol-1-yl)-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CC(=O)N3CCC(N4CCC(C5=CC6=C(C=C5)C5(CCCCC5)C5=NC(=O)C7=C(C=CC=C7Cl)N56)CC4)CC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C(C4CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C59H69ClN10O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-F10L8Z	SCHEMBL30843652	(2S,4R)-N-[(1S)-3-[9-[4-(4'-bromo-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]-3-azaspiro[5.5]undecan-3-yl]-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]-3-oxopropyl]-1-[(2S)-2-(4-cyclopropyltriazol-1-yl)-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CC(=O)N3CCC4(CCC(N5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Br)N67)CC5)CC4)CC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C(C4CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C64H77BrN10O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-L30NEH	SCHEMBL30843486	methyl (3S)-3-[[(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4'-chloro-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carbonyl]amino]-3-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]propanoate	COC(=O)C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](N1C=C([C@H]2CC[C@H](CN3CCC(C4=CC5=C(C=C4)C4(CCCCC4)C4=NC(=O)C6=C(C=CC=C6Cl)N45)CC3)CC2)N=N1)C(C)(C)C)C1=CC=C(C2=C(C)N=CS2)C=C1	C59H70ClN9O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-KXBZTQ	SCHEMBL30843733	(3S)-3-[[(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4'-chloro-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carbonyl]amino]-3-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]propanoic acid	CC1=C(C2=CC=C([C@H](CC(=O)O)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C([C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C58H68ClN9O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-MLDMLG	WO2024064328A1_A147	.	CC1=C(C2=CC=C([C@H](CC(=O)N(C)C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C([C@H]4CC[C@H](CN5CCC(C6=CC(N7C=NC(=O)C8=C7C=CC=C8Cl)=C(C7CCCCC7)C=C6)CC5)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C60H75ClN10O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-VJMXV0	SCHEMBL30843716	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4'-chloro-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1R)-2-[2-[2-(2-methoxyethoxy)ethoxy]ethoxy]-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	COCCOCCOCCOC[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](N1C=C([C@H]2CC[C@H](CN3CCC(C4=CC5=C(C=C4)C4(CCCCC4)C4=NC(=O)C6=C(C=CC=C6Cl)N45)CC3)CC2)N=N1)C(C)(C)C)C1=CC=C(C2=C(C)N=CS2)C=C1	C64H82ClN9O8S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-KSN7N6	SCHEMBL30843596	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4'-chloro-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1R)-2-[2-[2-[2-(2-methoxyethoxy)ethoxy]ethoxy]ethoxy]-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	COCCOCCOCCOCCOC[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](N1C=C([C@H]2CC[C@H](CN3CCC(C4=CC5=C(C=C4)C4(CCCCC4)C4=NC(=O)C6=C(C=CC=C6Cl)N45)CC3)CC2)N=N1)C(C)(C)C)C1=CC=C(C2=C(C)N=CS2)C=C1	C66H86ClN9O9S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-JNOC95	SCHEMBL27395483	(2S,4R)-1-[(2S)-2-[[4-[[4-(4'-bromo-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-9'-yl)piperidin-1-yl]methyl]cyclohexanecarbonyl]amino]-3,3-dimethylbutanoyl]-N-[(1R)-2-(dimethylamino)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]-4-hydroxypyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CN(C)C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)[C@H]3CC[C@H](CN4CCC(C5=CC6=C(C=C5)N5C(=NC(=O)C7=C5C=CC=C7Br)C65CCCCC5)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C58H73BrN8O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-C0QHYT	SCHEMBL30843741	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-10-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1R)-2-[2-[2-(2-methoxyethoxy)ethoxy]ethoxy]-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	COCCOCCOCCOC[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](N1C=C([C@H]2CC[C@H](CN3CCC(C4=CC5=C(C=C4)C(C)(C)C4=NC(=O)C6=C(C=CC=C6Cl)N45)CC3)CC2)N=N1)C(C)(C)C)C1=CC=C(C2=C(C)N=CS2)C=C1	C61H78ClN9O8S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-TTNSO2	WO2024064328A1_A151	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-10-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1R)-2-[2-[2-[2-(2-methoxyethoxy)ethoxy]ethoxy]ethoxy]-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	COCCOCCOCCOCCOC[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](N1C=C([C@H]2CC[C@H](CN3CCC(C4=CC5=C(C=C4)C(C)(C)C4=NC(=O)C6=C(C=CC=C6Cl)N45)CC3)CC2)N=N1)C(C)(C)C)C1=CC=C(C2=C(C)N=CS2)C=C1	C63H82ClN9O9S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-1HM5XI	SCHEMBL30843653	methyl 2-[(2R)-2-[[(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4'-chloro-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carbonyl]amino]-2-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethoxy]acetate	COC(=O)COC[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](N1C=C([C@H]2CC[C@H](CN3CCC(C4=CC5=C(C=C4)C4(CCCCC4)C4=NC(=O)C6=C(C=CC=C6Cl)N45)CC3)CC2)N=N1)C(C)(C)C)C1=CC=C(C2=C(C)N=CS2)C=C1	C60H72ClN9O7S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-S3O77P	SCHEMBL30843393	methyl 1-[(2R)-2-[[(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4'-chloro-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carbonyl]amino]-2-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]piperidine-4-carboxylate	COC(=O)C1CCN(C[C@H](NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](N2C=C([C@H]3CC[C@H](CN4CCC(C5=CC6=C(C=C5)C5(CCCCC5)C5=NC(=O)C7=C(C=CC=C7Cl)N56)CC4)CC3)N=N2)C(C)(C)C)C2=CC=C(C3=C(C)N=CS3)C=C2)CC1	C64H79ClN10O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-BK5F21	SCHEMBL30843619	methyl 1-[(2R)-2-[[(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4'-chloro-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carbonyl]amino]-2-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]azetidine-3-carboxylate	COC(=O)C1CN(C[C@H](NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](N2C=C([C@H]3CC[C@H](CN4CCC(C5=CC6=C(C=C5)C5(CCCCC5)C5=NC(=O)C7=C(C=CC=C7Cl)N56)CC4)CC3)N=N2)C(C)(C)C)C2=CC=C(C3=C(C)N=CS3)C=C2)C1	C62H75ClN10O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-LBHREN	SCHEMBL30843606	2-[(2R)-2-[[(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4'-chloro-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carbonyl]amino]-2-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethoxy]acetic acid	CC1=C(C2=CC=C([C@H](COCC(=O)O)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C([C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C59H70ClN9O7S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-SF2QU3	SCHEMBL30843650	1-[(2R)-2-[[(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4'-chloro-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carbonyl]amino]-2-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]piperidine-4-carboxylic acid	CC1=C(C2=CC=C([C@H](CN3CCC(C(=O)O)CC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C([C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C63H77ClN10O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-SINAQX	SCHEMBL30843706	1-[(2R)-2-[[(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4'-chloro-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carbonyl]amino]-2-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]azetidine-3-carboxylic acid	CC1=C(C2=CC=C([C@H](CN3CC(C(=O)O)C3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C([C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C61H73ClN10O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-PUP3I3	WO2024064328A1_A158	.	CC1=C(C2=CC=C([C@H](CN3CCOCC3)NC(=O)[C@@H]3CC(=O)CN3C(=O)[C@@H](N3C=C([C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N3)C(C)(C)O)C=C2)SC=N1	C60H71ClN10O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-7EW0MT	WO2024064328A1_A159	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-10-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3-hydroxy-3-methylbutanoyl]-4-hydroxy-N-[(1R)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]-2-morpholin-4-ylethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CN3CCOCC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C(C4CCC(CN5CCC(C6=CC7=C(C=C6)C(C)(C)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N3)C(C)(C)O)C=C2)SC=N1	C57H69ClN10O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-N99X39	SCHEMBL30843424	(2S,4R)-1-[(2S)-2-[[4-[[4-(4'-bromo-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-9'-yl)piperidin-1-yl]methyl]cyclohexanecarbonyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1R)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]-2-morpholin-4-ylethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CN3CCOCC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)[C@H]3CC[C@H](CN4CCC(C5=CC6=C(C=C5)N5C(=NC(=O)C7=C5C=CC=C7Br)C65CCCCC5)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C60H75BrN8O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-3QFL18	WO2024064328A1_A160	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4'-bromo-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3-hydroxy-3-methylbutanoyl]-4-hydroxy-N-[(1R)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]-2-morpholin-4-ylethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CN3CCOCC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C([C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Br)N67)CC5)CC4)N=N3)C(C)(C)O)C=C2)SC=N1	C60H73BrN10O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-8UCNMX	SCHEMBL30843389	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4'-chloro-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3,3-dimethylbutanoyl]-N-[(1R)-1-[4-(2,4-dimethyl-1,3-thiazol-5-yl)phenyl]-2-morpholin-4-ylethyl]-4-hydroxypyrrolidine-2-carboxamide	CC1=NC(C)=C(C2=CC=C([C@H](CN3CCOCC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C([C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N3)C(C)(C)C)C=C2)S1	C62H77ClN10O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-VEO449	SCHEMBL30843700	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4'-chloro-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1R)-2-morpholin-4-yl-1-(4-phenylphenyl)ethyl]pyrrolidine-2-carboxamide	CC(C)(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](CN1CCOCC1)C1=CC=C(C2=CC=CC=C2)C=C1)N1C=C([C@H]2CC[C@H](CN3CCC(C4=CC5=C(C=C4)C4(CCCCC4)C4=NC(=O)C6=C(C=CC=C6Cl)N45)CC3)CC2)N=N1	C63H76ClN9O5	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-V5A157	WO2024064328A1_A163	.	CC1=CC=CC=C1C1=CC=C2C(=C1)C1COCCN1C[C@@H]2NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](N1C=C([C@H]2CC[C@H](CN3CCC(C4=CC5=C(C=C4)C4(CCCCC4)C4=NC(=O)C6=C(C=CC=C6Cl)N45)CC3)CC2)N=N1)C(C)(C)C	C64H76ClN9O5	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-8TDOBL	WO2024064328A1_A164	.	CC(C)(C)[C@@H](C(=O)N1C[C@H](O)CC1C(=O)N[C@@H](CN1CCOCC1)C1=CC=C(C2=CC=CC=C2F)C=C1)N1C=C([C@H]2CC[C@H](CN3CCC(C4=CC5=C(C=C4)C4(CCCCC4)C4=NC(=O)C6=C(C=CC=C6Cl)N45)CC3)CC2)N=N1	C63H75ClFN9O5	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-DZJUAV	SCHEMBL30843705	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4'-chloro-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1R)-1-[4-(4-methyl-1,3-oxazol-5-yl)phenyl]-2-morpholin-4-ylethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CN3CCOCC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C([C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N3)C(C)(C)C)C=C2)OC=N1	C61H75ClN10O6	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-EXFS0Q	SCHEMBL30843647	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4'-chloro-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3,3-dimethylbutanoyl]-N-[(1R)-1-[4-(2,4-dimethyl-1,3-oxazol-5-yl)phenyl]-2-morpholin-4-ylethyl]-4-hydroxypyrrolidine-2-carboxamide	CC1=NC(C)=C(C2=CC=C([C@H](CN3CCOCC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C([C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N3)C(C)(C)C)C=C2)O1	C62H77ClN10O6	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-FK8CE7	WO2024064328A1_A167	.	CC(C)(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](CN1CCOCC1)C1=CC=C(C2=C(C(F)(F)F)N=CS2)C=C1)N1C=C([C@H]2CC[C@H](CN3CCC(C4=CC5=C(C=C4)C4(CCCCC4)C4=NC(=O)C6=C(C=CC=C6Cl)N45)CC3)CC2)N=N1	C61H72ClF3N10O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-NIBG2T	WO2024064328A1_A168	.	CC1=C(C2=CC=C([C@H](CN3CCOCC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C(C4CCN(CC5CCN(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C60H74ClN11O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-MCXL31	SCHEMBL30843522	(2S,4R)-1-[(2S)-2-[4-[1-[[1-(4'-bromo-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-4-yl]methyl]piperidin-4-yl]triazol-1-yl]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1R)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]-2-morpholin-4-ylethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CN3CCOCC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C(C4CCN(CC5CCN(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Br)N67)CC5)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C60H74BrN11O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-RG3KKR	SCHEMBL30843530	(2S,4R)-N-[(1S)-6-[4-(4'-bromo-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-9'-yl)piperidin-1-yl]-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]hexyl]-1-[(2S)-2-[[1-(dimethylamino)cyclopropanecarbonyl]amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CCCCCN3CCC(C4=CC5=C(C=C4)N4C(=NC(=O)C6=C4C=CC=C6Br)C54CCCCC4)CC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3(N(C)C)CC3)C(C)(C)C)C=C2)SC=N1	C58H73BrN8O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-BHG38J	SCHEMBL30843676	(2S,4R)-1-[(2S)-3,3-dimethyl-2-[4-[4-[[4-(5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]butanoyl]-4-hydroxy-N-[(1R)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]-2-morpholin-4-ylethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CN3CCOCC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C(C4CCC(CN5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8)N67)CC5)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C61H76N10O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-AZYNM2	SCHEMBL30843717	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4'-chloro-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1R)-2-morpholin-4-yl-1-(4-pyridin-3-ylphenyl)ethyl]pyrrolidine-2-carboxamide	CC(C)(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](CN1CCOCC1)C1=CC=C(C2=CC=CN=C2)C=C1)N1C=C([C@H]2CC[C@H](CN3CCC(C4=CC5=C(C=C4)C4(CCCCC4)C4=NC(=O)C6=C(C=CC=C6Cl)N45)CC3)CC2)N=N1	C62H75ClN10O5	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-S1UTQI	SCHEMBL30843666	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4'-chloro-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1R)-2-morpholin-4-yl-1-(4-pyridin-4-ylphenyl)ethyl]pyrrolidine-2-carboxamide	CC(C)(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](CN1CCOCC1)C1=CC=C(C2=CC=NC=C2)C=C1)N1C=C([C@H]2CC[C@H](CN3CCC(C4=CC5=C(C=C4)C4(CCCCC4)C4=NC(=O)C6=C(C=CC=C6Cl)N45)CC3)CC2)N=N1	C62H75ClN10O5	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-W0AIOZ	SCHEMBL30843452	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4'-chloro-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1R)-2-morpholin-4-yl-1-(4-pyridin-2-ylphenyl)ethyl]pyrrolidine-2-carboxamide	CC(C)(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](CN1CCOCC1)C1=CC=C(C2=CC=CC=N2)C=C1)N1C=C([C@H]2CC[C@H](CN3CCC(C4=CC5=C(C=C4)C4(CCCCC4)C4=NC(=O)C6=C(C=CC=C6Cl)N45)CC3)CC2)N=N1	C62H75ClN10O5	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-F7HJVH	SCHEMBL30843569	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4'-chloro-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1R)-1-[4-(2-methylpyridin-3-yl)phenyl]-2-morpholin-4-ylethyl]pyrrolidine-2-carboxamide	CC1=NC=CC=C1C1=CC=C([C@H](CN2CCOCC2)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](N2C=C([C@H]3CC[C@H](CN4CCC(C5=CC6=C(C=C5)C5(CCCCC5)C5=NC(=O)C7=C(C=CC=C7Cl)N56)CC4)CC3)N=N2)C(C)(C)C)C=C1	C63H77ClN10O5	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-SSJV5C	SCHEMBL30843382	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4'-chloro-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1R)-1-[4-(4-methylpyridin-3-yl)phenyl]-2-morpholin-4-ylethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CN3CCOCC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C([C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N3)C(C)(C)C)C=C2)C=NC=C1	C63H77ClN10O5	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-PZIW4W	WO2024064328A1_A18	(2S,4R)-N-[(1S)-6-[4-(4'-bromo-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-9'-yl)piperidin-1-yl]-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]hexyl]-1-[(2S)-2-[[1-[(dimethylamino)methyl]cyclopropanecarbonyl]amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CCCCCN3CCC(C4=CC5=C(C=C4)N4C(=NC(=O)C6=C4C=CC=C6Br)C54CCCCC4)CC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3(CN(C)C)CC3)C(C)(C)C)C=C2)SC=N1	C59H75BrN8O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-ZWEMUJ	WO2024064328A1_A19	(2S,4R)-1-[(2S)-2-[[4-[[4-(4'-bromo-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-9'-yl)piperidin-1-yl]methyl]bicyclo[2.2.1]heptane-1-carbonyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)[C@]34CC[C@@](CN5CCC(C6=CC7=C(C=C6)N6C(=NC(=O)C8=C6C=CC=C8Br)C76CCCCC6)CC5)(CC3)C4)C(C)(C)C)C=C2)SC=N1	C57H68BrN7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-EFY8S0	SCHEMBL27394630	(2S,4R)-N-[(1S)-6-[4-(4'-chloro-5'-oxospiro[cyclopentane-1,7'-indolo[1,2-a]quinazoline]-9'-yl)piperidin-1-yl]-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]hexyl]-1-[(2S)-2-[(1-fluorocyclopropanecarbonyl)amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide; SCHEMBL30843616	CC1=C(C2=CC=C([C@H](CCCCCN3CCC(C4=CC5=C(C=C4)N4C(=NC(=O)C6=C4C=CC=C6Cl)C54CCCC4)CC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3(F)CC3)C(C)(C)C)C=C2)SC=N1	C55H65ClFN7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-O5RN4O	SCHEMBL30843507	(2S,4R)-1-[(2S)-2-[[3-[[4-(4'-bromo-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-9'-yl)piperidin-1-yl]methyl]cyclobutanecarbonyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3CC(CN4CCC(C5=CC6=C(C=C5)N5C(=NC(=O)C7=C5C=CC=C7Br)C65CCCCC5)CC4)C3)C(C)(C)C)C=C2)SC=N1	C54H64BrN7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-O3HB26	SCHEMBL30843410	(2S,4R)-1-[(2S)-2-[[3-[[4-(4'-bromo-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-9'-yl)piperidin-1-yl]methyl]cyclobutanecarbonyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1R)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]-2-morpholin-4-ylethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CN3CCOCC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3CC(CN4CCC(C5=CC6=C(C=C5)N5C(=NC(=O)C7=C5C=CC=C7Br)C65CCCCC5)CC4)C3)C(C)(C)C)C=C2)SC=N1	C58H71BrN8O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-MIP256	WO2024064328A1_A22	(2S,4R)-1-[(2S)-2-[[4-[[4-(4'-bromo-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-9'-yl)piperidin-1-yl]methyl]bicyclo[2.2.1]heptane-1-carbonyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1R)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]-2-morpholin-4-ylethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CN3CCOCC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C34CCC(CN5CCC(C6=CC7=C(C=C6)N6C(=NC(=O)C8=C6C=CC=C8Br)C76CCCCC6)CC5)(CC3)C4)C(C)(C)C)C=C2)SC=N1	C61H75BrN8O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-H99XA7	SCHEMBL30843458	(2S,4R)-1-[(2S)-2-[[4-[[4-(4'-bromo-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]bicyclo[2.2.1]heptane-1-carbonyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C34CCC(CN5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Br)N67)CC5)(CC3)C4)C(C)(C)C)C=C2)SC=N1	C57H68BrN7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-9EYBL3	WO2024064328A1_A24	(2S,4R)-1-[(2S)-2-[[4-[[4-(4'-bromo-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]bicyclo[2.2.1]heptane-1-carbonyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1R)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]-2-morpholin-4-ylethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CN3CCOCC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C34CCC(CN5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Br)N67)CC5)(CC3)C4)C(C)(C)C)C=C2)SC=N1	C61H75BrN8O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-JX5WDT	SCHEMBL30843691	(2S,4R)-N-[(1S)-6-[4-(4'-bromo-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-9'-yl)piperidin-1-yl]-1-(4-chlorophenyl)hexyl]-1-[(2S)-2-[(1-fluorocyclopropanecarbonyl)amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide	CC(C)(C)[C@H](NC(=O)C1(F)CC1)C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](CCCCCN1CCC(C2=CC3=C(C=C2)N2C(=NC(=O)C4=C2C=CC=C4Br)C32CCCCC2)CC1)C1=CC=C(Cl)C=C1	C52H63BrClFN6O5	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-EXN24A	SCHEMBL30843495	(2S,4R)-N-[(1S)-6-[4-(4'-bromo-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]-1-(4-chlorophenyl)hexyl]-1-[(2S)-2-[(1-fluorocyclopropanecarbonyl)amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide	CC(C)(C)[C@H](NC(=O)C1(F)CC1)C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](CCCCCN1CCC(C2=CC3=C(C=C2)C2(CCCCC2)C2=NC(=O)C4=C(C=CC=C4Br)N23)CC1)C1=CC=C(Cl)C=C1	C52H63BrClFN6O5	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-HZRJO6	SCHEMBL30843673	(2S,4R)-1-[(2S)-2-[[4-[[4-(4'-bromo-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-9'-yl)piperidin-1-yl]methyl]bicyclo[2.2.2]octane-1-carbonyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C34CCC(CN5CCC(C6=CC7=C(C=C6)N6C(=NC(=O)C8=C6C=CC=C8Br)C76CCCCC6)CC5)(CC3)CC4)C(C)(C)C)C=C2)SC=N1	C58H70BrN7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-2OLST6	SCHEMBL30843659	(2S,4R)-1-[(2S)-2-[[4-[[4-(4'-bromo-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-9'-yl)piperidin-1-yl]methyl]bicyclo[2.2.2]octane-1-carbonyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1R)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]-2-morpholin-4-ylethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CN3CCOCC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C34CCC(CN5CCC(C6=CC7=C(C=C6)N6C(=NC(=O)C8=C6C=CC=C8Br)C76CCCCC6)CC5)(CC3)CC4)C(C)(C)C)C=C2)SC=N1	C62H77BrN8O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-LKA1WI	SCHEMBL30843722	(2S,4R)-1-[(2S)-2-[[4-[[4-(4'-bromo-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]bicyclo[2.2.2]octane-1-carbonyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C34CCC(CN5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Br)N67)CC5)(CC3)CC4)C(C)(C)C)C=C2)SC=N1	C58H70BrN7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-701UEY	SCHEMBL30843504	(2S,4R)-N-[(1S)-6-[4-(4'-chloro-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-9'-yl)piperidin-1-yl]-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]hexyl]-1-[(2S)-2-[(1-fluorocyclopropanecarbonyl)amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CCCCCN3CCC(C4=CC5=C(C=C4)N4C(=NC(=O)C6=C4C=CC=C6Cl)C54CCCCC4)CC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3(F)CC3)C(C)(C)C)C=C2)SC=N1	C56H67ClFN7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-DCC1D8	SCHEMBL30843488	(2S,4R)-1-[(2S)-2-[[4-[[4-(4'-bromo-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]bicyclo[2.2.2]octane-1-carbonyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1R)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]-2-morpholin-4-ylethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CN3CCOCC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C34CCC(CN5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Br)N67)CC5)(CC3)CC4)C(C)(C)C)C=C2)SC=N1	C62H77BrN8O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-IDU95V	WO2024064328A1_A31	.	CC1=C(C2=CC=C([C@H](C)NC(=O)C3C[C@@H](O)CN3C(=O)[C@@H](N3C=C([C@H]4CC[C@H](CN5CCC(C6=NC7=C(C=N6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Br)N67)CC5)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C55H66BrN11O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-ZYOBXB	SCHEMBL30843727	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(6-bromo-8-oxospiro[1,9,14,16-tetrazatetracyclo[8.7.0.02,7.012,17]heptadeca-2(7),3,5,9,12,14,16-heptaene-11,1'-cyclohexane]-15-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1R)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]-2-morpholin-4-ylethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CN3CCOCC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C([C@H]4CC[C@H](CN5CCC(C6=NC7=C(C=N6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Br)N67)CC5)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C59H73BrN12O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-924GZK	SCHEMBL30843718	(2S,4R)-N-[(1R)-2-[4-[4-[[4-(4'-bromo-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-9'-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]-1-[(2S)-2-[(1-fluorocyclopropanecarbonyl)amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CN3C=C([C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)N6C(=NC(=O)C8=C6C=CC=C8Br)C76CCCCC6)CC5)CC4)N=N3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3(F)CC3)C(C)(C)C)C=C2)SC=N1	C61H72BrFN10O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-NUJ7D7	WO2024064328A1_A34	(2S,4R)-N-[(1R)-2-[4-[4-[[4-(6-bromo-8-oxospiro[1,9,16-triazatetracyclo[8.7.0.02,7.012,17]heptadeca-2(7),3,5,9,12(17),13,15-heptaene-11,1'-cyclohexane]-15-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]-1-[(2S)-2-[(1-fluorocyclopropanecarbonyl)amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CN3C=C([C@H]4CC[C@H](CN5CCC(C6=NC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Br)N67)CC5)CC4)N=N3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3(F)CC3)C(C)(C)C)C=C2)SC=N1	C60H71BrFN11O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-2BYGLT	SCHEMBL30843474	(2R,4S)-N-[(1S)-6-[4-(4'-bromo-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-9'-yl)piperidin-1-yl]-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]hexyl]-1-[(2S)-2-(4-cyclopropyltriazol-1-yl)-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CCCCCN3CCC(C4=CC5=C(C=C4)N4C(=NC(=O)C6=C4C=CC=C6Br)C54CCCCC4)CC3)NC(=O)[C@H]3C[C@H](O)CN3C(=O)[C@@H](N3C=C(C4CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C57H68BrN9O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-X5S20P	WO2024064328A1_A36	.	CC1=C(C2=CC=C([C@H](CCCCCN3C=CC(C4=CC5=C(C=C4)C4(CCCCC4)C4=NC(=O)C6=C(C=CC=C6Br)N45)CC3)NC(=O)[C@H]3C[C@H](O)CN3C(=O)[C@@H](N3C=C(C4CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C57H66BrN9O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-IW09VR	SCHEMBL30843545	(2R,4S)-N-[(1S)-6-[4-(6-bromo-8-oxospiro[1,9,16-triazatetracyclo[8.7.0.02,7.012,17]heptadeca-2(7),3,5,9,12(17),13,15-heptaene-11,1'-cyclohexane]-15-yl)piperidin-1-yl]-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]hexyl]-1-[(2S)-2-(4-cyclopropyltriazol-1-yl)-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CCCCCN3CCC(C4=NC5=C(C=C4)C4(CCCCC4)C4=NC(=O)C6=C(C=CC=C6Br)N45)CC3)NC(=O)[C@H]3C[C@H](O)CN3C(=O)[C@@H](N3C=C(C4CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C56H67BrN10O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-RMKPWK	SCHEMBL30843568	(2R,4S)-N-[(1S)-6-[4-(4'-bromo-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-9'-yl)piperidin-1-yl]-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]hexyl]-1-[(2S)-3,3-dimethyl-2-[[1-(morpholin-4-ylmethyl)cyclopropanecarbonyl]amino]butanoyl]-4-hydroxypyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CCCCCN3CCC(C4=CC5=C(C=C4)N4C(=NC(=O)C6=C4C=CC=C6Br)C54CCCCC4)CC3)NC(=O)[C@H]3C[C@H](O)CN3C(=O)[C@@H](NC(=O)C3(CN4CCOCC4)CC3)C(C)(C)C)C=C2)SC=N1	C61H77BrN8O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-A8LQOP	WO2024064328A1_A39	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCC(C4=CC5=C(C=C4)C4(CC=CCC4)C4=NC(=O)C6=C(C=CC=C6Cl)N45)CC3)C(C)(C)C)C=C2)SC=N1	C50H56ClN7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-MKQW67	SCHEMBL30843449	(2S,4R)-N-[(1S)-6-[4-(4'-bromo-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-9'-yl)piperidin-1-yl]-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]hexyl]-1-[(2S)-2-[(1-fluorocyclopropanecarbonyl)amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CCCCCN3CCC(C4=CC5=C(C=C4)N4C(=NC(=O)C6=C4C=CC=C6Br)C54CCCCC4)CC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3(F)CC3)C(C)(C)C)C=C2)SC=N1	C56H67BrFN7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-MW8AVJ	WO2024064328A1_A40	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCC(C4=CC5=C(C=C4)C4(CC=CCC4)C4=NC(=O)C6=C(C=CC=C6Br)N45)CC3)C(C)(C)C)C=C2)SC=N1	C50H56BrN7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-D7C2RG	WO2024064328A1_A41	.	CC1=C(C2=CC=C([C@H](C)NC(=O)C3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)[C@H]3CC[C@H](CN4CCC(C5=CC6=C(C=C5)C5(CCCCC5)C5=NC(=O)C7=C(C=CC=C7Br)N56)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C56H68BrN7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-D9IXKL	orb2944974	(2S,4R)-1-[(2S)-2-[[4-[[4-(4'-chloro-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]cyclohexanecarbonyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL30843448; 3033586-04-5	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)[C@H]3CC[C@H](CN4CCC(C5=CC6=C(C=C5)C5(CCCCC5)C5=NC(=O)C7=C(C=CC=C7Cl)N56)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C56H68ClN7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-3QNN5I	SCHEMBL30843736	(2S,4R)-1-[(2S)-2-[4-[[4-(4'-bromo-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]triazol-1-yl]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C(CN4CCC(C5=CC6=C(C=C5)C5(CCCCC5)C5=NC(=O)C7=C(C=CC=C7Br)N56)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C51H58BrN9O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-4SHKHX	SCHEMBL30843598	(2S,4R)-1-[(2S)-2-[4-[3-[4-(4'-bromo-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]propyl]triazol-1-yl]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C(CCCN4CCC(C5=CC6=C(C=C5)C5(CCCCC5)C5=NC(=O)C7=C(C=CC=C7Br)N56)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C53H62BrN9O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-BUKQB1	SCHEMBL30843631	(2S,4R)-1-[(2S)-2-[4-[4-[4-(4'-bromo-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]butyl]triazol-1-yl]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C(CCCCN4CCC(C5=CC6=C(C=C5)C5(CCCCC5)C5=NC(=O)C7=C(C=CC=C7Br)N56)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C54H64BrN9O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-9QG9WO	WO2024064328A1_A46	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C(CCCCCN4CCC(C5=CC6=C(C=C5)C5(CCCCC5)C5NC(=O)C7=C(C=CC=C7Br)N65)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C55H68BrN9O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-B9QD8O	SCHEMBL30843703	(2S,4R)-1-[(2S)-2-[4-[6-[4-(4'-bromo-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]hexyl]triazol-1-yl]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C(CCCCCCN4CCC(C5=CC6=C(C=C5)C5(CCCCC5)C5=NC(=O)C7=C(C=CC=C7Br)N56)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C56H68BrN9O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-922X24	SCHEMBL30843683	(2S,4R)-1-[(2S)-2-[4-[2-[4-(4'-bromo-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]ethyl]triazol-1-yl]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C(CCN4CCC(C5=CC6=C(C=C5)C5(CCCCC5)C5=NC(=O)C7=C(C=CC=C7Br)N56)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C52H60BrN9O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-N6E9II	WO2024064328A1_A49	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4'-chloro-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C([C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C57H68ClN9O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-ORLE1X	WO2024064328A1_A5	(2S,4R)-1-[(2S)-2-[[2-[4-(4'-chloro-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-9'-yl)piperidin-1-yl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCC(C4=CC5=C(C=C4)N4C(=NC(=O)C6=C4C=CC=C6Cl)C54CCCCC4)CC3)C(C)(C)C)C=C2)SC=N1	C50H58ClN7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-MB0OI8	WO2024064328A1_A50	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C([C@H]4CC[C@H](CN5C=CC(C6=NC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Br)N67)CC5)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C56H65BrN10O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-EQFNF5	WO2024064328A1_A51	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3CCC(CN4CCC(C5=NC6=C(C=C5)C5(CCCCC5)C5=NC(=O)C7=C(C=CC=C7Br)N56)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C55H67BrN8O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-U5HWOF	SCHEMBL30843623	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(6-bromo-8-oxospiro[1,9,16-triazatetracyclo[8.7.0.02,7.012,17]heptadeca-2(7),3,5,9,12(17),13,15-heptaene-11,1'-cyclohexane]-15-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1R)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]-2-morpholin-4-ylethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CN3CCOCC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C([C@H]4CC[C@H](CN5CCC(C6=NC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Br)N67)CC5)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C60H74BrN11O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-ZUD3YD	WO2024064328A1_A53	.	CC1=C(C2=CC=C([C@H](C)NC(=O)C3C[C@@H](O)CN3C(=O)[C@@H](N3C=C(CN4CCC(C5=CC6=C(C=C5)N5C(=NC(=O)C7=C5C=CC=C7Br)C65CCCCC5)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C51H58BrN9O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-5C3FAO	WO2024064328A1_A54	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C(CCN4CCC(C5=CC6=C(C=C5)N5C(=NC(=O)C7=C5C=CC=C7Br)C65CC=CCC5)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C52H58BrN9O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-80LT5E	SCHEMBL30843516	(2S,4R)-1-[(2S)-2-[4-[3-[4-(4'-bromo-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-9'-yl)piperidin-1-yl]propyl]triazol-1-yl]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C(CCCN4CCC(C5=CC6=C(C=C5)N5C(=NC(=O)C7=C5C=CC=C7Br)C65CCCCC5)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C53H62BrN9O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-QCWX0T	SCHEMBL30843421	(2S,4R)-1-[(2S)-2-[4-[4-[4-(4'-bromo-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-9'-yl)piperidin-1-yl]butyl]triazol-1-yl]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C(CCCCN4CCC(C5=CC6=C(C=C5)N5C(=NC(=O)C7=C5C=CC=C7Br)C65CCCCC5)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C54H64BrN9O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-0XRLKD	SCHEMBL30843738	(2S,4R)-1-[(2S)-2-[4-[5-[4-(4'-bromo-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-9'-yl)piperidin-1-yl]pentyl]triazol-1-yl]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C(CCCCCN4CCC(C5=CC6=C(C=C5)N5C(=NC(=O)C7=C5C=CC=C7Br)C65CCCCC5)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C55H66BrN9O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-VL2F5U	WO2024064328A1_A58	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C(CCCCCCN4CCC(C5=CC6=C(C=C5)N5C(=NC(=O)C7=C5C=CC=C7Br)C65CC=CCC5)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C56H66BrN9O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-BZPHPB	SCHEMBL30843607	(2S,4R)-1-[2-[3-[4-[[4-(4'-bromo-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-9'-yl)piperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1R)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCC(CN5CCC(C6=CC7=C(C=C6)N6C(=NC(=O)C8=C6C=CC=C8Br)C76CCCCC6)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C56H65BrN8O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-QIM3T2	SCHEMBL27394848	(2S,4R)-1-[(2S)-2-[3-[4-(4'-chloro-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-9'-yl)piperidin-1-yl]propanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL30843571	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCN3CCC(C4=CC5=C(C=C4)N4C(=NC(=O)C6=C4C=CC=C6Cl)C54CCCCC4)CC3)C(C)(C)C)C=C2)SC=N1	C51H60ClN7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-9M9VI1	SCHEMBL30843541	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4'-bromo-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-9'-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C([C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)N6C(=NC(=O)C8=C6C=CC=C8Br)C76CCCCC6)CC5)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C57H68BrN9O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-7P48SB	WO2024064328A1_A61	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CC3C(=O)[C@@H](N3C=C([C@H]4C[C@H](CN5CCC(C6=CC7=C(C=C6)N6C(=NC(=O)C8=C6C=CC=C8Br)C76CCCCC6)CC5)C4)N=N3)C(C)(C)C)C=C2)SC=N1	C56H65BrN8O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-7C4SR7	SCHEMBL30843701	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4'-bromo-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C([C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Br)N67)CC5)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C57H68BrN9O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-N4T6TB	SCHEMBL30843608	(2S,4R)-1-[(2S)-2-[4-[3-[[4-(4'-bromo-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]cyclobutyl]triazol-1-yl]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C([C@H]4C[C@H](CN5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Br)N67)CC5)C4)N=N3)C(C)(C)C)C=C2)SC=N1	C55H64BrN9O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-M9N7BW	SCHEMBL30843704	(2S,4R)-1-[(2S)-2-[4-[1-[[4-(4'-bromo-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]cyclopropyl]triazol-1-yl]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C(C4(CN5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Br)N67)CC5)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C54H62BrN9O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-ESE190	SCHEMBL30843724	(2S,4R)-1-[(2S)-2-[4-[1-[2-[4-(4'-bromo-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]ethyl]cyclopropyl]triazol-1-yl]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C(C4(CCN5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Br)N67)CC5)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C55H64BrN9O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-8ZYALX	WO2024064328A1_A66	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C(C4=CN=C(CN5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Br)N67)CC5)C=C4)N=N3)C(C)(C)C)C=C2)SC=N1	C56H61BrN10O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-JNLFVS	WO2024064328A1_A67	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C([C@H]4CC[C@H](NN5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Br)N67)CC5)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C55H65BrN10O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-GRXSHM	SCHEMBL30843461	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4'-bromo-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3,3-dimethylbutanoyl]-N-[(1S)-1-(4-chlorophenyl)ethyl]-4-hydroxypyrrolidine-2-carboxamide	C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](N1C=C([C@H]2CC[C@H](CN3CCC(C4=CC5=C(C=C4)C4(CCCCC4)C4=NC(=O)C6=C(C=CC=C6Br)N45)CC3)CC2)N=N1)C(C)(C)C)C1=CC=C(Cl)C=C1	C53H64BrClN8O4	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-R8K8HC	SCHEMBL30843633	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4'-bromo-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1R)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]-2-morpholin-4-ylethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CN3CCOCC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C([C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Br)N67)CC5)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C61H75BrN10O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-R0IAUC	SCHEMBL30843640	(2S,4R)-1-[(2S)-2-[4-[4-(4'-chloro-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-9'-yl)piperidin-1-yl]butanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCN3CCC(C4=CC5=C(C=C4)N4C(=NC(=O)C6=C4C=CC=C6Cl)C54CCCCC4)CC3)C(C)(C)C)C=C2)SC=N1	C52H62ClN7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-96AKYH	orb2944727	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4'-chloro-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1R)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]-2-morpholin-4-ylethyl]pyrrolidine-2-carboxamide; SCHEMBL30843614; 3033586-31-8	CC1=C(C2=CC=C([C@H](CN3CCOCC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C([C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C61H75ClN10O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-MQATSM	SCHEMBL30843743	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4'-chloro-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1R)-2-(3-hydroxy-3-methylazetidin-1-yl)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CN3CC(C)(O)C3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C([C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C61H75ClN10O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-1J5UQ9	SCHEMBL30843630	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4'-chloro-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3,3-dimethylbutanoyl]-N-[(1R)-2-(1,1-dioxo-1,4-thiazinan-4-yl)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]-4-hydroxypyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CN3CCS(=O)(=O)CC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C([C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C61H75ClN10O6S2	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-X6GT52	SCHEMBL30843465	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4'-chloro-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1R)-2-(4-hydroxypiperidin-1-yl)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CN3CCC(O)CC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C([C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C62H77ClN10O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-GEKNBP	SCHEMBL30843746	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4'-chloro-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3,3-dimethylbutanoyl]-N-[(1R)-2-(3-fluoro-3-methylazetidin-1-yl)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]-4-hydroxypyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CN3CC(C)(F)C3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C([C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C61H74ClFN10O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-NBSWP6	WO2024064328A1_A75	.	C=N/C(=C\N(N)[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](CN1CCC(F)(F)CC1)C1=CC=C(C2=C(C)N=CS2)C=C1)C(C)(C)C)[C@H]1CC[C@H](CN2CCC(C3=CC4=C(C=C3)C3(CCCCC3)C3=NC(=O)C5=C(C=CC=C5Cl)N34)CC2)CC1	C63H79ClF2N10O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-F3WR9N	SCHEMBL30843726	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(6-bromo-8-oxospiro[1,9,13-triazatetracyclo[8.7.0.02,7.012,17]heptadeca-2(7),3,5,9,12(17),13,15-heptaene-11,1'-cyclohexane]-15-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C([C@H]4CC[C@H](CN5CCC(C6=CC7=C(N=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Br)N67)CC5)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C56H67BrN10O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-5NA8ZS	WO2024064328A1_A77	.	CC1=C(C2=CC=C([C@H](CN3CCOCC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C(C4CCC(NN5CCC(C6=NC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C59H73ClN12O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-3PIT2D	WO2024064328A1_A78	.	C=N/C(=C\N(N)[C@H](C(=O)N1C[C@H](O)CC1C(=O)N[C@@H](C)C1=CC=C(C2=C(C)N=CS2)C=C1)C(C)(C)C)[C@H]1CC[C@H](CN2CCC(C3=NC4=C(C=C3)C3(CCCCC3)C3=NC(=O)C5=C(C=CC=C5Cl)N34)CC2)CC1	C57H71ClN10O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-OVPA3K	SCHEMBL30843696	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4'-chloro-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3,3-dimethylbutanoyl]-N-[(1S)-3-(3-fluoro-3-methylazetidin-1-yl)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]propyl]-4-hydroxypyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CCN3CC(C)(F)C3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C([C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C62H76ClFN10O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-1STQ0N	SCHEMBL27394964	(2S,4R)-1-[(2S)-2-[5-[4-(4'-chloro-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-9'-yl)piperidin-1-yl]pentanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL30843668	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCN3CCC(C4=CC5=C(C=C4)N4C(=NC(=O)C6=C4C=CC=C6Cl)C54CCCCC4)CC3)C(C)(C)C)C=C2)SC=N1	C53H64ClN7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-TUOVEN	SCHEMBL30843599	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4'-chloro-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-3-(3-hydroxy-3-methylazetidin-1-yl)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]propyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CCN3CC(C)(O)C3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C([C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C62H77ClN10O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-B4EQ07	WO2024064328A1_A81	.	CC1=C(C2=CC=C([C@H](CCN3CCOCC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C([C@H]4CC[C@H](NN5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C61H76ClN11O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-7R356Q	SCHEMBL30843685	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4'-chloro-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-3-[2-(2-methoxyethoxy)ethoxy]-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]propyl]pyrrolidine-2-carboxamide	COCCOCCOCC[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](N1C=C([C@H]2CC[C@H](CN3CCC(C4=CC5=C(C=C4)C4(CCCCC4)C4=NC(=O)C6=C(C=CC=C6Cl)N45)CC3)CC2)N=N1)C(C)(C)C)C1=CC=C(C2=C(C)N=CS2)C=C1	C63H80ClN9O7S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-FG922D	WO2024064328A1_A83	.	CC1=C(C2=CC=C([C@H](CN3CCC(C(F)(F)F)CC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C([C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C63H76ClF3N10O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-811TLH	WO2024064328A1_A84	.	CC1=C(C2=CC=C([C@H](CN3CCC(C(F)F)CC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(N3C=C([C@H]4CC[C@H](ON5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6NC(=O)C8=C(C=CC=C8Cl)N76)CC5)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C62H77ClF2N10O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-PTLVKR	SCHEMBL30843398	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4'-chloro-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1R)-2-(4-methylpiperazin-1-yl)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CN3CCN(C)CC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C([C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C62H78ClN11O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-AXU0J1	WO2024064328A1_A86	.	CC1=C(C2=CC=C([C@H](COCCO)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C([C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C59H72ClN9O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-T12VU1	WO2024064328A1_A87	.	COCCOCCOC[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](N1C=C([C@H]2CC[C@H](CN3CCC(C4=CC5=C(C=C4)C4(CCCCC4)C4=NC(=O)C6=C(C=CC=C6Cl)N45)CC3)CC2)NN1)C(C)(C)C)C1=CC=C(C2=C(C)N=CS2)C=C1	C62H80ClN9O7S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-41DVZU	SCHEMBL30843455	(2S,4R)-1-[(2S)-2-[4-[3-[[7-(4'-chloro-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)-2-azaspiro[3.5]nonan-2-yl]methyl]cyclobutyl]triazol-1-yl]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1R)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]-2-morpholin-4-ylethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CN3CCOCC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C([C@H]4C[C@H](CN5CC6(CCC(C7=CC8=C(C=C7)C7(CCCCC7)C7=NC(=O)C9=C(C=CC=C9Cl)N78)CC6)C5)C4)N=N3)C(C)(C)C)C=C2)SC=N1	C62H75ClN10O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-Y4431J	WO2024064328A1_A89	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C([C@H]4CC[C@H](ON5CCC(C6=CC7=C(C=C6)C(C)(C)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C53H62ClN9O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-F7EA04	SCHEMBL27395027	(2S,4R)-1-[(2S)-2-[6-[4-(4'-chloro-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-9'-yl)piperidin-1-yl]hexanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; SCHEMBL30843543	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCN3CCC(C4=CC5=C(C=C4)N4C(=NC(=O)C6=C4C=CC=C6Cl)C54CCCCC4)CC3)C(C)(C)C)C=C2)SC=N1	C54H66ClN7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-JT2EC5	SCHEMBL30843401	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-10-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1R)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]-2-morpholin-4-ylethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CN3CCOCC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C([C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)C(C)(C)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C58H71ClN10O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-6Z91SL	WO2024064328A1_A91	.	COCCOC[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](N1C=C([C@H]2CC[C@H](CN3CCC(C4=CC5=C(C=C4)C(C)(C)C4=NC(=O)C6=C(C=CC=C6Cl)N45)CC3)CC2)N=N1)C(C)(C)C)C1=CC=C(C2=C(C)N=CS2)C=C1	C57H70ClN9O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-2CPIV1	WO2024064328A1_A92	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-10-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1R)-2-[2-(2-methoxyethoxy)ethoxy]-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	COCCOCCOC[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](N1C=C([C@H]2CC[C@H](CN3CCC(C4=CC5=C(C=C4)C(C)(C)C4=NC(=O)C6=C(C=CC=C6Cl)N45)CC3)CC2)N=N1)C(C)(C)C)C1=CC=C(C2=C(C)N=CS2)C=C1	C59H74ClN9O7S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-L2NYLD	WO2024064328A1_A93	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-10-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3,3-dimethylbutanoyl]-N-[(1R)-2-(3-fluoro-3-methylazetidin-1-yl)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]-4-hydroxypyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CN3CC(C)(F)C3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C(C4CCC(CN5CCC(C6=CC7=C(C=C6)C(C)(C)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C58H70ClFN10O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-0PS12K	SCHEMBL30843747	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-10-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3,3-dimethylbutanoyl]-N-[(1R)-2-(4,4-difluoropiperidin-1-yl)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]-4-hydroxypyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CN3CCC(F)(F)CC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C([C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)C(C)(C)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C59H71ClF2N10O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-I226WX	SCHEMBL30843651	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-10-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1R)-2-(3-hydroxy-3-methylazetidin-1-yl)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CN3CC(C)(O)C3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C([C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)C(C)(C)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C58H71ClN10O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-9KNXCL	WO2024064328A1_A96	.	CC1=C(C2=CC=C([C@H](CN3CC4(COC4)C3)NC(=O)[C@@H]3CC(=O)CN3C(=O)[C@@H](N3C=C([C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C62H73ClN10O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-IZAN0X	WO2024064328A1_A97	.	CC1=C(C2=CC=C([C@H](CN3CCC4(COC4)C3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C([C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=C=C=C8Cl)N67)CC5)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C63H75ClN10O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-H1R0IR	SCHEMBL30843603	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-10-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1R)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]-2-(2-oxa-6-azaspiro[3.3]heptan-6-yl)ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CN3CC4(COC4)C3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C([C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)C(C)(C)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C59H71ClN10O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-7NP30W	WO2024064328A1_A99	.	CC1=C(C2=CC=C([C@H](CN3CCC4(CO4)C3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C([C@H]4CC[C@H](NN5CCC(C6=CC7=C(C=C6)C(C)(C)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C58H70ClN11O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-IF28B3	WO2024064328A1_B1	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)[C@H]3CC[C@H](CN4CCC(C5=CC6=C(C=C5)N5C(=NC(=O)C7=C5C=CC=C7Cl)C6(C)C)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C53H64ClN7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-3XMEER	WO2024064328A1_B100	(2S,4R)-1-[(2R)-2-[3-[[4-[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-8-yl)piperidin-1-yl]cyclohexyl]methoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(OCC4CCC(N5CCC(C6=CC=CC7=C6C(C)(C)C6=NC(=O)C8=C(Cl)C=CC=C8N67)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C54H62ClN7O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-786PT3	WO2024064328A1_B101	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCN3C=C(C4=CC5=C(C=C4)N4C6=CC=CC(Cl)=C6C(=O)N=C4C5(C)C)C=N3)C(C)(C)C)C=C2)SC=N1	C46H49ClN8O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-1TOZJD	SCHEMBL30843594	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-10-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3,3-dimethylbutanoyl]-N-[(1R)-1-(4-ethynylphenyl)-2-morpholin-4-ylethyl]-4-hydroxypyrrolidine-2-carboxamide	C#CC1=CC=C([C@H](CN2CCOCC2)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](N2C=C([C@H]3CC[C@H](CN4CCC(C5=CC6=C(C=C5)C(C)(C)C5=NC(=O)C7=C(C=CC=C7Cl)N56)CC4)CC3)N=N2)C(C)(C)C)C=C1	C56H68ClN9O5	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-T42TE8	WO2024064328A1_B103	(2S,4R)-N-[(1S)-1-[4-[4-[3-[3-[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-10-yl)piperidin-1-yl]propoxy]prop-1-ynyl]-1,3-thiazol-5-yl]phenyl]ethyl]-4-hydroxy-1-[3-methyl-2-(3-methyl-1,2-oxazol-5-yl)butanoyl]pyrrolidine-2-carboxamide	CC1=NOC(C(C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=C(C#CCOCCCN4CCC(C5=CC6=C(C=C5)C(C)(C)C5=NC(=O)C7=C(C=CC=C7Cl)N56)CC4)N=CS3)C=C2)C(C)C)=C1	C53H58ClN7O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-GDF9XA	SCHEMBL30843567	(2S,4R)-N-[(1S)-1-[4-[4-[3-[2-[2-[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-10-yl)piperidin-1-yl]ethoxy]ethoxy]prop-1-ynyl]-1,3-thiazol-5-yl]phenyl]ethyl]-4-hydroxy-1-[3-methyl-2-(3-methyl-1,2-oxazol-5-yl)butanoyl]pyrrolidine-2-carboxamide	CC1=NOC(C(C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=C(C#CCOCCOCCN4CCC(C5=CC6=C(C=C5)C(C)(C)C5=NC(=O)C7=C(C=CC=C7Cl)N56)CC4)N=CS3)C=C2)C(C)C)=C1	C54H60ClN7O7S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-GYQY8D	SCHEMBL30843600	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4-bromo-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-10-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1R)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]-2-morpholin-4-ylethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CN3CCOCC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C([C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)C(C)(C)C6=NC(=O)C8=C(C=CC=C8Br)N67)CC5)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C58H71BrN10O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-LNCQF3	WO2024064328A1_B106	.	CC1=C(C2=CC=C([C@H](CN3CCOCC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C([C@H]4CC[C@H](CN5CCC(C6=CC7=C(CC6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Br)N67)CC5)CC4)N=N3)C=C2)SC=N1	C60H75BrN10O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-S5VMSL	WO2024064328A1_B107	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C([C@H]4CC[C@H](CN5CCC(C6=CC=CC7=C6C(C)(C)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N3)C=C2)SC=N1	C53H62ClN9O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-Y232GE	WO2024064328A1_B108	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4'-chloro-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-[4-(3-morpholin-4-ylpropyl)-1,3-thiazol-5-yl]phenyl]ethyl]pyrrolidine-2-carboxamide	C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](N1C=C([C@H]2CC[C@H](CN3CCC(C4=CC5=C(C=C4)C4(CCCCC4)C4=NC(=O)C6=C(C=CC=C6Cl)N45)CC3)CC2)N=N1)C(C)(C)C)C1=CC=C(C2=C(CCCN3CCOCC3)N=CS2)C=C1	C63H79ClN10O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-XJTV7H	WO2024064328A1_B109	(2S,4R)-1-[(2S)-2-[3-[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-9-yl)piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1R)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]-2-morpholin-4-ylethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CN3CCOCC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3=CC(N4CCC(C5=CC6=C(C=C5)N5C(=NC(=O)C7=C5C=CC=C7Cl)C6(C)C)CC4)=NO3)C(C)C)C=C2)SC=N1	C51H57ClN8O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-Q1EHFN	WO2024064328A1_B11	(2S,4R)-1-[(2R)-2-[3-[3-[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-9-yl)piperidin-1-yl]propoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(OCCCN4CCC(C5=CC6=C(C=C5)N5C(=NC(=O)C7=C5C=CC=C7Cl)C6(C)C)CC4)=NO3)C(C)C)C=C2)SC=N1	C50H56ClN7O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-FPOCU2	WO2024064328A1_B110	(2S,4R)-1-[(2R)-2-[3-[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-9-yl)piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1R)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]-2-morpholin-4-ylethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CN3CCOCC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(C5=CC6=C(C=C5)N5C(=NC(=O)C7=C5C=CC=C7Cl)C6(C)C)CC4)=NO3)C(C)C)C=C2)SC=N1	C51H57ClN8O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-FO670T	WO2024064328A1_B111	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCN(C6=CC7=C(C=C6)C(C)(C)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C52H60ClN9O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-04CJZ5	WO2024064328A1_B113	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-10-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3,3-dimethylbutanoyl]-4-hydroxy-N-[3-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]azetidin-3-yl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(C3(NC(=O)[C@@H]4C[C@@H](O)CN4C(=O)[C@@H](N4C=C([C@H]5CC[C@H](CN6CCC(C7=CC8=C(C=C7)C(C)(C)C7=NC(=O)C9=C(C=CC=C9Cl)N78)CC6)CC5)N=N4)C(C)(C)C)CNC3)C=C2)SC=N1	C55H65ClN10O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-MK69M5	WO2024064328A1_B114	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C(C4CCC(N5CCC(C6=CC=CC7=C6C(C)(C)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N3)C=C2)SC=N1	C52H60ClN9O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-C8WMOE	WO2024064328A1_B115	.	CC1=C(C2=CC=C([C@H](CN3CCOCC3)NC(=O)C3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCC(CN5CCC(C6=CC7=C(C=C6)C(C)(C)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C57H68ClN9O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-NE4C7E	SCHEMBL30843491	(2S,4R)-1-[(2R)-2-[3-[2-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-8-yl)ethoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(OCCC4=CC=CC5=C4C(C)(C)C4=NC(=O)C6=C(C=CC=C6Cl)N45)=NO3)C(C)C)C=C2)SC=N1	C44H45ClN6O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-BQFGDP	WO2024064328A1_B117	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-10-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3,3-dimethylbutanoyl]-N-[(1S)-1-[4-(4-chloro-1,3-thiazol-5-yl)phenyl]ethyl]-4-hydroxypyrrolidine-2-carboxamide	C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](N1C=C([C@H]2CC[C@H](CN3CCC(C4=CC5=C(C=C4)C(C)(C)C4=NC(=O)C6=C(C=CC=C6Cl)N45)CC3)CC2)N=N1)C(C)(C)C)C1=CC=C(C2=C(Cl)N=CS2)C=C1	C53H61Cl2N9O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-9YBI4Q	WO2024064328A1_B118	.	CC1=C(C2=CC=C([C@H](CN3CCOCC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C([C@H]4CC[C@H](S(=O)(=O)N5CCC(C6=CC=C7C(=C6)N6C(=NC(=O)C8=C6C=CC=C8Cl)C76CCCCC6)CC5)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C60H73ClN10O7S2	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-2O59X5	WO2024064328A1_B119	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C(C4=CC=CC(CN5CCC(C6=CC7=C(C=C6)C(C)(C)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)=C4)N=N3)C(C)(C)C)C=C2)SC=N1	C54H58ClN9O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-ZIBMSO	WO2024064328A1_B12	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(OCCCCN4CCC(C5=CC6=C(C=C5)N5C7=CC=CC(Cl)=C7C(=O)N=C5C6(C)C)CC4)=NO3)C(C)C)C=C2)SC=N1	C51H58ClN7O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-FXCNRU	WO2024064328A1_B120	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-10-yl)piperazin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C([C@H]4CC[C@H](CN5CCN(C6=CC7=C(C=C6)C(C)(C)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N3)C=C2)SC=N1	C52H61ClN10O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-MFHM71	WO2024064328A1_B121	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-10-yl)piperazin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C([C@H]4CC[C@H](CN5CCN(C6=CC7=C(C=C6)C(C)(C)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C53H63ClN10O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-IUCID1	WO2024064328A1_B122	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-10-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1R)-5-(4-methyl-1,3-thiazol-5-yl)-2,3-dihydro-1H-inden-1-yl]pyrrolidine-2-carboxamide	CC1=C(C2=CC3=C(C=C2)[C@H](NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](N2C=C([C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)C(C)(C)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N2)C(C)(C)C)CC3)SC=N1	C55H64ClN9O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-7MZKCA	WO2024064328A1_B123	.	CC1=C(C2=CC3=C(C=C2)[C@@H](NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](N2C=C([C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)C(C)(C)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N2)C(C)(C)C)CC3)SC=N1	C55H64ClN9O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-KKOSSE	WO2024064328A1_B124	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-10-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3,3-dimethylbutanoyl]-4-hydroxy-N-[1-methyl-3-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]azetidin-3-yl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C(C3(NC(=O)[C@@H]4C[C@@H](O)CN4C(=O)[C@@H](N4C=C([C@H]5CC[C@H](CN6CCC(C7=CC8=C(C=C7)C(C)(C)C7=NC(=O)C9=C(C=CC=C9Cl)N78)CC6)CC5)N=N4)C(C)(C)C)CN(C)C3)C=C2)SC=N1	C56H67ClN10O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-USH3TY	WO2024064328A1_B125	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-10-yl)piperazin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(2-methylpyrazol-3-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](N1C=C([C@H]2CC[C@H](CN3CCN(C4=CC5=C(C=C4)C(C)(C)C4=NC(=O)C6=C(C=CC=C6Cl)N45)CC3)CC2)N=N1)C(C)(C)C)C1=CC=C(C2=CC=NN2C)C=C1	C53H64ClN11O4	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-PRJYUG	WO2024064328A1_B126	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C(C4CCC(CN5CCN(C6=CC7=C(C=C6)C(C)(C)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N3)C(C)(C)C)C=C2)OC=N1	C53H63ClN10O5	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-TUYM6O	WO2024064328A1_B127	.	C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](N1C=C([C@H]2CC[C@H](CN3CCN(C4=CC5=C(C=C4)C(C)(C)C4=NC(=O)C6=C(C=CC=C6Cl)N45)CC3)CC2)N=N1)C(C)(C)C)C1=CC=C(C2=CC=NN2)C=C1	C52H62ClN11O4	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-DZHZ3O	WO2024064328A1_B128	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-10-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3-methylbutanoyl]-N-[(1S)-1-(4-ethynylphenyl)ethyl]-4-hydroxypyrrolidine-2-carboxamide	C#CC1=CC=C([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](C(C)C)N2C=C([C@H]3CC[C@H](CN4CCC(C5=CC6=C(C=C5)C(C)(C)C5=NC(=O)C7=C(C=CC=C7Cl)N56)CC4)CC3)N=N2)C=C1	C51H59ClN8O4	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-4WZPL8	WO2024064328A1_B129	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-10-yl)piperazin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1R)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]-2-morpholin-4-ylethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CN3CCOCC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C([C@H]4CC[C@H](CN5CCN(C6=CC7=C(C=C6)C(C)(C)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N3)C=C2)SC=N1	C56H68ClN11O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-18WB1B	WO2024064328A1_B13	(2S,4R)-1-[(2S)-2-[[3-[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-9-yl)piperidin-1-yl]cyclobutanecarbonyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3CC(N4CCC(C5=CC6=C(C=C5)N5C(=NC(=O)C7=C5C=CC=C7Cl)C6(C)C)CC4)C3)C(C)(C)C)C=C2)SC=N1	C50H58ClN7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-ASJFP3	WO2024064328A1_B130	(2S,4R)-1-[(2R)-2-[3-[3-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-8-yl)prop-2-ynoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(OCC#CC4=CC=CC5=C4C(C)(C)C4=NC(=O)C6=C(C=CC=C6Cl)N45)=NO3)C(C)C)C=C2)SC=N1	C45H43ClN6O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-NFJT7Z	WO2024064328A1_B131	.	CC#CC1=CC=C([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](C(C)C)N2C=C([C@H]3CC[C@H](CN4CCC(C5=CC6=C(C=C5)C(C)(C)C5=NC(=O)C7=C(C=CC=C7Cl)N56)CC4)CC3)N=N2)C=C1	C52H61ClN8O4	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-QSP6NF	SCHEMBL30843528	(2S,4R)-1-[(2S)-2-[4-[[4-[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-8-yl)piperidin-1-yl]cyclohexyl]methyl]triazol-1-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C(CC4CCC(N5CCC(C6=CC=CC7=C6C(C)(C)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N3)C=C2)SC=N1	C53H62ClN9O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-OY48KW	WO2024064328A1_B133	.	CC1=NC(C)=C(C2=CC=C([C@H](C)NC(=O)C3C[C@@H](O)CN3C(=O)[C@@H](N3C=C([C@H]4CC[C@H](CN5CCN(C6=CC7=C(C=C6)C(C)(C)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N3)C(C)(C)C)C=C2)S1	C54H65ClN10O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-WI3XZ2	WO2024064328A1_B134	(2S,4R)-N-[(1S)-1-(4-acetylphenyl)ethyl]-1-[(2S)-2-[4-[4-[[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-10-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3-methylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide	CC(=O)C1=CC=C([C@H](C)NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@H](C(C)C)N2C=C([C@H]3CC[C@H](CN4CCC(C5=CC6=C(C=C5)C(C)(C)C5=NC(=O)C7=C(C=CC=C7Cl)N56)CC4)CC3)N=N2)C=C1	C51H61ClN8O5	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-6MAAEP	WO2024064328A1_B135	.	C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](N1C=C(C2CCC(CN3CCN(C4=CC5=C(C=C4)C(C)(C)C4=NC(=O)C6=C(C=CC=C6Cl)N45)CC3)CC2)N=N1)C(C)(C)C)C1=CC=C(C2=C(C#CCN3CCOCC3)N=CS2)C=C1	C59H70ClN11O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-GBFEWZ	WO2024064328A1_B136	.	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=C(C#CCN3CCOCC3)N=CS2)C=C1)N1C=C([C@H]2CC[C@H](CN3CCN(C4=CC5=C(C=C4)C(C)(C)C4=NC(=O)C6=C(C=CC=C6Cl)N45)CC3)CC2)N=N1	C58H68ClN11O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-5QOC5H	WO2024064328A1_B137	(2S,4R)-1-[(2S)-2-[4-[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-8-yl)cyclohexyl]triazol-1-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C(C4CCC(C5=CC=CC6=C5C(C)(C)C5=NC(=O)C7=C(C=CC=C7Cl)N56)CC4)N=N3)C=C2)SC=N1	C47H51ClN8O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-JHMLHO	WO2024064328A1_B138	.	CC1=C(C2=CC=C([C@H](CN3CCOCC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(O[C@H]4CC[C@H](CN5CCN(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(Cl)C=CC=C8N67)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C60H72ClN9O7S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-92PW3H	SCHEMBL30843478	(2S,4R)-N-[(1R)-2-[4-[[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-8-yl)piperidin-1-yl]methyl]piperidin-1-yl]-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]-4-hydroxy-1-[3-methyl-2-(3-methyl-1,2-oxazol-5-yl)butanoyl]pyrrolidine-2-carboxamide	CC1=NOC(C(C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](CN2CCC(CN3CCC(C4=CC=CC5=C4C(C)(C)C4=NC(=O)C6=C(C=CC=C6Cl)N45)CC3)CC2)C2=CC=C(C3=C(C)N=CS3)C=C2)C(C)C)=C1	C54H63ClN8O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-80D3QL	WO2024064328A1_B140	.	C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](N1C=C(C2CCC(CN3CCN(C4=CC5=C(C=C4)C4(CCCCC4)C4=NC(=O)C6=C(C=CC=C6Cl)N45)CC3)CC2)N=N1)C(C)(C)C)C1=CC=C(C2=C(C#CCN3CCOCC3)N=CS2)C=C1	C62H74ClN11O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-MYBUNC	WO2024064328A1_B141	.	C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](N(C)/C=C(\N=N)[C@H]1CC[C@H](CN2CCC(C3=CC4=C(C=C3)C(C)(C)C3=NC(=O)C5=C(C=CC=C5Cl)N34)CC2)CC1)C(C)(C)C)C1=CC=C(C2=C(C#N)N=CS2)C=C1	C55H65ClN10O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-SFA448	WO2024064328A1_B143	.	CC1=C(C2=CC3=C(C=C2)C(NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](N2C=C([C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)C(C)(C)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N2)C(C)(C)C)=NC=C3)SC=N1	C55H61ClN10O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-VVNHXW	SCHEMBL30843412	(2S,4R)-N-[(1S)-1-[4-[4-[3-[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-9-yl)piperidin-1-yl]prop-1-ynyl]-1,3-thiazol-5-yl]phenyl]ethyl]-4-hydroxy-1-[3-methyl-2-(3-methyl-1,2-oxazol-5-yl)butanoyl]pyrrolidine-2-carboxamide; SCHEMBL30843422	CC1=NOC(C(C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=C(C#CCN4CCC(C5=CC6=C(C=C5)N5C(=NC(=O)C7=C5C=CC=C7Cl)C6(C)C)CC4)N=CS3)C=C2)C(C)C)=C1	C50H52ClN7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-X13RAG	WO2024064328A1_B145	(2S,4R)-N-[(1S)-1-[4-[4-[3-[3-[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-8-yl)piperidin-1-yl]propoxy]prop-1-ynyl]-1,3-thiazol-5-yl]phenyl]ethyl]-4-hydroxy-1-[3-methyl-2-(3-methyl-1,2-oxazol-5-yl)butanoyl]pyrrolidine-2-carboxamide	CC1=NOC(C(C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=C(C#CCOCCCN4CCC(C5=CC=CC6=C5C(C)(C)C5=NC(=O)C7=C(C=CC=C7Cl)N56)CC4)N=CS3)C=C2)C(C)C)=C1	C53H58ClN7O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-LO1NB3	WO2024064328A1_B146	.	CC1=C(C2=CC3=C(C=C2)C(NC(=O)C2C[C@@H](O)CN2C(=O)[C@@H](N2C=C([C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)C(C)(C)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N2)C(C)(C)C)CCC3)SC=N1	C56H66ClN9O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-WKGIC2	SCHEMBL30843562	N-[4-[2-[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-10-yl)piperidin-1-yl]ethoxy]butyl]-5-[4-[(1S)-1-[[(2S,4R)-4-hydroxy-1-[3-methyl-2-(3-methyl-1,2-oxazol-5-yl)butanoyl]pyrrolidine-2-carbonyl]amino]ethyl]phenyl]-1,3-thiazole-4-carboxamide	CC1=NOC(C(C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=C(C(=O)NCCCCOCCN4CCC(C5=CC6=C(C=C5)C(C)(C)C5=NC(=O)C7=C(C=CC=C7Cl)N56)CC4)N=CS3)C=C2)C(C)C)=C1	C54H63ClN8O7S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-YURGEM	WO2024064328A1_B148	.	CC1=C(C2=CC3=C(C=C2)C(NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](N2C=C(C4CCC(CN5CCC(C6=CC7=C(C=C6)C(C)(C)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N2)C(C)(C)C)=NN3)SC=N1	C53H60ClN11O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-RG4MG9	WO2024064328A1_B149	.	CC1=C([C@H](C)NC(=O)C2C[C@@H](C)CN2C(=O)[C@@H](N2C=C([C@H]3CC[C@H](CN4CCC(C5=CC6=C(C=C5)C(C)(C)C5=NC(=O)C7=C(C=CC=C7Cl)N56)CC4)CC3)N=N2)C(C)(C)C)C=CC(C2=C(C)N=CS2)=C1	C56H68ClN9O3S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-RR1DMR	WO2024064328A1_B15	(2S,4R)-1-[2-[3-[2-[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-9-yl)piperidin-1-yl]ethyl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(CCN4CCC(C5=CC6=C(C=C5)N5C(=NC(=O)C7=C5C=CC=C7Cl)C6(C)C)CC4)=NO3)C(C)C)C=C2)SC=N1	C49H54ClN7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-LWBS8J	WO2024064328A1_B150	.	CC1=NOC(C(C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](C)C2=CC=C(C3=C(C#CCN4CCC(C5=CC=CC6=C5C(C)(C)C5=NC(=O)C7=C(C=CC=C7Cl)N56)CC4)N=CS3)C=C2)C(C)C)=C1	C50H52ClN7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-MTG1C7	WO2024064328A1_B151	.	CC1=C(C2=CC3=C(C=C2)[C@H](NC(=O)[C@@H]2C[C@@H](O)CN2C(=O)[C@@H](N2C=C(C4CCC(CN5CCC(C6=CC7=C(C=C6)C(C)(C)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N2)C(C)(C)C)CCC3)SC=N1	C56H66ClN9O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-J58TW1	SCHEMBL30843591	(2S,4R)-N-[(1S)-3-[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-8-yl)piperidin-1-yl]-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]propyl]-4-hydroxy-1-[3-methyl-2-(3-methyl-1,2-oxazol-5-yl)butanoyl]pyrrolidine-2-carboxamide	CC1=NOC(C(C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](CCN2CCC(C3=CC=CC4=C3C(C)(C)C3=NC(=O)C5=C(C=CC=C5Cl)N34)CC2)C2=CC=C(C3=C(C)N=CS3)C=C2)C(C)C)=C1	C49H54ClN7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-J7RMTE	WO2024064328A1_B153	(2S,4R)-N-[(1R)-2-[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-8-yl)piperidin-1-yl]-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]-4-hydroxy-1-[3-methyl-2-(3-methyl-1,2-oxazol-5-yl)butanoyl]pyrrolidine-2-carboxamide	CC1=NOC(C(C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](CN2CCC(C3=CC=CC4=C3C(C)(C)C3=NC(=O)C5=C(C=CC=C5Cl)N34)CC2)C2=CC=C(C3=C(C)N=CS3)C=C2)C(C)C)=C1	C48H52ClN7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-9A2ZXJ	WO2024064328A1_B154	.	CC1=NOC(C(C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](CN2CCC(C3=CC=CC4=C3C(C)(C)C3=NC(=O)C5=C(C=CC=C5CI)N34)CC2)C2=CC=C(C3=C(C)N=CS3)C=C2)C(C)C)=C1	C49H54IN7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-NGX9PB	WO2024064328A1_B155	.	CC1=NOC(C(C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](CN2CCC(N3CCC(C4=CC=CC5=C4C(C)(C)C4=NC(=O)C6=C(C=CC=C6Cl)N45)CC3)CC2)C2=CC=C(C3=C(C)N=CS3)C=C2)C(C)C)=C1	C53H61ClN8O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-PXJUEG	WO2024064328A1_B156	.	C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@H](N1C=C([C@H]2CC[C@H](CN3CCC(C4=CC5=C(C=C4)C(C)(C)C4=NC(=O)C6=C(C=CC=C6Cl)N45)CC3)CC2)N=N1)C(C)(C)C)C1=CC=C(C2=C(C#CCN3CCOCC3)N=CS2)C=C1	C60H71ClN10O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-XQCMTY	WO2024064328A1_B157	(2S,4R)-1-[(2R)-2-[3-[4-[[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-10-yl)piperidin-1-yl]methyl]cyclohexyl]oxy-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1R)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]-2-morpholin-4-ylethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CN3CCOCC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(O[C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)C(C)(C)C6=NC(=O)C8=C(Cl)C=CC=C8N67)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C58H69ClN8O7S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-817XLH	WO2024064328A1_B158	.	CC1=C(C2=CC=C(C(CN3CCOCC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(O[C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(Cl)C=CC=C8N67)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C61H73ClN8O7S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-BJUFNP	SCHEMBL30843407	(2S,4R)-1-[(2R)-2-[3-[4-[[4-(4'-bromo-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidin-1-yl]methyl]cyclohexyl]oxy-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1R)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]-2-morpholin-4-ylethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CN3CCOCC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(O[C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(Br)C=CC=C8N67)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C61H73BrN8O7S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-UQMKKJ	SCHEMBL30843481	(2S,4R)-1-[(2S)-2-[[3-[[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-9-yl)piperidin-1-yl]methyl]benzoyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3=CC(CN4CCC(C5=CC6=C(C=C5)N5C(=NC(=O)C7=C5C=CC=C7Cl)C6(C)C)CC4)=CC=C3)C(C)(C)C)C=C2)SC=N1	C53H58ClN7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-8SOFVW	WO2024064328A1_B160	(2S,4R)-1-[(2S)-2-[3-[4-[[4-(4'-chloro-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperazin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]-2-morpholin-4-ylethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@@H](CN3CCOCC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3=CC(N4CCC(CN5CCN(C6=CC7=C(C=C6)C6(CCCCC6)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C59H71ClN10O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-MY3KAZ	WO2024064328A1_B163	.	CC1=C(C2=CC=C([C@H](CN3CCOCC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(O[C@H]4CC[C@H](CN5CCN(C6=CC7=C(C=C6)C(C)(C)C6=NC(=O)C8=C(Cl)C=CC=C8N67)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C57H68ClN9O7S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-BQ55ER	WO2024064328A1_B164	.	CC1=NC(C)=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C([C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)C(C)(C)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N3)C(C)(C)C)C=C2)S1	C55H66ClN9O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-97ZB9U	WO2024064328A1_B167	.	CC1=NC(C)=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCC(C5CC=CC6=C5C(C)(C)C5=NC(=O)C7=C(C=CC=C7Cl)N56)CC4)=NO3)C(C)C)C=C2)S1	C48H54ClN7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-KR2AQS	WO2024064328A1_B168	.	CC1=NC(C)=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C([C@H]4CC[C@H](CN5CCN(C6=CC=C7C(=C6)N6C(=NC(=O)C8=C6C=CC=C8Cl)C76CCCCC6)CC5)CC4)N=N3)C(C)(C)C)C=C2)S1	C57H69ClN10O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-8GFHDQ	SCHEMBL30843442	(2S,4R)-1-[(2S)-2-[4-[3-[4-(4'-chloro-5'-oxospiro[cyclohexane-1,7'-indolo[1,2-a]quinazoline]-10'-yl)piperidine-1-carbonyl]-1-bicyclo[1.1.1]pentanyl]triazol-1-yl]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C(C45CC(C(=O)N6CCC(C7=CC=C8C(=C7)N7C(=NC(=O)C9=C7C=CC=C9Cl)C87CCCCC7)CC6)(C4)C5)N=N3)C(C)(C)C)C=C2)SC=N1	C56H62ClN9O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-QFQV07	WO2024064328A1_B17	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C(CCN4CCC(C5=CC6=C(C=C5)N5C(=NC(=O)C7=C5C=CC=C7Cl)C6(C)C)CC4)N=N3)C=C2)SC=N1	C48H54ClN9O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-KWT1YG	WO2024064328A1_B18	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C34CCC(CN5CCC(C6=CC7=C(C=C6)N6C(=NC(=O)C8=C6C=CC=C8Cl)C7(C)C)CC5)(CC3)C4)C(C)(C)C)C=C2)SC=N1	C54H64ClN7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-KSPH9A	WO2024064328A1_B19	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C(C4CCC(CN5CCC(C6=CC7=C(C=C6)N6C(=NC(=O)C8=C6C=CC=C8Cl)C7(C)C)CC5)CC4)N=N3)C=C2)SC=N1	C53H62ClN9O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-U7DET7	WO2024064328A1_B20	(2S,4R)-1-[(2S)-2-[[5-[[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-9-yl)piperidin-1-yl]methyl]thiophene-2-carbonyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3=CC=C(CN4CCC(C5=CC6=C(C=C5)N5C(=NC(=O)C7=C5C=CC=C7Cl)C6(C)C)CC4)S3)C(C)(C)C)C=C2)SC=N1	C51H56ClN7O5S2	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-O62CB1	WO2024064328A1_B21	.	CC1=C(C2=CC=C([C@H](CCCCCN3CCC(C4=CC5=C(C=C4)C(C)(C)C4=NC(=O)C6=C(Cl)C=CC=C6N45)CC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3(F)CC3)C(C)(C)C)C=C2)SC=N1	C53H63ClFN7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-M4DX06	WO2024064328A1_B22	.	CC1=C(C2=CC=C([C@H](CC(=O)N[C@H]3CC[C@H](CN4CCC(C5=CC6=C(C=C5)C(C)(C)C5=NC(=O)C7=C(C=CC=C7Cl)N56)CC4)CC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3(F)CC3)C(C)(C)C)C=C2)SC=N1	C57H68ClFN8O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-5OJP6B	WO2024064328A1_B23	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C34CC(CN5CCC(C6=CC7=C(C=C6)N6C(=NC(=O)C8=C6C=CC=C8Cl)C7(C)C)CC5)(C3)C4)C(C)(C)C)C=C2)SC=N1	C52H60ClN7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-1FKQ73	SCHEMBL30843615	(2S,4R)-1-[(2S)-2-[4-[3-[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-9-yl)piperidin-1-yl]propyl]triazol-1-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C(CCCN4CCC(C5=CC6=C(C=C5)N5C(=NC(=O)C7=C5C=CC=C7Cl)C6(C)C)CC4)N=N3)C=C2)SC=N1	C49H56ClN9O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-0BGDP5	WO2024064328A1_B25	.	CC1=C(C2=CC=C([C@H](CC(=O)NCCCN3CCC(C4=CC5=C(C=C4)C(C)(C)C4NC(=O)C6=C(C=CC=C6Cl)N54)CC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3(F)CC3)C(C)(C)C)C=C2)SC=N1	C53H64ClFN8O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-FXMUMW	WO2024064328A1_B26	(2S,4R)-1-[(2R)-2-[3-[3-[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-10-yl)piperidin-1-yl]propoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(OCCCN4CCC(C5=CC6=C(C=C5)C(C)(C)C5=NC(=O)C7=C(C=CC=C7Cl)N56)CC4)=NO3)C(C)C)C=C2)SC=N1	C50H56ClN7O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-FTFTGP	WO2024064328A1_B27	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(OCCCCN4CCC(C5=CC6=C(C=C5)C(C)(C)C5=NC(=O)C7=C(C=CC=C7Cl)N56)CC4)=NO3)C(C)C)C=C2)SC=N1	C51H58ClN7O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-NX71JN	WO2024064328A1_B28	(2S,4R)-1-[(2R)-2-[3-[4-[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-9-yl)piperidin-1-yl]cyclohexyl]oxy-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(OC4CCC(N5CCC(C6=CC7=C(C=C6)N6C(=NC(=O)C8=C6C=CC=C8Cl)C7(C)C)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C53H60ClN7O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-VTOD78	SCHEMBL30843419	(2S,4R)-1-[(2S)-2-[4-[[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-9-yl)piperidin-1-yl]methyl]triazol-1-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C(CN4CCC(C5=CC6=C(C=C5)N5C(=NC(=O)C7=C5C=CC=C7Cl)C6(C)C)CC4)N=N3)C=C2)SC=N1	C47H52ClN9O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-7ZAFBK	WO2024064328A1_B30	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(OC4CCC(CN5CCC(C6=CC7=C(C=C6)N6C8=CC=CC(Cl)=C8C(=O)N=C6C7(C)C)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C54H62ClN7O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-VAN6T6	WO2024064328A1_B31	.	CC1=C(C2=CC=C([C@H](CC(=O)NC3CCC(N4CCC(C5=CC6=C(C=C5)C(C)(C)C5NC(=O)C7=C(C=CC=C7Cl)N65)CC4)CC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3(F)CC3)C(C)(C)C)C=C2)SC=N1	C56H68ClFN8O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-YCKO53	WO2024064328A1_B32	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(OCCN4CCC(C5=CC6=C(C=C5)C(C)(C)C5=NC(=O)C7=C(C=CC=C7Cl)N56)CC4)=NO3)C(C)C)C=C2)SC=N1	C49H54ClN7O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-E6OT3L	SCHEMBL30843501	(2S,4R)-N-[(1S)-3-[4-[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-10-yl)piperidin-1-yl]butylamino]-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]-3-oxopropyl]-1-[(2S)-2-[(1-fluorocyclopropanecarbonyl)amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CC(=O)NCCCCN3CCC(C4=CC5=C(C=C4)C(C)(C)C4=NC(=O)C6=C(C=CC=C6Cl)N45)CC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3(F)CC3)C(C)(C)C)C=C2)SC=N1	C54H64ClFN8O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-FNEPMF	WO2024064328A1_B34	.	CC1=C(C2=CC(OCCN3CCC(C4=CC5=C(C=C4)C(C)(C)C4=NC(=O)C6=C(CCC=C6Cl)N45)CC3)=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3(F)CC3)C(C)(C)C)C=C2)SC=N1	C50H59ClFN7O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-LEGEF5	SCHEMBL30843462	(2S,4R)-N-[[2-[4-[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-10-yl)piperidin-1-yl]butoxy]-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-1-[(2S)-2-[(1-fluorocyclopropanecarbonyl)amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3(F)CC3)C(C)(C)C)C(OCCCCN3CCC(C4=CC5=C(C=C4)C(C)(C)C4=NC(=O)C6=C(C=CC=C6Cl)N45)CC3)=C2)SC=N1	C52H61ClFN7O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-SNOPSW	WO2024064328A1_B36	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C(CCN4CCC(C5=CC6=C(C=C5)C(C)(C)C5=NC(=O)C7=C(C=CC=C7Cl)N56)CC4)N=N3)C=C2)SC=N1	C48H54ClN9O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-YNZ4P5	WO2024064328A1_B37	(2S,4R)-1-[(2R)-2-[3-[4-[[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-10-yl)piperidin-1-yl]methyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(CN5CCC(C6=CC7=C(C=C6)C(C)(C)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C53H61ClN8O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-EHZFTI	WO2024064328A1_B38	(2S,4R)-1-[(2R)-2-[3-[4-[[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-10-yl)piperidin-1-yl]methyl]cyclohexyl]oxy-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(OC4CCC(CN5CCC(C6=CC7=C(C=C6)C(C)(C)C6=NC(=O)C8=C(Cl)C=CC=C8N67)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C54H62ClN7O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-OQAIQK	WO2024064328A1_B39	(2S,4R)-N-[[2-[3-[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-10-yl)piperidin-1-yl]propoxy]-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-1-[(2S)-2-[(1-fluorocyclopropanecarbonyl)amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide	CC1=C(C2=CC(OCCCN3CCC(C4=CC5=C(C=C4)C(C)(C)C4=NC(=O)C6=C(C=CC=C6Cl)N45)CC3)=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3(F)CC3)C(C)(C)C)C=C2)SC=N1	C51H59ClFN7O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-K9NGQM	WO2024064328A1_B4	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(OCCN4CCC(C5=CC6=C(C=C5)N5C(=NC(=O)C7=C5C=CC=C7Cl)C6(C)C)CC4)=NO3)C(C)C)C=C2)SC=N1	C48H52ClN7O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-6LKR2G	WO2024064328A1_B40	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)[C@H]3CC[C@H](CN4CCC(C5=CC6=C(C=C5)C(C)(C)C5=NC(=O)C7=C(C=CC=C7Cl)N56)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C53H64ClN7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-7QPBZ1	WO2024064328A1_B41	.	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CN=CS2)C=C1)N1C=C([C@H]2CC[C@H](CN3CCC(C4=CC5=C(C=C4)C(C)(C)C4=NC(=O)C6=C(C=CC=C6Cl)N45)CC3)CC2)N=N1	C52H60ClN9O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-5W9R1X	SCHEMBL30843551	(2S,4R)-1-[2-[3-[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-9-yl)piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(N4CCC(C5=CC6=C(C=C5)N5C(=NC(=O)C7=C5C=CC=C7Cl)C6(C)C)CC4)=NO3)C(C)C)C=C2)SC=N1	C47H50ClN7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-J4ALGR	SCHEMBL30843584	(2S,4R)-1-[(2S)-2-[3-[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-10-yl)piperidin-1-yl]propanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCN3CCC(C4=CC5=C(C=C4)C(C)(C)C4=NC(=O)C6=C(C=CC=C6Cl)N45)CC3)C(C)(C)C)C=C2)SC=N1	C48H56ClN7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-DHNIZK	WO2024064328A1_B44	.	CC1=C(C2=CC=C([C@H](CC(=O)NCCN3CCC(C4=CC5=C(C=C4)C(C)(C)C4=NC(=O)C6=C(C=CC=C6Cl)N45)CC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3(F)CC3)C(C)(C)C)C=C2)SC=N1	C52H60ClFN8O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-C1O83Q	WO2024064328A1_B45	(2S,4R)-1-[(2S)-2-[4-[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-10-yl)piperidin-1-yl]butanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCN3CCC(C4=CC5=C(C=C4)C(C)(C)C4=NC(=O)C6=C(C=CC=C6Cl)N45)CC3)C(C)(C)C)C=C2)SC=N1	C49H58ClN7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-67PXK1	WO2024064328A1_B46	(2S,4R)-N-[(1S)-6-[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-10-yl)pyrazol-1-yl]-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]hexyl]-1-[(2S)-2-[(1-fluorocyclopropanecarbonyl)amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CCCCCN3C=C(C4=CC5=C(C=C4)C(C)(C)C4=NC(=O)C6=C(C=CC=C6Cl)N45)C=N3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3(F)CC3)C(C)(C)C)C=C2)SC=N1	C51H56ClFN8O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-KMIF4W	WO2024064328A1_B47	(2S,4R)-1-[(2S)-2-[[4-[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-10-yl)piperidin-1-yl]cyclohexanecarbonyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3CCC(N4CCC(C5=CC6=C(C=C5)C(C)(C)C5=NC(=O)C7=C(C=CC=C7Cl)N56)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C52H62ClN7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-C3JHPH	SCHEMBL30843477	(2S,4R)-1-[(2S)-2-[[4-[[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-9-yl)pyrazol-1-yl]methyl]cyclohexanecarbonyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)[C@H]3CC[C@H](CN4C=C(C5=CC6=C(C=C5)N5C(=NC(=O)C7=C5C=CC=C7Cl)C6(C)C)C=N4)CC3)C(C)(C)C)C=C2)SC=N1	C51H57ClN8O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-FBBO1B	WO2024064328A1_B49	(2S,4R)-1-[(2S)-2-[4-[[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-10-yl)piperidin-1-yl]methyl]triazol-1-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C(CN4CCC(C5=CC6=C(C=C5)C(C)(C)C5=NC(=O)C7=C(C=CC=C7Cl)N56)CC4)N=N3)C=C2)SC=N1	C47H52ClN9O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-3QLRWE	WO2024064328A1_B5	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CN3CCC(C4=CC5=C(C=C4)N4C(=NC(=O)C6C(Br)=CC=CC64)C5(C)C)CC3)C(C)(C)C)C=C2)SC=N1	C47H56BrN7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-UD1OYQ	WO2024064328A1_B50	(2S,4R)-1-[(2S)-2-[5-[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-10-yl)piperidin-1-yl]pentanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCN3CCC(C4=CC5=C(C=C4)C(C)(C)C4=NC(=O)C6=C(C=CC=C6Cl)N45)CC3)C(C)(C)C)C=C2)SC=N1	C50H60ClN7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-4J3TUN	PROTAC SMARCA2 degrader-32	orb2814492; PROTAC SMARCA2 degrader-32; SCHEMBL30843698; HY-170343; 3033586-50-1	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C([C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)C(C)(C)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C54H64ClN9O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-EWY4YX	WO2024064328A1_B52	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(OCCN4C=C(C5=CC6=C(C=C5)N5C(=NC(=O)C7=C5C=CC=C7Cl)C6(C)C)C=N4)=NO3)C(C)C)C=C2)SC=N1	C47H47ClN8O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-2ANHJK	WO2024064328A1_B53	(2S,4R)-N-[(1S)-3-[[4-[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-10-yl)piperidin-1-yl]cyclohexyl]methylamino]-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]-3-oxopropyl]-1-[(2S)-2-[(1-fluorocyclopropanecarbonyl)amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CC(=O)NCC3CCC(N4CCC(C5=CC6=C(C=C5)C(C)(C)C5=NC(=O)C7=C(C=CC=C7Cl)N56)CC4)CC3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3(F)CC3)C(C)(C)C)C=C2)SC=N1	C57H68ClFN8O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-JKQJKM	SCHEMBL30843493	(2S,4R)-N-[(1S)-6-[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-9-yl)pyrazol-1-yl]-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]hexyl]-1-[(2S)-2-[(1-fluorocyclopropanecarbonyl)amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](CCCCCN3C=C(C4=CC5=C(C=C4)N4C(=NC(=O)C6=C4C=CC=C6Cl)C5(C)C)C=N3)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3(F)CC3)C(C)(C)C)C=C2)SC=N1	C51H56ClFN8O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-K9OYWM	SCHEMBL30843467	(2S,4R)-1-[2-[4-[2-[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-9-yl)piperidin-1-yl]ethoxy]pyrazol-1-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C(C)C)N3C=C(OCCN4CCC(C5=CC6=C(C=C5)N5C(=NC(=O)C7=C5C=CC=C7Cl)C6(C)C)CC4)C=N3)C=C2)SC=N1	C49H55ClN8O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-K33UIL	WO2024064328A1_B58	.	CC(C)[C@@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=CN=CS2)C=C1)N1C=C(CCCN2CCC(C3=CC4=C(C=C3)C(C)(C)C3=NC(=O)C5=C(C=CC=C5Cl)N34)CC2)N=N1	C48H54ClN9O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-7X6TYO	SCHEMBL30843482	(2S,4R)-1-[(2S)-2-[4-[4-[[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-10-yl)piperidin-1-yl]methyl]cyclohexyl]triazol-1-yl]-3-methylbutanoyl]-4-hydroxy-N-methylpyrrolidine-2-carboxamide	CNC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@H](C(C)C)N1C=C([C@H]2CC[C@H](CN3CCC(C4=CC5=C(C=C4)C(C)(C)C4=NC(=O)C6=C(C=CC=C6Cl)N45)CC3)CC2)N=N1	C42H53ClN8O4	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-04PZUC	WO2024064328A1_B60	(2S,4R)-1-[(2R)-2-[3-[2-[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-10-yl)pyrazol-1-yl]ethoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(OCCN4C=C(C5=CC6=C(C=C5)C(C)(C)C5=NC(=O)C7=C(C=CC=C7Cl)N56)C=N4)=NO3)C(C)C)C=C2)SC=N1	C47H47ClN8O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-H3WI8D	WO2024064328A1_B61	(2S,4R)-1-[(2S)-2-[4-[5-[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-10-yl)piperidin-1-yl]pentyl]triazol-1-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C(CCCCCN4CCC(C5=CC6=C(C=C5)C(C)(C)C5=NC(=O)C7=C(C=CC=C7Cl)N56)CC4)N=N3)C=C2)SC=N1	C51H60ClN9O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-E8O1KD	WO2024064328A1_B62	(2S,4R)-1-[2-[3-[[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-10-yl)piperidin-1-yl]methyl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(CN4CCC(C5=CC6=C(C=C5)C(C)(C)C5=NC(=O)C7=C(C=CC=C7Cl)N56)CC4)=NO3)C(C)C)C=C2)SC=N1	C48H52ClN7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-DUSXTT	WO2024064328A1_B63	(2S,4R)-1-[(2S)-2-[[2-[4-[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-10-yl)piperidin-1-yl]cyclohexyl]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CC3CCC(N4CCC(C5=CC6=C(C=C5)C(C)(C)C5=NC(=O)C7=C(C=CC=C7Cl)N56)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C53H64ClN7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-EOJ2DV	WO2024064328A1_B64	(2S,4R)-1-[(2S)-2-[5-[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-10-yl)pyrazol-1-yl]pentanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCN3C=C(C4=CC5=C(C=C4)C(C)(C)C4=NC(=O)C6=C(Cl)C=CC=C6N45)C=N3)C(C)(C)C)C=C2)SC=N1	C48H53ClN8O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-6TFIRY	WO2024064328A1_B65	.	C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](NC(=O)[C@H]1CC[C@H](C(=O)N2CCC(C3=CC4=C(C=C3)C(C)(C)C3=NC(=O)C5=C(C=CC=C5Cl)N34)CC2)CC1)C(C)(C)C)C1=CC=C(C2=NC=NN2C)C=C1	C52H62ClN9O6	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-PO7LI2	SCHEMBL30843494	(2S,4R)-1-[(2S)-2-[4-[1-[3-[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-10-yl)piperidin-1-yl]propyl]piperidin-4-yl]triazol-1-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C(C4CCN(CCCN5CCC(C6=CC7=C(C=C6)C(C)(C)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N3)C=C2)SC=N1	C54H65ClN10O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-KG7XIT	WO2024064328A1_B67	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C(C4CCN(CCN5CCC(C6=CC7=C(C=C6)C(C)(C)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)N=N3)C=C2)SC=N1	C53H63ClN10O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-WSZP3F	WO2024064328A1_B68	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C([C@H](C)N4CCC(C5=CC6=C(C=C5)C(C)(C)C5=NC(=O)C7=C(C=CC=C7Cl)N56)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C49H56ClN9O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-O05KPW	WO2024064328A1_B69	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C(CN4CCC(C5=CC6=C(C=C5)C(C)(C)C5=NC(=O)C7=C(C=CC=C7Cl)N56)CC4)N=N3)C(C)(C)C)C=C2)SC=N1	C48H54ClN9O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-9B80W1	WO2024064328A1_B70	(2S,4R)-1-[(2S)-2-[[4-[[4-(4-bromo-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-10-yl)piperidin-1-yl]methyl]cyclohexanecarbonyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)[C@H]3CC[C@H](CN4CCC(C5=CC6=C(C=C5)C(C)(C)C5=NC(=O)C7=C(C=CC=C7Br)N56)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C53H64BrN7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-B0DHYW	WO2024064328A1_B71	.	CC1=C(C2=CC=C([C@H](C)NC(=O)C3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(OCCCN4C=C(C5=CC6=C(C=C5)N5C(=NC(=O)C7=C5C=CC=C7Cl)C6(C)C)C=N4)=NO3)C(C)C)C=C2)SC=N1	C48H49ClN8O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-DO2XW6	WO2024064328A1_B72	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(OCCCN4C=C(C5=CC6=C(C=C5)C(C)(C)C5=NC(=O)C7=C(C=CC=C7Cl)N56)C=N4)=NO3)C(C)C)C=C2)SC=N1	C48H49ClN8O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-KLNIND	WO2024064328A1_B73	(2S,4R)-1-[(2S)-2-[4-[4-[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-10-yl)piperidin-1-yl]butyl]triazol-1-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C(CCCCN4CCC(C5=CC6=C(C=C5)C(C)(C)C5=NC(=O)C7=C(C=CC=C7Cl)N56)CC4)N=N3)C=C2)SC=N1	C50H58ClN9O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-7E8EAD	WO2024064328A1_B74	(2S,4R)-1-[2-[3-[2-[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-9-yl)piperidin-1-yl]ethoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(2-methyl-1,2,4-triazol-3-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC(C)C(C(=O)N1C[C@H](O)C[C@H]1C(=O)N[C@@H](C)C1=CC=C(C2=NC=NN2C)C=C1)C1=CC(OCCN2CCC(C3=CC4=C(C=C3)N3C(=NC(=O)C5=C3C=CC=C5Cl)C4(C)C)CC2)=NO1	C48H54ClN9O6	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-HDRYVZ	WO2024064328A1_B76	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3CCC(CN4CCC(C5=CC6=C(C=C5)N5C(=NC(=O)C7=C5C=CC=C7Cl)C6(C)C(F)(F)F)CC4)CC3)C(C)(C)C)C=C2)SC=N1	C53H61ClF3N7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-BPIFWR	WO2024064328A1_B77	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C34CCC(CN5CCC(C6=CC7=C(C=C6)C(C)(C)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)(CC3)C4)C(C)(C)C)C=C2)SC=N1	C54H64ClN7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-8KE74O	WO2024064328A1_B78	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C(C)C)N3C=C([C@H]4CC[C@H](CN5CCC(C6=CC7=C(C=C6)N6C(=NC(=O)C8=C6C=CC=C8Cl)C7(C)C)CC5)CC4)N=N3)C=C2)SC=N1	C53H62ClN9O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-XIWUV8	WO2024064328A1_B79	.	C=C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](NC(=O)[C@H]1CC[C@H](CN2CCC(C3=CC4=C(C=C3)N3C(=NC(=O)C5=C3C=CC=C5Cl)C4(C)C)CC2)CC1)C(C)(C)C)C1=CC=C(C2=C(C)N=CS2)C=C1	C54H64ClN7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-958UKQ	WO2024064328A1_B80	(2S,4R)-N-[[2-[[4-[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-10-yl)piperidin-1-yl]cyclohexyl]methoxy]-4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]-1-[(2S)-2-[(1-fluorocyclopropanecarbonyl)amino]-3,3-dimethylbutanoyl]-4-hydroxypyrrolidine-2-carboxamide	CC1=C(C2=CC(OCC3CCC(N4CCC(C5=CC6=C(C=C5)C(C)(C)C5=NC(=O)C7=C(C=CC=C7Cl)N56)CC4)CC3)=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3(F)CC3)C(C)(C)C)C=C2)SC=N1	C55H65ClFN7O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-HY1ZXF	SCHEMBL30843489	(2S,4R)-1-[(2R)-2-[3-[4-[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-10-yl)piperidin-1-yl]cyclohexyl]oxy-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(OC4CCC(N5CCC(C6=CC7=C(C=C6)C(C)(C)C6=NC(=O)C8=C(Cl)C=CC=C8N67)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C53H60ClN7O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-PDER1J	WO2024064328A1_B82	(2S,4R)-1-[(2R)-2-[3-[[1-[[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-9-yl)piperidin-1-yl]methyl]cyclopropyl]methoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(OCC4(CN5CCC(C6=CC7=C(C=C6)N6C(=NC(=O)C8=C6C=CC=C8Cl)C7(C)C)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C52H58ClN7O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-CP45RT	WO2024064328A1_B83	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCN3C=C(C4=CC5=C(C=C4)C(C)(C)C4=NC(=O)C6=C(Cl)C=CC=C6N45)C=N3)C(C)(C)C)C=C2)SC=N1	C47H51ClN8O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-CEOK9N	WO2024064328A1_B84	.	CC1=NOC(C(C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](CCCCCN2C=CC(C3=CC4=C(C=C3)C(C)(C)C3=NC(=O)C5=C(C=CC=C5Cl)N34)CC2)C2=CC=C(C3=C(C)N=CS3)C=C2)C(C)C)=C1	C52H58ClN7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-7Y7AGR	WO2024064328A1_B85	(2S,4R)-N-[(1S)-6-[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-9-yl)piperidin-1-yl]-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]hexyl]-4-hydroxy-1-[3-methyl-2-(3-methyl-1,2-oxazol-5-yl)butanoyl]pyrrolidine-2-carboxamide	CC1=NOC(C(C(=O)N2C[C@H](O)C[C@H]2C(=O)N[C@@H](CCCCCN2CCC(C3=CC4=C(C=C3)N3C(=NC(=O)C5=C3C=CC=C5Cl)C4(C)C)CC2)C2=CC=C(C3=C(C)N=CS3)C=C2)C(C)C)=C1	C52H60ClN7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-W5STM2	SCHEMBL30843744	(2S,4R)-1-[(2S)-2-[4-[2-[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-10-yl)piperidin-1-yl]spiro[3.3]heptan-6-yl]triazol-1-yl]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](N3C=C(C4CC5(C4)CC(N4CCC(C6=CC7=C(C=C6)C(C)(C)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC4)C5)N=N3)C(C)(C)C)C=C2)SC=N1	C54H62ClN9O4S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-YK4OVR	WO2024064328A1_B87	.	CC1=C2C(=O)N=C3N(C2=CC=C1)C1=C(C=C(C2=CN(CCCCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)N[C@@H](C)C4=CC=C(C5=C(C)N=CS5)C=C4)C(C)(C)C)N=C2)C=C1)C3(C)C	C49H56N8O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-AE8LLM	WO2024064328A1_B88	.	C[C@H](NC(=O)[C@@H]1C[C@@H](O)CN1C(=O)[C@@H](NC(=O)[C@H]1CC[C@H](CN2CCC(C3=CC4=C(C=C3)N3C(=NC(=O)C5=C3C=CC=C5Cl)C4(C)C)CC2)CC1)C(C)(C)C)C1=CC=C(C2=NC=NN2C)C=C1	C52H64ClN9O5	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-T7CBHT	WO2024064328A1_B89	(2S,4R)-1-[(2S)-2-[3-[4-[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-9-yl)piperidine-1-carbonyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@H](C3=CC(N4CCC(C(=O)N5CCC(C6=CC7=C(C=C6)N6C(=NC(=O)C8=C6C=CC=C8Cl)C7(C)C)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C53H59ClN8O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-30GW0O	WO2024064328A1_B90	(2S,4R)-1-[(2R)-2-[3-[4-[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-9-yl)piperidine-1-carbonyl]piperidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(N4CCC(C(=O)N5CCC(C6=CC7=C(C=C6)N6C(=NC(=O)C8=C6C=CC=C8Cl)C7(C)C)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C53H59ClN8O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-ZOAVL9	WO2024064328A1_B91	(2S,4R)-1-[(2R)-2-[3-[[1-[[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-10-yl)piperidin-1-yl]methyl]cyclopropyl]methoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(OCC4(CN5CCC(C6=CC7=C(C=C6)C(C)(C)C6=NC(=O)C8=C(C=CC=C8Cl)N67)CC5)CC4)=NO3)C(C)C)C=C2)SC=N1	C52H58ClN7O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-CEHZVA	WO2024064328A1_B92	(2S,4R)-1-[(2S)-2-[3-[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-10-yl)pyrazol-1-yl]propanoylamino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCN3C=C(C4=CC5=C(C=C4)C(C)(C)C4=NC(=O)C6=C(C=CC=C6Cl)N45)C=N3)C(C)(C)C)C=C2)SC=N1	C46H49ClN8O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-J3KV22	WO2024064328A1_B93	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCC3C=C(C4=CC5=C(C=C4)N4C(=NC(=O)C6=C4C=CC=C6Cl)C5(C)C)C=N3)C(C)(C)C)C=C2)SC=N1	C48H52ClN7O5S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-P4KH12	WO2024064328A1_B94	(2S,4R)-1-[(2R)-2-[3-[3-[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-10-yl)piperidin-1-yl]-2-methylpropoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(OCC(C)CN4CCC(C5=CC6=C(C=C5)C(C)(C)C5=NC(=O)C7=C(C=CC=C7Cl)N56)CC4)=NO3)C(C)C)C=C2)SC=N1	C51H58ClN7O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-7I6WCY	WO2024064328A1_B95	(2S,4R)-1-[(2R)-2-[3-[4-[[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-10-yl)pyrazol-1-yl]methyl]cyclohexyl]oxy-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(OC4CCC(CN5C=C(C6=CC7=C(C=C6)C(C)(C)C6=NC(=O)C8=C(C=CC=C8Cl)N67)C=N5)CC4)=NO3)C(C)C)C=C2)SC=N1	C52H55ClN8O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-943K7N	WO2024064328A1_B97	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](C3=CC(OCCCCN4C=C(C5=CC6=C(C=C5)C(C)(C)C5=NC(=O)C7=C(C=CC=C7Cl)N56)C=N4)=NO3)C(C)C)C=C2)SC=N1	C49H51ClN8O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-RITXQW	WO2024064328A1_B98	(2S,4R)-1-[2-[3-[4-[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-8-yl)piperidin-1-yl]butoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(OCCCCN4CCC(C5=CC=CC6=C5C(C)(C)C5=NC(=O)C7=C(C=CC=C7Cl)N56)CC4)=NO3)C(C)C)C=C2)SC=N1	C51H58ClN7O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-T3QOYO	WO2024064328A1_B99	(2S,4R)-1-[2-[3-[4-[4-(4-chloro-7,7-dimethyl-5-oxoindolo[1,2-a]quinazolin-9-yl)pyrazol-1-yl]butoxy]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(C3=CC(OCCCCN4C=C(C5=CC6=C(C=C5)N5C(=NC(=O)C7=C5C=CC=C7Cl)C6(C)C)C=N4)=NO3)C(C)C)C=C2)SC=N1	C49H51ClN8O6S	SMARCA2;SMARCA4	P51531/P51532	VHL	WO-2024064328-A1
TPD-8H7X20	WO2024083256A1_100	.	C#CC1=C(F)C=CC2=CC(OC(=O)NC)=CC(C3=C(F)C4=C(C=N3)C(N3CCC[C@@](C)(O)C3)NC(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(Cl)C=C6)CC7)CC5)CC3)=N4)=C21	C58H67ClF2N10O7	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-442RHP	WO2024083256A1_101	.	C#CC1=C(F)C=CC2=CC(OCCOC)=CC(C3=C(F)C4=C(C=N3)C(N3CCC[C@@](C)(O)C3)=NC(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(Cl)C=C6)CC7)CC5)CC3)=N4)=C21	C59H68ClF2N9O7	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-1Z5DBK	WO2024083256A1_102	.	C#CC1=C(F)C=CC2=CC(O)=CC(C3CC4N=C(OCC5(CN6CCN(CC7CCC8(CC7)CCN(C(=O)C7=CC(N9CCC(=O)NC9=O)=C(Cl)C=C7)CC8)CC6)CC5)N=C(N5CCC[C@@](C)(O)C5)C4CO3)=C21	C56H68ClFN8O7	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-XRHH1B	WO2024083256A1_103	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=C1OC)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCN(CC5CCC6(CC5)CCN(C(=O)C5=CC(N7CCC(=O)NC7=O)=C(Cl)C=C5)CC6)CC4)CC1)=N3)=CC(O)=C2	C58H65ClF2N8O7	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-9V8FWP	WO2024083256A1_104	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=C1OCC)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCN(CC5CCC6(CC5)CCN(C(=O)C5=CC(N7CCC(=O)NC7=O)=C(Cl)C=C5)CC6)CC4)CC1)=N3)=CC(O)=C2	C59H67ClF2N8O7	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-E54M6E	WO2024083256A1_105	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=C1F)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCN(CC5CCC6(CC5)CCN(C(=O)C5=CC(N7CCC(=O)NC7=O)=C(Cl)C=C5)CC6)CC4)CC1)=N3)=CC(O)=C2	C57H62ClF3N8O6	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-MP08UN	WO2024083256A1_106	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=C(C=C1Cl)C(N1CCC[C@@](C)(O)C1)=NC(OCC1(CN4CCN(CC5CCC6(CC5)CCN(C(=O)C5=CC(N7CCC(=O)NC7=O)=C(Cl)C=C5)CC6)CC4)CC1)=N3)=CC(O)=C2	C57H62Cl2F2N8O6	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-4XRC8O	WO2024083256A1_107	.	C#CC1=CC=CC2=CC(O)=CC(N3CCC4=C(C3)N=C(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(OC)C=C6)CC7)CC5)CC3)N=C4N3CCC[C@@](C)(O)C3)=C12	C57H71N9O7	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-L9EIQV	WO2024083256A1_108	.	C#CC1=CC=CC2=CC(O)=CC(N3CCC4=C(C3)N=C(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(C)C=C6)CC7)CC5)CC3)N=C4N3CCC[C@@](C)(O)C3)=C12	C57H71N9O6	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-XZ5Z9S	WO2024083256A1_109	.	C#CC1=CC=CC2=CC(O)=CC(N3CCC4=C(C3)N=C(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(Cl)C=C6)CC7)CC5)CC3)N=C4N3CCC[C@@](C)(O)C3)=C12	C56H68ClN9O6	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-DEMSHA	WO2024083256A1_110	.	C#CC1=CC=CC2=CC(O)=CC(N3CCC4=C(C3)N=C(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(F)C=C6)CC7)CC5)CC3)N=C4N3CCC[C@@](C)(O)C3)=C12	C56H68FN9O6	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-UL5W28	WO2024083256A1_112	.	CCC1=CC=CC2=CC(O)=CC(N3CCC4=C(C3)N=C(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(C)C=C6)CC7)CC5)CC3)N=C4N3CCC[C@@](C)(O)C3)=C21	C57H75N9O6	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-IPBCU4	WO2024083256A1_113	.	CCC1=CC=CC2=CC(O)=CC(N3CCC4=C(C3)N=C(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(Cl)C=C6)CC7)CC5)CC3)N=C4N3CCC[C@@](C)(O)C3)=C21	C56H72ClN9O6	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-FT4M6Q	WO2024083256A1_114	.	C#CC1=C(F)C=CC2=CC(O)=CC(N3CCC4=C(C3)N=C(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(OC)C=C6)CC7)CC5)CC3)N=C4N3CCC[C@@](C)(O)C3)=C21	C57H70FN9O7	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-Y6UCGA	WO2024083256A1_115	.	C#CC1=C(F)C=CC2=CC(O)=CC(N3CCC4=C(C3)N=C(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(C)C=C6)CC7)CC5)CC3)N=C4N3CCC[C@@](C)(O)C3)=C21	C57H70FN9O6	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-4U046F	WO2024083256A1_116	.	C#CC1=C(F)C=CC2=CC(O)=CC(N3CCC4=C(C3)N=C(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(Cl)C=C6)CC7)CC5)CC3)N=C4N3CCC[C@@](C)(O)C3)=C21	C56H67ClFN9O6	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-975JW5	WO2024083256A1_117	.	C#CC1=C(F)C=CC2=CC(O)=CC(N3CCC4=C(C3)N=C(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(F)C=C6)CC7)CC5)CC3)N=C4N3CCC[C@@](C)(O)C3)=C21	C56H67F2N9O6	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-QI1UTI	WO2024083256A1_118	.	C#CC1=CC=CC2=CC(O)=CC(C(=O)N3CC4=C(C3)C(N3CCC[C@@](C)(O)C3)=NC(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(OC)C=C6)CC7)CC5)CC3)=N4)=C12	C57H69N9O8	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-LM0F69	WO2024083256A1_119	.	C#CC1=CC=CC2=CC(O)=CC(C(=O)N3CC4=C(C3)C(N3CCC[C@@](C)(O)C3)=NC(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(C)C=C6)CC7)CC5)CC3)=N4)=C12	C57H69N9O7	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-0W0H44	WO2024083256A1_120	.	C#CC1=CC=CC2=CC(O)=CC(C(=O)N3CC4=C(C3)C(N3CCC[C@@](C)(O)C3)=NC(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(CI)C=C6)CC7)CC5)CC3)=N4)=C12	C57H68IN9O7	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-AZCH47	WO2024083256A1_121	.	CCC1=CC=CC2=CC(O)=CC(C(=O)N3CC4=C(C3)C(N3CCC[C@@](C)(O)C3)=NC(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(C)C=C6)CC7)CC5)CC3)=N4)=C21	C57H73N9O7	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-KPNKT8	WO2024083256A1_122	.	CCC1=CC=CC2=CC(O)=CC(C(=O)N3CC4=C(C3)C(N3CCC[C@@](C)(O)C3)=NC(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(Cl)C=C6)CC7)CC5)CC3)=N4)=C21	C56H70ClN9O7	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-KYQEH6	WO2024083256A1_123	.	C#CC1=C(F)C=CC2=CC(O)=CC(C(=O)N3CC4=C(C3)C(N3CCC[C@@](C)(O)C3)=NC(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(OC)C=C6)CC7)CC5)CC3)=N4)=C21	C57H68FN9O8	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-QG5IBG	WO2024083256A1_124	.	C#CC1=C(F)C=CC2=CC(O)=CC(C(=O)N3CC4=C(C3)C(N3CCC[C@@](C)(O)C3)=NC(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(C)C=C6)CC7)CC5)CC3)=N4)=C21	C57H68FN9O7	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-NEGFEI	WO2024083256A1_125	.	C#CC1=C(F)C=CC2=CC(O)=CC(C(=O)N3CC4=C(C3)C(N3CCC[C@@](C)(O)C3)=NC(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(Cl)C=C6)CC7)CC5)CC3)=N4)=C21	C56H65ClFN9O7	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-EBUPH8	WO2024083256A1_126	.	C#CC1=C(F)C=CC2=CC(O)=CC(C(=O)N3CC4=C(C3)C(N3CCC[C@@](C)(O)C3)=NC(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(F)C=C6)CC7)CC5)CC3)=N4)=C21	C56H65F2N9O7	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-869LRU	WO2024083256A1_127	.	C=CC1=CC=CC2=CC(O)=CC(C3CC4=C(CO3)C(N3CCC[C@@](C)(O)C3)=NC(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(OC)C=C6)CC7)CC5)CC3)=N4)=C12	C57H72N8O8	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-Z0CLMR	WO2024083256A1_128	.	C#CC1=CC=CC2=CC(O)=CC(C3CC4=C(CO3)C(N3CCC[C@@](C)(O)C3)=NC(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(C)C=C6)CC7)CC5)CC3)=N4)=C12	C57H70N8O7	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-OZJ0XA	WO2024083256A1_129	.	C#CC1=CC=CC2=CC(O)=CC(C3CC4=C(CO3)C(N3CCC[C@@](C)(O)C3)=NC(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(Cl)C=C6)CC7)CC5)CC3)=N4)=C12	C56H67ClN8O7	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-5XTDOZ	WO2024083256A1_130	.	CCC1=CC=CC2=CC(O)=CC(C3CC4=C(CO3)C(N3CCC[C@@](C)(O)C3)=NC(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(OC)C=C6)CC7)CC5)CC3)=N4)=C21	C57H74N8O8	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-QOGI7K	WO2024083256A1_131	.	CCC1=CC=CC2=CC(O)=CC(C3CC4=C(CO3)C(N3CCC[C@@](C)(O)C3)=NC(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(C)C=C6)CC7)CC5)CC3)=N4)=C21	C57H74N8O7	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-XNJK8C	WO2024083256A1_134	.	CCC1=CC=CC2=CC(O)=CC(C3CC4=C(CO3)C(N3CCC[C@@](C)(O)C3)=NC(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(Cl)C=C6)CC7)CC5)CC3)=N4)=C21	C56H71ClN8O7	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-3KSC1A	WO2024083256A1_135	.	C#CC1=C(F)C=CC2=CC(O)=CC(C3CC4=C(CO3)C(N3CCC[C@@](C)(O)C3)=NC(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(OC)C=C6)CC7)CC5)CC3)=N4)=C21	C57H69FN8O8	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-9G0E3H	WO2024083256A1_136	.	C#CC1=C(F)C=CC2=CC(O)=CC(C3CC4=C(CO3)C(N3CCC[C@@](C)(O)C3)=NC(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(C)C=C6)CC7)CC5)CC3)=N4)=C21	C57H69FN8O7	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-NCZ59S	WO2024083256A1_137	.	C#CC1=C(F)C=CC2=CC(O)=CC(C3CC4=C(CO3)C(N3CCC[C@@](C)(O)C3)=NC(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(Cl)C=C6)CC7)CC5)CC3)=N4)=C21	C56H66ClFN8O7	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-4ZP94Q	WO2024083256A1_138	.	COC1=C(N2CCC(=O)NC2=O)C=C(C(=O)N2CCC3(CCC(CN4CCN(CC5(COC6=NC7=C(CCN(C8=C(C9CC9)C(Cl)=CC(O)=C8)C7)C(N7CCC[C@@](C)(O)C7)=N6)CC5)CC4)CC3)CC2)C=C1	C54H72ClN9O7	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-QDPBXX	WO2024083256A1_139	.	COC1=C(N2CCC(=O)NC2=O)C=C(C(=O)N2CCC3(CCC(CN4CCN(CC5(COC6=NC7=C(CN(C(=O)C8=C(C9CC9)C(Cl)=CC(O)=C8)C7)C(N7CCC[C@@](C)(O)C7)=N6)CC5)CC4)CC3)CC2)C=C1	C54H70ClN9O8	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-QC7H9O	WO2024083256A1_140	.	C#CC1=CC=CC2=CC(O)=CC(N3CCC4=C(C3)N=C(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(OC)C=C6)CC7)CC5)CC3)N=C4N3CCCN4N=C(C(=O)N(C)C)C=C4C3)=C12	C61H74N12O7	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-GO9WJF	WO2024083256A1_141	.	C#CC1=CC=CC2=CC(O)=CC(N3CCC4=C(C3)N=C(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(OC)C=C6)CC7)CC5)CC3)N=C4N3CC4C(=O)NC(=O)C4C3)=C12	C57H66N10O8	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-X8G8W8	WO2024083256A1_142	.	COCC1=C(N2CCC(=O)NC2=O)C=C(C(=O)N2CCC3(CCC(CN4CCN(CC5(COC6=NC7=C(C=NC(C8=C(C#N)C(Cl)=CC(O)=C8)=C7F)C(N7CCC[C@@](C)(O)C7)=N6)CC5)CC4)CC3)CC2)C=C1	C53H64ClFN10O7	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-2BV1V3	WO2024083256A1_143	.	C#CC1=CC=CC2=CC(O)=CC(C3=C(F)C4=C(C=N3)C(N3CCOC[C@@](C)(O)C3)=NC(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(OC)C=C6)CC7)CC5)CC3)=N4)=C12	C57H66FN9O8	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-X2KUG1	WO2024083256A1_144	.	C#CC1=CC=CC2=CC(O)=CC(C3=C(F)C4=C(C=C3)C(N3CCC[C@@](C)(O)C3)=NC(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(Cl)C=C6)CC7)CC5)CC3)=N4)=C12	C57H64ClFN8O6	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-O3SLY5	WO2024083256A1_145	.	C#CC1=CC=CC2=CC(C)=CC(C3=C(F)C4=C(C=C3)C(N3CCC[C@@](C)(O)C3)=NC(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(C)C=C6)CC7)CC5)CC3)=N4)=C12	C59H69FN8O5	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-I7WNOM	WO2024083256A1_146	.	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=C(C=N3)C(N3CCC[C@@](C)(N)C3)=NC(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(Cl)C=C6)CC7)CC5)CC3)=N4)=C21	C56H63ClF2N10O5	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-OO0O54	WO2024083256A1_147	.	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=C(C=C3)C(N3CCC[C@@](C)(N)C3)=NC(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(Cl)C=C6)CC7)CC5)CC3)=N4)=C21	C57H64ClF2N9O5	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-PJUTGR	WO2024083256A1_148	.	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=C(C=N3)C(N3CCNC[C@@](C)(O)C3)=NC(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(Cl)C=C6)CC7)CC5)CC3)=N4)=C21	C56H63ClF2N10O6	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-Q2CRCY	WO2024083256A1_149	.	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=C(C=C3)C(N3CCNC[C@@](C)(O)C3)=NC(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(Cl)C=C6)CC7)CC5)CC3)=N4)=C21	C57H64ClF2N9O6	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-J4UHZ7	WO2024083256A1_150	.	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=C(C=C3)C(N3CCCNCC3)=NC(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(Cl)C=C6)CC7)CC5)CC3)=N4)=C21	C56H62ClF2N9O5	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-ZMXVFU	WO2024083256A1_151	.	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=C(C=N3)C(N3CCCNCC3)=NC(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(Cl)C=C6)CC7)CC5)CC3)=N4)=C21	C55H61ClF2N10O5	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-NA64YW	WO2024083256A1_152	.	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=C(C=N3)C(N3CCC[C@@](C)(O)C3)=NC(OCC(C)CN3CCN(CC5CCC6(CC5)CCN(C(=O)C5=CC(N7CCC(=O)NC7=O)=C(Cl)C=C5)CC6)CC3)=N4)=C21	C55H62ClF2N9O6	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-46J7D5	WO2024083256A1_153	.	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=C(C=N3)C(N3CCC[C@@](C)(O)C3)=NC(OCC(C)CN3CCN(CC5CCC6(CC5)CCN(C(=O)C5=CC(N7CCC(=O)NC7=O)=C(C)C=C5)CC6)CC3)=N4)=C21	C56H65F2N9O6	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-4BYZWS	WO2024083256A1_154	.	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=C(C=N3)C(N3CCC[C@@](C)(O)C3)=NC(OCC(C)CN3CCN(CC5CCC6(CC5)CCN(C(=O)C5=CC(N7CCC(=O)NC7)=C(OC)C=C5)CC6)CC3)=N4)=C21	C56H67F2N9O6	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-04M5QG	WO2024083256A1_155	.	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=C(C=N3)C(N3CCC[C@@](C)(O)C3)=NC(OC[C@@H](C)CN3CCN(CC5CCC6(CC5)CCN(C(=O)C5=CC(N7CCC(=O)NC7=O)=C(OC)C=C5)CC6)CC3)=N4)=C21	C56H65F2N9O7	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-OQYPTH	WO2024083256A1_156	.	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=C(C=N3)C(N3CCCC(C)(N)C3)=NC(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(Cl)C=C6)CC7)CC5)CC3)=N4)=C21	C56H63ClF2N10O5	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-FDE2TP	WO2024083256A1_157	.	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=C(C=N3)C(N3CCOC[C@@](C)(O)C3)=NC(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(Cl)C=C6)CC7)CC5)CC3)=N4)=C21	C56H62ClF2N9O7	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-Q26FTF	WO2024083256A1_158	.	COC1=C(N2CCC(=O)NC2=O)C=C(C(=O)N2CCC3(CCC(CN4CCN(CC5(COC6=NC7=C(CN(C(=O)C8=C9C(I)=CC=CC9=CC(O)=C8)C7)C(N7CCC[C@@](C)(O)C7)=N6)CC5)CC4)CC3)CC2)C=C1	C55H68IN9O8	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-GGQCK8	WO2024083256A1_159	.	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=C(C=N3)C(N3CCCNCC3)=NC(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(OC)C=C6)CC7)CC5)CC3)=N4)=C21	C56H64F2N10O6	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-ZCHGG9	WO2024083256A1_160	.	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=C(C=N3)C(N3CCC[C@@](C)(O)C3)=NC(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(OC)C=C6F)CC7)CC5)CC3)=N4)=C21	C57H64F3N9O7	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-PLPHXK	WO2024083256A1_161	.	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=C(C=N3)C(N3CCC[C@@](C)(O)C3)=NC(OCC3(CN5CCN(CC6CCC7(CCN(C(=O)C8=CC(N9CCC(=O)NC9=O)=C(OC)C=C8)CC7)OC6)CC5)CC3)=N4)=C21	C56H63F2N9O8	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-OJAENV	WO2024083256A1_171	.	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=C(C=N3)C(N3CCC[C@@](C)(O)C3)=NC(OCC3(CN5CCN(CC6CCC7(CCN(C(=O)C8=CC(N9CCC(=O)NC9=O)=C(OC)C=C8)CC7)CO6)CC5)CC3)=N4)=C21	C56H63F2N9O8	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-RQ2A63	WO2024083256A1_172	.	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=C(C=N3)C(N3CCC[C@@](C)(O)C3)=NC(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(OC)C=C6)CC7)C(F)(F)C5)CC3)=N4)=C21	C57H63F4N9O7	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-PBF5WR	WO2024083256A1_173	.	C#CC1=C(F)C=CC2=CC(C)=CC(C3=C(F)C4=C(C=N3)C(N3CCC[C@@](C)(O)C3)=NC(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(OC)C=C6)CC7)C(F)C5)CC3)=N4)=C21	C58H66F3N9O6	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-BVS0RO	WO2024083256A1_174	.	C=CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=C(C=N3)C(N3CCC[C@@](C)(O)C3)=NC(OC[C@@H](C)CN3CCN(CC5CCC6(CC5)CCN(C(=O)C5=CC(N7CCC(=O)NC7=O)=C(C)C=C5)CC6)CC3)=N4)=C21	C56H67F2N9O6	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-MCOMT8	WO2024083256A1_175	.	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=C(C=N3)C(N3CCC[C@@](C)(O)C3)=NC(OC[C@@H](C)CN3CCN(CC5CCC6(CC5)CCN(C(=O)C5=CC(N7CCC(=O)NC7=O)=C(Cl)C=C5)CC6)CC3)=N4)=C21	C55H62ClF2N9O6	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-1NL74X	WO2024083256A1_51	.	CCC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=C(C=N3)C(N3CCC[C@@](C)(O)C3)=NC(OCC3(CN5CCC(COCCC6CCN(C(=O)C7=CC(N8CCC(=O)NC8=O)=C(Cl)C=C7)CC6)CC5)CC3)=N4)=C21	C54H63ClF2N8O7	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-OJZWSL	WO2024083256A1_52	.	CCC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=C(C=N3)C(N3CCCN5NC(C(=O)NC)C=C5C3)=NC(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(C)C=C6)CC7)CC5)CC3)=N4)=C21	C60H72F2N12O6	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-U85Y94	WO2024083256A1_53	.	CCC1=C(F)C=CC2=CC(O)=CC(N3CCC4=C(C3)N=C(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(C)C=C6)CC7)CC5)CC3)NC4N3CCCN4N=C(C(=O)N(C)C)C=C4C3)=C21	C61H79FN12O6	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-ECABFK	WO2024083256A1_54	.	CCC1=C(F)C=CC2=CC(O)=CC(N3CCC4=C(C3)N=C(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(C)C=C6)CC7)CC5)CC3)N=C4N3CC4C(=O)NC(=O)C4C3)=C21	C57H69FN10O7	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-1NFE22	WO2024083256A1_55	.	CCC1=C(F)C=CC2=CC(O)=CC(N3CCC4=C(C3)N=C(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(C)C=C6)CC7)CC5)CC3)N=C4N3CCCC4(CNC(=O)N4)C3)=C21	C58H74FN11O6	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-IKASE6	WO2024083256A1_56	.	C[C@@]1(O)CCCN(C2=NC(OCC3(CN4CCC(CCOCC5CCN(C(=O)C6=CC(N7CCC(=O)NC7=O)=C(Cl)C=C6)CC5)CC4)CC3)=NC3=C2CCC2(CCCC4=C2C=C(O)C=C4)C3)C1	C52H68ClN7O7	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-5UJL2I	WO2024083256A1_57	.	C[C@@]1(O)CCCN(C2=NC(OCC3(CN4CCC(CCOCC5CCN(C(=O)C6=CC(N7CCC(=O)NC7=O)=C(Cl)C=C6)CC5)CC4)CC3)=NC3=C2CCC2(CCC4=C2C=C(O)C=C4)C3)C1	C51H66ClN7O7	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-CPI3FZ	WO2024083256A1_58	.	C[C@@H]1C[C@H]1C1=C(C2=C(F)C3=C(C=N2)C(N2CCC[C@@](C)(O)C2)=NC(OCC2(CN4CCN(CC5CCC6(CC5)CCN(C(=O)C5=CC(N7CCC(=O)NC7=O)=C(Cl)C=C5)CC6)CC4)CC2)=N3)C=C(O)C=C1Cl	C54H66Cl2FN9O6	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-UN54OR	WO2024083256A1_59	.	CC1=C(N2CCC(=O)NC2=O)C=C(C(=O)N2CCC3(CCC(CN4CCN(CC5(COC6=NC7=C(C=NC(C8=C(C(F)(F)F)C(Cl)=CC(O)=C8)=C7F)C(N7CCC[C@@](C)(O)C7)=N6)CC5)CC4)CC3)CC2)C=C1	C52H62ClF4N9O6	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-YK0WBI	WO2024083256A1_62	.	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=C(C=N3)C(N3CCC[C@@](C)(O)C3)=NC(OCC3(CN5CCN(CCC6CCN(C(=O)C7=CC=C(CI)C(N8CCC(=O)NC8=O)=C7)CC6)CC5)CC3)=N4)=C21	C53H58F2IN9O6	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-1D4UX0	WO2024083256A1_63	.	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=C(C=N3)C(N3CCC[C@@](C)(O)C3)=NC(OCC3(CN5CCN(CCCC6CCC7(CC6)CCN(C(=O)C6=CC=C(Cl)C(N8CCC(=O)NC8=O)=C6)CC7)CC5)CC3)=N4)=C21	C58H66ClF2N9O6	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-D9TBVI	WO2024083256A1_65	.	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=C(C=N3)C(N3CCC[C@@](C)(O)C3)=NC(OCC3(CN5CCN(CCCCC6CCC7(CC6)CCN(C(=O)C6=CC=C(Cl)C(N8CCC(=O)NC8=O)=C6)CC7)CC5)CC3)=N4)=C21	C59H68ClF2N9O6	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-HA6L0D	WO2024083256A1_66	.	CC1=C(C(F)(F)F)C(C2=C(F)C3=C(C=C2Cl)C(N2CCC[C@@](C)(O)C2)=NC(OCC2(CN4CCC(CCOCC5CCN(C(=O)C6=CC(N7CCC(=O)NC7=O)=C(Cl)C=C6)CC5)CC4)CC2)=N3)=NC(N)=C1	C50H59Cl2F4N9O6	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-EVW6YM	WO2024083256A1_68	.	CCC1=CC=CC2=CC(O)=CC(N3CCC4=C(C3)N=C(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(OC)C=C6)CC7)CC5)CC3)N=C4N3CCC[C@@](C)(O)C3)=C21	C57H75N9O7	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-EK1QFA	WO2024083256A1_69	.	CCC1=CC=CC2=CC(O)=CC(C(=O)N3CC4=C(C3)C(N3CCC[C@@](C)(O)C3)=NC(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(O[Mc])C=C6)CC7)CC5)CC3)=N4)=C21	C56H70McN9O8	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-LWRHOS	WO2024083256A1_70	.	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=C(C=N3)C(N3CCC[C@@](C)(O)C3)=NC(OCC3(CN5CCN(CCCC6CCN(C(=O)C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)CC3)=N4)=C21	C56H59F2N9O8	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-QDARIZ	WO2024083256A1_71	.	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=C(C=N3)C(N3CCC[C@@](C)(O)C3)=NC(OCC3(CN5CCN(CC6CCN(C(=O)C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)CC3)=N4)=C21	C54H55F2N9O8	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-705H5D	WO2024083256A1_73	.	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=C(C=N3)C(N3CCC[C@@](C)(O)C3)=NC(OCC3(CN5CCN(CCC6CCN(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)CC3)=N4)=C21	C54H57F2N9O7	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-DGAOW7	WO2024083256A1_74	.	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=C(C=N3)C(N3CCCC5(CC(=O)N5)C3)=NC(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(C)C=C6)CC7)CC5)CC3)=N4)=C21	C58H64F2N10O6	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-2AKO87	WO2024083256A1_75	.	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=C(C=N3)C(N3CC5CC(C3)[C@H](O)C5)=NC(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(C)C=C6)CC7)CC5)CC3)=N4)=C21	C58H65F2N9O6	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-VKJHGK	WO2024083256A1_76	.	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=C(C=N3)C(N3CCOC[C@@](C)(O)C3)=NC(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(C)C=C6)CC7)CC5)CC3)=N4)=C21	C57H65F2N9O7	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-UP15HD	WO2024083256A1_77	.	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=C(C=N3)C(N3CCCN5N=C(C(=O)N(C)C)C=C5C3)=NC(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(Cl)C=C6)CC7)CC5)CC3)=N4)=C21	C60H65ClF2N12O6	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-HBEVNW	WO2024083256A1_78	.	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=C(C=N3)C(N3CCC[C@@H](N)C3)=NC(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(C)C=C6)CC7)CC5)CC3)=N4)=C21	C56H64F2N10O5	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-MHKO23	WO2024083256A1_79	.	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=C(C=N3)C(N3CC[C@@H](O)C3)=NC(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(C)C=C6)CC7)CC5)CC3)=N4)=C21	C55H61F2N9O6	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-V5G40Y	WO2024083256A1_80	.	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=C(C=N3)C(N3CC5C(=O)NC(=O)C5C3)=NC(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(C)C=C6)CC7)CC5)CC3)=N4)=C21	C57H60F2N10O7	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-OGG9XN	WO2024083256A1_81	.	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=C(C=N3)C(C3CCC[C@@](C)(O)C3)=NC(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(OC)C=C6)CC7)CC5)CC3)=N4)=C21	C58H66F2N8O7	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-GOINDY	WO2024083256A1_82	.	CCC1=CC=CC2=CC(O)=CC(C3=C(F)C4=C(C=N3)C(N3CCC[C@@](C)(O)C3)=NC(OCC3(CN5CCN(CC6CCN(C(=O)COC7=CC=CC(N8CCC(=O)NC8=O)=C7C)CC6)CC5)CC3)=N4)=C21	C53H64FN9O7	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-JHEN8M	WO2024083256A1_83	.	CCC1=CC=CC2=CC(O)=CC(C3=C(F)C4=C(C=N3)C(N3CCC[C@@](C)(O)C3)=NC(OCC3(CN5CCN(CC6CCN(C(=O)COC7=CC=C(C)C(N8CCC(=O)NC8=O)=C7)CC6)CC5)CC3)=N4)=C21	C53H64FN9O7	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-2I5E58	WO2024083256A1_84	.	CCC1=CC=CC2=CC(O)=CC(C3=C(F)C4=C(C=N3)C(C3CCC[C@@](C)(O)C3)=NC(OCC3(CN5CCN(CC6CCN(CC#CC7=CC=CC(N8CCC(=O)NC8=O)=C7C)CC6)CC5)CC3)=N4)=C21	C55H65FN8O5	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-F4SCN6	WO2024083256A1_85	.	CCC1=CC=CC2=CC(O)=CC(C3=C(F)C4=C(C=N3)C(N3CCC[C@@](C)(O)C3)=NC(OCC3(CN5CCN(CC6CCN(CC#CC7=CC=C(C)C(N8CCC(=O)NC8=O)=C7)CC6)CC5)CC3)=N4)=C21	C54H64FN9O5	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-NL1XZ1	WO2024083256A1_87	1-[5-[9-[[4-[[1-[[4-[Cyclopropyl(methyl)amino]-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperazin-1-yl]methyl]-3-azaspiro[5.5]undecane-3-carbonyl]-2-methoxyphenyl]-1,3-diazinane-2,4-dione	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=C(C=N3)C(N(C)C3CC3)=NC(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(OC)C=C6)CC7)CC5)CC3)=N4)=C21	C55H61F2N9O6	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-ZLAAKS	WO2024083256A1_88	.	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=C(C=N3)C(N(C)[C@H]3C[C@@H]3F)=NC(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(OC)C=C6)CC7)CC5)CC3)=N4)=C21	C55H60F3N9O6	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-KXHJFR	WO2024083256A1_89	.	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=C(C=N3)C(N(C)C3C[C@H]3F)=NC(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(OC)C=C6)CC7)CC5)CC3)=N4)=C21	C55H60F3N9O6	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-2N2D6H	WO2024083256A1_90	.	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=C(C=C3)C(N(C)C3CC3)=NC(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(OC)C=C6)CC7)CC5)CC3)=N4)=C21	C56H62F2N8O6	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-YAOOLR	WO2024083256A1_93	.	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=C(C=N3)C(N3CC5COC(C5)C3)=NC(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(C)C=C6)CC7)CC5)CC3)=N4)=C21	C57H63F2N9O6	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-2XMJ6R	WO2024083256A1_94	.	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=C(C=N3)C(N3CCOCC(F)(F)C3)=NC(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(C)C=C6)CC7)CC5)CC3)=N4)=C21	C56H61F4N9O6	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-S12XZL	WO2024083256A1_95	.	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=C(C=N3)C(NCCSC)=NC(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(OC)C=C6)CC7)CC5)CC3)=N4)=C21	C54H61F2N9O6S	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-R4AQK8	WO2024083256A1_96	.	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=C(C=N3)C(N3CCCCC(F)(F)C3)=NC(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(C)C=C6)CC7)CC5)CC3)=N4)=C21	C57H63F4N9O5	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-275PAF	WO2024083256A1_97	.	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=C(C=N3)C(N3CCCSCC3)=NC(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(C)C=C6)CC7)CC5)CC3)=N4)=C21	C56H63F2N9O5S	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-VVRI8V	WO2024083256A1_98	.	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=C(C=N3)C(N3CCCCC(F)C3)=NC(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(C)C=C6)CC7)CC5)CC3)=N4)=C21	C57H64F3N9O5	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-RA54SF	WO2024083256A1_99	.	C#CC1C2=C(C3=C(F)C4=C(C=N3)C(N3CCCC(F)CC3)=NC(OCC3(CC5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(C)C=C6)CC7)CC5)CC3)=N4)C=C(O)C=C2C=CC1F	C58H67F3N8O5	KRAS	P01116	CRBN	WO-2024083256-A1
TPD-DLUAU1	WO2024099441A1_1	.	CC1=C(C2=CC3=C(N=C2)C2=NN(C)C(C(=O)NCCOCCOCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)=C2N3C(C2=C(F)C=CC=N2)C2CCOCC2)N(C)NN1	C44H49FN12O8	BRD2;BRD3;BRD4;BRDT	P25440/Q15059/O60885/Q58F21	CRBN	WO-2024099441-A1
TPD-37DH4K	WO2024099441A1_10	.	CC1=C(C2=CC3=C(N=C2)C2=NN(C)C(C(=O)NCCCC(C)CCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)=C2N3C(C2=C(F)C=CC=N2)C2CCOCC2)N(C)N=N1	C46H51FN12O6	BRD2;BRD3;BRD4;BRDT	P25440/Q15059/O60885/Q58F21	CRBN	WO-2024099441-A1
TPD-T44YJX	WO2024099441A1_11	.	CC1=C(C2=CC3=C(N=C2)C2=NN(C)C(C(=O)NCCCCCCCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)=C2N3C(C2=CC=CC=C2)C2CCOCC2)N(C)N=N1	C47H53N11O6	BRD2;BRD3;BRD4;BRDT	P25440/Q15059/O60885/Q58F21	CRBN	WO-2024099441-A1
TPD-33MZWY	WO2024099441A1_12	.	CC1=C(C2=CC3=C(N=C2)C2=NN(C)C(C(=O)NCCCCCCCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)=C2N3C(C2=C(F)C=CC=N2)C2CCOCC2)N(C)N=N1	C46H51FN12O6	BRD2;BRD3;BRD4;BRDT	P25440/Q15059/O60885/Q58F21	CRBN	WO-2024099441-A1
TPD-KMMCC5	WO2024099441A1_14	.	CC1=C(C2=CC3=C(N=C2)C2=NN(C)C(C(=O)NCCCCCCCCNC4=C5CN(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)=C2N3C(C2=C(F)C=CC=N2)C2CCOCC2)N(C)N=N1	C46H53FN12O5	BRD2;BRD3;BRD4;BRDT	P25440/Q15059/O60885/Q58F21	CRBN	WO-2024099441-A1
TPD-YGD5OY	WO2024099441A1_15	.	CC1=C(C2=CC3=C(N=C2)C2=NN(C)C(C(=O)NCCCCCCCCNC4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)=C2N3C(C2=C(F)C=CC=N2)C2CCOCC2)N(C)N=N1	C46H51FN12O6	BRD2;BRD3;BRD4;BRDT	P25440/Q15059/O60885/Q58F21	CRBN	WO-2024099441-A1
TPD-K7XY0E	WO2024099441A1_16	.	CC1=C(C2=CC3=C(N=C2)C2=C(C(C(=O)NCCOCCOCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)=NN2C)N3C(C2=C(F)C=CC=N2)C2CCOCC2)N(C)N=N1	C44H47FN12O8	BRD2;BRD3;BRD4;BRDT	P25440/Q15059/O60885/Q58F21	CRBN	WO-2024099441-A1
TPD-0RQ8W5	WO2024099441A1_17	.	CC1=C(C2=CC3=C(N=C2)C2=C(C(C(=O)NCCOCCOCCOC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)=NN2C)N3C(C2=C(F)C=CC=N2)C2CCOCC2)N(C)N=N1	C44H46FN11O9	BRD2;BRD3;BRD4;BRDT	P25440/Q15059/O60885/Q58F21	CRBN	WO-2024099441-A1
TPD-KINV4B	WO2024099441A1_18	.	CC1=C(C2=CC3=C(N=C2)C2=C(C(C(=O)NCCCCCCCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)=NN2C)N3C(C2=C(F)C=CC=N2)C2CCOCC2)N(C)N=N1	C46H51FN12O6	BRD2;BRD3;BRD4;BRDT	P25440/Q15059/O60885/Q58F21	CRBN	WO-2024099441-A1
TPD-B1TE0S	WO2024099441A1_19	.	CC1=C(C2=CC3=C(N=C2)C2=C(C(C(=O)NCCOCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)=NN2C)N3C(C2=C(F)C=CC=N2)C2CCOCC2)N(C)N=N1	C42H43FN12O7	BRD2;BRD3;BRD4;BRDT	P25440/Q15059/O60885/Q58F21	CRBN	WO-2024099441-A1
TPD-W8G7SQ	WO2024099441A1_2	.	CC1=C(C2=CC3=C(N=C2)C2=NN(C)C(C(=O)NCCOCCOCCOC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)=C2N3C(C2=C(F)C=CC=N2)C2CCOCC2)N(C)NN1	C44H48FN11O9	BRD2;BRD3;BRD4;BRDT	P25440/Q15059/O60885/Q58F21	CRBN	WO-2024099441-A1
TPD-QJ2P6G	WO2024099441A1_20	.	CC1=C(C2=CC3=C(N=C2)C2=C(C(C(=O)NCCCCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)=NN2C)N3C(C2=C(F)C=CC=N2)C2CCOCC2)N(C)N=N1	C43H45FN12O6	BRD2;BRD3;BRD4;BRDT	P25440/Q15059/O60885/Q58F21	CRBN	WO-2024099441-A1
TPD-WNK8DD	WO2024099441A1_21	.	CC1=C(C2=CC3=C(N=C2)C2=C(C(COCCOCCOCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)=NN2C)N3C(C2=C(F)C=CC=N2)C2CCOCC2)N(C)N=N1	C44H48FN11O8	BRD2;BRD3;BRD4;BRDT	P25440/Q15059/O60885/Q58F21	CRBN	WO-2024099441-A1
TPD-LNUEJH	WO2024099441A1_22	.	CC1=C(C2=CC3=C(N=C2)C2=C(C(C(=O)NCCCCCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)=NN2C)N3C(C2=C(F)C=CC=N2)C2CCOCC2)N(C)N=N1	C44H47FN12O6	BRD2;BRD3;BRD4;BRDT	P25440/Q15059/O60885/Q58F21	CRBN	WO-2024099441-A1
TPD-S8BBJM	WO2024099441A1_23	.	CC1=C(C2=CC3=C(N=C2)C2=C(C(C(=O)NCCCCCCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)=NN2C)N3C(C2=C(F)C=CC=N2)C2CCOCC2)N(C)N=N1	C45H49FN12O6	BRD2;BRD3;BRD4;BRDT	P25440/Q15059/O60885/Q58F21	CRBN	WO-2024099441-A1
TPD-8S0M1G	WO2024099441A1_24	.	CC1=C(C2=CC3=C(N=C2)C2=C(C(C(=O)NCCCCCCCCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)=NC2C)N3C(C2=C(F)C=CC=N2)C2CCOCC2)N(C)N=N1	C48H54FN11O6	BRD2;BRD3;BRD4;BRDT	P25440/Q15059/O60885/Q58F21	CRBN	WO-2024099441-A1
TPD-GQOG3K	WO2024099441A1_25	.	CC1=C(C2=CC3=C(N=C2)C2=C(C(C(=O)NCCCC(C)CCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)=NN2C)N3C(C2=C(F)C=CC=N2)C2CCOCC2)N(C)N=N1	C46H51FN12O6	BRD2;BRD3;BRD4;BRDT	P25440/Q15059/O60885/Q58F21	CRBN	WO-2024099441-A1
TPD-795TMX	WO2024099441A1_28	.	CC1=C(C2=CC3=C(N=C2)C2=C(C=C(C(=O)NCCOCCOCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C2)N3C(C2=C(F)C=CC=N2)C2CCOCC2)N(C)N=N1	C46H47FN10O8	BRD2;BRD3;BRD4;BRDT	P25440/Q15059/O60885/Q58F21	CRBN	WO-2024099441-A1
TPD-2YTCI3	WO2024099441A1_29	.	CC1=C(C(C2CCOCC2)N2C3=C(C=CC(C(=O)NCCOCCOCCOC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)=C3)C3=C2C=C(C2=C(C)N=NN2C)C=N3)N=CC=C1	C47H49N9O9	BRD2;BRD3;BRD4;BRDT	P25440/Q15059/O60885/Q58F21	CRBN	WO-2024099441-A1
TPD-W932JR	WO2024099441A1_30	.	CC1=C(C2=CC3=C(N=C2)C2=C(C=C(C(=O)NCCCCCCCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C2)N3C(C2=C(F)C=CC=N2)C2CCOCC2)N(C)N=N1	C48H51FN10O6	BRD2;BRD3;BRD4;BRDT	P25440/Q15059/O60885/Q58F21	CRBN	WO-2024099441-A1
TPD-2GGTTS	WO2024099441A1_31	.	CC1=C(C2=CC3=C(N=C2)C2=C(C=C(C(=O)NCCOCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C2)N3C(C2=C(F)C=CC=N2)C2CCOCC2)N(C)N=N1	C44H43FN10O7	BRD2;BRD3;BRD4;BRDT	P25440/Q15059/O60885/Q58F21	CRBN	WO-2024099441-A1
TPD-UGTLCL	WO2024099441A1_32	.	CC1=C(C2=CC3=C(N=C2)C2=C(C=C(C(=O)NCCCCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C2)N3C(C2=C(F)C=CC=N2)C2CCOCC2)N(C)N=N1	C45H45FN10O6	BRD2;BRD3;BRD4;BRDT	P25440/Q15059/O60885/Q58F21	CRBN	WO-2024099441-A1
TPD-LLWOM2	WO2024099441A1_33	.	CC1=C(C2=CC3=C(N=C2)C2=C(C=C(COCCOCCOCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C2)N3C(C2=C(F)C=CC=N2)C2CCOCC2)N(C)N=N1	C46H48FN9O8	BRD2;BRD3;BRD4;BRDT	P25440/Q15059/O60885/Q58F21	CRBN	WO-2024099441-A1
TPD-ADNTX8	WO2024099441A1_34	.	CC1=C(C2=CC3=C(N=C2)C2=C(C=C(C(=O)NCCCCCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C2)N3C(C2=C(F)C=CC=N2)C2CCOCC2)N(C)N=N1	C46H47FN10O6	BRD2;BRD3;BRD4;BRDT	P25440/Q15059/O60885/Q58F21	CRBN	WO-2024099441-A1
TPD-RDCA5G	WO2024099441A1_35	.	CC1=C(C2=CC3=C(N=C2)C2=C(C=C(C(=O)NCCCCCCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C2)N3C(C2=C(F)C=CC=N2)C2CCOCC2)N(C)N=N1	C47H49FN10O6	BRD2;BRD3;BRD4;BRDT	P25440/Q15059/O60885/Q58F21	CRBN	WO-2024099441-A1
TPD-35RXX7	WO2024099441A1_36	.	CC1=C(C2=CC3=C(N=C2)C2=C(C=C(C(=O)NCCCCCCCCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C2)N3C(C2=C(F)C=CC=N2)C2CCOCC2)N(C)N=N1	C49H53FN10O6	BRD2;BRD3;BRD4;BRDT	P25440/Q15059/O60885/Q58F21	CRBN	WO-2024099441-A1
TPD-TW1VRW	WO2024099441A1_37	.	CC1=C(C2=CC3=C(N=C2)C2=C(C=C(C(=O)NCCCC(C)CCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C2)N3C(C2=C(F)C=CC=N2)C2CCOCC2)N(C)N=N1	C48H51FN10O6	BRD2;BRD3;BRD4;BRDT	P25440/Q15059/O60885/Q58F21	CRBN	WO-2024099441-A1
TPD-NTDYIX	WO2024099441A1_4	.	CC1=C(C2=CC3=C(N=C2)C2=NN(C)C(C(=O)NCCOCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)=C2N3C(C2=C(F)C=CC=N2)C2CCOCC2)N(C)N=N1	C42H43FN12O7	BRD2;BRD3;BRD4;BRDT	P25440/Q15059/O60885/Q58F21	CRBN	WO-2024099441-A1
TPD-8TIR1L	WO2024099441A1_41	.	CC1=C(C2=CC3=C(N=C2)C2=C(C=C(C(=O)NCCOCCOCCOC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C2)N3C(C2=C(F)C=CC=N2)C2CCOCC2)N(C)N=N1	C46H46FN9O9	BRD2;BRD3;BRD4;BRDT	P25440/Q15059/O60885/Q58F21	CRBN	WO-2024099441-A1
TPD-G8T2US	WO2024099441A1_5	.	CC1=C(C2=CC3=C(N=C2)C2=NN(C)C(C(=O)NCCCCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)=C2N3C(C2=C(F)C=CC=N2)C2CCOCC2)N(C)N=N1	C43H45FN12O6	BRD2;BRD3;BRD4;BRDT	P25440/Q15059/O60885/Q58F21	CRBN	WO-2024099441-A1
TPD-EL71JW	WO2024099441A1_6	.	CC1=C(C2=CC3=C(N=C2)C2=NN(C)C(COCCOCCOCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)=C2N3C(C2=C(F)C=CC=N2)C2CCOCC2)N(C)N=N1	C44H48FN11O8	BRD2;BRD3;BRD4;BRDT	P25440/Q15059/O60885/Q58F21	CRBN	WO-2024099441-A1
TPD-8D6LMM	WO2024099441A1_7	.	CC1=C(C2=CC3=C(N=C2)C2=NN(C)C(C(=O)NCCCCCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)=C2N3C(C2=C(F)C=CC=N2)C2CCOCC2)N(C)N=N1	C44H47FN12O6	BRD2;BRD3;BRD4;BRDT	P25440/Q15059/O60885/Q58F21	CRBN	WO-2024099441-A1
TPD-SIZIFB	WO2024099441A1_8	.	CC1=C(C2=CC3=C(N=C2)C2=NN(C)C(C(=O)NCCCCCCCNC4C=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C54)=C2N3C(C2=C(F)C=CC=N2)C2CCOCC2)N(C)N=N1	C45H51FN12O6	BRD2;BRD3;BRD4;BRDT	P25440/Q15059/O60885/Q58F21	CRBN	WO-2024099441-A1
TPD-LQY13B	WO2024099441A1_9	.	CC1=C(C2=CC3=C(N=C2)C2=NN(C)C(C(=O)NCCCCCCCCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)=C2N3C(C2=C(F)C=CC=N2)C2CCOCC2)N(C)N=N1	C47H53FN12O6	BRD2;BRD3;BRD4;BRDT	P25440/Q15059/O60885/Q58F21	CRBN	WO-2024099441-A1
TPD-MTMKBK	WO2024146617A1_10	.	COC1(CN2CC3(CCC4=CC5=C(C=C4O3)CN(C3CCC(=O)NC3=O)C5=O)C2)CCN(C2=NN=C(C(=O)N[C@H]3CC[C@H](OC4=CC=C(C#N)C(Cl)=C4)CC3)C=C2)CC1	C43H47ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-AYXSOA	WO2024146617A1_100	.	CC1(C)C(=O)N(C2=CC(C(F)(F)F)=C(C#N)C=C2)C(=S)N1C1=CC=C(C(=O)N2CC3(CC(N4CCC5(CCC6=CC7=C(C=C6O5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)C3)C2)C(F)=C1	C46H41F4N7O7S	AR	P10275	CRBN	WO-2024146617-A1
TPD-TMM554	WO2024146617A1_101	.	CC1(C)C(=O)N(C2=CC(C(F)(F)F)=C(C#N)C=C2)C(=S)N1C1=CC=C(C(=O)N2CCC(N3CCC4(CCC5=CC6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6C=C5O4)CC3)CC2)C(F)=C1	C45H43F4N7O7S	AR	P10275	CRBN	WO-2024146617-A1
TPD-B4G633	WO2024146617A1_102	.	CC1(C)C(=O)N(C2=CC(C(F)(F)F)=C(C#N)C=C2)C(=S)N1C1=CC=C(C(O)N2CC(N3CCC4(CCC5=CC6=C(C=C5O4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C2)C(F)=C1	C43H39F4N7O7S	AR	P10275	CRBN	WO-2024146617-A1
TPD-F4X5MA	WO2024146617A1_103	.	CC1(C)C(=O)N(C2=CC(C(F)(F)F)=C(C#N)C=C2)C(=S)N1C1=CC=C(C(=O)N2CCC3(CC2)CC(N2CCC4(CCC5=CC6=C(C=C5O4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC2)C3)C(F)=C1	C48H45F4N7O7S	AR	P10275	CRBN	WO-2024146617-A1
TPD-FYFN0U	WO2024146617A1_106	.	CC1(CN2CCC3(CCC4=CC5=C(C=C4O3)C(=O)N(C3CCC(=O)NC3=O)C5)CC2)CCN(C2=NN=C(C(=O)N[C@H]3CC[C@H](OC4=CC=C(C#N)C(Cl)=C4)CC3)C=C2)CC1	C45H51ClN8O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-AEGVB6	WO2024146617A1_107	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC(O)(CN5CC6(CCC7=CC8=C(C=C7O6)C(=O)N(C6CCC(=O)NC6=O)C8=O)C5)CC4)C=C3)CC2)C=C1Cl	C42H43ClN8O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-O7L8MP	WO2024146617A1_11	.	CC1(CN2CC3(CCC4=CC5=C(C=C4O3)C(=O)N(C3CCC(=O)NC3=O)C5)C2)CCN(C2=NN=C(C(=O)N[C@H]3CC[C@H](OC4=CC=C(C#N)C(Cl)=C4)CC3)C=C2)CC1	C43H47ClN8O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-X10J2Z	WO2024146617A1_110	.	CC1(C)C(=O)N(C2=CC(C(F)(F)F)=C(C#N)C=C2)C(=S)N1C1=CC=C(C(=O)N2CC(CN3CCC4(CC3)COC3C=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC34)C2)C(F)=C1	C43H39F4N7O7S	AR	P10275	CRBN	WO-2024146617-A1
TPD-2ND0WN	WO2024146617A1_117	.	CC1(C)C(=O)N(C2=CC(C(F)(F)F)=C(C#N)C=C2)C(=S)N1C1=CC=C(C(=O)N2CC3(CCC(N4CCC5(CCC6=CC7=C(C=C6O5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)CC3)C2)C(F)=C1	C48H45F4N7O7S	AR	P10275	CRBN	WO-2024146617-A1
TPD-4R0BRF	WO2024146617A1_118	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC(F)(CN5CCC6(CC5)COC5=C6C=CC6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)CC2)C=C1Cl	C43H44ClFN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-HDBATM	WO2024146617A1_12	.	CC1(CN2CC3(CCC4=CC5=C(C=C4O3)CN(C3CCC(=O)NC3=O)C5=O)C2)CCN(C2=NN=C(C(=O)N[C@H]3CC[C@H](OC4=CC=C(C#N)C(Cl)=C4)CC3)C=C2)CC1	C43H47ClN8O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-AUAJDU	WO2024146617A1_122	.	CC1(C)C(=O)N(C2=CC(C(F)(F)F)=C(C#N)C=C2)C(=S)N1C1=CC=C(C(=O)N2CCC3(CC2)CC(N2CCC4(CC2)COC2=CC5=C(C=C24)C(=O)N(C2CCC(=O)NC2=O)C5=O)C3)C(F)=C1	C47H43F4N7O7S	AR	P10275	CRBN	WO-2024146617-A1
TPD-EGEPWN	WO2024146617A1_124	.	CC1(C)C(=O)N(C2=CC(C(F)(F)F)=C(C#N)C=C2)C(=S)N1C1=CC=C(C(=O)N2CCC(CN3CC4(CCC5=C(C=C6CN(C7CCC(=O)NC7=O)C(=O)C6C5)O4)C3)CC2)C(F)=C1	C44H43F4N7O6S	AR	P10275	CRBN	WO-2024146617-A1
TPD-WLSVMS	WO2024146617A1_127	.	CC1(C)C(=O)N(C2=CC(C(F)(F)F)=C(C#N)C=C2)C(=S)N1C1=CC=C(C(=O)N2CC[C@@H](CN3CCC4(CCC5=CC6=C(C=C5O4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C2)C(F)=C1	C45H41F4N7O7S	AR	P10275	CRBN	WO-2024146617-A1
TPD-W46ZWT	WO2024146617A1_128	.	CC1(C)C(=O)N(C2=CC(C(F)(F)F)=C(C#N)C=C2)C(=S)N1C1=CC=C(C(=O)N2CC(CN3CCC4(CC3)COC3=CC5=C(C=C3C4)C(=O)N(C3CCC(=O)NC3=O)C5=O)C2)C(F)C1	C44H41F4N7O7S	AR	P10275	CRBN	WO-2024146617-A1
TPD-BMWOX0	WO2024146617A1_129	.	CC1(C)C(=O)N(C2=CC(C(F)(F)F)=C(C#N)C=C2)C(=S)N1C1=CC=C(C(=O)N2CCC3(CCC(N4CCC5(CCC6=CC7=C(C=C6O5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)CC3)C2)C(F)=C1	C49H47F4N7O7S	AR	P10275	CRBN	WO-2024146617-A1
TPD-YWB6UD	WO2024146617A1_13	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC(F)(CN5CC6(CCC7=CC8=C(C=C7O6)C(=O)N(C6CCC(=O)NC6=O)C8)C5)CC4)C=C3)CC2)C=C1Cl	C42H44ClFN8O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-2NMDAB	WO2024146617A1_131	.	COC1(CN2CCC3(CCC4=CC5=C(C=C4O3)C(=O)N(C3CCC(=O)NC3=O)C5)CC2)CCN(C2=NN=C(C(=O)N[C@H]3CC[C@H](OC4=CC=C(C#N)C(Cl)=C4)CC3)C=C2)CC1	C45H51ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-Z82HJN	WO2024146617A1_132	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC(F)(CN5CCC6(CCC7=C(O6)C6=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C6)CC5)CC4)C=C3)CC2)C=C1Cl	C44H48ClFN8O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-447IFO	WO2024146617A1_133	.	COC1(CN2CCC3(CCC4=C(O3)C3=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C3)CC2)CCN(C2=NN=C(C(=O)N[C@H]3CC[C@H](OC4=CC=C(C#N)C(Cl)=C4)CC3)C=C2)CC1	C45H51ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-8QSMM1	WO2024146617A1_134	.	COC1=CC(O[C@H]2CC[C@H](NC(=O)C3=CN=C(N4CCC(CN5CCC6(CC5)COC5=C6C=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)(OC)CC4)C=C3)CC2)=CC=C1C#N	C46H53N7O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-ONQ7IP	WO2024146617A1_135	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC(F)(CN5CCC6(CC5)COC5=C6C=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)CC2)C=C1Cl	C43H46ClFN8O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-E6A1OZ	WO2024146617A1_136	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CC5(CC(N6CCC7(CC6)COC6=C7C=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)C5)C4)C=C3)CC2)C=C1Cl	C43H45ClN8O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-079QI3	WO2024146617A1_137	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC5(CCC(N6CCC7(CC6)COC6=C7C=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)CC5)CC4)C=C3)CC2)C=C1Cl	C47H53ClN8O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-AS4EBQ	WO2024146617A1_138	.	COC1(CN2CC3(CCC4=C(O3)C3=C(C=C4)CN(C4CCC(=O)NC4=O)C3=O)C2)CCN(C2=NN=C(C(=O)N[C@H]3CC[C@H](OC4=CC=C(C#N)C(Cl)=C4)CC3)C=C2)CC1	C43H47ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-S1G8L0	WO2024146617A1_139	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC(F)(CN5CC6(CCC7=C(O6)C6=C(C=C7)CN(C7CCC(=O)NC7=O)C6=O)C5)CC4)C=C3)CC2)C=C1Cl	C42H44ClFN8O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-M6LR59	WO2024146617A1_14	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC(F)(CN5CC6(CCC7=CC8=C(C=C7O6)CN(C6CCC(=O)NC6=O)C8=O)C5)CC4)C=C3)CC2)C=C1Cl	C42H44ClFN8O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-LMTGBN	WO2024146617A1_140	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CC5(CC(N6CCC7(CC6)COC6=C7C=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7=O)C5)C4)C=C3)CC2)C=C1Cl	C43H43ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-TK9K7W	WO2024146617A1_141	.	N#CC1=CCC(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC5(CCC(N6CCC7(COC8=C7C=CC7=C8C(=O)N(C8CCC(=O)NC8=O)C7=O)OC6)CC5)CC4)C=C3)CC2)C=C1Cl	C46H51ClN8O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-H7XLVC	WO2024146617A1_142	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CC(N5CCC6(CC5)COC5=C6C=CC6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)C=C3)CC2)C=C1Cl	C40H39ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-YZRWQE	WO2024146617A1_143	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC5(CC4)CC(N4CCC6(CC4)COC4=C6C=CC6=C4C(=O)N(C4CCC(=O)NC4=O)C6=O)C5)C=C3)CC2)C=C1Cl	C45H47ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-ZL19GT	WO2024146617A1_144	.	N#CC1=CCC(OC2CCC(NC(=O)C3=NN=C(N4CCC(N5CC(N6CCC7(CC6)COC6=C7C=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)C5)CC4)C=C3)CC2)C=C1Cl	C45H52ClN9O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-QV1SCQ	WO2024146617A1_145	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC(CN5CCC6(CC5)COC5=C6C=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)CC2)C=C1Cl	C43H47ClN8O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-079DNL	WO2024146617A1_146	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CC(N5CC(N6CCC7(CC6)COC6=C7C=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)C5)C4)C=C3)CC2)C=C1Cl	C43H46ClN9O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-6BNNN6	WO2024146617A1_147	.	N#CC1=CC=C(OC2CCC(NC(=O)C3=NN=C(N4CCC(F)(CN5CCC6(CC5)COC5=C(C6)C6=C(C=C5)CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)CC2)C=C1Cl	C44H48ClFN8O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-BSG1S5	WO2024146617A1_148	.	C/C=C(C#N)\C(Cl)=C/COC1CCC(NC(=O)C2=NN=C(N3CCC(CN4CCC5(CC4)COC4=C(C5)C5=C(C=C4)CN(C4CCC(=O)NC4=O)C5=O)(OC)CC3)C=C2)CC1	C45H55ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-6TSRH9	WO2024146617A1_149	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3C=CC(N4CCC5(CCC(N6CCC7(CC6)COC6=C(C7)C7=C(C=C6)CN(C6CCC(=O)NC6=O)C7=O)CC5)CC4)=NN3)CC2)C=C1Cl	C48H57ClN8O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-D3LIOF	WO2024146617A1_15	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC(F)(CN5CCC6(CCC7=CC8=C(C=C7O6)C(=O)N(C6CCC(=O)NC6=O)C8=O)CC5)CC4)C=C3)CC2)C=C1Cl	C44H46ClFN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-A2Z3DC	WO2024146617A1_150	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC5(CCC(N6CCC7(CCC8=C(O7)C7=C(C=C8)C(=O)N(C8CCC(=O)NC8=O)C7)CC6)CC5)CC4)C=C3)CC2)C=C1Cl	C48H55ClN8O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-76PEV3	WO2024146617A1_151	.	CC1(CN2CCC3(CCC4=C(O3)C3=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C3)CC2)CCN(C2=NN=C(C(=O)N[C@H]3CC[C@H](OC4=CC=C(C#N)C(Cl)=C4)CC3)C=C2)CC1	C45H51ClN8O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-UA32S6	WO2024146617A1_152	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CC5(CC(N6CCC7(CCC8=C(O7)C7CN(C9CCC(=O)NC9=O)C(=O)C7C=C8)CC6)C5)C4)C=C3)CC2)C=C1Cl	C44H49ClN8O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-LLC5CN	WO2024146617A1_153	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CC5(CCC(N6CCC7(CCC8=C(O7)C7=C(C=C8)C(=O)N(C8CCC(=O)NC8=O)C7)CC6)CC5)C4)C=C3)CC2)C=C1Cl	C46H51ClN8O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-YCYADA	WO2024146617A1_154	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC5(CC4)CC(N4CCC6(CCC7=C(O6)C6=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C6)CC4)C5)C=C3)CC2)C=C1Cl	C46H51ClN8O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-HKXYAE	WO2024146617A1_155	.	CCOC1(CN2CCC3(CC2)COC2=C3C=CC3=C2CN(C2CCC(=O)NC2=O)C3=O)CCN(C2=NN=C(C(=O)N[C@H]3CC[C@H](OC4=CC=C(C#N)C(Cl)=C4)CC3)C=C2)CC1	C45H51ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-XI3H1O	WO2024146617A1_156	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NC=C(N4CCC(C#N)(CN5CCC6(CC5)COC5=C6C=CC6C(=O)N(C7CCC(=O)NC7=O)CC56)CC4)C=C3)CC2)CC1Cl	C45H51ClN8O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-JA4PH3	WO2024146617A1_157	.	C=C1OCC2(C/C=C\C3=C1CN(C1CCC(=O)NC1=O)C3=O)CCN(CC1(F)CCN(C3=NC=C(C(=O)N[C@H]4CC[C@H](OC5C=C(Cl)C(C#N)=CC5)CC4)N=C3)CC1)CC2	C44H52ClFN8O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-HJYJZ6	WO2024146617A1_158	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=CN=C(N4CCC(F)(CN5CCC6(CC5)COC5=C6C=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)N=C3)CC2)C=C1Cl	C43H46ClFN8O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-9ZLSGX	WO2024146617A1_159	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CC5(CCC(CN6CCC7(CC6)COC6=C7C=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)CC5)C4)C=C3)CC2)C=C1Cl	C46H51ClN8O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-T9DIGM	WO2024146617A1_16	.	N#C/C=C/C=C(\C=C\Cl)O[C@H]1CC[C@H](NC(=O)C2=NN=C(N3CCC(CN4CCC5(CCC6=CC7=C(C=C6O5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)CC3)C=C2)CC1	C44H49ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-2IH2IT	WO2024146617A1_160	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC(N5CCC(C(=O)N6CCC7(CC6)COC6=C7C=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)CC5)CC4)C=C3)CC2)C=C1Cl	C48H54ClN9O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-NVGKUC	WO2024146617A1_161	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC(C(=O)N5CCC(N6CCC7(CC6)COC6=C7C=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)CC5)CC4)C=C3)CC2)C=C1Cl	C48H54ClN9O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-FFES7C	WO2024146617A1_162	.	COC1(CN2CCC3(CCC4=C(O3)C3=C(C=C4)CN(C4CCC(=O)NC4=O)C3=O)CC2)CCN(C2=NN=C(C(=O)N[C@H]3CC[C@H](OC4=CC=C(C#N)C(Cl)=C4)CC3)C=C2)CC1	C45H51ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-PN3O2M	WO2024146617A1_163	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC(F)(CN5CCC6(CCC7=C(O6)C6=C(C=C7)CN(C7CCC(=O)NC7=O)C6=O)CC5)CC4)C=C3)CC2)C=C1Cl	C44H48ClFN8O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-N2FRAW	WO2024146617A1_164	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC(F)(CN5CC6(CCC7=C(O6)C6=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C6=O)C5)CC4)C=C3)CC2)C=C1Cl	C42H42ClFN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-P5VWZK	WO2024146617A1_165	.	COC1(CN2CC3(CCC4=C(O3)C3=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C3=O)C2)CCN(C2=NN=C(C(=O)N[C@H]3CC[C@H](OC4=CC=C(C#N)C(Cl)=C4)CC3)C=C2)CC1	C43H45ClN8O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-RFNXWD	WO2024146617A1_168	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CC5(CCC(N6CCC7(CC6)COC6=C7C=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)CC5)C4)C=C3)CC2)C=C1Cl	C45H49ClN8O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-OLAE2H	WO2024146617A1_169	.	O=NC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC(N5CCC6(CC5)COC5=C6C=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)CC2)C=C1Cl	C41H45ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-8YRY1G	WO2024146617A1_17	.	CC1(CN2CCC3(CCC4=CC5=C(C=C4O3)C(=O)N(C3CCC(=O)NC3=O)C5=O)CC2)CCN(C2=NN=C(C(=O)N[C@H]3CC[C@H](OC4=CCC(C#N)C(Cl)=C4)CC3)C=C2)CC1	C45H51ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-7YDENL	WO2024146617A1_170	.	N#CC1=CC=C(OC2CCC(NC(=O)C3=NN=C(N4CCC(O)(CN5CCC6(CC5)COC5=C6C=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)CC2)C=C1Cl	C43H47ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-2CNYZQ	WO2024146617A1_171	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC(N5CCC6(CCC7=C(O6)C6=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C6)CC5)CC4)C=C3)CC2)C=C1Cl	C43H47ClN8O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-53W5E7	WO2024146617A1_172	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CC(N5CCC6(CCC7=C(O6)C6=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C6)CC5)C4)C=C3)CC2)C=C1Cl	C41H43ClN8O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-VXJXV1	WO2024146617A1_173	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC(N5CCC(N6CCC7(CC6)COC6=C7C=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)CC5)CC4)C=C3)CC2)C=C1Cl	C47H54ClN9O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-KXH05W	WO2024146617A1_174	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CC(N5CCC(N6CCC7(CC6)COC6=C7C=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)CC5)C4)C=C3)CC2)C=C1Cl	C45H50ClN9O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-VI4XR4	WO2024146617A1_175	.	N#CC1=CC=C(OC2CCC(NC(=O)C3=NN=C(N4CC5(CCC(N6CCC(N7CCC8(CC7)COC7=C8C=CC8=C7CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)C4)C=C3)CC2)C=C1Cl	C50H58ClN9O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-A1F3WP	WO2024146617A1_178	.	CC1(CN2CCC3(CC2)COC2=C3C=CC3=C2CN(C2CCC(=O)NC2=O)C3=O)CCN(C2=NC=C(C(=O)N[C@H]3CC[C@H](OC4=CC=C(C#N)C(Cl)=C4)CC3)C=C2)CC1	C45H50ClN7O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-F82ET8	WO2024146617A1_179	.	CC1(CN2CCC3(CC2)COC2=C3C=CC3=C2C(=O)N(C2CCC(=O)NC2=O)C3=O)CCN(C2=NN=C(C(=O)N[C@H]3CC[C@H](OC4=CC=C(C#N)C(Cl)=C4)CC3)C=C2)CC1	C44H47ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-78LL4G	WO2024146617A1_18	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC(CN5CCC6(CC5)OC5=CC7=C(C=C5CC6(F)F)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)C=C3)CC2)C=C1Cl	C44H45ClF2N8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-GRAQ3T	WO2024146617A1_180	.	COC1=CC(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC(C)(CN5CCC6(CC5)COC5=C6C=CC6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)CC2)=CC=C1C#N	C45H50N8O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-2W44MU	WO2024146617A1_181	.	CC1(CCN2CCC3(CC2)COC2=C3C=CC3=C2C(=O)N(C2CCC(=O)NC2=O)C3=O)CCN(C2=NN=C(C(=O)N[C@H]3CC[C@H](OC4=CC=C(C#N)C(C(F)(F)F)=C4)CC3)C=C2)CC1	C46H49F3N8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-HZDZ2J	WO2024146617A1_182	.	CC1(CN2CCC3(CC2)COC2=C3C=CC3=C2CN(C2CCC(=O)NC2=O)C3=O)CCN(C2=NN=C(C(=O)N[C@H]3CC[C@H](OC4=CC=C(C#N)C(Cl)=C4)CC3)C=C2)CC1	C44H49ClN8O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-SBLUG1	WO2024146617A1_183	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CC(N5CCC6(CC5)COC5=C6C=CC6C(=O)N(C7CCC(=O)NC7=O)CC56)C4)C=C3)CC2)C=C1Cl	C40H43ClN8O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-6VJ9H9	WO2024146617A1_184	.	CC1(C2=C(O)C3=C(C=C2)C(=O)N(C2CCC(=O)NC2=O)C3)CCN(C2CC3(CCN(C4=NN=C(C(=O)N[C@H]5CC[C@H](OC6=CC=C(C#N)C(Cl)=C6)CC5)C=C4)CC3)C2)CC1	C45H51ClN8O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-JLKO0R	WO2024146617A1_185	.	N#CC1=CC=C(OC2CCC(NC(=O)C3=NN=C(N4CCC(F)(CN5CCC6(CC5)COC5C7=C(C=CC5C6)CN(C5CCC(=O)NC5=O)C7=O)CC4)C=C3)CC2)C=C1Cl	C44H50ClFN8O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-IUEPES	WO2024146617A1_186	.	COC1(CN2CCC3(CC2)COC2=C(C=CC4=C2C(=O)N(C2CCC(=O)NC2=O)C4)C3)CCN(C2=NN=C(C(=O)NC3CCC(OC4=CC=C(C#N)C(Cl)=C4)CC3)C=C2)CC1	C45H51ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-WO9WVD	WO2024146617A1_187	.	CC1(CN2CCC3(CC2)COC2=C(C=CC4=C2C(=O)N(C2CCC(=O)NC2=O)C4)C3)CCN(C2=NN=C(C(=O)NC3CCC(OC4=CC=C(C#N)C(Cl)=C4)CC3)C=C2)CC1	C45H51ClN8O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-APJ3UI	WO2024146617A1_188	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC5(CC4)CC(N4CCC6(CC4)COC4=C(C=CC7=C4C(=O)N(C4CCC(=O)NC4=O)C7)C6)C5)C=C3)CC2)C=C1Cl	C46H51ClN8O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-8NGUBC	WO2024146617A1_189	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC(N5CCC6(CC5)COC5=C(C=CC7=C5C(=O)N(C5CCC(=O)NC5=O)C7)C6)CC4)C=C3)CC2)C=C1Cl	C43H47ClN8O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-BAAOR1	WO2024146617A1_19	.	COC1CN(C2=NN=C(C(=O)N[C@H]3CC[C@H](OC4=CC=C(C#N)C(Cl)=C4)CC3)C=C2)CCC1CN1CCC2(CCC3=CC4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4C=C3O2)CC1	C45H51ClN8O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-BMRDMP	WO2024146617A1_190	.	N#CC1=CC=C(OC2CCC(NC(=O)C3=NN=C(N4CCC5(CCC(C6CCC7(CC6)COC6=C(C=CC8=C6C(=O)N(C6CCC(=O)NC6=O)C8)C7)CC5)CC4)C=C3)CC2)C=C1Cl	C49H56ClN7O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-ZMQKCK	WO2024146617A1_191	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CC(N5CCC6(CC5)COC5=C(C=CC7=C5C(=O)N(C5CCC(=O)NC5=O)C7)C6)C4)C=C3)CC2)C=C1Cl	C41H43ClN8O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-J83EG7	WO2024146617A1_192	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC(CC(=O)N5CCC6(CC5)COC5=C6C=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)CC2)C=C1Cl	C44H47ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-526GCJ	WO2024146617A1_193	.	CC1(CN2CCC3(CC2)COC2=C3C=CC3=C2CN(C2CCC(=O)NC2=O)C3=O)CCN(C2=NC=C(C(=O)N[C@H]3CC[C@H](OC4=CC=C(C#N)C(Cl)=C4)CC3)C=N2)CC1	C44H49ClN8O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-XK3OE0	WO2024146617A1_194	.	COC1(CN2CCC3(CC2)COC2=C3C=CC3=C2C(=O)N(C2CCC(=O)NC2=O)C3=O)CCN(C2=NN=C(C(=O)N[C@H]3CC[C@H](OC4=CC=C(C#N)C(Cl)=C4)CC3)C=C2)CC1	C44H47ClN8O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-FY7BCD	WO2024146617A1_195	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC(C(=O)N5CCC6(CC5)COC5=C6C=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)CC2)C=C1Cl	C43H45ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-0ZFBAQ	WO2024146617A1_196	.	COC(=O)C1(CN2CCC3(CC2)COC2=C3C=CC3=C2CN(C2CCC(=O)NC2=O)C3=O)CCN(C2=NN=C(C(=O)N[C@H]3CC[C@H](OC4=CC=C(C#N)C(Cl)=C4)CC3)C=C2)CC1	C45H49ClN8O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-JUHN35	WO2024146617A1_199	.	COC1(CN2CCC3(CC2)CC2=C(C=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C2)O3)CCN(C2=NN=C(C(=O)N[C@H]3CC[C@H](OC4=CC=C(C#N)C(Cl)=C4)CC3)C=C2)CC1	C44H47ClN8O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-LOQEFC	WO2024146617A1_2	.	CC1(CN2CC3(CC/C=C/C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4/C=C/O3)C2)CCN(C2=NN=C(C(O)NC3CCC(OC4=CC=C(C#N)C(Cl)=C4)CC3)C=C2)CC1	C43H51ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-NZZGYK	WO2024146617A1_20	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CC(CN5CCC6(CCC7=CC8=C(C=C7O6)C(=O)N(C6CCC(=O)NC6=O)C8=O)CC5)C4)C=C3)CC2)C=C1Cl	C42H43ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-420E36	WO2024146617A1_200	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC5(CC4)COC4=C5C=CC5=C4CN(C4CCC(=O)NC4=O)C5=O)C=C3)CC2)C=C1Cl	C37H36ClN7O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-AOPKN5	WO2024146617A1_201	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=CN=C(N4CCC5(CC4)COC4=C5C=CC5=C4CN(C4CCC(=O)NC4=O)C5=O)N=C3)CC2)C=C1Cl	C37H36ClN7O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-OXD6CG	WO2024146617A1_202	.	CCOC1(CN2CCC3(CC2)COC2=C3C=CC3=C2CN(C2CCC(=O)NC2=O)C3=O)CCN(C2=NN=C(C(=O)N[C@H]3CC[C@H](OC4=CC=C(C#N)C(C(F)(F)F)=C4)CC3)C=C2)CC1	C46H51F3N8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-M3DDCU	WO2024146617A1_205	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC(F)(CN5CCC6(CC5)CC5=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C5)O6)CC4)C=C3)CC2)C=C1Cl	C43H44ClFN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-T8HJ4E	WO2024146617A1_206	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(C#CC4CCC(N5CCC6(CC5)COC5=C6C=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)CC2)C=C1Cl	C45H46ClN7O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-2XP3ER	WO2024146617A1_207	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(C#N)(CN5CCC6(CC5)COC5=C6C=CC6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)C2(C)C)=CC=C1C#N	C49H53N7O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-Z2GHWV	WO2024146617A1_208	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(C#N)(CN5CCC6(CC5)COC5=C6C=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)C2(C)C)=CC=C1C#N	C49H55N7O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-9RRQH6	WO2024146617A1_209	.	COC1=CC(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC(F)(CN5CC6(CCC7=CC8=C(C=C7O6)CN(C6CCC(=O)NC6=O)C8=O)C5)CC4)C=C3)CC2)=CC=C1C#N	C43H47FN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-2WCXAG	WO2024146617A1_21	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CC[C@@H](CN5CCC6(CCC7=CC8=C(C=C7O6)C(=O)N(C6CCC(=O)NC6=O)C8=O)CC5)C4)C=C3)CC2)C=C1Cl	C43H45ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-DV9JCI	WO2024146617A1_210	.	CC1(C)[C@H](NC(=O)C2=NN=C(N3CCC(CN4CCC5(CC4)COC4=C5C=CC5=C4CN(C4CCC(=O)NC4=O)C5=O)CC3)C=C2)C(C)(C)[C@H]1OC1C=C(Cl)C(C#N)=CC1	C45H53ClN8O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-GCGJWC	WO2024146617A1_211	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC(CC5CC5)(CN5CCC6(CC5)COC5C7=C(C=CC56)C(=O)N(C5CCC(=O)NC5=O)C7)CC4)C=C3)CC2)C=C1Cl	C47H55ClN8O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-Y9KKJ3	WO2024146617A1_212	.	C[C@H]1CN(C2=NN=C(C(=O)N[C@H]3CC[C@H](OC4=CC=C(C#N)C(Cl)=C4)CC3)C=C2)C[C@@H]1CN1CCC2(CC1)COC1=C2C=CC2=C1CN(C1CCC(=O)NC1=O)C2=O	C43H47ClN8O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-0EUK34	WO2024146617A1_213	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC(O)(CN5CCC6(CC5)COC5=C6C=CC6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)CC2)C=C1Cl	C43H45ClN8O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-WMFR5Z	WO2024146617A1_214	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC(O)(CN5CCC6(CC5)COC5=C6C=CC6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)CC2)C=C1C(F)(F)F	C44H45F3N8O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-J3QZ9M	WO2024146617A1_215	.	COC1=CC(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC(O)(CN5CCC6(CC5)COC5=C6C=CC6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)CC2)=CC=C1C#N	C44H48N8O9	AR	P10275	CRBN	WO-2024146617-A1
TPD-Q053O8	WO2024146617A1_216	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=CN=C(N4CCC(F)(CN5CCC6(CC5)COC5=C6C=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)CC2)C=C1Cl	C44H47ClFN7O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-RVULNA	WO2024146617A1_217	.	COC1=CC(OC2C(C)(C)C(NC(=O)C3=CC=C(N4CCC(CN5CCC6(CC5)COC5=C6C=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)(OC)CC4)C=C3)C2(C)C)=CC=C1C#N	C49H58N6O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-TLLNKU	WO2024146617A1_218	.	COC1=CC(OC2C(C)(C)C(NC(=O)C3=CC=C(N4CCC(CN5CCC6(CC5)COC5=C6C=CC6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)(OC)CC4)C=C3)C2(C)C)CC=C1C#N	C49H58N6O9	AR	P10275	CRBN	WO-2024146617-A1
TPD-XFE8F2	WO2024146617A1_219	.	COC1=CC(OC2CCC(NC(=O)C3=CC=C(N4CCC(CN5CCC6(CC5)COC5=C6C=CC6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)(OC)CC4)C=C3)CC2)=CC=C1C#N	C47H52N6O9	AR	P10275	CRBN	WO-2024146617-A1
TPD-P84RAB	WO2024146617A1_22	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CC[C@H](CN5CCC6(CCC7=CC8=C(C=C7O6)C(=O)N(C6CCC(=O)NC6=O)C8=O)CC5)C4)C=C3)CC2)C=C1Cl	C43H45ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-9Y1F3G	WO2024146617A1_221	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(C)(CN5CCC6(CC5)COC5=C6C=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)C2(C)C)=CN=C1C#N	C48H57N7O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-AQM6MV	WO2024146617A1_222	.	CC1(CN2CCC3(CC2)COC2=C3C=CC3=C2CN(C2CCC(=O)NC2=O)C3=O)CCN(C2=CC=C(C(=O)N[C@H]3C(C)(C)[C@H](OC4=CC=C(C#N)C(Cl)=C4)C3(C)C)C=C2)CC1	C48H55ClN6O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-ZVBM1P	WO2024146617A1_223	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(F)(CN5CCC6(CC5)COC5=C6C=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)C2(C)C)CC=C1C#N	C48H57FN6O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-PARV8R	WO2024146617A1_224	.	COC1=CC(OC2C(C)(C)C(NC(=O)C3=NN=C(N4CCC(C#N)(CN5CCC6(CC5)COC5=C6C=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)C2(C)C)=CC=C1C#N	C47H53N9O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-U56I56	WO2024146617A1_225	.	CC1(C)[C@H](NC(=O)C2=NN=C(N3CCC(C#N)(CN4CCC5(CC4)COC4=C5C=CC5=C4CN(C4CCC(=O)NC4=O)C5=O)CC3)C=C2)C(C)(C)[C@H]1OC1C=C(Cl)C(C#N)=CC1	C46H52ClN9O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-9HY32I	WO2024146617A1_226	.	[H]C1CN(C2=NN=C(C(=O)NC3CCC(OC4=CC=C(C#N)C(Cl)=C4)CC3)C=C2)CC[C@@H]1CN1CCC2(CC1)COC1=C2C=CC2=C1CN(C1CCC(=O)NC1=O)C2=O	C43H47ClN8O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-KVQ5S8	WO2024146617A1_227	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC(C#N)(CN5CCC6(CC5)COC5=C6C=CC6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)CC2)C=C1Cl	C44H44ClN9O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-0J120P	WO2024146617A1_228	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC(C#N)(CN5CCC6(CC5)COC5=C6C=CC6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)CC2)C=C1C(F)(F)F	C45H44F3N9O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-N85CHH	WO2024146617A1_229	.	COC1=CC(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC(C#N)(CN5CCC6(CC5)COC5=C6C=CC6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)CC2)=CC=C1C#N	C45H47N9O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-JWWLPJ	WO2024146617A1_23	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC(N5CCC6(CCC7=CC8=C(C=C7O6)C(=O)N(C6CCC(=O)NC6=O)C8=O)CC5)[C@@H](F)C4)C=C3)CC2)C=C1Cl	C43H44ClFN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-ICC044	WO2024146617A1_230	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(C)(CN5CCC6(CC5)COC5=C6C=CC6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)C2(C)C)=CC=C1C#N	C49H56N6O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-MYF4HN	WO2024146617A1_231	.	COC1=CC(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC(CN5CC6(CCC7=CC8=C(C=C7O6)C(=O)N(C6CCC(=O)NC6=O)C8=O)C5)(OC)CC4)C=C3)CC2)=CC=C1C#N	C44H48N8O9	AR	P10275	CRBN	WO-2024146617-A1
TPD-47WZAO	WO2024146617A1_232	.	COC1=CC(O[C@H]2CC[C@H](NC(=O)C3=CN=C(N4CCC(CN5CC6(CCC7=CC8=C(C=C7O6)C(=O)N(C6CCC(=O)NC6=O)C8=O)C5)(OC)CC4)N=C3)CC2)=CC=C1C#N	C44H48N8O9	AR	P10275	CRBN	WO-2024146617-A1
TPD-7GEHQK	WO2024146617A1_233	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCN(C(=O)CN5CCC6(CC5)COC5=C6C=CC6C(=O)N(C7CCC(=O)NC7=O)CC56)CC4)C=C3)CC2)C=C1Cl	C43H48ClN9O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-8D7SOO	WO2024146617A1_234	.	COC1=CC(OC2C(C)(C)C(NC(=O)C3=CC=C(N4CCC(CN5CCC6(CC5)COC5=C6C=CC6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)C2(C)C)=CC=C1C#N	C48H54N6O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-PKGJS6	WO2024146617A1_235	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=CN=C(C#CC4CCC(N5CCC6(CC5)COC5=C6C=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)CC2)C=C1Cl	C46H47ClN6O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-26DU2W	WO2024146617A1_236	.	CCC1(CN2CCC3(CC2)COC2=C3C=CC=C2CN(C=O)C2CCC(=O)NC2=O)CCN(C2=NN=C(C(=O)NC3CCC(OC4=CC=C(C#N)C(CI)=C4)CC3)C=C2)CC1	C46H55IN8O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-G0VI5M	WO2024146617A1_237	.	CC1(C)[C@H](NC(=O)C2=NN=C(N3CCC(F)(CN4CCC5(CC4)COC4=C5C=CC5=C4CN(C4CCC(=O)NC4=O)C5=O)CC3)C=C2)C(C)(C)[C@H]1OC1=CCC(C#N)C(C(F)(F)F)=C1	C46H52F4N8O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-DVQK0K	WO2024146617A1_238	.	N#CC1=C(Cl)C=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC(CN5CCC6(CC5)COC5=C6C=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)(C5CC5)CC4)C=C3)CC2)C=C1	C46H51ClN8O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-AZ1YLI	WO2024146617A1_239	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(C#CC4=CN=C(N5CCC6(CC5)COC5=C6C=CC6C(=O)N(C7CCC(=O)NC7=O)CC56)C=C4)C=C3)CC2)C=C1Cl	C44H41ClN8O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-G7MR86	WO2024146617A1_24	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NC(F)=C(N4CCC(N5CCC6(CCC7=CC8=C(C=C7O6)C(=O)N(C6CCC(=O)NC6=O)C8=O)CC5)[C@H](F)C4)C=C3)CC2)C=C1Cl	C44H44ClF2N7O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-GOINOW	WO2024146617A1_241	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCN(CC(=O)N5CCC6(CC5)COC5=C7CN(C8CCC(=O)NC8=O)C(=O)C7=CC=C56)CC4)CC3)CC2)C=C1Cl	C43H48ClN9O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-YSXBNX	WO2024146617A1_242	.	CCOC1(CN2CCC3(CC2)COC2=C3C=CC3=C2C(=O)N(C2CCC(=O)NC2=O)C3=O)CCN(C2=NN=C(C(=O)N[C@H]3CC[C@H](OC4=CC=C(C#N)C(C(F)(F)F)=C4)CC3)C=C2)CC1	C46H49F3N8O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-F51JY9	WO2024146617A1_243	.	CCOC1(CN2CCC3(CC2)COC2=C3C=CC3=C2C(=O)N(C2CCC(=O)NC2=O)C3=O)CCN(C2=NN=C(C(=O)N[C@H]3CC[C@H](OC4=CC=C(C#N)C(OC)=C4)CC3)C=C2)CC1	C46H52N8O9	AR	P10275	CRBN	WO-2024146617-A1
TPD-SZ3B86	WO2024146617A1_244	.	CCOC1(CN2CCC3(CC2)COC2=C3C=CC3=C2C(=O)N(C2CCC(=O)NC2=O)C3=O)CCN(C2=NN=C(C(=O)N[C@H]3CC[C@H](OC4=CC=C(C#N)C(Cl)=C4)CC3)C=C2)CC1	C45H49ClN8O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-1E2FDG	WO2024146617A1_245	.	CC1(CN2CCC3(CC2)COC2=C3C=CC3=C2C(=O)N(C2CCC(=O)NC2=O)C3=O)CCN(C2=NC=C(C(=O)NC3CCC(OC4=CC=C(C#N)C(Cl)=C4)CC3)C=N2)CC1	C44H47ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-42C0NE	WO2024146617A1_246	.	COC1=CC(OC2CCC(NC(=O)C3=CN=C(N4CCC(C)(CN5CCC6(CC5)COC5=C6C=CC6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)N=C3)CC2)=CC=C1C#N	C45H50N8O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-1NG7X4	WO2024146617A1_247	.	COC1=CC(O[C@H]2CC[C@H](NC(=O)C3=CN=C(N4CCC(C)(CN5CCC6(CC5)COC5=C6C=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)N=C3)CC2)=CC=C1C#N	C45H52N8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-J45W4B	WO2024146617A1_248	.	CCC1(CN2CCC3(CC2)COC2=C3C=CC3=C2C(=O)N(C2CCC(=O)NC2=O)C3=O)CCN(C2=NN=C(C(=O)N[C@H]3CC[C@H](OC4=CCC(C#N)C(C(F)(F)F)=C4)CC3)C=C2)CC1	C46H51F3N8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-SQHJZR	WO2024146617A1_249	.	CCC1(CN2CCC3(CC2)COC2=C3C=CC3=C2C(=O)N(C2CCC(=O)NC2=O)C3=O)CCN(C2=NN=C(C(=O)N[C@H]3CC[C@H](OC4=CC=C(C#N)C(Cl)=C4)CC3)C=C2)CC1	C45H49ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-A9PV0O	WO2024146617A1_25	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CC(N5CCC6(CCC7=CC8=C(C=C7O6)C(=O)N(C6CCC(=O)NC6=O)C8=O)CC5)C4)C=C3)CC2)C=C1Cl	C41H41ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-WCT5UE	WO2024146617A1_250	.	CCC1(CN2CCC3(CC2)COC2=C3C=CC3=C2C(=O)N(C2CCC(=O)NC2=O)C3=O)CCN(C2=NN=C(C(=O)N[C@H]3CC[C@H](OC4=CC=C(C#N)C(OC)=C4)CC3)C=C2)CC1	C46H52N8O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-IY764N	WO2024146617A1_251	.	COC1=CC(O[C@H]2CC[C@H](NC(=O)C3=CC=C(N4CC(CN5CCC6(CC5)COC5=C6C=CC6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)C4)N=N3)CC2)=CC=C1C#N	C42H44N8O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-J4NGJX	WO2024146617A1_252	.	N#CC1CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(C#CC4CC5(C4)CC(N4CCC6(CC4)COC4=C6C=CC6=C4CN(C4CCC(=O)NC4=O)C6=O)C5)C=C3)CC2)C=C1Cl	C46H48ClN7O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-UQPIPE	WO2024146617A1_253	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC5(CCC(C(=O)N6CCC7(CC6)COC6=C7C=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)CC5)CC4)C=C3)CC2)C=C1Cl	C48H53ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-C0LA91	WO2024146617A1_254	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC5(CC4)CC(C(=O)N4CCC6(CC4)COC4=C6C=CC6=C4CN(C4CCC(=O)NC4=O)C6=O)C5)C=C3)CC2)C=C1Cl	C46H49ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-JK6NSQ	WO2024146617A1_255	.	N#CC1=CCC(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CC5(CCC(C(=O)N6CCC7(CC6)COC6=C7C=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)CC5)C4)C=C3)CC2)C=C1Cl	C46H51ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-8ARYDB	WO2024146617A1_256	.	N#CC1=CC=C(OC2CCC(NC(=O)C3=NN=C(N4CC5(CC(C(=O)N6CCC7(CC6)COC6=C7C=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)C5)C4)C=C3)CC2)C=C1Cl	C44H45ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-JKDY80	WO2024146617A1_257	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC(CO)(CN5CCC6(CC5)COC5=C6C=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)CC2)C=C1Cl	C44H49ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-C8VE2A	WO2024146617A1_258	.	COCC1(CN2CCC3(CC2)COC2=C3CCC3=C2CN(C2CCC(=O)NC2=O)C3=O)CCN(C2=NN=C(C(=O)N[C@H]3CC[C@H](OC4=CC=C(C#N)C(Cl)=C4)CC3)C=C2)CC1	C45H53ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-H291Z8	WO2024146617A1_259	.	CC1(CN2CCC3(CC2)COC2=C3C=CC3=C2CN(C2CCC(=O)NC2=O)C3=O)CCN(C2=CN=C(C(=O)NC3CCC(OC4=CC=C(C#N)C(Cl)=C4)CC3)C=C2)CC1	C45H50ClN7O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-MST4SF	WO2024146617A1_26	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC(N5CCC6(CCC7=CC8=C(C=C7O6)C(=O)N(C6CCC(=O)NC6=O)C8=O)CC5)CC4)C=C3)CC2)C=C1Cl	C43H45ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-PPHTYK	WO2024146617A1_260	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NC=C(N4CCC(F)(CN5CCC6(CC5)COC5=C6C=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)CC2)C=C1Cl	C44H47ClFN7O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-HMJJG5	WO2024146617A1_265	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(C)(CNCC5CCC6=CC7=C(C=C6O5)C(=O)N(C5CCC(=O)NC5=O)C7)CC4)C=C3)C2(C)C)=CC=C1C#N	C47H56N6O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-AT78LD	WO2024146617A1_266	.	CO/C=C/C(=C\C=C\C#N)OC1C(C)(C)C(NC(=O)C2=CC=C(N3CCC(CN4CCC5(CC4)COC4=C(C=CC6CN(C7CCC(=O)NC7=O)C(=O)C46)C5)CC3)C=C2)C1(C)C	C49H62N6O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-FQ5W0W	WO2024146617A1_267	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(C)(CN5CCC6(CCC7=CC8=C(C=C7O6)C(=O)N(C6CCC(=O)NC6=O)C8)CC5)CC4)C=C3)C2(C)C)=CC=C1C#N	C50H60N6O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-Y0VHRW	WO2024146617A1_268	.	C=C1C2=C(C(=O)N1C1CCC(=O)NC1=O)C1=C(C=C2)CCC2(CCN(CC3(C)CCN(C4=CC=C(C(=O)N[C@H]5C(C)(C)[C@H](OC6=CC=C(C#N)C(O)=C6)C5(C)C)C=C4)CC3)CC2)O1	C50H58N6O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-2GA95K	WO2024146617A1_269	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(F)(CN5CC6(CCC7=CC8=C(C=C7O6)C(=O)N(C6CCC(=O)NC6=O)C8=O)C5)CC4)C=C3)C2(C)C)=CC=C1C#N	C47H51FN6O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-I0G5V6	WO2024146617A1_27	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NNC(N4CCC(N5CCC6(CCC7=CC8=C(C=C7O6)C(=O)N(C6CCC(=O)NC6=O)C8=O)CC5)C(F)(F)C4)C=C3)CC2)C=C1Cl	C43H45ClF2N8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-NTQIW9	WO2024146617A1_270	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(F)(CN5CCC6(CCC7=CC8=C(C=C7O6)C(=O)N(C6CCC(=O)NC6=O)C8=O)CC5)CC4)C=C3)C2(C)C)=CC=C1C#N	C49H55FN6O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-6PGGDT	WO2024146617A1_271	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(C)(CN5CCC6(CC5)COC5=CC7=C(C=C5C6)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)C=C3)C2(C)C)=CC=C1C#N	C50H58N6O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-RNVL9X	WO2024146617A1_272	.	COC1=CC(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC(CN5CCC6(CC5)COC5=C6C=CC6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)(OC)CC4)C=C3)CC2)=CC=C1C#N	C45H50N8O9	AR	P10275	CRBN	WO-2024146617-A1
TPD-J65QM0	WO2024146617A1_273	.	COC1=CC(OC2C(C)(C)C(NC(=O)C3=CC=C(N4CCC(C)(CN5CCC6(CC5)COC5=CC7=C(C=C56)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)C=C3)C2(C)C)=CC=C1C#N	C49H56N6O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-YWXDMW	WO2024146617A1_274	.	COC1=CC(O[C@@H](C(C)(C)C)C(C)(C)CNC(=O)C2=CCC(N3CCC(F)(CN4CC5(CCC6=C(O5)C5=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C5=O)C4)CC3)C=C2)=CC=C1C#N	C48H57FN6O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-WW5NOK	WO2024146617A1_275	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(F)(CN5CCC6(CC5)COC5=C6C=CC6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)C2(C)C)CC=C1C#N	C48H55FN6O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-O5UJCE	WO2024146617A1_277	.	COC1=CC(OC2C(C)(C)C(NC(=O)C3=CC=C(N4CCC(CN5CC6(CCC7=CC8=C(C=C7O6)C(=O)N(C6CCC(=O)NC6=O)C8=O)C5)CC4)C=C3)C2(C)C)=CC=C1C#N	C47H52N6O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-FHGZRH	WO2024146617A1_278	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(CN5CCC6(CCC7=NC8=C(C=C7O6)C(=O)N(C6CCC(=O)NC6=O)C8=O)CC5)CC4)C=C3)C2(C)C)=CC=C1C#N	C48H55N7O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-94FPX6	WO2024146617A1_279	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(CN5CCC6(CC5)COC5=CC7=C(C=C5C6)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)C=C3)C2(C)C)=CC=C1C#N	C49H56N6O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-ZWJ8YH	WO2024146617A1_28	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC5(CCC6=CC7=C(C=C6O5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)C=C3)CC2)C=C1Cl	C38H36ClN7O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-IYQCVH	WO2024146617A1_280	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(CN5CCC6(CC5)COC5=CC7=C(C=C56)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)C=C3)C2(C)C)=CC=C1C#N	C48H54N6O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-XK68BD	WO2024146617A1_281	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(C)(CN5CCC6(CCC7=CC8=C(C=C7O6)CN(C6CCC(=O)NC6=O)C8=O)CC5)CC4)C=C3)C2(C)C)=CC=C1C#N	C50H60N6O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-DE77ZI	WO2024146617A1_282	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CCC(N4CCC(CN5CC6(CCC7=CC8=C(C=C7O6)CN(C6CCC(=O)NC6=O)C8=O)C5)CC4)C=C3)C2(C)C)=CC=C1C#N	C47H56N6O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-VCVMWZ	WO2024146617A1_283	.	COC1=CC(OC2C(C)(C)C(NC(=O)C3=CCC(N4CCC(C)(CN5CCC6(CCC7=C(O6)C6=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C6)CC5)CC4)C=C3)C2(C)C)=CC=C1C#N	C50H62N6O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-AGGSVT	WO2024146617A1_284	.	COCC1(OC2=CC3=C(C=C2)C(=O)N(C2CCC(=O)NC2=O)C3)CCN(CC2(F)CCN(C3=CC=C(C(=O)NC4C(C)(C)C(OC5=CC=C(C#N)C(OC)=C5)C4(C)C)C=C3)CC2)CC1	C49H59FN6O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-1XATUN	WO2024146617A1_285	.	COC1=CC(O[C@H]2CC[C@H](NC(=O)C3=CC=C(N4CCC(CN5CC6(CCC7=CC8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8C=C7O6)C5)(OC)CC4)C=C3)CC2)=CC=C1C#N	C46H52N6O9	AR	P10275	CRBN	WO-2024146617-A1
TPD-NVPQNV	WO2024146617A1_286	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(C)(CN5CCC6(CC5)COC5=C6C=CC6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)C2(C)C)=CCC1C#N	C49H58N6O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-6FK99F	WO2024146617A1_287	.	CO/C=C/C(=C\C=C\C#N)O[C@H]1C(C)(C)[C@H](NC(=O)C2=CC=C(N3CCC(C)(CN4CCC5(CCC6=CC7=C(C=C6O5)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)CC3)C=C2)C1(C)C	C50H60N6O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-K7POKU	WO2024146617A1_288	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(C)(CN5CCC6(CC5)COC5=CC7=C(C=C56)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)C=C3)C2(C)C)=CC=C1C#N	C49H56N6O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-AE3C3K	WO2024146617A1_289	.	COC1=CC(OC2C(C)(C)C(NC(=O)C3=CC=C(N4CCC(C)(CN5CCC6(CC5)COC5=CC7=C(C=C5C6)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)C=C3)C2(C)C)=CC=C1C#N	C50H58N6O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-DX9TXY	WO2024146617A1_29	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCN(C5CCC6(CCC7=CC8=C(C=C7O6)C(=O)N(C6CCC(=O)NC6=O)C8=O)CC5)CC4)C=C3)CC2)C=C1Cl	C43H45ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-FFGIUK	WO2024146617A1_290	.	COC1=CC(OC2C(C)(C)C(NC(=O)C3=CC=C(N4CCC(C)(CN5CC6(CCC7=C(O6)C6=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C6=O)C5)CC4)C=C3)C2(C)C)=CC=C1C#N	C48H54N6O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-GPGWRJ	WO2024146617A1_291	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(C)(CN5CC6(CCC7=CC8=C(C=C7O6)C(=O)N(C6CCC(=O)NC6=O)C8=O)C5)CC4)C=C3)C2(C)C)=CC=C1C#N	C48H54N6O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-8954TL	WO2024146617A1_294	.	CCC(C1CCN(C2=CC=C(C(=O)N[C@H]3C(C)[C@H](OC4=CC=C(C#N)C(O)=C4)C3(C)C)C=C2)CC1)N1CCC2(CC1)COC1=C2C=CC2=C1CN(C1CCC(=O)NC1=O)C2=O	C48H56N6O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-2Q50PB	WO2024146617A1_295	.	CCOC1(CN2CCC3(CC2)COC2=C3C=CC3=C2C(=O)N(C2CCC(=O)NC2=O)C3=O)CCN(C2=CC=C(C(=O)N[C@H]3C(C)(C)[C@H](OC4=CC=C(C#N)C(OC)=C4)C3(C)C)C=C2)CC1	C50H58N6O9	AR	P10275	CRBN	WO-2024146617-A1
TPD-3CQN34	WO2024146617A1_296	.	COC1=CC(OC2C(C)(C)C(NC(=O)C3=CCC(N4CCC(CN5CCC6(CCC7=CC8=C(C=C7O6)CN(C6CCC(=O)NC6=O)C8=O)CC5)CC4)C=C3)C2(C)C)=CC=C1C#N	C49H60N6O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-0A74FZ	WO2024146617A1_297	.	COC1=CC(OC2C(C)(C)C(NC(=O)C3=CC=C(N4CCC(CN5CC6(CCC7=NC8=C(C=C7O6)CN(C6CCC(=O)NC6=O)C8=O)C5)CC4)C=C3)C2(C)C)=CC=C1C#N	C46H53N7O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-K4WPVT	WO2024146617A1_298	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(CN5CCC6(CCC7=C(O6)C6=C(C=C7)[C@@H](C)N(C7CCC(=O)NC7=O)C6)CC5)CC4)C=C3)C2(C)C)=CC=C1C#N	C50H62N6O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-IAW40P	WO2024146617A1_299	.	COC1=CC(O[C@H]2CC[C@H](NC(=O)C3=CN=C4CN(C(=O)CN5CCC6(CC5)COC5=C6C=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CCC4=C3)CC2)=CC=C1C#N	C44H47N7O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-M91XIQ	WO2024146617A1_3	.	COC1(CN2CC3(CCC4=CC5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5C=C4O3)C2)CCN(C2=NN=C(C(=O)N[C@H]3CC[C@H](OC4=CC=C(C#N)C(Cl)=C4)CC3)C=C2)CC1	C43H47ClN8O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-WD0FT4	WO2024146617A1_30	.	CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC5(CCC(N6CCC7(CCC8=CC9=C(C=C8O7)C(=O)N(C7CCC(=O)NC7=O)C9=O)CC6)CC5)CC4)C=C3)CC2)C=C1Cl	C48H56ClN7O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-MM3UU7	WO2024146617A1_300	.	COC1=CC(O[C@H]2CC[C@H](NC(=O)C3=CN=C4CN(CC(=O)N5CCC6(CC5)COC5=C6C=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CCC4=C3)CC2)=CC=C1C#N	C44H47N7O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-X5NYSM	WO2024146617A1_301	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(CN5CCC6(CCC7=CC8=C(C=C7O6)C(=O)N(C6CCC(=O)NC6=O)C8)CC5)CC4)C=C3)C2(C)C)=CC=C1C#N	C49H58N6O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-EVNVSE	WO2024146617A1_302	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(CN5CC6(CCC7=CC8CN(C9CCC(=O)NC9=O)C(=O)C8C=C7O6)C5)CC4)C=C3)C2(C)C)=CC=C1C#N	C47H56N6O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-QB57PD	WO2024146617A1_303	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(C4CCC(CN5CCC6(CC5)COC5=C(C=CC7=C5C(=O)N(C5CCC(=O)NC5=O)C7)C6)CC4)C=C3)C2(C)C)=CC=C1C#N	C50H59N5O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-I0WJ5M	WO2024146617A1_304	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(CN5CCC6(CC5)COC5=CC7=C(C=C5O6)CN(C5CCC(=O)NC5=O)C7=O)CC4)C=C3)C2(C)C)=CC=C1C#N	C48H56N6O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-DO7NN7	WO2024146617A1_305	.	C=C1C2=C(C(=O)N1C1CCC(=O)NC1=O)C1=C(C=C2)CCC2(CCN(CC3CCN(C4=CC=C(C(=O)N[C@H]5C(C)(C)[C@H](OC6C=C(OC)C(C#N)=CC6)C5(C)C)C=C4)CC3)CC2)C1	C51H62N6O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-RY2B2C	WO2024146617A1_306	.	COC1=CC(OC2CCC(NC(=O)C3=CC=C4CN(C(=O)CN5CCC6(CC5)COC5=C6C=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CCC4N3)CC2)=CC=C1C#N	C44H49N7O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-L4W9T4	WO2024146617A1_307	.	COC1=CC(O[C@H]2CC[C@H](NC(=O)C3=CC=C4CN(CC(=O)N5CCC6(CC5)COC5=C6C=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CCC4=N3)CC2)=CC=C1C#N	C44H47N7O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-6F3JSP	WO2024146617A1_308	.	COC1=CC(O[C@H]2CC[C@H](NC(=O)C3=NC=C(N4CCC(CN5CCC6(CC5)COC5=C6C=CC6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)(OC)CC4)C=N3)CC2)=CC=C1C#N	C45H50N8O9	AR	P10275	CRBN	WO-2024146617-A1
TPD-VA5P1K	WO2024146617A1_309	.	COC1=CC(O[C@H]2CC[C@H](NC(=O)C3=NC=C(N4CCC(CN5CC6(CCC7=CC8=C(C=C7O6)C(=O)N(C6CCC(=O)NC6=O)C8=O)C5)(OC)CC4)C=N3)CC2)=CC=C1C#N	C44H48N8O9	AR	P10275	CRBN	WO-2024146617-A1
TPD-ISYTYU	WO2024146617A1_310	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(F)(CN5CCC6(CCC7=CC8=C(C=C7O6)CN(C6CCC(=O)NC6=O)C8=O)CC5)CC4)C=C3)C2(C)C)=CC=C1C#N	C49H57FN6O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-8PX6WU	WO2024146617A1_311	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(F)(CN5CC6(CCC7=CC8=C(C=C7O6)CN(C6CCC(=O)NC6=O)C8=O)C5)CC4)C=C3)C2(C)C)=CC=C1C#N	C47H53FN6O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-8CP4TQ	WO2024146617A1_312	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(F)(CN5CCC6(CCC7=C(O6)C6=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C6)CC5)CC4)C=C3)C2(C)C)=CC=C1C#N	C49H57FN6O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-GNQ0GF	WO2024146617A1_317	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(F)(CN5CC6(CCC7=CC8=C(C=C7O6)C(=O)N(C6CCC(=O)NC6=O)C8)C5)OC4)C=C3)C2(C)C)=CC=C1C#N	C46H51FN6O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-UPF94C	WO2024146617A1_319	.	C[C@H]1CC2(CCN(C3=CC=C(C(=O)N4CCC(C)(CN5CCC6(CC5)COC5=C6C=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)CC2)CN1C1=CC=C(C#N)C(Cl)=C1	C49H56ClN7O5	AR	P10275	CRBN	WO-2024146617-A1
TPD-HJQ1FT	WO2024146617A1_32	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CC5(CC(N6CCC7(CCC8=CC9=C(C=C8O7)C(=O)N(C7CCC(=O)NC7=O)C9=O)CC6)C5)C4)C=C3)CC2)C=C1Cl	C44H45ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-D4H376	WO2024146617A1_320	.	COC1(CN2CC3(CCC4=C(C=C5CN(C6CCC(=O)NC6=O)C(=O)C5=C4)O3)C2)CCN(C(=O)C2=CC=C(N3CCC4(CC3)CCN(C3=CC=C(C#N)C(Cl)=C3)C4)C=C2)CC1	C47H52ClN7O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-XECVVP	WO2024146617A1_322	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(O)C3=CC=C(N4CCC(F)(CN5CCC6(CC5)COC5=C(C=CC7=C5C(=O)N(C5CCC(=O)NC5=O)C7)C6)CC4)C=C3)C2(C)C)=CC=C1C#N	C49H59FN6O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-K3YYOB	WO2024146617A1_323	.	O=C1CCC(N2CC3=C(C=CC4=C3OCC43CCN(C4CC5(C4)CN(C4=NN=C(C(=O)N[C@H]6CC[C@H](OC7=CC=CC=C7)CC6)C=C4)C5)CC3)C2=O)C(=O)N1	C42H47N7O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-DPR3NZ	WO2024146617A1_324	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC(CN5CCC6(CC5)COC5=C6C=CC6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)CC2)C=C1Cl	C43H45ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-KCU2O4	WO2024146617A1_325	.	COC1=CC(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC(C)(CN5CCC6(CC5)COC5=C6C=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)CC2)=CC=C1C#N	C45H52N8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-FPH8YC	WO2024146617A1_326	.	COC1=CC(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC(CN5CCC6(CC5)COC5=C6C=CC6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)CC2)=CC=C1C#N	C44H48N8O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-306HG1	WO2024146617A1_327	.	COC1=CC(O[C@H]2CC[C@H](NC(=O)C3=NN=C(C4CCC(F)(CN5CCC6(CC5)COC5=C6C=CC6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)CC2)=CC=C1C#N	C45H48FN7O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-TLDJ2R	WO2024146617A1_328	.	COC1(N2CCC3(CC2)COC2=C3C=CC3=C2C(=O)N(C2CCC(=O)NC2=O)C3=O)CCN(C2=NN=C(C(=O)N(C)[C@H]3CC[C@H](OC4=CCC(C#N)C(Cl)=C4)CC3)C=C2)CC1	C44H49ClN8O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-97J4YJ	WO2024146617A1_329	.	COC1=CC(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC(F)(CN5CCC6(CC5)COC5=CC7=C(C=C56)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)C=C3)CC2)=CC=C1C#N	C44H47FN8O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-TYGT1Z	WO2024146617A1_33	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CC5(CCC(N6CCC7(CCC8=CC9=C(C=C8O7)C(=O)N(C7CCC(=O)NC7=O)C9=O)CC6)CC5)C4)C=C3)CC2)C=C1Cl	C46H49ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-PZMEU5	WO2024146617A1_330	.	C=C1NC(=O)CCC1N1C(=O)C2=C(C=C3C(=C2)OCC3CCN(CCC)CC2(OCC)CCN(C3=NN=C(C(=O)N[C@H]4CC[C@H](OC5=CC=C(C#N)C(OC)=C5)CC4)C=C3)CC2)C1=O	C48H58N8O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-WOFJQJ	WO2024146617A1_331	.	CC1=CC=C(N2CC3(CCN(C4=CC=C(C(=O)N5CCC(CN6CCC7(CC6)COC6=C7C=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)CC5)C=C4)CC3)C[C@@H]2C)C=C1Cl	C48H57ClN6O5	AR	P10275	CRBN	WO-2024146617-A1
TPD-2DY1P2	WO2024146617A1_332	.	C[C@H]1CC2(CCN(C3=CC=C(C(=O)N4CCC(F)(CN5CCC6(CC5)COC5=C6C=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)CC2)CN1C1=CC=C(C#N)C(Cl)=C1	C48H53ClFN7O5	AR	P10275	CRBN	WO-2024146617-A1
TPD-M3WGMV	WO2024146617A1_333	.	C[C@H]1CC2(CCN(C3=NN=C(C(=O)N4CCC(CN5CCC6(CC5)COC5=C6C=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)CC2)CN1C1=CC=C(C#N)C(Cl)=C1	C46H52ClN9O5	AR	P10275	CRBN	WO-2024146617-A1
TPD-7UOXYH	WO2024146617A1_334	.	COC1(CN2CCC3(CC2)COC2=C3C=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=C2)CCN(C2=NN=C(C(=O)N[C@H]3CC[C@H](OC4=CC=C(C#N)C(Cl)=C4)CC3)C=C2)CC1	C44H47ClN8O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-2KBQQN	WO2024146617A1_335	.	C[C@H]1CC2(CCN(C3=CC=C(N4CCC(CN5CCC6(CC5)COC5=C6C=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)CC2)CN1C1=CC=C(C#N)C(Cl)=C1	C47H54ClN7O4	AR	P10275	CRBN	WO-2024146617-A1
TPD-2TCQ53	WO2024146617A1_336	.	N#CC1=CCC(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC(C#N)(CN5CCC6(CC5)COC5=C6C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)C=C3)CC2)C=C1Cl	C44H46ClN9O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-MJ46CT	WO2024146617A1_337	.	COC1=CC(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC(CN5CCC6(CC5)COC5=C6C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)C=C3)CC2)=CC=C1C#N	C44H48N8O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-BJP2I6	WO2024146617A1_338	.	CC1(CN2CCC3(CC2)COC2=C3C=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=C2)CCN(C2=NN=C(C(=O)N[C@H]3CC[C@H](OC4=CC=C(C#N)C(Cl)=C4)CC3)C=C2)CC1	C44H47ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-NFVQKA	WO2024146617A1_339	.	COC1=CC(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC(F)(CN5CCC6(CCC7=CC8=C(C=C7O6)C(=O)N(C6CCC(=O)NC6=O)C8=O)CC5)CC4)C=C3)CC2)=CC=C1C#N	C45H49FN8O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-ZY9GBQ	WO2024146617A1_34	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC5(CCC(N6CCC7(CCC8=CC9=C(C=C8O7)C(=O)N(C7CCC(=O)NC7=O)C9=O)CC6)CC5)C4)C=C3)CC2)C=C1Cl	C47H51ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-UBOQOZ	WO2024146617A1_340	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CCC(N4CCC(C)(CC5CCC6(CC5)COC5=CC7=C(C=C5O6)CN(C5CCC(=O)NC5=O)C7=O)CC4)C=C3)C2(C)C)=CC=C1C#N	C50H61N5O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-TJQ7VJ	WO2024146617A1_341	.	CN(C(=O)C1=NN=C(N2CCC(C)(CN3CCC4(CC3)COC3=C4C=CC4=C3CN(C3CCC(=O)NC3=O)C4=O)CC2)C=C1)[C@H]1CC[C@H](OC2=CC=C(C#N)C(Cl)=C2)CC1	C45H51ClN8O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-90E536	WO2024146617A1_342	.	N#CC1=C(C(F)(F)F)C=C(N2CCC(C3=CC=C(N4CCC(CN5CCC6(CC5)COC5=C6C=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)CC2)C=C1	C44H47F3N6O4	AR	P10275	CRBN	WO-2024146617-A1
TPD-KSZ53O	WO2024146617A1_343	.	C[C@H]1CC2(CCN(C3=CC=C(C(=O)N4CCC(F)(CN5CCC6(CC5)COC5=C6C=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)CC2)CN1C1=CC=C(C#N)C(C(F)(F)F)=C1	C49H53F4N7O5	AR	P10275	CRBN	WO-2024146617-A1
TPD-FB37N1	WO2024146617A1_344	.	C[C@H]1CC2(CCN(C3=CC=C(N4CCC(CN5CCC6(CCC7=CC8=C(C=C7O6)C(=O)N(C6CCC(=O)NC6=O)C8=O)CC5)CC4)C=C3)CC2)CN1C1=CC=C(C#N)C(Cl)=C1	C48H54ClN7O5	AR	P10275	CRBN	WO-2024146617-A1
TPD-FYOXFM	WO2024146617A1_345	.	C[C@H]1CC2(CCN(C3=CC=C(N4CCC(CN5CCC6(CC5)COC5=C6C=CC6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)CC2)CN1C1=CC=C(C#N)C(Cl)=C1	C47H52ClN7O5	AR	P10275	CRBN	WO-2024146617-A1
TPD-ZW1IPT	WO2024146617A1_346	.	C[C@H]1CC2(CCN(C3=NN=C(N4CCC(CN5CCC6(CC5)COC5=C6C=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)CC2)CN1C1=CC=C(C#N)C(Cl)=C1	C45H52ClN9O4	AR	P10275	CRBN	WO-2024146617-A1
TPD-NXN12H	WO2024146617A1_347	.	COC1(CN2CCC3(CC2)COC2=C3C=CC3=C2CN(C2CCC(=O)NC2=O)C3=O)CCN(C2=CC=C(N3CCC4(CC3)C[C@H](C)N(C3=CC=C(C#N)C(Cl)=C3)C4)C=C2)CC1	C48H56ClN7O5	AR	P10275	CRBN	WO-2024146617-A1
TPD-OO5TQU	WO2024146617A1_348	.	C[C@H]1CC2(CCN(C3=CC=C(CN4CCC(CN5CCC6(CC5)COC5=CC7=C(C=C56)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)C=C3)CC2)CN1C1=CC=C(C#N)C(Cl)=C1	C48H54ClN7O5	AR	P10275	CRBN	WO-2024146617-A1
TPD-9D2ZZ5	WO2024146617A1_349	.	C[C@H]1CC2(CCN(C3=CC=C(N4CCC(CN5CCC6(CC5)COC5=C(C=CC7=C5C(=O)N(C5CCC(=O)NC5=O)C7)C6)CC4)C=C3)CC2)CN1C1=CC=C(C#N)C(CI)=C1	C49H58IN7O4	AR	P10275	CRBN	WO-2024146617-A1
TPD-4DDSIC	WO2024146617A1_35	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC5(CC(N6CCC7(CCC8=CC9=C(C=C8O7)C(=O)N(C7CCC(=O)NC7=O)C9=O)CC6)C5)C4)C=C3)CC2)C=C1Cl	C45H47ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-E38UPX	WO2024146617A1_350	.	C[C@H]1CC2(CCN(C3=CC=C(C(=O)N4CCC(C)(CN5CCC6(CC5)COC5=C6C=CC6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)CC2)CN1C1=CC=C(C#N)C(Cl)=C1	C49H54ClN7O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-Q347KO	WO2024146617A1_351	.	N#CC1=CC=C(N2CCC3(CCN(C4=CC=C(C(=O)N5CCC(CN6CCC7(CC6)COC6=C7C=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)CC5)C=C4)CC3)C2)C=C1Cl	C47H52ClN7O5	AR	P10275	CRBN	WO-2024146617-A1
TPD-R51Z5X	WO2024146617A1_352	.	N#CC1=CC=C(N2CCC3(CCN(C4=CC=C(C(=O)N5CCC(CN6CCC7(CC6)COC6=C7C=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)CC5)C=C4)C3)C2)C=C1Cl	C46H50ClN7O5	AR	P10275	CRBN	WO-2024146617-A1
TPD-WUDVUO	WO2024146617A1_353	.	C[C@H]1CC2(CCN(C3=CC=C(N4CCC(CN5CCC6(CCC7=CC8=C(C=C7O6)CN(C6CCC(=O)NC6=O)C8=O)CC5)CC4)C=C3)CC2)CN1C1=CC=C(C#N)C(Cl)=C1	C48H56ClN7O4	AR	P10275	CRBN	WO-2024146617-A1
TPD-VRLODY	WO2024146617A1_354	.	C[C@H]1CC2(CCN(C3=CC=C(N4CCC(CN5CCC6(CCC7=C(O6)C6=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C6)CC5)CC4)C=C3)CC2)CN1C1=CC=C(C#N)C(Cl)=C1	C48H56ClN7O4	AR	P10275	CRBN	WO-2024146617-A1
TPD-O0G8FF	WO2024146617A1_355	.	N#CC1=C(C(F)(F)F)C=C(N2CCC(C3=CC=C(CN4CCC(CN5CC6(CCC7=CC8=C(C=C7O6)C(=O)N(C6CCC(=O)NC6=O)C8=O)C5)CC4)C=C3)CC2)C=C1	C44H45F3N6O5	AR	P10275	CRBN	WO-2024146617-A1
TPD-7PJ3DN	WO2024146617A1_356	.	C[C@H]1CC2(CCN(C3=NC=C(C(=O)N4CCC(CN5CCC6(CC5)COC5=C6C=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)CC2)CN1C1=CC=C(C#N)C(Cl)=C1	C47H53ClN8O5	AR	P10275	CRBN	WO-2024146617-A1
TPD-D7SUIS	WO2024146617A1_357	.	C[C@H]1CC2(CCN(C3=CN=C(C(=O)N4CCC(CN5CCC6(CC5)COC5=C6C=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)CC2)CN1C1=CC=C(C#N)C(Cl)=C1	C47H53ClN8O5	AR	P10275	CRBN	WO-2024146617-A1
TPD-CU9YDG	WO2024146617A1_358	.	COC1=CC(N2CC3(CCN(C4=CC=C(N5CCC(CN6CCC7(CC6)COC6=C7C=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)CC5)C=C4)CC3)C[C@@H]2C)=CC=C1C#N	C48H57N7O5	AR	P10275	CRBN	WO-2024146617-A1
TPD-CHTC1P	WO2024146617A1_359	.	C[C@H]1CC2(CCN(C3=CC=C(N4CCC(CN5CCC6(CC5)COC5=C6C=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)CC2)CN1C1=CC=C(C#N)C(C(F)(F)F)=C1	C48H54F3N7O4	AR	P10275	CRBN	WO-2024146617-A1
TPD-R9XJYD	WO2024146617A1_36	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC5(CC4)CC(F)(F)C4=CC6=C(C=C4O5)C(=O)N(C4CCC(=O)NC4=O)C6=O)C=C3)CC2)C=C1Cl	C38H34ClF2N7O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-4ULAHK	WO2024146617A1_360	.	C[C@H]1CC2(CCN(C3=CC=C(N4CCC(CN5CC6(CCC7=CC8=C(C=C7O6)C(=O)N(C6CCC(=O)NC6=O)C8=O)C5)CC4)C=C3)CC2)CN1C1=CC=C(C#N)C(Cl)=C1	C46H50ClN7O5	AR	P10275	CRBN	WO-2024146617-A1
TPD-G0FCE8	WO2024146617A1_361	.	C[C@H]1CC2(CCN(C3=CN=C(N4CCC(CN5CCC6(CC5)COC5=C6C=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)CC2)CN1C1=CC=C(C#N)C(Cl)=C1	C46H53ClN8O4	AR	P10275	CRBN	WO-2024146617-A1
TPD-EGVYMF	WO2024146617A1_362	.	N#CC1=CC=C(N2CCC3(CCN(C4=CC=C(C(=O)N5CCC(CN6CCC7(CC6)COC6=C7C=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)CC5)C=C4)CC3)CC2)C=C1Cl	C48H54ClN7O5	AR	P10275	CRBN	WO-2024146617-A1
TPD-U8MNMZ	WO2024146617A1_363	.	N#CC1=CC=C(N2CCC3(C2)CN(C2=CC=C(C(=O)N4CCC(CN5CCC6(CC5)COC5=C6C=CC6C(=O)N(C7CCC(=O)NC7=O)CC56)CC4)C=C2)C3)C=C1Cl	C45H50ClN7O5	AR	P10275	CRBN	WO-2024146617-A1
TPD-FVY9HB	WO2024146617A1_364	.	C[C@H]1CC2(CCN(C3=CC=C(N4CCC(CN5CC6(CCC7=CC8=C(C=C7O6)CN(C6CCC(=O)NC6=O)C8=O)C5)CC4)C=C3)CC2)CN1C1=CC=C(C#N)C(Cl)=C1	C46H52ClN7O4	AR	P10275	CRBN	WO-2024146617-A1
TPD-ZXWU4C	WO2024146617A1_365	.	C[C@H]1CC2(CCN(C3=CC=C(N4CCC(CN5CCC6(CC5)COC5=CC7=C(C=C56)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)C=C3)CC2)CN1C1=CC=C(C#N)C(Cl)=C1	C47H52ClN7O5	AR	P10275	CRBN	WO-2024146617-A1
TPD-0XT8DN	WO2024146617A1_366	.	N#CC1=C(Cl)C=C2CC3(CCN(C4=CC=C(N5CCC(CN6CCC7(CC6)COC6=C7C=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)CC5)C=C4)CC3)COC2=C1	C45H49ClN6O5	AR	P10275	CRBN	WO-2024146617-A1
TPD-PWYVNZ	WO2024146617A1_367	.	CC1CC2(CCN(C3=NN=C(C(=O)N4CCC(F)(CN5CCC6(CC5)COC5=C6C=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)CC2)CN1C1=CC=C(C#N)C(Cl)=C1	C46H51ClFN9O5	AR	P10275	CRBN	WO-2024146617-A1
TPD-TO10B7	WO2024146617A1_368	.	C[C@H]1CC2(CCN(C3=CC=C(N4CCC(CN5CCC6(CCC7=C(O6)C6=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C6=O)CC5)CC4)C=C3)CC2)CN1C1=CC=C(C#N)C(Cl)=C1	C48H54ClN7O5	AR	P10275	CRBN	WO-2024146617-A1
TPD-GG7J1U	WO2024146617A1_369	.	C[C@H]1CC2(CCN(C3=CC=C(N4CCC(CN5CC6(CCC7=C(O6)C6=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C6=O)C5)CC4)C=C3)CC2)CN1C1=CC=C(C#N)C(Cl)=C1	C46H50ClN7O5	AR	P10275	CRBN	WO-2024146617-A1
TPD-GOM9MU	WO2024146617A1_37	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CC(N5CCC6(CC5)OC5=NC7=C(C=C5CC6(F)F)C(=O)N(C5CCC(=O)NC5=O)C7=O)C4)C=C3)CC2)C=C1Cl	C40H38ClF2N9O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-0WPMGH	WO2024146617A1_370	.	COC1=CC(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC(CN5CCC6(CC5)COC5=CC7=C(C=C56)C(=O)N(C5CCC(=O)NC5=O)C7)CC4)C=C3)CC2)=CC=C1C#N	C44H50N8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-YVW7NX	WO2024146617A1_371	.	COC1(CN2CCC3(CC2)COC2=C3C=CC3=C2CN(C2CCC(=O)NC2=O)C3=O)CCN(C(=O)C2=CC=C(N3CCC4(CC3)C[C@H](C)N(C3=CC=C(C#N)C(Cl)=C3)C4)C=C2)CC1	C49H56ClN7O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-KEO1Q0	WO2024146617A1_372	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC(CN5CCC6(CC5)COC5=CC7=C(C=C56)C(=O)N(C5CCC(=O)NC5=O)C7)CC4)C=C3)CC2)C=C1Cl	C43H47ClN8O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-TYD5E9	WO2024146617A1_375	.	COC1=CC(N2CC3(CCN(C4=CC=C(C(=O)N5CCC(C)(CN6CCC7(CC6)COC6=C7C=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)CC5)C=C4)CC3)CC2C)=CC=C1C#N	C50H59N7O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-TKS3GI	WO2024146617A1_377	.	C[C@H]1CC2(CCN(C3=CC=C(C(=O)C4CCC(C)(CN5CCC6(CC5)COC5=C6C=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)CC2)CN1C1=CC=C(C#N)C(C(F)(F)F)=C1	C51H57F3N6O5	AR	P10275	CRBN	WO-2024146617-A1
TPD-SRNCHO	WO2024146617A1_378	.	C[C@H]1CC2(CCN(C3=CC=C(N4CCC(CN5CCC6(CC5)COC5=CC7=C(C=C56)C(=O)N(C5CCC(=O)NC5=O)C7)CC4)C=C3)CC2)CN1C1=CC=C(C#N)C(Cl)=C1	C47H54ClN7O4	AR	P10275	CRBN	WO-2024146617-A1
TPD-9WZMYB	WO2024146617A1_379	.	C[C@H]1CC2(CCN(C3=NN=C(C(=O)N4CCC(CN5CCC6(CC5)COC5=CC7=C(C=C56)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)C=C3)CC2)CN1C1=CC=C(C#N)C(Cl)=C1	C46H50ClN9O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-NV2255	WO2024146617A1_38	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC(N5CCC6(CC5)CC(F)(F)C5=CC7=C(C=C5O6)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)C=C3)CC2)C=C1Cl	C43H43ClF2N8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-AIKK6L	WO2024146617A1_380	.	C[C@H]1CC2(CCN(C3=CC=C(C(=O)N4CCC(C)(CN5CCC6(CC5)COC5=CC7=C(C=C56)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)C=C3)CC2)CN1C1=CC=C(C#N)C(Cl)=C1	C49H54ClN7O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-9DXNPG	WO2024146617A1_381	.	C[C@H]1CC2(CCN(C3=CC=C(C(=O)N4CCC(N5CCC6(CC5)COC5=C6C=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)CC2)CN1C1=CC=C(C#N)C(Cl)=C1	C47H52ClN7O5	AR	P10275	CRBN	WO-2024146617-A1
TPD-P2ED1I	WO2024146617A1_382	.	C[C@H]1CC2(CCN(CC3=CC=C(C(=O)N4CCC(CN5CCC6(CC5)COC5=CC7=C(C=C56)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)C=C3)CC2)CN1C1=CC=C(C#N)C(Cl)=C1	C49H54ClN7O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-LNQPM1	WO2024146617A1_383	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(CN4CCC5(CC4)COC4=C5C=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(CO)=C1	C48H54N6O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-FPPIFT	WO2024146617A1_385	.	C[C@H]1CC2(CCN(C3=CC=C(N4CCC(CN5CCC6(CC5)CC5=C(C=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C5)O6)CC4)C=C3)CC2)CN1C1=CC=C(C#N)C(Cl)=C1	C47H52ClN7O5	AR	P10275	CRBN	WO-2024146617-A1
TPD-WRSK3W	WO2024146617A1_386	.	C[C@H]1CC2(CCN(C3=CC=C(C(=O)N4CCC(CN5CCC6(CC5)COC5=CC7=C(C=C56)C(=O)N(C5CCC(=O)NC5=O)C7)CC4)C=C3)CC2)CN1C1=CN=C(C#N)C(Cl)=C1	C47H53ClN8O5	AR	P10275	CRBN	WO-2024146617-A1
TPD-9RMF8H	WO2024146617A1_387	.	N#CC1=C(C(F)(F)F)C=C(N2CCC(C3=CC=C(N4CCC(CN5CC6(CCC7=CC8=C(C=C7O6)C(=O)N(C6CCC(=O)NC6=O)C8=O)C5)CC4)C=C3)CC2)C=C1	C43H43F3N6O5	AR	P10275	CRBN	WO-2024146617-A1
TPD-KKAOYV	WO2024146617A1_388	.	N#CC1=CC=C(N2CCC3(CC2)CCN(C2=CC=C(C(=O)N4CCC(CN5CCC6(CC5)COC5=C6C=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C2)C3)C=C1Cl	C47H52ClN7O5	AR	P10275	CRBN	WO-2024146617-A1
TPD-87AO3Y	WO2024146617A1_389	.	N#CC1=CC=C(N2CCC3(CC2)CN(C2=CC=C(C(=O)N4CCC(CN5CCC6(CC5)COC5=C6C=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C2)C3)C=C1Cl	C46H50ClN7O5	AR	P10275	CRBN	WO-2024146617-A1
TPD-O3CO6G	WO2024146617A1_39	.	CC1(CN2CCC3(CCC4=CC5=C(C=C4O3)CN(C3CCC(=O)NC3=O)C5=O)CC2)CCN(C2=NN=C(C(=O)N[C@H]3CC[C@H](OC4=CC=C(C#N)C(Cl)=C4)CC3)C=C2)CC1	C45H51ClN8O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-WITXWZ	WO2024146617A1_390	.	N#CC1=CC=C(N2CC3(CCN(C4=CC=C(C(=O)N5CCC(CN6CCC7(CC6)COC6=C7C=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)CC5)C=C4)CC3)C2)C=C1Cl	C46H50ClN7O5	AR	P10275	CRBN	WO-2024146617-A1
TPD-5RH5IO	WO2024146617A1_391	.	N#CC1=C(Cl)C=C2CC3(CCN(C4=CC=C(C(=O)N5CCC(CN6CCC7(CC6)COC6=C7C=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)CC5)C=C4)CC3)COC2=C1	C46H49ClN6O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-V77I33	WO2024146617A1_392	.	CCN(CC1CN(C2=CC=C(C(=O)N3CCC(CN4CCC5(CC4)COC4=C5C=CC5=C4CN(C4CCC(=O)NC4=O)C5=O)CC3)C=C2)C1)C1=CC=C(C#N)C(Cl)=C1	C45H50ClN7O5	AR	P10275	CRBN	WO-2024146617-A1
TPD-T8HCAU	WO2024146617A1_393	.	N#CC1=CC=C(N2CC3(CCN(C4=CC=C(C(=O)N5CCC(CN6CCC7(CC6)COC6=C7C=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)CC5)C=C4)C3)C2)C=C1Cl	C45H48ClN7O5	AR	P10275	CRBN	WO-2024146617-A1
TPD-10UNQ7	WO2024146617A1_394	.	C[C@H]1CC2(CCN(C3=CC=C(N4CCC(C)(CN5CCC6(CC5)COC5=C6C=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)CC2)CN1C1=CC=C(C#N)C(Cl)=C1	C48H56ClN7O4	AR	P10275	CRBN	WO-2024146617-A1
TPD-QURDVC	WO2024146617A1_395	.	CC1=CC=C(N2CC3(CCN(C4=CC=C(N5CCC(CN6CC7(CCC8=C(C=C9C(=O)N(C%10CCC(=O)NC%10=O)CC9=C8)O7)C6)CC5)C=C4)CC3)C[C@@H]2C)C=C1Cl	C46H55ClN6O4	AR	P10275	CRBN	WO-2024146617-A1
TPD-NI5ZQ0	WO2024146617A1_397	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=CN=C(N4CCC(CN5CCC6(CC5)COC5=CC7=C(C=C56)C(=O)N(C5CCC(=O)NC5=O)C7)CC4)C=C3)CC2)C=C1Cl	C44H48ClN7O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-F57VUM	WO2024146617A1_398	.	N#CC1=C(Cl)C=C2OCC3(CCN(C(=O)C4=CC=C(N5CCC(CN6CCC7(CC6)COC6=C7C=CC7C(=O)N(C8CCC(=O)NC8=O)C(=O)C67)CC5)C=C4)CC3)OC2=C1	C45H47ClN6O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-ZAOWFK	WO2024146617A1_399	.	N#CC1=C(Cl)C=C2OCC3(CCN(C(=O)C4=CC=C(N5CCC(CN6CCC7(CC6)COC6=C7C=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)CC5)C=C4)CC3)OC2=C1	C45H47ClN6O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-FOJ3DU	WO2024146617A1_4	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC(CN5CC6(CCC7=CC8=C(C=C7O6)C(=O)N(C6CCC(=O)NC6=O)C8=O)C5)C(F)C4)C=C3)CC2)C=C1Cl	C42H42ClFN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-KHZQ58	WO2024146617A1_40	.	COC1(CN2CCC3(CCC4=CC5=C(C=C4O3)CN(C3CCC(=O)NC3=O)C5=O)CC2)CCN(C2=NN=C(C(=O)NC3CCC(OC4=CC=C(C#N)C(Cl)=C4)CC3)C=C2)CC1	C45H51ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-N89UC1	WO2024146617A1_400	.	C[C@H]1CC2(CCN(C3=CC=C(C(=O)N4CCC(CN5CCC6(CC5)COC5=C6C=CC6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)CC2)CN1C1=CC=C(C#N)C(Cl)=C1	C48H52ClN7O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-9FIPMD	WO2024146617A1_401	.	C[C@H]1CC2(CCN(C3=CC=C(N4CCC(C)(CN5CC6(CCC7=CC8=C(C=C7O6)CN(C6CCC(=O)NC6=O)C8=O)C5)CC4)C=C3)CC2)CN1C1=CC=C(C#N)C(Cl)=C1	C47H54ClN7O4	AR	P10275	CRBN	WO-2024146617-A1
TPD-6RK92Z	WO2024146617A1_403	.	C[C@H]1CC2(CCN(C3=CC=C(C(=O)N4CCC(CN5CC6(CCC7=C(C=C8CN(C9CCC(=O)NC9=O)C(=O)C8=C7)O6)C5)CC4)C=C3)CC2)CN1C1=CC=C(C#N)C(Cl)=C1	C47H52ClN7O5	AR	P10275	CRBN	WO-2024146617-A1
TPD-TH1J0J	WO2024146617A1_404	.	N#CC1=C(Cl)C=C2OC3(CCN(C(=O)C4=CC=C(N5CCC(CN6CCC7(CC6)COC6=C7C=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C=C4)CC3)COC2=C1	C45H45ClN6O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-R9L8X4	WO2024146617A1_405	.	N#CC1=C(Cl)C=C2OC3(CCN(C(=O)C4=CC=C(N5CCC(CN6CCC7(CC6)COC6=C7C=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)CC5)C=C4)CC3)COC2=C1	C45H47ClN6O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-093BIZ	WO2024146617A1_406	.	COC1(CN2CC3(CCC4=CC5=C(C=C4O3)CN(C3CCC(=O)NC3=O)C5=O)C2)CCN(C2=CC=C(N3CCC4(CC3)C[C@H](C)N(C3=CC=C(C#N)C(Cl)=C3)C4)C=C2)CC1	C47H54ClN7O5	AR	P10275	CRBN	WO-2024146617-A1
TPD-XS1UL5	WO2024146617A1_408	.	C[C@H]1CC2(CCN(C3=CC=C(N4CCC(CN5CCC6(CC5)COC5=CC7=C(C=C5C6)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)C=C3)CC2)CN1C1=CC=C(C#N)C(Cl)=C1	C48H54ClN7O5	AR	P10275	CRBN	WO-2024146617-A1
TPD-LL1HI9	WO2024146617A1_409	.	N#CC1=C(Cl)C=C2CC3(CCN(C(=O)C4=CC=C(N5CCC(CN6CCC7(CC6)COC6=C7C=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C=C4)CC3)COC2=C1	C46H47ClN6O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-1KZP0Z	WO2024146617A1_41	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC(CN5CCC6(CCC7=CC8C(=O)N(C9CCC(=O)NC9=O)CC8C=C7O6)CC5)CC4)C=C3)CC2)C=C1Cl	C44H51ClN8O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-4EQ4OM	WO2024146617A1_410	.	N#CC1=C(Cl)C=C2OC3(CCN(C4=CC=C(C(=O)N5CCC(CN6CCC7(CC6)COC6=C7C=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C=C4)CC3)COC2=C1	C45H45ClN6O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-8H4ROV	WO2024146617A1_411	.	C[C@H]1CC2(CCN(C3=CC=C(C(=O)N4CCC(C)(CN5CC6(CCC7=C(C=C8CN(C9CCC(=O)NC9=O)C(=O)C8=C7)O6)C5)CC4)C=C3)CC2)CN1C1=CC=C(C#N)C(Cl)=C1	C48H54ClN7O5	AR	P10275	CRBN	WO-2024146617-A1
TPD-GWC7NX	WO2024146617A1_412	.	N#CC1=C(Cl)C=C2OC3(CCN(C(=O)C4=NN=C(N5CCC(CN6CCC7(CC6)COC6=C7C=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)CC5)C=C4)CC3)CC(=O)C2=C1	C44H45ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-VARHTN	WO2024146617A1_413	.	N#CC1=C(Cl)C=C2CC3(CCN(C(=O)C4=CC=C(N5CCC(CN6CCC7(CC6)COC6C8=C(C=CC67)C(=O)N(C6CCC(=O)NC6=O)C8)CC5)C=C4)CC3)COC2=C1	C46H51ClN6O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-RNHH7T	WO2024146617A1_414	.	N#CC1=C(Cl)C=C2OC3(CCN(C4=CC=C(C(=O)N5CCC(CN6CCC7(CC6)COC6=C7C=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)CC5)C=C4)CC3)COC2=C1	C45H47ClN6O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-BWCSQR	WO2024146617A1_415	.	COC1(CN2CCC3(CCC4=CC5=C(C=C4O3)C(=O)N(C3CCC(=O)NC3=O)C5)CC2)CCN(C2=CC=C(N3CCC4(CC3)C[C@H](C)N(C3=CC=C(C#N)C(Cl)=C3)C4)C=C2)CC1	C49H58ClN7O5	AR	P10275	CRBN	WO-2024146617-A1
TPD-7UYSYF	WO2024146617A1_416	.	C[C@H]1CC2(CCN(C3=CC=C(N4CCC(CN5CCC6(CCC7=CC8=C(C=C7O6)C(=O)N(C6CCC(=O)NC6=O)C8)CC5)CC4)C=C3)CC2)CN1C1=CC=C(C#N)C(Cl)=C1	C48H56ClN7O4	AR	P10275	CRBN	WO-2024146617-A1
TPD-G4E775	WO2024146617A1_417	.	CC1CC2(CCN(C3=CC=C(C(=O)N4CCC(CN5CCC6(CCC7=CC8=C(C=C7O6)CN(C6CCC(=O)NC6=O)C8=O)CC5)CC4)C=C3)CC2)CN1C1=CC=C(C#N)C(Cl)=C1	C49H56ClN7O5	AR	P10275	CRBN	WO-2024146617-A1
TPD-GSY17E	WO2024146617A1_418	.	C[C@H]1CC2(CCN(C3=CC=C(C(=O)N4CCC(CN5CCC6(CCC7=CC8=C(C=C7O6)C(=O)N(C6CCC(=O)NC6=O)C8)CC5)CC4)C=C3)CC2)CN1C1=CC=C(C#N)C(Cl)=C1	C49H56ClN7O5	AR	P10275	CRBN	WO-2024146617-A1
TPD-W9AZ8J	WO2024146617A1_419	.	CC1CC2(CCN(C3=CC=C(C(O)N4CCC(F)(CN5CC6(CCC7=C(C=C8CN(C9CCC(=O)NC9=O)C(=O)C8=C7)O6)C5)CC4)C=C3)CC2)CN1C1=CC=C(C#N)C(Cl)=C1	C47H53ClFN7O5	AR	P10275	CRBN	WO-2024146617-A1
TPD-DKVMXS	WO2024146617A1_42	.	CCC(=O)NC(=O)C(C)N1CC2=C(C=C3CCC4(CCN(C5CN(C6=NN=C(C(=O)N[C@H]7CC[C@H](OC8=CC(Cl)=C(C#N)C=C8)CC7)C=C6)C5)CC4)OC3=C2)C1=O	C42H47ClN8O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-UPG59U	WO2024146617A1_420	.	C[C@H]1CC2(CCN(C3=CCC(C(O)N4CCC(CN5CC6(CCC7=CC8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8C=C7O6)C5)CC4)C=C3)CC2)CN1C1=CC=C(C#N)C(Cl)=C1	C47H56ClN7O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-22K0KG	WO2024146617A1_421	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(CN5CCC6(CC5)COC5=CC7=C(C=C56)C(=O)N(C5CCC(=O)NC5=O)C7)CC4)C=C3)C2(C)C)=CC=C1C#N	C48H56N6O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-IJ3V9O	WO2024146617A1_424	.	N#CC1=C(Cl)C=C2CC3(CCN(C(=O)C4=NN=C(N5CCC(CN6CCC7(CC6)COC6=C7C=CC7=C6CN(C6CCC(=O)NC6=O)C7=O)CC5)C=C4)CC3)COC2=C1	C44H47ClN8O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-GYA3V7	WO2024146617A1_43	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC(F)(CN5CCC6(CCC7=CC8=C(C=C7O6)CN(C6CCC(=O)NC6=O)C8=O)CC5)CC4)C=C3)CC2)C=C1Cl	C44H48ClFN8O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-O4BPLL	WO2024146617A1_44	.	CC[C@@H](CCCOC1=CC=C(C#N)C(Cl)=C1)NC(=O)C1=NN=C(N2CCC(CN3CCC4(CCC5=CC6=C(C=C5O4)C(=O)N(C4CCC(=O)NC4=O)C6)CC3)CC2)C=C1	C44H51ClN8O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-8BBL4B	WO2024146617A1_45	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC(F)(CN5CCC6(CCC7=CC8=C(C=C7O6)C(=O)N(C6CCC(=O)NC6=O)C8)CC5)CC4)C=C3)CC2)C=C1Cl	C44H48ClFN8O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-8XQT56	WO2024146617A1_46	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CC(N5CCC6(CCC7=CC8=C(C=C7O6)C(=O)N(C6CCC(=O)NC6=O)C8)CC5)C4)C=C3)CC2)C=C1Cl	C41H43ClN8O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-4G2A07	WO2024146617A1_47	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC5(CC4)CC(N4CCC6(CC4)COC4=CC7=C(C=C46)C(=O)N(C4CCC(=O)NC4)C7=O)C5)C=C3)CC2)C=C1Cl	C45H49ClN8O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-F438QA	WO2024146617A1_48	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC(N5CCC6(CC5)COC5=C6C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)C=C3)CC2)C=C1Cl	C42H43ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-TUEGOV	WO2024146617A1_49	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CC(N5CCC6(CC5)COC5=C6C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)C=C3)CC2)C=C1Cl	C40H39ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-NKW2S5	WO2024146617A1_5	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CC(N5CC6(CCC7=CC8=C(C=C7O6)C(=O)N(C6CCC(=O)NC6=O)C8=O)C5)C4)C=C3)CC2)C=C1Cl	C39H37ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-7918EY	WO2024146617A1_50	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CC5(CC(N6CCC7(CC6)COC6=CC8=C(C=C67)C(=O)N(C6CCC(=O)NC6=O)C8=O)C5)C4)C=C3)CC2)C=C1Cl	C43H43ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-IXSO1I	WO2024146617A1_51	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC5(CCC(N6CCC7(CC6)COC6=CC8=C(C=C67)C(=O)N(C6CCC(=O)NC6=O)C8=O)CC5)CC4)C=C3)CC2)C=C1Cl	C47H51ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-URNZXF	WO2024146617A1_52	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC5(CC4)COC4=CC6=C(C=C45)C(=O)N(C4CCC(=O)NC4=O)C6=O)C=C3)CC2)C=C1Cl	C37H34ClN7O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-DT5SGZ	WO2024146617A1_53	.	N#CC1=CCC(O[C@H]2CC[C@H](NC(=O)C3=NN=C(C4CC5(CCC(N6CCC7(CC6)COC6=CC8=C(C=C67)C(=O)N(C6CCC(=O)NC6=O)C8=O)CC5)C4)C=C3)CC2)C=C1Cl	C46H50ClN7O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-PE6N1S	WO2024146617A1_54	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC5(CC(N6CCC7(CC6)COC6=CC8=C(C=C67)C(=O)N(C6CCC(=O)NC6=O)C8=O)C5)C4)C=C3)CC2)C=C1Cl	C44H45ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-H97GCA	WO2024146617A1_55	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CC(CN5CCC6(CC5)COC5=C6/C=C/C(=O)N(C6CCC(=O)NC6=O)C(=O)/C=C/5)C4)C=C3)CC2)C=C1Cl	C41H43ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-G2J6YG	WO2024146617A1_56	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC(CN5CCC6(CC5)COC5=C6C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)C=C3)CC2)C=C1Cl	C43H45ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-PRFKUF	WO2024146617A1_57	.	N#CC1=C(Cl)C=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CC[C@@H](CN5CCC6(CC5)COC5=C6C=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)C4)C=C3)CC2)C=C1	C42H43ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-CVWAML	WO2024146617A1_58	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CC[C@H](CN5CCC(COC6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C4)C=C3)CC2)C=C1Cl	C42H45ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-PV52CI	WO2024146617A1_59	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CC(CN5CCC6(CC5)COC5=CC7=C(C=C5C6)C(=O)N(C5CCC(=O)NC5=O)C7=O)C4)C=C3)CC2)C=C1Cl	C42H43ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-MDR8I6	WO2024146617A1_6	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CC5(CCC6=CC7=C(C=C6O5)C(=O)N(C5CCC(=O)NC5=O)C7=O)C4)C=C3)CC2)C=C1Cl	C36H32ClN7O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-JWCB85	WO2024146617A1_60	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC5(CC4)COC4=CC6=C(C=C4C5)C(=O)N(C4CCC(=O)NC4=O)C6=O)C=C3)CC2)C=C1Cl	C38H36ClN7O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-VYM7NO	WO2024146617A1_62	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC5(CCC(N6CCC7(CC6)COC6=CC8=C(C=C6C7)C(=O)N(C6CCC(=O)NC6=O)C8=O)CC5)C4)C=C3)CC2)C=C1Cl	C47H51ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-YLC7OU	WO2024146617A1_63	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC5(CC(N6CCC7(CC6)COC6=CC8=C(C=C6C7)C(=O)N(C6CCC(=O)NC6=O)C8=S)C5)C4)C=C3)CC2)C=C1Cl	C45H47ClN8O6S	AR	P10275	CRBN	WO-2024146617-A1
TPD-WLTIKY	WO2024146617A1_64	.	N#CC1=CCC(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC5(CCC(N6CCC7(CC6)COC6=CC8=C(C=C6C7)C(=O)N(C6CCC(=O)NC6=O)C8=O)CC5)CC4)C=C3)CC2)C=C1Cl	C48H55ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-CC9IB2	WO2024146617A1_65	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CC5(CCC(N6CCC7(CC6)COC6=CC8=C(C=C6C7)C(=O)N(C6CCC(=O)NC6=O)C8=O)CC5)C4)C=C3)CC2)C=C1Cl	C46H49ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-OUAOE5	WO2024146617A1_66	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CC5(CC(N6CCC7(CC6)COC6=CC8=C(C=C6C7)C(=O)N(C6CCC(=O)NC6=O)C8=O)C5)C4)C=C3)CC2)C=C1Cl	C44H45ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-NPW5Q1	WO2024146617A1_67	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC(F)(CN5CCC6(CC5)COC5=CC7=C(C=C5C6)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)C=C3)CC2)C=C1Cl	C44H46ClFN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-MXK03Z	WO2024146617A1_68	.	CCN(CCCCN1CCC2(CC1)COC1=CC3=C(C=C1C2)C(=O)N(C1CCC(=O)NC1=O)C3=O)C1=NN=C(C(=O)N[C@H]2CC[C@H](OC3=CC=C(C#N)C(Cl)=C3)CC2)C=C1	C44H49ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-X4XOXT	WO2024146617A1_69	.	COC1(CN2CCC3(CC2)COC2=CC4=C(C=C2C3)C(=O)N(C2CCC(=O)NC2=O)C4=O)CCN(C2=NN=C(C(=O)N[C@H]3CC[C@H](OC4=CC=C(C#N)C(Cl)=C4)CC3)C=C2)CC1	C45H49ClN8O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-K05KRB	WO2024146617A1_7	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC(CN5CC6(CCC7=CC8C(=O)N(C9CCC(=O)NC9=O)CC8C=C7O6)C5)CC4)C=C3)CC2)C=C1O	C42H48N8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-32V97H	WO2024146617A1_70	.	N#CC1=CC=C(OC2CCC(NC(=O)C3=NN=C(N4CCC(N5CCC6(CC5)COC5=CC7=C(C=C5C6)C(=O)N(C5CCC(=O)NC5=O)C7=O)CC4)C=C3)CC2)C=C1Cl	C43H45ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-CNFPOH	WO2024146617A1_71	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC5(CC4)CC(N4CCC6(CC4)COC4=CC7=C(C=C4C6)C(=O)N(C4CCC(=O)NC4=O)C7=O)C5)C=C3)CC2)C=C1Cl	C46H49ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-F1T6S1	WO2024146617A1_72	.	CC[C@H](CCCNC(=O)C1=NN=C(N2CCC(CN3CCC4(CC3)COC3=CC5=C(C=C3C4)C(=O)N(C3CCC(=O)NC3=O)C5=O)CC2)C=C1)OC1=CC=C(C#N)C(Cl)=C1	C44H49ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-0I6Y9U	WO2024146617A1_73	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CC[C@@H](CN5CCC6(CC5)COC5=CC7=C(C=C5C6)C(=O)N(C5CCC(=O)NC5=O)C7=O)C4)C=C3)CC2)C=C1Cl	C43H45ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-SFK6V5	WO2024146617A1_74	.	N#CC1=CC=C(C[C@H]2CC[C@H](NC(=O)C3=CN=C(N4CC[C@H](CN5CCC6(CC5)COC5=CC7=C(C=C5C6)C(=O)N(C5CCC(=O)NC5=O)C7=O)C4)C=C3)CC2)C=C1Cl	C45H48ClN7O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-3TIJ4L	WO2024146617A1_75	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC5(CC4)CO/C=C/C4=C(/C=C/O5)C(=O)N(C5CCC(=O)NC5=O)C4=O)C=C3)CC2)C=C1Cl	C37H36ClN7O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-GL482I	WO2024146617A1_77	.	N#CC1=CC=C(O[C@H]2CC[C@@H](NC(=O)C3=CC=C(N4CCC(F)(CN5CCC6(CC5)COC5=CC7=C(C=C5O6)CN(C5CCC(=O)NC5=O)C7=O)CC4)N=N3)CC2)C=C1Cl	C43H46ClFN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-R1JHK7	WO2024146617A1_8	.	N#CC1CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC(CN5CC6(CCC7=C(C=C8C(=O)N(C9CCC(=O)NC9=O)CC8=C7)O6)C5)CC4)C=C3)CC2)C=C1Cl	C42H47ClN8O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-D9ZG5J	WO2024146617A1_80	.	CC1(CN2CC3(CCC4=CC5=C(C=C4O3)CN(C3CCC(=O)NC3=O)C5=O)C2)CCN(C2=NN=C(C(=O)N[C@H]3CC[C@H](OC4C=C(Cl)C(C#N)=CC4)CC3)C=C2)CC1	C43H49ClN8O6	AR	P10275	CRBN	WO-2024146617-A1
TPD-N1WUUE	WO2024146617A1_84	.	CC1(C)C(=O)N(C2=CC(C(F)(F)F)=C(C#N)C=C2)C(=S)N1C1=CC=C(C(=O)N2CC(CN3CCC4(CCC5CC6=C(C=C5O4)C(=O)N(C4CCC(=O)NC4=O)C6=O)CC3)C2)C(F)=C1	C44H41F4N7O7S	AR	P10275	CRBN	WO-2024146617-A1
TPD-IFL1EZ	WO2024146617A1_87	.	CC1(C)C(=O)N(C2=CC(C(F)(F)F)=C(C#N)C=C2)C(=S)N1C1=CC=C(C(=O)N2CCC(CN3CCN(C4=C(F)C=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)C(F)=C1	C43H39F5N8O6S	AR	P10275	CRBN	WO-2024146617-A1
TPD-HD9SPT	WO2024146617A1_9	.	COC1(CN2CC3(CCC4=CC5=C(C=C4O3)C(=O)N(C3CCC(=O)NC3=O)C5)C2)CCN(C2=NN=C(C(=O)N[C@H]3CC[C@H](OC4=CC=C(C#N)C(Cl)=C4)CC3)C=C2)CC1	C43H47ClN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-HXCD5E	WO2024146617A1_90	.	CC1(C)C(=O)N(C2=CC(C(F)(F)F)=C(C#N)C=C2)C(=S)N1C1=CC=C(C(=O)N2CC(N3CC4(CCC5=CC6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6C=C5O4)C3)C2)C(F)=C1	C41H35F4N7O7S	AR	P10275	CRBN	WO-2024146617-A1
TPD-8ZRXGI	WO2024146617A1_94	.	CC1(C)C(=O)N(C2=CC(C(F)(F)F)=C(C#N)C=C2)C(=S)N1C1=CC=C(C(=O)N2CC(N3CCC4(CC3)COC3=C4C=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=C3)C2)C(F)=C1	C42H35F4N7O7S	AR	P10275	CRBN	WO-2024146617-A1
TPD-GHR2MN	WO2024146617A1_95	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=NN=C(N4CCC(F)(CN5CCC6(CCC7=C(O6)C6=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C6=O)CC5)CC4)C=C3)CC2)C=C1Cl	C44H46ClFN8O7	AR	P10275	CRBN	WO-2024146617-A1
TPD-60HDAL	WO2024146617A1_96	.	COC1(CN2CCC3(CCC4=C(O3)C3=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C3=O)CC2)CCN(C2=NN=C(C(=O)N[C@H]3CC[C@H](OC4=CC=C(C#N)C(Cl)=C4)CC3)C=C2)CC1	C45H49ClN8O8	AR	P10275	CRBN	WO-2024146617-A1
TPD-97JLFR	WO2024187066A1_1	.	CC(=O)N1CCC2=C(C1)C(C1=CC=CC3=C1C=NC(C1=CN=C(C(=O)NCC#CC4=CC=CC5=C4CN(C4CCC(=O)NC4=O)C5=O)C=C1)=C3)NN2C1CCOCC1	C44H42N8O6	CBP;P300	Q92793/Q09472	CRBN	WO-2024187066-A1
TPD-8Z62IC	SCHEMBL31086957	5-[8-[5-acetyl-1-(oxan-4-yl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-3-yl]isoquinolin-3-yl]-N-[4-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]but-3-ynyl]pyridine-2-carboxamide	CC(=O)N1CCC2=C(C1)C(C1=CC=CC3=C1C=NC(C1=CN=C(C(=O)NCCC#CC4=CC=CC5=C4CN(C4CCC(=O)NC4=O)C5=O)C=C1)=C3)=NN2C1CCOCC1	C45H42N8O6	CBP;P300	Q92793/Q09472	CRBN	WO-2024187066-A1
TPD-636SL3	WO2024187066A1_3	.	CC(=O)N1CCC2=C(C1)C(C1=CC=CC3=C1C=NC(C1=CN=C(C(=O)NCCCC#CC4=CC=CC5=C4CN(C4CCC(=O)NC4=O)C5=O)C=C1)=C3)NN2C1CCOCC1	C46H46N8O6	CBP;P300	Q92793/Q09472	CRBN	WO-2024187066-A1
TPD-MM6LG8	SCHEMBL31086901	5-[8-[5-acetyl-1-(oxan-4-yl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-3-yl]isoquinolin-3-yl]-N-[5-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]pent-4-ynyl]pyridine-2-carboxamide	CC(=O)N1CCC2=C(C1)C(C1=CC=CC3=C1C=NC(C1=CN=C(C(=O)NCCCC#CC4=CC=CC5=C4CN(C4CCC(=O)NC4=O)C5=O)C=C1)=C3)=NN2C1CCOCC1	C46H44N8O6	CBP;P300	Q92793/Q09472	CRBN	WO-2024187066-A1
TPD-WE44D4	WO2024187066A1_5	.	CC(=O)N1CCC2=C(C1)C(C1=CC=CC3=C1C=NC(C1=CN=C(C(=O)NCCCCCC#CC4=CC=CC5=C4CN(C4CCC(=O)NC4=O)C5=O)C=C1)=C3)NN2C1CCOCC1	C48H50N8O6	CBP;P300	Q92793/Q09472	CRBN	WO-2024187066-A1
TPD-9THZ9N	SCHEMBL31086910	5-[8-[5-acetyl-1-(oxan-4-yl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-3-yl]isoquinolin-3-yl]-N-[4-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]but-3-ynyl]pyridine-2-carboxamide	CC(=O)N1CCC2=C(C1)C(C1=CC=CC3=C1C=NC(C1=CN=C(C(=O)NCCC#CC4=CC=CC5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)C=C1)=C3)=NN2C1CCOCC1	C45H40N8O7	CBP;P300	Q92793/Q09472	CRBN	WO-2024187066-A1
TPD-IAP4F2	SCHEMBL31086938	3-[7-[2-[1-[5-[8-[5-acetyl-1-(oxan-4-yl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-3-yl]isoquinolin-3-yl]pyridine-2-carbonyl]piperidin-4-yl]ethynyl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione	CC(=O)N1CCC2=C(C1)C(C1=CC=CC3=C1C=NC(C1=CN=C(C(=O)N4CCC(C#CC5=CC=CC6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)C=C1)=C3)=NN2C1CCOCC1	C48H46N8O6	CBP;P300	Q92793/Q09472	CRBN	WO-2024187066-A1
TPD-FE59NA	SCHEMBL31134269	US20240374588, Example 1; BDBM704307; BDBM704308; US20240374588, Example 1; US20240374588, Example 2	COC1=CC2=NN(C3CCC(N(C)CCCCC4=C5C(=CC=C4)N(C4CCC(=O)NC4=O)C(=O)N5C)CC3)C=C2C=C1C(=O)NC1=CN=C2C=CC=NN12	C39H44N10O5	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-Y84FO8	SCHEMBL31134291	US20240374588, Example 9; BDBM704317; BDBM704319; US20240374588, Example 9; US20240374588, Example 10	COC1=CC2=NN(C3CCC(N(C)C4CCN(CCCC5=C6C(=CC=C5)N(C5CCC(=O)NC5=O)C(=O)N6C)CC4)CC3)C=C2C=C1C(=O)NC1=CN=C2C=CC=NN12	C43H51N11O5	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-S9KS9Y	WO2024209044A1_100	.	COC1=CC2=NN([C@H]3CC[C@@H](CN4CCC(C5=CC6=CC=C(N7CCC(=O)NC7=O)C=C6N5C)CC4)CC3)C=C2C=C1C(=O)NC1=CN=C2C=CC=NN12	C40H44N10O4	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-E6S59D	SCHEMBL31134400	US20240374588, Example 11; BDBM704321; BDBM704323; US20240374588, Example 11; US20240374588, Example 12; 2-(4-(4-(4-(1-(2,6-Dioxopiperidin-3-yl)-3-methyl-2-oxo-2,3-dihydro-1H-benzo[d]imidazol-5-yl)piperazin-1-yl)piperidin-1-yl)cyclohexyl)-N-(imidazo[1,2-b]pyridazin-3-yl)-6-methoxy-2H-indazole-5-carboxamide-Isomer 1 & Isomer 2	COC1=CC2=NN(C3CCC(N4CCC(N5CCN(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC5)CC4)CC3)C=C2C=C1C(=O)NC1=CN=C2C=CC=NN12	C43H50N12O5	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-0NF9TL	SCHEMBL31134526	US20240374588, Example 13; BDBM704324; BDBM704325; US20240374588, Example 13; US20240374588, Example 14	COC1=CC2=NN(C3CCC(N(C)C4CCN(CC5=C6C(=CC=C5)N(C5CCC(=O)NC5=O)C(=O)N6C)CC4)CC3)C=C2C=C1C(=O)NC1=CN=C2C=CC=NN12	C41H47N11O5	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-6EQKEL	SCHEMBL31134369	2-[4-[3-[3-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-4-yl]propoxy]propyl-methylamino]cyclohexyl]-N-imidazo[1,2-b]pyridazin-3-yl-6-methoxyindazole-5-carboxamide	COC1=CC2=NN(C3CCC(N(C)CCCOCCCC4=C5C(=CC=C4)N(C4CCC(=O)NC4=O)C(=O)N5C)CC3)C=C2C=C1C(=O)NC1=CN=C2C=CC=NN12	C41H48N10O6	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-9MZSSM	SCHEMBL31134430	US20240374588, Example 19; BDBM704352; BDBM704353; US20240374588, Example 19; US20240374588, Example 20	COC1=CC2=NN(C3CCC(NCCOC4=CC=C5C(=O)N(C6CCC(=O)NC6=O)CC5=C4)CC3)C=C2C=C1C(=O)NC1=CN=C2C=CC=NN12	C36H37N9O6	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-AZ5FI3	SCHEMBL31134385	US20240374588, Example 21; BDBM704354; BDBM704355; US20240374588, Example 21; US20240374588, Example 22	COC1=CC2=NN(C3CCC(NCCN4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)CC6=C5)CC4)CC3)C=C2C=C1C(=O)NC1=CN=C2C=CC=NN12	C40H45N11O5	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-MPCOYU	SCHEMBL31134384	US20240374588, Example 23; BDBM704356; BDBM704357; US20240374588, Example 23; US20240374588, Example 24; 2-((1r,4r)-4-((4-(4-(1-(2,6-Dioxopiperidin-3-yl)-3-methyl-2-oxo-2,3-dihydro-1H-benzo[d]imidazol-5-yl)piperazin-1-yl)piperidin-1-yl)methyl)cyclohexyl)-N-(imidazo[1,2-b]pyridazin-3-yl)-6-methoxy-2H-indazole-5-carboxamide	COC1=CC2=NN(C3CCC(NCCN4CCC(CN5CCN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)CC7=C6)CC5)CC4)CC3)C=C2C=C1C(=O)NC1=CN=C2C=CC=NN12	C46H56N12O5	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-5EK4I5	SCHEMBL31134263	2-[4-[[4-[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperazin-1-yl]piperidin-1-yl]methyl]cyclohexyl]-N-imidazo[1,2-b]pyridazin-3-yl-6-methoxyindazole-5-carboxamide	COC1=CC2=NN([C@H]3CC[C@H](CN4CCC(N5CCN(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC5)CC4)CC3)C=C2C=C1C(=O)NC1=CN=C2C=CC=NN12	C44H52N12O5	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-L1HL36	SCHEMBL31134494	US20240374588, Example 25; BDBM704358; US20240374588, Example 25; N-(1-Cyclopropyl-2-oxo-1,2-dihydropyridin-3-yl)-2-((1r,4r)-4-((4-(4-(1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxo-2,3-dihydro-1H-benzo[d]imidazol-5-yl)piperazin-1-yl)piperidin-1-yl)methyl)cyclohexyl)-6-methoxy-2H-indazole-5-carboxamide	COC1=CC2=NN([C@H]3CC[C@H](CN4CCC(N5CCN(C6=CC7=C(C=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC5)CC4)CC3)C=C2C=C1C(=O)NC1=CC=CN(C2CC2)C1=O	C46H56N10O6	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-067VZH	SCHEMBL31134311	US20240374588, Example 26; BDBM704359; US20240374588, Example 26; 2-((1r,4r)-4-((4-((3-(1-(2,6-Dioxopiperidin-3-yl)-3-methyl-2-oxo-2,3-dihydro-1H-benzo[d]imidazol-4-yl)prop-2-yn-1-yl)oxy)piperidin-1-yl)methyl)cyclohexyl)-N-(imidazo[1,2-b]pyridazin-3-yl)-6-methoxy-2H-indazole-5-carboxamide	COC1=CC2=NN([C@H]3CC[C@H](CN4CCC(OCC#CC5=C6C(=CC=C5)N(C5CCC(=O)NC5=O)C(=O)N6C)CC4)CC3)C=C2C=C1C(=O)NC1=CN=C2C=CC=NN12	C43H46N10O6	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-REQNJW	WO2024209044A1_27	.	COC1=CC2=NN([C@H]3CC[C@H](CN4CCC(OCC#CC5=C6NC(=O)N(C7CCC(=O)NC7=O)C6=CC=C5)CC4)CC3)C=C2C=C1C(=O)NC1=CC=CN(C2CC2)C1=O	C44H48N8O7	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-K8D0AP	SCHEMBL31134284	US20240374588, Example 28; BDBM704361; US20240374588, Example 28; 2-((1r,4r)-4-(4-((3-(1-(2,6-Dioxopiperidin-3-yl)-3-methyl-2-oxo-2,3-dihydro-1H-benzo[d]imidazol-4-yl)prop-2-yn-1-yl)oxy)piperidine-1-carbonyl)cyclohexyl)-N-(imidazo[1,2-b]pyridazin-3-yl)-6-methoxy-2H-indazole-5-carboxamide	COC1=CC2=NN([C@H]3CC[C@H](C(=O)N4CCC(OCC#CC5=C6C(=CC=C5)N(C5CCC(=O)NC5=O)C(=O)N6C)CC4)CC3)C=C2C=C1C(=O)NC1=CN=C2C=CC=NN12	C43H44N10O7	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-BSQXWK	SCHEMBL31134342	US20240374588, Example 29; BDBM704362; US20240374588, Example 29; N-(1-Cyclopropyl-2-oxo-1,2-dihydropyridin-3-yl)-2-((1r,4r)-4-(4-((3-(1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxo-2,3-dihydro-1H-benzo[d]imidazol-4-yl)prop-2-yn-1-yl)oxy)piperidine-1-carbonyl)cyclohexyl)-6-methoxy-2H-indazole-5-carboxamide	COC1=CC2=NN([C@H]3CC[C@H](C(=O)N4CCC(OCC#CC5=C6C(=CC=C5)N(C5CCC(=O)NC5=O)C(=O)N6C)CC4)CC3)C=C2C=C1C(=O)NC1=CC=CN(C2CC2)C1=O	C45H48N8O8	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-LQ5SWN	SCHEMBL31134475	US20240374588, Example 3; BDBM704310; BDBM704311; US20240374588, Example 3; US20240374588, Example 4	COC1=CC2=NN(C3CCC(N(C)C4CCN(CC#CC5=C6C(=CC=C5)N(C5CCC(=O)NC5=O)C(=O)N6C)CC4)CC3)C=C2C=C1C(=O)NC1=CN=C2C=CC=NN12	C43H47N11O5	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-U94I24	SCHEMBL31134295	US20240374588, Example 30; BDBM704363; US20240374588, Example 30; 2-((1r,4r)-4-((4-(2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindolin-5-yl)piperazin-1-yl)methyl)cyclohexyl)-N-(imidazo[1,2-b]pyridazin-3-yl)-6-methoxy-2H-indazole-5-carboxamide	COC1=CC2=NN([C@H]3CC[C@H](CN4CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)C=C2C=C1C(=O)NC1=CN=C2C=CC=NN12	C39H40N10O6	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-IVEIZZ	WO2024209044A1_31	.	CO/C(=C/C1=NN([C@H]2CC[C@H](CN3CCN(C4=CC5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5C=C4)CC3)CC2)C=C1C)CC(=O)NC1=CC=CN(C2CC2)C1=O	C41H50N8O7	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-2W2UYB	WO2024209044A1_32	.	COC1=CC2=NN([C@H]3CC[C@H](CN4CCC(N5C=CC6=C5C=CC=C6N5CCC(=O)NC5=O)CC4)CC3)C=C2C=C1C(=O)NC1=CN=C2C=CC=NN12	C39H42N10O4	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-UYVYT7	SCHEMBL31134392	US20240374588, Example 33; BDBM704366; US20240374588, Example 33; 2-((1r,4r)-4-((4-(4-(2,6-dioxopiperidin-3-yl)phenyl)piperazin-1-yl)methyl)cyclohexyl)-N-(imidazo[1,2-b]pyridazin-3-yl)-6-methoxy-2H-indazole-5-carboxamide	COC1=CC2=NN([C@H]3CC[C@H](CN4CCN(C5=CC=C(C6CCC(=O)NC6=O)C=C5)CC4)CC3)C=C2C=C1C(=O)NC1=CN=C2C=CC=NN12	C37H41N9O4	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-4HBDY7	SCHEMBL31134304	US20240374588, Example 34; BDBM704367; US20240374588, Example 34; 2-((1r,4r)-4-((4-(2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindolin-5-yl)piperazin-1-yl)methyl)cyclohexyl)-N-(imidazo[1,2-b]pyridazin-3-yl)-6-methoxy-2H-indazole-5-carboxamide	COC1=CC2=NN([C@H]3CC[C@H](CN4CCN(C5=CC6=C(C=C5F)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)C=C2C=C1C(=O)NC1=CN=C2C=CC=NN12	C39H39FN10O6	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-IIJ4XO	SCHEMBL31134445	US20240374588, Example 35; BDBM704368; US20240374588, Example 35; N-(1-Cyclopropyl-2-oxo-1,2-dihydropyridin-3-yl)-2-((1r,4r)-4-((4-(2-(2,6-dioxopiperidin-3-yl)-6-fluoro-1,3-dioxoisoindolin-5-yl)piperazin-1-yl)methyl)cyclohexyl)-6-methoxy-2H-indazole-5-carboxamide	COC1=CC2=NN(C3CCC(CN4CCN(C5=CC6=C(C=C5F)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)C=C2C=C1C(=O)NC1=CC=CN(C2CC2)C1=O	C41H43FN8O7	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-23HAP4	SCHEMBL31134409	US20240374588, Example 36; BDBM704369; US20240374588, Example 36; 2-((1r,4r)-4-(4-(2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindolin-5-yl)piperazine-1-carbonyl)cyclohexyl)-N-(imidazo[1,2-b]pyridazin-3-yl)-6-methoxy-2H-indazole-5-carboxamide	COC1=CC2=NN([C@H]3CC[C@H](C(=O)N4CCN(C5=CC6=C(C=C5)C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)C=C2C=C1C(=O)NC1=CN=C2C=CC=NN12	C39H38N10O7	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-HEOID3	SCHEMBL31134358	US20240374588, Example 37; BDBM704370; US20240374588, Example 37; N-(1-Cyclopropyl-2-oxo-1,2-dihydropyridin-3-yl)-2-((1r,4r)-4-((4-(4-(2,4-dioxotetrahydropyrimidin-1(2H)-yl)-1H-indol-1-yl)piperidin-1-yl)methyl)cyclohexyl)-6-methoxy-2H-indazole-5-carboxamide	COC1=CC2=NN([C@H]3CC[C@H](CN4CCC(N5C=CC6=C(N7CCC(=O)NC7=O)C=CC=C65)CC4)CC3)C=C2C=C1C(=O)NC1=CC=CN(C2CC2)C1=O	C41H46N8O5	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-ZAVWAY	SCHEMBL31134429	2-[4-[[4-[4-(2,6-dioxopiperidin-3-yl)indol-1-yl]piperidin-1-yl]methyl]cyclohexyl]-N-imidazo[1,2-b]pyridazin-3-yl-6-methoxyindazole-5-carboxamide	COC1=CC2=NN([C@H]3CC[C@H](CN4CCC(N5C=CC6=C5C=CC=C6C5CCC(=O)NC5=O)CC4)CC3)C=C2C=C1C(=O)NC1=CN=C2C=CC=NN12	C40H43N9O4	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-A8ASIE	SCHEMBL31134319	US20240374588, Example 39; BDBM704371; US20240374588, Example 39; N-(1-Cyclopropyl-2-oxo-1,2-dihydropyridin-3-yl)-2-((1r,4r)-4-((4-(4-(2,6-dioxopiperidin-3-yl)-1H-indol-1-yl)piperidin-1-yl)methyl)cyclohexyl)-6-methoxy-2H-indazole-5-carboxamide	COC1=CC2=NN([C@H]3CC[C@H](CN4CCC(N5C=CC6=C5C=CC=C6C5CCC(=O)NC5=O)CC4)CC3)C=C2C=C1C(=O)NC1=CC=CN(C2CC2)C1=O	C42H47N7O5	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-4GRNQA	SCHEMBL31134348	US20240374588, Example 40; BDBM704372; US20240374588, Example 40; 6-Cyclopropoxy-2-((1r,4r)-4-((4-(4-(2,4-dioxotetrahydropyrimidin-1(2H)-yl)-1H-indol-1-yl)piperidin-1-yl)methyl)cyclohexyl)-N-(imidazo[1,2-b]pyridazin-3-yl)-2H-indazole-5-carboxamide	O=C1CCN(C2=C3C=CN(C4CCN(C[C@H]5CC[C@H](N6C=C7C=C(C(=O)NC8=CN=C9C=CC=NN89)C(OC8CC8)=CC7=N6)CC5)CC4)C3=CC=C2)C(=O)N1	C41H44N10O4	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-INPNOO	SCHEMBL31134248	US20240374588, Example 41; BDBM704373; US20240374588, Example 41; 2-((1r,4r)-4-((4-(4-(2,4-Dioxotetrahydropyrimidin-1(2H)-yl)-2-methyl-1H-indol-1-yl)piperidin-1-yl)methyl)cyclohexyl)-N-(imidazo[1,2-b]pyridazin-3-yl)-6-methoxy-2H-indazole-5-carboxamide	COC1=CC2=NN([C@H]3CC[C@H](CN4CCC(N5C(C)=CC6=C(N7CCC(=O)NC7=O)C=CC=C65)CC4)CC3)C=C2C=C1C(=O)NC1=CN=C2C=CC=NN12	C40H44N10O4	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-WCG3PJ	SCHEMBL31134464	US20240374588, Example 42; BDBM704374; US20240374588, Example 42; 2-((1r,4r)-4-((4-(4-(2,4-Dioxotetrahydropyrimidin-1(2H)-yl)-3-methyl-1H-indol-1-yl)piperidin-1-yl)methyl)cyclohexyl)-N-(imidazo[1,2-b]pyridazin-3-yl)-6-methoxy-2H-indazole-5-carboxamide	COC1=CC2=NN([C@H]3CC[C@H](CN4CCC(N5C=C(C)C6=C5C=CC=C6N5CCC(=O)NC5=O)CC4)CC3)C=C2C=C1C(=O)NC1=CN=C2C=CC=NN12	C40H44N10O4	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-S5D221	SCHEMBL31134245	US20240374588, Example 43; BDBM704375; US20240374588, Example 43; 2-((1r,4r)-4-((4-(4-(2,4-Dioxotetrahydropyrimidin-1(2H)-yl)-1H-indol-1-yl)-[1,4''-bipiperidin]-1''-yl)methyl)cyclohexyl)-N-(imidazo[1,2-b]pyridazin-3-yl)-6-methoxy-2H-indazole-5-carboxamide	COC1=CC2=NN([C@H]3CC[C@H](CN4CCC(N5CCC(N6C=CC7=C6C=CC=C7N6CCC(=O)NC6=O)CC5)CC4)CC3)C=C2C=C1C(=O)NC1=CN=C2C=CC=NN12	C44H51N11O4	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-W8LKJS	SCHEMBL31134289	US20240374588, Example 44; BDBM704376; US20240374588, Example 44; 2-((1r,4r)-4-(4-(4-(2,4-Dioxotetrahydropyrimidin-1(2H)-yl)-1H-indol-1-yl)-[1,4''-bipiperidine]-1''-carbonyl)cyclohexyl)-N-(imidazo[1,2-b]pyridazin-3-yl)-6-methoxy-2H-indazole-5-carboxamide	COC1=CC2=NN([C@H]3CC[C@H](C(=O)N4CCC(N5CCC(N6C=CC7=C6C=CC=C7N6CCC(=O)NC6=O)CC5)CC4)CC3)C=C2C=C1C(=O)NC1=CN=C2C=CC=NN12	C44H49N11O5	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-BJ1Q32	SCHEMBL31134410	US20240374588, Example 45; BDBM704377; US20240374588, Example 45; 2-((1r,4r)-4-((4-((4-(2,4-Dioxotetrahydropyrimidin-1(2H)-yl)-1H-indol-1-yl)methyl)piperidin-1-yl)methyl)cyclohexyl)-N-(imidazo[1,2-b]pyridazin-3-yl)-6-methoxy-2H-indazole-5-carboxamide	COC1=CC2=NN([C@H]3CC[C@H](CN4CCC(CN5C=CC6=C5C=CC=C6N5CCC(=O)NC5=O)CC4)CC3)C=C2C=C1C(=O)NC1=CN=C2C=CC=NN12	C40H44N10O4	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-HML5ZM	SCHEMBL31134278	US20240374588, Example 46; BDBM704378; US20240374588, Example 46; 2-((1r,4r)-4-(2-(4-(4-(2,4-Dioxotetrahydropyrimidin-1(2H)-yl)-1H-indol-1-yl)piperidin-1-yl)ethyl)cyclohexyl)-N-(imidazo[1,2-b]pyridazin-3-yl)-6-methoxy-2H-indazole-5-carboxamide	COC1=CC2=NN([C@H]3CC[C@H](CCN4CCC(N5C=CC6=C5C=CC=C6N5CCC(=O)NC5=O)CC4)CC3)C=C2C=C1C(=O)NC1=CN=C2C=CC=NN12	C40H44N10O4	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-9DPNB1	SCHEMBL31134274	N-(1-cyclopropyl-2-oxopyridin-3-yl)-2-[4-[2-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]ethyl]cyclohexyl]-6-methoxyindazole-5-carboxamide	COC1=CC2=NN([C@H]3CC[C@H](CCN4CCC(N5C=CC6=C5C=CC=C6N5CCC(=O)NC5=O)CC4)CC3)C=C2C=C1C(=O)NC1=CC=CN(C2CC2)C1=O	C42H48N8O5	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-JWTY5Z	SCHEMBL31134434	US20240374588, Example 48; BDBM704380; US20240374588, Example 48; 2-((1r,4r)-4-((4-((4-(4-(2,4-Dioxotetrahydropyrimidin-1(2H)-yl)-1H-indol-1-yl)piperidin-1-yl)methyl)piperidin-1-yl)methyl)cyclohexyl)-N-(imidazo[1,2-b]pyridazin-3-yl)-6-methoxy-2H-indazole-5-carboxamide	COC1=CC2=NN([C@H]3CC[C@H](CN4CCC(CN5CCC(N6C=CC7=C(N8CCC(=O)NC8=O)C=CC=C76)CC5)CC4)CC3)C=C2C=C1C(=O)NC1=CN=C2C=CC=NN12	C45H53N11O4	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-WJUSCM	SCHEMBL31134493	US20240374588, Example 49; BDBM704381; US20240374588, Example 49	COC1=CC2=NN([C@H]3CC[C@H](C(=O)N4CCC(CN5CCC(N6C=CC7=C(N8CCC(=O)NC8=O)C=CC=C76)CC5)CC4)CC3)C=C2C=C1C(=O)NC1=CN=C2C=CC=NN12	C45H51N11O5	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-E0RZMI	SCHEMBL31134254	US20240374588, Example 5; BDBM704312; BDBM704313; US20240374588, Example 5; US20240374588, Example 6	COC1=CC2=NN(C3CCC(N(C)CCC#CC4=C5C(=CC=C4)N(C4CCC(=O)NC4=O)C(=O)N5C)CC3)C=C2C=C1C(=O)NC1=CN=C2C=CC=NN12	C39H40N10O5	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-GKHW62	SCHEMBL31134322	US20240374588, Example 50; BDBM704382; BDBM704383; US20240374588, Example 50; US20240374588, Example 51; 2-((1r,4r)-4-((4-(2-(4-(2,4-Dioxotetrahydropyrimidin-1(2H)-yl)-1H-indol-1-yl)ethyl)piperazin-1-yl)methyl)cyclohexyl)-N-(imidazo[1,2-b]pyridazin-3-yl)-6-methoxy-2H-indazole-5-carboxamide	COC1=CC2=NN(C3CCC(CN4CCC(CCN5CCC(N6C=CC7=C6C=CC=C7N6CCC(=O)NC6=O)CC5)CC4)CC3)C=C2C=C1C(=O)NC1=CN=C2C=CC=NN12	C46H55N11O4	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-S245BX	SCHEMBL31134460	2-[4-[[4-[2-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]ethyl]piperazin-1-yl]methyl]cyclohexyl]-N-imidazo[1,2-b]pyridazin-3-yl-6-methoxyindazole-5-carboxamide	COC1=CC2=NN([C@H]3CC[C@H](CN4CCN(CCN5C=CC6=C5C=CC=C6N5CCC(=O)NC5=O)CC4)CC3)C=C2C=C1C(=O)NC1=CN=C2C=CC=NN12	C40H45N11O4	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-H1YYQF	SCHEMBL31134420	US20240374588, Example 52; BDBM704384; US20240374588, Example 52	O=C1CCN(C2=CC=CC3=C2C=CN3C2CCN(CC(=O)N3CCC(N4C=C5C=C(C(=O)NC6=CN=C7C=CC=NN67)C(OC6CC6)=CC5=N4)CC3)CC2)C(=O)N1	C41H43N11O5	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-RDHRDM	SCHEMBL31134281	US20240374588, Example 53; BDBM704385; BDBM704386; US20240374588, Example 53; US20240374588, Example 54; 6-Cyclopropoxy-2-(1-(2-(4-((4-(2,4-dioxotetrahydropyrimidin-1(2H)-yl)-1H-indol-1-yl)methyl)piperidin-1-yl)acetyl)piperidin-4-yl)-N-(imidazo[1,2-b]pyridazin-3-yl)-2H-indazole-5-carboxamide	O=C1CCN(C2=CC=CC3=C2C=CN3C2CCN(C(=O)CN3CCC(N4C=C5C=C(C(=O)NC6=CN=C7C=CC=NN67)C(OC6CC6)=CC5=N4)CC3)CC2)C(=O)N1	C41H43N11O5	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-W0BZ1W	SCHEMBL31134395	6-cyclopropyloxy-2-[1-[2-[4-[[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]methyl]piperidin-1-yl]acetyl]piperidin-4-yl]-N-imidazo[1,2-b]pyridazin-3-ylindazole-5-carboxamide	O=C1CCN(C2=CC=CC3=C2C=CN3CC2CCN(CC(=O)N3CCC(N4C=C5C=C(C(=O)NC6=CN=C7C=CC=NN67)C(OC6CC6)=CC5=N4)CC3)CC2)C(=O)N1	C42H45N11O5	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-JQACLQ	WO2024209044A1_55	.	COC1=CC2=NN([C@H]3CC[C@H](CN4CCC(C5=CC6=CC=C(N7CCC(=O)NC7=O)C=C6N5C)CC4)CC3)C=C2C=C1C(=O)NC1=CN=C2C=CC=NN12	C40H44N10O4	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-5P1OS6	SCHEMBL31134375	2-[4-[[4-[1-(2,6-dioxopiperidin-3-yl)-3-methylindol-4-yl]piperazin-1-yl]methyl]cyclohexyl]-N-imidazo[1,2-b]pyridazin-3-yl-6-methoxyindazole-5-carboxamide	COC1=CC2=NN([C@H]3CC[C@H](CN4CCN(C5=C6C(C)=CN(C7CCC(=O)NC7=O)C6=CC=C5)CC4)CC3)C=C2C=C1C(=O)NC1=CN=C2C=CC=NN12	C40H44N10O4	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-6MD7V1	SCHEMBL31134271	US20240374588, Example 57; BDBM704387; US20240374588, Example 57; 2-((1r,4r)-4-((4-(4-((2,6-Dioxopiperidin-3-yl)carbamoyl)-3-fluorophenyl)piperazin-1-yl)methyl)cyclohexyl)-N-(imidazo[1,2-b]pyridazin-3-yl)-6-methoxy-2H-indazole-5-carboxamide	COC1=CC2=NN([C@H]3CC[C@H](CN4CCN(C5=CC(F)=C(C(=O)NC6CCC(=O)NC6=O)C=C5)CC4)CC3)C=C2C=C1C(=O)NC1=CN=C2C=CC=NN12	C38H41FN10O5	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-VUYZH6	SCHEMBL31134442	US20240374588, Example 58; BDBM704388; US20240374588, Example 58; N-(1-Cyclopropyl-2-oxo-1,2-dihydropyridin-3-yl)-2-((1r,4r)-4-((4-(4-((2,6-dioxopiperidin-3-yl)carbamoyl)-3-fluorophenyl)piperazin-1-yl)methyl)cyclohexyl)-6-methoxy-2H-indazole-5-carboxamide	COC1=CC2=NN([C@H]3CC[C@H](CN4CCN(C5=CC(F)=C(C(=O)NC6CCC(=O)NC6=O)C=C5)CC4)CC3)C=C2C=C1C(=O)NC1=CC=CN(C2CC2)C1=O	C40H45FN8O6	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-668P7R	SCHEMBL31134490	US20240374588, Example 59; BDBM704389; US20240374588, Example 59; 2-((1r,4r)-4-((4-(1-(2,6-Dioxopiperidin-3-yl)-3-methyl-2-oxo-2,3-dihydro-1H-benzo[d]imidazol-5-yl)piperidin-1-yl)methyl)cyclohexyl)-N-(imidazo[1,2-b]pyridazin-3-yl)-6-methoxy-2H-indazole-5-carboxamide	COC1=CC2=NN([C@H]3CC[C@H](CN4CCC(C5=CC6=C(C=C5)N(C5CCC(=O)NC5=O)C(=O)N6C)CC4)CC3)C=C2C=C1C(=O)NC1=CN=C2C=CC=NN12	C40H44N10O5	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-F1PEX3	SCHEMBL31134396	US20240374588, Example 60; BDBM704390; US20240374588, Example 60; N-(1-Cyclopropyl-2-oxo-1,2-dihydropyridin-3-yl)-2-((1r,4r)-4-((4-(1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxo-2,3-dihydro-1H-benzo[d]imidazol-5-yl)piperidin-1-yl)methyl)cyclohexyl)-6-methoxy-2H-indazole-5-carboxamide	COC1=CC2=NN([C@H]3CC[C@H](CN4CCC(C5=CC6=C(C=C5)N(C5CCC(=O)NC5=O)C(=O)N6C)CC4)CC3)C=C2C=C1C(=O)NC1=CC=CN(C2CC2)C1=O	C42H48N8O6	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-1KX7QR	WO2024209044A1_61	.	CNC(=O)C(CCC=O)N1C(=O)N(C)C2=C1C=CC(C1CCN(C[C@H]3CC[C@H](N4C=C5C=C(C(=O)NC6=CN=C7C=CC=NN67)C(OC6CC6)=CC5=N4)CC3)CC1)=C2	C43H50N10O5	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-LFRGDX	SCHEMBL31134667	US20240374588, Example 62; BDBM704392; US20240374588, Example 62; 2-((1r,4r)-4-((4-(1-(2,6-Dioxopiperidin-3-yl)-3-methyl-2-oxo-2,3-dihydro-1H-benzo[d]imidazol-4-yl)piperazin-1-yl)methyl)cyclohexyl)-N-(imidazo[1,2-b]pyridazin-3-yl)-6-methoxy-2H-indazole-5-carboxamide	COC1=CC2=NN([C@H]3CC[C@H](CN4CCN(C5=CC=CC6=C5N(C)C(=O)N6C5CCC(=O)NC5=O)CC4)CC3)C=C2C=C1C(=O)NC1=CN=C2C=CC=NN12	C39H43N11O5	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-PAD43R	SCHEMBL31134671	US20240374588, Example 63; BDBM704393; US20240374588, Example 63; 6-Cyclopropoxy-2-((1r,4r)-4-((4-(1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxo-2,3-dihydro-1H-benzo[d]imidazol-4-yl)piperazin-1-yl)methyl)cyclohexyl)-N-(imidazo[1,2-b]pyridazin-3-yl)-2H-indazole-5-carboxamide	CN1C(=O)N(C2CCC(=O)NC2=O)C2=C1C(N1CCN(C[C@H]3CC[C@H](N4C=C5C=C(C(=O)NC6=CN=C7C=CC=NN67)C(OC6CC6)=CC5=N4)CC3)CC1)=CC=C2	C41H45N11O5	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-GO3B6F	SCHEMBL31134425	US20240374588, Example 64; BDBM704394; US20240374588, Example 64; 2-((1r,4r)-4-((4-((1-(2,6-Dioxopiperidin-3-yl)-3-methyl-2-oxo-2,3-dihydro-1H-benzo[d]imidazol-4-yl)methyl)piperazin-1-yl)methyl)cyclohexyl)-N-(imidazo[1,2-b]pyridazin-3-yl)-6-methoxy-2H-indazole-5-carboxamide	COC1=CC2=NN([C@H]3CC[C@H](CN4CCN(CC5=CC=CC6=C5N(C)C(=O)N6C5CCC(=O)NC5=O)CC4)CC3)C=C2C=C1C(=O)NC1=CN=C2C=CC=NN12	C40H45N11O5	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-AZQXQ0	SCHEMBL31134449	US20240374588, Example 65; BDBM704395; US20240374588, Example 65; 2-((1r,4r)-4-((4-((1-(4-(2,4-Dioxotetrahydropyrimidin-1(2H)-yl)-3-methylphenyl)piperidin-4-yl)methyl)piperazin-1-yl)methyl)cyclohexyl)-N-(imidazo[1,2-b]pyridazin-3-yl)-6-methoxy-2H-indazole-5-carboxamide	COC1=CC2=NN([C@H]3CC[C@H](CN4CCN(CC5CCN(C6=CC(C)=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)CC3)C=C2C=C1C(=O)NC1=CN=C2C=CC=NN12	C43H53N11O4	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-TRMQEV	SCHEMBL31134242	N-(1-cyclopropyl-2-oxopyridin-3-yl)-2-[4-[[4-[[1-[4-(2,4-dioxo-1,3-diazinan-1-yl)-3-methylphenyl]piperidin-4-yl]methyl]piperazin-1-yl]methyl]cyclohexyl]-6-methoxyindazole-5-carboxamide	COC1=CC2=NN([C@H]3CC[C@H](CN4CCN(CC5CCN(C6=CC(C)=C(N7CCC(=O)NC7=O)C=C6)CC5)CC4)CC3)C=C2C=C1C(=O)NC1=CC=CN(C2CC2)C1=O	C45H57N9O5	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-E5UZOQ	WO2024209044A1_67	.	COC1=CC2=NN([C@H]3CC[C@H](CN4CCC(C5=CC6=C(C=C(N7CCC(=O)NC7=O)C=C6)N5C)CC4)CC3)C=C2C=C1C(=O)CC1=CC=CN(C2CC2)C1=O	C43H49N7O5	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-N8BD26	SCHEMBL31134344	US20240374588, Example 68; BDBM704398; US20240374588, Example 68; 6-Cyclopropoxy-2-((1r,4r)-4-((4-(4-(2,6-dioxopiperidin-3-yl)phenyl)piperazin-1-yl)methyl)cyclohexyl)-N-(imidazo[1,2-b]pyridazin-3-yl)-2H-indazole-5-carboxamide	O=C1CCC(C2=CC=C(N3CCN(C[C@H]4CC[C@H](N5C=C6C=C(C(=O)NC7=CN=C8C=CC=NN78)C(OC7CC7)=CC6=N5)CC4)CC3)C=C2)C(=O)N1	C39H43N9O4	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-43K6K4	SCHEMBL31134371	US20240374588, Example 69; BDBM704399; US20240374588, Example 69; N-(1-Cyclopropyl-2-oxo-1,2-dihydropyridin-3-yl)-2-((1r,4r)-4-((4-(4-(2,6-dioxopiperidin-3-yl)phenyl)piperazin-1-yl)methyl)cyclohexyl)-6-methoxy-2H-indazole-5-carboxamide	COC1=CC2=NN([C@H]3CC[C@H](CN4CCN(C5=CC=C(C6CCC(=O)NC6=O)C=C5)CC4)CC3)C=C2C=C1C(=O)NC1=CC=CN(C2CC2)C1=O	C39H45N7O5	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-91666R	SCHEMBL31134481	US20240374588, Example 7; BDBM704314; BDBM704316; US20240374588, Example 7; US20240374588, Example 8	COC1=CC2=NN(C3CCC(N(C)CCC4CCN(CC5=C6C(=CC=C5)N(C5CCC(=O)NC5=O)C(=O)N6C)CC4)CC3)C=C2C=C1C(=O)NC1=CN=C2C=CC=NN12	C43H51N11O5	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-PDJXK7	SCHEMBL31134341	US20240374588, Example 70; BDBM704400; US20240374588, Example 70; 2-((1r,4r)-4-((4-(4-(2,6-Dioxopiperidin-3-yl)-3-methylphenyl)piperazin-1-yl)methyl)cyclohexyl)-N-(imidazo[1,2-b]pyridazin-3-yl)-6-methoxy-2H-indazole-5-carboxamide	COC1=CC2=NN([C@H]3CC[C@H](CN4CCN(C5=CC(C)=C(C6CCC(=O)NC6=O)C=C5)CC4)CC3)C=C2C=C1C(=O)NC1=CN=C2C=CC=NN12	C38H43N9O4	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-7X796K	SCHEMBL31134331	US20240374588, Example 71; BDBM704401; US20240374588, Example 71; N-(1-Cyclopropyl-2-oxo-1,2-dihydropyridin-3-yl)-2-((1r,4r)-4-((4-(4-(2,6-dioxopiperidin-3-yl)-3-methylphenyl)piperazin-1-yl)methyl)cyclohexyl)-6-methoxy-2H-indazole-5-carboxamide	COC1=CC2=NN([C@H]3CC[C@H](CN4CCN(C5=CC(C)=C(C6CCC(=O)NC6=O)C=C5)CC4)CC3)C=C2C=C1C(=O)NC1=CC=CN(C2CC2)C1=O	C40H47N7O5	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-LTVSTE	SCHEMBL31134338	US20240374588, Example 72; SCHEMBL31134339; BDBM704402; US20240374588, Example 72	COC1=CC2=NN([C@H]3CC[C@H](CN4CCC(N5CCN(C6=CC=C(C7CCC(=O)NC7=O)C=C6)CC5)CC4)CC3)C=C2C=C1C(=O)NC1=CN=C2C=CC=NN12	C42H50N10O4	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-62Z4OX	SCHEMBL31134300	US20240374588, Example 73; BDBM704403; BDBM704404; US20240374588, Example 73; US20240374588, Example 74; 2-((1r,4r)-4-(2-(4-(4-(2,6-Dioxopiperidin-3-yl)phenyl)piperazin-1-yl)ethyl)cyclohexyl)-N-(imidazo[1,2-b]pyridazin-3-yl)-6-methoxy-2H-indazole-5-carboxamide	COC1=CC2=NN([C@H]3CC[C@H](CN4CCN(C5=CC(OC)=C(C6CCC(=O)NC6=O)C=C5)CC4)CC3)C=C2C=C1C(=O)NC1=CN=C2C=CC=NN12	C38H43N9O5	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-LXE4UH	SCHEMBL31134336	2-[4-[2-[4-[4-(2,6-dioxopiperidin-3-yl)phenyl]piperazin-1-yl]ethyl]cyclohexyl]-N-imidazo[1,2-b]pyridazin-3-yl-6-methoxyindazole-5-carboxamide	COC1=CC2=NN([C@H]3CC[C@H](CCN4CCN(C5=CC=C(C6CCC(=O)NC6=O)C=C5)CC4)CC3)C=C2C=C1C(=O)NC1=CN=C2C=CC=NN12	C38H43N9O4	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-QDNC1Y	SCHEMBL31134387	N-(1-cyclopropyl-2-oxopyridin-3-yl)-2-[4-[2-[4-[4-(2,6-dioxopiperidin-3-yl)phenyl]piperazin-1-yl]ethyl]cyclohexyl]-6-methoxyindazole-5-carboxamide	COC1=CC2=NN([C@H]3CC[C@H](CCN4CCN(C5=CC=C(C6CCC(=O)NC6=O)C=C5)CC4)CC3)C=C2C=C1C(=O)NC1=CC=CN(C2CC2)C1=O	C40H47N7O5	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-BH8BUB	SCHEMBL31134432	US20240374588, Example 76; BDBM704405; US20240374588, Example 76; 2-((1r,4r)-4-((4-(6-(2,6-Dioxopiperidin-3-yl)pyridin-3-yl)piperazin-1-yl)methyl)cyclohexyl)-N-(imidazo[1,2-b]pyridazin-3-yl)-6-methoxy-2H-indazole-5-carboxamide	COC1=CC2=NN([C@H]3CC[C@H](CN4CCN(C5=CN=C(C6CCC(=O)NC6=O)C=C5)CC4)CC3)C=C2C=C1C(=O)NC1=CN=C2C=CC=NN12	C36H40N10O4	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-MOOWXX	SCHEMBL31134252	US20240374588, Example 77; BDBM704406; US20240374588, Example 77; 2-((1r,4r)-4-((4-(2-(2,6-Dioxopiperidin-3-yl)-3-oxoisoindolin-5-yl)piperazin-1-yl)methyl)cyclohexyl)-N-(imidazo[1,2-b]pyridazin-3-yl)-6-methoxy-2H-indazole-5-carboxamide	COC1=CC2=NN([C@H]3CC[C@H](CN4CCN(C5=CC6=C(C=C5)CN(C5CCC(=O)NC5=O)C6=O)CC4)CC3)C=C2C=C1C(=O)NC1=CN=C2C=CC=NN12	C39H42N10O5	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-D85B3G	SCHEMBL31134508	US20240374588, Example 78; BDBM704407; US20240374588, Example 78; N-(1-Cyclopropyl-2-oxo-1,2-dihydropyridin-3-yl)-2-((1r,4r)-4-((4-(2-(2,6-dioxopiperidin-3-yl)-3-oxoisoindolin-5-yl)piperazin-1-yl)methyl)cyclohexyl)-6-methoxy-2H-indazole-5-carboxamide	COC1=CC2=NN([C@H]3CC[C@H](CN4CCN(C5=CC=C6CN(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)CC3)C=C2C=C1C(=O)NC1=CC=CN(C2CC2)C1=O	C41H46N8O6	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-F9BS64	SCHEMBL31134265	US20240374588, Example 79; BDBM704408; BDBM704409; US20240374588, Example 79; US20240374588, Example 80; 2-((1r,4r)-4-((4-(2-(2,6-Dioxopiperidin-3-yl)-7-methoxy-1-oxoisoindolin-5-yl)piperazin-1-yl)methyl)cyclohexyl)-N-(imidazo[1,2-b]pyridazin-3-yl)-6-methoxy-2H-indazole-5-carboxamide	COC1=CC2=NN([C@H]3CC[C@H](CN4CCN(CC5CCN(C6=CC7=C(C=C6)CN(C6CCC(=O)NC6=O)C7=O)CC5)CC4)CC3)C=C2C=C1C(=O)NC1=CN=C2C=CC=NN12	C45H53N11O5	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-197S4M	SCHEMBL31134380	2-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]cyclohexyl]-N-imidazo[1,2-b]pyridazin-3-yl-6-methoxyindazole-5-carboxamide	COC1=CC2=NN([C@H]3CC[C@H](CN4CCN(C5=CC6=C(C(=O)N(C7CCC(=O)NC7=O)C6)C(OC)=C5)CC4)CC3)C=C2C=C1C(=O)NC1=CN=C2C=CC=NN12	C40H44N10O6	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-F0UDJQ	SCHEMBL31134343	N-(1-cyclopropyl-2-oxopyridin-3-yl)-2-[4-[[4-[2-(2,6-dioxopiperidin-3-yl)-7-methoxy-1-oxo-3H-isoindol-5-yl]piperazin-1-yl]methyl]cyclohexyl]-6-methoxyindazole-5-carboxamide	COC1=CC2=NN([C@H]3CC[C@H](CN4CCN(C5=CC(OC)=C6C(=O)N(C7CCC(=O)NC7=O)CC6=C5)CC4)CC3)C=C2C=C1C(=O)NC1=CC=CN(C2CC2)C1=O	C42H48N8O7	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-SM4XFF	SCHEMBL31134365	2-[4-[[4-[3-(2,4-dioxo-1,3-diazinan-1-yl)-1-methylindazol-7-yl]piperidin-1-yl]methyl]cyclohexyl]-N-imidazo[1,2-b]pyridazin-3-yl-6-methoxyindazole-5-carboxamide	COC1=CC2=NN([C@H]3CC[C@H](CN4CCC(C5=C6C(=CC=C5)C(N5CCC(=O)NC5=O)=NN6C)CC4)CC3)C=C2C=C1C(=O)NC1=CN=C2C=CC=NN12	C39H43N11O4	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-XUECOA	SCHEMBL31134308	2-[4-[[4-[3-(2,4-dioxo-1,3-diazinan-1-yl)-1-methylindazol-7-yl]piperazin-1-yl]methyl]cyclohexyl]-N-imidazo[1,2-b]pyridazin-3-yl-6-methoxyindazole-5-carboxamide	COC1=CC2=NN([C@H]3CC[C@H](CN4CCN(C5=CC=CC6=C5N(C)N=C6N5CCC(=O)NC5=O)CC4)CC3)C=C2C=C1C(=O)NC1=CN=C2C=CC=NN12	C38H42N12O4	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-DB1YLG	SCHEMBL31134499	2-[4-[[2-[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]piperidin-1-yl]acetyl]-methylamino]cyclohexyl]-N-imidazo[1,2-b]pyridazin-3-yl-6-methoxyindazole-5-carboxamide	COC1=CC2=NN([C@H]3CC[C@H](N(C)C(=O)CN4CCC(N5C=CC6=C5C=CC=C6N5CCC(=O)NC5=O)CC4)CC3)C=C2C=C1C(=O)NC1=CN=C2C=CC=NN12	C41H45N11O5	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-AFYS09	SCHEMBL31134237	2-[4-[[4-[2-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]acetyl]piperazin-1-yl]methyl]cyclohexyl]-N-imidazo[1,2-b]pyridazin-3-yl-6-methoxyindazole-5-carboxamide	COC1=CC2=NN([C@H]3CC[C@H](CN4CCN(C(=O)CN5C=CC6=C5C=CC=C6N5CCC(=O)NC5=O)CC4)CC3)C=C2C=C1C(=O)NC1=CN=C2C=CC=NN12	C40H43N11O5	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-7Q9RYQ	SCHEMBL31134283	US20240374588, Example 86; BDBM704411; BDBM704412; US20240374588, Example 86; US20240374588, Example 89; 2-((1r,4r)-4-((4-(1-(2,6-Dioxopiperidin-3-yl)-3-methyl-1H-indazol-4-yl)piperazin-1-yl)methyl)cyclohexyl)-N-(imidazo[1,2-b]pyridazin-3-yl)-6-methoxy-2H-indazole-5-carboxamide	COC1=CC2=NN([C@H]3CC[C@H](CN4CCN(C5CCC(N6C=CC7=C6C=CC=C7N6CCC(=O)NC6=O)CC5)CC4)CC3)C=C2C=C1C(=O)NC1=CN=C2C=CC=NN12	C44H51N11O4	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-BI3DCI	SCHEMBL31134401	6-cyclopropyloxy-2-[1-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)indol-1-yl]cyclohexyl]methyl]piperidin-4-yl]-N-imidazo[1,2-b]pyridazin-3-ylindazole-5-carboxamide	O=C1CCN(C2=CC=CC3=C2C=CN3[C@H]2CC[C@H](CN3CCC(N4C=C5C=C(C(=O)NC6=CN=C7C=CC=NN67)C(OC6CC6)=CC5=N4)CC3)CC2)C(=O)N1	C41H44N10O4	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-OJHZ6D	SCHEMBL31134479	2-[4-[[4-[1-(2,6-dioxopiperidin-3-yl)-3-methylindazol-4-yl]piperazin-1-yl]methyl]cyclohexyl]-N-imidazo[1,2-b]pyridazin-3-yl-6-methoxyindazole-5-carboxamide	COC1=CC2=NN([C@H]3CC[C@H](CN4CCN(C5=CC=CC6=C5C(C)=NN6C5CCC(=O)NC5=O)CC4)CC3)C=C2C=C1C(=O)NC1=CN=C2C=CC=NN12	C39H43N11O4	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-DERDGR	SCHEMBL31134472	US20240374588, Example 90; BDBM704413; US20240374588, Example 90; 6-Cyclopropoxy-2-((1r,4r)-4-((4-(1-(2,6-dioxopiperidin-3-yl)-3-methyl-1H-indazol-4-yl)piperazin-1-yl)methyl)cyclohexyl)-N-(imidazo[1,2-b]pyridazin-3-yl)-2H-indazole-5-carboxamide	CC1=NN(C2CCC(=O)NC2=O)C2=C1C(N1CCN(C[C@H]3CC[C@H](N4C=C5C=C(C(=O)NC6=CN=C7C=CC=NN67)C(OC6CC6)=CC5=N4)CC3)CC1)=CC=C2	C41H45N11O4	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-HBEABJ	SCHEMBL31134390	US20240374588, Example 91; BDBM704414; US20240374588, Example 91	COC1=CC2=NN([C@H]3CC[C@H](CN4CCN(C5=CC6=C(C=C5)N(C5CCC(=O)NC5=O)N=C6C)CC4)CC3)C=C2C=C1C(=O)NC1=CN=C2C=CC=NN12	C39H43N11O4	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-DWTDKE	SCHEMBL31134550	US20240374588, Example 92; BDBM704415; BDBM704416; US20240374588, Example 92; US20240374588, Example 93; 2-((1r,4r)-4-((4-(4-(2,4-Dioxotetrahydropyrimidin-1(2H)-yl)isoquinolin-8-yl)piperazin-1-yl)methyl)cyclohexyl)-N-(imidazo[1,2-b]pyridazin-3-yl)-6-methoxy-2H-indazole-5-carboxamide	COC1=CC2=NN([C@H]3CC[C@H](CN4C=C(C5=CC=CC6=C5C(C)=NN6C5CCC(=O)NC5=O)C=N4)CC3)C=C2C=C1C(=O)NC1=CN=C2C=CC=NN12	C38H37N11O4	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-9QUZH0	SCHEMBL31134440	2-[4-[[4-[4-(2,4-dioxo-1,3-diazinan-1-yl)isoquinolin-8-yl]piperazin-1-yl]methyl]cyclohexyl]-N-imidazo[1,2-b]pyridazin-3-yl-6-methoxyindazole-5-carboxamide	COC1=CC2=NN([C@H]3CC[C@H](CN4CCN(C5=C6C=NC=C(N7CCC(=O)NC7=O)C6=CC=C5)CC4)CC3)C=C2C=C1C(=O)NC1=CN=C2C=CC=NN12	C39H41N11O4	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-5WYG0C	SCHEMBL31134533	US20240374588, Example 94; BDBM704417; US20240374588, Example 94	COC1=CC2=NN([C@H]3CC[C@H](CN4CCN(C5=C6OC(=O)N(C7CCC(=O)NC7=O)C6=CC=C5)CC4)CC3)C=C2C=C1C(=O)NC1=CN=C2C=CC=NN12	C38H40N10O6	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-FSKUE9	SCHEMBL31134419	US20240374588, Example 95; BDBM704418; US20240374588, Example 95	COC1=CC2=NN([C@H]3CC[C@H](CN4CCN(C5=CC=C6C(=C5)C5(CC5)C(=O)N6C5CCC(=O)NC5=O)CC4)CC3)C=C2C=C1C(=O)NC1=CN=C2C=CC=NN12	C41H44N10O5	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-49UOM6	SCHEMBL31134487	US20240374588, Example 96; BDBM704419; US20240374588, Example 96	COC1=CC2=NN([C@H]3CC[C@H](CN4CCC(C5=CN(C)C6=C5C=CC=C6N5CCC(=O)NC5=O)CC4)CC3)C=C2C=C1C(=O)NC1=CN=C2C=CC=NN12	C40H44N10O4	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-1GIYD4	SCHEMBL31134326	2-[4-[[4-[3-(2,4-dioxo-1,3-diazinan-1-yl)imidazo[1,5-a]pyridin-8-yl]piperazin-1-yl]methyl]cyclohexyl]-N-imidazo[1,2-b]pyridazin-3-yl-6-methoxyindazole-5-carboxamide	COC1=CC2=NN([C@H]3CC[C@H](CN4CCN(C5=CC=CN6C5=CN=C6N5CCC(=O)NC5=O)CC4)CC3)C=C2C=C1C(=O)NC1=CN=C2C=CC=NN12	C37H40N12O4	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-R6CBAE	SCHEMBL31134497	N-(1-cyclopropyl-2-oxopyridin-3-yl)-2-[4-[[4-[3-(2,4-dioxo-1,3-diazinan-1-yl)-1,2-benzoxazol-6-yl]piperazin-1-yl]methyl]cyclohexyl]-6-methoxyindazole-5-carboxamide	COC1=CC2=NN([C@H]3CC[C@H](CN4CCN(C5=CC=C6C(=C5)ON=C6N5CCC(=O)NC5=O)CC4)CC3)C=C2C=C1C(=O)NC1=CC=CN(C2CC2)C1=O	C39H43N9O6	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-MQMZJ4	WO2024209044A1_99	.	COC1=CC2=NN([C@H]3CC[C@@H](CN4CCC(N5C=CC6=C5C=CC=C6N5CCC(=O)NC5=O)CC4)CC3)C=C2C=C1C(=O)NC1=CN=C2C=CC=NN12	C39H42N10O4	IRAK4	Q9NWZ3	CRBN	WO-2024209044-A1
TPD-T4OSEA	WO2024263586A1_1	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-1,2-dihydropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl N-[3-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]propyl]carbamate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)NCCCC4=CC=C6C(=C4)N(C)C(=O)N6C4CCC(=O)NC4=O)CC5)NC(N4CC5CCC(C4)N5)=C3C=N1)=CC(O)=C2	C51H54F2N10O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-R0U2PV	WO2024263586A1_102	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=CC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(COC6CN(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)C6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C58H62F2N10O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-EZUKJ6	WO2024263586A1_103	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CC6CCC(C4)C6CN4CCC(C6=CC=C7C(=C6)N(C)C(=O)N7C6CCC(=O)NC6=O)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C61H67F2N11O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-DB4AX1	WO2024263586A1_104	.	[H]=C(OC[C@@H]1CC[C@]2(COC3=NC(N4CC5CCC(C4)N5)=C4C=NC(C5=CC=CC6=C5C(C#C)=C(F)C=C6)=C(F)C4=N3)CCCN12)N1CC(COC2CCN(C3=CC=C4C(=C3)N(C)C(=O)N4C3CCC(=O)NC3=O)CC2)C1	C57H63F2N11O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-21NGJK	SCHEMBL26634914	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 4-[2-[3-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]prop-2-ynoxy]ethyl]piperidine-1-carboxylate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CCOCC#CC6=CC=C7C(=C6)N(C)C(=O)N7C6CCC(=O)NC6=O)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C58H60F2N10O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-0SBR40	WO2024263586A1_106	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCN(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C58H66F2N12O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-8DW8PG	WO2024263586A1_107	.	C#CC1=C(F)C=CC2=C1C(C1=CC3=NC(OC[C@@]45CCCN4[C@H](COCN4CCC(OCCC#CC6=C7C(=CC=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C57H61FN10O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-L4AAU5	WO2024263586A1_108	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN(C)C6CCN(C7=C8C(=CC=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C60H68F2N12O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-I7A8MD	WO2024263586A1_109	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CC=CN4[C@H](COC(=O)NCCCN(C)C4CCN(C6=C7C(=CC=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C57H62F2N12O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-WKZR6S	WO2024263586A1_110	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CC=CN4[C@H](COC(=O)NCCCC(=O)N4CCN(C6=C7C(=CC=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C56H58F2N12O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-I3J2AE	WO2024263586A1_111	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCO[C@@H](CN6CCN(C7=C8C(=CC=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)CC6)C4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C57H62F2N12O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-0YB1BG	WO2024263586A1_112	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCN(C7=C8C(=CC=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C58H64F2N12O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-BXXYVS	SCHEMBL26635155	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 3-[[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-4-yl]piperazin-1-yl]methyl]azetidine-1-carboxylate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CC(CN6CCN(C7=C8C(=CC=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)CC6)C4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C56H60F2N12O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-48CPQC	WO2024263586A1_114	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCCCC#CC6=CC=C7C(=C6)N(C)C(=O)N7C6CCC(=O)NC6=O)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C58H62F2N10O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-WTX7V4	SCHEMBL26634980	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 4-[3-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]prop-2-ynoxy]piperidine-1-carboxylate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCC#CC6=CC=C7C(=C6)N(C)C(=O)N7C6CCC(=O)NC6=O)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C56H56F2N10O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-SP5SFF	WO2024263586A1_116	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4C(COC(=O)N4CCC(OCC6=CC=C7C(=C6)N(C)C(=O)N7C6CCC(=O)NC6=O)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C54H56F2N10O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-V7ZTCT	WO2024263586A1_117	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCCCCC6=C7C(=CC=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C57H64F2N10O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-Q5E1Z1	WO2024263586A1_118	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCCCCC6=CC=C7C(=C6)NC(=O)N7C6CCC(=O)NC6=O)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C56H60F2N10O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-WHKPGO	WO2024263586A1_119	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CC=CN4[C@H](COC(=O)N4CCC(OCCCC#CC6=C7C(=CC=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C58H58F2N10O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-T06B1W	SCHEMBL26634919	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 4-[5-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]pentoxy]piperidine-1-carboxylate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCCCCCC6=CC=C7C(=C6)N(C)C(=O)N7C6CCC(=O)NC6=O)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C58H64F2N10O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-0YW7AQ	SCHEMBL26634952	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 7-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-4-yl]-2,7-diazaspiro[3.5]nonane-2-carboxylate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CC6(CCN(C7=C8C(=CC=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)CC6)C4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C55H57F2N11O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-NJUXU9	WO2024263586A1_122	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCCCCCC6=C7C(=CC=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C58H64F2N10O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-1USUS6	SCHEMBL26634878	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl N-[2-[2-[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-4-yl]piperazin-1-yl]ethoxy]ethyl]carbamate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)NCCOCCN4CCN(C6=C7C(=CC=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C56H62F2N12O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-AJN3PJ	SCHEMBL26634941	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 2-[2-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-4-yl]ethyl]-7-azaspiro[3.5]nonane-7-carboxylate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC6(CC4)CC(CCC4=C7C(=CC=C4)N(C4CCC(=O)NC4=O)C(=O)N7C)C6)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C58H62F2N10O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-PIN0VM	WO2024263586A1_125	.	[H]C1=C(C2=CC=CC3=C2C(C#C)=C(F)C=C3)N=CC2=C(N3CC4CCC(C3)N4)N=C(OC[C@@]34CCCN3[C@H](COC(=O)NC[C@@H]3CN(CC#CC5=C6C(=CC=C5)N(C5CCC(=O)NC5=O)C(=O)N6C)CCO3)CC4)N=C12	C56H58FN11O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-5XSEZG	SCHEMBL26635054	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 4-[1-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-4-yl]piperidin-4-yl]piperidine-1-carboxylate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(C6CCN(C7=C8C(=CC=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C58H63F2N11O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-C5WYLU	WO2024263586A1_128	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(COC6CCN(CC7=C8C(=CC=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C60H67F2N11O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-R7K6YP	WO2024263586A1_129	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CC=CN4[C@H](COC(=O)N4CCC6(CC4)CCN(C4=C7C(=CC=C4)N(C4CCC(=O)NC4=O)C(=O)N7C)CC6)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C57H59F2N11O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-NXCJ8Y	WO2024263586A1_131	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(N6CCN(C7=C8C(=CC=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C57H62F2N12O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-W54PLW	WO2024263586A1_132	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CC6CCN(CC7=C8C(=CC=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C60H67F2N11O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-92N4H7	WO2024263586A1_136	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCCCC6=CC=C7C(=C6)N(C)C(=O)N7C6CCC(=O)NC6=O)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C56H60F2N10O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-MI118K	WO2024263586A1_138	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)NCCCCCCCCC4=CC=C6C(=C4)N(C)C(=O)N6C4CCC(=O)NC4=O)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC(O)=C2	C56H62F2N10O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-96FY3D	WO2024263586A1_14	.	C#CC1=C(F)C=CC2=C1C(C1=CC3=NC(OCC45CCCN4[C@H](COC(=O)NCCCCCCCCCCC4=C6C(=CC=C4)N(C4CCC(=O)NC4=O)C(=O)N6C)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C58H67FN10O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-72YMN1	WO2024263586A1_140	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)NCCCCCCCCC4=C6C(=CC=C4)N(C4CCC(=O)NC4=O)C(=O)N6C)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC(O)=C2	C56H62F2N10O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-6C8B54	WO2024263586A1_141	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=CC(OC[C@@]45CCCN4[C@H](COC(=O)NCCCCCCCC4=C6C(=CC=C4)N(C4CCC(=O)NC4=O)C(=O)N6C)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC(O)=C2	C56H61F2N9O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-S34724	WO2024263586A1_144	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CC=CN4[C@H](COC(=O)N4CCC(OCCCC6=C7C(=CC=C6)N(C6CCC(=O)N(C)C6=O)C(=O)N7C)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C57H60F2N10O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-6V1SL0	SCHEMBL26634934	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 4-[[[1-[[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-4-yl]methyl]piperidin-4-yl]amino]methyl]piperidine-1-carboxylate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CNC6CCN(CC7=C8C(=CC=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C60H68F2N12O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-GJWITB	WO2024263586A1_147	.	C#CC1=C(F)C=CC2=C1C(C1N=CC3=C(N4CC5CCC(C4)N5)N=C(OC[C@@]45CCCN4[C@H](COC(=O)NCCCCC(=O)N4CCN(C6=CC=C(N7CCC(=O)NC7=O)C=C6)CC4)CC5)N=C3C1F)=CC=C2	C54H61F2N11O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-BWV7AH	WO2024263586A1_148	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)NCCCCCC(=O)N4CCN(C6=CC=C(N7CCC(=O)NC7=O)C=C6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3CN1)=CC=C2	C55H63F2N11O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-4I8Y0C	WO2024263586A1_149	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)NCCCCCCC(=O)N4CCN(C6=CC=C(N7CCC(=O)NC7=O)C=C6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C56H63F2N11O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-UTXV00	WO2024263586A1_15	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)NCCCCCCCCCCNC4=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C4)CC5)=NC(C4CC5CCC(C4)N5)=C3C=N1)=CC(O)=C2	C59H65F2N9O8	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-LUIN5B	SCHEMBL31003864	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl N-[9-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]nonyl]carbamate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)NCCCCCCCCCNC4=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC(O)=C2	C57H62F2N10O8	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-WF4WWB	SCHEMBL26635002	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl N-[6-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-5-yl]amino]hexyl]carbamate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)NCCCCCCNC4=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC(O)=C2	C54H56F2N10O8	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-ZP2TMF	WO2024263586A1_2	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=CC(OC[C@@]45CCCN4[C@H](COC(=O)NCCC4=CC=C6C(=C4)N(C)C(=O)N6C4CCC(=O)NC4=O)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC(O)=C2	C51H51F2N9O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-1M4NP7	WO2024263586A1_201	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=CC(CCCOC3CCN(C(=O)OC[C@@H]4CC[C@]5(COC6=NC(N7CC8CCC(C7)N8)=C7C=NC(C8=CC=CC=C8F)=C(F)C7=N6)CCCN45)CC3)=C21	C50H58F2N10O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-TFYQU4	WO2024263586A1_202	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CC(C7=C8C(=CC=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)C6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C57H61F2N11O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-VNNYXG	WO2024263586A1_203	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CC(CN6CCC(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)C4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C57H61F2N11O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-FGFRQH	WO2024263586A1_204	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CC(CN6CCC(C7=C8C(=CC=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)CC6)C4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C57H61F2N11O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-C96WNM	WO2024263586A1_205	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CC(OCCCC#CC6=CC=C7C(=C6)N(C)C(=O)N7C6CCC(=O)NC6=O)C4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C56H56F2N10O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-INTY3G	WO2024263586A1_206	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(C6(N7CCC(C8=CC=C9C(=C8)N(C)C(=O)N9C8CCC(=O)NC8=O)CC7)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C61H67F2N11O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-3VLMKP	WO2024263586A1_207	.	[H]C1=C(C2=CC=CC3=C2C(C#C)=C(F)C=C3)N=CC2=C(N3CC4CCC(C3)N4)N=C(OC[C@@]34CCCN3[C@H](COC(=O)N3CC(CN5CCC(OC6=CC=C7C(=C6)N(C)C(=O)N7C6CCC(=O)NC6=O)CC5)C3)CC4)N=C12	C57H62FN11O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-TQZKFD	WO2024263586A1_208	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CCCC5(CCO5)C4)=C3C=N1)=CC(O)=C2	C60H70F2N10O8	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-2ZGTZT	WO2024263586A1_209	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=C8C(=CC=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)CC6)CC4)CC5)=NC(N4CCCC5(CCO5)C4)=C3C=N1)=CC(O)=C2	C60H70F2N10O8	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-MIZ4UB	WO2024263586A1_21	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]4(CC[C@H](C)COC(=O)NCCCCCCNC5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)CCCN4)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC(O)=C2	C55H60F2N10O8	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-GAH12B	WO2024263586A1_210	.	[H]=C(OC[C@H]1CC[C@@]2(COC3=NC(N4CC5CCC(C4)N5)=C4C=NC(C5=CC=CC6=C5C(C#C)=C(F)C=C6)=C(F)C4=N3)CCCN12)N1CCC(CN2CCC(C3=C4C(=CC=C3)N(C3CCC(=O)NC3=O)C(=O)N4C)CC2)CC1	C59H67F2N11O5	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-MNQ8VX	WO2024263586A1_211	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(COCCC#CC6=CC=C7C(=C6)N(C)C(=O)N7C6CCC(=O)NC6=O)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C58H60F2N10O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-WYPVV8	WO2024263586A1_212	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CC6CC(C4)C6CN4CCC(C6=CC=C7C(=C6)N(C)C(=O)N7C6CCC(=O)NC6=O)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C60H65F2N11O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-IHEFU9	WO2024263586A1_213	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CC6CC4CC6CN4CCC(C6=CC=C7C(=C6)N(C)C(=O)N7C6CCC(=O)NC6=O)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C60H65F2N11O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-XCDQNR	WO2024263586A1_214	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CC7(CC(C8=C9C(=CC=C8)N(C8CCC(=O)NC8=O)C(=O)N9C)C7)C6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C60H65F2N11O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-GTLC8D	WO2024263586A1_215	.	C#CC1=C(CF)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CC7(CC(C8=CC=C9C(=C8)N(C)C(=O)N9C8CCC(=O)NC8=O)C7)C6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C61H67F2N11O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-X45BOH	WO2024263586A1_216	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CC(OC7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)C6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C57H61F2N11O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-C674BN	WO2024263586A1_217	.	C#CC1=CC=CC2=C1C(C1=C(F)C3=CC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C60H67FN10O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-TOYJFN	WO2024263586A1_218	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(C3CCN(CC4CCN(C(=O)OC[C@@H]5CC[C@]6(COC7=NC(N8CC9CC(C8)N9)=C8C=NC(C9=CC=CC%10=C9C=C(F)C=C%10)=C(F)C8=N7)CCCN56)CC4)CC3)C=C21	C56H63F2N11O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-U7SHSN	WO2024263586A1_219	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N[C@H]4CC[C@@H](OC6CCN(CC7=C8C(=CC=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C60H67F2N11O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-OZMHE9	WO2024263586A1_22	[(3R,8R)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl N-[6-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]hexyl]carbamate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@]45CCCN4[C@@H](COC(=O)NCCCCCCNC4=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC(O)=C2	C54H56F2N10O8	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-U4FGJE	WO2024263586A1_220	.	[H]C1=C(C2=CC=CC3=C2C(C#C)=C(F)C=C3)N=CC2=C(N3CC4CCC(C3)N4)N=C(OC[C@@]34CCCN3[C@H](COC(O)N[C@H]3CC[C@H](OC5CCN(CC6=C7C(=CC=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC5)CC3)CC4)N=C12	C60H70FN11O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-6I5CYG	WO2024263586A1_221	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=C8C(=CC=C7)N(C7CCC(=O)NC7=O)C(=C)N8C)C6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C59H65F2N11O5	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-SRNCN1	WO2024263586A1_222	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCCC#CC#CC6=CC=C7C(=C6)N(C)C(=O)N7C6CCC(=O)NC6=O)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C59H58F2N10O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-M1E34D	WO2024263586A1_223	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)C6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C58H63F2N11O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-KW3BNN	WO2024263586A1_224	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CC(CN6CCC(CC7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)C4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C58H63F2N11O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-85GP12	WO2024263586A1_225	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CC(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)C6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C57H61F2N11O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-8AJSOO	WO2024263586A1_226	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(CC7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C60H67F2N11O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-ZB7VXY	WO2024263586A1_227	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=CC(CCCOC3CCN(C(=O)OC[C@@H]4CC[C@]5(COC6=NC(N7CC8CCC(C7)N8)=C7C=NC(C8=CC=CC=C8C(F)(F)F)=C(F)C7=N6)CC=CN45)CC3)=C21	C51H56F4N10O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-T7YPRI	WO2024263586A1_228	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(CCCOC3CCN(C(=O)OC[C@@H]4CC[C@]5(COC6=NC(N7CC8CCC(C7)N8)=C7C=NC(C8=CC=CC=C8F)=C(F)C7=N6)CCCN45)CC3)C=C21	C50H58F2N10O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-U0WU4I	WO2024263586A1_229	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=C8C(=CC=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC(O)=C2	C59H65F2N11O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-QMWIG3	WO2024263586A1_230	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(NC6CCC(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C59H65F2N11O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-QGUS9Z	WO2024263586A1_231	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(CCCOC3CCN(C(=O)OC[C@@H]4CC[C@]5(COC6=NC(N7CC8CCC(C7)N8)=C7C=NC(C8=CC(O)=CC=C8OC(F)(F)F)=C(F)C7=N6)CCCN45)CC3)C=C21	C51H58F4N10O9	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-LB00XG	WO2024263586A1_232	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=CC(CCCOC3CCN(C(=O)OC[C@@H]4CC[C@]5(COC6=NC(N7CC8CCC(C7)N8)=C7C=NC(C8=CC(O)=CC=C8OC(F)(F)F)=C(F)C7=N6)CCCN45)CC3)=C21	C51H58F4N10O9	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-MVLGST	WO2024263586A1_233	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(CCCOC3CCN(C(=O)OC[C@@H]4CC[C@]5(COC6=NC(N7CC8CCC(C7)N8)=C7C=NC(C8=CC=CC(Cl)=C8C(F)(F)F)=C(F)C7=N6)CC=CN45)CC3)C=C21	C51H55ClF4N10O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-KPP14K	WO2024263586A1_234	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(CCCOC3CCN(C(=O)OC[C@@H]4CC[C@]5(COC6=CC(N7CC8CCC(C7)N8)=C7C=NC(C8=CC=CC=C8OC(F)(F)F)=C(F)C7=N6)CCCN45)CC3)C=C21	C52H59F4N9O8	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-TKDDI0	WO2024263586A1_235	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=CC(CCCOC3CCN(C(=O)OC[C@@H]4CC[C@]5(COC6=NC(N7CC8CCC(C7)N8)=C7C=NC(C8=CC=CC=C8OC(F)(F)F)=C(F)C7=N6)CC=CN45)CC3)=C21	C51H56F4N10O8	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-XBVKSL	WO2024263586A1_236	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4C(COC(=O)N4CCC(CN6CCC(CC7=C8C(=CC=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C60H67F2N11O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-X5J6VD	WO2024263586A1_237	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CC(CC7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)N=NC7=O)C6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C58H62F2N12O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-RTIX8Y	WO2024263586A1_238	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCCC#CC#CC6=C7C(=CC=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C59H58F2N10O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-H24WWY	WO2024263586A1_239	.	[H]C1=C(C2=CC(O)=CC=C2F)N=CC2=C(N3CC4CCC(C3)N4)N=C(OC[C@@]34CCCN3[C@H](COC(=O)N3CCC(OCCCC5=CC=C6C(=C5)N(C)C(=O)N6C5CCC(=O)NC5=O)CC3)CC4)N=C12	C50H59FN10O8	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-6S5VUV	WO2024263586A1_24	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)NCCCCCCNC4=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C4)CC5)=CC(N4CC5CCC(C4)N5)=C3C=N1)=CC(O)=C2	C55H57F2N9O8	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-W7VSU4	WO2024263586A1_240	.	CC1=C(C2=CC(O)=CC=C2F)N=CC2=C(N3CC4CCC(C3)N4)N=C(OC[C@@]34CCCN3[C@H](COC(=O)N3CCC(OCCCC5=C6C(=CC=C5)N(C5CCC(=O)NC5=O)C(=O)N6C)CC3)CC4)N=C12	C51H61FN10O8	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-YVMLES	WO2024263586A1_241	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=CC=C8C(=C7)N(C)N=C8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C59H65F2N11O5	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-TEVT3W	WO2024263586A1_242	.	C#CC1C2=C(C=CC=C2C2=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=C8C(=CC=C7)C(C7CCC(=O)NC7=O)=NN8C)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N2)C=CC1F	C59H67F2N11O5	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-V1ORQ9	WO2024263586A1_243	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CC=CN4[C@H](COC(=O)N4CCC(OCCOCCOCCCC6C=CC=C7C(C8CCC(=O)NC8=O)=NN(C)C76)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C60H68F2N10O8	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-71ALGQ	WO2024263586A1_244	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCCCC6=C7C(=CC=C6)C(C6CCC(=O)NC6=O)=NN7C)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C56H60F2N10O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-CTE121	WO2024263586A1_245	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCCOCCOCCCC6=CC=C7C(=C6)N(C)N=C7C6CCC(=O)NC6=O)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C60H68F2N10O8	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-3EDML8	WO2024263586A1_246	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCCOCCC6=CC=C(C7CCC(=O)NC7=O)C=C6)CC4)CC5)=CC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C56H61F2N7O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-2I0LMY	WO2024263586A1_247	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CC=CN4[C@H](COC(=O)N4CCC(OCCOCCOCCOCCC6=CC=C(C7CCC(=O)NC7=O)C=C6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C59H66F2N8O9	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-D82G63	WO2024263586A1_248	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CC(CN6CCC(CC7=C8C(=CC=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)CC6)C4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C58H63F2N11O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-L48OVI	WO2024263586A1_249	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CC(CC7=C8C(=CC=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)C6)CC4)CC5)=NC(C4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C59H64F2N10O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-JPU45T	WO2024263586A1_250	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CC(C#CC7=C8C(=CC=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)C6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C59H61F2N11O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-DIUVTA	WO2024263586A1_251	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=CC=C8C(=C7F)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C59H64F3N11O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-6AFRTR	WO2024263586A1_252	.	CC1=C2C(=CC3=C(N4CC5CCC(C4)N5)N=C(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=C8C(=CC=C7)C(N7CCC(=O)NC7=O)=NN8C)CC6)CC4)CC5)N=C13)CC1=C(F)C=CC3=C1C2=CC=C3	C59H68FN11O5	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-LMQDQK	WO2024263586A1_253	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCCOCCOCCCC6=C7C(=CC=C6)C(N6CCC(=O)NC6=O)=NN7C)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C59H67F2N11O8	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-B8HROO	WO2024263586A1_254	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCCCC6=C7C(=CC=C6)C(N6CCC(=O)NC6=O)=NN7C)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C55H59F2N11O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-MIVEQ2	WO2024263586A1_255	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCCCC6=CC=C7C(=C6)N(C)NC7C6CCC(=O)NC6=O)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C56H62F2N10O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-AFKVMN	WO2024263586A1_256	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CC(C#CC7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)C6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C59H61F2N11O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-QO2RJ0	WO2024263586A1_257	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(C(=O)N6CCC(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C59H63F2N11O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-OKJS02	WO2024263586A1_258	.	COC1=C(C2CC2)C(C2=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCCCC6=CC=C7C(=C6)N(C)C(=O)N7C6CCC(=O)NC6=O)CC4)CC5)=NC(C4CC5CCC(C4)N5)=C3C=N2)=CC=C1	C55H66FN9O8	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-YIHJIN	WO2024263586A1_259	.	[H][C@]1(CN2CCC(C3=C4C(=CC=C3)N(C3CCC(=O)NC3=O)C(=O)N4C)CC2)[C@]2([H])CN(C(=O)OC[C@@H]3CC[C@]4(COC5=NC(N6CC7CCC(C6)N7)=C6C=NC(C7=CC=CC8=C7C(C#C)=C(F)C=C8)=C(F)C6=N5)CCCN34)C[C@]12[H]	C59H63F2N11O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-W6L5BA	WO2024263586A1_260	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4C(COC(=O)C4CC6C(C4)C6CN4CCC(C6=C7C(=CC=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C60H64F2N10O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-719T0Q	WO2024263586A1_261	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(CCCOC3CCN(C(=O)OC[C@@H]4CC[C@]5(COC6=NC(N7CC8CCC(C7)N8)=C7C=NC(C8=CC(O)=CC(Cl)=C8C8CC8)=C(F)C7=N6)CCCN45)CC3)C=C21	C53H62ClFN10O8	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-271FGN	WO2024263586A1_262	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=CC(CCCOC3CCN(C(=O)OC[C@@H]4CC[C@]5(COC6=NC(N7CC8CCC(C7)N8)=C7C=NC(C8=CC(O)=CC(Cl)=C8C8CC8)=C(F)C7=N6)CCCN45)CC3)=C21	C53H62ClFN10O8	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-YD2SQC	WO2024263586A1_263	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=CC=C8C(=C7)N(C)N=C8N7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CC5CC[C@H](C4)N5)=C3C=N1)=CC=C2	C58H64F2N12O5	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-BRSOK8	WO2024263586A1_264	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCCCC6=CC=C7C(=C6)N(C)N=C7N6CCC(=O)NC6=O)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C55H59F2N11O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-OTGIH0	WO2024263586A1_265	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CC=CN4C(COC(=O)N4CCC(OCC#CCC#CC6=CC=C7C(=C6)N(C)C(=O)N7C6CCC(=O)NC6=O)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C59H56F2N10O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-EODQYN	WO2024263586A1_266	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCC#CCC#CC6=C7C(=CC=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C59H58F2N10O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-EHWVAM	WO2024263586A1_267	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=C(F)C=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C59H64F3N11O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-K29VP9	WO2024263586A1_268	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CC6CC7(C6)CN(C6=CC=C8C(=C6)N(C)C(=O)N8C6CCC(=O)NC6=O)C7)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C60H65F2N11O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-IVBIY0	WO2024263586A1_269	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(O[C@H]6CC[C@@H](C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C59H64F2N10O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-4Q62XR	WO2024263586A1_27	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@]45CCCN4[C@@H](COC(=O)NCCOCCOCCOCCNC4=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC(O)=C2	C56H60F2N10O11	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-9L0QTS	WO2024263586A1_270	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=CC(CCCOC3CCN(C(=O)OC[C@@H]4CC[C@]5(COC6=NC(N7CC8CCC(C7)N8)=C7C=NC(C8=CC=CC(Cl)=C8C8CC8)=C(F)C7=N6)CCCN45)CC3)=C21	C53H62ClFN10O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-IDGXXS	WO2024263586A1_271	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCCOCCOCCCC6=CC=C7C(=C6)N(C)N=C7N6CCC(=O)NC6=O)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C59H67F2N11O8	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-URQBWM	WO2024263586A1_272	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(O[C@H]6CC[C@H](C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C59H64F2N10O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-83HF23	WO2024263586A1_273	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CC=CN4[C@H](COC(=O)N4CCC(OCCOCCOC6=CC=C(NC7CCC(=O)NC7=O)C=C6)CC4)CC5)NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C55H61F2N9O8	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-RDO10K	WO2024263586A1_274	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)C(F)(F)C6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C59H63F4N11O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-4XRS5S	WO2024263586A1_275	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N[C@H]4CC[C@H](OC6CCN(CC7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C60H67F2N11O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-ZAG976	WO2024263586A1_276	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=CC(OC[C@@]45CCCN4[C@H](COC(=O)N[C@H]4CC[C@@H](OC6CCN(CC7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C61H68F2N10O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-NNUDVU	WO2024263586A1_277	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OC6CCN(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CCCC5(CCO5)C4)=C3C=N1)=CC(O)=C2	C59H68F2N10O9	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-9XK14G	WO2024263586A1_278	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(CCCOC3CCN(C(=O)OC[C@@H]4CC[C@]5(COC6=NC(N7CC8CCC(C7)N8)=C7C=NC(C8=CC(O)=CC(Cl)=C8C(F)(F)F)=C(F)C7=N6)CCCN45)CC3)C=C21	C51H57ClF4N10O8	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-F501TQ	WO2024263586A1_279	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CC=CN4[C@H](COC(=O)N4CCC(OCCOCCOC6=CC=CC(NC7CCC(=O)NC7=O)=C6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C55H59F2N9O8	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-EBQ53F	SCHEMBL26830273	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl N-[2-[2-[2-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]ethoxy]ethoxy]ethoxy]ethyl]carbamate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)NCCOCCOCCOCCNC4=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC(O)=C2	C56H60F2N10O11	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-TFI9ON	WO2024263586A1_280	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCCOCCC6=CC=CC(N7CCC(=O)NC7=O)=C6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C54H59F2N9O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-D3Z0XV	WO2024263586A1_281	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=CC=C8C(=C7)N(C)N=C8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CCCC5(CCO5)C4)=C3C=N1)=CC(O)=C2	C60H70F2N10O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-TO2POB	WO2024263586A1_282	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OC6CCN(C7=CC=C8C(=C7)N(C)N=C8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C58H63F2N11O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-XHFFI6	WO2024263586A1_283	.	C#CC1=C(F)C=CC2=C1C(C1=C(C)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CCC6CC7(C6)CN(C6=CC=C8C(=C6)N(C)C(=O)N8C6CCC(=O)NC6=O)C7)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C62H70FN11O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-87OW2N	WO2024263586A1_284	.	[H]C1=C(C2=CC(O)=CC(O)=C2C(F)(F)F)N=CC2=C(N3CC4CCC(C3)N4)N=C(OC[C@@]34CCCN3[C@H](COC(=O)N3CCC(OCCCC5=C6C(=CC=C5)N(C5CCC(=O)NC5=O)C(=O)N6C)CC3)CC4)N=C12	C51H59F3N10O9	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-KGBFS9	WO2024263586A1_285	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CCCC5(CCO5)C4)=C3C=N1)=CC=C2	C60H70F2N10O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-O7S39J	WO2024263586A1_286	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=C8C(=CC=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)CC6)CC4)CC5)=NC(N4CCCC5(CCO5)C4)=C3C=N1)=CC=C2	C60H70F2N10O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-QNF05E	WO2024263586A1_287	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OC6CC7(C6)CN(C6=CC=C8C(=C6)N(C)C(=O)N8C6CCC(=O)NC6=O)C7)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C59H63F2N11O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-WV2I9T	WO2024263586A1_288	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(C3CCN(CC4CCN(C(=O)OC[C@@H]5CC[C@]6(COC7=NC(N8CC9CCC(C8)N9)=C8C=NC(C9=CC(O)=CC=C9OC(F)(F)F)=C(F)C8=N7)CCCN56)CC4)CC3)C=C21	C54H63F4N11O8	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-UTIJ7P	WO2024263586A1_289	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(CN3CCN(CCC4CCN(C(=O)OC[C@@H]5CC[C@]6(COC7=NC(N8CC9CCC(C8)N9)=C8C=NC(C9=CC(O)=CC=C9OC(F)(F)F)=C(F)C8=N7)CCCN56)CC4)CC3)C=C21	C55H66F4N12O8	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-HFGLD5	WO2024263586A1_29	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)NCCCCCCCCC4=CC=C6C(=C4)N(C)C(=O)N6C4CCC(=O)NC4=O)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C56H62F2N10O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-AJGCBU	WO2024263586A1_290	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(C3CCN(CC4CCN(C(=O)OC[C@@H]5CC[C@]6(COC7=NC(N8CC9CCC(C8)N9)=C8C=NC(C9=CC(O)=CC(Cl)=C9C9CC9)=C(F)C8=N7)CCCN56)CC4)CC3)C=C21	C56H67ClFN11O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-UB0NXI	WO2024263586A1_291	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(CN3CCN(CCC4CCN(C(=O)OC[C@@H]5CC[C@]6(COC7=NC(N8CC9CCC(C8)N9)=C8C=NC(C9=CC(O)=CC(Cl)=C9C9CC9)=C(F)C8=N7)CCCN56)CC4)CC3)C=C21	C57H70ClFN12O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-AOXZBJ	WO2024263586A1_292	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(O[C@H]6CC[C@H](C7=C8C(=CC=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C59H64F2N10O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-488YT2	WO2024263586A1_293	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(O[C@H]6CC[C@@H](C7=C8C(=CC=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C59H64F2N10O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-FFQAFO	WO2024263586A1_294	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=CC=C8C(C9CCC(=O)NC9=O)=NN(C)C8=C7F)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C59H64F3N11O5	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-LG0N26	WO2024263586A1_295	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=C(F)C=C8C(=C7)N(C)N=C8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C59H64F3N11O5	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-5BJ3TR	WO2024263586A1_296	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(O[C@H]6CC[C@@H](C7=CC=C8C(=C7)N(C)N=C8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C59H64F2N10O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-IAX6AP	WO2024263586A1_297	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(O[C@H]6CC[C@H](C7=CC=C8C(=C7)N(C)N=C8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C59H64F2N10O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-CFRKWT	WO2024263586A1_298	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(O[C@H]6CC[C@@H](C7=CC=C8C(=C7)N(C)N=C8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CCCC5(CCO5)C4)=C3C=N1)=CC(O)=C2	C60H69F2N9O8	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-J89WWC	WO2024263586A1_299	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(O[C@H]6CC[C@H](C7=CC=C8C(=C7)N(C)N=C8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CCCC5(CCO5)C4)=C3C=N1)=CC(O)=C2	C60H69F2N9O8	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-GJRJJO	WO2024263586A1_3	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)NCCCC4=C6C(=CC=C4)N(C4CCC(=O)NC4=O)C(=O)N6C)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC(O)=C2	C51H52F2N10O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-IO0I0V	WO2024263586A1_300	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(O[C@H]6CC[C@@H](C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CCCC5(CCO5)C4)=C3C=N1)=CC(O)=C2	C60H69F2N9O9	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-4RPPLR	WO2024263586A1_301	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(O[C@H]6CC[C@H](C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CCCC5(CCO5)C4)=C3C=N1)=CC(O)=C2	C60H69F2N9O9	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-DFLSDY	WO2024263586A1_302	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCN(CC6CCN(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C58H64F2N12O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-SU9BRD	WO2024263586A1_303	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCN(CC6CCN(C7=CC=C8C(=C7)N(C)N=C8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C58H64F2N12O5	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-MVUXLT	WO2024263586A1_304	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CC6CC7(C6)CN(C6=CC=C8C(=C6)N(C)N=C8C6CCC(=O)NC6=O)C7)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C60H65F2N11O5	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-T0I3GP	WO2024263586A1_305	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCC6CN(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)C6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C57H61F2N11O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-9SKI9M	WO2024263586A1_306	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OC6CC(C#CC7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)C6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C59H60F2N10O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-R0S2P1	WO2024263586A1_307	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OC6CC(C#CC7=C8C(=CC=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)C6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C59H60F2N10O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-JLMSY2	WO2024263586A1_308	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4C(COC(=O)N4CCC(OCC#CC#CCC6=CC=C7C(=C6)N(C)C(=O)N7C6CCC(=O)NC6=O)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C59H58F2N10O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-IC569Z	WO2024263586A1_309	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CC(OCC6CCN(C7=C8C(=CC=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)CC6)C4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C57H61F2N11O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-O1N6GH	WO2024263586A1_310	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CC(COC6CCN(C7=C8C(=CC=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)CC6)C4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C57H61F2N11O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-2LV4FO	WO2024263586A1_311	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@]45CCCN4[C@@H](COC(=O)N4CCC(CN6CCC(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CCCC5(CCO5)C4)=C3C=N1)=CC(O)=C2	C60H70F2N10O8	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-R2FVHY	WO2024263586A1_312	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(COC6CN(C7=C8C(=CC=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)C6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C57H61F2N11O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-HRDN1W	WO2024263586A1_313	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OC6CC7(C6)CN(C6=C8C(=CC=C6)N(C6CCC(=O)NC6=O)C(=O)N8C)C7)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C59H63F2N11O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-7PUSJ6	WO2024263586A1_314	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CC6CC7(C6)CN(C6=C8C(=CC=C6)N(C6CCC(=O)NC6=O)C(=O)N8C)C7)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C60H65F2N11O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-2IA6I3	WO2024263586A1_315	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CCC6CC7(C6)CN(C6=C8C(=CC=C6)N(C6CCC(=O)NC6=O)C(=O)N8C)C7)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C61H67F2N11O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-ZRZI6I	WO2024263586A1_316	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCCOCCOC6=CC=CC(C(=O)NC7CCC(=O)NC7=O)=C6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C56H61F2N9O9	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-4UG3G8	WO2024263586A1_317	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCCOCCOC6=CC=CC(C(=O)N[C@H]7CCC(=O)NC7=O)=C6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C56H61F2N9O9	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-I1YL0P	WO2024263586A1_318	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OCC45CCCN4[C@H](COC(=O)N4CCC(OCCOCCOCCOCCOC6=CC=C(C(=O)N[C@H]7CCC(=O)NC7=O)C=C6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C60H69F2N9O11	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-32JKBN	WO2024263586A1_319	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCCOCCOCCOCCOC6=CC=C(C(=O)N[C@@H]7CCC(=O)NC7=O)C=C6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C60H69F2N9O11	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-D56939	WO2024263586A1_32	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCCCC6=C7C(=CC=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC4)CC5)=NC(C4CC5CCC(C4)N5)=C3C=N1)=CC(O)=C2	C57H61F2N9O8	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-WT8T4F	SCHEMBL31282175	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 4-[2-[2-[2-[2-[3-[[(3S)-2,6-dioxopiperidin-3-yl]carbamoyl]phenoxy]ethoxy]ethoxy]ethoxy]ethoxy]piperidine-1-carboxylate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCCOCCOCCOCCOC6=CC=CC(C(=O)N[C@H]7CCC(=O)NC7=O)=C6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C60H69F2N9O11	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-QKWIYL	WO2024263586A1_321	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCCOCCOCCOCCOC6=CC=CC(C(=O)NC7CCC(=O)NC7=O)=C6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C60H69F2N9O11	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-6FRFC7	WO2024263586A1_322	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCCOCCOC6=CC=C(C(=O)N[C@H]7CCC(=O)NC7=O)C=C6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C56H61F2N9O9	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-ZN3LQ2	WO2024263586A1_323	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCCOCCOC6=CC=C(C(=O)N[C@@H]7CCC(=O)NC7=O)C=C6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C56H61F2N9O9	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-HWDJQ6	WO2024263586A1_324	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCCOCCOCCOCCC6=CC=CC(C7CCC(=O)NC7=O)=C6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C59H68F2N8O9	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-8TA048	WO2024263586A1_325	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCCOCCC6=CC=CC(C7CCC(=O)NC7=O)=C6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C55H60F2N8O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-R1AD2D	WO2024263586A1_326	.	[H]C1=C(C2=CC=CC3=C2C(C#C)=C(F)C=C3)N=CC2=C(N3CC4CCC(C3)N4)N=C(OC[C@@]34CCCN3[C@H](COC(=O)N3CCC(OCCOCCOCCOCCOC5=CC=CC(NC6CCC(=O)NC6=O)=C5)CC3)CC4)N=C12	C59H70FN9O10	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-8YGU54	WO2024263586A1_327	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=CC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCCOCCOCCOCCOC6=CC=C(NC7CCC(=O)NC7=O)C=C6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C60H70F2N8O10	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-XANCA4	WO2024263586A1_328	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCCOCCC6=CC=C(N7CCC(=O)NC7=O)C=C6)CC4)CC5)=CC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C55H60F2N8O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-BOJCRV	WO2024263586A1_329	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCCOCCOCCOCCC6=CC=CC(N7CCC(=O)NC7=O)=C6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C58H67F2N9O9	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-207PG0	WO2024263586A1_330	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCCOCCOCCOCCC6=CC=C(N7CCC(=O)NC7=O)C=C6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C58H67F2N9O9	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-E4SNY4	WO2024263586A1_331	.	[H]C1=C(C2=CC(O)=CC3=C2C(CC)=C(F)C=C3)N=CC2=C(N3CCCC4(CCO4)C3)N=C(OC[C@@]34CCCN3[C@H](COC(=O)N3CCC(CN5CCC(C6=CC=C7C(C8CCC(=O)NC8=O)=NN(C)C7=C6F)CC5)CC3)CC4)N=C12	C60H70F2N10O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-3F71GC	WO2024263586A1_332	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCN(C7=CC=C8C(=C7)N(C)N=C8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C58H64F2N12O5	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-GNLPVB	WO2024263586A1_333	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCN(CC6CCN(C7=CC=C8C(C9CCC(=O)NC9=O)=NN(C)C8=C7F)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C58H63F3N12O5	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-8Z5DK4	WO2024263586A1_334	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCN(CC6CCN(C7=C(F)C=C8C(=C7)N(C)N=C8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C58H63F3N12O5	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-7LRQDG	WO2024263586A1_335	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=CC=C8C(=C7)N(C)N=C8C7CCC(=O)NC7=O)C(F)(F)C6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C59H63F4N11O5	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-83WFT1	WO2024263586A1_336	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=C(F)C=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)C(F)(F)C6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C59H62F5N11O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-KX3O6I	WO2024263586A1_337	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=C(F)C=C8C(=C7)N(C)N=C8C7CCC(=O)NC7=O)C(F)(F)C6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C59H62F5N11O5	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-L3OS2Y	WO2024263586A1_338	.	CCC1=C(F)C=CC2=C1C(C1=C(N)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=CC=C8C(=C7F)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CCCC5(CCO5)C4)=C3C=N1)=CC(O)=C2	C60H71F2N11O8	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-0XIMHP	WO2024263586A1_339	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=C(F)C=C8C(=C7)N(C)N=C8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CCCC5(CCO5)C4)=C3C=N1)=CC(O)=C2	C60H69F3N10O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-L13Z2X	WO2024263586A1_34	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCCCC6=C7C(=CC=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC4)CC5)=NC(N4C=CCC5(CCO5)C4)=C3C=N1)=CC(O)=C2	C57H63F2N9O9	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-F5ZXFC	WO2024263586A1_340	.	[H]=C(OC[C@@H]1CC[C@]2(COC3=NC(N4CCCC5(CCO5)C4)=C4C=NC(C5=CC(O)=CC6=C5C(CC)=C(F)C=C6)=C(F)C4=N3)CCCN12)N1CCN(CC2CCN(C3=CC=C4C(=C3)N(C)N=C4C3CCC(=O)NC3=O)CC2)CC1	C59H71F2N11O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-LILCGF	WO2024263586A1_341	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCN(CC6CCN(C7=CC=C8C(C9CCC(=O)NC9=O)=NN(C)C8=C7F)CC6)CC4)CC5)=NC(N4CCCC5(CCO5)C4)=C3C=N1)=CC(O)=C2	C59H68F3N11O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-9G5LYB	WO2024263586A1_342	.	CCC1=C(F)C=CC2=C1C(C1=C(S)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCN(CC6CCN(C7=C(F)C=C8C(=C7)N(C)N=C8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CCCC5(CCO5)C4)=C3C=N1)=CC(O)=C2	C59H69F2N11O7S	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-UNQ0VZ	WO2024263586A1_343	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCN(CC6CCN(C7=C(F)C=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C58H63F3N12O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-RIS7UX	WO2024263586A1_344	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=CC=C8C(=C7F)N(C)C(=O)N8C7CCC(=O)NC7=O)C(F)(F)C6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C59H62F5N11O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-UHM56P	WO2024263586A1_345	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=CC=C8C(C9CCC(=O)NC9=O)=NN(C)C8=C7F)C(F)(F)C6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C59H62F5N11O5	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-491W9K	WO2024263586A1_346	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=CC=C8C(=C7)N(C)N=C8C7CCC(=O)NC7=O)C(F)(F)C6)CC4)CC5)=NC(N4CCCC5(CCO5)C4)=C3C=N1)=CC(O)=C2	C60H68F4N10O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-S49R77	WO2024263586A1_347	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCN(CC6CCN(C7=CC=C8C(=C7F)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C58H63F3N12O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-L9DFOW	WO2024263586A1_348	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCN(CC6CCN(C7=CC=C8C(=C7F)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CCCC5(CCO5)C4)=C3C=N1)=CC(O)=C2	C59H68F3N11O8	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-SGXW8L	WO2024263586A1_349	.	CCC1=C(F)C=CC2=C1C(C1=C(S)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCN(CC6CCN(C7=C(F)C=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CCCC5(CCO5)C4)=C3C=N1)=CC(O)=C2	C59H69F2N11O8S	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-IBCHL2	WO2024263586A1_35	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4C(COC(=O)N4CCC(OCCCC6=C7C(=CC=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC4)CC5)=NC(N4CCCC5(CCO5)C4)=C3C=N1)=CC(O)=C2	C57H61F2N9O9	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-KXX952	WO2024263586A1_350	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCN(CC6CCN(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CCCC5(CCO5)C4)=C3C=N1)=CC(O)=C2	C59H69F2N11O8	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-PXR7AX	WO2024263586A1_351	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=C(F)C=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CCCC5(CCO5)C4)=C3C=N1)=CC(O)=C2	C60H69F3N10O8	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-EPSDRB	WO2024263586A1_352	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)C(F)(F)C6)CC4)CC5)=NC(N4CCCC5(CCO5)C4)=C3C=N1)=CC(O)=C2	C60H68F4N10O8	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-93L3XW	WO2024263586A1_353	.	CCC1=C(F)C=CC(/C=C(O)\C=C\C2=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OC6CCN(C7=C(F)C=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CCCC5(CCO5)C4)=C3C=N2)=C1	C59H69F3N10O9	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-ZK99R4	WO2024263586A1_354	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OC6CCN(C7=CC=C8C(=C7F)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CCCC5(CCO5)C4)=C3C=N1)=CC(O)=C2	C59H67F3N10O9	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-QTN7L9	WO2024263586A1_355	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OC6CCN(C7=C(F)C=C8C(=C7)N(C)N=C8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CCCC5(CCO5)C4)=C3C=N1)=CC(O)=C2	C59H67F3N10O8	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-NOOKD7	WO2024263586A1_356	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OC6CCN(C7=CC=C8C(=C7)N(C)N=C8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CCCC5(CCO5)C4)=C3C=N1)=CC(O)=C2	C59H68F2N10O8	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-K500UX	WO2024263586A1_357	.	CCC1=C(F)C=CC(/C=C(O)\C=C\C2=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CCC[C@]5(CCO5)C4)=C3C=N2)=C1	C60H72F2N10O8	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-J60J0T	WO2024263586A1_358	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CCC[C@@]5(CCO5)C4)=C3C=N1)=CC(O)=C2	C60H70F2N10O8	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-NCLINY	WO2024263586A1_359	.	CCC1=C(F)C=CC2=C1C(C1=C(N)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=CC=C8C(=C7)N(C)N=C8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CCC[C@]5(CCO5)C4)=C3C=N1)=CC(O)=C2	C60H72FN11O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-ZC1Z25	WO2024263586A1_36	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COCN4CCC(OCCCC6=C7C(=CC=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC4)CC5)=NC(N4CCCC5(CCO5)C4)=C3C=N1)=CC=C2	C57H63F2N9O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-SP94RE	WO2024263586A1_360	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=CC=C8C(=C7)N(C)N=C8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CCC[C@@]5(CCO5)C4)=C3C=N1)=CC(O)=C2	C60H70F2N10O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-0PA53V	WO2024263586A1_361	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@]45CCCN4[C@@H](COC(=O)N4CCC(CN6CCC(C7=CC=C8C(=C7)N(C)N=C8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CCCC5(CCO5)C4)=C3C=N1)=CC(O)=C2	C60H70F2N10O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-JXV8ND	WO2024263586A1_362	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OC6CCN(C7=CC=C8C(=C7F)N(C)NC8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CCCC5(CCO5)C4)=C3C=N1)=CC(O)=C2	C59H69F3N10O8	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-MXD9H9	WO2024263586A1_38	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=CC(OCC45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=C8C(=CC=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C60H66F2N10O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-3G8N4S	WO2024263586A1_39	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl N-[4-[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-4-yl]piperidin-1-yl]-4-oxobutyl]carbamate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)NCCCC(=O)N4CCC(C6=C7C(=CC=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C57H61F2N11O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-2IQC7H	SCHEMBL31556826	[(3S,8S)-8-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(4S)-1-oxa-8-azaspiro[3.5]nonan-8-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 4-[3-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]prop-2-ynyl]piperidine-1-carboxylate	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CC#CC6=CC=C7C(=C6)N(C)C(=O)N7C6CCC(=O)NC6=O)CC4)CC5)=NC(N4CCC[C@]5(CCO5)C4)=C3C=N1)=CC(O)=C2	C57H61F2N9O8	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-QED0EQ	WO2024263586A1_401	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCCC#CC6=CC=C7C(=C6)N(C)C(=O)N7C6CCC(=O)NC6=O)CC4)CC5)=NC(N4CCC[C@]5(CCO5)C4)=C3C=N1)=CC(O)=C2	C58H63F2N9O9	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-EJ96DM	WO2024263586A1_402	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(C#CC6=CC=C7C(=C6)N(C)C(=O)N7C6CCC(=O)NC6=O)CC4)CC5)=NC(N4CCC[C@]5(CCO5)C4)=C3C=N1)=CC(O)=C2	C56H59F2N9O8	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-D9HD79	SCHEMBL31282938	[(3S,8S)-8-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(4S)-1-oxa-8-azaspiro[3.5]nonan-8-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 2-[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidin-1-yl]-7-azaspiro[3.5]nonane-7-carboxylate	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC6(CC4)CC(N4CCC(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC4)C6)CC5)=NC(N4CCC[C@]5(CCO5)C4)=C3C=N1)=CC(O)=C2	C62H72F2N10O8	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-V3CH6K	WO2024263586A1_404	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CC6(CC(N7CCC(C8=CC=C9C(=C8)N(C)C(=O)N9C8CCC(=O)NC8=O)CC7)C6)C4)CC5)=CC(N4CCC[C@]5(CCO5)C4)=C3C=N1)=CC(O)=C2	C61H69F2N9O8	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-4NOUQU	WO2024263586A1_405	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CC6(CC(CN7CCC(C8=CC=C9C(=C8)N(C)C(=O)N9C8CCC(=O)NC8=O)CC7)C6)C4)CC5)=NC(N4CCC[C@]5(CCO5)C4)=C3C=N1)=CC(O)=C2	C61H70F2N10O8	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-UIJTIC	WO2024263586A1_406	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)C(F)(F)C6)CC4)CC5)=NC(N4CCC[C@]5(CCO5)C4)=C3C=N1)=CC(O)=C2	C60H68F4N10O8	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-ES4K2R	WO2024263586A1_407	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=C(F)C=C8C(=C7)N(C)N=C8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CCC[C@]5(CCO5)C4)=C3C=N1)=CC(O)=C2	C60H69F3N10O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-AILECY	SCHEMBL31281842	[(3S,8S)-8-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(4R)-1-oxa-8-azaspiro[3.5]nonan-8-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 4-[[4-[3-(2,6-dioxopiperidin-3-yl)-5-fluoro-1-methylindazol-6-yl]piperidin-1-yl]methyl]piperidine-1-carboxylate	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=C(F)C=C8C(=C7)N(C)N=C8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CCC[C@@]5(CCO5)C4)=C3C=N1)=CC(O)=C2	C60H69F3N10O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-LVYT85	SCHEMBL31282671	[(3S,8S)-8-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-(2-oxa-8-azaspiro[3.5]nonan-8-yl)pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 4-[[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidin-1-yl]methyl]piperidine-1-carboxylate	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CCCC5(COC5)C4)=C3C=N1)=CC(O)=C2	C60H70F2N10O8	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-KGS61F	SCHEMBL26830689	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 4-[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-4-yl]butyl]piperidine-1-carboxylate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CCCCC6=C7C(=CC=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C57H62F2N10O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-GERMF6	WO2024263586A1_410	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@]45CCCN4[C@@H](COC(=O)N4CCC(CN6CCC(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CCC[C@]5(CCO5)C4)=C3C=N1)=CC(O)=C2	C60H70F2N10O8	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-FLBKNT	WO2024263586A1_411	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=CC=C8C(=C7)C(C7CCC(=O)NC7=O)=NN8C)CC6)CC4)CC5)=NC(N4CCC[C@]5(CCO5)C4)=C3C=N1)=CC(O)=C2	C60H70F2N10O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-0MFGKS	WO2024263586A1_412	.	[H]C1=C(C2=CC(O)=CC3=C2C(CC)=C(F)C=C3)N=CC2=C(N3CCC[C@]4(CCO4)C3)N=C(OC[C@@]34CCCN3[C@H](COC(=O)N3CCC(CN5CCC(C6=C7C(=CC=C6)C(C6CCC(=O)NC6=O)=NN7C)CC5)CC3)CC4)N=C12	C60H71FN10O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-QL9RD8	SCHEMBL31281746	[(3S,8S)-8-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(4S)-1-oxa-8-azaspiro[3.5]nonan-8-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 4-[[4-[1-(2,6-dioxopiperidin-3-yl)-6-fluoro-3-methyl-2-oxobenzimidazol-5-yl]piperidin-1-yl]methyl]piperidine-1-carboxylate	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=C(F)C=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CCC[C@]5(CCO5)C4)=C3C=N1)=CC(O)=C2	C60H69F3N10O8	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-U57YFP	SCHEMBL31282578	[(3S,8S)-8-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(4R)-1-oxa-8-azaspiro[3.5]nonan-8-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 4-[[4-[1-(2,6-dioxopiperidin-3-yl)-6-fluoro-3-methyl-2-oxobenzimidazol-5-yl]piperidin-1-yl]methyl]piperidine-1-carboxylate	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=C(F)C=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CCC[C@@]5(CCO5)C4)=C3C=N1)=CC(O)=C2	C60H69F3N10O8	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-M4I42F	WO2024263586A1_415	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OC6CCN(C7=CC=C8C(=C7)N(C)N=C8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CCC[C@]5(CCO5)C4)=C3C=N1)=CC(O)=C2	C59H68F2N10O8	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-GRCFHJ	SCHEMBL31282071	[(3S,8S)-8-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(4R)-1-oxa-8-azaspiro[3.5]nonan-8-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 4-[1-[3-(2,6-dioxopiperidin-3-yl)-1-methylindazol-6-yl]piperidin-4-yl]oxypiperidine-1-carboxylate	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OC6CCN(C7=CC=C8C(=C7)N(C)N=C8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CCC[C@@]5(CCO5)C4)=C3C=N1)=CC(O)=C2	C59H68F2N10O8	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-CX4PIF	SCHEMBL31282906	[(3S,8S)-8-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(4S)-1-oxa-8-azaspiro[3.5]nonan-8-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 4-[1-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidin-4-yl]oxypiperidine-1-carboxylate	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OC6CCN(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CCC[C@]5(CCO5)C4)=C3C=N1)=CC(O)=C2	C59H68F2N10O9	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-NH6K07	SCHEMBL31282327	[(3S,8S)-8-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(4R)-1-oxa-8-azaspiro[3.5]nonan-8-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 4-[1-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidin-4-yl]oxypiperidine-1-carboxylate	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OC6CCN(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CCC[C@@]5(CCO5)C4)=C3C=N1)=CC(O)=C2	C59H68F2N10O9	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-1E1MMM	SCHEMBL31282252	[(3R,8R)-8-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-[(4R)-1-oxa-8-azaspiro[3.5]nonan-8-yl]pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 4-[[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidin-1-yl]methyl]piperidine-1-carboxylate	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@]45CCCN4[C@@H](COC(=O)N4CCC(CN6CCC(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CCC[C@@]5(CCO5)C4)=C3C=N1)=CC(O)=C2	C60H70F2N10O8	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-8VFCVY	WO2024263586A1_42	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CC(CN6CCN(C7=CC=C8C(=C7)N(C)C(=O)C8C7CCC(=O)NC7=O)CC6)C4)CC5)=CC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C58H62F2N10O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-DYXHF2	SCHEMBL31282299	[(3S,8S)-8-[[7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoro-4-(1-oxa-8-azaspiro[3.5]nonan-8-yl)pyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 4-[[4-[3-(2,6-dioxopiperidin-3-yl)-1-methyl-2-oxobenzimidazol-5-yl]piperidin-1-yl]methyl]piperidine-1-carboxylate	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=CC=C8C(=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)CC6)CC4)CC5)=NC(N4CCCC5(CCO5)C4)=C3C=N1)=CC(O)=C2	C60H70F2N10O8	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-82YDI9	WO2024263586A1_421	.	C#CC1=CC=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=CC=C8C(=C7)N(C)N=C8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC4=C3C(=N1)OC[C@@H]1[C@@H]3CC[C@H](CN41)N3)=CC=C2	C60H66FN11O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-NH5PWZ	WO2024263586A1_422	.	C#CC1=CC=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC4=C3C(=N1)O[C@@H]1[C@@H]3CC[C@H](CN41)N3)=CC=C2	C59H64FN11O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-3XOXHY	WO2024263586A1_423	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=CC=C8C(=C7)N(C)N=C8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC4=C3C(=N1)OC[C@@H]1[C@@H]3CC[C@H](CN41)N3)=CC=C2	C60H65F2N11O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-D8XRO6	WO2024263586A1_424	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC4=C3C(=N1)OC[C@@H]1[C@@H]3CC[C@H](CN41)N3)=CC=C2	C60H65F2N11O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-L1PA2T	WO2024263586A1_427	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CC6CN(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)C6)CC4)CC5)=NC(N4CCC[C@]5(CCO5)C4)=C3C=N1)=CC(O)=C2	C58H66F2N10O8	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-2OIUY4	WO2024263586A1_428	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(NC6CCN(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CCC[C@]5(CCO5)C4)=C3C=N1)=CC(O)=C2	C59H69F2N11O8	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-GL9ATU	SCHEMBL31282010	[(3S,8R)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 2-[4-[1-(2,6-dioxopiperidin-3-yl)-6-fluoro-3-methyl-2-oxobenzimidazol-5-yl]piperidin-1-yl]-7-azaspiro[3.5]nonane-7-carboxylate	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@]45CCCN4[C@H](COC(=O)N4CCC6(CC4)CC(N4CCC(C7=C(F)C=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC4)C6)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C61H70F3N11O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-54X811	WO2024263586A1_43	.	C#CC1=C(F)C=CC2=C1C(C1=C(C)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CCCCC6=CC=C7C(=C6)N(C)C(=O)N7C6CCC(=O)NC6=O)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C58H65FN10O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-3P7SMP	WO2024263586A1_430	.	[H]C1=C(C2CCN(C3CC4(CCN(C(=O)OC[C@@H]5CC[C@]6(COC7=NC(N8CC9CCC(C8)N9)=C8C=NC(C9=CC=CC%10=C9C(CC)=C(F)C=C%10)=C(F)C8=N7)CCCN56)CC4)C3)CC2)C=C2C(=C1)N(C1CCC(=O)NC1=O)C(=O)N2C	C61H71F2N11O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-7HMJ7G	WO2024263586A1_431	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC6(CC4)CC(C4CCC(C7=C(F)C=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC4)C6)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C62H67F3N10O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-WSKXNR	WO2024263586A1_432	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=CC=C8C(=C7)N(C)N=C8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=C1F)=CC=C2	C60H65F3N10O5	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-ZMYN7J	SCHEMBL31282479	[(3S,8R)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 2-[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidin-1-yl]-7-azaspiro[3.5]nonane-7-carboxylate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@]45CCCN4[C@H](COC(=O)N4CCC6(CC4)CC(N4CCC(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC4)C6)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C61H67F2N11O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-VA76DC	WO2024263586A1_434	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(F)(CN6CCC(C7=C(F)C=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C59H63F4N11O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-ZOB83L	WO2024263586A1_435	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@]45CCCN4[C@H](COC(=O)N4CCC6(CC4)CC(N4CCC(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC4)C6)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C61H71F2N11O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-VCDQB0	WO2024263586A1_437	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(F)(CN6CCC(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C59H64F3N11O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-IO24BW	WO2024263586A1_438	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@]45CCCN4[C@H](COC(=O)N4CCC(CC6CCN(CC7=C8C(=CC=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C60H67F2N11O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-DJW9GA	WO2024263586A1_439	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=C8C(=CC=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C59H65F2N11O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-1ID2ZA	WO2024263586A1_440	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C59H62F2N10O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-RBUSE4	WO2024263586A1_441	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=CC=C8C(=C7)N(C)N=C8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=C1)=CC=C2	C60H66F2N10O5	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-7QO0BW	WO2024263586A1_442	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=C1F)=CC=C2	C60H65F3N10O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-RVGLRQ	WO2024263586A1_443	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=CC=C8C(=C7)N(C)N=C8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C59H65F2N11O5	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-DMIG9U	WO2024263586A1_444	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=C(F)C=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C59H64F3N11O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-XDVVQF	WO2024263586A1_445	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=C1)=CC=C2	C60H66F2N10O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-QIBXG3	WO2024263586A1_446	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC6(CC4)CC(N4CCC(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC4)C6)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C61H67F2N11O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-PB0CV0	SCHEMBL31282398	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 2-[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperazin-1-yl]-7-azaspiro[3.5]nonane-7-carboxylate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC6(CC4)CC(N4CCN(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC4)C6)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C60H66F2N12O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-3GILJH	SCHEMBL31281899	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-7-fluoro-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 4-[[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidin-1-yl]methyl]piperidine-1-carboxylate	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC(O)=C2	C59H69F2N11O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-W9PG9A	SCHEMBL31282692	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 4-[[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidin-1-yl]methyl]piperidine-1-carboxylate	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C59H69F2N11O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-WDWNYD	WO2024263586A1_450	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@]45CCCN4[C@H](COC(=O)N4CCC(CN6CCC(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C59H65F2N11O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-FSK1SE	WO2024263586A1_451	.	CCC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC6(CC4)CC(N4CCC(C7=C(F)C=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC4)C6)CC5)=NC(N4CCC[C@]5(CCO5)C4)=C3C=N1)=CC(O)=C2	C62H71F3N10O8	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-SKJYM9	WO2024263586A1_46	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC6(CC4)CN(CC#CC4=C7C(=CC=C4)N(C4CCC(=O)NC4=O)C(=O)N7C)CCO6)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C59H61F2N11O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-INOTFP	WO2024263586A1_47	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CC=CN4[C@H](COC(=O)N4CCC(CC6CCN(CC7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C60H65F2N11O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-AECHAD	WO2024263586A1_5	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)NCCCCCC4=CC=C6C(=C4)N(C)C(=O)N6C4CCC(=O)NC4=O)CC5)=CC(N4CC5CCC(C4)N5)=C3C=N1)=CC(O)=C2	C54H57F2N9O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-IA9EP5	WO2024263586A1_57	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(NC6CCN(CC7=C8C(=CC=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C59H68F2N12O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-65IK4Y	WO2024263586A1_59	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 4-[7-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-4-yl]heptoxy]piperidine-1-carboxylate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCCCCCCCC6=C7C(=CC=C6)N(C6CCC(=O)NC6=O)C(=O)N7C)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C60H68F2N10O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-1YMLI3	WO2024263586A1_60	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 9-[2-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-4-yl]ethyl]-3-azaspiro[5.5]undecane-3-carboxylate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC6(CCC(CCC7=C8C(=CC=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C60H66F2N10O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-9AVXZ4	WO2024263586A1_61	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCC4[C@H](COC(=O)N4CC6(CC(CCC7=C8C(=CC=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)C6)C4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C57H59F2N9O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-C2XPXR	SCHEMBL26831749	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 4-[[1-[[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-4-yl]methyl]piperidin-4-yl]methoxy]piperidine-1-carboxylate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCC6CCN(CC7=C8C(=CC=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C60H67F2N11O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-EJL8SI	WO2024263586A1_63	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(COC6CN(CC7=C8C(=CC=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)C6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C58H63F2N11O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-M4E1VB	SCHEMBL26831916	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 4-[1-[[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-4-yl]methyl]piperidin-4-yl]piperazine-1-carboxylate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCN(C6CCN(CC7=C8C(=CC=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C58H64F2N12O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-IUVL30	WO2024263586A1_65	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=CC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(N6CCC(CC7=C8C(=CC=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C60H66F2N10O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-O7RAZP	WO2024263586A1_66	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CC=CN4[C@H](COC(=O)N4CCC(N6CCC(OC7=C8C(=CC=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C58H61F2N11O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-TNR4CB	WO2024263586A1_68	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 4-[[1-[[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]methyl]piperidin-4-yl]oxymethyl]piperidine-1-carboxylate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(COC6CCN(CC7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C60H67F2N11O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-NBGLUJ	WO2024263586A1_69	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CCC6CCN(CC7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C61H69F2N11O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-R3MYHA	WO2024263586A1_78	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CC=CN4[C@H](COC(=O)N4CC(CN6CCC(OC7=C8C(=CC=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)CC6)C4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C57H59F2N11O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-FLL5HC	WO2024263586A1_80	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CC[C@H](CN6CCC(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)C4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C58H65F2N11O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-S1LWG0	WO2024263586A1_81	.	C#CC1=C(F)C=CC2=C1C(C1=CC3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CC[C@@H](CN6CCC(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)C4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C58H64FN11O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-KR8UA8	WO2024263586A1_82	.	[H]C1=C(C2=CC(O)=CC3=C2C(C#C)=C(F)C=C3)N=CC2=C(N3CC4CCC(C3)N4)N=C(OC[C@@]34CCCN3[C@H](COC(=O)N3CCC(CN5CCC(C6=CC=C7C(=C6)N(C)C(=O)N7C6CCC(=O)NC6=O)CC5)CC3)CC4)NC12	C59H68FN11O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-33OJEL	WO2024263586A1_83	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CC=CN4[C@H](COC(=O)N4CC(OC6CCN(CC7=C8C(=CC=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)CC6)C4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C57H59F2N11O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-P9OZYE	WO2024263586A1_84	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CCN6CCN(CC7=C8C(=CC=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C60H68F2N12O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-388RN5	WO2024263586A1_85	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCN(CCC6CCN(CC7=C8C(=CC=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C60H68F2N12O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-PKKOSY	WO2024263586A1_88	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCN(CCC6CCN(CC7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C60H68F2N12O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-HRT0EI	WO2024263586A1_90	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CC6CCN(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C59H65F2N11O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-J9XIRA	SCHEMBL26635044	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 4-[5-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]penta-2,4-diynoxy]piperidine-1-carboxylate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OCC#CC#CC6=CC=C7C(=C6)N(C)C(=O)N7C6CCC(=O)NC6=O)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C58H56F2N10O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-9EZ8SU	SCHEMBL26634864	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 4-[2-[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]triazol-1-yl]ethyl]piperidine-1-carboxylate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CCN6C=C(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)N=N6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C57H59F2N13O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-A1FTCH	WO2024263586A1_97	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 4-[2-[4-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-4-yl]triazol-1-yl]ethyl]piperidine-1-carboxylate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(CCN6C=C(C7=C8C(=CC=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)N=N6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C57H59F2N13O6	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-1305FW	SCHEMBL26635056	[(3S,8S)-8-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethynyl-7-fluoronaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]-1,2,3,5,6,7-hexahydropyrrolizin-3-yl]methyl 4-[1-[1-(2,6-dioxopiperidin-3-yl)-3-methyl-2-oxobenzimidazol-5-yl]piperidin-4-yl]oxypiperidine-1-carboxylate	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OC6CCN(C7=CC=C8C(=C7)N(C)C(=O)N8C7CCC(=O)NC7=O)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C58H63F2N11O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-R7AZ3E	WO2024263586A1_99	.	C#CC1=C(F)C=CC2=C1C(C1=C(F)C3=NC(OC[C@@]45CCCN4[C@H](COC(=O)N4CCC(OC6CCN(C7=C8C(=CC=C7)N(C7CCC(=O)NC7=O)C(=O)N8C)CC6)CC4)CC5)=NC(N4CC5CCC(C4)N5)=C3C=N1)=CC=C2	C58H63F2N11O7	KRAS	P01116	CRBN	WO-2024263586-A1
TPD-JJVTP8	SCHEMBL31343124	(2S,4R)-1-[(2R)-2-[3-[3-[[1-[(2S)-1-[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxypropan-2-yl]piperidin-4-yl]methyl]azetidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	[H]N1C2CCC1CN(C1=C3C=NC(C4=C5C(=CC(O)=C4)C=CC=C5CC)=C(F)C3=NC(OC[C@H](C)N3CCC(CC4CN(C5=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C5)C4)CC3)=N1)C2	C62H74FN11O6S	KRAS	P01116	VHL	WO-2025024732-A1
TPD-1L5CB2	WO2025024732A1_10	.	[H]N1C2CCC1CN(C1=C3C=NC(C4=C5C(=CC(O)=C4)C=CC(F)=C5C#C)=C(F)C3=NC(OCCN3CCC(CC4(F)CCN(C5=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C5)CC4)CC3)=N1)C2	C63H70F3N11O6S	KRAS	P01116	VHL	WO-2025024732-A1
TPD-FI8PMN	WO2025024732A1_11	.	[H]N1C2CCC1CN(C1=C3C=NC(C4=C5C(=CC(O)=C4)C=CC(F)=C5C#C)=C(F)C3=NC(OC[C@H](C)N3CCC(CC4CN(C5=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C5)C4)CC3)=N1)C2	C62H69F2N11O6S	KRAS	P01116	VHL	WO-2025024732-A1
TPD-NPT0QL	WO2025024732A1_12	.	[H]N1C2CCC1CN(C1=C3C=NC(C4=C5C(=CC(O)=C4)C=CC(F)=C5C#C)=C(F)C3=NC(OC[C@H](C)N3CCC(CC4CN(C5=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C5)C4)CC3)=N1)C2	C62H69F2N11O6S	KRAS	P01116	VHL	WO-2025024732-A1
TPD-5P2PN8	WO2025024732A1_13	.	[H]N1C2CCC1CN(C1=C3C=NC(C4=C5C(=CC(O)=C4)C=CC=C5CC)=C(F)C3=NC(OC[C@H](C)N3CCC(CC4CN(C5=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C5)C4)CC3)=N1)C2	C62H74FN11O6S	KRAS	P01116	VHL	WO-2025024732-A1
TPD-4DAET3	WO2025024732A1_14	.	[H]N1C2CCC1CN(C1=C3C=NC(C4=C5C(=CC(O)=C4)C=CC=C5CC)=C(F)C3=NC(OC[C@@H](C)N3CCC(CC4CN(C5=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C5)C4)CC3)=N1)C2	C62H74FN11O6S	KRAS	P01116	VHL	WO-2025024732-A1
TPD-QI28QF	WO2025024732A1_15	.	CCC1=CC=CC2=CC(O)=CC(C3=C(F)C4=NC(N5CC[C@@H](N6CCC(CC7CN(C8=NOC([C@@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)C9=CC=C(C%10=C(C)N=CS%10)C=C9)C(C)C)=C8)C7)CC6)C5)=NC(N5CC6CCC(C5)N6)=C4C=N3)=C21	C63H75FN12O5S	KRAS	P01116	VHL	WO-2025024732-A1
TPD-2FX9JC	WO2025024732A1_16	.	[H]N1C2CCC1CN(C1=C3C=NC(C4=C5C(=CC(O)=C4)C=CC=C5CC)=C(F)C3=NC(OCC3(CN4CCC(CC5CN(C6=NOC([C@@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)C)=C6)C5)CC4)CC3)=N1)C2	C64H76FN11O6S	KRAS	P01116	VHL	WO-2025024732-A1
TPD-RX4O5L	WO2025024732A1_17	.	[H]N1C2CCC1CN(C1=C3C=NC(C4=C5C(=CC(O)=C4)C=CC=C5CC)=C(F)C3=NC(OC[C@@H]3C[C@@H](OC4CCN(C5=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C5)CC4)CN3C)=N1)C2	C61H72FN11O7S	KRAS	P01116	VHL	WO-2025024732-A1
TPD-JGZ27J	WO2025024732A1_18	.	CCC1=CC=CC2=CC(O)=CC(C3=C(F)C4=NC(N5CC[C@H](N6CCC(CC7CN(C8=NOC([C@@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)C9=CC=C(C%10=C(C)N=CS%10)C=C9)C(C)C)=C8)C7)CC6)C5)=NC(N5CC6CCC(C5)N6)=C4C=N3)=C21	C63H75FN12O5S	KRAS	P01116	VHL	WO-2025024732-A1
TPD-I3NRQ1	WO2025024732A1_19	.	[H]N1C2CCC1CN(C1=C3C=NC(C4=C5C(=CC(O)=C4)C=CC(F)=C5C#C)=C(F)C3=NC(OCCN3CCC(CC4(F)CCN(C5=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C5)CC4)CC3)=N1)C2	C63H70F3N11O6S	KRAS	P01116	VHL	WO-2025024732-A1
TPD-07I5FO	WO2025024732A1_2	.	[H]N1C2CCC1CN(C1=C3C=NC(C4=C5C(=CC(O)=C4)C=CC=C5CC)=C(F)C3=NC(OC[C@@H](C)N3CCC(CC4CN(C5=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C5)C4)CC3)=N1)C2	C62H74FN11O6S	KRAS	P01116	VHL	WO-2025024732-A1
TPD-QZY4FJ	WO2025024732A1_20	.	[H]N1C2CCC1CN(C1=C3C=NC(C4=C5C(=CC=C4)C=CC(F)=C5C#C)=C(F)C3=NC(OCCN3CCC(CC4CN(C5=NOC([C@@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C5)C4)CC3)=N1)C2	C61H67F2N11O5S	KRAS	P01116	VHL	WO-2025024732-A1
TPD-R0O01O	WO2025024732A1_21	.	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=NC(OCCN5CCC(CC6CN(C7=NOC([C@@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)C8=CC=C(C9=C(C)N=CS9)C=C8)C(C)C)=C7)C6)CC5)=NC(N5CCCCCC5)=C4C=N3)=C21	C61H68F2N10O6S	KRAS	P01116	VHL	WO-2025024732-A1
TPD-PA6RWT	WO2025024732A1_3	.	CCC1=CC=CC2=CC(O)=CC(C3=C(F)C4=NC(N5CC[C@@H](N6CCC(CC7CN(C8=NOC([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)C9=CC=C(C%10=C(C)N=CS%10)C=C9)C(C)C)=C8)C7)CC6)C5)=NC(N5CC6CCC(C5)N6)=C4C=N3)=C21	C63H75FN12O5S	KRAS	P01116	VHL	WO-2025024732-A1
TPD-3Q699G	SCHEMBL31343156	(2S,4R)-1-[(2R)-2-[3-[3-[[1-[[1-[[4-(3,8-diazabicyclo[3.2.1]octan-3-yl)-7-(8-ethyl-3-hydroxynaphthalen-1-yl)-8-fluoropyrido[4,3-d]pyrimidin-2-yl]oxymethyl]cyclopropyl]methyl]piperidin-4-yl]methyl]azetidin-1-yl]-1,2-oxazol-5-yl]-3-methylbutanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	[H]N1C2CCC1CN(C1=C3C=NC(C4=C5C(=CC(O)=C4)C=CC=C5CC)=C(F)C3=NC(OCC3(CN4CCC(CC5CN(C6=NOC([C@H](C(=O)N7C[C@H](O)C[C@H]7C(=O)N[C@@H](C)C7=CC=C(C8=C(C)N=CS8)C=C7)C(C)C)=C6)C5)CC4)CC3)=N1)C2	C64H76FN11O6S	KRAS	P01116	VHL	WO-2025024732-A1
TPD-Q0M3L9	WO2025024732A1_5	.	[H]N1C2CCC1CN(C1=C3C=NC(C4=C5C(=CC(O)=C4)C=CC=C5CC)=C(F)C3=NC(OC[C@@H]3C[C@@H](OC4CCN(C5=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C5)CC4)CN3C)=N1)C2	C61H72FN11O7S	KRAS	P01116	VHL	WO-2025024732-A1
TPD-IB8QJQ	WO2025024732A1_6	.	[H]N1C2CCC1CN(C1=C3C=NC(C4=C5C(=CC=C4)C=CC(F)=C5C#C)=C(F)C3=NC(OCCN3CCC(CC4CN(C5=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C5)C4)CC3)=N1)C2	C61H67F2N11O5S	KRAS	P01116	VHL	WO-2025024732-A1
TPD-RXFZPW	WO2025024732A1_7	.	CCC1=CC=CC2=CC(O)=CC(C3=C(F)C4=NC(N5CC[C@H](N6CCC(CC7CN(C8=NOC([C@H](C(=O)N9C[C@H](O)C[C@H]9C(=O)N[C@@H](C)C9=CC=C(C%10=C(C)N=CS%10)C=C9)C(C)C)=C8)C7)CC6)C5)=NC(N5CC6CCC(C5)N6)=C4C=N3)=C21	C63H75FN12O5S	KRAS	P01116	VHL	WO-2025024732-A1
TPD-I62A6K	WO2025024732A1_8	.	[H]N1C2CCC1CN(C1=C3C=NC(C4=C5C(=CC(O)=C4)C=CC(F)=C5C#C)=C(F)C3=NC(OCCN3CCC(OC4CN(C5=NOC([C@H](C(=O)N6C[C@H](O)C[C@H]6C(=O)N[C@@H](C)C6=CC=C(C7=C(C)N=CS7)C=C6)C(C)C)=C5)C4)CC3)=N1)C2	C60H65F2N11O7S	KRAS	P01116	VHL	WO-2025024732-A1
TPD-H2105H	WO2025024732A1_9	.	C#CC1=C(F)C=CC2=CC(O)=CC(C3=C(F)C4=NC(OCCN5CCC(CC6CN(C7=NOC([C@H](C(=O)N8C[C@H](O)C[C@H]8C(=O)N[C@@H](C)C8=CC=C(C9=C(C)N=CS9)C=C8)C(C)C)=C7)C6)CC5)=NC(N5CCCCCC5)=C4C=N3)=C21	C61H68F2N10O6S	KRAS	P01116	VHL	WO-2025024732-A1
TPD-LDALXC	WO2025036489A1_1	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(CN5CCN6C7=C(C=C(C8CCC(=O)NC8=O)C(F)=C7)CC[C@H]6C5)CC4)C=C3)C2(C)C)=CC=C1C#N	C46H55FN6O5	AR	P10275	CRBN	WO-2025036489-A1
TPD-MBTT57	WO2025036489A1_10	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC5(CC4)CC(CN4CCN6C7=C(C=C(C8CCC(=O)NC8=O)C(F)=C7)CCC6C4)C5)C=C3)C2(C)C)=CC=C1C#N	C49H59FN6O5	AR	P10275	CRBN	WO-2025036489-A1
TPD-4C41I2	WO2025036489A1_100	.	CC#CCOC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(CN5CCN6C7=CC(F)=C(C(=O)N[C@H]8CCC(=O)NC8=O)C=C7CC[C@H]6C5)CC4)C=C3)C2(C)C)=CC=C1C#N	C50H58FN7O6	AR	P10275	CRBN	WO-2025036489-A1
TPD-WW59AG	WO2025036489A1_101	.	CC1=CC=C(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(CN5CCN6C7=CC(F)=C(C8CCC(=O)NC8=O)C=C7CC[C@H]6C5)CC4)C=C3)C2(C)C)C=C1OCCOC1CC1	C50H64FN5O6	AR	P10275	CRBN	WO-2025036489-A1
TPD-XN7PU4	WO2025036489A1_102	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(CN4CCN5C6=CC(F)=C(C7CCC(=O)NC7=O)C=C6CC[C@@H]5C4)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(OCCOC2CC2)=C1	C50H61FN6O6	AR	P10275	CRBN	WO-2025036489-A1
TPD-A2N8K7	WO2025036489A1_103	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(CN4CCN5C6=CC(F)=C(C(=O)N[C@H]7CCC(=O)NC7=O)C=C6CC[C@@H]5C4)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(OCCOC2CC2)=C1	C51H62FN7O7	AR	P10275	CRBN	WO-2025036489-A1
TPD-7THDRY	WO2025036489A1_104	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(CN4CCN5C6=CC(F)=C(C(=O)N[C@H]7CCC(=O)NC7=O)C=C6CC[C@H]5C4)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(OCCOC2CC2)=C1	C51H62FN7O7	AR	P10275	CRBN	WO-2025036489-A1
TPD-K4MX0M	WO2025036489A1_105	.	COCCOC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(CN5CCN6C7=CC(F)=C(C8CCC(=O)NC8=O)C=C7CC[C@@H]6C5)CC4)C=C3)C2(C)C)=CC=C1C#N	C48H59FN6O6	AR	P10275	CRBN	WO-2025036489-A1
TPD-KAO5RF	WO2025036489A1_106	.	COCCOC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(CN5CCN6C7=CC(F)=C(C8CCC(=O)NC8=O)C=C7CC[C@H]6C5)CC4)C=C3)C2(C)C)=CC=C1C#N	C48H59FN6O6	AR	P10275	CRBN	WO-2025036489-A1
TPD-IM91C9	WO2025036489A1_107	.	COCCOC1=CC(O[C@H]2C(C)(C)[C@@H](NC(=O)C3=CC=C(N4CCC(CN5CCN6C7=CC(F)=C(C(=O)N[C@H]8CCC(=O)NC8=O)C=C7CC[C@@H]6C5)CC4)C=C3)C2(C)C)=CC=C1C#N	C49H60FN7O7	AR	P10275	CRBN	WO-2025036489-A1
TPD-B2N8CQ	WO2025036489A1_108	.	COCCOC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(CN5CCN6C7=CC(F)=C(C(=O)NC8CCC(=O)NC8=O)C=C7CC[C@H]6C5)CC4)C=C3)C2(C)C)=CC=C1C#N	C49H60FN7O7	AR	P10275	CRBN	WO-2025036489-A1
TPD-E0DKXC	WO2025036489A1_109	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(CN4CCN5C6=CC(F)=C(C7CCC(=O)NC7=O)C=C6CC[C@@H]5C4)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(OCC2CC2)=C1	C49H59FN6O5	AR	P10275	CRBN	WO-2025036489-A1
TPD-RIZH6A	WO2025036489A1_11	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(CN5CCN6C7=C(C=C(C(=O)N[C@H]8CCC(=O)NC8=O)C(F)=C7)CC[C@@H]6C5)CC4)C=C3)C2(C)C)=CC=C1C#N	C47H56FN7O6	AR	P10275	CRBN	WO-2025036489-A1
TPD-MP5YOS	WO2025036489A1_110	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(CN4CCN5C6=CC(F)=C(C7CCC(=O)NC7=O)C=C6CC[C@H]5C4)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(OCC2CC2)=C1	C49H59FN6O5	AR	P10275	CRBN	WO-2025036489-A1
TPD-GV9HOG	WO2025036489A1_111	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(CN4CCN5C6=CC(F)=C(C(=O)N[C@H]7CCC(=O)NC7=O)C=C6CC[C@@H]5C4)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(OCC2CC2)=C1	C50H60FN7O6	AR	P10275	CRBN	WO-2025036489-A1
TPD-MYOFPY	WO2025036489A1_112	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(CN4CCN5C6=CC(F)=C(C(=O)N[C@@H]7CCC(=O)NC7=O)C=C6CC[C@H]5C4)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(OCC2CC2)=C1	C50H60FN7O6	AR	P10275	CRBN	WO-2025036489-A1
TPD-8UU9L9	WO2025036489A1_113	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(CN4CCN5C6=CC(F)=C(C7CCC(=O)NC7=O)C=C6CC[C@@H]5C4)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(CC2CC2)=C1	C49H59FN6O4	AR	P10275	CRBN	WO-2025036489-A1
TPD-5G1TBQ	WO2025036489A1_114	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(CN4CCN5C6=CC(F)=C(C7CCC(=O)NC7=O)C=C6CC[C@H]5C4)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(CC2CC2)=C1	C49H59FN6O4	AR	P10275	CRBN	WO-2025036489-A1
TPD-HIRX5Z	WO2025036489A1_115	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(CN4CCN5C6=CC(F)=C(C(=O)N[C@H]7CCC(=O)NC7=O)C=C6CC[C@@H]5C4)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(CC2CC2)=C1	C50H60FN7O5	AR	P10275	CRBN	WO-2025036489-A1
TPD-E3025Y	WO2025036489A1_116	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(CN4CCN5C6=CC(F)=C(C(=O)N[C@H]7CCC(=O)NC7=O)C=C6CC[C@H]5C4)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(CC2CC2)=C1	C50H60FN7O5	AR	P10275	CRBN	WO-2025036489-A1
TPD-SBY04N	WO2025036489A1_117	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(CN4CCN5C6=C(C=C(C7CCC(=O)NC7=O)C(F)=C6)CC[C@@H]5C4)CC3)C=C2)C(C)(C)[C@H]1OC1=CC(C2CC2)=C(C#N)C=C1	C48H57FN6O4	AR	P10275	CRBN	WO-2025036489-A1
TPD-TT2DTK	WO2025036489A1_118	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(CN4CCN5C6=C(C=C(C7CCC(=O)NC7=O)C(F)=C6)CC[C@H]5C4)CC3)C=C2)C(C)(C)[C@H]1OC1=CC(C2CC2)=C(C#N)C=C1	C48H57FN6O4	AR	P10275	CRBN	WO-2025036489-A1
TPD-ES4LR4	WO2025036489A1_119	.	CC1(C)C(NC(=O)C2=CC=C(N3CCC(CN4CCN5C6=CC(F)=C(C(=O)N[C@@H]7CCC(=O)NC7=O)C=C6CC[C@@H]5C4)CC3)C=C2)C(C)(C)C1OC1=CC=C(C#N)C(C2CC2)=C1	C49H58FN7O5	AR	P10275	CRBN	WO-2025036489-A1
TPD-BXTG0G	WO2025036489A1_12	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(CN5CCN6C7=C(C=C(C(=O)N[C@@H]8CCC(=O)NC8=O)C(F)=C7)CC[C@@H]6C5)CC4)C=C3)C2(C)C)=CC=C1C#N	C47H56FN7O6	AR	P10275	CRBN	WO-2025036489-A1
TPD-Z09M8P	WO2025036489A1_120	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(CN4CCN5C6=CC(F)=C(C(=O)N[C@H]7CCC(=O)NC7=O)C=C6CC[C@H]5C4)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(C2CC2)=C1	C49H58FN7O5	AR	P10275	CRBN	WO-2025036489-A1
TPD-JINBZ7	WO2025036489A1_121	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NCC3=CC=C(N4CCC5(CC4)CC(N4CCN6C7=C(C=C(C8CCC(=O)NC8=O)C(F)=C7)CC[C@H]6C4)C5)C=C3)C2(C)C)=CC=C1C#N	C48H59FN6O4	AR	P10275	CRBN	WO-2025036489-A1
TPD-CF73AS	WO2025036489A1_122	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC5(CC4)CC(N4CCN6C7=C(C=C(C8CCC(=O)NC8=O)C(F)=C7)CCC6C4)C5)C=C3)C2(C)C)=CC=C1C#N	C48H57FN6O5	AR	P10275	CRBN	WO-2025036489-A1
TPD-JXBRLX	WO2025036489A1_127	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(O[C@H]5C[C@H](N6CCN7C8=CC(F)=C(C9CCC(=O)NC9=O)C=C8CC[C@@H]7C6)C5)CC4)C=C3)C2(C)C)=CC=C1C#N	C49H59FN6O6	AR	P10275	CRBN	WO-2025036489-A1
TPD-5YJ2D9	WO2025036489A1_128	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(OC5CC(N6CCN7C8=CC(F)=C(C9CCC(=O)NC9=O)C=C8CCC7C6)C5)CC4)C=C3)C2(C)C)=CC=C1C#N	C49H59FN6O6	AR	P10275	CRBN	WO-2025036489-A1
TPD-1HBTT7	WO2025036489A1_129	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(O[C@H]5C[C@H](N6CCN7C8=CC(F)=C(N9CCC(=O)NC9=O)C=C8CC[C@@H]7C6)C5)CC4)C=C3)C2(C)C)=CC=C1C#N	C48H58FN7O6	AR	P10275	CRBN	WO-2025036489-A1
TPD-ZILXWO	WO2025036489A1_13	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(CN5CCN6C7=C(C=C(C(=O)N[C@H]8CCC(=O)NC8=O)C(F)=C7)CC[C@H]6C5)CC4)C=C3)C2(C)C)=CC=C1C#N	C47H56FN7O6	AR	P10275	CRBN	WO-2025036489-A1
TPD-WH2D7A	WO2025036489A1_130	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(OC5CC(N6CCN7C8=CC(F)=C(N9CCC(=O)NC9=O)C=C8CC[C@H]7C6)C5)CC4)C=C3)C2(C)C)=CC=C1C#N	C48H58FN7O6	AR	P10275	CRBN	WO-2025036489-A1
TPD-QEF47J	WO2025036489A1_14	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(CN5CCN6C7=C(C=C(C(=O)N[C@@H]8CCC(=O)NC8=O)C(F)=C7)CC[C@H]6C5)CC4)C=C3)C2(C)C)=CC=C1C#N	C47H56FN7O6	AR	P10275	CRBN	WO-2025036489-A1
TPD-GBL9EN	WO2025036489A1_15	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(CN5CCN6C7=CC=C(N8CCC(=O)NC8=O)C=C7CCC6C5)CC4)C=C3)C2(C)C)=CC=C1C#N	C45H55N7O5	AR	P10275	CRBN	WO-2025036489-A1
TPD-V702P5	WO2025036489A1_16	.	COC1=CC(OC2C(C)(C)C(NC(=O)C3=CC=C(N4CCC5(CC4)CC(N4CCN6C7=C(C=C(C(=O)NC8CCC(=O)NC8=O)C(F)=C7)CC[C@@H]6C4)C5)C=C3)C2(C)C)=CC=C1C#N	C49H58FN7O6	AR	P10275	CRBN	WO-2025036489-A1
TPD-VA0U5M	WO2025036489A1_17	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC5(CC4)CC(N4CCN6C7=C(C=C(C(=O)N[C@@H]8CCC(=O)NC8=O)C(F)=C7)CC[C@@H]6C4)C5)C=C3)C2(C)C)=CC=C1C#N	C49H58FN7O6	AR	P10275	CRBN	WO-2025036489-A1
TPD-DGAFVD	WO2025036489A1_18	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC5(CC4)CC(N4CCN6C7=C(C=C(C(=O)N[C@H]8CCC(=O)NC8=O)C(F)=C7)CC[C@H]6C4)C5)C=C3)C2(C)C)=CC=C1C#N	C49H58FN7O6	AR	P10275	CRBN	WO-2025036489-A1
TPD-6B4Q6I	WO2025036489A1_19	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC5(CC4)CC(N4CCN6C7=C(C=C(C(=O)N[C@@H]8CCC(=O)NC8=O)C(F)=C7)CC[C@H]6C4)C5)C=C3)C2(C)C)=CC=C1C#N	C49H58FN7O6	AR	P10275	CRBN	WO-2025036489-A1
TPD-0O8AMP	WO2025036489A1_2	.	C#CC1=CC=C(OC2C(C)(C)C(NC(=O)C3=CC=C(N4CCC(CN5CCN6C7=C(C=C(C8CCC(=O)NC8=O)C(F)=C7)CC[C@@H]6C5)CC4)C=C3)C2(C)C)C=C1OC	C47H56FN5O5	AR	P10275	CRBN	WO-2025036489-A1
TPD-VE012O	WO2025036489A1_20	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(N5CCN6C7=CC(F)=C(C8CCC(=O)NC8=O)C=C7CC[C@@H]6C5)CC4)C=C3)C2(C)C)=CC=C1C#N	C45H53FN6O5	AR	P10275	CRBN	WO-2025036489-A1
TPD-LWBF3Q	WO2025036489A1_21	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(N5CCN6C7=CC(F)=C(C8CCC(=O)NC8=O)C=C7CC[C@H]6C5)CC4)C=C3)C2(C)C)=CC=C1C#N	C45H53FN6O5	AR	P10275	CRBN	WO-2025036489-A1
TPD-S6YFVZ	WO2025036489A1_22	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(N5CCN6C7=CC(F)=C(C(=O)NC8CCC(=O)NC8=O)C=C7CC[C@@H]6C5)CC4)C=C3)C2(C)C)=CC=C1C#N	C46H54FN7O6	AR	P10275	CRBN	WO-2025036489-A1
TPD-LFUEES	WO2025036489A1_23	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(N5CCN6C7=CC(F)=C(C(=O)N[C@@H]8CCC(=O)NC8=O)C=C7CC[C@@H]6C5)CC4)C=C3)C2(C)C)=CC=C1C#N	C46H54FN7O6	AR	P10275	CRBN	WO-2025036489-A1
TPD-SDIXIT	WO2025036489A1_24	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(N5CCN6C7=CC(F)=C(C(=O)N[C@H]8CCC(=O)NC8=O)C=C7CC[C@H]6C5)CC4)C=C3)C2(C)C)=CC=C1C#N	C46H54FN7O6	AR	P10275	CRBN	WO-2025036489-A1
TPD-4X6RCZ	WO2025036489A1_25	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(N5CCN6C7=CC(F)=C(C(=O)N[C@@H]8CCC(=O)NC8=O)C=C7CC[C@H]6C5)CC4)C=C3)C2(C)C)=CC=C1C#N	C46H54FN7O6	AR	P10275	CRBN	WO-2025036489-A1
TPD-TDJKZX	WO2025036489A1_26	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(F)(CN5CCN6C7=CC(F)=C(C8CCC(=O)NC8=O)C=C7CC[C@@H]6C5)CC4)C=C3)C2(C)C)=CC=C1C#N	C46H54F2N6O5	AR	P10275	CRBN	WO-2025036489-A1
TPD-4D54EK	WO2025036489A1_27	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(F)(CN5CCN6C7=CC(F)=C(C8CCC(=O)NC8=O)C=C7CC[C@H]6C5)CC4)C=C3)C2(C)C)=CC=C1C#N	C46H54F2N6O5	AR	P10275	CRBN	WO-2025036489-A1
TPD-D6XAVW	WO2025036489A1_28	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(CN5CCN6C7=CC(F)=C(N8CCC(=O)NC8=O)C=C7CC[C@@H]6C5)CC4)C=C3)C2(C)C)=CC=C1C#N	C45H54FN7O5	AR	P10275	CRBN	WO-2025036489-A1
TPD-1IZ68B	WO2025036489A1_29	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(CN5CCN6C7=CC(F)=C(N8CCC(=O)NC8=O)C=C7CC[C@H]6C5)CC4)C=C3)C2(C)C)=CC=C1C#N	C45H54FN7O5	AR	P10275	CRBN	WO-2025036489-A1
TPD-GHFD7M	WO2025036489A1_3	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(CN5CCN6C7=C(C=C(C(=O)NC8CCC(=O)NC8=O)C(F)=C7)CC[C@H]6C5)CC4)C=C3)C2(C)C)=CC=C1C#N	C47H56FN7O6	AR	P10275	CRBN	WO-2025036489-A1
TPD-MZBGV7	WO2025036489A1_30	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(CN4CCN5C6=CC(F)=C(C7CCC(=O)NC7=O)C=C6CC[C@@H]5C4)CC3)C=C2)C(C)(C)[C@H]1OC1=C2C=CC=NC2=C(C#N)C=C1	C48H54FN7O4	AR	P10275	CRBN	WO-2025036489-A1
TPD-58DC5Y	WO2025036489A1_31	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(CN4CCN5C6=CC(F)=C(C7CCC(=O)NC7=O)C=C6CC[C@H]5C4)CC3)C=C2)C(C)(C)[C@H]1OC1=C2C=CC=NC2=C(C#N)C=C1	C48H54FN7O4	AR	P10275	CRBN	WO-2025036489-A1
TPD-T9DNR6	WO2025036489A1_32	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(CN4CCN5C6=CC(F)=C(N7CCC(=O)NC7=O)C=C6CC[C@@H]5C4)CC3)C=C2)C(C)(C)[C@H]1OC1=C2C=CC=NC2=C(C#N)C=C1	C47H53FN8O4	AR	P10275	CRBN	WO-2025036489-A1
TPD-G8GM11	WO2025036489A1_33	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(CN4CCN5C6=CC(F)=C(N7CCC(=O)NC7=O)C=C6CC[C@H]5C4)CC3)C=C2)C(C)(C)[C@H]1OC1=C2C=CC=NC2=C(C#N)C=C1	C47H53FN8O4	AR	P10275	CRBN	WO-2025036489-A1
TPD-BTS4OO	WO2025036489A1_34	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(CN4CCN5C6=CC(F)=C(C(=O)N[C@H]7CCC(=O)NC7=O)C=C6CC[C@@H]5C4)CC3)C=C2)C(C)(C)[C@H]1OC1=C2C=CC=NC2=C(C#N)C=C1	C49H55FN8O5	AR	P10275	CRBN	WO-2025036489-A1
TPD-ZEMG80	WO2025036489A1_35	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(CN4CCN5C6=CC(F)=C(C(=O)N[C@H]7CCC(=O)NC7=O)C=C6CC[C@H]5C4)CC3)C=C2)C(C)(C)[C@H]1OC1=C2C=CC=NC2=C(C#N)C=C1	C49H55FN8O5	AR	P10275	CRBN	WO-2025036489-A1
TPD-WQUET0	WO2025036489A1_36	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(CN4CCN5C6=CC(F)=C(C7CCC(=O)NC7=O)C=C6CC[C@@H]5C4)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(OC(=O)OO)=C1	C46H53FN6O8	AR	P10275	CRBN	WO-2025036489-A1
TPD-CWGH90	WO2025036489A1_37	.	CC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(CN5CCN6C7=CC(F)=C(C8CCC(=O)NC8=O)C=C7CC[C@H]6C5)CC4)C=C3)C2(C)C)=CC=C1C#N	C46H55FN6O4	AR	P10275	CRBN	WO-2025036489-A1
TPD-9L3Q5E	WO2025036489A1_38	.	CC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(CN5CCN6C7=CC(F)=C(N8CCC(=O)NC8=O)C=C7CC[C@@H]6C5)CC4)C=C3)C2(C)C)=CC=C1C#N	C45H54FN7O4	AR	P10275	CRBN	WO-2025036489-A1
TPD-29PE8U	WO2025036489A1_39	.	CC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(CN5CCN6C7=CC(F)=C(N8CCC(=O)NC8=O)C=C7CC[C@H]6C5)CC4)C=C3)C2(C)C)=CC=C1C#N	C45H54FN7O4	AR	P10275	CRBN	WO-2025036489-A1
TPD-Y5THPK	WO2025036489A1_4	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(C4CCC(CN5CCN6C7=C(C=C(C(=O)NC8CCC(=O)NC8=O)C(F)=C7)CC[C@@H]6C5)CC4)C=C3)C2(C)C)=CC=C1C#N	C48H57FN6O6	AR	P10275	CRBN	WO-2025036489-A1
TPD-KLCKWK	WO2025036489A1_40	.	CC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(CN5CCN6C7=CC(F)=C(C(=O)N[C@H]8CCC(=O)NC8=O)C=C7CC[C@@H]6C5)CC4)C=C3)C2(C)C)=CC=C1C#N	C47H56FN7O5	AR	P10275	CRBN	WO-2025036489-A1
TPD-83DFE5	WO2025036489A1_41	.	CC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(CN5CCN6C7=CC(F)=C(C(=O)N[C@H]8CCC(=O)NC8=O)C=C7CC[C@H]6C5)CC4)C=C3)C2(C)C)=CC=C1C#N	C47H56FN7O5	AR	P10275	CRBN	WO-2025036489-A1
TPD-9S18D8	WO2025036489A1_42	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC4(CC3)CC(CN3CCN5C6=CC(F)=C(C7CCC(=O)NC7=O)C=C6CC[C@@H]5C3)C4)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(OC(=O)OO)=C1	C49H57FN6O8	AR	P10275	CRBN	WO-2025036489-A1
TPD-LNP01R	WO2025036489A1_43	.	CC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC5(CC4)CC(CN4CCN6C7=CC(F)=C(C8CCC(=O)NC8=O)C=C7CC[C@H]6C4)C5)C=C3)C2(C)C)=CC=C1C#N	C49H59FN6O4	AR	P10275	CRBN	WO-2025036489-A1
TPD-WB6DCS	WO2025036489A1_44	.	CC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC5(CC4)CC(CN4CCN6C7=CC(F)=C(N8CCC(=O)NC8=O)C=C7CC[C@@H]6C4)C5)C=C3)C2(C)C)=CC=C1C#N	C48H58FN7O4	AR	P10275	CRBN	WO-2025036489-A1
TPD-4NVF09	WO2025036489A1_46	.	CC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC5(CC4)CC(CN4CCN6C7=CC(F)=C(C(=O)N[C@H]8CCC(=O)NC8=O)C=C7CC[C@@H]6C4)C5)C=C3)C2(C)C)=CC=C1C#N	C50H60FN7O5	AR	P10275	CRBN	WO-2025036489-A1
TPD-4V81E3	WO2025036489A1_47	.	CC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC5(CC4)CC(CN4CCN6C7=CC(F)=C(C(=O)N[C@H]8CCC(=O)NC8=O)C=C7CC[C@H]6C4)C5)C=C3)C2(C)C)=CC=C1C#N	C50H60FN7O5	AR	P10275	CRBN	WO-2025036489-A1
TPD-BAHA33	WO2025036489A1_48	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(CN4CCN5C6=CC(F)=C(C7CCC(=O)NC7=O)C=C6CC[C@@H]5C4)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C45H52ClFN6O4	AR	P10275	CRBN	WO-2025036489-A1
TPD-R5D4ZR	WO2025036489A1_49	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(CN4CCN5C6=CC(F)=C(C7CCC(=O)NC7=O)C=C6CC[C@H]5C4)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C45H52ClFN6O4	AR	P10275	CRBN	WO-2025036489-A1
TPD-LIHJFM	WO2025036489A1_5	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC5(CC4)CC(CN4CCN6C7=C(C=C(C(=O)N[C@H]8CCC(=O)NC8=O)C(F)=C7)CC[C@@H]6C4)C5)C=C3)C2(C)C)=CC=C1C#N	C50H60FN7O6	AR	P10275	CRBN	WO-2025036489-A1
TPD-NSK7M3	WO2025036489A1_50	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(CN4CCN5C6=CC(F)=C(N7CCC(=O)NC7=O)C=C6CC[C@@H]5C4)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C44H51ClFN7O4	AR	P10275	CRBN	WO-2025036489-A1
TPD-POTQAB	WO2025036489A1_51	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(CN4CCN5C6=CC(F)=C(N7CCC(=O)NC7=O)C=C6CC[C@H]5C4)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C44H51ClFN7O4	AR	P10275	CRBN	WO-2025036489-A1
TPD-H10PXO	WO2025036489A1_52	.	C=C(N[C@H]1CCC(=O)NC1=O)C1=C(F)C=C2C(=C1)CC[C@@H]1CN(CC3CCN(C4=CC=C(C(=O)N[C@H]5C(C)(C)[C@H](OC6=CC=C(C#N)C(Cl)=C6)C5(C)C)C=C4)CC3)CCN21	C47H55ClFN7O4	AR	P10275	CRBN	WO-2025036489-A1
TPD-3NBYNT	WO2025036489A1_53	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(CN4CCN5C6=CC(F)=C(C(=O)N[C@H]7CCC(=O)NC7=O)C=C6CC[C@H]5C4)CC3)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C46H53ClFN7O5	AR	P10275	CRBN	WO-2025036489-A1
TPD-B6H0WV	WO2025036489A1_54	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC4(CC3)CC(CN3CCN5C6=CC(F)=C(C7CCC(=O)NC7=O)C=C6CC[C@@H]5C3)C4)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C48H56ClFN6O4	AR	P10275	CRBN	WO-2025036489-A1
TPD-EQBZ25	WO2025036489A1_55	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC4(CC3)CC(CN3CCN5C6=CC(F)=C(C7CCC(=O)NC7=O)C=C6CC[C@H]5C3)C4)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C48H56ClFN6O4	AR	P10275	CRBN	WO-2025036489-A1
TPD-Z0ZA28	WO2025036489A1_56	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC4(CC3)CC(CN3CCN5C6=CC(F)=C(N7CCC(=O)NC7=O)C=C6CC[C@@H]5C3)C4)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C47H55ClFN7O4	AR	P10275	CRBN	WO-2025036489-A1
TPD-XTJS3H	WO2025036489A1_57	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC4(CC3)CC(CN3CCN5C6=CC(F)=C(N7CCC(=O)NC7=O)C=C6CC[C@H]5C3)C4)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C47H55ClFN7O4	AR	P10275	CRBN	WO-2025036489-A1
TPD-Y96D4F	WO2025036489A1_58	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC4(CC3)CC(CN3CCN5C6=CC(F)=C(C(=O)N[C@H]7CCC(=O)NC7=O)C=C6CC[C@@H]5C3)C4)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C49H57ClFN7O5	AR	P10275	CRBN	WO-2025036489-A1
TPD-5Q239B	WO2025036489A1_59	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC4(CC3)CC(CN3CCN5C6=CC(F)=C(C(=O)N[C@H]7CCC(=O)NC7=O)C=C6CC[C@H]5C3)C4)C=C2)C(C)(C)[C@H]1OC1=CC=C(C#N)C(Cl)=C1	C49H57ClFN7O5	AR	P10275	CRBN	WO-2025036489-A1
TPD-J7OYJV	WO2025036489A1_6	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC5(CC4)CC(CN4CCN6C7=C(C=C(C(=O)N[C@@H]8CCC(=O)NC8=O)C(F)=C7)CC[C@@H]6C4)C5)C=C3)C2(C)C)=CC=C1C#N	C50H60FN7O6	AR	P10275	CRBN	WO-2025036489-A1
TPD-FOTXTV	WO2025036489A1_60	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(CN5CCN6C7=CC(F)=C(C8CCC(=O)NC8=O)C=C7CC[C@@H]6C5)CC4)N=N3)C2(C)C)=CC=C1C#N	C44H53FN8O5	AR	P10275	CRBN	WO-2025036489-A1
TPD-P4YHC5	WO2025036489A1_61	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(CN5CCN6C7=CC(F)=C(C8CCC(=O)NC8=O)C=C7CC[C@H]6C5)CC4)N=N3)C2(C)C)=CC=C1C#N	C44H53FN8O5	AR	P10275	CRBN	WO-2025036489-A1
TPD-1LFZFN	WO2025036489A1_62	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(CN5CCN6C7=CC(F)=C(N8CCC(=O)NC8=O)C=C7CC[C@@H]6C5)CC4)N=N3)C2(C)C)=CC=C1C#N	C43H52FN9O5	AR	P10275	CRBN	WO-2025036489-A1
TPD-PSDE4Y	WO2025036489A1_63	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(CN5CCN6C7=CC(F)=C(N8CCC(=O)NC8=O)C=C7CC[C@H]6C5)CC4)N=N3)C2(C)C)=CC=C1C#N	C43H52FN9O5	AR	P10275	CRBN	WO-2025036489-A1
TPD-3OOYP6	WO2025036489A1_64	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(CN5CCN6C7=CC(F)=C(C8CCC(=O)NC8=O)C=C7CC[C@@H]6C5)CC4)N=C3)C2(C)C)=CC=C1C#N	C45H54FN7O5	AR	P10275	CRBN	WO-2025036489-A1
TPD-TKI65X	WO2025036489A1_65	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(CN5CCN6C7=CC(F)=C(C8CCC(=O)NC8=O)C=C7CC[C@H]6C5)CC4)N=C3)C2(C)C)=CC=C1C#N	C45H54FN7O5	AR	P10275	CRBN	WO-2025036489-A1
TPD-WD894G	WO2025036489A1_66	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(CN5CCN6C7=CC(F)=C(N8CCC(=O)NC8=O)C=C7CC[C@@H]6C5)CC4)N=C3)C2(C)C)=CC=C1C#N	C44H53FN8O5	AR	P10275	CRBN	WO-2025036489-A1
TPD-DBFRMB	WO2025036489A1_67	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(CN5CCN6C7=CC(F)=C(N8CCC(=O)NC8=O)C=C7CC[C@H]6C5)CC4)N=C3)C2(C)C)=CC=C1C#N	C44H53FN8O5	AR	P10275	CRBN	WO-2025036489-A1
TPD-VZZVST	WO2025036489A1_68	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(CN5CCN6C7=CC(F)=C(C(=O)N[C@H]8CCC(=O)NC8=O)C=C7CC[C@@H]6C5)CC4)N=C3)C2(C)C)=CC=C1C#N	C46H55FN8O6	AR	P10275	CRBN	WO-2025036489-A1
TPD-KXK9LN	WO2025036489A1_69	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(CN5CCN6C7=CC(F)=C(C(=O)N[C@H]8CCC(=O)NC8=O)C=C7CC[C@H]6C5)CC4)N=C3)C2(C)C)=CC=C1C#N	C46H55FN8O6	AR	P10275	CRBN	WO-2025036489-A1
TPD-WC79RA	WO2025036489A1_7	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC5(CC4)CC(CN4CCN6C(=CCC7=C6C=C(F)C(C(=O)N[C@H]6CCC(=O)NC6=O)=C7)C4)C5)C=C3)C2(C)C)=CC=C1C#N	C50H58FN7O6	AR	P10275	CRBN	WO-2025036489-A1
TPD-9PS3S5	WO2025036489A1_70	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(CN5CCN6C7=CC(F)=C(C(=O)N[C@H]8CCC(=O)NC8=O)C=C7CC[C@@H]6C5)CC4)NN3)C2(C)C)=CC=C1C#N	C45H56FN9O6	AR	P10275	CRBN	WO-2025036489-A1
TPD-70CI4X	WO2025036489A1_71	.	COC1=CC(OC2C(C)(C)C(NC(=O)C3=CC=C(N4CCC(CN5CCN6C7=CC(F)=C(C(=O)N[C@H]8CCC(=O)NC8=O)C=C7CC[C@H]6C5)CC4)N=N3)C2(C)C)=CC=C1C#N	C45H54FN9O6	AR	P10275	CRBN	WO-2025036489-A1
TPD-FUX6YR	WO2025036489A1_72	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC4(CC3)CC(CN3CCN5C6=C(C=C(C7CCC(=O)NC7=O)C(F)=C6)CC[C@@H]5C3)C4)C=C2)C(C)(C)[C@H]1OC1=C2C=CC=NC2=C(C#N)C=C1	C51H58FN7O4	AR	P10275	CRBN	WO-2025036489-A1
TPD-TX1PCP	WO2025036489A1_73	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC4(CC3)CC(CN3CCN5C6=C(C=C(C7CCC(=O)NC7=O)C(F)=C6)CC[C@H]5C3)C4)C=C2)C(C)(C)[C@H]1OC1=C2C=CC=NC2=C(C#N)C=C1	C51H58FN7O4	AR	P10275	CRBN	WO-2025036489-A1
TPD-SKQJY2	WO2025036489A1_74	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC4(CC3)CC(CN3CCN5C6=C(C=C(N7CCC(=O)NC7=O)C(F)=C6)CC[C@H]5C3)C4)C=C2)C(C)(C)[C@H]1OC1=C2C=CC=NC2=C(C#N)C=C1	C50H57FN8O4	AR	P10275	CRBN	WO-2025036489-A1
TPD-BZ806X	WO2025036489A1_75	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC4(CC3)CC(CN3CCN5C6=C(C=C(N7CCC(=O)NC7=O)C(F)=C6)CC[C@@H]5C3)C4)C=C2)C(C)(C)[C@H]1OC1=C2C=CC=NC2=C(C#N)C=C1	C50H57FN8O4	AR	P10275	CRBN	WO-2025036489-A1
TPD-0HIV64	WO2025036489A1_76	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC4(CC3)CC(CN3CCN5C6=C(C=C(C(=O)N[C@H]7CCC(=O)NC7=O)C(F)=C6)CC[C@H]5C3)C4)C=C2)C(C)(C)[C@H]1OC1=C2C=CC=NC2=C(C#N)C=C1	C52H59FN8O5	AR	P10275	CRBN	WO-2025036489-A1
TPD-WUDZNY	WO2025036489A1_77	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC4(CC3)CC(CN3CCN5C6=C(C=C(C(=O)N[C@H]7CCC(=O)NC7=O)C(F)=C6)CC[C@@H]5C3)C4)C=C2)C(C)(C)[C@H]1OC1=C2C=CC=NC2=C(C#N)C=C1	C52H59FN8O5	AR	P10275	CRBN	WO-2025036489-A1
TPD-T5HEF8	WO2025036489A1_78	.	CC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(CN5CCN6C7=C(C=C(C8CCC(=O)NC8=O)C(F)=C7)CC[C@H]6C5)CC4)C=C3)C2(C)C)=CC(C)=C1C#N	C47H57FN6O4	AR	P10275	CRBN	WO-2025036489-A1
TPD-1WP8WA	WO2025036489A1_79	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC5(CC4)CC(N4CCN6C7=CC(F)=C(N8CCC(=O)NC8=O)C=C7CC[C@@H]6C4)C5)C=C3)C2(C)C)=CC=C1C#N	C47H56FN7O5	AR	P10275	CRBN	WO-2025036489-A1
TPD-SLRK4L	WO2025036489A1_8	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC5(CC4)CC(CN4CCN6C7=C(C=C(C(=O)N[C@H]8CCC(=O)NC8=O)C(F)=C7)CC[C@H]6C4)C5)C=C3)C2(C)C)=CC=C1C#N	C50H60FN7O6	AR	P10275	CRBN	WO-2025036489-A1
TPD-KECYUE	WO2025036489A1_80	.	CC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(CN5CCN6C7=C(C=C(N8CCC(=O)NC8=O)C(F)=C7)CC[C@H]6C5)CC4)C=C3)C2(C)C)=CC(C)=C1C#N	C46H56FN7O4	AR	P10275	CRBN	WO-2025036489-A1
TPD-O5Z0SX	WO2025036489A1_81	.	CC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(CN5CCN6C7=C(C=C(C8CCC(=O)NC8=O)C(F)=C7)CC[C@@H]6C5)CC4)C=C3)C2(C)C)=CC(C)=C1C#N	C47H57FN6O4	AR	P10275	CRBN	WO-2025036489-A1
TPD-Q55LV5	WO2025036489A1_82	.	CC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(CN5CCN6C7=C(C=C(N8CCC(=O)NC8=O)C(F)=C7)CC[C@@H]6C5)CC4)C=C3)C2(C)C)=CC(C)=C1C#N	C46H56FN7O4	AR	P10275	CRBN	WO-2025036489-A1
TPD-FN5NM8	WO2025036489A1_83	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(CN5CCN6C7=C(C=C(C8CCC(=O)NC8=O)C=N7)CC[C@H]6C5)CC4)C=C3)C2(C)C)=CC=C1C#N	C45H55N7O5	AR	P10275	CRBN	WO-2025036489-A1
TPD-RG7QIF	WO2025036489A1_84	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC5(CC4)CC(N4CCN6C7=CC(F)=C(N8CCC(=O)NC8=O)C=C7CCC6C4)C5)C=C3)C2(C)C)=CC=C1C#N	C47H56FN7O5	AR	P10275	CRBN	WO-2025036489-A1
TPD-3U8I52	WO2025036489A1_85	.	CC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(CN5CCN6C7=CC(F)=C(C8CCC(=O)NC8=O)C=C7CC[C@@H]6C5)CC4)N=N3)C2(C)C)=CC=C1C#N	C44H53FN8O4	AR	P10275	CRBN	WO-2025036489-A1
TPD-A6LRMB	WO2025036489A1_86	.	CC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(CN5CCN6C7=CC(F)=C(C8CCC(=O)NC8=O)C=C7CC[C@H]6C5)CC4)N=N3)C2(C)C)=CC=C1C#N	C44H53FN8O4	AR	P10275	CRBN	WO-2025036489-A1
TPD-GC8QPD	WO2025036489A1_87	.	CC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(CN5CCN6C7=CC(F)=C(C(=O)N[C@H]8CCC(=O)NC8=O)C=C7CC[C@@H]6C5)CC4)N=N3)C2(C)C)=CC=C1C#N	C45H54FN9O5	AR	P10275	CRBN	WO-2025036489-A1
TPD-N31SZZ	WO2025036489A1_88	.	CC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(CN5CCN6C7=CC(F)=C(C(=O)N[C@H]8CCC(=O)NC8=O)C=C7CC[C@H]6C5)CC4)N=N3)C2(C)C)=CC=C1C#N	C45H54FN9O5	AR	P10275	CRBN	WO-2025036489-A1
TPD-YGURGN	WO2025036489A1_89	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(CN4CCN5C6=CC(F)=C(C7CCC(=O)NC7=O)C=C6CC[C@@H]5C4)CC3)N=N2)C(C)(C)[C@H]1OC1=C2C=CC=NC2=C(C#N)C=C1	C46H52FN9O4	AR	P10275	CRBN	WO-2025036489-A1
TPD-XOSPGY	WO2025036489A1_9	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC5(CC4)CC(CN4CCN6C7=C(C=C(C8CCC(=O)NC8=O)C(F)=C7)CC[C@@H]6C4)C5)C=C3)C2(C)C)=CC=C1C#N	C49H59FN6O5	AR	P10275	CRBN	WO-2025036489-A1
TPD-7CYM2T	WO2025036489A1_90	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(CN4CCN5C6=CC(F)=C(C7CCC(=O)NC7=O)C=C6CC[C@H]5C4)CC3)N=C2)C(C)(C)[C@H]1OC1=C2C=CC=NC2=C(C#N)C=C1	C47H53FN8O4	AR	P10275	CRBN	WO-2025036489-A1
TPD-XHAO3U	WO2025036489A1_91	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(CN4CCN5C6=CC(F)=C(C(=O)N[C@H]7CCC(=O)NC7=O)C=C6CC[C@@H]5C4)CC3)N=N2)C(C)(C)[C@H]1OC1=C2C=CC=NC2=C(C#N)C=C1	C47H53FN10O5	AR	P10275	CRBN	WO-2025036489-A1
TPD-SC6BL6	WO2025036489A1_92	.	CC1(C)[C@H](NC(=O)C2=CC=C(N3CCC(CN4CCN5C6=CC(F)=C(C(=O)N[C@H]7CCC(=O)NC7=O)C=C6CC[C@H]5C4)CC3)N=N2)C(C)(C)[C@H]1OC1=C2C=CC=NC2=C(C#N)C=C1	C47H53FN10O5	AR	P10275	CRBN	WO-2025036489-A1
TPD-KJ2210	WO2025036489A1_93	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(CN5CCN6C7=C(C=C(C8CCC(=O)NC8=O)C=N7)CC[C@@H]6C5)CC4)C=C3)C2(C)C)=CC=C1C#N	C45H55N7O5	AR	P10275	CRBN	WO-2025036489-A1
TPD-GX4M67	WO2025036489A1_94	.	CC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC5(CC4)CC(N4CCN6C7=CC(F)=C(N8CCC(=O)NC8=O)C=C7CC[C@@H]6C4)C5)C=C3)C2(C)C)=CC=C1C#N	C47H56FN7O4	AR	P10275	CRBN	WO-2025036489-A1
TPD-JZVPJ4	WO2025036489A1_95	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC5(CC4)CC(N4CCN6C(=NC7=C6C=C(F)C(C6CCC(=O)NC6=O)=C7)C4)C5)C=C3)C2(C)C)=CC=C1C#N	C46H52FN7O5	AR	P10275	CRBN	WO-2025036489-A1
TPD-0V0PKJ	WO2025036489A1_96	.	COC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(CN5CCN6C(=NC7=C6C=C(F)C(C6CCC(=O)NC6=O)=C7)C5)CC4)C=C3)C2(C)C)=CC=C1C#N	C44H50FN7O5	AR	P10275	CRBN	WO-2025036489-A1
TPD-HE45SC	WO2025036489A1_97	.	CC#CCOC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(CN5CCN6C7=CC(F)=C(C8CCC(=O)NC8=O)C=C7CC[C@H]6C5)CC4)C=C3)C2(C)C)=CC=C1C#N	C49H57FN6O5	AR	P10275	CRBN	WO-2025036489-A1
TPD-1QGBTG	WO2025036489A1_98	.	CC#CCOC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(CN5CCN6C7=CC(F)=C(C8CCC(=O)NC8=O)C=C7CC[C@@H]6C5)CC4)C=C3)C2(C)C)=CC=C1C#N	C49H57FN6O5	AR	P10275	CRBN	WO-2025036489-A1
TPD-LVS4IN	WO2025036489A1_99	.	CC#CCOC1=CC(O[C@H]2C(C)(C)[C@H](NC(=O)C3=CC=C(N4CCC(CN5CCN6C7=CC(F)=C(C(=O)N[C@H]8CCC(=O)NC8=O)C=C7CC[C@@H]6C5)CC4)C=C3)C2(C)C)=CC=C1C#N	C50H58FN7O6	AR	P10275	CRBN	WO-2025036489-A1
TPD ID	TPD Name	PubChem synonyms	SMILES	Formula	Target	Target ID	Ligase	Source
TPD-04W1C4	AU2011272860A1_1	.	C=C(CC)C(=O)C1=CC=C(OCC(=O)NCCCCCCCC(=O)C(CCCN/C(=N/C(=O)OC(C)(C)C)NC(=O)OC(C)(C)C)NC(=O)OC(C)(C)C)C(Cl)=C1Cl	C41H63Cl2N5O10	eDHFR-KRas;IMPDH	P00374/A0A384N6C2	.	AU2011272860A1
TPD-05Q017	SCHEMBL254271	SCHEMBL254271; SCHEMBL15122458; SCHEMBL19362578	COC1=CC(CC2=CN=C(N)N=C2N)=CC(OC)=C1OCC(=O)NCCCCCCNC(=O)C(CCCN/C(=N/C(=O)OC(C)(C)C)NC(=O)OC(C)(C)C)NC(=O)OC(C)(C)C	C42H68N10O11	eDHFR-KRas;IMPDH	P00374/A0A384N6C2	.	AU2011272860A1
TPD-0A13QN	CN-110642849-B_1	.	[H][C@@]12CC[C@]3(CC=C(C(=O)OC)CC[C@@]31OC(C)=O)C(=O)O[C@]2(C)/C=C/C=C(\C)C(=O)OCOC1=C2C(=O)N(C3CCC(=O)NC3=O)C(=O)C2=CC=C1	C37H38N2O13	CD147	P35613	CRBN	CN-110642849-B
TPD-0F6692	CN-110642849-B_2	.	[H][C@@]12CC[C@]3(CC=C(C(=O)OC)CC[C@@]31OC(C)=O)C(=O)O[C@]2(C)/C=C/C=C(\C)C(=O)OCCCOC1=C2C(=O)N(C3CCC(=O)NC3=O)C(=O)C2=CC=C1	C39H42N2O13	CD147	P35613	CRBN	CN-110642849-B
TPD-0F7MF4	CN-110642849-B_3	.	[H][C@@]12CC[C@]3(CC=C(C(=O)OC)CC[C@@]31OC(C)=O)C(=O)O[C@]2(C)/C=C/C=C(\C)C(=O)OCCCCCOC1=C2C(=O)N(C3CCC(=O)NC3=O)C(=O)C2=CC=C1	C41H46N2O13	CD147	P35613	CRBN	CN-110642849-B
TPD-0K8ZRR	CN-110642849-B_4	.	[H][C@@]12CC[C@]3(CC=C(C(=O)OC)CC[C@@]31OC(C)=O)C(=O)O[C@]2(C)/C=C/C=C(\C)C(=O)OCCCCCCCOC1=C2C(=O)N(C3CCC(=O)NC3=O)C(=O)C2=CC=C1	C43H50N2O13	CD147	P35613	CRBN	CN-110642849-B
TPD-0PGK2O	CN-115043831-A_P30	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCOC3=CC=CC=C3C3=CSC(C4=CSC(NC5=CC=C(Cl)C=C5)=N4)=N3)C(C)(C)C)C=C2)SC=N1	C47H52ClN7O5S3	CYP1B1	Q16678	VHL	CN-115043831-A
TPD-0RP7MW	CN-115043831-A_P31	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCOC3=CC=CC=C3C3=CSC(C4=CSC(NC5=CC=C(Cl)C=C5)=N4)=N3)C(C)(C)C)C=C2)SC=N1	C48H54ClN7O5S3	CYP1B1	Q16678	VHL	CN-115043831-A
TPD-11DXZN	PROTAC CYP1B1 degrader-2	PROTAC CYP1B1 degrader-2; 2836297-26-6; orb2646303; HY-158429; CS-1054653	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCOC3=CC=CC=C3C3=CSC(C4=CSC(NC5=CC=C(Cl)C=C5)=N4)=N3)C(C)(C)C)C=C2)SC=N1	C49H56ClN7O5S3	CYP1B1	Q16678	VHL	CN-115043831-A
TPD-11IE8F	SCHEMBL28962487	SCHEMBL28962487	COC1=NC(CCCNC(=O)CN/C2=C/C=C\C3=C2CN(C2CCC(=O)NC2=O)C3=O)=CN=C1NS(=O)(=O)C1=CC=C(NC(=O)/C=C/C2=CC=C([N+](=O)[O-])S2)C=C1	C36H35N9O10S2	MLKL	Q8NB16	CRBN	CN-115745979-A
TPD-12FMJ8	SCHEMBL28962475	SCHEMBL28962475	COC1=NC(CCCNC(=O)CCN/C2=C/C=C\C3=C2CN(C2CCC(=O)NC2=O)C3=O)=CN=C1NS(=O)(=O)C1=CC=C(NC(=O)/C=C/C2=CC=C([N+](=O)[O-])S2)C=C1	C37H37N9O10S2	MLKL	Q8NB16	CRBN	CN-115745979-A
TPD-12LY7I	SCHEMBL28962541	SCHEMBL28962541	COC1=NC(CCCNC(=O)CCCN/C2=C/C=C\C3=C2CN(C2CCC(=O)NC2=O)C3=O)=CN=C1NS(=O)(=O)C1=CC=C(NC(=O)/C=C/C2=CC=C([N+](=O)[O-])S2)C=C1	C38H39N9O10S2	MLKL	Q8NB16	CRBN	CN-115745979-A
TPD-14EHSV	CN-116640123-A_4H3PM	.	COC1=CC=C(C2=NC(C3=CC=C(Cl)C=C3)C(C3=CC=C(Cl)C=C3)N2C(=O)N2CCN(CC(=O)NCCOCCOCCOCCN3C=C(COC4=CC(C(=O)N/N=C/C5=CC=C(O)C(O)=C5O)=CC=C4[N+](=O)[O-])N=N3)C(=O)C2)C(OC(C)C)=C1	C57H61Cl2N11O15	HK2	P52789	MDM2	CN-116640123-A
TPD-1B89ZY	CN-116640123-A_4H5PM	.	COC1=CC=C(C2=NC(C3=CC=C(Cl)C=C3)C(C3=CC=C(Cl)C=C3)N2C(=O)N2CCN(CC(=O)NCCOCCOCCOCCOCCOCCN3C=C(COC4=CC(C(=O)N/N=C\C5=CC=C(O)C(O)=C5O)=CC=C4[N+](=O)[O-])N=N3)C(=O)C2)C(OC(C)C)=C1	C61H69Cl2N11O17	HK2	P52789	MDM2	CN-116640123-A
TPD-1BVLMW	CN-117486875-A_93	.	[H][C@]12C[C@](O)(CC3=CN(CCC(=O)NC4=C5\C(=O)N(C6CCC(=O)NC6=O)C(=O)\C5=C/C=C\4)N=N3)C[C@H](C)N1CCC1=C/C(OCC3=CC(C)=CC(C)=C3)=C(OCC3=CC(C)=CC(C)=C3)\C=C\12	C51H55N7O8	GDI2	P50395	CRBN	CN-117486875-A
TPD-1C3NR8	CN-117486875-A_94	.	[H][C@]12C[C@](O)(CC3=CN(CCCCCCCCCCC(=O)NC4=C5\C(=O)N(C6CCC(=O)NC6=O)C(=O)\C5=C/C=C\4)N=N3)C[C@H](C)N1CCC1=CC(OCC3=CC(C)=CC(C)=C3)=C(OCC3=CC(C)=CC(C)=C3)C=C12	C59H71N7O8	GDI2	P50395	CRBN	CN-117486875-A
TPD-1G5REP	CN-117486875-A_95	.	[H][C@]12C[C@](O)(CC3=CN(CCOCCOCCOCCOCC(=O)NC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)N=N3)C[C@H](C)N1CCC1=CC(OCC3=CC(C)=CC(C)=C3)=C(OCC3=CC(C)=CC(C)=C3)C=C12	C58H69N7O12	GDI2	P50395	CRBN	CN-117486875-A
TPD-1GGOKB	CN109422753B_10	.	N#CCC1(N2C=C(C3=C4C=CNC4=NC=N3)C=N2)CN(C(=O)COCCOCCNC2=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=CC=C2)C1	C33H32N10O7	JAK1;JAK2	P23458/O60674	CRBN	CN109422753B
TPD-1N1KXE	CN109422753B_13	.	N#CCC1(N2C=C(C3=C4C=CNC4=NC=N3)C=N2)CN(S(=O)(=O)CCCCCO/C2=C/C=C\C3=C2C(=O)N(C2CCC(=O)NC2=O)C3=O)C1	C32H31N9O7S	JAK1;JAK2	P23458/O60674	CRBN	CN109422753B
TPD-1ON5W5	CN109422753B_14	.	N#CCC1(N2C=C(C3=C4C=CNC4=NC=N3)C=N2)CN(CCOCCOCCOCCNC2=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=CC=C2)C1	C35H38N10O7	JAK1;JAK2	P23458/O60674	CRBN	CN109422753B
TPD-1Q6GFB	CN109422753B_15	.	N#CCC1(N2C=C(C3=C4C=CNC4=NC=N3)C=N2)CN(CCOCCOCCOCCOC2=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=CC=C2)C1	C35H37N9O8	JAK1;JAK2	P23458/O60674	CRBN	CN109422753B
TPD-1UHJGA	CN109422753B_3	.	N#CCC1(N2C=C(C3=C4C=CNC4=NC=N3)C=N2)CN(CCCCCC(=O)NC2=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=CC=C2)C1	C33H32N10O5	JAK1;JAK2	P23458/O60674	CRBN	CN109422753B
TPD-1VJ9RL	CN109422753B_7	.	N#CCC1(N2C=C(C3=C4C=CNC4=NC=N3)C=N2)CN(CCOCCOCCOC2=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=CC=C2)C1	C33H33N9O7	JAK1;JAK2	P23458/O60674	CRBN	CN109422753B
TPD-1Y03CR	PROTAC BRD9 Degrader-1	PROTAC BRD9 Degrader-1; 2097971-01-0; N-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyacetyl]amino]butyl]-2-[4-[2-[N'-(1,1-dioxothian-4-yl)carbamimidoyl]-5-methyl-4-oxothieno[3,2-c]pyridin-7-yl]-2-methoxyphenoxy]acetamide; orb1708798; CHEMBL5199808; SCHEMBL21259422; SCHEMBL29881137; C42H45N7O12S2; BCP30517; EX-A3889; XID97101; AKOS037653394; DA-77136; PD102755; HY-103632; CS-0028482; G16554; EN300-22942797; (Z)-2-(4-(2-(N'-(1,1-dioxidotetrahydro-2H-thiopyran-4-yl)carbamimidoyl)-5-methyl-4-oxo-4,5-dihydrothieno[3,2-c]pyridin-7-yl)-2-methoxyphenoxy)-N-(4-(2-((2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindolin-4-yl)oxy)acetamido)butyl)acetamide; 2-(4-{2-[N-(1,1-dioxo-1lambda6-thian-4-yl)carbamimidoyl]-5-methyl-4-oxo-4H,5H-thieno[3,2-c]pyridin-7-yl}-2-methoxyphenoxy)-N-[4-(2-{[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]oxy}acetamido)butyl]acetamide; N-[4-[[2-[2-(2,6-dioxo-3-piperidyl)-1,3-dioxo-isoindolin-4-yl]oxyacetyl]amino]butyl]-2-[4-[2-[N'-(1,1-dioxothian-4-yl)carbamimidoyl]-5-methyl-4-oxo-thieno[3,2-c]pyridin-7-yl]-2-methoxy-phenoxy]acetamide	COC1=CC(/C2=C/N(C)C(=O)C3=C2SC(C(=N)NC2CCS(=O)(=O)CC2)=C3)=CC=C1OCC(=O)NCCCCNC(=O)CO/C1=C/C=C\C2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O	C42H45N7O12S2	BRD9	Q9H8M2	CRBN	US-11285218-B2
TPD-1Y80PI	SCHEMBL21259469	SCHEMBL21259469; PD141263	COC1=CC(C2=CN(C)C(=O)C3=C2SC(C(=N)NC2CCS(=O)(=O)CC2)=C3)=CC=C1OCC(=O)NCCCCCCCCNC(=O)CO/C1=C/C=C\C2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O	C46H53N7O12S2	BRD9	Q9H8M2	CRBN	US-11285218-B2
TPD-222HXX	SCHEMBL21259388	SCHEMBL21259388; PD141262	COC1=CC(C2=CN(C)C(=O)C3=C2SC(C(=N)NC2CCS(=O)(=O)CC2)=C3)=CC=C1OCC(=O)NCCCOCCOCCOCCCNC(=O)CO/C1=C/C=C\C2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O	C48H57N7O15S2	BRD9	Q9H8M2	CRBN	US-11285218-B2
TPD-22GCC8	SCHEMBL24764858	SCHEMBL24764858	CCCCNC1=NC2=C(C=N1)/C(C1=CC=C(CN3CCN(CCOCCOCCOCCOCCN/C4=C/C=C\C5=C4N(C)C(=O)N5C4CCC(=O)NC4=O)CC3)C=C1)=C\N2[C@H]1CC[C@H](O)CC1	C50H70N10O8	MerTK;TYRO3	Q12866/Q06418	CRBN	US-2022356185-A1
TPD-2DLEU2	SCHEMBL24764500	SCHEMBL24764500	CCCCNC1=NC2=C(C=N1)C(C1=CC=C(CN3CCN(CCOCCOCCOCCOCCCC4=C/C5=C(\C=C/4)N(C4CCC(=O)NC4=O)C(=O)N5C)CC3)C=C1)=NN2[C@H]1CC[C@H](O)CC1	C50H70N10O8	MerTK;TYRO3	Q12866/Q06418	CRBN	US-2022356185-A1
TPD-2FOQWN	SCHEMBL24764650	SCHEMBL24764650; SCHEMBL30042131	CCCCNC1=NC2=C(C=N1)/C(C1=CC=C(CN3CCN(CCOCCOCCOCCCC4=C/C5=C(\C=C/4)N(C4CCC(=O)NC4=O)C(=O)N5C)CC3)C=C1)=C\N2[C@H]1CC[C@H](O)CC1	C49H67N9O7	MerTK;TYRO3	Q12866/Q06418	CRBN	US-2022356185-A1
TPD-2GTCYU	SCHEMBL23866825	SCHEMBL23866825; SCHEMBL30462110	CCN1CC[C@H]2CC[C@@H](C(=O)N[C@@H](CCS(N)(=O)=O)C(=O)N[C@@H](CC3=CC=C(C(C)(C)C)C=C3)C(=O)N3CCC(CCC#C/C4=C/C=C\C5=C4CN(C4CCC(=O)NC4=O)C5=O)CC3)N2C(=O)[C@@H](NC(=O)C2=CC3=C(/C=C\C(C(F)(F)P(=O)(O)O)=C/3)S2)C1	C61H74F2N9O13PS2	STAT3	P40763	CRBN	US-2023159573-A1
TPD-2HBB74	SCHEMBL25209445	SCHEMBL25209445; SCHEMBL25266621	CCN1CC[C@H]2CC[C@@H](C(=O)N[C@@H](CCN3C=CN=C3[N+](=O)[O-])C(=O)N[C@@H](CC3=CC=C(C(C)(C)C)C=C3)C(=O)N3CCC(CCC#CC4=CC=CC5=C4CN(C4CCC(=O)NC4=O)C5=O)CC3)N2C(=O)[C@@H](NC(=O)/C2=C/C3=C(C=CC(C(F)(F)P(=O)(O)O)=C3)S2)C1	C64H74F2N11O13PS	STAT3	P40763	CRBN	US-2023159573-A1
TPD-2MSKM0	US-2023159573-A1_22	.	CCN1CC[C@H]2CC[C@@H](C(=O)N[C@@H](CCN3C=CN=C3N)C(=O)N[C@@H](CC3=CC=C(C(C)(C)C)C=C3)C(=O)N3CCC(CCC#CC4=CC=CC5=C4CN(C4CCC(=O)NC4=O)C5=O)CC3)N2C(=O)[C@@H](NC(=O)/C2=C/C3=C(C=CC(C(F)(F)P(=O)(O)O)=C3)S2)C1	C64H76F2N11O11PS	STAT3	P40763	CRBN	US-2023159573-A1
TPD-2OZGKM	US-2023257380-A1_TR-029	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCC(=O)N3CCN(C4=NC(/C5=C/N=C6/C=CC(N7CCCC7C7=CC=CC(F)=C7)=NN56)=CC=C4)CC3)C(C)(C)C)C=C2)SC=N1	C55H66FN11O5S	TRKA;TRKB;TRKC	P04629/Q16620/Q16288	VHL	US-2023257380-A1
TPD-2P0YAN	SCHEMBL22463980	SCHEMBL22463980; SCHEMBL30502226	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCC(=O)N3CCN(C4=CC=C(C(=O)N/C5=N/NC6=C5C=C(CC5=CC(F)=CC(F)=C5)C=C6)C(NC5CCOCC5)=C4)CC3)C(C)(C)C)C=C2)SC=N1	C60H72F2N10O7S	TRKA;TRKB;TRKC	P04629/Q16620/Q16288	VHL	US-2023257380-A1
TPD-2TE3Q0	SCHEMBL21759414	SCHEMBL21759414	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCCCC(=O)N3CCN(C4=CC=C(C(=O)N/C5=N/NC6=C5C=C(CC5=CC(F)=CC(F)=C5)C=C6)C(NC5CCOCC5)=C4)CC3)C(C)(C)C)C=C2)SC=N1	C63H78F2N10O7S	TRKA;TRKB;TRKC	P04629/Q16620/Q16288	VHL	US-2023257380-A1
TPD-2TU5WT	CHEMBL5424239	CHEMBL5424239; SCHEMBL25396162; SCHEMBL30617666; PD216026	CC(C)(C)[C@H](NC(=O)/C1=C/C2=C(C=CC(C(F)(F)P(=O)(O)O)=C2)S1)C(=O)N1CCC[C@H]1C(=O)N(CCC(=O)NCCCCCCC#CC1=C2CN(C3CCC(=O)NC3=O)C(=O)C2=CC=C1)C1=CC=C(Br)C=C1	C51H56BrF2N6O10PS	STAT5	P42229	CRBN	US-2023295197-A1
TPD-2TVZRQ	CHEMBL5407249	CHEMBL5407249; SCHEMBL25396595; SCHEMBL30617618; AK-023; PD216024	CC(C)(C)[C@H](NC(=O)C1=CC2=C(/C=C\C(C(F)(F)P(=O)(O)O)=C/2)S1)C(=O)N1CCC[C@H]1C(=O)N(CCC(=O)NCCCCCC#CC1=C2CN(C3CCC(=O)NC3=O)C(=O)C2=CC=C1)C1=CC=C(Br)C=C1	C50H54BrF2N6O10PS	STAT5	P42229	CRBN	US-2023295197-A1
TPD-2YRAP6	CHEMBL5409467	CHEMBL5409467; SCHEMBL25396995; SCHEMBL30617629; AK-021; PD216020	CC(C)(C)[C@H](NC(=O)/C1=C/C2=C(C=CC(C(F)(F)P(=O)(O)O)=C2)S1)C(=O)N1CCC[C@H]1C(=O)N(CCC(=O)NCCCC#CC1=C2CN(C3CCC(=O)NC3=O)C(=O)C2=CC=C1)C1=CC=C(Br)C=C1	C48H50BrF2N6O10PS	STAT5	P42229	CRBN	US-2023295197-A1
TPD-30GKWT	CPD-1224	CPD-1224; 2891620-68-9; CHEMBL5395301; orb1982284; SCHEMBL31093896; EX-A7859; BDBM50625494; DA-62488; HY-153386; CS-0694733	COC1=C(NC2=NC=C(Cl)C(NC3=C(S(=O)(=O)C(C)C)C=CC=C3)=N2)C=C(C)C(C2CCN(CC3CN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)CC2)=C1	C43H47ClN8O7S	EML4-ALK	Q9HC35	CRBN	US-2024336643-A1
TPD-32O5U4	SCHEMBL24852275	SCHEMBL24852275	COC1=C(NC2=NC=C(Cl)C(NC3=C(S(=O)(=O)C(C)C)C=CC=C3)=N2)C=C(C)C(C2CCN(CCC3CN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)CC2)=C1	C44H49ClN8O7S	EML4-ALK	Q9HC35	CRBN	US-2024336643-A1
TPD-35XMID	US-2024336643-A1_3	.	COC1=C(NC2=NC=C(Cl)C(NC3=C(S(=O)(=O)C(C)C)C=CC=C3)=N2)C=C(C)C(C2CCN(C(=O)CC3CN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)CC2)=C1	C44H47ClN8O8S	EML4-ALK	Q9HC35	CRBN	US-2024336643-A1
TPD-361BJN	CHEMBL5430072	CHEMBL5430072; CPD-1793; BDBM50625493	COC1=C(NC2=NC=C(Cl)C(NC3=C(S(=O)(=O)C(C)C)C=CC=C3)=N2)C=C(C)C(C2CCN(CC3CN(C4=CC5=C(C=C4)C(=O)N(C4CCC(=O)NC4=O)C5)C3)CC2)=C1	C43H49ClN8O6S	EML4-ALK	Q9HC35	CRBN	US-2024336643-A1
TPD-3625EW	SCHEMBL31249504	SCHEMBL31249504; JMF4605; 4-((2-(2-((2-(4-(dimethylamino)phenyl)benzo[d]thiazol-6-yl)oxy)ethoxy)ethyl)amino)-2-(2,6-dioxopiperidin-3-yl)isoindoline-1,3-dione	CN(C)C1=CC=C(C2=NC3=C\C=C(OCCOCCN/C4=C/C=C\C5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)/C=C\3S2)C=C1	C32H31N5O6S	TDP-43	Q13148	CRBN	US-2024400549-A1
TPD-385K5Y	US-2024400549-A1_II-2a	.	[H]N(C)C1=CC=C(/C=C/C2=CN=C(OCCOCCN/C3=C/C=C\C4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)C=C2)C=C1	C31H31N5O6	TDP-43	Q13148	CRBN	US-2024400549-A1
TPD-3A0F62	CHEMBL4515966	CHEMBL4515966; SCHEMBL19475571; PD140856	O=C1CCC(N2C(=O)C3=C\C=C/C(NCCOCCOCCOCCC(=O)N4CCN(C5=CC=C(C6=C/C7=C(\C=C/6)CN(C(C(=O)NC6=NC=CS6)C6=CC=CC=C6)C7=O)C=C5)CC4)=C\3C2=O)C(=O)N1	C51H52N8O10S	EGFR L858R/T790M;EGFR L858R/T790M/C797S	P00533/P00533	CRBN	US10450310B2
TPD-3DQXJ3	SCHEMBL19475574	SCHEMBL19475574; PD140756	O=C1CCC(N2C(=O)C3=C\C=C/C(NCCOCCOCCOCCOCCOCCC(=O)N4CCN(C5=CC=C(C6=CC7=C(C=C6)CN(C(C(=O)NC6=NC=CS6)C6=CC=CC=C6)C7=O)C=C5)CC4)=C\3C2=O)C(=O)N1	C55H60N8O12S	EGFR L858R/T790M;EGFR L858R/T790M/C797S	P00533/P00533	CRBN	US10450310B2
TPD-3I8DKX	SCHEMBL19475629	SCHEMBL19475629	O=C1CCC(N2C(=O)C3=C\C=C/C(NCCOCCOCCOCCC(=O)N4CCN(C5=CC=C(C6=C/C7=C(\C=C/6)CN(C(C(=O)NC6=NC=CS6)C6=CC(F)=CC=C6O)C7=O)C=C5)CC4)=C\3C2=O)C(=O)N1	C51H51FN8O11S	EGFR L858R/T790M;EGFR L858R/T790M/C797S	P00533/P00533	CRBN	US10450310B2
TPD-3KDBRD	SCHEMBL20322437	SCHEMBL20322437	O=C1CCC(N2C(=O)C3=C\C=C/C(OCCN4CCN(CCOC5=CC=C6C=C5COC/C=C/COCC5=CC=CC(=C5)C5=NC(=NC=C5)N6)CC4)=C\3C2=O)C(=O)N1	C43H45N7O8	FLT3-ITD	P36888	CRBN	US10806737B2
TPD-3SP7WJ	SCHEMBL22560492	SCHEMBL22560492	O=C1CCC(N2C(=O)C3=CC=CC(OCCOCCN4CCN(CCOC5=C\C=C6/C=C\5COC/C=C/COCC5=CC=CC(=C5)C5=NC(=NC=C5)N6)CC4)=C3C2=O)C(=O)N1	C45H49N7O9	FLT3-ITD	P36888	CRBN	US10806737B2
TPD-3X1Q5B	SCHEMBL22560491	SCHEMBL22560491	O=C1CCC(N2C(=O)C3=CC=CC(OCCOCCOCCN4CCN(CCOC5=C\C=C6/C=C\5COC/C=C/COCC5=CC=CC(=C5)C5=NC(=NC=C5)N6)CC4)=C3C2=O)C(=O)N1	C47H53N7O10	FLT3-ITD	P36888	CRBN	US10806737B2
TPD-416BO3	SCHEMBL21330773	SCHEMBL21330773	C=CC(=O)NC1=CC=CC=C1NC1=C(Cl)C=NC(NC2=CC(C#CCCNC(=O)OC3CC/C=C/CCC3)=NC=C2)=N1	C31H32ClN7O3	ERK1;ERK2	P27361/P28482	CRBN	US11786600B2
TPD-45FBJT	SCHEMBL19709461	SCHEMBL19709461	CC1=NN=C(C2=CC=C(CNC(=O)CCCOC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)C=C2)N=N1	C27H25N7O6	ERK1;ERK2	P27361/P28482	CRBN	US11786600B2
TPD-4C3QIB	SCHEMBL19709435	SCHEMBL19709435	CC1=NN=C(C2=CC=C(CNC(=O)CCCCOC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)C=C2)N=N1	C28H27N7O6	ERK1;ERK2	P27361/P28482	CRBN	US11786600B2
TPD-4E3AIG	SCHEMBL19692280	SCHEMBL19692280	CC1=NN=C(C2=CC=C(CNC(=O)CCCCCCOC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)C=C2)N=N1	C30H31N7O6	ERK1;ERK2	P27361/P28482	CRBN	US11786600B2
TPD-4FHXDG	SCHEMBL19692368	SCHEMBL19692368	CC1=NN=C(C2=CC=C(CNC(=O)CCCCCCCOC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)C=C2)N=N1	C31H33N7O6	ERK1;ERK2	P27361/P28482	CRBN	US11786600B2
TPD-4KC7DO	SCHEMBL25566215	SCHEMBL25566215	COC1=C(NC2=NC=C(Cl)C(NC3=CC=CC=C3S(=O)(=O)C(C)C)=N2)C=C(C)C(CCN(C)C(=O)CCCNC2=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=CC=C2)=C1	C41H45ClN8O8S	EML4-ALK;EML4-ALK G1202R	Q9HC35/Q9HC35	CRBN	WO-2021173677-A1
TPD-4OBSQQ	WO-2021173677-A1_2	.	COC1=C(NC2=NC=C(Cl)C(NC3=CC=CC=C3S(=O)(=O)C(C)C)=N2)C=C(C)C(CCN(C)C(=O)CCCCCNC2=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=CC=C2)=C1	C43H49ClN8O8S	EML4-ALK;EML4-ALK G1202R	Q9HC35/Q9HC35	CRBN	WO-2021173677-A1
TPD-4XBP6F	SCHEMBL25575738	SCHEMBL25575738; SCHEMBL30165764	COC1=C(NC2=NC=C(Cl)C(NC3=CC=CC=C3S(=O)(=O)C(C)C)=N2)C=C(C)C(CCN(C)C(=O)CCCCCCCCNC2=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=CC=C2)=C1	C46H55ClN8O8S	EML4-ALK;EML4-ALK G1202R	Q9HC35/Q9HC35	CRBN	WO-2021173677-A1
TPD-4ZIW4H	WO-2021187766-A1_1	.	CC1=CC=C(C(=O)NC2CC2)C=C1C1=CC=C(C(=O)C2=CC=C(OCCOC(=O)N/C3=C/C=C\C4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)C=C2)C=C1	C40H34N4O9	p-p38	Q16539	CRBN	WO-2021187766-A1
TPD-5AQ9VN	PRZ-18002	PRZ-18002	CC1=CC=C(C(=O)NC2CC2)C=C1C1=CC=C(C(=O)C2=CC=C(OCCOCCOC(=O)NC3=CC=CC4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)C=C2)C=C1	C42H38N4O10	p-p38	Q16539	CRBN	WO-2021187766-A1
TPD-5BWPHF	WO-2021187766-A1_3	.	CC1=CC=C(C(=O)NC2CC2)C=C1C1=CC=C(C(=O)C2=CC=C(OCCOCCOCCOC(=O)N/C3=C/C=C\C4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)C=C2)C=C1	C44H42N4O11	p-p38	Q16539	CRBN	WO-2021187766-A1
TPD-5CGAC2	CN-109651395-B_1	.	CO[C@H]1C[C@@H]2CC[C@@H](C)[C@@](O)(O2)C(=O)C(=O)N2CCCC[C@H]2C(=O)O[C@H]([C@H](C)C[C@H]2CC[C@@H](OCCOC3=CN(CCOCCOCCOCCOCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)N=N3)[C@H](OC)C2)CC(=O)[C@H](C)/C=C(\C)[C@@H](O)[C@@H](OC)C(=O)[C@H](C)C[C@H](C)/C=C/C=C/C=C/1C	C78H113N7O22	FKBP12.6	P68106	CRBN	CN-109651395-B
TPD-5DHI5A	CHEMBL4748741	CHEMBL4748741; BDBM50562312; PG1	COC1=C(C(=O)NCCCNC(=O)COC2=CC=CC3=C2C(=O)N(C2CCC(=O)NC2=O)C3=O)SC(C2=CC=NC(NC(=O)C3CC3)=C2)=N1	C32H31N7O9S	GSK-3beta	P49841	CRBN	CN-110078725-A
TPD-5E44I7	CN-112533918-A_11JQ1	.	CC1=NN=C2[C@H](CC(=O)NCCOCCNC(=O)C3=CC4=C(/N=C\C(C(=O)NCCC5=NC=CS5)=C/4)C(S)=C3)/N=C(/C3=CC=C(Cl)C=C3)C3=C(SC(C)=C3C)N12	C39H38ClN9O4S3	RPN11;BRD4	O00487/O60885	.	CN-112533918-A
TPD-5F8C7R	CN-112585127-A_05JQ1	.	CCCC(NC(=O)/C(C#N)=C/C1=NC(Br)=CC=C1)C1=CC=C(OC/C=N/OCC(=O)NCCOCCNC(=O)C[C@@H]2/N=C(/C3=CC=C(Cl)C=C3)C3=C(SC(C)=C3C)N3C(C)=NN=C23)C=C1	C46H48BrClN10O6S	uchl5	Q9Y5K5	.	CN-112585127-A
TPD-5FDTGB	SCHEMBL21759402	SCHEMBL21759402	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCC(=O)N3CCN(C4=NC(/C5=C/N=C6/C=CC(N7CCC[C@@H]7C7=CC=CC(F)=C7)=NN56)=CC=C4)CC3)C(C)(C)C)C=C2)SC=N1	C53H62FN11O5S	TPM3-TRKA;AGBL4-TRKB;ETV6-TRKC	P04629/Q16620/Q16288	VHL	CN-112888681-A
TPD-5HUB73	CHEMBL5088417	CHEMBL5088417; SCHEMBL24072458; BDBM50582386; PD155646	CCN(C1=CC(C2=CC=C(CN3CCN(CCCCOC4=C5\C(=O)N(C6CCC(=O)NC6=O)C(=O)\C5=C/C=C\4)CC3)C=C2)=CC(C(=O)NCC2=C(C)C=C(C)NC2=O)=C1C)C1CCOCC1	C51H61N7O8	EZH2;EED;SUZ12;RbAp48;RbAp46	Q15910/O75530/Q15022/Q09028/Q16576	CRBN	CN-112920176-A
TPD-5K5TC4	CHEMBL5089116	CHEMBL5089116; SCHEMBL24072455; BDBM50582377; PD155663	CC[C@H](C)N1C=C(C)C2=C1/C=C(C1=CC=C(N3CCN(CCCCO/C4=C/C=C\C5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)N=C1)\C=C/2C(=O)NCC1=C(C)C=C(C)NC1=O	C48H54N8O7	EZH2;EED;SUZ12;RbAp48;RbAp46	Q15910/O75530/Q15022/Q09028/Q16576	CRBN	CN-112920176-A
TPD-5OHMS7	SCHEMBL27092274	SCHEMBL27092274; SCHEMBL29921224	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCC(=O)NCCN3CCN(CC4=CC=CC(C5=CC=C(N6CCN(C)CC6)C(NC(=O)C6=CNC(=O)C=C6C(F)(F)F)=C5)=C4)CC3)C(C)(C)C)C=C2)SC=N1	C57H70F3N11O8S	WDR5	P61964	VHL	CN-112996518-A
TPD-5QKNCQ	SCHEMBL27092258	SCHEMBL27092258; SCHEMBL29921728	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCOCCC(=O)NCCN3CCN(CC4=CC=CC(C5=CC=C(N6CCN(C)CC6)C(NC(=O)C6=CNC(=O)C=C6C(F)(F)F)=C5)=C4)CC3)C(C)(C)C)C=C2)SC=N1	C59H74F3N11O8S	WDR5	P61964	VHL	CN-112996518-A
TPD-5R4XSV	SCHEMBL30308515	SCHEMBL30308515	NC(=O)CC[C@H](NC(=O)[C@@H]1CC[C@@H]2CCCC[C@H](NC(=O)/C3=C/C4=C(C=CC(C(F)(F)P(=O)(O)O)=C4)N3)C(=O)N21)C(=O)NCCCOCCOCCOCCCN/C1=C/C=C\C2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O	C49H62F2N9O15P	STAT3	P40763	CRBN	CN-114269763-A
TPD-5RDTWD	SCHEMBL24833575	SCHEMBL24833575; SCHEMBL31260226	CC1(C2=CC=C(NC3=C(C(N)=O)N=CC(N4CCCC(N5CCN(C6CCCC6)C5=O)C4)=N3)C=C2)CCN(C2CN(C3=C/C=C4/C(=O)N(C5CCC(=O)NC5=O)C(=O)/C4=C\3)C2)CC1	C46H55N11O6	BTK C481S	Q06187	CRBN	CN-115557933-A
TPD-5SJ5F5	SCHEMBL31121732	SCHEMBL31121732	CC1=C(/C=C2\C(=O)NC3=CC=C(F)C=C32)NC=C1NC(=O)CN1CCN(C(=O)CCOCCNC(=O)COC2=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=CC=C2)CC1	C40H41FN8O10	FLT3	P36888	CRBN	CN-116444495-A
TPD-5VBZUS	CN-116813622-A_GDPU-1	.	NC1=C2N=C(SC3=C/C4=C(\C=C/3I)OCO4)N(CCNC(=O)CN3C=C(COC4=C(Cl)C=C(N(C(=O)CCl)C(C(=O)NCCC5=CC=CC=C5)C5=CC=CS5)C=C4)N=N3)C2=NC=N1	C41H36Cl2IN11O6S2	GPX4	P36969	.	CN-116813622-A
TPD-5VDCXZ	CN-117447466-A_LL-K9-001	.	CCC(=O)N1CCC(C(=O)NC2=NC=C(SCC3=NC=C(C)O3)S2)CC1	C17H22N4O3S2	CDK9-cyclin T1	P50750	.	CN-117447466-A
TPD-5Z69OJ	CHEMBL5405221	CHEMBL5405221; SCHEMBL29227644; BDBM50622584	CC1=CC(NC2=C3C=NN(C4CCN(C(=O)COC5=C/C=C6/C(=O)N(C7CCC(=O)NC7=O)C(=O)/C6=C\5)CC4)C3=NC(NCC3=CC=C(F)C=C3F)=N2)=NN1	C36H33F2N11O6	PLK4	O00444	CRBN	CN-117886820-A
TPD-60X8GJ	CN-117886820-A_2	.	CC1=CC(NC2=C3C=NN(C4CCN(C(=O)CCCO/C5=C/C=C6/C(=O)N(C7CCC(=O)NC7=O)C(=O)C6C5)CC4)C3=NC(NCC3=CC=C(F)C=C3F)=N2)=NN1	C38H39F2N11O6	PLK4	O00444	CRBN	CN-117886820-A
TPD-62729G	CN-118027068-A_1	.	[H][C@@]12N(C3=NC=C(C4=CC(C5=CN([C@H]6CC[C@@H](N7CCC(C8=C(F)C=C(NC9CCC(=O)NC9=O)C=C8)CC7)CC6)N=C5)=CN5N=CC(C#N)=C45)C=C3)C[C@]1([H])N(CC1=CN=C(OC)C=C1)CC2(C)N	C51H56FN13O3	RET-G810R	P07949	CRBN	CN-118027068-A
TPD-6I85WD	CN-118027068-A_2	.	[H][C@@]12N(C3=NC=C(C4=CC(C5=CN([C@H]6CC[C@H](N7CCC(C8=C(F)C=C(NC9CCC(=O)NC9=O)C=C8)CC7)CC6)N=C5)=CN5/N=C\C(C#N)=C\45)C=C3)C[C@]1([H])N(CC1=CN=C(OC)C=C1)CC2(C)N	C51H56FN13O3	RET-G810R	P07949	CRBN	CN-118027068-A
TPD-6RLP4W	CN-118139860-A_1	.	CCC1=CC2=C(/C=C(CN3CCN(C4=CC=C(C(=O)NC5CCN(C6CN(C7=C/C=C8/C(=O)N(C9CCC(=O)NC9=O)C(=O)/C8=C\7)C6)CC5)N=C4)CC3)\C=N/2)NC1=O	C42H46N10O6	PARP1	P09874	CRBN	CN-118139860-A
TPD-6RWL5U	SCHEMBL26088901	SCHEMBL26088901; SCHEMBL30384950	CCC1=CC2=C(/C=C(CN3CCN(C4=CC=C(C(=O)NC5CCN(C6CCN(C7=C/C=C8/C(=O)N(C9CCC(=O)NC9=O)C(=O)/C8=C\7)CC6)CC5)N=C4)CC3)\C=N/2)NC1=O	C44H50N10O6	PARP1	P09874	CRBN	CN-118139860-A
TPD-6SPER9	CN-119431379-A_I-A-1	.	CC/C1=C(\N2CCN(CC(=O)NC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)CC2)C(=O)N2N=C(C3=CCOCC3)N=C2N1CC(=O)NC1=CC=C(C(F)(F)F)C=C1Cl	C40H38ClF3N10O8	WRN	Q14191	CRBN	CN-119431379-A
TPD-6TDE0A	CN-119431379-A_I-A-2	.	CC/C1=C(\N2CCN(CCCC(=O)NC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)CC2)C(=O)N2N=C(C3=CCOCC3)N=C2N1CC(=O)NC1=CC=C(C(F)(F)F)C=C1Cl	C42H42ClF3N10O8	WRN	Q14191	CRBN	CN-119431379-A
TPD-6TEJ0K	CN-119504718-A_DhpB	.	[H][C@]1([C@H](C2=CC(OC)=C(OC)C(OC)=C2)C2=CC(OC)=C3OCOC3=C2)COC(=O)C1CN(C)CCO	C26H33NO9	RPS7	P62081	MKRN2	CN-119504718-A
TPD-6TI25H	CN-119775213-A_A15	.	COC1=CC=C(C(=O)NC2=CC(CN(C)C)=CC(C(F)(F)F)=C2)C=C1C#CC1=CN=C(NC2CCN(CCC(=O)NC3=CC=C4C(=O)N(C5CCC(=O)NC5=O)CC4=C3)CC2)N=C1	C45H46F3N9O6	DDR1	Q08345	CRBN	CN-119775213-A
TPD-6UYALG	CN-119823115-A_2	.	COC1=CC=CC=C1C1=CN=CC=C1C(=O)NC1=NN=C(OCC2=CC=C(C(=O)NC34CC5CC(CC(C5)C3)C4)C=C2)S1	C33H33N5O4S	Pol胃	O75417	.	CN-119823115-A
TPD-6VY8QH	CN-120172981-A_NT-01	.	COC1=CC(C#CC2=NN(C3CCN(C(=O)CO/C4=C/C=C\C5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)C3=NC=NC(N)=C23)=CC(OC)=C1	C34H30N8O8	FGFR2	P21802	CRBN	CN-120172981-A
TPD-77UIZ0	CN-120172981-A_NT-02	.	COC1=CC(C#CC2=NN(C3CCN(C(=O)CN/C4=C/C=C\C5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)C3=NC=NC(N)=C23)=CC(OC)=C1	C34H31N9O7	FGFR2	P21802	CRBN	CN-120172981-A
TPD-792LVA	CN-120271564-A_1	.	C[C@H](NC(=O)C1=CC2=CC=CC(C3=CC=C(C(F)(F)F)C=C3)=C2C=C1)C1=CC=CC(NC2CCN(CC3CN(C4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C3)CC2)=N1	C47H44F3N7O5	tead1;tead2;tead3;tead4	P28347/Q15562/Q99594/Q15561	CRBN	CN-120271564-A
TPD-7CBLT3	CN-120271564-A_2	.	C[C@H](NC(=O)C1=CC2=CC=CC(C3=CC=C(C(F)(F)F)C=C3)=C2C=C1)C1=CC=CC(NC2CCN(CC3CN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)C3)CC2)=N1	C47H44F3N7O5	tead1;tead2;tead3;tead4	P28347/Q15562/Q99594/Q15561	CRBN	CN-120271564-A
TPD-7EJ6V8	SCHEMBL22221627	SCHEMBL22221627	CC(C)N(C[C@H]1O[C@@H](N2C=NC3=C2N=CN=C3NCCCCNC(=O)CCCC(=O)NCCCCCCCC(=O)N[C@H](CC2=CC=CC=C2)C(=O)N2C/C(=C\C3=CC=C(Cl)C(Cl)=C3)C(=O)/C(=C/C3=CC(Cl)=C(Cl)C=C3)C2)C(O)C1O)C1CC(CCC2=NC3=C(C=CC(C(C)(C)C)=C3)N2)C1	C75H92Cl4N12O8	DOT1L	Q8TEK3	.	US-12331069-B2
TPD-7K6DT8	ARV-102	ARV-102; EX-A12186	CN1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(N3CCC(O[C@H]4CC[C@H](CN5CCN(C6=CC(C7=NNC8=CN=C(OC9(C)CC9)C=C87)=NC=N6)CC5)CC4)CC3)C=C21	C43H53N11O5	LRRK2	Q5S007	CRBN	WO-2025072629-A1
TPD-7KS0JL	WO-2025072629-A1_2	.	CC(C)N1C(=O)N(C2CCC(=O)NC2=O)C2=CC=C(N3CCC(CN4CCN(CC5CCN(C6=CC(C7=NNC8=CC=C(OC9(C)CC9)C=C87)=NC=N6)CC5)C(C)(C)C4)CC3)C=C21	C48H63N11O4	LRRK2	Q5S007	CRBN	WO-2025072629-A1
TPD-7PBYL1	WO-2025083594-A1_1	.	CC1(C)CC(NC2=CC=CC(C3=C(F)C(OCC(=O)O)=C(C(=O)O)S3)=C2)CCN1S(=O)(=O)CC1=CC(NC(=O)N2CCC(/C3=C/C=C4\C5=C3C=CC=C5C(=O)N4C3CCC(=O)NC3=O)CC2)=CC=C1	C49H49FN6O11S2	PTPN2;PTPN1	P17706/P18031	CRBN	WO-2025083594-A1
TPD-7RIOG1	SCHEMBL31642793	SCHEMBL31642793	CC1=C(C2=CC=C(NC(=O)C3CC3)C=C2)N=C(NC(=O)CC2=CC=CC(OCCOCCN/C3=C/C=C\C4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)=C2)S1	C39H38N6O8S	Nrf2	Q16236	CRBN	WO-2025137606-A1
TPD-7XLH0J	SCHEMBL31643067	SCHEMBL31643067	CC1=CC(C2=C(C)SC(NC(=O)CC3=CC=CC(OCCOCCN/C4=C/C=C\C5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)=C3)=N2)=CC=C1NC(=O)C1CC1	C40H40N6O8S	Nrf2	Q16236	CRBN	WO-2025137606-A1
TPD-811VN3	US-20220185831-A1_1	.	NC(=O)CC[C@H](NC(=O)[C@@H]1CC[C@@H]2C[C@H](NC(=O)CCCCCC#C/C3=C/C=C\C4=C3CN(C3CCC(=O)NC3=O)C4=O)CC[C@H](NC(=O)/C3=C/C4=C(C=CC(C(F)(F)P(=O)(O)O)=C4)N3)C(=O)N21)C(=O)NC(C1=CC=CC=C1)C1=CC=CC=C1	C60H64F2N9O12P	STAT3	P40763	CRBN	US-20220185831-A1
TPD-82FK9I	US-20220185831-A1_2	.	NC(=O)CC[C@H](NC(=O)[C@@H]1CC[C@@H]2C[C@@H](NC(=O)CCCCCC#C/C3=C/C=C\C4=C3CN(C3CCC(=O)NC3=O)C4=O)CC[C@H](NC(=O)/C3=C/C4=C(C=CC(C(F)(F)P(=O)(O)O)=C4)N3)C(=O)N21)C(=O)NC(C1=CC=CC=C1)C1=CC=CC=C1	C60H64F2N9O12P	STAT3	P40763	CRBN	US-20220185831-A1
TPD-89NA0G	US-20220185831-A1_3	.	NC(=O)CC[C@H](NC(=O)[C@@H]1CC[C@@H]2C[C@H](NCCCCCCC#C/C3=C/C=C\C4=C3CN(C3CCC(=O)NC3=O)C4=O)CC[C@H](NC(=O)/C3=C/C4=C(C=CC(C(F)(F)P(=O)(O)O)=C4)N3)C(=O)N21)C(=O)NC(C1=CC=CC=C1)C1=CC=CC=C1	C60H66F2N9O11P	STAT3	P40763	CRBN	US-20220185831-A1
TPD-8KJM6M	US-20220185831-A1_4	.	NC(=O)CC[C@H](NC(=O)[C@@H]1CC[C@@H]2C[C@@H](NCCCCCCC#C/C3=C/C=C\C4=C3CN(C3CCC(=O)NC3=O)C4=O)CC[C@H](NC(=O)/C3=C/C4=C(C=CC(C(F)(F)P(=O)(O)O)=C4)N3)C(=O)N21)C(=O)NC(C1=CC=CC=C1)C1=CC=CC=C1	C60H66F2N9O11P	STAT3	P40763	CRBN	US-20220185831-A1
TPD-8KW8PO	SCHEMBL29622166	SCHEMBL29622166	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCNC(=O)CC3CCN(CC4=NC5=CC(NC(=O)C6=CC=C7C(=C6)C=NN7C)=CC=C5N4)C3)C(C)(C)C)C=C2)SC=N1	C49H59N11O7S	MLLT1	Q03111	VHL	US-20230391765-A1
TPD-8L7VZU	SCHEMBL26911693	SCHEMBL26911693; SCHEMBL30704519	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCOCCNC(=O)CC3CCN(CC4=NC5=CC(NC(=O)C6=C\C=C7C(=C/6)/C=NN/7C)=CC=C5N4)C3)C(C)(C)C)C=C2)SC=N1	C50H61N11O7S	MLLT1	Q03111	VHL	US-20230391765-A1
TPD-8MW84P	SCHEMBL26911606	SCHEMBL26911606; SCHEMBL30704665	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCNC(=O)CC3CCN(CC4=NC5=CC(NC(=O)C6=C/C=C7C(=C/6)\C=NN\7C)=CC=C5N4)C3)C(C)(C)C)C=C2)SC=N1	C51H63N11O8S	MLLT1	Q03111	VHL	US-20230391765-A1
TPD-8NAC5D	SCHEMBL30704662	SCHEMBL30704662	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCOCCOCCNC(=O)CC3CCN(CC4=NC5=CC(NC(=O)C6=CC=C7C(=C6)C=NN7C)=CC=C5N4)C3)C(C)(C)C)C=C2)SC=N1	C52H65N11O8S	MLLT1	Q03111	VHL	US-20230391765-A1
TPD-8OPTM7	SCHEMBL26911439	SCHEMBL26911439; SCHEMBL30704617	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCOCCOCCNC(=O)CC3CCN(CC4=NC5=CC(NC(=O)C6=CC=C7C(=C6)C=NN7C)=CC=C5N4)C3)C(C)(C)C)C=C2)SC=N1	C53H67N11O9S	MLLT1	Q03111	VHL	US-20230391765-A1
TPD-8T3RGR	SCHEMBL25511698	SCHEMBL25511698; SCHEMBL30462372	CC1=C(OCC2=CC=CC=C2)C(C(=O)N2CC3=C(/C=C(CN4CCN(CCOCCOCCNC5=CC=CC6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)\C=C/3)C2)=C(O)C=C1O	C47H52N6O10	PMS2	P54278	CRBN	US-20240425483-A1
TPD-8W7A35	SCHEMBL30462383	SCHEMBL30462383	CC1=C(OCC2=CC=CC=C2)C(C(=O)N2CC3=C(/C=C(CN4CCN(CCOCCOCCOCCOCCNC5=CC=CC6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)\C=C/3)C2)=C(O)C=C1O	C51H60N6O12	PMS2	P54278	CRBN	US-20240425483-A1
TPD-8WE7TG	US-20240425483-A1_4	.	CC1=C(OCC2=CC=CC=C2)C(C(=O)N2CC3=C(/C=C(CN4CCN(CCOCCOCCOCCOCCOCNC5=CC=CC6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)\C=C/3)C2)=C(O)C=C1O	C52H62N6O13	PMS2	P54278	CRBN	US-20240425483-A1
TPD-8XM8FO	CHEMBL5421882	CHEMBL5421882; SCHEMBL20113926; PD141637	CN[C@@H](C)C(=O)N[C@H](C(=O)N1CC2=C(C=CC(OCCOCCOCCOCCOC3=C/C4=C(\C=C/3S(=O)(=O)C(C)(C)C)C(NC3=C/C5=C(\C=C/3)SC=N5)=CC=N4)=C2)C[C@H]1C(=O)N[C@@H]1CCCC2=C1C=CC=C2)C(C)(C)C	C58H73N7O10S2	RIPK2	O43353	VHL	US10435391B2
TPD-91WS9R	SCHEMBL18181853	SCHEMBL18181853	CN[C@@H](C)C(=O)N[C@H](C(=O)N1CC2=C(/C=C\C(OCCOCCOCCOCCOC3=CC4=C(C=C3S(=O)(=O)C(C)(C)C)/C(NC3=CC5=C(C=C3)S/C=N\5)=C\C=N/4)=C/2)C[C@H]1C(=O)N[C@H]1CCCC2=C1C=CC=C2)C(C)(C)C	C58H73N7O10S2	RIPK2	O43353	VHL	US10435391B2
TPD-94PW5J	SCHEMBL20137249	SCHEMBL20137249; PD172236	CN[C@@H](C)C(=O)N[C@H](C(=O)N1CC2=C(/C=C\C(OCCOCCOCCOCCOC3=CC4=C(C=C3S(=O)(=O)C(C)(C)C)/C(NC3=NNC(C)=C3C)=N\C=N/4)=C/2)C[C@H]1C(=O)N[C@@H]1CCCC2=C1C=CC=C2)C(C)(C)C	C55H75N9O10S	RIPK2	O43353	VHL	US10435391B2
TPD-97W5IF	dBET1	dBET1; 1799711-21-9; MFCD31544503; 2-((S)-4-(4-chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl)-N-(4-(2-((2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindolin-4-yl)oxy)acetamido)butyl)acetamide; CHEMBL4094346; 2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]-N-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyacetyl]amino]butyl]acetamide; dBET1?; JQ1-Thalidomide conjugate; C38H37ClN8O7S; orb1302813; SCHEMBL17553399; SCHEMBL29566239; GLXC-06330; EX-A1817; ZWC71121; BDBM50544938; s8296; AKOS032962867; SG5-025; AC-35891; BP-27851; DA-62701; SY388958; HY-101838; CS-0021961; D70029; EN300-26567647; F986769; Z3070465669; (6S)-4-(4-Chlorophenyl)-N-[4-[[2-[[2-(2,6-dioxo-3-piperidinyl)-2,3-dihydro-1,3-dioxo-1H-isoindol-4-yl]oxy]acetyl]amino]butyl]-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetamide;; 2-((S,Z)-4-(4-Chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl)-N-(4-(2-(2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindolin-4-yloxy)acetamido)butyl)acetamide; 2-[(S)-4-(4-Chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl]-N-[4-[2-[[2-(2,6-dioxo-3-piperidyl)-1,3-dioxo-4-isoindolinyl]oxy]acetamido]butyl]acetamide; N-(4-{2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetraazatricyclo[8.3.0.0,2,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetamido}butyl)-2-{[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]oxy}acetamide; N-[4-[2-[2-[2,6-bis(oxidanylidene)piperidin-3-yl]-1,3-bis(oxidanylidene)isoindol-4-yl]oxyethanoylamino]butyl]-2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]ethanamide	CC1=NN=C2[C@H](CC(=O)NCCCCNC(=O)CO/C3=C/C=C\C4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)/N=C(/C3=CC=C(Cl)C=C3)C3=C(SC(C)=C3C)N12	C38H37ClN8O7S	MYCN	P04198	CRBN	US10464925B2
TPD-9C53XQ	SCHEMBL17859030	SCHEMBL17859030; BDBM511595; US11059801, Compound dBET3	CC1=NN=C2[C@H](CC(=O)NCCNC(=O)CO/C3=C/C=C\C4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)/N=C(/C3=CC=C(Cl)C=C3)C3=C(SC(C)=C3C)N12	C36H33ClN8O7S	MYCN	P04198	CRBN	US10464925B2
TPD-9F3LRK	SCHEMBL17859034	SCHEMBL17859034; BDBM511596; US11059801, Compound dBET4	CC1=C(C)C2=C(S1)N1/C(C)=N\N=C/1[C@@H](CC(=O)NCCCCNC(=O)CO/C1=C/C=C\C3=C1C(=O)N(C1CCC(=O)NC1=O)C3=O)/N=C\2C1=CC=C(Cl)C=C1	C38H37ClN8O7S	MYCN	P04198	CRBN	US10464925B2
TPD-9JYL49	dBET6	dBET6; DTXSID901022545; RefChem:131047; DTXCID701507230; 1950634-92-0; 2-((S)-4-(4-Chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl)-N-(8-(2-((2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindolin-4-yl)oxy)acetamido)octyl)-acetamide; 2-((S)-4-(4-chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl)-N-(8-(2-((2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindolin-4-yl)oxy)acetamido)octyl)acetamide; MFCD31692407; 2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]-N-[8-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyacetyl]amino]octyl]acetamide; C42H45ClN8O7S; dBET 6; dBET6?; orb1302063; CHEMBL4303781; SCHEMBL17859031; GTPL10534; CHEBI:189651; BDBM511598; GLXC-10995; 2-((S)-4-(4-Chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2- f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl)-N-(8-(2-((2-(2,6- dioxopiperidin-3-yl)-1,3-dioxoisoindolin-4- yl)oxy)acetamido)octyl)acetamide; EX-A3094; US11059801, Compound dBET6; s8762; AKOS037653363; AT14156; AC-35571; BD177448; BP-28374; DA-52347; SY389665; HY-112588; CS-0047679; EN300-23308290; F837796; 2-[(S)-4-(4-Chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl]-N-[8-[2-[[2-(2,6-dioxo-3-piperidyl)-1,3-dioxo-4-isoindolinyl]oxy]acetamido]octyl]acetamide; N-(8-{2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetraazatricyclo[8.3.0.0,2,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetamido}octyl)-2-{[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]oxy}acetamide; N-(8-{2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetraazatricyclo[8.3.0.0,trideca-2(6),4,7,10,12-pentaen-9-yl]acetamido}octyl)-2-{[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]oxy}acetamide; N-[8-[2-[2-[2,6-bis(oxidanylidene)piperidin-3-yl]-1,3-bis(oxidanylidene)isoindol-4-yl]oxyethanoylamino]octyl]-2-[(9S)-7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]ethanamide	CC1=NN=C2[C@H](CC(=O)NCCCCCCCCNC(=O)CO/C3=C/C=C\C4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)/N=C(/C3=CC=C(Cl)C=C3)C3=C(SC(C)=C3C)N12	C42H45ClN8O7S	MYCN	P04198	CRBN	US10464925B2
TPD-9LQHLK	CHEMBL4591946	CHEMBL4591946; SCHEMBL18379499	CCC(C)(C)C(=O)C(=O)N1CCCCC1C(=O)O[C@H](CCC1=CC=C(OC)C(OC)=C1)C1=CC=CC(NC(=O)CCC(=O)NCCCCNC(=O)CO/C2=C/C=C\C3=C2C(=O)N(C2CCC(=O)NC2=O)C3=O)=C1	C53H64N6O14	MYCN	P04198	CRBN	US10464925B2
TPD-A8UGWU	SCHEMBL18019930	SCHEMBL18019930	CCC(C)(C)C(=O)C(=O)N1CCCCC1C(=O)O[C@H](CCC1=CC=C(OC)C(OC)=C1)C1=CC=CC(NC(=O)CCC(=O)NCCCOCCOCCOCCCNC(=O)CO/C2=C/C=C\C3=C2C(=O)N(C2CCC(=O)NC2=O)C3=O)=C1	C59H76N6O17	MYCN	P04198	CRBN	US10464925B2
TPD-AC6CJA	SCHEMBL25096384	SCHEMBL25096384	O=C(CN1CCN(C(=O)C2=CC(F)=C(NC3=NC(C4CC4)=CN4/C(C5=CNN=C5)=C\N=C\34)C=C2)CC1)NCCCN/C1=C/C=C\C2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O	C41H41FN12O6	PTK6	Q13882	CRBN	WO-2020010204-A1
TPD-ACN6ZT	SCHEMBL25096072	SCHEMBL25096072	O=C(CN1CCN(C(=O)C2=CC(F)=C(NC3=NC(C4CC4)=CN4C(C5=CNN=C5)=CN=C34)C=C2)CC1)NCCN/C1=C/C=C\C2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O	C40H39FN12O6	PTK6	Q13882	CRBN	WO-2020010204-A1
TPD-ACU3EO	SCHEMBL25096490	SCHEMBL25096490	O=C(CN1CCN(C(=O)C2=CC(F)=C(NC3=NC(C4CC4)=CN4/C(C5=CNN=C5)=C\N=C\34)C=C2)CC1)NCCCCN/C1=C/C=C\C2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O	C42H43FN12O6	PTK6	Q13882	CRBN	WO-2020010204-A1
TPD-AFGWRS	SCHEMBL25096362	SCHEMBL25096362	O=C(CN1CCN(C(=O)C2=CC(F)=C(NC3=NC(C4CC4)=CN4C(C5=CNN=C5)=CN=C34)C=C2)CC1)NCCCCCN/C1=C/C=C\C2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O	C43H45FN12O6	PTK6	Q13882	CRBN	WO-2020010204-A1
TPD-AOL2KZ	DGY-03-081	DGY-03-081; CHEMBL5198513; SCHEMBL23975093	[H][C@@]12CCC[C@]1([H])[C@@H](C(=O)N[C@@H](CCC)C(=O)C(=O)NC1CC1)N(C(=O)[C@@H](NC(=O)[C@@H](NC(=O)C1=NC=C(C(=O)NCCCCCCNC3=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)N=C1)C1CCCCC1)C(C)(C)C)C2	C56H77N11O10	ns3;ns4a;NS3-V55A;NS3-Al56S;NS3-eGFP	P27958/P26663/P27958/P27958/P27958	CRBN	WO-2020069125-A1
TPD-ARD5PP	WO-2020069125-A1_11	.	[H][C@@]12CCC[C@]1([H])[C@@H](C(=O)N[C@@H](CCC)C(O)C(=O)NC1CC1)N(C(=O)[C@@H](NC(=O)[C@@H](NC(=O)C1=NC=C(C(=O)NCCOCCOCCNC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)N=C1)C1CCCCC1)C(C)(C)C)C2	C56H77N11O13	ns3;ns4a;NS3-V55A;NS3-Al56S;NS3-eGFP	P27958/P26663/P27958/P27958/P27958	CRBN	WO-2020069125-A1
TPD-AT5E26	DGY-04-035	DGY-04-035; CHEMBL5196237; SCHEMBL23975015	[H][C@@]12CCC[C@]1([H])[C@@H](C(=O)N[C@@H](CCC)C(=O)C(=O)NC1CC1)N(C(=O)[C@@H](NC(=O)[C@@H](NC(=O)C1=NC=C(C(=O)NCCOCCOCCNC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)N=C1)C1CCCCC1)C(C)(C)C)C2	C56H75N11O13	ns3;ns4a;NS3-V55A;NS3-Al56S;NS3-eGFP	P27958/P26663/P27958/P27958/P27958	CRBN	WO-2020069125-A1
TPD-AW01PN	SCHEMBL23975116	SCHEMBL23975116	[H][C@@]12CCC[C@]1([H])[C@@H](C(=O)N[C@@H](CCC)C(=O)C(=O)NC1CC1)N(C(=O)[C@@H](NC(=O)[C@@H](NC(=O)C1=NC=C(C(=O)NCCCCCCCC(=O)NC3=C4CN(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)N=C1)C1CCCCC1)C(C)(C)C)C2	C58H79N11O11	ns3;ns4a;NS3-V55A;NS3-Al56S;NS3-eGFP	P27958/P26663/P27958/P27958/P27958	CRBN	WO-2020069125-A1
TPD-B10XCX	WO-2020069125-A1_9	.	[H][C@@]12CCC[C@]1([H])[C@@H](C(=O)N[C@@H](CCC)C(=O)C(=O)NC1CCCC1)N(C(=O)[C@@H](NC(=O)[C@@H](NC(=O)C1=NC=C(C(=O)NCCOCCOCCNC(=O)CCOCCOCCNC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)N=C1)C1CCCCC1)C(C)(C)C)C2	C65H92N12O16	ns3;ns4a;NS3-V55A;NS3-Al56S;NS3-eGFP	P27958/P26663/P27958/P27958/P27958	CRBN	WO-2020069125-A1
TPD-BDGORK	SCHEMBL21938874	SCHEMBL21938874	CNC1=NC(NC2=CC=C(C(=O)N3CCN(CCOCCOCCOCCOCCNC4=CC=CC5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)C=C2OC)=NC=C1Cl	C40H50ClN9O10	LRRK2 G2019S;LRRK2	Q5S007/Q5S007	CRBN	WO-2020081682-A1
TPD-BHHCB7	SCHEMBL21938878	SCHEMBL21938878; FSAWYWAIHFCKHA-UHFFFAOYSA-N; 2-(2,6-Dioxopiperidin-3-yl)-4-[2-[2-[2-[2-[2-[4-[3-methoxy-4-[[4-(methylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino]benzoyl]piperazin-1-yl]ethoxy]ethoxy]ethoxy]ethoxy]ethylamino]isoindole-1,3-dione	CNC1=NC(NC2=CC=C(C(=O)N3CCN(CCOCCOCCOCCOCCNC4=CC=CC5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)C=C2OC)=NC=C1C(F)(F)F	C41H50F3N9O10	LRRK2 G2019S;LRRK2	Q5S007/Q5S007	CRBN	WO-2020081682-A1
TPD-BQ1E8Z	CHEMBL4759913	CHEMBL4759913; SCHEMBL21939590; BDBM50628343; PD215259	CC1(OC2=CC=C3NN=C(C4=NC=NC(N5CCN(C(=O)CCOCCOCCNC6=C7\C(=O)N(C8CCC(=O)NC8=O)C(=O)\C7=C/C=C\6)CC5)=C4)C3=C2)CC1	C39H43N9O8	LRRK2 G2019S;LRRK2	Q5S007/Q5S007	CRBN	WO-2020081682-A1
TPD-BQ2XJ6	JH-XII-03-02	JH-XII-03-02; 2415900-86-4; CHEMBL4752225; orb2278011; SCHEMBL21939268; GTPL12908; BDBM50628346; EX-A12436; compound 6 [PMID: 37591317]; DA-74643; HY-155150; CS-0887715; 2-(2,6-dioxopiperidin-3-yl)-4-[2-[2-[2-[2-[3-[4-[6-[5-(1-methylcyclopropyl)oxy-1H-indazol-3-yl]pyrimidin-4-yl]piperazin-1-yl]-3-oxopropoxy]ethoxy]ethoxy]ethoxy]ethylamino]isoindole-1,3-dione	CC1(OC2=CC=C3N/N=C(/C4=NC=NC(N5CCN(C(=O)CCOCCOCCOCCOCCNC6=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)CC5)=C4)C3=C2)CC1	C43H51N9O10	LRRK2 G2019S;LRRK2	Q5S007/Q5S007	CRBN	WO-2020081682-A1
TPD-BZO74I	SCHEMBL22468630	SCHEMBL22468630	NC(=O)CC[C@H](NC(=O)[C@@H]1CC[C@@H]2CCN(C(=O)CCCCCC#C/C3=C/C=C\C4=C3CN(C3CCC(=O)NC3=O)C4=O)C[C@H](NC(=O)/C3=C/C4=C(C=CC(C(F)(F)P(=O)(O)O)=C4)S3)C(=O)N21)C(=O)NC(C1=CC=CC=C1)C1=CC=CC=C1	C59H61F2N8O12PS	STAT3;STAT1	P40763/P42224	CRBN	WO-2020198435-A1
TPD-C0OM6T	SD-36	SD-36; CHEMBL4452527; [[2-[[(5S,8S,10aR)-8-[[(2S)-5-amino-1-(benzhydrylamino)-1,5-dioxopentan-2-yl]carbamoyl]-3-[8-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-3H-isoindol-4-yl]oct-7-ynoyl]-6-oxo-1,2,4,5,8,9,10,10a-octahydropyrrolo[1,2-a][1,5]diazocin-5-yl]carbamoyl]-1H-indol-5-yl]-difluoromethyl]phosphonic acid; ((2-(((5S,8S,10aR)-8-(((S)-5-Amino-1-(benzhydrylamino)-1,5-dioxopentan-2-yl)carbamoyl)-3-(8-(2-(2,6-dioxopiperidin-3-yl)-1-oxoisoindolin-4-yl)oct-7-ynoyl)-6-oxodecahydropyrrolo[1,2-a][1,5]diazocin-5-yl)carbamoyl)-1H-indol-5-yl)difluoromethyl)phosphonic acid; orb1987750; SD36; SCHEMBL22468769; SCHEMBL30308498; GTPL12915; GLXC-21755; EX-A5026; BDBM50514302; AKOS040743878; compound 14 [PMID: 31747516]; BP-41602; HY-129602; CS-0106866; EN300-33135220; ((2-(((5S,8S,10aR)-8-(((S)-5-Amino-1-(benzhydrylamino)-1,5-dioxopentan-2-yl)carbamoyl)-3-(8-(2-(2,6-dioxopiperidin-3-yl)-1-oxoiSoindolin-4-yl)oct-7-ynoyl)-6-oxodecahydropyrrolo[1,2-a][1,5]diazocin-5-yl)carbamoyl)-1H-indol-5-yl)difluoromethyl)phosphonic ac; [(2-{[(5S,8S,10aR)-8-{[(1S)-3-carbamoyl-1-[(diphenylmethyl)carbamoyl]propyl]carbamoyl}-3-{8-[2-(2,6-dioxopiperidin-3-yl)-1-oxo-2,3-dihydro-1H-isoindol-4-yl]oct-7-ynoyl}-6-oxo-decahydropyrrolo[1,2-a][1,5]diazocin-5-yl]carbamoyl}-1H-indol-5-yl)difluoromethyl]phosphonic acid	NC(=O)CC[C@H](NC(=O)[C@@H]1CC[C@@H]2CCN(C(=O)CCCCCC#CC3=CC=CC4=C3CN(C3CCC(=O)NC3=O)C4=O)C[C@H](NC(=O)/C3=C/C4=C(C=CC(C(F)(F)P(=O)(O)O)=C4)N3)C(=O)N21)C(=O)NC(C1=CC=CC=C1)C1=CC=CC=C1	C59H62F2N9O12P	STAT3;STAT1	P40763/P42224	CRBN	WO-2020198435-A1
TPD-C2M6JE	CHEMBL4532980	CHEMBL4532980; SCHEMBL22468638; SCHEMBL30308493	CN1C(=O)CCC(N2CC3=C(/C=C\C=C/3C#CCCCCCC(=O)N3CC[C@H]4CC[C@@H](C(=O)N[C@@H](CCC(N)=O)C(=O)NC(C5=CC=CC=C5)C5=CC=CC=C5)N4C(=O)[C@@H](NC(=O)/C4=C/C5=C(C=CC(C(F)(F)P(=O)(O)O)=C5)N4)C3)C2=O)C1=O	C60H64F2N9O12P	STAT3;STAT1	P40763/P42224	CRBN	WO-2020198435-A1
TPD-C6CDWQ	SCHEMBL22737251	SCHEMBL22737251	NC1=C2C(C3=CC=C(OC4=CC=CC=C4)C=C3)=NN(C3CCN(CC4CN(C5CCN(C6=C/C=C7/C(=O)N(C8CCC(=O)NC8=O)C(=O)/C7=C\6)CC5)C4)CC3)C2=NC=N1	C44H46N10O5	BTK C481S	Q06187	CRBN	WO-2020239103-A1
TPD-CEN42H	SCHEMBL22720885	SCHEMBL22720885; SCHEMBL29439233	NC1=C2C(C3=CC=C(OC4=CC=CC=C4)C=C3)=NN(C3CCN(C4CCN(C5CCN(C6=C/C=C7\C(=O)N(C8CCC(=O)NC8=O)C(=O)\C7=C\6)CC5)CC4)CC3)C2=NC=N1	C45H48N10O5	BTK C481S	Q06187	CRBN	WO-2020239103-A1
TPD-CH9LA2	SCHEMBL22737431	SCHEMBL22737431	NC1=C2C(C3=CC=C(OC4=CC=CC=C4)C=C3)=NN(C3CCN(CC4CCN(C5CN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C2=NC=N1	C44H46N10O5	BTK C481S	Q06187	CRBN	WO-2020239103-A1
TPD-CIPZZM	SCHEMBL22720886	SCHEMBL22720886; SCHEMBL29439101	NC1=C2C(C3=CC=C(OC4=CC=CC=C4)C=C3)=NN(C3CCN(C4CCN(C5CN(C6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)C5)CC4)CC3)C2=NC=N1	C43H44N10O5	BTK C481S	Q06187	CRBN	WO-2020239103-A1
TPD-CTO7BY	SCHEMBL22737475	SCHEMBL22737475	NC1=C2C(C3=CC=C(OC4=CC=CC=C4)C=C3)=NN(C3CCN(CC4CCN(C5CCN(C6=C/C=C7/C(=O)N(C8CCC(=O)NC8=O)C(=O)/C7=C\6)CC5)CC4)CC3)C2=NC=N1	C46H50N10O5	BTK C481S	Q06187	CRBN	WO-2020239103-A1
TPD-CYJZPS	SCHEMBL20120831	SCHEMBL20120831; SCHEMBL29547405	CN1C2=CC=NC=C2C2=C1/C=C(C1=CN=C(OCC#CCOCCCCOCCCCOC3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C=C1)\C=C/2	C42H41N5O8	tauP301L	P10636	CRBN	WO-2021011913-A1
TPD-D94MHK	SCHEMBL20120813	SCHEMBL20120813; SCHEMBL20120814; SCHEMBL29547810	CN1C2=CC=NC=C2C2=C1/C=C(C1=CN=C(O[C@H]3C[C@H](OCCCCCCCCN4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)C3)C=C1)\C=C/2	C46H51N7O6	tauP301L	P10636	CRBN	WO-2021011913-A1
TPD-DA9HOR	SCHEMBL20120399	SCHEMBL20120399; SCHEMBL29548307; JTOIMQJVGOJKQP-UHFFFAOYSA-N; 5-[6-[5-[2,2-Difluoro-2-[5-(5-methylpyrido[4,3-b]indol-7-yl)pyridin-2-yl]ethoxy]pentoxy]hexoxy]-2-(2,6-dioxopiperidin-3-yl)isoindole-1,3-dione	CN1C2=CC=NC=C2C2=C1/C=C(C1=CN=C(C(F)(F)COCCCCCOCCCCCCOC3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4=O)C=C1)\C=C/2	C43H45F2N5O7	tauP301L	P10636	CRBN	WO-2021011913-A1
TPD-DB3L10	SCHEMBL22954513	SCHEMBL22954513	COC1=C(NC(=O)C2=NC(C3=CC=NN3)=CC=C2)C=CC(N2CCN(C(=O)CCCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCC3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)CC2)=C1	C47H56N10O7S	IRAK1	P51617	VHL	WO-2021018118-A1
TPD-DGXHF7	SCHEMBL22954590	SCHEMBL22954590	COC1=C(NC(=O)C2=NC(C3=CC=NN3)=CC=C2)C=CC(N2CCN(C(=O)CCCCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCC3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)CC2)=C1	C48H58N10O7S	IRAK1	P51617	VHL	WO-2021018118-A1
TPD-DU6ONM	SCHEMBL22954621	SCHEMBL22954621	COC1=C(NC(=O)C2=NC(C3=CC=NN3)=CC=C2)C=CC(N2CCN(C(=O)CC(C)CC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCC3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)CC2)=C1	C48H58N10O7S	IRAK1	P51617	VHL	WO-2021018118-A1
TPD-DVKJC9	SCHEMBL22955662	SCHEMBL22955662	COC1=C(NC(=O)C2=NC(C3=CC=NN3)=CC=C2)C=CC(N2CCN(C(=O)CCCCCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCC3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)CC2)=C1	C49H60N10O7S	IRAK1	P51617	VHL	WO-2021018118-A1
TPD-DXUP51	WO-2021194878-A1_1	.	CC1=C(C(=O)NC2=CC=C3NN=C(C4=CC=NC(N5C[C@@H](C)N(CC6CCN(CC7CCN(C8=C/C9=C(\C=C/8)C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)CC6)[C@@H](C)C5)=C4)C3=C2)CN2N=NN=C2N1	C49H57N15O5	LRRK2	Q5S007	CRBN	WO-2021194878-A1
TPD-E0ILKN	SCHEMBL23860627	SCHEMBL23860627; SCHEMBL29450395	CC1=C(C(=O)NC2=CC=C3NN=C(C4=CC=NC(N5CCN(CCC6CCN(CC7CCN(C8=CC=C9C(=O)N(C%10CCC(=O)NC%10=O)C(=O)C9=C8)CC7)CC6)CC5)=C4)C3=C2)[C@@H](C)N2N=NN=C2N1C	C50H59N15O5	LRRK2	Q5S007	CRBN	WO-2021194878-A1
TPD-E1VB0L	SCHEMBL23860663	SCHEMBL23860663; SCHEMBL29450421	C/C1=C(\C(=O)NC2=CC=C3NN=C(C4=CC=NC(N5CCN(CCCN6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)CC5)=C4)C3=C2)[C@@H](C)N2N=NN=C2N1C	C44H49N15O5	LRRK2	Q5S007	CRBN	WO-2021194878-A1
TPD-E2TCJT	SCHEMBL23860621	SCHEMBL23860621; SCHEMBL29450410	C/C1=C(\C(=O)NC2=CC=C3NN=C(C4=CC=NC(N5CCN(CC6CN(C7CCN(C8=CC9=C(C=C8)C(=O)N(C8CCC(=O)NC8=O)C9=O)CC7)C6)CC5)=C4)C3=C2)[C@@H](C)N2N=NN=C2N1C	C46H51N15O5	LRRK2	Q5S007	CRBN	WO-2021194878-A1
TPD-E2YK33	SCHEMBL23860601	SCHEMBL23860601; SCHEMBL29450405	CC1=C(C(=O)NC2=CC=C3NN=C(C4=CC=NC(N5C[C@@H](C)N(CCOCCN6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)[C@@H](C)C5)=C4)C3=C2)CN2N=NN=C2N1C	C46H53N15O6	LRRK2	Q5S007	CRBN	WO-2021194878-A1
TPD-E6O531	SCHEMBL23860596	SCHEMBL23860596; SCHEMBL29450399	C/C1=C(\C(=O)NC2=CC=C3NN=C(C4=CC=NC(N5C[C@@H](C)N(CCN6CCN(C7=CC=C8C(=O)N(C9CCC(=O)NC9=O)C(=O)C8=C7)CC6)[C@@H](C)C5)=C4)C3=C2)CN2N=NN=C2N1C	C44H49N15O5	LRRK2	Q5S007	CRBN	WO-2021194878-A1
TPD-EBPGAT	SCHEMBL30085081	SCHEMBL30085081	C=CC(=O)N1CCN(C2=C3C=C(Cl)C(C4=C5C=CC=CC5=CC(O)=C4)=C(F)C3=NC(OCCN3CCC(C)(COCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)N[C@@H](C)C4=CC=C(C5=C(C)N=CS5)C=C4)C(C)(C)C)CC3)=N2)C[C@@H]1CC#N	C61H70ClFN10O8S	KRAS G12C	P01116	VHL	WO-2021207172-A1
TPD-ECGPPX	SCHEMBL30085061	SCHEMBL30085061	C=CC(=O)N1CCN(C2=C3C=C(Cl)C(C4=C5C=CC=CC5=CC(O)=C4)=C(F)C3=NC(OCCN3CCC(F)(COCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)N[C@@H](C)C4=CC=C(C5=C(C)N=CS5)C=C4)C(C)(C)C)CC3)=N2)C[C@@H]1CC#N	C60H67ClF2N10O8S	KRAS G12C	P01116	VHL	WO-2021207172-A1
TPD-EE5MZK	SCHEMBL30085055	SCHEMBL30085055	C=CC(=O)N1CCN(C2=C3C=C(Cl)C(C4=C5C=CC=CC5=CC(O)=C4)=C(F)C3=NC(O[C@H](C)CN3CCC(COCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)N[C@@H](C)C4=CC=C(C5=C(C)N=CS5)C=C4)C(C)(C)C)CC3)=N2)C[C@@H]1CC#N	C61H70ClFN10O8S	KRAS G12C	P01116	VHL	WO-2021207172-A1
TPD-EGJE5G	SCHEMBL29521654	SCHEMBL29521654	NC1=NC=C(C2=CN(C3CCN(CC4CCN(C5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)CC4)CC3)N=C2)N=C1C(=O)O[C@@H](C(=O)NC1=CC=C(F)C=C1)C1=CC=CC=C1	C46H45FN10O7	MLKL	Q8NB16	CRBN	WO-2022065962-A1
TPD-EGKPH9	SCHEMBL29521794	SCHEMBL29521794	NC1=C(C(=O)O[C@@H](C(=O)NC2=CC=C(F)C=C2)C2=CC=CC=C2)N=C(C2=CN(C3CCN(C(=O)C4CCN(C(=O)COC5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)CC4)CC3)N=C2)C=N1	C48H45FN10O10	MLKL	Q8NB16	CRBN	WO-2022065962-A1
TPD-EZUD7F	SCHEMBL29521812	SCHEMBL29521812	NC1=C(C(=O)O[C@@H](C(=O)NC2=CC=C(F)C=C2)C2=CC=CC=C2)N=C(C2=CN(C3CCN(C(=O)C4CCN(C5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)CC4)CC3)N=C2)C=N1	C46H43FN10O8	MLKL	Q8NB16	CRBN	WO-2022065962-A1
TPD-F0URNS	SCHEMBL29522155	SCHEMBL29522155	NC1=C(C(=O)O[C@@H](C(=O)NC2=CC=C(F)C=C2)C2=CC=CC=C2)N=C(C2=CN(C3CCN(CCCN4CCN(C(=O)COC5=C/C=C6/C(=O)N(C7CCC(=O)NC7=O)C(=O)/C6=C\5)CC4)CC3)N=C2)C=N1	C49H50FN11O9	MLKL	Q8NB16	CRBN	WO-2022065962-A1
TPD-F1PPT3	WO-2022068933-A1_JA-189	.	O=C1CCC(N2C(=O)C3=CC=C(NCCCCCC(=O)N4CCC(C5C=C(C6=NC7=C(C8=CC(F)=C(CN9CCOCC9)C(F)=C8)C=CC=C7N=C6)C=N5)CC4)C=C3C2=O)C(=O)N1	C47H48F2N8O6	TYK2	P29597	CRBN	WO-2022068933-A1
TPD-F2934C	CHEMBL4747645	CHEMBL4747645; SCHEMBL22512126	CS(=O)(=O)C1=CC=C(C2=CC=CC3=NC(NC4=CC=C(N5CCN(CC(=O)NCCCCCCCCNC6=C/C=C7\C(=O)N(C8CCC(=O)NC8=O)C(=O)\C7=C\6)CC5)C=C4)=NN23)C=C1	C46H52N10O7S	TYK2	P29597	CRBN	WO-2022068933-A1
TPD-F5FVI3	CHEMBL4786620	CHEMBL4786620; SCHEMBL22512372	CS(=O)(=O)C1=CC=C(C2=CC=C/C3=N/C(NC4=CC=C(N5CCN(CC(=O)NCCCCCCCNC6=CC=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=C6)CC5)C=C4)=N\N23)C=C1	C45H50N10O7S	TYK2	P29597	CRBN	WO-2022068933-A1
TPD-F6RN6J	WO-2022068933-A1_JA-322	.	O=C1CCC(N2C(=O)C3=C(C=C(NCCCCCC(=O)N4CCC(N5C=C(C6=CN=C7C=CC=C(C8=CC(F)=C(CO)C(F)=C8)C7=N6)C=N5)CC4)C=C3)C2=O)C(=O)N1	C42H40F2N8O6	TYK2	P29597	CRBN	WO-2022068933-A1
TPD-FI1G21	WO-2022068933-A1_JA-323	.	O=C1CCC(N2C(=O)C3=C(C=C(NCCCCCC(=O)N4CCC(N5C=C(C6=CN=C7C=CC=C(C8=CC(F)=C(CN9CCC(O)CC9)C(F)=C8)C7=N6)C=N5)CC4)C=C3)C2=O)C(=O)N1	C47H49F2N9O6	TYK2	P29597	CRBN	WO-2022068933-A1
TPD-FR2WES	SCHEMBL29961650	SCHEMBL29961650	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC(=O)NCCCCC#CC3=CC=CC(CN4C5=C(C(=N)N([C@H]6CC[C@H](O)CC6)/C=N\5)C(C5=CC=CC=C5)=C4C4=CC=CC=C4)=C3)C(C)(C)C)C=C2)SC=N1	C68H81N9O6S	eEF1A2	Q05639	VHL	WO-2022159650-A1
TPD-FRU3Y7	SCHEMBL29961543	SCHEMBL29961543	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCCC(=O)NCCCCC#CC3=CC=CC(CN4C5=C(C(=N)N([C@H]6CC[C@H](O)CC6)C=N5)/C(C5=CC=CC=C5)=C\4C4=CC=CC=C4)=C3)C(C)(C)C)C=C2)SC=N1	C69H83N9O6S	eEF1A2	Q05639	VHL	WO-2022159650-A1
TPD-FS1E8D	SCHEMBL29961306	SCHEMBL29961306	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCCCC(=O)NCCCCC#CC3=CC=CC(CN4C5=C(C(=N)N([C@H]6CC[C@H](O)CC6)/C=N\5)C(C5=CC=CC=C5)=C4C4=CC=CC=C4)=C3)C(C)(C)C)C=C2)SC=N1	C70H85N9O6S	eEF1A2	Q05639	VHL	WO-2022159650-A1
TPD-FU6I4W	WO-2022228576-A1_30	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCN3CCC[C@H]3COC3=N/C4=C(F)C(C5=C/C(O)=C\C6=C5C=CC=C6)=C(Cl)C=C4/C(N4CC5CCC(C4)N5)=N\3)C(C)(C)C)C=C2)SC=N1	C54H61ClFN9O6S	KRAS G12D	P01116	VHL	WO-2022228576-A1
TPD-FVGQX1	WO-2022228576-A1_31	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCN3CCC[C@H]3COC3=N/C4=C(F)C(C5=C/C(O)=C\C6=C5C=CC=C6)=C(Cl)C=C4/C(N4CC5CCC(C4)N5)=N\3)C(C)(C)C)C=C2)SC=N1	C55H63ClFN9O6S	KRAS G12D	P01116	VHL	WO-2022228576-A1
TPD-FW0XJQ	WO-2022228576-A1_32	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCOCCCCN3CCC[C@H]3COC3=N/C4=C(C=C(Cl)C(C5=C/C(O)=C\C6=C5C=CC=C6)=C4F)/C(N4CC5CCC(C4)N5)=N\3)C(C)(C)C)C=C2)SC=N1	C59H71ClFN9O7S	KRAS G12D	P01116	VHL	WO-2022228576-A1
TPD-G1MD3X	WO-2022228576-A1_33	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCN3CCC[C@H]3COC3=N/C4=C(F)C(C5=C/C(O)=C\C6=C5C=CC=C6)=C(Cl)C=C4/C(N4CC5CCC(C4)N5)=N\3)C(C)(C)C)C=C2)SC=N1	C58H69ClFN9O6S	KRAS G12D	P01116	VHL	WO-2022228576-A1
TPD-G24IDJ	SCHEMBL27172848	SCHEMBL27172848	CN(CCOCCN1CCN(C2=C/C3=C(\C=C/2)C(=O)N(C2CCC(=O)NC2=O)C3)CC1)CCOC1=CC=C(O/C2=C(C3=CC=C(S(C)(=O)=O)C=C3)/C=C\C3=C2C=CC(O)=C3)C=C1	C47H51N5O9S	ER	P03372	CRBN	WO-2022237904-A1
TPD-G2V4A8	SCHEMBL27172854	SCHEMBL27172854	CS(=O)(=O)C1=CC=C(C2=C(\OC3=CC=C(N4CCN(CCCCCOCC(=O)N5CCN(C6=CC7=C(C=C6)C(=O)N(C6CCC(=O)NC6=O)C7)CC5)CC4)C=C3)C3=C(C=C(O)C=C3)/C=C\2)C=C1	C51H56N6O9S	ER	P03372	CRBN	WO-2022237904-A1
TPD-G6U5YF	SCHEMBL27172824	SCHEMBL27172824	CCN(CCOC1=CC=C(O/C2=C(C3=CC=C(S(C)(=O)=O)C=C3)/C=C\C3=C2C=CC(O)=C3)C=C1)CC(=O)N1CCN(C2=CC=C3C(=O)N(C4CCC(=O)NC4=O)CC3=C2)CC1	C46H47N5O9S	ER	P03372	CRBN	WO-2022237904-A1
TPD-G7ZIAG	SCHEMBL27172766	SCHEMBL27172766	CCN(CCOC1=CC=C(O/C2=C(C3=CC=C(S(C)(=O)=O)C=C3)/C=C\C3=C2C=CC(O)=C3)C=C1)CC(=O)N1CCN(C2=CC=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=C2)CC1	C46H45N5O10S	ER	P03372	CRBN	WO-2022237904-A1
TPD-G9YEKE	SCHEMBL27172880	SCHEMBL27172880	C[C@@H]1CN(CCOC2=CC=C(OC3=C(C4=CC=C(S(C)(=O)=O)C=C4)C=CC4=CC(O)=CC=C43)C=C2)[C@@H](C)CN1CCOCC(=O)N1CCN(C2=C/C=C3/C(=O)N(C4CCC(=O)NC4=O)C/C3=C\2)CC1	C52H58N6O10S	ER	P03372	CRBN	WO-2022237904-A1
TPD-GGV3TA	SCHEMBL26089936	SCHEMBL26089936; SCHEMBL30384112	CC/C1=C/C2=C(C=C(CN3CCN(C4=CC=C(C(=O)NC5CCN(C6=C/C7=C(\C=C/6)C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)N=C4)CC3)C=N2)NC1=O	C39H41N9O6	PARP1	P09874	CRBN	WO-2023066363-A1
TPD-GKD03E	SCHEMBL26090013	SCHEMBL26090013; SCHEMBL30383697	CCC1=CC2=C(C=C(CN3CCN(C4=CC=C(C(=O)NC5=CN(C6CCN(C7=C/C8=C(\C=C/7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)N=C5)N=C4)CC3)C=N2)NC1=O	C42H43N11O6	PARP1	P09874	CRBN	WO-2023066363-A1
TPD-GR1Y92	SCHEMBL26091571	SCHEMBL26091571; SCHEMBL30384121	CCC1=CC2=C(C=C(CN3CC=C(C4=CC=C(C(=O)NC5=CN(C6CCN(C7=C/C8=C(\C=C/7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)N=C5)N=C4)CC3)C=N2)NC1=O	C43H42N10O6	PARP1	P09874	CRBN	WO-2023066363-A1
TPD-GU7P55	SCHEMBL25474010	SCHEMBL25474010; SCHEMBL30400887	O=C1CCC(N2CC3=C(C=CC(C(=O)NCCCCCCCNC(=O)C4=C/C5=C(\C(NC(=O)C6=CC(C(F)(F)F)=CC(F)=C6)=C/4)[C@@H](C4=CC(F)=CC=C4Cl)NC5=O)=C3)C2=O)C(=O)N1	C44H38ClF5N6O7	PI3Kalpha	P42336	CRBN	WO-2023081759-A1
TPD-GX8I04	SCHEMBL25171971	SCHEMBL25171971; SCHEMBL30400656	CC1=CC=CC=C1NC1=NC=C(C(=O)NCCCC#CC2=C/C3=C(\C=C/2)C(=O)N(C2CCC(=O)NC2=O)C3)C=C1NC(=O)C1=CS/C2=C\C=C/C=C\12	C40H34N6O5S	PI3Kalpha	P42336	CRBN	WO-2023081759-A1
TPD-H17L2V	SCHEMBL25438593	SCHEMBL25438593; SCHEMBL30401440	CC1=CC=CC=C1NC1=NC=C(C(=O)NC2=CC=C(N3CCN(C4=C/C5=C(\C=C/4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)C=C2)C=C1NC(=O)C1=CSC2=CC=CC=C21	C45H38N8O6S	PI3Kalpha	P42336	CRBN	WO-2023081759-A1
TPD-H7U3X7	SCHEMBL25437480	SCHEMBL25437480; SCHEMBL30398994	O=C1CCC(N2C(=O)C3=C(/C=C(NCCCCCNC(=O)C4=CN=C(NC5=CC(F)=CC=C5Cl)C(NC(=O)C5=CSC6=CC=CC=C65)=C4)\C=C/3)C2=O)C(=O)N1	C39H33ClFN7O6S	PI3Kalpha	P42336	CRBN	WO-2023081759-A1
TPD-H83BE5	SCHEMBL24833209	SCHEMBL24833209; SCHEMBL30161152	CN1CCN(C2CC3CC2N(C2=NN=C(C(N)=O)C(NC4=CC=C(N5CCN(CC6CCN(C7=C/C8=C(\C=C/7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)C=C4)=N2)C3)C1=O	C43H51N13O6	BTK C481S	Q06187	CRBN	WO-2023274390-A1
TPD-HACQO3	SCHEMBL24833193	SCHEMBL24833193; SCHEMBL30161241	CN1CCN(C2CC3CC2N(C2=NN=C(C(N)=O)C(NC4=CC=C(C5CCN(C6CCN(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)C=C4)=N2)C3)C1=O	C43H50N12O6	BTK C481S	Q06187	CRBN	WO-2023274390-A1
TPD-HBOTK3	SCHEMBL24833701	SCHEMBL24833701	CN1CCN(C2CC3CC2N(C2=NN=C(C(N)=O)C(NC4=CC=C(N5CCC(N6CCN(CC#CC7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8)CC6)CC5)C=C4)=N2)C3)C1=O	C45H53N13O5	BTK C481S	Q06187	CRBN	WO-2023274390-A1
TPD-HHRU9Q	SCHEMBL24833098	SCHEMBL24833098; SCHEMBL30161123	CN1CCN(C2CC3CC2N(C2=NN=C(C(N)=O)C(NC4=CC=C(C5CCN(CC6CCN(C7=CC8=C(C=C7F)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)CC5)C=C4)=N2)C3)C1=O	C44H51FN12O6	BTK C481S	Q06187	CRBN	WO-2023274390-A1
TPD-HIAWHR	SCHEMBL24833335	SCHEMBL24833335; SCHEMBL30160788	CN1CCN(C2CC3CC2N(C2=NN=C(C(N)=O)C(NC4=CC=C(C5CCN(CC6CCN(C7=CC8=C(C=C7)CN(C7CCC(=O)NC7=O)C8=O)CC6)CC5)C=C4)=N2)C3)C1=O	C44H54N12O5	BTK C481S	Q06187	CRBN	WO-2023274390-A1
TPD-HL9L99	SCHEMBL27354433	SCHEMBL27354433; SCHEMBL30696678	CC1=C(C(=O)N2CCC3=C\C(C4=C(C)SC(NC(=O)CC5=CC=CC(OCCCN6CCN(C7=CC8=C(C=C7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)=C5)=N4)=C/C=C\32)C=CC=C1	C48H47N7O7S	Nrf2	Q16236	CRBN	WO-2024006742-A2
TPD-HLSZ8F	SCHEMBL27354502	SCHEMBL27354502; SCHEMBL30696666	CC1=C(C(=O)N2CCC3=C\C(C4=C(C)SC(NC(=O)CC5=CC=CC(OCCCCN6CCN(C7=C/C8=C(\C=C/7)C(=O)N(C7CCC(=O)NC7=O)C8=O)CC6)=C5)=N4)=C/C=C\32)C=CC=C1	C49H49N7O7S	Nrf2	Q16236	CRBN	WO-2024006742-A2
TPD-HPWBEN	SCHEMBL30696688	SCHEMBL30696688	CC1=C(C2=C/C=C3C(=C/2)\CCN\3C(=O)C2CC2)N=C(NC(=O)CC2=CC=C(F)C(OCCOCCNC3=CC4=C(C=C3)C(=O)N(C3CCC(=O)NC3=O)C4=O)=C2)S1	C41H39FN6O8S	Nrf2	Q16236	CRBN	WO-2024006742-A2
TPD-HT07UU	WO-2024054591-A1_198	.	N#CC1=C(OC2=C/C3=C(\C=C/2)N=CN(C2=CC=C(N4CC(CN5CCN(C6CCN(C7=C/C8=C(\C=C/7)C(=O)N(C7CCC(=O)NC7=O)C8)CC6)CC5)C4)C=C2)C3=O)C(F)=CC=C1NS(=O)(=O)N1CC[C@@H](F)C1	C51H53F2N11O7S	ARAF;BRAF;CRAF	P10398/P15056/P04049	CRBN	WO-2024054591-A1
TPD-HXJ0J3	SCHEMBL27194448	SCHEMBL27194448; SCHEMBL30873170	O=C1CCC(N2CC3=C(/C=C\C(N4CCC(CN5CCN(C6=CC=C(N7/C=N\C8=C(C=C(OC9=C(Cl)C(NS(=O)(=O)N%10CC[C@@H](F)C%10)=CC=C9F)C=C8)C7=O)C=C6)CC5)CC4)=C/3)C2=O)C(=O)N1	C47H48ClF2N9O7S	ARAF;BRAF;CRAF	P10398/P15056/P04049	CRBN	WO-2024054591-A1
TPD-HZ1O71	SCHEMBL27194281	SCHEMBL27194281; SCHEMBL30873288	N#CC1=C(OC2=CC3=C(C=C2)/N=C\N(C2=CC=C(N4CCC5(CCN(CC6CCN(C7=C/C8=C(\C=C/7)C(=O)N([C@H]7CCC(=O)NC7=O)C8)CC6)CC5)CC4)C=C2)C3=O)C(F)=CC=C1NS(=O)(=O)N1CC[C@@H](F)C1	C53H56F2N10O7S	ARAF;BRAF;CRAF	P10398/P15056/P04049	CRBN	WO-2024054591-A1
TPD-HZ2VQ3	SCHEMBL27194422	SCHEMBL27194422; SCHEMBL30873164	N#CC1=C(OC2=CC3=C(C=C2)/N=C\N(C2=CC=C(N4CCC5(CCN(CC6CCN(C7=C/C8=C(\C=C/7)C(=O)N([C@@H]7CCC(=O)NC7=O)C8)CC6)CC5)CC4)C=C2)C3=O)C(F)=CC=C1NS(=O)(=O)N1CC[C@@H](F)C1	C53H56F2N10O7S	ARAF;BRAF;CRAF	P10398/P15056/P04049	CRBN	WO-2024054591-A1
TPD-I1KOG3	WO-2024083258-A1_222	.	C#CC1=CC=CC2=CC(O)=CC(C3CC4=C(CO3)C(N3CC5CCC(C3)N5)=NC(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(C)C=C6)CC7)CC5)CC3)=N4)=C12	C57H69N9O6	KRAS G12C	P01116	VHL	WO-2024083258-A1
TPD-I4AU8J	WO-2024083258-A1_223	.	C#CC1=CC=CC2=CC(O)=CC(C3CC4=C(CO3)/C(N3CC5CCC(C3)N5)=N\C(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(Cl)C=C6)CC7)CC5)CC3)=N/4)=C12	C56H66ClN9O6	KRAS G12C	P01116	VHL	WO-2024083258-A1
TPD-IABSWZ	WO-2024083258-A1_224	.	CCC1=CC=CC2=CC(O)=CC(C3CC4=C(CO3)/C(N3CC5CCC(C3)N5)=N\C(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(OC)C=C6)CC7)CC5)CC3)=N/4)=C21	C57H73N9O7	KRAS G12C	P01116	VHL	WO-2024083258-A1
TPD-IM1IDO	WO-2024083258-A1_225	.	CCC1=CC=CC2=CC(O)=CC(C3CC4=C(CO3)/C(N3CC5CCC(C3)N5)=N\C(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(C)C=C6)CC7)CC5)CC3)=N/4)=C21	C57H73N9O6	KRAS G12C	P01116	VHL	WO-2024083258-A1
TPD-ITVPSO	WO-2024083258-A1_226	.	CCC1=CC=CC2=CC(O)=CC(C3CC4=C(CO3)/C(N3CC5CCC(C3)N5)=N\C(OCC3(CN5CCN(CC6CCC7(CC6)CCN(C(=O)C6=CC(N8CCC(=O)NC8=O)=C(Cl)C=C6)CC7)CC5)CC3)=N/4)=C21	C56H70ClN9O6	KRAS G12C	P01116	VHL	WO-2024083258-A1
TPD-IVWCKU	SCHEMBL27301011	SCHEMBL27301011; SCHEMBL30941902	CC/C1=C(F)/C=C\C2=C1C(C1=C(\F)C3=C(\C=N/1)C(N1CC4CCC(C1)N4)=NC(OCC1(CN4CCC5(CC4)CC(N4CCN(C6=C/C7=C(\C=C/6)C(=O)N([C@H]6CCC(=O)NC6=O)C7)CC4)C5)CC1)=N3)=CC(O)=C2	C55H62F2N10O5	KRAS G12D	P01116	CRBN	WO-2024118960-A1
TPD-IX474L	SCHEMBL27301013	SCHEMBL27301013; SCHEMBL30942034	O=C1CC[C@H](N2CC3=C(/C=C\C(N4CCN(C5CC6(CCN(CC7(COC8=N/C9=C(C=NC(C%10=CC(O)=CC%11=C%10C(F)=C(F)C=C%11)=C9F)/C(N9CC%10CCC(C9)N%10)=N\8)CC7)CC6)C5)CC4)=C/3)C2=O)C(=O)N1	C53H57F3N10O5	KRAS G12D	P01116	CRBN	WO-2024118960-A1
TPD-J899AV	SCHEMBL27301018	SCHEMBL27301018; SCHEMBL30941894	CCC1=CC=CC2=C1/C(C1=C(F)C3=C(C=N1)/C(N1CC4CCC(C1)N4)=N\C(OCC1(CN4CC5(CCC(N6CCN(C7=C/C8=C(\C=C/7)C(=O)N([C@H]7CCC(=O)NC7=O)C8)CC6)CC5)C4)CC1)=N/3)=C\C(O)=C/2	C55H63FN10O5	KRAS G12D	P01116	CRBN	WO-2024118960-A1
TPD-JATL2Y	SCHEMBL29320168	SCHEMBL29320168	CN1C(=O)N(C2CCC(=O)NC2=O)C2=C/C=C(CCN3CCC(CC4=CC5=NN([C@H]6CC[C@H](CNC(=O)C7=CC(F)=C(O)C(F)=C7F)CC6)C=C5C=C4)C(F)(F)C3)/C=C\21	C42H44F5N7O5	HSD17B13	Q7Z5P4	CRBN	WO-2024127297-A1
TPD-JCWCPL	SCHEMBL29320179	SCHEMBL29320179	CN1C(=O)N(C2CCC(=O)NC2=O)C2=C1/C=C(CCCN1CC(F)(F)CC3(CCN(C4=CC5=NN([C@H]6CC[C@H](CNC(=O)C7=C(F)C(F)=C(O)C(F)=C7)CC6)C=C5C=C4)C3=O)C1)\C=C/2	C45H47F5N8O6	HSD17B13	Q7Z5P4	CRBN	WO-2024127297-A1
TPD-JEXENS	SCHEMBL29320184	SCHEMBL29320184	CN1C(=O)N(C2CCC(=O)NC2=O)C2=C1/C=C(CCCN1CCN(C3=NN=C(C4=NC([C@]56CC[C@](CNC(=O)C7=C(F)C(F)=C(O)C(F)=C7)(CC5)CC6)=NO4)C=C3)CC1)\C=C/2	C42H45F3N10O6	HSD17B13	Q7Z5P4	CRBN	WO-2024127297-A1
TPD-JFC3EN	SCHEMBL29320191	SCHEMBL29320191	CN1C(=O)N(C2CCC(=O)NC2=O)C2=C1/C=C(CCCN1CCN(C3=NC=C(C4=NC([C@]56CC[C@](CNC(=O)C7=C(F)C(F)=C(O)C(F)=C7)(CC5)CC6)=NO4)C=N3)CC1)\C=C/2	C42H45F3N10O6	HSD17B13	Q7Z5P4	CRBN	WO-2024127297-A1
TPD-JFOLOC	WO-2025021075-A1_LLC0635	.	CC1(NC(=O)C2=CC=C(NC(=O)C3=CC=C(CN(C(=O)C4=C/C5=C(\C=C/4)NC(=O)CO5)C4CC4)C=C3)C=C2)CCN(C2=C/C3=C(\C=C/2)C(=O)N(C2CCC(=O)NC2=O)C3=O)CC1	C46H43N7O9	NSD2;NSD1;NSD3;KLK3;NKX3.1	O96028/Q96L73/Q9BZ95/P07288/Q99801	CRBN	WO-2025021075-A1
TPD-JV6286	SCHEMBL31337874	SCHEMBL31337874	O=C1CCC(N2C(=O)C3=C(C2=O)/C(NCCNC(=O)C2=CC=C(CN(C(=O)C4=C/C5=C(\C=C/4)NC(=O)CO5)C4CC4)C=C2)=C\C=C/3)C(=O)N1	C35H32N6O8	NSD2;NSD1;NSD3;KLK3;NKX3.1	O96028/Q96L73/Q9BZ95/P07288/Q99801	CRBN	WO-2025021075-A1
TPD-JW93KH	SCHEMBL31337881	SCHEMBL31337881	O=C1CCC(N2C(=O)C3=C(C2=O)/C(NCCCCNC(=O)C2=CC=C(CN(C(=O)C4=C/C5=C(\C=C/4)NC(=O)CO5)C4CC4)C=C2)=C\C=C/3)C(=O)N1	C37H36N6O8	NSD2;NSD1;NSD3;KLK3;NKX3.1	O96028/Q96L73/Q9BZ95/P07288/Q99801	CRBN	WO-2025021075-A1
TPD-K7QHEH	WO-2025021075-A1_LLC0638	.	O=C1CCC(N2C(=O)C3=C(C2=O)C(NCCCCCCNC(=O)C2=CC=C(CN(C(=O)C4=C/C5=C(\C=C/4)NC(=O)CO5)C4CC4)C=C2)=CC=C3)C(=O)N1	C39H40N6O8	NSD2;NSD1;NSD3;KLK3;NKX3.1	O96028/Q96L73/Q9BZ95/P07288/Q99801	CRBN	WO-2025021075-A1
TPD-KCR4U8	WO-2025021075-A1_LLC0639	.	O=C1CCC(N2C(=O)C3=C(C2=O)/C(NCCCCCCCCNC(=O)C2=CC=C(CN(C(=O)C4=C/C5=C(\C=C/4)NC(=O)CO5)C4CC4)C=C2)=C\C=C/3)C(=O)N1	C41H44N6O8	NSD2;NSD1;NSD3;KLK3;NKX3.1	O96028/Q96L73/Q9BZ95/P07288/Q99801	CRBN	WO-2025021075-A1
TPD-KD5MJH	SCHEMBL31287020	SCHEMBL31287020	CC1=C(C2=CC(OCCCCCCCCC(=O)NC3=NC4=C/C=C(C5=CC6=C(N=C5)OCCN6C(=O)OC5CCCCC5)/C=C\4S3)=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)C3(F)CC3)C(C)(C)C)C=C2)SC=N1	C56H69FN8O9S2	RIPK1	Q13546	VHL	WO-2025022093-A1
TPD-KMC9J8	SCHEMBL31287012	SCHEMBL31287012	CC1=NC=C(C2=C/C3=C(\C=C/2)N=C(NC(=O)CCCCCCCCCCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(C4=C(C)N=CS4)C=C2)C(C)(C)C)S3)C=C1NC(=O)OC12CCC(CC1)CC2	C56H72N8O7S2	RIPK1	Q13546	VHL	WO-2025022093-A1
TPD-KUFE7T	SCHEMBL31287103	SCHEMBL31287103	CC1=NC=C(C2=CC3=C(C=C2)/N=C(/NC(=O)CCCCCCCCCCC(=O)N[C@H](C(=O)N2C[C@H](O)C[C@H]2C(=O)NCC2=CC=C(C4=C(C)N=CS4)C=C2)C(C)(C)C)S3)N=C1NC(=O)OC(C)C	C50H65N9O7S2	RIPK1	Q13546	VHL	WO-2025022093-A1
TPD-KUFNCB	PD155841	PD155841	O=C1CCC(N2CC3=C(NC(=O)COCCOCCNCCNC4=NON=C4/C(=N/O)NC4=CC(Br)=C(F)C=C4)/C=C/C=C\3C2=O)C(=O)N1	C30H33BrFN9O8	IDO1	P14902	CRBN	CN-111217804-A
TPD-L0H65K	CN-111303133-A_1	.	CCN(C1=C(C)C(C(=O)NCC2=C(C)C=C(C)NC2=O)=CC(C2=CC=C(CN3CCN(C(=O)CCCC4=CN(CCOCCNC5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)N=N4)CC3)C=C2)=C1)C1CCOCC1	C57H69N11O9	EZH2	Q15910	CRBN	CN-111303133-A
TPD-LDS4KN	DA-PROTAC	DA-PROTAC; 2488660-12-2; N-(2-Bromo-4,6-difluorophenyl)-3-(2-(3-(2-((1-((2S,4R)-4-hydroxy-2-((4-(4-methylthiazol-5-yl)benzyl)carbamoyl)pyrrolidin-1-yl)-3,3-dimethyl-1-oxobutan-2-yl)amino)-2-oxoethoxy)propoxy)acetamido)-6,7-dihydro-5H-cyclopenta[b]thieno[3,2-e]pyridine-2-carboxamide; orb1942160; YQF1969; DA-62669; HY-147373; CS-0567671; EN300-44826004; N-(2-bromo-4,6-difluorophenyl)-6-(2-{3-[({1-[(2S,4R)-4-hydroxy-2-({[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl}carbamoyl)pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl}carbamoyl)methoxy]propoxy}acetamido)-4-thia-2-azatricyclo[7.3.0.0,3,7]dodeca-1,3(7),5,8-tetraene-5-carboxamide; N-(2-bromo-4,6-difluorophenyl)-6-[[2-[3-[2-[[1-[(2S,4R)-4-hydroxy-2-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methylcarbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]amino]-2-oxoethoxy]propoxy]acetyl]amino]-4-thia-2-azatricyclo[7.3.0.03,7]dodeca-1,3(7),5,8-tetraene-5-carboxamide	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)C(NC(=O)COCCCOCC(=O)NC3=C(C(=O)NC4=C(Br)C=C(F)C=C4F)SC4=NC5=C(C=C43)CCC5)C(C)(C)C)C=C2)SC=N1	C46H50BrF2N7O8S2	ATOX1;CCS	O00244/O14618	VHL	CN-111471054-A
TPD-LDSQRR	CN-111646977-A_PP2	.	CC1=CN(C2=CC=C(OCCOCCN3C=C(CO/C4=C/C=C\C5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)N=N3)C=C2)C(=O)C=C1	C32H30N6O8	TGFBR1	P36897	CRBN	CN-111646977-A
TPD-LGTKIE	SCHEMBL28514080	SCHEMBL28514080	COC1=NC=C(C2=CC3=C(C=C2)/N=C\C=C/3C2=CC=C(OCCOCCNC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)C=C2)C=C1NS(=O)(=O)C1=CC=C(F)C=C1F	C44H36F2N6O9S	PI3K;mTOR	P42336/P42345	CRBN	CN-112341434-B
TPD-LM604T	CN-112430229-A_1-2	.	NC(=O)C1=CC=CC2=CN(C3=CC=C([C@@H]4CCCN(C(=O)CCOCCNC5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)C4)C=C3)NC21	C37H39N7O7	PARP1	P09874	CRBN	CN-112430229-A
TPD-LMTAZH	CHEMBL5090540	CHEMBL5090540; PD172807	NC1=NC=C(C2=CC=C(S(=O)(=O)N3CCN(CC4=CN(CCOCCOCCN/C5=C/C=C\C6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)N=N4)CC3)C=C2)N=C1C(=O)NC1=CC=CN=C1	C42H45N13O9S	GSK3A;GSK-3beta	P49840/P49841	CRBN	CN-113248473-B
TPD-LUCO8J	CN-113512035-A_8b	.	CCOC(=O)C1=C(CN2CCN(C(=O)CCCCCNC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)CC2)NC(C2=NC=CS2)=NC1C1=C(Br)C=C(F)C=C1	C40H42BrFN8O7S	HBV	P03146	CRBN	CN-113512035-A
TPD-LW2EMJ	CHEMBL4849375	CHEMBL4849375; PD172056	N/C1=C(\C2=NC3=C(/C=C\C(N4CCN(C(=O)CCCC#CC5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)CC4)=C/3)N2)C(=O)NC2=C1C(F)=CC=C2	C39H33FN8O6	FLT3-ITD	P36888	CRBN	CN-113527263-A
TPD-M2J57C	CN-113527270-B_PROTAC-1	.	CC(C)OC1=CC(OC(C)C)=C(C2=N[C@@H](C3=CC=C(Cl)C=C3)[C@@H](C3=CC=C(Cl)C=C3)N2C(=O)N2CCN(C(=O)COCCOC3=CC=C([C@@](O)(C4=C/C5=C(\C=C/4)OCO5)C4CCN(C(=O)OC5=CC=C([N+](=O)[O-])C=C5)CC4)C=C3)CC2)C=C1	C62H64Cl2N6O13	MGLL	Q99685	MDM2	CN-113527270-B
TPD-M3TMC4	CN-113861213-A_TSM-1	.	[H][C@@]12C[C@@H](O)C3[C@@]45O[C@]4([H])C[C@@H](C4=COC=C4)[C@]5(C)[C@@H](OC(C)=O)C(=O)[C@]3([H])[C@]13CO[C@@H](OC(=O)CCC(=O)N1CC(CN/C4=C/C=C\C5=C4C(=O)N(C4CCC(=O)NC4=O)C5)C1)[C@@]2(C)[C@H](OC(C)=O)C[C@@H]3O	C50H58N4O16	STAT3	P40763	CRBN	CN-113861213-A
TPD-M9B7FT	SCHEMBL28732616	SCHEMBL28732616	O=C1CCC(N2C(=O)C3=CC=C(N4CCC(CN5CCC(C(=O)N6CCN(C(=O)C7=C(F)C=CC(C/C8=N/NC(=O)C9=C8C=CC=C9)=C7)CC6)CC5)CC4)C=C3C2=O)C(=O)N1	C45H47FN8O7	PARP1;PARP2	P09874/Q9UGN5	CRBN	CN-114181196-A
TPD-MMHVXJ	CN-114409638-A_11a	.	O=C1CCC(N2C(=O)C3=C(C2=O)/C(NCC2=CN(CCOC4=CC=C(CN5C=CC6=C/C=C(C(=O)NO)\C=C\65)C=C4)N=N2)=C\C=C/3)C(=O)N1	C34H30N8O7	HDAC8	Q9BY41	CRBN	CN-114409638-A
TPD-MOEJB1	CN-114621310-A_1-1	.	[H][C@@]12C[C@](C)(C(=O)NCCOCCNC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)CC[C@@]1(C)CC[C@]1(C)C3=CC=C4C(=CC(=O)C(O)=C4C)[C@]3(C)CC[C@@]21C	C46H56N4O8	PRDX2	P32119	CRBN	CN-114621310-A
TPD-MOWGC5	CN-114650989-A_25	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCOCCN3C=C(CNC(=O)C4=CC(NC5=NNC(C6CC6)=C5)=NC(NC5=CC=C(CC#N)C=C5)=N4)N=N3)C(C)(C)C)C=C2)SC=N1	C49H57N15O6S	CHEK1;CHK2	O14757/O96017	VHL	CN-114650989-A
TPD-MRCRFQ	SCHEMBL29175252	SCHEMBL29175252	O=C1CCC(N2C(=O)C3=CC=CC(OCCOCCC(=O)N4CCN(CCCN5C6=CC(Cl)=CC=C6SC6=C5C=CC=C6)CC4)=C3C2=O)C(=O)N1	C37H38ClN5O7S	S100A4	P26447	CRBN	CN-114853751-A
TPD-MYWLEB	CN-114890995-A_SI-3	.	C#CCOC1=CC(O)=C2C(=O)C(OCC(=O)NCCCCCC(=O)N/C3=C/C=C\C4=C3CN(C3CCC(=O)NC3=O)C4=O)=C(C3=CC=C(OC)C=C3)OC2=C1CC=C(C)C	C45H46N4O11	AFF4;GRIA3;NLRP13;NMD3;TECPR2;TMEM18;ARHGEF3;BTN3A3;CCM2;CCNDBP1;CD63;CRIPT;CUTC;FLYWCH2;FSD1;HAUS8;HDAC3;INF2;KDM7A;MCL-1;MRPL2;MTHFS;NAB2;NDUFA13;NDUFS2;P4HA1;PAXX;PDK3;PSEN1;RNASET2;SFXN4;TAF6L;TXNIP;UPRT;ZNF354A	Q9UHB7/P42263/Q86W25/Q96D46/O15040/Q96B42/Q9NR81/O00478/Q9BSQ5/O95273/P08962/Q9P021/Q9NTM9/Q96CP2/Q9BTV5/Q9BT25/O15379/Q27J81/Q6ZMT4/Q07820/Q5T653/P49914/P32505/Q9P0J0/O75306/P13674/Q9BUH6/Q15120/P49768/O00584/Q6P4A7/Q9Y6J9/Q9H3M7/Q96BW1/O60765	CRBN	CN-114890995-A
TPD-N9AVJM	CN-114890995-A_SI-4	.	C#CCOC1=CC(O)=C2C(=O)/C(OCCCC(=O)NCCCCCC(=O)N/C3=C/C=C\C4=C3CN(C3CCC(=O)NC3=O)C4=O)=C(/C3=CC=C(OC)C=C3)OC2=C1CC=C(C)C	C47H50N4O11	AFF4;GRIA3;NLRP13;NMD3;TECPR2;TMEM18;ARHGEF3;BTN3A3;CCM2;CCNDBP1;CD63;CRIPT;CUTC;FLYWCH2;FSD1;HAUS8;HDAC3;INF2;KDM7A;MCL-1;MRPL2;MTHFS;NAB2;NDUFA13;NDUFS2;P4HA1;PAXX;PDK3;PSEN1;RNASET2;SFXN4;TAF6L;TXNIP;UPRT;ZNF354A	Q9UHB7/P42263/Q86W25/Q96D46/O15040/Q96B42/Q9NR81/O00478/Q9BSQ5/O95273/P08962/Q9P021/Q9NTM9/Q96CP2/Q9BTV5/Q9BT25/O15379/Q27J81/Q6ZMT4/Q07820/Q5T653/P49914/P32505/Q9P0J0/O75306/P13674/Q9BUH6/Q15120/P49768/O00584/Q6P4A7/Q9Y6J9/Q9H3M7/Q96BW1/O60765	CRBN	CN-114890995-A
TPD-N9LWAT	CN-114890995-A_SI-5	.	C#CCOC1=CC(O)=C2C(=O)C(OCCCCC(=O)NCCCCCC(=O)N/C3=C/C=C\C4=C3CN(C3CCC(=O)NC3=O)C4=O)=C(C3=CC=C(OC)C=C3)OC2=C1CC=C(C)C	C48H52N4O11	AFF4;GRIA3;NLRP13;NMD3;TECPR2;TMEM18;ARHGEF3;BTN3A3;CCM2;CCNDBP1;CD63;CRIPT;CUTC;FLYWCH2;FSD1;HAUS8;HDAC3;INF2;KDM7A;MCL-1;MRPL2;MTHFS;NAB2;NDUFA13;NDUFS2;P4HA1;PAXX;PDK3;PSEN1;RNASET2;SFXN4;TAF6L;TXNIP;UPRT;ZNF354A	Q9UHB7/P42263/Q86W25/Q96D46/O15040/Q96B42/Q9NR81/O00478/Q9BSQ5/O95273/P08962/Q9P021/Q9NTM9/Q96CP2/Q9BTV5/Q9BT25/O15379/Q27J81/Q6ZMT4/Q07820/Q5T653/P49914/P32505/Q9P0J0/O75306/P13674/Q9BUH6/Q15120/P49768/O00584/Q6P4A7/Q9Y6J9/Q9H3M7/Q96BW1/O60765	CRBN	CN-114890995-A
TPD-N9QMPR	CN-114920728-B_6c	.	O=C1CCC(N2CC3=C(NCCOCCN4C=C(CN5C(=O)/C(=C6/C(=O)NC7=C6/C=C\C=C/7)C6=C5C=CC=C6)N=N4)/C=C\C=C\3C2=O)C(=O)N1	C36H32N8O6	ATM	Q13315	CRBN	CN-114920728-B
TPD-NCCR6L	CN-115109047-B_GPX4-3	.	O=C1CC(N2C(=O)C3=C(C2=O)/C(NCCOCCOCCOCCN2C=C(COC4=CC=C(N(C(=O)CCl)C(C(=O)NCCC5=CC=CC=C5)C5=CC=CS5)C=C4Cl)N=N2)=C\C=C/3)CC(=O)N1	C46H48Cl2N8O10S	GPX4	P36969	CRBN	CN-115109047-B
TPD-NFD959	SCHEMBL26161762	SCHEMBL26161762	CC1=C(C2CCN(CC(=O)NCCOC3=C/C4=C(\C=C/3)OC=C4C3CCC(=O)NC3=O)CC2)C=C(OC(C)C)C(NC2=NC=C(Cl)C(NC3=CC=CC=C3S(=O)(=O)C(C)C)=N2)=C1	C45H52ClN7O8S	p-ALK;EML4-ALK	Q9UM73/Q9HC35	CRBN	CN-115380026-A
TPD-NLRITT	CN-115557965-A_22a	.	CC1=C(C2=CC=C([C@H](C)NC(=O)C3C[C@@H](O)CN3C(NC(=O)CCCOC3=CC=C(N(CC(F)(F)F)S(=O)(=O)C4CC5OC4C(C4=CC=C(N6C=CN=C6)C=C4)=C5C4=CC=C(O)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C55H60F3N7O8S2	CYP19A1	P11511	VHL	CN-115557965-A
TPD-NVPSEO	CN-115677815-A_1	.	CC1(C)CC[C@]2(C(=O)NCCCCCCOCCOCC(=O)N/C3=C/C=C\C4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC[C@]3(C)C(=CCC4[C@@]5(C)CC[C@H](O)C(C)(C)C5CC[C@]43C)C2C1	C53H76N4O9	PTPN1	P18031	CRBN	CN-115677815-A
TPD-NXJKZ0	CHEMBL5431842	CHEMBL5431842	C[C@@H]1CCC2[C@@H](C)[C@@H](OCCN(CCO[C@H]3O[C@@H]4O[C@@]5(C)CCC6[C@H](C)CCC([C@H]3C)[C@]64OO5)C(=O)CCCCNC3=C4\C(=O)N(C5CCC(=O)NC5=O)C(=O)\C4=C\C=C\3)O[C@@H]3O[C@@]4(C)CCC1[C@@]23OO4	C52H72N4O15	ETS1;ZFAND5;PCLAF	P14921/O76080/Q15004	CRBN	CN-115724850-B
TPD-NZG0PB	CN-116283915-A_1	.	CC1=CC(NC2=NC=C(Cl)C(NC3=CC=CC=C3S(=O)(=O)C(C)C)=N2)=C(OC(C)C)C=C1C1CCN(C(=O)COCCOCCOCCCCCCO/C2=C/C=C\C3=C2C(=O)N(C2CCC(=O)NC2=O)C3=O)CC1	C53H66ClN7O12S	EML4-ALK	Q9HC35	CRBN	CN-116283915-A
TPD-O20TOG	CN-116284202-A_B1	.	[H][C@]12CC[C@@]3([H])[C@@](C)(CC[C@@]4(C(=O)NCCC(=O)NC5=C6CN(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)CC[C@@H](C(=C)C)[C@@]43[H])[C@]1(C)CC[C@@]1([H])C(C)(C)C(=O)CC[C@]21C	C46H62N4O6	KDM5A	P29375	CRBN	CN-116284202-A
TPD-O2P395	CN-116375713-B_P1	.	COC1=C(NC2=NC3=C(C=N2)N(C)C(=O)C2=C(C=CC=C2)N3C)C=CC(C(=O)NC2CCN(C(=O)CC(=O)N[C@H](C(=O)N3C[C@H](O)CC3C(=O)N[C@@H](C)C3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)CC2)=C1	C52H61N11O8S	DCLK1	O15075	VHL	CN-116375713-B
TPD-O3GIKJ	CN-116425733-A_3	.	CC(C)(CNC(=O)CCC(=O)NCCOCCOCCOCCNC1=C/C2=C(\C=C/1)C(=O)N(C1CCC(=O)NC1=O)C2=O)CN(C(=O)CCl)C1CCS(=O)(=O)C1	C36H51ClN6O12S	Pin1	Q13526	CRBN	CN-116425733-A
TPD-OAJPRR	SCHEMBL29040424	SCHEMBL29040424	CN1C=C(N2C=NC3=C2/N=C(N2CCOCC2)\N=C/3NCC2=NC3=CC(Cl)=C(NCCOCCNC(=O)COC4=C/C=C5C(=C/4)\CCCN\5C(=O)CCl)C=C3N2)C=N1	C38H43Cl2N13O5	BUB1B;BUB1	O60566/O43683	DACF16	CN-116444494-A
TPD-OBTBOC	CN-116640123-A_4h1pm	.	COC1=CC=C(C2=N[C@H](C3=CC=C(Cl)C=C3)[C@H](C3=CC=C(Cl)C=C3)N2C(=O)N2CCN(CC(=O)NCCOCCN3C=C(COC4=CC(C(=O)N/N=C/C5=CC=C(O)C(O)=C5O)=CC=C4[N+](=O)[O-])N=N3)C(=O)C2)C(OC(C)C)=C1	C53H53Cl2N11O13	HK2	P52789	MDM2	CN-116640123-A
TPD-OCOT52	PROTAC ATR degrader-2	PROTAC ATR degrader-2; 3010273-12-5; orb2565426; HY-161615; CS-1054163	NC1=NC=C(C2=CC=C(C(=O)N3CCN(CCCCC(=O)NC4=C5CN(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)C=C2)N=C1C(=O)NC1=CC=CC=C1	C40H41N9O6	ATR	Q13535	CRBN	CN-117003736-B
TPD-OD0JLT	CN-117065022-A_279	.	N#CC1=CC=C(O[C@H]2CC[C@H](NC(=O)C3=CN=C(N4CCC(CN5CCC6(CC5)CN(C5=C/C=C7/C(=O)N(C8CCC(=O)NC8=O)C(=O)/C7=C\5)C6)CC4)N=N3)CC2)C=C1Cl	C43H47ClN10O6	PI3Kalpha	P42336	CRBN	CN-117065022-A
TPD-OE7DDU	SCHEMBL29160539	SCHEMBL29160539	O=C(COC1=CN=C(/C2=N/C3=CC(OC(F)(F)F)=CC=C3N2)C=C1)NCCCCNC(=O)COC1=C2\C(=O)N(C3CCC(=O)NC3=O)C(=O)\C2=C/C=C\1	C34H30F3N7O9	CBF尾鈥揝MMHC	P35749	CRBN	CN-117567434-A
TPD-OM6SRS	SCHEMBL29160533	SCHEMBL29160533	O=C(COC1=CN=C(C2=NC3=CC(OC(F)(F)F)=CC=C3N2)C=C1)NCCCCCCNC(=O)COC1=C2\C(=O)N(C3CCC(=O)NC3=O)C(=O)\C2=C/C=C\1	C36H34F3N7O9	CBF尾鈥揝MMHC	P35749	CRBN	CN-117567434-A
TPD-OMT5Y1	CN-117586230-B_EP-1226	.	COC(=O)C1=C(C2=C/C3=C(C=CN3)/C=C\2)C(C#CC2=CC=C(OC3CCN(CC4CCN(C5=CC=CC6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)C=C2)=CC=C1	C48H45N5O7	EBNA1	P03211	CRBN	CN-117586230-B
TPD-OOFF2U	CN-117586230-B_EP-1228	.	COC(=O)C1=C(C2=C/C3=C(C=CN3)/C=C\2)C(C#CC2=CC=C(OC3CCN(C4CCN(/C5=C/C=C\C6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)C=C2)=CC=C1	C47H43N5O7	EBNA1	P03211	CRBN	CN-117586230-B
TPD-ORB675	CN-117603190-A_1-1	.	CC(C)C1=CC(C(=O)N2CC3=CC=C(CN4CCN(CCC(=O)NC5=C6\C(=O)N(C7CCC(=O)NC7=O)C(=O)\C6=C/C=C\5)CC4)C=C3C2)=CC=C1O	C39H42N6O7	Hsp90 alpha	P07900	CRBN	CN-117603190-A
TPD-OT3U5G	PROTAC STAT3 degrader-3	PROTAC STAT3 degrader-3; HY-163502; CS-1049710	CN(CC(=O)NC1=CC=C(C(=O)NCCOCCNC2=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=CC=C2)C=C1)S(=O)(=O)C1=C(F)C(F)=C(F)C(F)=C1F	C33H29F5N6O9S	STAT3	P40763	CRBN	CN-117720443-A
TPD-OUZXCD	CN-117720515-B_1	.	O=C1CCC(N2C(=O)C3=C(C2=O)/C(OCCOCCOCCOCCOC(=O)C2=CC(O)=C(O)C(O)=C2)=C\C=C/3)C(=O)N1	C28H30N2O13	GSDMD;GSDME	P57764/O60443	CRBN	CN-117720515-B
TPD-OYJS5K	PD216539	PD216539	COC1=C(OC)C=C(/C2=C/NC3=C2C=C(C2=CC=C(N4CCN(C(=O)COC5=C/C=C6/C(=O)N(C7CCC(=O)NC7=O)C(=O)/C6=C\5)CC4)C=C2)C=N3)C=C1	C40H36N6O8	HPK1;LCK;MAP4K3;PCK胃;ITK	Q92918/P06239/Q8IVH8/Q04759/Q08881	CRBN	CN-117777125-A
TPD-OZLI75	CN-117777223-A_AREprotac	.	CCCC1=CN(CCCNC(=O)CCCC(=O)NC2=C3CN(C4CCC(=O)NC4=O)C(=O)C3=CC=C2)N=N1	C26H33N7O5	Nrf2	Q16236	CRBN	CN-117777223-A
TPD-P2O9B1	5-((2-(2,6-dioxopiperidin-3-yl)-1-oxoisoindolin-4-yl)amino)-5-oxopentyl (2r,4as,6as,12br,14as,14br)-10-hydroxy-2,4a,6a,9,12b,14a-hexamethyl-11-oxo-1,2,3,4,4a,5,6,6a,11,12b,13,14,14a,14b-tetradecahydropicene-2-carboxylate	5-((2-(2,6-dioxopiperidin-3-yl)-1-oxoisoindolin-4-yl)amino)-5-oxopentyl (2r,4as,6as,12br,14as,14br)-10-hydroxy-2,4a,6a,9,12b,14a-hexamethyl-11-oxo-1,2,3,4,4a,5,6,6a,11,12b,13,14,14a,14b-tetradecahydropicene-2-carboxylate	[H][C@@]12C[C@](C)(C(=O)OCCCCC(=O)N/C3=C/C=C\C4=C3CN(C3CCC(=O)NC3=O)C4=O)CC[C@]1(C)CC[C@]1(C)C3=CC=C4C(=CC(=O)C(O)=C4C)[C@]3(C)CC[C@@]21C	C47H57N3O8	HSP90	P07900	CRBN	CN-117924404-A
TPD-P61U0V	6-((2-(2,6-dioxopiperidin-3-yl)-1-oxoisoindolin-4-yl)amino)-6-oxohexyl (2r,4as,6as,12br,14as,14br)-10-hydroxy-2,4a,6a,9,12b,14a-hexamethyl-11-oxo-1,2,3,4,4a,5,6,6a,11,12b,13,14,14a,14b-tetradecahydropicene-2-carboxylate	6-((2-(2,6-dioxopiperidin-3-yl)-1-oxoisoindolin-4-yl)amino)-6-oxohexyl (2r,4as,6as,12br,14as,14br)-10-hydroxy-2,4a,6a,9,12b,14a-hexamethyl-11-oxo-1,2,3,4,4a,5,6,6a,11,12b,13,14,14a,14b-tetradecahydropicene-2-carboxylate	[H][C@@]12C[C@](C)(C(=O)OCCCCCC(=O)N/C3=C/C=C\C4=C3CN(C3CCC(=O)NC3=O)C4=O)CC[C@]1(C)CC[C@]1(C)C3=CC=C4C(=CC(=O)C(O)=C4C)[C@]3(C)CC[C@@]21C	C48H59N3O8	HSP90	P07900	CRBN	CN-117924404-A
TPD-P9D9BD	CN-118026997-A_1-3	.	NS(=O)(=O)C1=C2C(=O)C=C(NC3=CC=CC=C3N3CCN(C(=O)CCCCNC4=CC=CC5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)C(=O)C2=CC=C1	C38H37N7O9S	STAT3;pSTAT3	P40763/P40763	CRBN	CN-118026997-A
TPD-PAQ519	CN-118027001-A_W1-L4-C1	.	N#CC1=CC=C(C2=CC=C(N3C=C(CC(NC(=O)C4(C5=CC=CC=C5)CC4)C(=O)NCCCCOC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)N=N3)C=C2)C=C1	C45H40N8O7	PIN1	Q13526	CRBN	CN-118027001-A
TPD-PBEYMB	CN-118027014-A_1A	.	O=C(CN1CCN(C2=CC(C3=CC=C4N=CC=C(NC5=C/C6=C(\C=C/5)SC=N6)C4=C3)=CC=C2)CC1)NCCCCCCCCCCN/C1=C/C=C\C2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O	C51H55N9O5S	RIPK3	Q9Y572	CRBN	CN-118027014-A
TPD-PE0MXR	CN-118239946-A_1	.	CC1=CC(OC2=CC=C(OCCOCCOCCOCCNC3=C4\C(=O)N(C5CCC(=O)NC5=O)C(=O)\C4=C\C=C\3)C=C2)=CC(C)=C1C1=CSC(NC(=O)C2=CC=NC=C2)=N1	C44H44N6O10S	HEC 1	O14777	CRBN	CN-118239946-A
TPD-PGKSYC	CN-118267388-A_1	.	CN1C(=O)N(C2CCC(=O)NC2=O)C2=C1C=C(C#CCCC1CCN(C(=O)[C@H](CC3=CC=C(C(C)(C)C)C=C3)NC(=O)[C@H](CCC(N)=O)NC(=O)C3CC[C@@H]4CCN(CC(F)F)C[C@H](NC(=O)C5=CC6=CC(C(F)(F)P(=O)(O)O)=CC=C6S5)C(=O)N34)CC1)C=C2	C62H73F4N10O12PS	MCP-1	P13500	CRBN	CN-118267388-A
TPD-PGL6EL	CN-118459451-A_1	.	CC(C)(C)C1=CC(NC(=O)NC2=CC=C(C3=CN(C4=CC=C(OCO/C5=C/C=C\C6=C5CN(C5CCC(=O)NC5=O)C6=O)C=C4Cl)N=N3)C=C2)=NO1	C36H33ClN8O7	FLT3	P36888	CRBN	CN-118459451-A
TPD-PNEVKL	CN-118598856-A_1	.	CC1=C(CCC(=O)NCCNC2=CC=CC3=C2C(=O)N(C2CCC(=O)NC2=O)C3=O)C(=O)N(NC2=NC(Cl)=C(C(F)(F)F)C=C2)C1=O	C29H25ClF3N7O7	XPO1	O14980	CRBN	CN-118598856-A
TPD-PNO498	CN-118619965-A_2	.	CC1=C(NC2CCCNC2)C(C2=C3SC(CNCCCCCCC(=O)N/C4=C/C=C\C5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)=CC3=NC=C2)=CC(Cl)=C1	C40H44ClN7O5S	USP7	Q93009	CRBN	CN-118619965-A
TPD-PR14JW	CN-118725001-A_G1	.	[H][C@@]12C[C@@](C)(C(=O)NCCN/C3=C/C=C\C4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC[C@]1(C)CC[C@]1(C)C2=CC(=O)[C@@]2([H])C1CC[C@@]1([H])C(C)(C)[C@@H](O)CC[C@]21C	C44H58N4O7	PRDX2;伪鈥慡MA	P32119/P62736	CRBN	CN-118725001-A
TPD-PSA84R	CN-118772112-B_15a	.	COC1=CC(NC2=NC(NC3=CC=C(NS(=O)(=O)C4=CC=C(C(=O)NCCNC5=CC=CC6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)C=C4)C=C3)=NC=C2)=CC(OC)=C1OC	C41H39N9O10S	FAM20C	Q8IXL6	CRBN	CN-118772112-B
TPD-Q1KIQL	CN-118772112-B_15b	.	COC1=CC(NC2=NC(NC3=CC=C(NS(=O)(=O)C4=CC=C(C(=O)NCCCNC5=CC=CC6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)C=C4)C=C3)=NC=C2)=CC(OC)=C1OC	C42H41N9O10S	FAM20C	Q8IXL6	CRBN	CN-118772112-B
TPD-Q1NIJJ	CN-118878517-A_IB-1	.	CN1C(=O)C(NC(=S)SCC(=O)NC(=O)NC2=CC(C(=O)NCC3=CN(CCC(=O)NC4=C5CN(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)N=N3)=CC=C2)/N=C(/C2=CC=CC=C2)C2=C1C=CC=C2	C46H42N12O8S2	ANXA3	P12429	CRBN	CN-118878517-A
TPD-Q2UII2	CN-118930546-A_1-1	.	CC(SC1=NC2=C(/C=N\N2C2=CC=CC(C(=O)NCCNC3=CC=CC4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)=C2)C(=O)N1)C(N)=O	C30H27N9O7S	DAPK1	P53355	CRBN	CN-118930546-A
TPD-Q7WOHS	CN-119119026-A_A2	.	CCCC(C1=CC=C(OCCCCN2CCN(/C3=N/C4=C(C=CC(F)=C4)N(CC(F)F)C4=C3C=C(Cl)C=C4)CC2)C=C1)N(C)C(=O)/C(C#N)=C/C1=NC=CS1	C41H43ClF3N7O2S	PAK1	Q13153	.	CN-119119026-A
TPD-Q84J1O	SCHEMBL31255746	SCHEMBL31255746	CC1=CC(CNCCCCCCNC(=O)[C@@H](N)CCCNC(=N)N)=CC(C)=C1C1=C(C2=CC=NC3=CC(F)=CC=C32)N(C)C=N1	C34H46FN9O	NSD3	Q9BZ95	.	CN-119241502-A
TPD-Q8TFNA	CN-119285612-A_A1	.	N/C1=C(\C2=NC3=C(/C=C(N4CCN(CC5CCN(CC(=O)N6CCN(C7=C/C=C8/C(=O)N(C9CCC(=O)NC9=O)C(=O)/C8=C\7)CC6)CC5)CC4)\C=C/3)N2)C(=O)NC2=C1C(F)=CC=C2	C45H48FN11O6	FLT3-ITD	P36888	CRBN	CN-119285612-A
TPD-Q9KLW1	SMART1	SMART1; EX-A11401; H38756	CNC(=O)C1=NC=CC(OC2=CC=C(N3C=C(C4=CC(NC(=O)C5CCCN(C6=C7C(=O)N(C8CCC(=O)NC8=O)C(=O)C7=CC=C6)C5)=CC=C4)N=N3)C=C2)=C1	C40H35N9O7	SMUF1	Q9HCE7	CRBN	CN-119330934-A
TPD-Q9NLKB	CN-119390701-A_1-2	.	COC1=C2N=C(NC(=O)C3=CN=C(N)N=C3)N3CCN=C3C2=CC=C1OCCCN1CCN(CCCCCC(=O)NC2=C3C(=O)N(C4CCC(=O)NC4=O)CC3=CC=C2)CC1	C42H50N12O7	PI3Kalpha	P42336	CRBN	CN-119390701-A
TPD-Q9ZUPB	CN-119504710-A_YZ-26	.	O=C1CCC(N2CC3=C(NCCCCCN4CCC(NC5=CC(C(=O)NCC(O)CN6CCC7=C(C=CC=C7)C6)=NC=N5)CC4)C=CC=C3C2=O)C(=O)N1	C40H51N9O5	PRMT5	O14744	CRBN	CN-119504710-A
TPD-QAEUD4	CN-119661504-A_P3	.	CCC1=NC2=CC=C(CN3CCN(C4=CN=C(C(=O)NCCOCCOCCNC5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)C=C4)CC3)C=C2NC1=O	C40H45N9O8	PARP1	P09874	CRBN	CN-119661504-A
TPD-QBA1Y8	CN-119751452-A_1	.	CC1=CC=C(C2=C(C#N)C3=NC4=CC=CC=C4N3C(NC(=O)CCC(=O)N3CCN(C4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)=C2C#N)C=C1	C41H33N9O6	FSP1	Q9BRQ8	CRBN	CN-119751452-A
TPD-QBUTGL	CN-119899171-A_B5C	.	COC1=CC=C(C2=CC=CC=C2)C=C1NS(=O)(=O)C1=C(OCCCCCNC2=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=CC=C2)C(Cl)=CC(Cl)=C1	C37H34Cl2N4O8S	ACLY	P53396	CRBN	CN-119899171-A
TPD-QCCAZ9	CN-120004853-A_RP-4	.	O=C1CCC(N2C(=O)C3=C(C2=O)/C(NCCOCCNC(=O)C(CC2=CC(O)=C(O)C=C2)OC(=O)/C=C/C2=CC(O)=C(O)C=C2)=C\C=C/3)C(=O)N1	C35H34N4O12	NEU1	Q99519	CRBN	CN-120004853-A
TPD-QE34HN	CN-120004875-A_1-1	.	NC1=NC2=CC(C3=NC(N4CCN(C(=O)CCC(=O)N/C5=C/C=C\C6=C5CN(C5CCC(=O)NC5=O)C6=O)CC4)=NC(N4CCOCC4)=N3)=CC=C2O1	C35H37N11O7	PI3Kalpha	P42336	CRBN	CN-120004875-A
TPD-QEOV76	CN-120097965-A_9A	.	O=C1CCC(N2C(=O)C3=CC=CC(NCCNC(=O)C4=CNC(C5=CC(OCC6CC6)=C(OC(F)F)C=C5)=N4)=C3C2=O)C(=O)N1	C30H28F2N6O7	PDE4	Q07343	CRBN	CN-120097965-A
TPD-QJET83	CN-120118070-A_GSAz-15	.	COC1=CC=C(C2=C(C3=CC=C(OC)C=C3)N(CC3=CC=C(C(=O)NCCOCCOCCC(=O)N4CCC(C5=C(C)C=C(NC6=NC=C(Cl)C(NC7=CC=CC=C7S(=O)(=O)C(C)C)=N6)C(OC(C)C)=C5)CC4)C=C3)C(C3=CC(C(F)(F)F)=CC(C(F)(F)F)=C3)=N2)C=C1	C68H71ClF6N8O9S	EML4-ALK	Q9HC35	.	CN-120118070-A
TPD-QK7VZD	CN-120136812-A_LS-26	.	CC1=C(C)C=C2SC(NC(=O)C3=CC=CC(NC(=O)CCOCCOCCNC4=C/C5=C(\C=C/4)C(=O)N(C4CCC(=O)NC4=O)C5=O)=C3)=NC2=C1	C36H36N6O8S	KLF5	Q13887	CRBN	CN-120136812-A
TPD-QLZM5Q	SCHEMBL31619679	SCHEMBL31619679	O=C1CCC(N2C(=O)C3=CC=CC(NCCOCCOCCOCCOCCC(=O)NC4=CC=C(/C=C/C(=O)C5=CC(O)=CC=C5O)C=C4)=C3C2=O)C(=O)N1	C39H42N4O12	SPT5-Pol II	O00267	CRBN	CN-120136841-A
TPD-QN8POL	CN-120136845-A_PS1	.	NC1=NC(N2C=C(C(=O)N3CCN(CCCCCC(=O)N/C4=C/C=C\C5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)C3=C2/C=C(C#CC2(O)CCCCC2)\C=C/3)=CC=N1	C44H47N9O7	PAK4	O96013	CRBN	CN-120136845-A
TPD-QS9G6F	CN-120136845-A_PS2	.	NC1=NC(N2C=C(C(=O)N3CCN(CCCCCCC(=O)N/C4=C/C=C\C5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)C3=C2/C=C(C#CC2(O)CCCCC2)\C=C/3)=CC=N1	C45H49N9O7	PAK4	O96013	CRBN	CN-120136845-A
TPD-QUF4LD	CN-120208920-A_5a	.	COC1=CC(CNC(=O)CCCC/C=C/C(C)C)=CC=C1OCCCOC1=C2C(=O)N(C3CCC(=O)NC3=O)C(=O)C2=CC=C1	C34H41N3O8	TRPV1	Q8NER1	CRBN	CN-120208920-A
TPD-QVWENL	CN-120289430-A_ND-F-2	.	COC1=CC(C(=O)NC2CCN(CC3CCN(C4=C/C5=C(\C=C/4)C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)CC2)=C(F)C=C1NC1=NC(O/C2=C/C=C\C3=C2C(=O)N(C)C3)=C(C(F)(F)F)C=N1	C46H45F4N9O8	FAK	Q05397	CRBN	CN-120289430-A
TPD-QY5MK8	CN-120309611-A_27	.	COC1=NC=C(C2=CC=C3NC(=O)C4=C(C3=C2)N(C2=CC=C(N3CCN(C(=O)/C=C/C(=O)C5=CC=C(F)C=C5)CC3)C(F)=C2)N=N4)C=C1	C35H27F2N7O4	RIOK2	Q9BVS4	.	CN-120309611-A
TPD-R3RAL0	EP-4313979-A1_P5	.	CC1=C(C2=CC=C(CNC(=O)C3CC(O)CN3C(=O)C(NC(=O)CCC(=O)NCCCCOC3=CC=C(OC4=CC=C(N(CC5=CC=CC=C5)C(=O)CCl)C=C4)C=C3)C(C)(C)C)C=C2)SC=N1	C51H59ClN6O8S	RNF4	P78317	VHL	EP-4313979-A1
TPD-R4AJ3T	EP-4526303-A1_8-4	.	CC1(C)CCN(CC2=CC=C(N3CC(=O)NC4(CCN(C5=CC(NCCCNC(=O)CCOCOCCNC6=C7\C(=O)N(C8CCC(=O)NC8=O)C(=O)\C7=C\C=C\6)=NC=N5)CC4)C3)C=C2)CC1	C48H63N11O8	METTL3-METTL14 complex	Q86U44	CRBN	EP-4526303-A1
TPD-RD4L8G	EP-4617271-A1_RBM3-395	.	CC1=CC(C(=O)N2CCC(CN3C=C(CCCCCCCCC(=O)N[C@@H](CO)C[C@H](O)C4=CC=CC=C4)N=N3)CC2)=C(C)N1C1=CC=C(F)C=C1	C40H53FN6O4	CERT	Q9Y5P4	.	EP-4617271-A1
TPD-RMP04V	SCHEMBL27215741	SCHEMBL27215741	O=C1CCC(N2C(=O)C3=C(C2=O)/C(NCCOCCOCCOCCOCCC(=O)N2CCN(C4=CC=C(C5=CN=C(NCC6=CC=CO6)N6C=NN=C56)C=C4)CC2)=C\C=C/3)C(=O)N1	C44H50N10O10	EED	O75530	CRBN	US-11981678-B2
TPD-RN5W8A	US-20240398800-A1_17	.	C[C@@H]1COCCN1C1=CC(C2([S@](C)(=N)=O)CC2)=NC(C2=C3C=CN(CCCCCCCCN4C=C(COC5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CCC5)N=N4)C3=NC=C2)=N1	C44H53N11O7S	TAF1	P21675	CRBN	US-20240398800-A1
TPD-RN7RF1	TBK1 PROTAC 3i	TBK1 PROTAC 3i; CHEMBL4227907; PROTAC TBK1 degrader-2; 2052306-13-3; (2S,4R)-1-[(2S)-2-[[2-[3-[4-[3-[4-[[5-bromo-4-[3-[cyclobutanecarbonyl(methyl)amino]propylamino]pyrimidin-2-yl]amino]phenoxy]propoxy]butoxy]propoxy]acetyl]amino]-3,3-dimethylbutanoyl]-4-hydroxy-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide; TBK1-PROTAC1; TBK1 PROTAC? 3i; SCHEMBL18282349; GTPL11661; GLXC-15899; BDBM50459898; AKOS040755150; compound 3i [PMID: 28692295]; BP-41579; HY-112557; CS-0046374	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)COCCCOCCCCOCCCOC3=CC=C(NC4=NC=C(Br)C(NCCCN(C)C(=O)C5CCC5)=N4)C=C3)C(C)(C)C)C=C2)SC=N1	C53H74BrN9O9S	TBK1	Q9UHD2	VHL	WO-2016197114-A1
TPD-S60NSQ	WO-2016197114-A1_18	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@H](O)CN3C(=O)C(NC(=O)COCCCOCCCCOCCCOC3=CC=C(NC4=NC=C(Br)C(NCCN(C)C(=O)C5CCC5)=N4)C=C3)C(C)(C)C)C=C2)SC=N1	C52H72BrN9O9S	TBK1	Q9UHD2	VHL	WO-2016197114-A1
TPD-S7YGQ2	WO-2017211924-A1_33	.	CNC(=O)C1=CC=CC=C1NC1=C(Cl)C=NC(NC2=CC=C(N3CCN(CCOCCOCCOCCOC4=CC(CNC(=O)[C@@H](NC(=O)[C@H](C)NC)C(C)(C)C)=C(CCC(=O)N[C@@H]5CCCC6=C5C=CC=C6)C=C4)CC3)C=C2)=N1	C60H80ClN11O8	RPS6KA1;IRAK3;GAK;TEC;PTK2B;AURKA;MAPK9;AKT2	Q15418/Q9Y616/O14976/P42680/Q14289/O14965/P45984/P31751	VHL	WO-2017211924-A1
TPD-SA4NUJ	SJF-6693	SJF-6693; CHEMBL4576361	COC1=CC2=C(OC3=C(F)C=C(NC(=O)C4(C(=O)NC5=CC=C(F)C=C5)CC4)C=C3)C=CN=C2C=C1OCCOCCOCCC(=O)N[C@H](C(=O)N1C[C@H](O)C[C@H]1C(=O)NCC1=CC=C(C2=C(C)N=CS2)C=C1)C(C)(C)C	C56H61F2N7O11S	p38;c-Met	Q16539/P08581	VHL	WO-2018226542-A1
TPD-SCE04R	PROTAC d9A-2	PROTAC d9A-2; d9A-2; SCHEMBL25906681; GLXC-22449; 2690350-15-1; N-(14-((2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindolin-4-yl)amino)-3,6,9,12-tetraoxatetradecyl)-4'-fluoro-3'-methyl-2-(4-(4-methyl-1H-imidazol-5-yl)piperidin-1-yl)-[1,1'-biphenyl]-4-carboxamide	CC1=CC(C2=CC=C(C(=O)NCCOCCOCCOCCOCCNC3=C4\C(=O)N(C5CCC(=O)NC5=O)C(=O)\C4=C\C=C\3)C=C2N2CCC(C3=C(C)N=CN3)CC2)=CC=C1F	C46H54FN7O9	SLC9A1;SLC9A4;SLC9A5;SLC9A8;SLC9B2;SLC9A6;SLC9A9;SLC9A3	P19634/Q6AI14/Q14940/Q9Y2E8/Q86UD5/Q92581/Q8IVB4/P48764	CRBN	WO-2021074429-A9
TPD-SGX7L7	SCHEMBL23578877	SCHEMBL23578877	CCN1C(=O)/C(=C/C2=CN(CC3=CN(CCOCCOCCOCC(=O)NC4=C5\C(=O)N(C6CCC(=O)NC6=O)C(=O)\C5=C/C=C\4)N=N3)C3=CC=CN=C23)NC1=S	C37H38N10O9S	p-tau S202-T205;p-tau S396;p-tau S356	P10636/P10636/P10636	CRBN	WO-2021133037-A1
TPD-SHKGS8	SCHEMBL23768517	SCHEMBL23768517	[H][C@]12C[C@@H](N(C)C(=O)CCOCCOCCNC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)[C@@H](OC)[C@](C)(O1)N1C3=C(C=CC=C3)/C3=C1/C1=C(/C4=C(C=CC=C4)N12)C1=C3CNC1=O	C48H47N7O10	c-KIT D816V;EGFR del19;EGFR C797S;EGFR del19-C797S;EGFR T790M-C797S;EGFR del19/T790M/C797S	P10721/P00533/P00533/P00533/P00533/P00533	CRBN	WO-2021162493-A1
TPD-SIRO9M	SCHEMBL24419189	SCHEMBL24419189; SCHEMBL29665293	O=C1CCC(N2C(=O)C3=C(C2=O)/C(NCCOCCOC2=CC=C(S(=O)(=O)NC(=O)NC4=C5CCCC5=CC5=C4CCC5)C=C2)=C\C=C/3)C(=O)N1	C36H37N5O9S	NLRP3	Q96P20	CRBN	WO-2022098108-A1
TPD-SJGBDY	SCHEMBL24634693	SCHEMBL24634693; SCHEMBL30876599	CCCC(=O)NC(C1=CC=CC(OCCCCCCNC(=O)CO/C2=C/C=C\C3=C2C(=O)N(C2CCC(=O)NC2=O)C3=O)=C1)C1=CC(Cl)=C2C=CC=NC2=C1O	C41H42ClN5O9	grp78	P11021	CRBN	WO-2022169834-A2
TPD-SNLD42	WO-2024005905-A2_1-4	.	CCOC(=O)C1=C(O)C=C(NC2=NC(C3=CC=C(NC(=O)CCOCCCOCCOCCOCCOCCNC(=O)COC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C3)=CS2)C=C1	C47H54N6O15S	SIRT1;SIRT2;SIRT3;SIRT4;SIRT5;SIRT6;SIRT7	Q96EB6/Q8IXJ6/Q9NTG7/Q9Y6E7/Q9NXA8/Q8N6T7/Q9NRC8	CRBN	WO-2024005905-A2
TPD-SW0D3T	SCHEMBL27162577	SCHEMBL27162577; EX-A9086G; 1H-Isoindole-1,3(2H)-dione, 5-[4-[[1-[4-[[5-bromo-4-[[4-cyclopropyl-2-(dimethylphosphinyl)phenyl]amino]-2-pyrimidinyl]amino]-5-methoxy-2-(1-methyl-1H-pyrazol-4-yl)phenyl]-4-piperidinyl]methyl]-1-piperazinyl]-2-(2,6-dioxo-3-piperidinyl)-; 2861227-35-0	COC1=C(NC2=NC=C(Br)C(NC3=C(P(C)(C)=O)C=C(C4CC4)C=C3)=N2)C=C(C2=CN(C)N=C2)C(N2CCC(CN3CCN(C4=CC=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=C4)CC3)CC2)=C1	C49H55BrN11O6P	EGFR L858R/T790M;EGFR L858R/T790M/C797S	P00533/P00533	CRBN	WO-2024083182-A1
TPD-SW0RSC	SCHEMBL27398043	SCHEMBL27398043	CC1=NC(NC2=NC=C(C(=O)NC3=C(C)C=CC=C3Cl)S2)=CC(N2CCN(C3CN(C4CCN(C5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)C3)CC2)=N1	C41H44ClN11O5S	c-Src	P12931	CRBN	WO-2024123819-A2
TPD-T1EUL1	WO-2024211154-A2_Defer-1	.	CCCCCCCC/C=C\CCCCCCCC(=O)NCC(=O)N[C@H](C(=O)N1CC(O)C[C@H]1C(=O)NCC1=CC=C(C2=C(C)N=CS2)C=C1)C(C)(C)C	C42H65N5O5S	Mitochondrial	Q8N4E7	VHL	WO-2024211154-A2
TPD-T1PDM1	WO-2025053796-A1_7	.	CCC1=NC(N)=NC(N)=C1OCCCOC1=CC=C(OCCOCCNC(=O)C2=CC(OC)=C(NC(=O)C3N[C@@H](CC(C)(C)C)[C@](C#N)(C4=CC=C(Cl)C=C4F)[C@H]3C3=C(F)C(Cl)=CC=C3)C=C2)C=C1CCC(=O)O	C53H60Cl2F2N8O9	DHFR-TS	A0A2Z4NBY2	VHL	WO-2025053796-A1
TPD-T4VBPW	WO-2025117674-A1_ZS3-046	.	C=CCCN1/C=C(/C2=C3N=CN(CCCCCCCN4CCC(CNC5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)CC4)C3=CC(C(=O)N3CCOCC3)=C2)C2=C(NC=C2)C1=O	C49H57N9O7	TAF1	P21675	CRBN	WO-2025117674-A1
TPD-T6YBZM	WO-2025155882-A1_4	.	COC1=CC2=C(C=C1OCCCN1CCCC1)N=C(N1CCC(F)(F)CC1)N=C2NC1CCN(CCCNC(=O)CCCCCNC2=CC=CC3=C2C(=O)N(C2CCC(=O)NC2=O)C3=O)CC1	C48H64F2N10O7	G9A;GLP	Q96KQ7/Q9H9B1	CRBN	WO-2025155882-A1
TPD-T7577B	PD155450	PD155450	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCCC(=O)NCCCNC3=NC(NC4=CC=C(CC#N)C=C4)=NC(NC4=NNC(C5CC5)=C4)=C3)C(C)(C)C)C=C2)SC=N1	C53H69N13O5S	AAK1;AURKA;AURKB;BMP2K;CDK9;EPHB2;GSK-3beta;ITK;LATS1;MAP4K2;NEK9	Q2M2I8/O14965/Q96GD4/Q9NSY1/P50750/P29323/P49841/Q08881/O95835/Q12851/Q8TD19	VHL	WO-2022093742-A1
TPD-T7S1NH	CDK4/6-IN-11	CDK4/6-IN-11; 2139329-47-6; BSJ-02-162; CHEMBL4646450; orb1983003; SCHEMBL19475278; SCHEMBL30338338; BDBM50545382; EX-A11478; MS-31547; HY-144995; CS-0436644; N-[4-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]butyl]-2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]acetamide	CC(=O)C1=C(C)C2=CN=C(NC3=CC=C(N4CCN(CCCCNC(=O)CN/C5=C/C=C\C6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C=N3)N=C2N(C2CCCC2)C1=O	C43H49N11O7	CDK4;CDK6;WEE1	P11802/Q00534/P30291	CRBN	WO-2022093742-A1
TPD-TBRCYP	BSJ-03-123	BSJ-03-123; 2361493-16-3; N-(2-(2-(2-(2-(4-(6-((6-Acetyl-8-cyclopentyl-5-methyl-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-2-yl)amino)pyridin-3-yl)piperazin-1-yl)ethoxy)ethoxy)ethoxy)ethyl)-2-((2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindolin-4-yl)oxy)acetamide; N-[2-[2-[2-[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]pyridin-3-yl]piperazin-1-yl]ethoxy]ethoxy]ethoxy]ethyl]-2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyacetamide; orb1301826; CHEMBL5204174; SCHEMBL22199840; SCHEMBL29678272; SCHEMBL30338263; GTPL10532; GLXC-21547; EX-A3877; LUD49316; C47H56N10O11; s8815; AKOS037653387; AT18355; BSJ-03-123?; AC-36701; BP-40150; N-[2-[2-[2-[2-[4-[6-[(6-Acetyl-8-cyclopentyl-7,8-dihydro-5-methyl-7-oxopyrido[2,3-d]pyrimidin-2-yl)amino]-3-pyridinyl]-1-piperazinyl]ethoxy]ethoxy]ethoxy]ethyl]-2-[[2-(2,6-dioxo-3-piperidinyl)-2,3-dihydro-1,3-dioxo-1H-isoindol-4-yl]oxy]acetamide; CID 137628658; HY-111556; CS-0087154; EN300-22946657; Z3847529695; N-(2-{2-[2-(2-{4-[6-({6-acetyl-8-cyclopentyl-5-methyl-7-oxo-7H,8H-pyrido[2,3-d]pyrimidin-2-yl}amino)pyridin-3-yl]piperazin-1-yl}ethoxy)ethoxy]ethoxy}ethyl)-2-{[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]oxy}acetamide; N-[2-[2-[2-[2-[4-[6-[(6-acetyl-8-cyclopentyl-5-methyl-7-oxo-pyrido[2,3-d]pyrimidin-2-yl)amino]-3-pyridyl]piperazin-1-yl]ethoxy]ethoxy]ethoxy]ethyl]-2-[2-(2,6-dioxo-3-piperidyl)-1,3-dioxo-isoindolin-4-yl]oxy-acetamide	CC(=O)C1=C(C)C2=CN=C(NC3=CC=C(N4CCN(CCOCCOCCOCCNC(=O)CO/C5=C/C=C\C6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C=N3)N=C2N(C2CCCC2)C1=O	C47H56N10O11	BCKDK;CDK4;CDK6;COQ8A;PDK1;PDK2;PDK3;WEE1	O14874/P11802/Q00534/Q8NI60/Q15118/Q15119/Q15120/P30291	CRBN	WO-2022093742-A1
TPD-TCYO30	WO-2022093742-A1_BSJ-03-204	.	CC(=O)C1=C(C)C2=CN=C(NC3=CC=C(N4CCN(CCCCNC(=O)CS/C5=C/C=C\C6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C=N3)N=C2N(C2CCCC2)C1=O	C43H48N10O7S	CDK4;CDK6;WEE1	P11802/Q00534/P30291	CRBN	WO-2022093742-A1
TPD-TDLU5M	BSJ-04-132	BSJ-04-132; 2349356-39-2; 7-Cyclopentyl-2-[[5-[4-[4-[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindolin-4-yl]oxy]acetamido]butyl]piperazin-1-yl]pyridin-2-yl]amino]-N,N-dimethyl-7H-pyrrolo[2,3d]pyrimidine-6-carboxamide; 7-cyclopentyl-2-[[5-[4-[4-[[2-[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]oxyacetyl]amino]butyl]piperazin-1-yl]pyridin-2-yl]amino]-N,N-dimethylpyrrolo[2,3-d]pyrimidine-6-carboxamide; CHEMBL5303541; SCHEMBL23974495; SCHEMBL29678499; GTPL10531; GLXC-20107; BP-42271; DA-61920; MS-31521; HY-136252; CS-0121012; G17656; EN300-33448895; 7-cyclopentyl-2-[(5-{4-[4-(2-{[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]oxy}acetamido)butyl]piperazin-1-yl}pyridin-2-yl)amino]-N,N-dimethyl-7H-pyrrolo[2,3-d]pyrimidine-6-carboxamide	CN(C)C(=O)C1=CC2=CN=C(NC3=CC=C(N4CCN(CCCCNC(=O)CO/C5=C/C=C\C6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C=N3)N=C2N1C1CCCC1	C42H49N11O7	BCKDK;CDK4;CDK6;COQ8A;PDK1;PDK2;PDK3	O14874/P11802/Q00534/Q8NI60/Q15118/Q15119/Q15120	CRBN	WO-2022093742-A1
TPD-TI9ODY	PD155191	PD155191	O=C(CO/C1=C/C=C\C2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O)NCCCCCCCN1CCC2=CC(NC3=NC=C(C4CC4)C(NCCCNC(=O)C4CCC4)=N3)=CC=C2C1	C46H57N9O7	AAK1;AURKA;AURKB;BMP2K;CDK10;CDK9;GAK;MARK2;MARK3;MARK4;SIK2;STK17A;STK17B;SNRK;ULK1;WEE1	Q2M2I8/O14965/Q96GD4/Q9NSY1/Q15131/P50750/O14976/Q7KZI7/P27448/Q96L34/Q9H0K1/Q9UEE5/O94768/Q9NRH2/O75385/P30291	CRBN	WO-2022093742-A1
TPD-TIHQRZ	PD155189	PD155189	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCN3CCC4=CC(NC5=NC=C(C6CC6)C(NCCCNC(=O)C6CCC6)=N5)=CC=C4C3)C(C)(C)C)C=C2)SC=N1	C53H72N10O5S	AAK1;GAK;MARK2;MARK3;MARK4;RPS6KB1;SIK2;SIK3;SNRK;STK17A;STK17B;ULK1;WEE1	Q2M2I8/O14976/Q7KZI7/P27448/Q96L34/P23443/Q9H0K1/Q9Y2K2/Q9NRH2/Q9UEE5/O94768/O75385/P30291	VHL	WO-2022093742-A1
TPD-TIU48A	DB-3-291	DB-3-291; 2769753-64-0; SCHEMBL21307398; SCHEMBL29750193; MS-31647; HY-137345; CS-0137849	CC1=CC=CC(Cl)=C1NC(=O)C1=CN=C(NC2=CC(N3CCN(CC(=O)NCCCCNC(=O)CO/C4=C/C=C\C5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)=NC(C)=N2)S1	C41H44ClN11O8S	ABL2;BLK;CSK;WEE1	P42684/P51451/P41240/P30291	CRBN	WO-2022093742-A1
TPD-TJB6Z2	WO-2022093742-A1_DB0646	.	CC1=CC=C(NC(=O)C2=CC=CC(C(F)(F)F)C2)C=C1N1CC2=CN=C(NC3=CC=C(N4CCN(CC5=CN(CCCCCOC6=CC=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7=O)C=N5)CC4)N=C3)N=C2N(C)C1=O	C53H54F3N13O7	ABL2;AURKA;BLK;BUB1;CDK11A;CDK11B;CDK4;CSK;DDR2;EPHA3;EPHB3;EPHB6;FER;FYN;GAK;LATS1;LCK;LIMK1;LIMK2;LRRK2;LYN;MAP3K1;MAP3K11;MAP3K20;MAP4K1;MAP4K2;MAP4K5;p38beta;MAPK12;p38alpha;MAPK8;MAPK9;MAPKAPK2;MKNK2;NLK;PLK1;FAK;PTK2B;RIPK1;RIPK2;RPS6KA3;SIK2;Src;TAOK2;TEC;TNK2;TTK;UHMK1;ULK1;WEE1;YES1	P42684/O14965/P51451/O43683/Q9UQ88/P21127/P11802/P41240/Q16832/P29320/P54753/O15197/P16591/P06241/O14976/O95835/P06239/P53667/P53671/Q5S007/P07948/Q13233/Q16584/Q9NYL2/Q92918/Q12851/Q9Y4K4/Q15759/P53778/Q16539/P45983/P45984/P49137/Q9HBH9/Q9UBE8/P53350/Q05397/Q14289/Q13546/O43353/P51812/Q9H0K1/P12931/Q9UL54/P42680/Q07912/P33981/Q8TAS1/O75385/P30291/P07947	CRBN	WO-2022093742-A1
TPD-TNBWMA	PD155184	PD155184	CC1=CC=C(NC(=O)C2=CC=CC(C(F)(F)F)=C2)C=C1N1CC2=CN=C(NC3=CC=C(N4CCN(CCOC5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)CC4)N=C3)N=C2N(C)C1=O	C46H42F3N11O7	BLK;CDK4;CLK1;CSK;FER;LCK;LIMK1;MAPK8;MAPK9;MKNK2;PLK1;PTK2B;SIK2;Src;TNK2;UHMK1;YES1	P51451/P11802/P49759/P41240/P16591/P06239/P53667/P45983/P45984/Q9HBH9/P53350/Q14289/Q9H0K1/P12931/Q07912/Q8TAS1/P07947	CRBN	WO-2022093742-A1
TPD-TW1Q2M	DB0662	DB0662; 2769753-51-5; orb2566519; DA-72576; MS-31739; HY-148066; CS-0609907	CC1=CC=C(NC(=O)C2=CC=CC(C(F)(F)F)=C2)C=C1N1CC2=CN=C(NC3=CC=C(N4CCN(CCCOC5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)CC4)N=C3)N=C2N(C)C1=O	C47H44F3N11O7	ABL1;ABL2;BLK;BUB1;CDK11B;CDK4;CSK;EPHB6;FER;FYN;GAK;LCK;LIMK1;MAP3K1;MAP3K11;MAP3K20;MAP4K1;p38alpha;MAPK8;MAPK9;MAPKAPK2;MKNK2;PAK4;PDIK1L;PTK2B;RPS6KA1;RPS6KA3;SIK2;Src;TNK2;UHMK1;ULK1;YES1	P00519/P42684/P51451/O43683/P21127/P11802/P41240/O15197/P16591/P06241/O14976/P06239/P53667/Q13233/Q16584/Q9NYL2/Q92918/Q16539/P45983/P45984/P49137/Q9HBH9/O96013/Q8N165/Q14289/Q15418/P51812/Q9H0K1/P12931/Q07912/Q8TAS1/O75385/P07947	CRBN	WO-2022093742-A1
TPD-U1H70Y	PD155182	PD155182	CC1=CC=C(NC(=O)C2=CC=CC(C(F)(F)F)=C2)C=C1N1CC2=C/N=C(NC3=CC=C(N4CCN(CCCCCCO/C5=C/C=C\C6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)N=C3)\N=C\2N(C)C1=O	C50H50F3N11O7	CDK4;BLK;FER;LIMK2;GAK;CSK;SIK2;LCK;PTK2B;Src;ABL2;MAPK9;MAP4K2;MKNK2;MAP3K20;TNK2	P11802/P51451/P16591/P53671/O14976/P41240/Q9H0K1/P06239/Q14289/P12931/P42684/P45984/Q12851/Q9HBH9/Q9NYL2/Q07912	CRBN	WO-2022093742-A1
TPD-U2D2KF	DB1113	DB1113; 2769753-53-7; orb1982760; SCHEMBL26446949; BP-42146; DA-72578; HY-148061; CS-0609884; EN300-44825953; (2S,4R)-1-[(2S)-3,3-dimethyl-2-[5-(4-{5-[(8-methyl-6-{2-methyl-5-[3-(trifluoromethyl)benzamido]phenyl}-7-oxo-5H,6H,7H,8H-pyrimido[4,5-d][1,3]diazin-2-yl)amino]pyridin-2-yl}piperazin-1-yl)pentanamido]butanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide; (2S,4R)-1-[(2S)-3,3-dimethyl-2-[5-[4-[5-[[1-methyl-3-[2-methyl-5-[[3-(trifluoromethyl)benzoyl]amino]phenyl]-2-oxo-4H-pyrimido[4,5-d]pyrimidin-7-yl]amino]pyridin-2-yl]piperazin-1-yl]pentanoylamino]butanoyl]-4-hydroxy-N-[(1S)-1-[4-(4-methyl-1,3-thiazol-5-yl)phenyl]ethyl]pyrrolidine-2-carboxamide	CC1=CC=C(NC(=O)C2=CC=CC(C(F)(F)F)=C2)C=C1N1CC2=CN=C(NC3=CC=C(N4CCN(CCCCC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=C(C)N=CS6)C=C5)C(C)(C)C)CC4)N=C3)N=C2N(C)C1=O	C59H68F3N13O6S	ABL1;ABL2;BLK;CDK11B;CDK4;CSK;EPHA3;FER;GAK;LIMK1;MAP3K20;MAP4K1;MAP4K2;MAP4K3;MAP4K4;MAP4K5;p38alpha;MAPK7;MAPK8;MAPK9;MAPKAPK2;MAPKAPK3;NLK;PDIK1L;PTK2B;RIPK1;RPS6KA1;RPS6KA3;SIK2;SIK3;STK35;TNK2;ULK1	P00519/P42684/P51451/P21127/P11802/P41240/P29320/P16591/O14976/P53667/Q9NYL2/Q92918/Q12851/Q8IVH8/O95819/Q9Y4K4/Q16539/Q13164/P45983/P45984/P49137/Q16644/Q9UBE8/Q8N165/Q14289/Q13546/Q15418/P51812/Q9H0K1/Q9Y2K2/Q8TDR2/Q07912/O75385	VHL	WO-2022093742-A1
TPD-U6DN51	SCHEMBL24847600	SCHEMBL24847600; PD155178	CC1=CC=C(NC(=O)C2=CC=CC(C(F)(F)F)=C2)C=C1N1CC2=CN=C(NC3=CC=C(N4CCN(CCCCCC(=O)N[C@H](C(=O)N5C[C@H](O)C[C@H]5C(=O)N[C@@H](C)C5=CC=C(C6=C(C)N=CS6)C=C5)C(C)(C)C)CC4)N=C3)N=C2N(C)C1=O	C60H70F3N13O6S	ABL1;ABL2;BLK;CDK11B;CDK4;CIT;CSK;EPHA3;FER;GAK;LCK;LIMK2;MAP3K20;MAP3K7;MAP4K1;MAP4K2;MAP4K5;p38alpha;MAPK7;MAPK9;MAPKAPK2;MAPKAPK3;PDIK1L;PTK2B;RIPK1;RPS6KA1;SIK2;STK35;TAOK2;TNK2;ULK1	P00519/P42684/P51451/P21127/P11802/O14578/P41240/P29320/P16591/O14976/P06239/P53671/Q9NYL2/O43318/Q92918/Q12851/Q9Y4K4/Q16539/Q13164/P45984/P49137/Q16644/Q8N165/Q14289/Q13546/Q15418/Q9H0K1/Q8TDR2/Q9UL54/Q07912/O75385	VHL	WO-2022093742-A1
TPD-UBK7ES	SCHEMBL29750021	SCHEMBL29750021; PD155176	CN[C@@H](C)C(=O)N[C@H](C(=O)N1CCC[C@H]1C1=NC(C(=O)C2=CC=CC(OCCCCCN3C=C(CN4CCN(C5=CC=C(NC6=NC7=C(C=N6)CN(C6=CC(NC(=O)C8=CC=CC(C(F)(F)F)=C8)=CC=C6C)C(=O)N7C)C=N5)CC4)N=N3)=C2)=CS1)C1CCCCC1	C65H75F3N16O6S	BLK;BUB1;CDK4;LIMK2;SIK2;STK17A;TEC;TNK2;UHMK1	P51451/O43683/P11802/P53671/Q9H0K1/Q9UEE5/P42680/Q07912/Q8TAS1	VHL	WO-2022093742-A1
TPD-UFGR9G	PD155174	PD155174	CC1=CC=C(NC(=O)C2=CC=CC(C(C)(C)C#N)=C2)C=C1NC1=CC=C2N=CN(CCOCCOCCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)NCC3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)C(=O)C2=C1	C55H63N9O8S	p38alpha	Q16539	VHL	WO-2022093742-A1
TPD-UPRCJV	PD155173	PD155173	CC(C)(C)C1=NC(C2=CC=CC(NS(=O)(=O)C3=C(F)C=CC=C3F)=C2F)=C(C2=CC=NC(NCCOCCNC(=O)CCOCCOCCN/C3=C/C=C\C4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)=N2)S1	C47H50F3N9O10S2	AURKA;BCKDK;CDK1;CDK16;CDK17;CDK2;CDK3;CDK4;CDK6;COQ8A;COQ8B;CSK;EIF2AK2;LIMK1;LIMK2;MAP3K20;NLK;PLK1;PDK1;PDK2;TESK2	O14965/O14874/P06493/Q00536/Q00537/P24941/Q00526/P11802/Q00534/Q8NI60/Q96D53/P41240/P19525/P53667/P53671/Q9NYL2/Q9UBE8/P53350/Q15118/Q15119/Q96S53	CRBN	WO-2022093742-A1
TPD-V1R691	WO-2022093742-A1_DD-03-107	.	CC(C)(C)C1=NC(C2=CC=CC(NS(=O)(=O)C3=C(F)C=CC=C3F)=C2F)=C(C2=CC=NC(CCCOCCNC(=O)CCOCCOCCN/C3=C/C=C\C4=C3CN(C3CCC(=O)NC3=O)C4=O)=N2)S1	C48H53F3N8O9S2	BCKDK;COQ8A;LIMK1;PDK1;PDK2;PDK3	O14874/Q8NI60/P53667/Q15118/Q15119/Q15120	CRBN	WO-2022093742-A1
TPD-V2F6DX	PD155170	PD155170	NC1=C2\C(C3=CC=C(OC4=CC=CC=C4)C=C3)=NN([C@@H]3CCCN(C(=O)CCCN4CCN(CCNC(=O)CCOCCOCCN/C5=C/C=C\C6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C3)\C2=N\C=N\1	C52H62N12O9	ABL2;BLK;CSK;FYN;LCK;Src;TEC	P42684/P51451/P41240/P06241/P06239/P12931/P42680	CRBN	WO-2022093742-A1
TPD-VFMWS0	DD-03-156	DD-03-156; 2769753-69-5; MS-31970; HY-137346; CS-0137850	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCOCCOCCNC3=NC=CC(C4=C(C5=CC=CC(NS(=O)(=O)C6=C(F)C=CC=C6F)=C5F)N=C(C(C)(C)C)S4)=N3)C(C)(C)C)C=C2)SC=N1	C53H62F3N9O8S3	CDK17;LIMK1;LIMK2	Q00537/P53667/P53671	VHL	WO-2022093742-A1
TPD-VIWVK6	SCHEMBL21307404	SCHEMBL21307404; PD155165	CCCS(=O)(=O)NC1=CC=C(F)C(C(=O)C2=CNC3=NC=C(C4=CC=C(C(=O)NCCCCCCCCNC(=O)CO/C5=C/C=C\C6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)C=C4)C=C23)=C1F	C47H47F2N7O10S	BLK;CSK;LCK;LIMK2;MAP2K5;MAP3K20	P51451/P41240/P06239/P53671/Q13163/Q9NYL2	CRBN	WO-2022093742-A1
TPD-VKJRIC	PD155164	PD155164	O=C1CCC(N2C(=O)C3=C(C2=O)/C(NCCOCCOCCOCCOCCC(=O)NC2=CC(CN4CCC(NC(=O)C5=C(NC(=O)C6=C(Cl)C=CC=C6Cl)C=NN5)CC4)=CC=C2)=C\C=C/3)C(=O)N1	C47H53Cl2N9O11	CDK11A;CDK9;CLK1;GSK3A;GSK-3beta;PIK3CG;SGK3	Q9UQ88/P50750/P49759/P49840/P49841/P48736/Q96BR1	CRBN	WO-2022093742-A1
TPD-VKPMHH	PD155162	PD155162	COC1=CC(N2CCN(CCOCCOCCC(=O)N[C@H](C(=O)N3C[C@H](O)C[C@H]3C(=O)N[C@@H](C)C3=CC=C(C4=C(C)N=CS4)C=C3)C(C)(C)C)CC2)=CC=C1NC1=NC=C2C(=N1)N(C)C1=CC=CC=C1C(=O)N2CC(F)(F)F	C55H68F3N11O8S	BLK;CSK	P51451/P41240	VHL	WO-2022093742-A1
TPD-VNXWCF	WO-2022093742-A1_FMF-06-098-1	.	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCOCCOCCN3CCN(C4=CC=C(NC5=NC=C(Cl)C(NC6=CC=CC=C6S(=O)(=O)C(C)C)=N5)C=C4)CC3)C(C)(C)C)C=C2)SCN1	C53H71ClN10O8S2	AAK1;ABL2;AURKA;AURKB;BUB1B;CDC7;CDK1;CDK12;KIAA1791;CDK2;CDK4;CDK6;CDK7;CDK9;CHEK1;CSNK1D;EPHA1;FER;FGFR1;GAK;IRAK4;ITK;LIMK2;MAP4K2;MAP4K3;MAPK6;MAPK7;MARK4;MELK;PKN3;PLK4;PRKAA1;FAK;PTK6;RPS6KA4;SIK2;STK35;TNK2;UHMK1;ULK1;WEE1	Q2M2I8/P42684/O14965/Q96GD4/O60566/O00311/P06493/Q9NYV4/Q14004/P24941/P11802/Q00534/P50613/P50750/O14757/P48730/P21709/P16591/P11362/O14976/Q9NWZ3/Q08881/P53671/Q12851/Q8IVH8/Q16659/Q13164/Q96L34/Q14680/Q6P5Z2/O00444/Q13131/Q05397/Q13882/O75676/Q9H0K1/Q8TDR2/Q07912/Q8TAS1/O75385/P30291	VHL	WO-2022093742-A1
TPD-VS7UA2	PD155157	PD155157	O=C(CO/C1=C/C=C\C2=C1C(=O)N(C1CCC(=O)NC1=O)C2=O)NCCCCCCCC(=O)NC1(C2=CC=C(C3=N/C4=C(\C=C/3C3=CC=CC=C3)C3=NNC(=O)N3C=C4)C=C2)CCC1	C48H46N8O8	PDK1;PDK2;PDK3	Q15118/Q15119/Q15120	CRBN	WO-2022093742-A1
TPD-VXT82I	SCHEMBL22533744	SCHEMBL22533744; PD155151	C[C@@H]1C[C@@H](O)C2=C1C(N1CCN(C(=O)[C@H](CNCCCCCCCCNC(=O)COC3=C4\C(=O)N(C5CCC(=O)NC5=O)C(=O)\C4=C\C=C\3)C3=CC=C(Cl)C=C3)CC1)=NC=N2	C44H53ClN8O8	Akt1;AKT2;AKT3;BCKDK;PDK1	P31749/P31751/Q9Y243/O14874/Q15118	CRBN	WO-2022093742-A1
TPD-VYUBZK	INY-03-041	INY-03-041; 2503017-97-6; 3-[7-[10-[[(2S)-2-(4-chlorophenyl)-3-[4-[(5R,7R)-7-hydroxy-5-methyl-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl]piperazin-1-yl]-3-oxopropyl]amino]decyl]-3-oxo-1H-isoindol-2-yl]piperidine-2,6-dione; orb1992823; SCHEMBL22533372; SCHEMBL29881317; GLXC-22005; EX-A7894; AKOS040733457; 3-(4-(10-(((S)-2-(4-Chlorophenyl)-3-(4-((5R,7R)-7-hydroxy-5-methyl-6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)piperazin-1-yl)-3-oxopropyl)amino)decyl)-1-oxoisoindolin-2-yl)piperidine-2,6-dione; BP-41601; MS-31470; HY-133120; CS-0112112; G18306	C[C@@H]1C[C@@H](O)C2=C1/C(N1CCN(C(=O)[C@H](CNCCCCCCCCCCC3=CC=CC4=C3CN(C3CCC(=O)NC3=O)C4=O)C3=CC=C(Cl)C=C3)CC1)=N\C=N/2	C44H56ClN7O5	Akt1;AKT2;AKT3;CDK4;MAPK6;STK17A	P31749/P31751/Q9Y243/P11802/Q16659/Q9UEE5	CRBN	WO-2022093742-A1
TPD-W63MC2	PD155145	PD155145	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCOC3=CC=CC=C3C3=CC=C4N=C(C5=C(N)N=CC=C5)N(C5=CC=C(C6(N)CCC6)C=C5)C4=N3)C(C)(C)C)C=C2)SC=N1	C55H62N10O5S	LATS1;STK17A	O95835/Q9UEE5	VHL	WO-2022093742-A1
TPD-W6P9X2	PD155144	PD155144	CC1=CN=C(NC2=CC=C(N3CCN(CCOCCOCCNC(=O)CO/C4=C/C=C\C5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)C=C2)N=C1NC1=CC=CC(S(=O)(=O)NC(C)(C)C)=C1	C46H56N10O10S	AAK1;AURKA;BMP2K;GAK;WEE1	Q2M2I8/O14965/Q9NSY1/O14976/P30291	CRBN	WO-2022093742-A1
TPD-WAV6BC	PD155139	PD155139	CC1=CN=C(NC2=CC=C(N3CCN(CCCCCCC(=O)N[C@H](C(=O)N4C[C@H](O)C[C@H]4C(=O)N[C@@H](C)C4=CC=C(C5=C(C)N=CS5)C=C4)C(C)(C)C)CC3)C=C2)N=C1NC1=CC=CC(S(=O)(=O)NC(C)(C)C)=C1	C55H75N11O6S2	AAK1;CDK16;WEE1;GAK;MARK4;NEK9;RPS6KB1;SIK2;SIK3;SNRK;STK17A;STK17B	Q2M2I8/Q00536/P30291/O14976/Q96L34/Q8TD19/P23443/Q9H0K1/Q9Y2K2/Q9NRH2/Q9UEE5/O94768	VHL	WO-2022093742-A1
TPD-WBXAE3	PD155135	PD155135	CC1=C(C2=CC=C([C@H](C)NC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCCCCCC3=CC=C(NC4=N\C=C5\NC(=O)NC6=CC=CC=C6\C5=N\4)C=C3)C(C)(C)C)C=C2)SC=N1	C47H55N9O5S	ABL2;EPHB2;SIK2;TYK2	P42684/P29323/Q9H0K1/P29597	VHL	WO-2022093742-A1
TPD-WD5W5A	SCHEMBL29750272	SCHEMBL29750272; PD155134	CC(C)S(=O)(=O)C1=C(NC2=NC(NC3=CC=C(N4CCN(CCOCCOCCNC(=O)CNC5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)C=C3)=NC=C2Cl)C=CC=C1	C44H51ClN10O9S	CDK4;AURKA;WEE1;BLK;FER;CDK6;LIMK2;AAK1;CDK5;CDK2;ITK;CDK17;LCK;PTK2B;CDK9;CDK7;KIAA1791;PRKAA1;CDK12;BMP2K;STK10	P11802/O14965/P30291/P51451/P16591/Q00534/P53671/Q2M2I8/Q00535/P24941/Q08881/Q00537/P06239/Q14289/P50750/P50613/Q14004/Q13131/Q9NYV4/Q9NSY1/O94804	CRBN	WO-2022093742-A1
TPD-WEMKIB	CHEMBL4642632	CHEMBL4642632; SCHEMBL29385285; CWHOUYZVKBUYQS-UHFFFAOYSA-N; PD155196; 2-[[2-[4-[4-[2-[2-[2-[[2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]acetyl]amino]ethoxy]ethoxy]ethyl]piperazin-1-yl]-2-methoxyanilino]-5-(trifluoromethyl)pyridin-4-yl]amino]-N-methylbenzamide	CNC(=O)C1=CC=CC=C1NC1=CC(NC2=CC=C(N3CCN(CCOCCOCCNC(=O)CNC4=CC=CC5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)C=C2OC)=NC=C1C(F)(F)F	C46H51F3N10O9	AURKA;CDK10;CDK7;MAPK7;PTK2B;RPS6KA1;RPS6KA3;STK33;WEE1	O14965/Q15131/P50613/Q13164/Q14289/Q15418/P51812/Q9BYT3/P30291	CRBN	WO-2022093742-A1
TPD-WMJI9V	PD155132	PD155132	CCC1=C2N=C(N3CCCC[C@H]3CCO)C=C(N(CC3=CC=C(N)N=C3)C(=O)CCOCCOCCOCCNC(=O)CN/C3=C/C=C\C4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)N2N=C1	C45H57N11O10	CDK4;WEE1;STK17A;PLK1;BUB1;TTK;UHMK1;MAP3K1;BUB1B;RIOK2;NUAK1;PIM2;CSNK1A1	P11802/P30291/Q9UEE5/P53350/O43683/P33981/Q8TAS1/Q13233/O60566/Q9BVS4/O60285/Q9P1W9/P48729	CRBN	WO-2022093742-A1
TPD-WNEV1Y	CHEMBL4636588	CHEMBL4636588; SCHEMBL29385704; DWHLPTIPTXJNCX-UHFFFAOYSA-N; PD155194; 2-[[2-[4-[4-[8-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]octyl]piperazin-1-yl]-2-methoxyanilino]-5-(trifluoromethyl)pyridin-4-yl]amino]-N-methylbenzamide	CNC(=O)C1=CC=CC=C1NC1=CC(NC2=CC=C(N3CCN(CCCCCCCCNC4=CC=CC5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)C=C2OC)=NC=C1C(F)(F)F	C46H52F3N9O6	AURKA;NUAK1;PTK2B;RPS6KA1;RPS6KA3;STK33;WEE1	O14965/O60285/Q14289/Q15418/P51812/Q9BYT3/P30291	CRBN	WO-2022093742-A1
TPD-WOCGX0	PD155131	PD155131	O=C1CCC(N2C(=O)C3=C(C2=O)/C(NCCCCCCCCN2CCC(NC(=O)C4=C(NC(=O)C5=C(Cl)C=CC=C5Cl)C=NN4)CC2)=C\C=C/3)C(=O)N1	C37H42Cl2N8O6	AURKA;BUB1;BUB1B;KIAA1791;CDK17;CDK4;CDK9;CHEK1;CLK1;CSNK1A1;CSNK1D;DAPK1;ERN1;GSK3A;GSK-3beta;MAP3K1;NUAK1;PIK3CG;PIM2;PLK1;RIOK2;STK17A;STK17B;TTK;UHMK1;WEE1	O14965/O43683/O60566/Q14004/Q00537/P11802/P50750/O14757/P49759/P48729/P48730/P53355/O75460/P49840/P49841/Q13233/O60285/P48736/Q9P1W9/P53350/Q9BVS4/Q9UEE5/O94768/P33981/Q8TAS1/P30291	CRBN	WO-2022093742-A1
TPD-WQM7YQ	PD155130	PD155130	CS(=O)(=O)NC1=CC=CC(C2=CS/C3=C\N=C(NC4=CC=C(N5CCN(CCOCCOCCOC6=CC=CC7=C6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C=C4)/N=C\23)=C1	C42H44N8O9S2	AAK1;AURKA;CAMKK1;CDK4;CDK6;LIMK2;NEK9;PTK2B;STK17A;STK17B;ULK1;ULK3;WEE1	Q2M2I8/O14965/Q8N5S9/P11802/Q00534/P53671/Q8TD19/Q14289/Q9UEE5/O94768/O75385/Q6PHR2/P30291	CRBN	WO-2022093742-A1
TPD-WRQ5US	DB0614	DB0614; 2769753-47-9; N-(3-(2-((4-(4-(5-((2-(2,6-DIOXOPIPERIDIN-3-YL)-1,3-DIOXOISOINDOLIN-4-YL)OXY)PENTYL)PIPERAZIN-1-YL)PHENYL)AMINO)THIENO[3,2-D]PYRIMIDIN-7-YL)PHENYL)METHANESULFONAMIDE; orb1982758; SCHEMBL29750429; BP-42213; DA-62683; HY-148063; CS-0609898; H54170	CS(=O)(=O)NC1=CC=CC(C2=CSC3=CN=C(NC4=CC=C(N5CCN(CCCCCO/C6=C/C=C\C7=C6C(=O)N(C6CCC(=O)NC6=O)C7=O)CC5)C=C4)N=C32)=C1	C41H42N8O7S2	AAK1;CDK1;CDK16;CDK2;CDK4;CDK6;EIF2AK4;GAK;LATS1;LIMK2;MAPK6;MAPKAPK5;MARK2;MARK4;MKNK2;NEK9;RPS6KB1;STK17A;STK17B;SIK2;SNRK;STK35;WEE1	Q2M2I8/P06493/Q00536/P24941/P11802/Q00534/Q9P2K8/O14976/O95835/P53671/Q16659/Q8IW41/Q7KZI7/Q96L34/Q9HBH9/Q8TD19/P23443/Q9UEE5/O94768/Q9H0K1/Q9NRH2/Q8TDR2/P30291	CRBN	WO-2022093742-A1
TPD-X4E6TU	SCHEMBL22835121	SCHEMBL22835121; SCHEMBL22835123; SCHEMBL29573923; PD155037; PD155038	NC1=C2C(C3=CC=C(OC4=CC=CC=C4)C=C3)=NN([C@H]3CC[C@H](N4CCN(CCOCCNC(=O)CN/C5=C/C=C\C6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)C2=NC=N1	C46H51N11O7	ABL1;ABL2;AURKA;BLK;CSK;CSNK1E;FYN;LATS1;LCK;LIMK1;MAP2K5;Src	P00519/P42684/O14965/P51451/P41240/P49674/P06241/O95835/P06239/P53667/Q13163/P12931	CRBN	WO-2022093742-A1
TPD-X5ITUK	SB1-G-187	SB1-G-187; 2769753-18-4; orb2279024; SCHEMBL29750164; EX-A8483; MS-31872; HY-137342; CS-0137845	CC1=CC=C(C(=O)NC2=CC=C(CN3CCN(CCCOCCOCCOCCNC(=O)CO/C4=C/C=C\C5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)C(C(F)(F)F)=C2)C=C1C#C/C1=C/N=C2/C=CC=NN12	C52H54F3N9O10	ABL1;ABL2;BLK;CDK14;CDK17;CDK5;CDK6;COQ8A;EPHA1;EPHA2;FER;FYN;GAK;IRAK1;LCK;LYN;MAP3K1;MAP3K20;MAP3K7;MAP4K2;MAP4K5;p38alpha;PDK1;PDK2;PDK3;RIPK1;RIPK2;Src;STK10;TAOK3;YES1	P00519/P42684/P51451/O94921/Q00537/Q00535/Q00534/Q8NI60/P21709/P29317/P16591/P06241/O14976/P51617/P06239/P07948/Q13233/Q9NYL2/O43318/Q12851/Q9Y4K4/Q16539/Q15118/Q15119/Q15120/Q13546/O43353/P12931/O94804/Q9H2K8/P07947	CRBN	WO-2022093742-A1
TPD-XAXURG	PD155035	PD155035	N#CCC1=CC=C(NC2=NC(NCCCNC(=O)CCCCCCNC(=O)CO/C3=C/C=C\C4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)=CC(NC3=CC(C4CC4)=NN3)=N2)C=C1	C43H48N12O7	AAK1;AURKA;BMP2K;GSK3A;GSK-3beta	Q2M2I8/O14965/Q9NSY1/P49840/P49841	CRBN	WO-2022093742-A1
TPD-XGQDA9	WO-2022093742-A1_SB1-G-192-1	.	CN1C(=O)C(C2=C(Cl)C=CC=C2Cl)CC2=CN=C(NC3=CC=C(OCCNC(=O)CCCCCCNC(=O)CO/C4=C/C=C\C5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)C=C3)N=C21	C44H44Cl2N8O9	ABL1;ABL2;AURKA;BLK;CSK;EPHA3;EPHB6;FYN;GAK;LCK;LIMK2;p38alpha;NLK;PDK1;PKMYT1;SIK2;Src;TNK2;WEE1;YES1	P00519/P42684/O14965/P51451/P41240/P29320/O15197/P06241/O14976/P06239/P53671/Q16539/Q9UBE8/Q15118/Q99640/Q9H0K1/P12931/Q07912/P30291/P07947	CRBN	WO-2022093742-A1
TPD-XLIKL5	PD155033	PD155033	O=C(CCCCCCNC(=O)COC1=C2C(=O)N(C3CCC(=O)NC3=O)C(=O)C2=CC=C1)NCCOC1=CC=C(NC2=NC=C3C=CC(=O)N(C4CC5CCC4C5)C3=N2)C=C1	C44H48N8O9	AAK1;AURKA;AURKB;CDK6;CDK9;STK17A;TTK	Q2M2I8/O14965/Q96GD4/Q00534/P50750/Q9UEE5/P33981	CRBN	WO-2022093742-A1
TPD-XPH790	SCHEMBL22845564	SCHEMBL22845564; PD155031; PD155032	NC1=C2C(C3=CC=C(OC4=CC=CC=C4)C=C3)=NN([C@H]3CC[C@H](N4CCN(CCCCCCNC(=O)CO/C5=C/C=C\C6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)CC3)C2=NC=N1	C48H54N10O7	ABL1;ABL2;BLK;CSK;FYN;LATS1;LCK;LIMK1;MAP2K5;Src	P00519/P42684/P51451/P41240/P06241/O95835/P06239/P53667/Q13163/P12931	CRBN	WO-2022093742-A1
TPD-XV1OTM	WO-2022093742-A1_SK-3-87	.	CC(C)S(=O)(=O)C1=C(NC2=NC(NC3=CC=C(C4CCN(CCOCCOCCOCCNC(=O)CNC5=C6\C(=O)N(C7CCC(=O)NC7=O)C(=O)\C6=C\C=C\5)CC4)C=C3)=NC=C2Cl)C=CC=C1	C47H56ClN9O10S	AAK1;AURKA;BLK;CDK12;CDK17;CDK2;CDK5;CDK7;CDK9;FER;ITK;LCK;LIMK2;PTK2B;WEE1	Q2M2I8/O14965/P51451/Q9NYV4/Q00537/P24941/Q00535/P50613/P50750/P16591/Q08881/P06239/P53671/Q14289/P30291	CRBN	WO-2022093742-A1
TPD-XY6KAL	PD155029	PD155029	CC(C)S(=O)(=O)C1=C(NC2=NC(NC3=CC=C(N4CCN(CCOCCOCCOCCNC(=O)CNC5=C/C=C6\C(=O)N(C7CCC(=O)NC7=O)C(=O)\C6=C\5)CC4)C=C3)=NC=C2Cl)C=CC=C1	C46H55ClN10O10S	AAK1;AURKA;BLK;CDK12;CDK17;CDK2;CDK4;CDK5;CDK6;CDK9;FER;ITK;LCK;LIMK2;PTK2B;STK10;WEE1	Q2M2I8/O14965/P51451/Q9NYV4/Q00537/P24941/P11802/Q00535/Q00534/P50750/P16591/Q08881/P06239/P53671/Q14289/O94804/P30291	CRBN	WO-2022093742-A1
TPD-XZR9ZP	SK-3-91	SK-3-91; 2769753-23-1; orb2565284; MS-31650; HY-137341; CS-0137844	CC(C)S(=O)(=O)C1=C(NC2=NC(NC3=CC=C(N4CCN(CCOCCNC(=O)CNC5=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=CC=C5)CC4)C=C3)=NC=C2Cl)C=CC=C1	C42H47ClN10O8S	AAK1;ABL1;ABL2;AKT2;AKT3;AURKA;AURKB;BCKDK;BLK;BMP2K;BMPR1A;BUB1;CDC7;CDK10;CDK12;KIAA1791;CDK14;CDK16;CDK17;CDK18;CDK2;CDK4;CDK5;CDK6;CDK7;CDK9;CSK;CSNK1D;EPHB2;EPHB4;FER;FYN;GAK;HIPK1;ITK;LATS1;LCK;LIMK1;LIMK2;LRRK2;MAP3K1;MAP3K11;MAP3K12;MAP3K21;MAP4K1;MAP4K3;MAPK6;MAPK7;MARK2;MARK4;MAST3;MKNK2;NEK2;PDK3;PLK1;PLK4;PRAG1;PRKAA1;PRKAA2;FAK;PTK2B;PTK6;RIOK2;RPS6KA1;RPS6KA6;RPS6KB1;RPS6KC1;SBK1;SIK2;Src;STK17A;STK17B;STK32C;STK33;STK40;TEC;TGFBR1;TNK1;TNK2;TRIB3;TRPM7;TTK;UHMK1;ULK1;ULK3;WEE1;YES1	Q2M2I8/P00519/P42684/P31751/Q9Y243/O14965/Q96GD4/O14874/P51451/Q9NSY1/P36894/O43683/O00311/Q15131/Q9NYV4/Q14004/O94921/Q00536/Q00537/Q07002/P24941/P11802/Q00535/Q00534/P50613/P50750/P41240/P48730/P29323/P54760/P16591/P06241/O14976/Q86Z02/Q08881/O95835/P06239/P53667/P53671/Q5S007/Q13233/Q16584/Q12852/Q5TCX8/Q92918/Q8IVH8/Q16659/Q13164/Q7KZI7/Q96L34/O60307/Q9HBH9/P51955/Q15120/P53350/O00444/Q86YV5/Q13131/P54646/Q05397/Q14289/Q13882/Q9BVS4/Q15418/Q9UK32/P23443/Q96S38/Q52WX2/Q9H0K1/P12931/Q9UEE5/O94768/Q86UX6/Q9BYT3/Q8N2I9/P42680/P36897/Q13470/Q07912/Q96RU7/Q96QT4/P33981/Q8TAS1/O75385/Q6PHR2/P30291/P07947	CRBN	WO-2022093742-A1
TPD-Y2GJ1H	PD155027	PD155027	CC(C)S(=O)(=O)C1=C(NC2=NC(NC3=CC=C(N4CCN(CCOCCNC(=O)CNC5=CC=C6C(=O)N(C7CCC(=O)NC7=O)C(=O)C6=C5)CC4)C=C3)=NC=C2Cl)C=CC=C1	C42H47ClN10O8S	AAK1;ABL2;AURKA;BLK;BMP2K;CDK12;KIAA1791;CDK17;CDK2;CDK5;CDK6;CDK7;CDK9;FER;GAK;ITK;LCK;LIMK2;PRKAA1;PTK2B;RPS6KA1;Src;WEE1	Q2M2I8/P42684/O14965/P51451/Q9NSY1/Q9NYV4/Q14004/Q00537/P24941/Q00535/Q00534/P50613/P50750/P16591/O14976/Q08881/P06239/P53671/Q13131/Q14289/Q15418/P12931/P30291	CRBN	WO-2022093742-A1
TPD-Y4ZR44	TL13-112	TL13-112; 2229037-19-6; TL 13-112; CHEMBL4213986; N-[2-[2-[2-[4-[4-[[5-chloro-4-(2-propan-2-ylsulfonylanilino)pyrimidin-2-yl]amino]-2-methyl-5-propan-2-yloxyphenyl]piperidin-1-yl]ethoxy]ethoxy]ethyl]-2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]acetamide; N-(2-(2-(2-(4-(4-((5-chloro-4-((2-(isopropylsulfonyl)phenyl)amino)pyrimidin-2-yl)amino)-5-isopropoxy-2-methylphenyl)piperidin-1-yl)ethoxy)ethoxy)ethyl)-2-((2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindolin-4-yl)amino)acetamide; orb1707795; SCHEMBL24801677; SCHEMBL29881183; GTPL10529; EPD03719; EX-A3972; BDBM50453140; AKOS037653466; AC-37753; BP-40505; DA-78497; HY-123919; CS-0087474; G16535	CC1=C(C2CCN(CCOCCOCCNC(=O)CN/C3=C/C=C\C4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)C=C(OC(C)C)C(NC2=NC=C(Cl)C(NC3=CC=CC=C3S(=O)(=O)C(C)C)=N2)=C1	C49H60ClN9O10S	FER;FAK	P16591/Q05397	CRBN	WO-2022093742-A1
TPD-YAEZZ2	2229037-04-9	2229037-04-9; TL13-12; TL 13-12; CHEMBL4217325; N-(2-(2-(2-(4-(4-((5-Chloro-4-((2-(isopropylsulfonyl)phenyl)amino)pyrimidin-2-yl)amino)-3-methoxyphenyl)piperazin-1-yl)ethoxy)ethoxy)ethyl)-2-((2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindolin-4-yl)amino)acetamide; N-[2-[2-[2-[4-[4-[[5-Chloro-4-(2-propan-2-ylsulfonylanilino)pyrimidin-2-yl]amino]-3-methoxyphenyl]piperazin-1-yl]ethoxy]ethoxy]ethyl]-2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]acetamide; orb1707794; SCHEMBL21844551; SCHEMBL29881935; GLXC-21967; EPD03704; EX-A3712; BDBM50453141; AKOS037653455; AC-36720; BP-40495; DA-58607; TL13-12?; HY-122582; CS-0087204; G16537; N-[2-[2-[2-[4-[4-[[5-Chloro-4-(2-propan-2-ylsulfonylanilino)pyrimidin-2-yl]amino]-3-methoxyphenyl]piperazin-1-yl]ethoxy]ethoxy]ethyl ]-2-[[2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindol-4-yl]amino]acetamide	COC1=CC(N2CCN(CCOCCOCCNC(=O)CN/C3=C/C=C\C4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)=CC=C1NC1=NC=C(Cl)C(NC2=CC=CC=C2S(=O)(=O)C(C)C)=N1	C45H53ClN10O10S	AURKA;FER;PRK2	O14965/P16591/Q9HC23	CRBN	WO-2022093742-A1
TPD-YHMMKO	SCHEMBL23015897	SCHEMBL23015897; PD155026	CC1=CC=C(C(=O)NC2=CC=C(CN3CCN(CCOCCOCCNC(=O)CNC4=CC=CC5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)CC3)C(C(F)(F)F)=C2)C=C1C#CC1=CN=C2C=CC=NN12	C49H49F3N10O8	BLK;CDK5;FER;GAK;IRAK1;LCK;MAP4K2;p38alpha;RIPK1;Src	P51451/Q00535/P16591/O14976/P51617/P06239/Q12851/Q16539/Q13546/P12931	CRBN	WO-2022093742-A1
TPD-YNDT9A	PD155025	PD155025	CC(C)(C)C1=NN(C2=CC=C3N=CC=CC3=C2)C(NC(=O)NC2=CC=C(OC3=CC=NC(C(=O)NCCOCCOCCNC(=O)CN/C4=C/C=C\C5=C4C(=O)N(C4CCC(=O)NC4=O)C5=O)=C3)C=C2F)=C1	C50H50FN11O10	CDK4;LIMK1;MAP3K20;p38alpha;MAST3	P11802/P53667/Q9NYL2/Q16539/O60307	CRBN	WO-2022093742-A1
TPD-YQ1DHF	WO-2022093742-A1_TL13-97	.	CC(C)S(=O)(=O)C1=CC=CC=C1NC1=NC(NC2=CC=C(N3CCN(CCOCCOCCC(=O)NCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)CC3)C=C2)=NC=C1Cl	C45H53ClN10O9S	AAK1;ABL2;AURKA;AURKB;BLK;BUB1B;KIAA1791;CDK17;CDK2;CDK4;CDK5;CDK6;CDK7;CDK9;FER;ITK;LCK;LIMK1;LIMK2;MAP3K11;MARK4;PLK4;PRKAA1;Src;STK10;STK38;TEC;TNK2;ULK1;ULK3;WEE1	Q2M2I8/P42684/O14965/Q96GD4/P51451/O60566/Q14004/Q00537/P24941/P11802/Q00535/Q00534/P50613/P50750/P16591/Q08881/P06239/P53667/P53671/Q16584/Q96L34/O00444/Q13131/P12931/O94804/Q15208/P42680/Q07912/O75385/Q6PHR2/P30291	CRBN	WO-2022093742-A1
TPD-YQJPNA	SCHEMBL22520938	SCHEMBL22520938; TMX-1160	NC(=O)C1=C(F)C=CC=C1NC1=C(Br)C=NC(NC2CCN(S(=O)(=O)CCNC(=O)CCCCCCCCO/C3=C/C=C\C4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)CC2)=N1	C40H47BrFN9O9S	AURKA;CDK1;CDK12;CDK16;CDK17;CDK2;CDK4;CDK5;CDK6;CDK7;CDK9;MAPK10;MAPK8;MAPK9;RPS6KA1	O14965/P06493/Q9NYV4/Q00536/Q00537/P24941/P11802/Q00535/Q00534/P50613/P50750/P53779/P45983/P45984/Q15418	CRBN	WO-2022093742-A1
TPD-YSZ869	TMX-2138	TMX-2138; 2488892-07-3; orb2945745; SCHEMBL22500899; SCHEMBL29392494; HY-164906	NC(=O)C1=C(NC2=NC(NC3=CC=C(S(=O)(=O)NCCOCCOCCOCCOCCNC4=C5C(=O)N(C6CCC(=O)NC6=O)C(=O)C5=CC=C4)C=C3)=NC=C2Br)C=CC=C1F	C40H43BrFN9O11S	AAK1;AURKA;AURKB;CDK1;CDK12;CDK16;CDK17;CDK2;CDK5;CDK7;CDK9;CLK1;FER;GSK3A;GSK-3beta;IRAK3;MAP3K11;MAPK8;MAPK9;NUAK1;PRKAA1;PRKAA2;PTK2B;RPS6KA1;RPS6KA3;STK33;STK38;TTK	Q2M2I8/O14965/Q96GD4/P06493/Q9NYV4/Q00536/Q00537/P24941/Q00535/P50613/P50750/P49759/P16591/P49840/P49841/Q9Y616/Q16584/P45983/P45984/O60285/Q13131/P54646/Q14289/Q15418/P51812/Q9BYT3/Q15208/P33981	CRBN	WO-2022093742-A1
TPD-Z3KHRH	CHEMBL5409959	CHEMBL5409959; TMX-2172; 2488892-09-5; orb2815195; SCHEMBL22520949; BDBM50622456; HY-155218	CC1=C(NC2=NC=C(Br)C(NC3=C(C(N)=O)C(F)=CC=C3)=N2)C=CC(S(=O)(=O)NCCOCCOCCOCCOCCNC2=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=CC=C2)=C1	C41H45BrFN9O11S	AURKA;AURKB;CDK1;CDK2;CDK5;MAPK8;MAPK9;FAK;RPS6KA1;RPS6KA3;STK33;TTK	O14965/Q96GD4/P06493/P24941/Q00535/P45983/P45984/Q05397/Q15418/P51812/Q9BYT3/P33981	CRBN	WO-2022093742-A1
TPD-Z4RCIY	WO-2022093742-A1_TMX-02-174	.	CC1=C(S(=O)(=O)N/C=C/OCCOCCOCCOCCNC2=C3C(=O)N(C4CCC(=O)NC4=O)C(=O)C3=CC=C2)C=CC(NC2=NC=C(Br)C(NC3=C(C(N)=O)C(F)=CC=C3)=N2)=C1	C41H43BrFN9O11S	AAK1;AURKA;AURKB;CDK1;CDK12;CDK16;CDK17;CDK2;CDK5;CDK7;CDK9;CLK1;FER;GSK3A;GSK-3beta;IRAK3;MAP3K11;MAPK8;MAPK9;NEK1;NEK3;NEK4;NEK9;NUAK1;PRKAA1;PRKAA2;FAK;PTK2B;RPS6KA1;RPS6KA3;RPS6KA4;STK33;STK35;STK38;TBK1;TEC;TTK;WEE1	Q2M2I8/O14965/Q96GD4/P06493/Q9NYV4/Q00536/Q00537/P24941/Q00535/P50613/P50750/P49759/P16591/P49840/P49841/Q9Y616/Q16584/P45983/P45984/Q96PY6/P51956/P51957/Q8TD19/O60285/Q13131/P54646/Q05397/Q14289/Q15418/P51812/O75676/Q9BYT3/Q8TDR2/Q15208/Q9UHD2/P42680/P33981/P30291	CRBN	WO-2022093742-A1
TPD-ZEIL94	WH-10417-099	WH-10417-099; 2769753-42-4; orb2278910; SCHEMBL29750498; MS-31889; HY-137340; CS-0137842; F82759	NC1=C(C2=C/C=C3/C(=O)NCC/C3=C\2)C=C(C2=CC=C(S(=O)(=O)N(CCCNC(=O)CCOCCOCCOCCOCCOCCNC3=C4C(=O)N(C5CCC(=O)NC5=O)C(=O)C4=CC=C3)C3CC3)C=C2)C=N1	C52H62N8O13S	CDK14;CSNK1A1;CSNK1D;CSNK1E;GSK3A;GSK-3beta;LIMK2;MAP3K1;MINK1;NUAK1;PAK4;PIM2;STK10;STK17B;STK35;STK4	O94921/P48729/P48730/P49674/P49840/P49841/P53671/Q13233/Q8N4C8/O60285/O96013/Q9P1W9/O94804/O94768/Q8TDR2/Q13043	CRBN	WO-2022093742-A1
TPD-ZHRB0P	SCHEMBL22580803	SCHEMBL22580803; PD155127	NC1=C(C2=CC=C3C(=O)NCCC3=C2)C=C(C2=C(F)C=C(S(=O)(=O)N(CCCNC(=O)CCOCCOCCOCCOCCOCCN/C3=C/C=C\C4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)C3CC3)C=C2)C=N1	C52H61FN8O13S	CDK14;CSNK1D;GSK3A;GSK-3beta;NUAK1;PIM2;STK17B;STK35;STK4	O94921/P48730/P49840/P49841/O60285/Q9P1W9/O94768/Q8TDR2/Q13043	CRBN	WO-2022093742-A1
TPD-ZI9VW8	WO-2022093742-A1_YKL-06-102	.	CC(=O)C1=C(C)C2=CN=C(NC3=CC=C(N4CCN(CC(=O)NCCOCCOCCOCCN/C5=C/C=C\C6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C=N3)C=C2N(C2CCCC2)C1=O	C48H58N10O10	CDK4;CDK6;WEE1	P11802/Q00534/P30291	CRBN	WO-2022093742-A1
TPD-ZIUHMY	2414418-49-6	2414418-49-6; Pomalidomide-C3-adavosertib; ZNL-02-096; ZNL 02-096; 4-((3-(4-(4-((2-allyl-1-(6-(2-hydroxypropan-2-yl)pyridin-2-yl)-3-oxo-2,3-dihydro-1H-pyrazolo[3,4-d]pyrimidin-6-yl)amino)phenyl)piperazin-1-yl)propyl)amino)-2-(2,6-dioxopiperidin-3-yl)isoindoline-1,3-dione; 4-((3-(4-(4-((2-Allyl-1-(6-(2-hydroxypropan-2-yl)pyridin-2-yl)-3-oxo-2,3-dihydro-1H-pyrazolo[3,4-d]pyrimidin-6-yl)amino)phenyl)piperazin-1-yl)propyl)amino)-2-(2,6-dioxopiperidin-3-yl)isoindolinedione; orb1690088; CHEMBL4638510; SCHEMBL24257345; SCHEMBL29986571; GLXC-21847; EX-A5766; ZNL-02-09; AKOS040758513; DA-66816; TS-08980; HY-133618; CS-0128444	C=CCN1C(=O)C2=CN=C(NC3=CC=C(N4CCN(CCCN/C5=C/C=C\C6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)N=C2N1C1=NC(C(C)(C)O)=CC=C1	C42H45N11O6	COQ8A;MKNK2;PAK4;PDK1;PDK2;PDK3;PRKCI;TBCK;WEE1	Q8NI60/Q9HBH9/O96013/Q15118/Q15119/Q15120/P41743/Q8TEA7/P30291	CRBN	WO-2022093742-A1
TPD-ZTC3A3	PD155126	PD155126	CN1C2=NC(NC3=CC=C(N4CCN(C(=O)CCOCCN/C5=C/C=C\C6=C5C(=O)N(C5CCC(=O)NC5=O)C6=O)CC4)C=C3)=NC=C2NC(=O)C2=C1C=CC=C2	C40H40N10O7	BLK;LIMK1;LIMK2;STK17A;TNK2	P51451/P53667/P53671/Q9UEE5/Q07912	CRBN	WO-2022093742-A1
TPD-ZVVVHB	WO-2022093742-A1_ZZ-1-31B	.	CC1=C(C2=CC=C(CNC(=O)[C@@H]3C[C@@H](O)CN3C(=O)[C@@H](NC(=O)CCOCCOCCOCCN3CCC(C(=O)NC4=NC=C(SCC5=NC=C(C(C)(C)C)O5)S4)CC3)C(C)(C)C)C=C2)SC=N1	C48H68N8O9S3	CDK9;CLK1	P50750/P49759	VHL	WO-2022093742-A1
TPD-ZZB0NE	WO-2022093742-A1_TL12-186	.	CC(C)S(=O)(=O)C1=CC=CC=C1NC1=C(Cl)C=NC(NC2=CC=C(N3CCN(CCOCCOCCNC(=O)CNC4=C5C(=O)N(C6CC(=O)NC6=O)C(=O)C5=CC=C4)CC3)C=C2)=N1	C43H49ClN10O9S	AAK1;ABL1;AURKA;AURKB;BLK;BMPR1A;BUB1;BUB1B;CDK10;CDK12;KIAA1791;CDK17;CDK2;CDK4;CDK5;CDK6;CDK7;CDK9;COQ8A;COQ8B;CSNK1D;CSNK1E;EEF2K;FER;FLT1;GAK;HASPIN;IRAK4;ITK;LCK;LIMK1;LIMK2;MAP3K11;MAP3K21;MAP4K1;MAP4K3;MAPK6;MAPK7;MARK2;MARK4;NEK2;NLK;PDK2;PLK4;PRAG1;PRKAA1;PTK2B;RIOK2;RPS6KA1;SIK2;Src;STK10;STK17A;STK35;TEC;TNK2;ULK1;ULK3;WEE1;YES1	Q2M2I8/P00519/O14965/Q96GD4/P51451/P36894/O43683/O60566/Q15131/Q9NYV4/Q14004/Q00537/P24941/P11802/Q00535/Q00534/P50613/P50750/Q8NI60/Q96D53/P48730/P49674/O00418/P16591/P17948/O14976/Q8TF76/Q9NWZ3/Q08881/P06239/P53667/P53671/Q16584/Q5TCX8/Q92918/Q8IVH8/Q16659/Q13164/Q7KZI7/Q96L34/P51955/Q9UBE8/Q15119/O00444/Q86YV5/Q13131/Q14289/Q9BVS4/Q15418/Q9H0K1/P12931/O94804/Q9UEE5/Q8TDR2/P42680/Q07912/O75385/Q6PHR2/P30291/P07947	CRBN	WO-2022093742-A1