TPD ID Activity Type Target Symbols Target IDs Cell Line Activity TPD-7WEF5B DC50 BRD4 O60885 HEK293 BRD4-HiBiT cell line 4nM TPD-RNQK6K IC50 E2F2 Q14209 HepG2 0.12μM TPD-RNQK6K IC50 E2F2 Q14209 HepG2 0.18μM TPD-1730LX EC50 CCNK O75909 HEK293T-Cas9 0.16μM TPD-1730LX EC50 CCNK O75909 HEK293T-Cas9 cells_DDB1(knock out) 1.12μM TPD-H36FEP AC50 STING Q86WV6 THP1-Dual 5.2μM TPD-UYX5KC EC50 CDK12 Q9NYV4 A549 1.9mM TPD-UYX5KC DC50 CDK12 Q9NYV4 HEK293T 0.132μM TPD-Q90952 EC50 GSPT2 Q8IYD1 . 0.2-4.8μM TPD-Q90952 DC50 GSPT2 Q8IYD1 RKO <1μM TPD-GP3QEF DC50 . . AML(KG-1) ≤10nM TPD-3GSS6I IC50 eRF1 P62495 HeLa RNF14 <10μM TPD-JFBQFN KDapp RBM39 Q14498 . 3.8μM TPD-JFBQFN EC50 RBM39 Q14498 . 0.74μM TPD-JFBQFN EC50 RBM23 Q86U06 . 1.0μM TPD-JFBQFN Ki . . . 2.9μM TPD-PCBVIQ MEC AR/AR-V7 P10275/P10275-3 22Rv1 cells-AR-HiBit 1.25μM TPD-PCBVIQ Dmax(20 μM) AR/AR-V7 P10275/P10275-3 22Rv1 cells-AR-HiBit 64.40% TPD-EBH1OJ EC50 . . . 9μM TPD-EBH1OJ EC50 . . . 45μM TPD-EBH1OJ EC50 . . . 107μM TPD-EBH1OJ EC50 . . . 253μM TPD-EBH1OJ EC50 . . . 187μM TPD-OTZLID GI50 . . . ≤100nmol/L TPD-OTZLID EC50 MEK1/ARAF Q02750/P10398 . 1.2nM TPD-OTZLID EC50 MEK1/BRAF Q02750/P15056 . 3.5nM TPD-OTZLID EC50 MEK1/CRAF Q02750/P04049 . 2.8nM TPD-T50FF4 IC50 PDE3A Q14432 . 30-80nM TPD-T50FF4 EC50 PDE3A Q14432 HeLa ~4nM TPD-5QPVXN EC50 HDAC1/HDAC2 Q13547/Q92769 . 542nM TPD-5QPVXN KD HDAC1/HDAC2 Q13547/Q92769 . 16nM TPD-5QPVXN IC50 HDAC1/HDAC2 Q13547/Q92769 K562 ~100nM TPD-L7AVW8 IC50 TrkA P04629 . 199nM TPD-W2HR7T IC50 . . PFSK-1 0.15nM TPD-W2HR7T IC50 . . HeLa 1nM TPD-3HGBX2 DC50 GSPT1 P15170 U937 35nM TPD-3HGBX2 IC50 . . U937 0.019μM TPD-3HGBX2 IC50 . . Molt-4 0.006μM TPD-3HGBX2 IC50 . . MV-4-11 0.027μM TPD-G1IE4T IC50 . . KURAMOCHI >>10μM TPD-G1IE4T IC50 . . COV 504 >>10μM TPD-Z1X484 DC50 ZBTB16 Q05516 HT-1080 0.47nM TPD-Z1X484 Ymin ZBTB16 Q05516 HT-1080 28 TPD-BVQ43A DC50 ZBTB16 Q05516 HT-1080 103nM TPD-BVQ43A Ymin ZBTB16 Q05516 HT-1080 37 TPD-VO0OTD EC50 SMAD4/SMAD3 Q13485/P84022 HEK293T 3.9±1.0μM TPD-VO0OTD EC50 SMAD4/SMAD3 Q13485/P84022 KBM7-WT 2.1±0.7μM TPD-7S830T IC50 . . U937 4.49μM TPD-7S830T IC50 . . OCI-AML-2 2.64μM TPD-7S830T IC50 . . K562 16.74μM TPD-ZR06I6 EC50 . . AML(KG-1) 0.46nM TPD-ZR06I6 EC50 . . TMD-8 5.2nM TPD-ZR06I6 EC50 . . HFL-1 0.011μM TPD-ZR06I6 EC50 . . VERO >1μM TPD-ZR06I6 Dmax(10nM) GSPT1 P15170 AML(KG-1) >95% TPD-ZR06I6 Dmax(10nM) GSPT1 P15170 TMD-8 80% TPD-ZR06I6 IC50 . . . 31.6μM TPD-ZR06I6 DC50 GSPT1 P15170 AML(KG-1) 0.269nM TPD-ZR06I6 DC50 GSPT1 P15170 TMD-8 5.8nM TPD-2459CI EC50 HIV-1 Integrase P12497 HeLa TZM-bl 12nM TPD-2459CI KD HIV-1 Integrase P12497 . ~5nM TPD-KW5UMU DC50 PDE6D O43924 Molt-4 <200nM TPD-3V2A7F DC50 CK1α P48729 Molt-4 <200nM TPD-SPNAYS KD 14-3-3σ P31947 . 0.60±0.10μM TPD-SPNAYS KD . . . 0.81±0.55μM TPD-SPNAYS IC50 . . . 3.2±0.5μM TPD-SPNAYS EC50 14-3-3σ P31947 . 67.1±41.1μM TPD-SJT3DV GI50 CDK12 Q9NYV4 Mino 0.010±0.001μM TPD-SJT3DV GI50 CDK12 Q9NYV4 UPF1H 0.010±0.002μM TPD-SJT3DV GI50 CDK12 Q9NYV4 NU-DUL-1 0.015μM TPD-SJT3DV GI50 CDK12 Q9NYV4 DB 0.020μM TPD-SJT3DV GI50 CDK12 Q9NYV4 OCI-LY2 0.011μM TPD-SJT3DV GI50 CDK12 Q9NYV4 OCI-LY19 0.465μM TPD-SJT3DV GI50 CDK12 Q9NYV4 U2932 0.055μM TPD-SJT3DV GI50 CDK12 Q9NYV4 SU-DHL4 0.028μM TPD-SJT3DV GI50 CDK12 Q9NYV4 RIVA 0.054μM TPD-SJT3DV IC50 . . . 0.004±0.001μM TPD-SJT3DV IC50 . . . >1μM TPD-SJT3DV IC50 . . . 0.039μM TPD-SJT3DV IC50 . . . 0.020μM TPD-SJT3DV IC50 . . . 0.064μM TPD-SJT3DV IC50 . . . 0.022μM TPD-9Y0C12 EC50 . . U2OS 2.9μM TPD-9Y0C12 DC50 CCNK/CDK12 O75909/Q9NYV4 A549 5.8μM TPD-AVN0IQ DC50 CK1α P48729 HEK293 6nM TPD-AVN0IQ IC50 CK1α P48729 MOLM-13 13nM TPD-AVN0IQ IC50 CK1α P48729 UCSD-AML1 0.844μM TPD-CUTKY4 IC50 . . TSC02 8.4μM TPD-CUTKY4 IC50 . . TSC03 1.0μM TPD-CUTKY4 IC50 . . TSC08 0.5μM TPD-CUTKY4 IC50 . . TSC14 0.9μM TPD-CUTKY4 IC50 . . TSC20 1.5μM TPD-CUTKY4 IC50 . . TSC23 11.8μM TPD-CUTKY4 IC50 . . TSC54 50.0μM TPD-YANNI5 IC50 MDM2 Q00987 . 33nM TPD-YANNI5 IC50 MDMX O15151 . 41nM TPD-YANNI5 KD MDMX/MDM2 O15151/Q00987 . 78nM TPD-C00IFX EC50 BCL6 P41182 . 64nM TPD-C00IFX KD BCL6 P41182 . 0.2μM TPD-MN1BRU KD 14-3-3-like protein E/PMA2 O49997/P19657 . 80μM TPD-9LTVEB KD 14-3-3-like protein E/PMA2 O49997/P19657 . 1.8μM TPD-OGMJJO EC50 . . . 206±54μM TPD-OGMJJO EC50 . . . 246±17μM TPD-OGMJJO EC50 . . . 129±33μM TPD-OGMJJO KD(500μM) β-Catenin P35222 . 68.0nM TPD-OGMJJO KD(250μM) β-Catenin P35222 . 78.1nM TPD-OGMJJO KD(125μM) β-Catenin P35222 . 143nM TPD-OGMJJO KD(62.5μM) β-Catenin P35222 . 244nM TPD-OGMJJO KD(0μM) β-Catenin P35222 . 689nM TPD-OGMJJO KD(500μM) β-Catenin P35222 . 4.8nM TPD-OGMJJO KD(250μM) β-Catenin P35222 . 5.8nM TPD-OGMJJO KD(125μM) β-Catenin P35222 . 4.5nM TPD-OGMJJO KD(62.5μM) β-Catenin P35222 . 4.5nM TPD-OGMJJO KD(0μM) β-Catenin P35222 . 4.8nM TPD-WBJSWU EC50 β-Catenin P35222 . 22.9±1.4μM TPD-WBJSWU KD β-Catenin P35222 . 54.8nM TPD-EZCI8K EC50 β-Catenin P35222 . 0.062±0.003μM TPD-EZCI8K KD β-Catenin P35222 . 0.6nM TPD-ZFGGFF EC50 β-Catenin P35222 . 0.163±0.006μM TPD-FJZ4T1 EC50 β-Catenin P35222 . 6.5±0.3nM TPD-FJZ4T1 KD β-Catenin P35222 . 0.4nM TPD-W2H9MC EC50 β-Catenin P35222 . 3.8±0.2nM TPD-1S2B5E CC50 MERS-CoV N-NTD K9N4V7 Vero E6 459.69μM TPD-1S2B5E EC50 MERS-CoV N-NTD K9N4V7 Vero E6 >100μM TPD-LAEQUR CC50 MERS-CoV N-NTD K9N4V7 Vero E6 569.77μM TPD-LAEQUR EC50 MERS-CoV N-NTD K9N4V7 Vero E6 >100μM TPD-CYUYFJ EC50 14-3-3β/CFTR P31946/P13569 . 36.1μM TPD-CYUYFJ KD 14-3-3β/CFTR P31946/P13569 . 0.056μM TPD-RT3T0Y IC50 PD-L1 Q9NZQ7 . 0.018μM TPD-G5SRU3 IC50 PD-1/PD-L1 Q15116/Q9NZQ7 . 33.65μM TPD-RC4V3F IC50 PD-1/PD-L1 Q15116/Q9NZQ7 . 22.35μM TPD-QQJ9IU KD CDC34A/Polyubiquitin-C P49427/P0CG48 . 12.2±2.6μM TPD-QQJ9IU KD CDC34A/Polyubiquitin-C P49427/P0CG48 . 14μM TPD-PQHOHR EC50 TTR P02766 . 2.7-3.2μM TPD-PQHOHR KD(high-affinity site) TTR P02766 . 3nM TPD-PQHOHR KD(lbinding affinitiesbinding affinitiesow-affinity site) TTR P02766 . 278nM TPD-4AM3TL KD USP7 Q93009 . 7.58±1.24μmol/L TPD-4AM3TL KD p53 P04637 . 4.39±0.75μmol/L TPD-EQXRZ7 EC50 14-3-3γ/SLP76 P61981/Q13094 . 19.1±7.7μM TPD-EQXRZ7 KD 14-3-3γ/SLP76 P61981/Q13094 . 3.3× TPD-EQXRZ7 SPR RU 14-3-3γ/SLP76 P61981/Q13094 . 66.40% TPD-AMC1OL EC50 14-3-3γ/SLP76 P61981/Q13094 . 18.6±5.5μM TPD-AMC1OL KD 14-3-3γ/SLP76 P61981/Q13094 . 4.1× TPD-AMC1OL SPR RU 14-3-3γ/SLP76 P61981/Q13094 . 67.60% TPD-B5KR2E EC50 14-3-3γ/SLP76 P61981/Q13094 . 14.4±1.9μM TPD-B5KR2E KD 14-3-3γ/SLP76 P61981/Q13094 . 10× TPD-B5KR2E SPR RU 14-3-3γ/SLP76 P61981/Q13094 . 66.90% TPD-3KUOHW EC50 14-3-3γ/SLP76 P61981/Q13094 . 17.4±4.9μM TPD-3KUOHW KD 14-3-3γ/SLP76 P61981/Q13094 . 3.4× TPD-3KUOHW SPR RU 14-3-3γ/SLP76 P61981/Q13094 . 57.10% TPD-XKXXE1 EC50 14-3-3γ/SLP76 P61981/Q13094 . 71.1±23.9μM TPD-XKXXE1 KD 14-3-3γ/SLP76 P61981/Q13094 . 4.7× TPD-PNTDM4 EC50 14-3-3γ/SLP76 P61981/Q13094 . 33.5±10.7μM TPD-PKT1A5 EC50 14-3-3γ/SLP76 P61981/Q13094 . 5.3±1.9μM TPD-PKT1A5 KD 14-3-3γ/SLP76 P61981/Q13094 . 4.4× TPD-PKT1A5 SPR RU 14-3-3γ/SLP76 P61981/Q13094 . 57.70% TPD-BPKF2E EC50 14-3-3γ/SLP76 P61981/Q13094 . 69.1±22.6μM TPD-BPKF2E EC50 14-3-3ζ/p27 P63104/P46527 . 53.9±17.1μM TPD-BPKF2E KD 14-3-3γ/SLP76 P61981/Q13094 . 3.5× TPD-BPKF2E SPR RU 14-3-3γ/SLP76 P61981/Q13094 . 61.20% TPD-VC0ZEK EC50 14-3-3γ/SLP76 P61981/Q13094 . 24.5±5.8μM TPD-VC0ZEK EC50 14-3-3ζ/p27 P63104/P46527 . 5.8±2.2μM TPD-VC0ZEK KD 14-3-3γ/SLP76 P61981/Q13094 . 11× TPD-VC0ZEK SPR RU 14-3-3γ/SLP76 P61981/Q13094 . 58.70% TPD-61KVG5 EC50 14-3-3γ/SLP76 P61981/Q13094 . 70.1±8.7μM TPD-61KVG5 EC50 14-3-3ζ/p27 P63104/P46527 . 16.5±10.6μM TPD-61KVG5 KD 14-3-3γ/SLP76 P61981/Q13094 . 1.4× TPD-T04VRE EC50 14-3-3γ/SLP76 P61981/Q13094 . 29.7±21.8μM TPD-T04VRE EC50 14-3-3ζ/p27 P63104/P46527 . 128.9±70.5μM TPD-YIW1S6 EC50 14-3-3γ/SLP76 P61981/Q13094 . 3.8±1.2μM TPD-YIW1S6 EC50 14-3-3ζ/p27 P63104/P46527 . 0.43±0.37μM TPD-YIW1S6 KD 14-3-3γ/SLP76 P61981/Q13094 . 5.2× TPD-YIW1S6 SPR RU 14-3-3γ/SLP76 P61981/Q13094 . 67.40% TPD-PP192J EC50 14-3-3γ/SLP76 P61981/Q13094 . 4.9±1.1μM TPD-PP192J KD 14-3-3γ/SLP76 P61981/Q13094 . 1.1× TPD-P6V7ZE EC50 14-3-3γ/SLP76 P61981/Q13094 . 21.2±11.3μM TPD-P6V7ZE EC50 14-3-3ζ/p27 P63104/P46527 . 12.6±14.4μM TPD-P6V7ZE KD 14-3-3γ/SLP76 P61981/Q13094 . 14.6× TPD-751CH5 EC50 14-3-3γ/SLP76 P61981/Q13094 . 17.1±5.2μM TPD-751CH5 EC50 14-3-3ζ/p27 P63104/P46527 . 11.6±6.1μM TPD-QGHBST EC50 14-3-3γ/SLP76 P61981/Q13094 . 1.2±0.7μM TPD-QGHBST EC50 14-3-3ζ/p27 P63104/P46527 . 80.6±53.4μM TPD-QGHBST KD 14-3-3γ/SLP76 P61981/Q13094 . 1.8× TPD-Q78N47 DR50 14-3-3σ/FOXO1 P31947/Q12778 . 0.36μM TPD-Q78N47 EC50 14-3-3σ/FOXO1 P31947/Q12778 . 5.1μM TPD-Q78N47 KD_app 14-3-3σ/FOXO1 P31947/Q12778 . 7.7nM TPD-Q78N47 KD_DMSO 14-3-3σ/FOXO1 P31947/Q12778 . 39nM TPD-N9LWHS DR50 14-3-3σ/FOXO1 P31947/Q12778 . 2.2μM TPD-N9LWHS KD_app 14-3-3σ/FOXO1 P31947/Q12778 . 10.6nM TPD-N9LWHS KD_DMSO 14-3-3σ/FOXO1 P31947/Q12778 . 42nM TPD-Q62XLU DR50 14-3-3σ/FOXO1 P31947/Q12778 . 143μM TPD-Q62XLU KD_app 14-3-3σ/FOXO1 P31947/Q12778 . 9.7nM TPD-Q62XLU KD_DMSO 14-3-3σ/FOXO1 P31947/Q12778 . 111nM TPD-954WHX DR50 14-3-3σ/CRAF P31947/P04049 . 0.58μM TPD-954WHX EC50 14-3-3σ/CRAF P31947/P04049 . 0.22μM TPD-954WHX KD_app 14-3-3σ/CRAF P31947/P04049 . 92nM TPD-954WHX KD_DMSO 14-3-3σ/CRAF P31947/P04049 . 23μM TPD-8T5U6Y DR50 14-3-3σ/CRAF P31947/P04049 . 8.78μM TPD-8T5U6Y EC50 14-3-3σ/CRAF P31947/P04049 . 1.33μM TPD-8T5U6Y KD_app 14-3-3σ/CRAF P31947/P04049 . 100nM TPD-8T5U6Y KD_DMSO 14-3-3σ/CRAF P31947/P04049 . 42μM TPD-VPD13O DR50 14-3-3σ/CRAF P31947/P04049 . 12.2μM TPD-VPD13O EC50 14-3-3σ/CRAF P31947/P04049 . 3.18μM TPD-VPD13O KD_app 14-3-3σ/CRAF P31947/P04049 . 294nM TPD-VPD13O KD_DMSO 14-3-3σ/CRAF P31947/P04049 . 23μM TPD-EUAJFT DR50 14-3-3σ/CRAF P31947/P04049 . 3.71μM TPD-EUAJFT EC50 14-3-3σ/CRAF P31947/P04049 . 13.5μM TPD-EUAJFT KD_app 14-3-3σ/CRAF P31947/P04049 . 207nM TPD-EUAJFT KD_DMSO 14-3-3σ/CRAF P31947/P04049 . 23μM TPD-AS3OHK EC50 ERα/14-3-3σ P03372/P31947 . 1μM TPD-AS3OHK KD ERα/14-3-3σ P03372/P31947 . 18nM TPD-ZGZ86Y KD FKBP12 P62942 . 0.03±0.006nM TPD-ZGZ86Y KD FKBP12.6 P68106 . 0.38±0.06nM TPD-ZGZ86Y KD FKBP51 Q13451 . 6.7±0.4nM TPD-ZGZ86Y KD FKBP52 Q02790 . 1.2±0.1nM TPD-0HBIV4 KD TAZ Q9GZV5 . 0.04±0.02μM TPD-AF17IW SF p65 Q04206 . 8 TPD-AF17IW KD_app p65 Q04206 . 1.1μM TPD-YOP33B DC50 BRD4 O60885 HEK293 12.2nM TPD-YOP33B IC50 . . MV-4-11 ~3nM TPD-YOP33B IC50(BD1) BRD4 O60885 . 10nmol/L TPD-YOP33B IC50(BD2) BRD4 O60885 . 30nmol/L TPD-4T271C Z-score KRAS P01116 HEK293T 3.2 TPD-4T271C Z-score KRAS P01116 HEK293T 2.46 TPD-PJUBUW Z-score KRAS P01116 HEK293T 4.64 TPD-U6BPLH EC50 14-3-3γ P61981 . 151μM TPD-W857PU IC50 . . HEK293 1.28mM TPD-W857PU IC50 . . P493-6 2.15μM TPD-TSH3L0 IC50 FXRα Q96RI1 . 3.4μM TPD-TSH3L0 KD FXRα Q96RI1 . 8.29μM TPD-J9DXH7 KDapp(10 μM Dose) 14-3-3γ P61981 . 2.0±0.4μM TPD-J9DXH7 KDapp(50 μM Dose) 14-3-3γ P61981 . 1.2±0.2μM TPD-J9DXH7 KDapp(100 μM Dose) 14-3-3γ P61981 . 0.9±0.1μM TPD-J9DXH7 KDapp(250 μM Dose) 14-3-3γ P61981 . 0.8±0.1μM TPD-HC4Q10 pEC50 ERα/14-3-3σ P03372/P31947 . 3.5 TPD-HC4Q10 pEC50 14-3-3η/ERα Q04917/P03372 . 3.22 TPD-HC4Q10 pIC50 14-3-3η Q04917 . 5.77 TPD-WG1VCU KDapp 14-3-3σ/ERα P31947/P03372 . 32nM TPD-WG1VCU EC50 14-3-3σ P31947 . 87nM TPD-DOUHJ1 KDapp 14-3-3σ P31947 . 92nM TPD-DOUHJ1 EC50 14-3-3σ P31947 . 209nM TPD-2BCDJ2 EC50 14-3-3ζ P63104 . 120μM TPD-9K946R KD 14-3-3ζ P63104 . 16μM TPD-MJSFOH KD 14-3-3ζ P63104 . 15μM TPD-G5DV19 EC50 . . hy926 0.9μM TPD-87TGUD EC50 14-3-3β/ChREBP P31946/Q9NP71 . 5.2±0.5μM TPD-KJ3470 EC50 14-3-3β P31946 . 6.4±0.4μM TPD-UMP01K EC50 14-3-3β P31946 . 7.0±0.4μM TPD-4XYRRV IC50 PD-L1 Q9NZQ7 . 6-100nM TPD-SRSU33 IC50 PD-L1 Q9NZQ7 . 80nM TPD-TCA2AY IC50 PD-L1 Q9NZQ7 . 2.25nM TPD-PJ9SR7 EC50 14-3-3σ P31947 . 12.4±2.3μM TPD-PJ9SR7 KD 14-3-3σ P31947 . 0.08±0.001μM TPD-ICBPJY KD LFA-1 P20701 . 52nM TPD-ICBPJY KD LFA-1 P20701 . 76nM TPD-RPBZ5Q EC50 14-3-3σ/ERα P31947/P03372 . 0.7±0.05μM TPD-D5B3MA EC50 14-3-3σ/ERα P31947/P03372 . 0.9±0.05μM TPD-XEL579 EC50 14-3-3σ/ERα P31947/P03372 . 0.3±0.01μM TPD-YDAQS8 EC50 14-3-3σ/ERα P31947/P03372 . 0.2±0.01μM TPD-QLCMM7 EC50 14-3-3σ/ERα P31947/P03372 . 0.5±0.03μM TPD-R6R3XV EC50 14-3-3σ/ERα P31947/P03372 . 0.8±0.09μM TPD-Q961B5 EC50 14-3-3σ/ERα P31947/P03372 . 0.4±0.03μM TPD-2V51GW EC50 14-3-3σ/ERα P31947/P03372 . 0.4±0.04μM TPD-IH1R0J KD KRAS P01116 . 0.7μM TPD-N62V45 CC50 14-3-3γ/p65 P61981/Q04206 . 430μM TPD-N62V45 KD 14-3-3γ/p65 P61981/Q04206 . 31μM TPD-N62V45 SF 14-3-3γ/p65 P61981/Q04206 . 10.6 TPD-APWKG9 CC50 14-3-3γ/p65 P61981/Q04206 . 140μM TPD-APWKG9 KD 14-3-3γ/p65 P61981/Q04206 . 4.3μM TPD-APWKG9 SF 14-3-3γ/p65 P61981/Q04206 . 81 TPD-LBWLTC IC50 PD-1/PD-L1 Q15116/Q9NZQ7 . 254nM TPD-L7HPA4 IC50 PD-1/PD-L1 Q15116/Q9NZQ7 . 408nM TPD-UDDJ1D IC50 PD-1/PD-L1 Q15116/Q9NZQ7 . 944nM TPD-LPI685 IC50 LOX-1 P78380 CHO-Trex-hLOX1 5.4μM TPD-OSMX1L EC50 EGFR P00533 MDA-MB-468 52μM TPD-BXO7WH IC50(Pr) HCMV P16753 . 4μM TPD-BXO7WH IC50(C-A) HCMV P16753 . 33μM TPD-FZU6JQ IC50 . . MIA PaCa-2 99.33μM TPD-FZU6JQ IC50 . . hTERT-HPNE 431.1μM TPD-X74G3T IC50 . . MIA PaCa-2 137.5μM TPD-X74G3T IC50 . . hTERT-HPNE 649.9μM TPD-MYT5P6 IC50 PD-1/PD-L1 Q15116/Q9NZQ7 . 8.9nmol/L TPD-MYT5P6 KD PD-L1 Q9NZQ7 . 24.4nmol/L TPD-BXM8LE KDapp CK1α P48729 . 1122±109nM TPD-QKBHW5 KDapp CK1α P48729 . 242±15nM TPD-QKBHW5 IC50 IKZF1 Q13422 . 712±11nM(Ki=89±3nM) TPD-X0AXX0 KDapp CK1α P48729 . 608±60nM TPD-YY6X3N IC50 REV1 Q9UBZ9 . 0.78±0.16μM TPD-YY6X3N KD REV1 Q9UBZ9 . 0.42μM TPD-REZY04 IC50 TLR8 Q9NR97 HEK-Blue hTLR2-TLR1 67±10nM TPD-REZY04 KD TLR8 Q9NR97 . 0.22μM TPD-9QW02U IC50 TLR8 Q9NR97 HEK-Blue hTLR2-TLR1 0.5±0.1nM TPD-QFTKZC IC50 TLR8 Q9NR97 HEK-Blue hTLR2-TLR1 0.7±0.2nM TPD-F7TT2C DC50 WIZ O95785 HEK293T 13nM TPD-F7TT2C EC50 WIZ O95785 . 547nM TPD-SGHDD9 IC50 . . . 60nM TPD-SGHDD9 EC50 IKZF1 Q13422 DF15 1nM TPD-SGHDD9 EC50 IKZF3 Q9UKT9 DF15 0.5nM TPD-06PRMR DC50 CDK4 P11802 . 1-5μM TPD-0N0SXN DC50 BRD4 O60885 HEK293T 0.01-0.1μM TPD-4VQHQ0 EC50 CDK12/CCNK Q9NYV4/O75909 . 17±1nM TPD-3OAEPG EC50 CDK12/CCNK Q9NYV4/O75909 . 57±3nM TPD-7MPHA6 EC50 CDK12/CCNK Q9NYV4/O75909 . 13±0.3nM TPD-KFU1V0 EC50 CDK12/CCNK Q9NYV4/O75909 . 9±0.2nM TPD-Q2IZ5C EC50 CDK12/CCNK Q9NYV4/O75909 . 14±0.4nM TPD-5IKCFI EC50 CDK12/CCNK Q9NYV4/O75909 . 36±2nM TPD-SAB574 EC50 CDK12/CCNK Q9NYV4/O75909 . 169±7nM TPD-5K0POH EC50 CDK12/CCNK Q9NYV4/O75909 . 18±1nM TPD-Y2TND7 EC50 CDK12/CCNK Q9NYV4/O75909 . 28±1nM TPD-YJ29RT EC50 CDK12/CCNK Q9NYV4/O75909 . 12±1nM TPD-1LG6JA EC50 CDK12/CCNK Q9NYV4/O75909 . 15±1nM TPD-4EKW3Y EC50 CDK12/CCNK Q9NYV4/O75909 . 20±1nM TPD-NLRZ5F EC50 CDK12/CCNK Q9NYV4/O75909 . 16±1nM TPD-7MPHA6 KD(50 nM CDK12-cyclin K +100 nM DDB1) CDK12/CCNK Q9NYV4/O75909 . <1nM TPD-4VQHQ0 KD(50 nM CDK12-cyclin K +100 nM DDB1) CDK12/CCNK Q9NYV4/O75909 . 6±2nM TPD-7MPHA6 KD(10 nM CDK12-cyclin K +100 nM DDB1) CDK12/CCNK Q9NYV4/O75909 . <<1nM TPD-4VQHQ0 KD(10 nM CDK12-cyclin K +100 nM DDB1) CDK12/CCNK Q9NYV4/O75909 . 4±1nM TPD-7MPHA6 IC50 CDK12 Q9NYV4 . 117nM TPD-KFU1V0 IC50 CDK12 Q9NYV4 . 289nM TPD-Q2IZ5C IC50 CDK12 Q9NYV4 . 163nM TPD-Q2IZ5C IC50 CDK9 P50750 . 143nM TPD-Y2TND7 IC50 CDK12 Q9NYV4 . 134nM TPD-YJ29RT IC50 CDK12 Q9NYV4 . 1nM TPD-1LG6JA IC50 CDK12 Q9NYV4 . 25nM TPD-4EKW3Y IC50 CDK12 Q9NYV4 . 25nM TPD-5K0POH IC50 CDK2 P24941 . 31nM TPD-5K0POH IC50 CDK9 P50750 . 5nM TPD-F9JHWF KD 14-3-3ζ/Gab2 P63104/Q9UQC2 . 1.25±0.072μM TPD-F9JHWF KD 14-3-3ζ/Gab2 P63104/Q9UQC2 . 0.19±0.014μM TPD-YQ5GU2 AC50 G6PD P11413 . 3.3μM TPD-YQ5GU2 Amax G6PD P11413 . 160% TPD-YQ5GU2 AC50(Trp509Ala) G6PD P11413 . 0.8μM TPD-YQ5GU2 Amax(Trp509Ala) G6PD P11413 . 170% TPD-LD1R2I EC50 14-3-3ζ P63104 . 4.3±0.3μM TPD-LD1R2I S 14-3-3ζ/TASK-3 P63104/Q9NPC2 . 42(0.5 μM FC-NAc) TPD-4KZKO6 IC50 GCase P04062 . 8nM TPD-7S830T IC50 . . U266 3.8μM TPD-G1IE4T IC50 . . OVSAHO >>10μM TPD-G1IE4T IC50 . . COV 318 >>10μM TPD-G1IE4T IC50 . . COV 644 >>10μM TPD-G1IE4T IC50 . . OVISE 10μM TPD-G1IE4T IC50 . . PEO4 1μM TPD-G1IE4T IC50 . . PEO1 0.25μM TPD-2BCDJ2 KD 14-3-3ζ P63104 . 1.01mM TPD-LPI685 KD LOX-1 P78380 . 4.3μM TPD-LPI685 KD LOX-1 P78380 . 6.99μM TPD-BXO7WH EC50 HCMV P16753 HFF-1 0.8μM TPD-FZU6JQ IC50 . . PanC-1 105μM TPD-FZU6JQ IC50 . . BxPC-3 252.85μM TPD-X74G3T IC50 . . PanC-1 108.5μM TPD-X74G3T IC50 . . BxPC-3 97.88μM TPD-BXM8LE KDapp IKZF1 Q13422 . 155±33nM TPD-QKBHW5 KDapp IKZF1 Q13422 . 101±2nM TPD-QKBHW5 Ki IKZF1 Q13422 . 89±3nM TPD-X0AXX0 KDapp IKZF1 Q13422 . 96±24nM TPD-QFTKZC KD TLR8 Q9NR97 . 21nM TPD-REZY04 KD TLR8 Q9NR97 . 220nM TPD-F7TT2C EC50 . . HbF 100nM TPD-F7TT2C KD WIZ O95785 . 3.5μM±0.6μM TPD-YQ5GU2 AC50 G6PD P11413 . 4.2μM TPD-YQ5GU2 Amax G6PD P11413 . 120% TPD-1LG6JA KD(50 nM CDK12-cyclin K +100 nM DDB1) CDK12/CCNK Q9NYV4/O75909 . 2±1nM TPD-1LG6JA KD(10 nM CDK12-cyclin K +100 nM DDB1) CDK12/CCNK Q9NYV4/O75909 . 0.2±0.3nM TPD-EE3ZSG IC50 PDE3A Q14432 . 82nM TPD-TU9F23 EC50_1 . . NCI-H358 0.082nM TPD-049ESM IC50_1 . . H929 R10-1 10μM TPD-3WSCIS IC50_1 . . H929 R10-1 0.51μM TPD-J1XBDQ IC50_1 . . H929 R10-1 0.0351μM TPD-HHQA5U IC50_1 . . H929 R10-1 0.0205μM TPD-QM5UZP IC50_1 . . H929 R10-1 0.00998μM TPD-YPBY07 IC50_1 . . H929 R10-1 0.00141μM TPD-S97N5C IC50_1 . . H929 R10-1 0.0083μM TPD-8GT4MX IC50_1 . . H929 R10-1 0.0351μM TPD-N17T1H IC50_1 . . H929 R10-1 0.00213μM TPD-AE1BU7 IC50_1 . . H929 R10-1 0.00285μM TPD-5EA3Q8 IC50_1 . . H929 R10-1 0.00459μM TPD-OQ6I6N IC50_1 . . H929 R10-1 0.146μM TPD-7G52P3 IC50_1 . . H929 R10-1 0.0017μM TPD-G7IGSR IC50_1 . . H929 R10-1 0.00364μM TPD-4S932U IC50_1 . . H929 R10-1 0.0092μM TPD-H4RLX4 IC50_1 . . H929 R10-1 0.00404μM TPD-ZJNNKD IC50_1 . . H929 R10-1 0.00369μM TPD-FC6JQP IC50_1 . . H929 R10-1 0.00504μM TPD-C9O9JF IC50_1 . . H929 R10-1 0.00709μM TPD-BBJ4HQ IC50_1 . . H929 R10-1 0.0074μM TPD-2IUM4C IC50_1 . . H929 R10-1 0.056μM TPD-V5SFQ5 IC50_1 . . H929 R10-1 0.00495μM TPD-EJ6Z25 IC50_1 . . H929 R10-1 0.00354μM TPD-49N0TZ IC50_1 . . H929 R10-1 0.00177μM TPD-VAMT79 IC50_1 . . H929 R10-1 0.0033μM TPD-04YR73 IC50_1 . . H929 R10-1 0.00373μM TPD-KIJ8SV IC50_1 . . H929 R10-1 0.00623μM TPD-1IBT9K IC50_1 . . H929 R10-1 0.0067μM TPD-FZARAW IC50_1 . . H929 R10-1 0.00384μM TPD-9QEZYK IC50_1 . . H929 R10-1 0.00431μM TPD-ZHDQXN IC50_1 . . H929 R10-1 0.0263μM TPD-ID4JCD IC50_1 . . H929 R10-1 0.632μM TPD-14ZFQ7 IC50_1 . . H929 R10-1 0.17μM TPD-W0U5JO IC50_1 . . H929 R10-1 0.159μM TPD-5HJED0 IC50_1 . . H929 R10-1 5.76μM TPD-19MYS5 IC50_1 . . H929 R10-1 0.496μM TPD-LF6F98 IC50_1 . . H929 R10-1 0.0023μM TPD-EE3ZSG EC50_1 . . HeLa 1.04nM TPD-EE3ZSG EC50_2 . . SK-MEL-3 2.81nM TPD-EE3ZSG EC5-_3 . . IGR37 3.1nM TPD-EE3ZSG EC50_4 . . DKMG 22nM TPD-EE3ZSG EC50_5 . . HS578T 33nM TPD-EE3ZSG EC50_6 . . H2172 38nM TPD-EE3ZSG EC50_7 . . NCI-H196 150nM TPD-EE3ZSG EC50_8 . . A2058 38nM TPD-EE3ZSG EC50_9 . . C32 58nM TPD-EE3ZSG EC50_10 . . RVH421 140nM TPD-EE3ZSG EC50_11 . . L3.3 82nM TPD-EE3ZSG EC50_12 . . GB1 8nM TPD-TU9F23 IC50_1 KRAS-RAF P01116 . 6.545nM TPD-TU9F23 IC50_2 pERK P27361 NCI-H358 0.614nM TPD-TU9F23 IC50_3 . . NCI-H358 0.082nM TPD-TU9F23 IC50_4 . . A375 238.238nM TPD-TU9F23 EC50_2 pERK P27361 NCI-H358 0.61nM TPD-049ESM IC50_2 . . . 0.2363μM TPD-3WSCIS IC50_2 . . . 0.1725μM TPD-J1XBDQ IC50_2 . . . 0.1394μM TPD-HHQA5U IC50_2 . . . 0.09521μM TPD-QM5UZP IC50_2 . . . 0.0957μM TPD-YPBY07 IC50_2 . . . 0.06249μM TPD-S97N5C IC50_2 . . . 0.1261μM TPD-8GT4MX IC50_2 . . . 0.1008μM TPD-N17T1H IC50_2 . . . 0.04103μM TPD-AE1BU7 IC50_2 . . . 0.07604μM TPD-5EA3Q8 IC50_2 . . . 0.08595μM TPD-OQ6I6N IC50_2 . . . 0.3218μM TPD-7G52P3 IC50_2 . . . 0.05513μM TPD-G7IGSR IC50_2 . . . 0.07996μM TPD-4S932U IC50_2 . . . 0.1244μM TPD-H4RLX4 IC50_2 . . . 0.1073μM TPD-ZJNNKD IC50_2 . . . 0.09994μM TPD-FC6JQP IC50_2 . . . 0.09505μM TPD-C9O9JF IC50_2 . . . 0.09029μM TPD-V5SFQ5 IC50_2 . . . 0.06889μM TPD-EJ6Z25 IC50_2 . . . 0.07097μM TPD-49N0TZ IC50_2 . . . 0.07467μM TPD-VAMT79 IC50_2 . . . 0.07716μM TPD-04YR73 IC50_2 . . . 0.08077μM TPD-KIJ8SV IC50_2 . . . 0.06507μM TPD-1IBT9K IC50_2 . . . 0.1178μM TPD-FZARAW IC50_2 . . . 1.158μM TPD-9QEZYK IC50_2 . . . 0.03736μM TPD-ZHDQXN IC50_2 . . . 0.1946μM TPD-ID4JCD IC50_2 . . . 28μM TPD-14ZFQ7 IC50_2 . . . 0.8773μM TPD-W0U5JO IC50_2 . . . 0.502μM TPD-5HJED0 IC50_2 . . . 96.18μM TPD-19MYS5 IC50_2 . . . >100μM TPD-LF6F98 IC50_2 . . . 0.0372μM TPD-049ESM EC50_1 IKZF3 Q9UKT9 DF15 0.00751μM TPD-3WSCIS EC50_1 IKZF3 Q9UKT9 DF15 0.00289μM TPD-J1XBDQ EC50_1 IKZF3 Q9UKT9 DF15 0.001μM TPD-HHQA5U EC50_1 IKZF3 Q9UKT9 DF15 0.0005μM TPD-QM5UZP EC50_1 IKZF3 Q9UKT9 DF15 0.0003μM TPD-YPBY07 EC50_1 IKZF3 Q9UKT9 DF15 0.0001μM TPD-S97N5C EC50_1 IKZF3 Q9UKT9 DF15 0.0006μM TPD-8GT4MX EC50_1 IKZF3 Q9UKT9 DF15 0.0003μM TPD-N17T1H EC50_1 IKZF3 Q9UKT9 DF15 0.0001μM TPD-AE1BU7 EC50_1 IKZF3 Q9UKT9 DF15 0.0001μM TPD-5EA3Q8 EC50_1 IKZF3 Q9UKT9 DF15 0.0004μM TPD-OQ6I6N EC50_1 IKZF3 Q9UKT9 DF15 0.0021μM TPD-7G52P3 EC50_1 IKZF3 Q9UKT9 DF15 0.0001μM TPD-G7IGSR EC50_1 IKZF3 Q9UKT9 DF15 0.0001μM TPD-4S932U EC50_1 IKZF3 Q9UKT9 DF15 0.0002μM TPD-H4RLX4 EC50_1 IKZF3 Q9UKT9 DF15 0.0003μM TPD-ZJNNKD EC50_1 IKZF3 Q9UKT9 DF15 0.0001μM TPD-FC6JQP EC50_1 IKZF3 Q9UKT9 DF15 0.0002μM TPD-C9O9JF EC50_1 IKZF3 Q9UKT9 DF15 0.0005μM TPD-BBJ4HQ EC50_1 IKZF3 Q9UKT9 DF15 0.0007μM TPD-2IUM4C EC50_1 IKZF3 Q9UKT9 DF15 0.001μM TPD-V5SFQ5 EC50_1 IKZF3 Q9UKT9 DF15 0.0001μM TPD-EJ6Z25 EC50_1 IKZF3 Q9UKT9 DF15 0.0004μM TPD-49N0TZ EC50_1 IKZF3 Q9UKT9 DF15 0.0001μM TPD-VAMT79 EC50_1 IKZF3 Q9UKT9 DF15 0.0001μM TPD-04YR73 EC50_1 IKZF3 Q9UKT9 DF15 0.0003μM TPD-KIJ8SV EC50_1 IKZF3 Q9UKT9 DF15 0.0001μM TPD-1IBT9K EC50_1 IKZF3 Q9UKT9 DF15 0.0006μM TPD-FZARAW EC50_1 IKZF3 Q9UKT9 DF15 0.0005μM TPD-9QEZYK EC50_1 IKZF3 Q9UKT9 DF15 0.0001μM TPD-ZHDQXN EC50_1 IKZF3 Q9UKT9 DF15 0.0015μM TPD-ID4JCD EC50_1 IKZF3 Q9UKT9 DF15 >0.01μM TPD-14ZFQ7 EC50_1 IKZF3 Q9UKT9 DF15 >0.003333μM TPD-W0U5JO EC50_1 IKZF3 Q9UKT9 DF15 0.0024μM TPD-5HJED0 EC50_1 IKZF3 Q9UKT9 DF15 >0.1μM TPD-19MYS5 EC50_1 IKZF3 Q9UKT9 DF15 >0.01μM TPD-LF6F98 EC50_1 IKZF3 Q9UKT9 DF15 0.0003μM TPD-049ESM EC50_2 GSPT1 P15170 DF15 >10μM TPD-3WSCIS EC50_2 GSPT1 P15170 DF15 >10μM TPD-J1XBDQ EC50_2 GSPT1 P15170 DF15 >10μM TPD-HHQA5U EC50_2 GSPT1 P15170 DF15 >10μM TPD-QM5UZP EC50_2 GSPT1 P15170 DF15 >10μM TPD-YPBY07 EC50_2 GSPT1 P15170 DF15 >10μM TPD-S97N5C EC50_2 GSPT1 P15170 DF15 >10μM TPD-8GT4MX EC50_2 GSPT1 P15170 DF15 >10μM TPD-N17T1H EC50_2 GSPT1 P15170 DF15 >10μM TPD-AE1BU7 EC50_2 GSPT1 P15170 DF15 >10μM TPD-5EA3Q8 EC50_2 GSPT1 P15170 DF15 >10μM TPD-OQ6I6N EC50_2 GSPT1 P15170 DF15 >10μM TPD-7G52P3 EC50_2 GSPT1 P15170 DF15 >10μM TPD-G7IGSR EC50_2 GSPT1 P15170 DF15 >10μM TPD-4S932U EC50_2 GSPT1 P15170 DF15 >10μM TPD-H4RLX4 EC50_2 GSPT1 P15170 DF15 >10μM TPD-ZJNNKD EC50_2 GSPT1 P15170 DF15 >10μM TPD-FC6JQP EC50_2 GSPT1 P15170 DF15 >10μM TPD-C9O9JF EC50_2 GSPT1 P15170 DF15 >10μM TPD-V5SFQ5 EC50_2 GSPT1 P15170 DF15 >10μM TPD-EJ6Z25 EC50_2 GSPT1 P15170 DF15 >10μM TPD-49N0TZ EC50_2 GSPT1 P15170 DF15 >10μM TPD-VAMT79 EC50_2 GSPT1 P15170 DF15 >10μM TPD-04YR73 EC50_2 GSPT1 P15170 DF15 >10μM TPD-KIJ8SV EC50_2 GSPT1 P15170 DF15 >10μM TPD-1IBT9K EC50_2 GSPT1 P15170 DF15 >10μM TPD-FZARAW EC50_2 GSPT1 P15170 DF15 >10μM TPD-9QEZYK EC50_2 GSPT1 P15170 DF15 >10μM TPD-ZHDQXN EC50_2 GSPT1 P15170 DF15 >10μM TPD-ID4JCD EC50_2 GSPT1 P15170 DF15 >10μM TPD-14ZFQ7 EC50_2 GSPT1 P15170 DF15 >10μM TPD-W0U5JO EC50_2 GSPT1 P15170 DF15 >10μM TPD-5HJED0 EC50_2 GSPT1 P15170 DF15 >10μM TPD-19MYS5 EC50_2 GSPT1 P15170 DF15 >10μM TPD-LF6F98 EC50_2 GSPT1 P15170 DF15 >10μM TPD-X7M15Q IC50 CDK12 Q9NYV4 A673 123.0nM TPD-4KFLOV IC50 CDK12 Q9NYV4 A673 716.0nM TPD-JAJD6G IC50 CDK12 Q9NYV4 A673 8.0nM TPD-756JVG IC50 CDK12 Q9NYV4 A673 12.0nM TPD-82YJFQ IC50 CDK12 Q9NYV4 A673 47.0nM TPD-P665RG IC50 CDK12 Q9NYV4 A673 52.0nM TPD-TMCCYH IC50 CDK12 Q9NYV4 A673 27.0nM TPD-4MO2W7 IC50 CDK12 Q9NYV4 A673 5.7nM TPD-F1N7DJ IC50 CDK12 Q9NYV4 A673 14.9nM TPD-CQ6L7B IC50 CDK12 Q9NYV4 A673 4.3nM TPD-67VB20 IC50 CDK12 Q9NYV4 A673 6.3nM TPD-XNB4UM IC50 CDK12 Q9NYV4 A673 21.8nM TPD-MLBW70 IC50 CDK12 Q9NYV4 A673 12.2nM TPD-CZWSLZ IC50 CDK12 Q9NYV4 A673 7.3nM TPD-9OYBDK IC50 CDK12 Q9NYV4 A673 151.0nM TPD-ORBEOJ IC50 CDK12 Q9NYV4 A673 14.8nM TPD-WVFRO6 IC50 CDK12 Q9NYV4 A673 8.3nM TPD-VWUYMY IC50 CDK12 Q9NYV4 A673 16.3nM TPD-LWEP3Q IC50_5 . . CAL-62 E TPD-QHYM7Q IC50_5 . . CAL-62 C TPD-8YPO9C IC50_5 . . CAL-62 D TPD-QHYM7Q IC50_4 . . CCRF-CEM B TPD-8YPO9C IC50_4 . . CCRF-CEM C TPD-JFVBR1 IC50_14 . . Caco-2 6.64nM TPD-86YMG4 IC50_14 . . Caco-2 4.46nM TPD-BYII1J IC50 . . Colo-205 100nM-300nM TPD-OQG9UV IC50 . . Colo-205 <=100nM TPD-HDR8DR IC50 . . Daudi 44.9nM TPD-9ROWSY IC50 . . Daudi 155.4nM TPD-BYII1J IC50 . . H69 <=100nM TPD-OQG9UV IC50 . . H69 <=100nM TPD-9X6CFO IC50 . . HNT-34 26.9nM TPD-1H21BH IC50 . . HNT-34 18.0nM TPD-TVMZU7 IC50 . . HNT-34 3.6nM TPD-JFVBR1 IC50_6 . . JIMT-1 0.25nM TPD-86YMG4 IC50_6 . . JIMT-1 0.64nM TPD-JFVBR1 IC50_12 . . KB-1 0.38nM TPD-DM1J6Z IC50_12 . . KB-1 4.95nM TPD-TO9J8L EC50 CDK12 Q9NYV4 KBM7-UBE2M Knockout 0.5μM10μM TPD-L1IH7O EC50 GSPT1 P15170 HEK293_hGSPT1_HiBiT >10μM TPD-WTXATR EC50 GSPT1 P15170 HEK293_hGSPT1_HiBiT <1μM TPD-CGSB62 EC50 GSPT1 P15170 HEK293_hGSPT1_HiBiT >10μM TPD-AB7Z5C EC50 GSPT1 P15170 HEK293_hGSPT1_HiBiT >10μM TPD-NYJQLX EC50 GSPT1 P15170 HEK293_hGSPT1_HiBiT >10μM TPD-SQAS76 EC50 GSPT1 P15170 HEK293_hGSPT1_HiBiT >10μM TPD-SFYTN6 EC50 GSPT1 P15170 HEK293_hGSPT1_HiBiT 1μM10μM TPD-Q4FMBC EC50 GSPT1 P15170 HEK293_hGSPT1_HiBiT >10μM TPD-DM274L EC50 GSPT1 P15170 HEK293_hGSPT1_HiBiT >10μM TPD-0944N9 EC50 GSPT1 P15170 HEK293_hGSPT1_HiBiT >10μM TPD-TO9J8L DC50 CCNK O75909 HEK293T 0.25μM10μM TPD-PMUOQ3 DC50 CCNK O75909 HEK293T 0.25μM10μM TPD-69N22M DC50 CCNK O75909 HEK293T ≤0.25μM TPD-WJY6M2 DC50 CCNK O75909 HEK293T ≤0.25μM TPD-KKCI08 DC50 CCNK O75909 HEK293T ≤0.25μM TPD-RQOG46 DC50 CCNK O75909 HEK293T >10μM TPD-8WGVWM DC50 CCNK O75909 HEK293T >10μM TPD-E9GU2W DC50 CCNK O75909 HEK293T ≤0.25μM TPD-N5ZTQQ DC50 CCNK O75909 HEK293T >10μM TPD-39VLK3 DC50 CCNK O75909 HEK293T 0.5μM10μM TPD-PMUOQ3 EC50 CDK12 Q9NYV4 HEK293T ≤0.25μM TPD-N7LN1T EC50 CDK12 Q9NYV4 HEK293T 0.5μM100μM TPD-ZCRP9Y EC50 RBM39 Q14498 HCT-116 >100μM TPD-9NX6LS EC50 RBM39 Q14498 HCT-116 <1μM TPD-NGH0ES EC50 RBM39 Q14498 HCT-116 <1μM TPD-1BJ31G EC50 RBM39 Q14498 HCT-116 >100μM TPD-IOE4P9 EC50 RBM39 Q14498 HCT-116 >100μM TPD-1AWXXH EC50 RBM39 Q14498 HCT-116 <10μM TPD-QJS15I EC50 RBM39 Q14498 HCT-116 <10μM TPD-K9QOCR EC50 RBM39 Q14498 HCT-116 <10μM TPD-DIIVRV EC50 RBM39 Q14498 HCT-116 >100μM TPD-JS5GP5 EC50 RBM39 Q14498 HCT-116 <10μM TPD-BX0BER EC50 RBM39 Q14498 HCT-116 <10μM TPD-FVCXIY EC50 RBM39 Q14498 HCT-116 <1μM TPD-C5LZQ0 EC50 RBM39 Q14498 HCT-116 <1μM TPD-HOIDP9 EC50 RBM39 Q14498 HCT-116 <10μM TPD-ED9HVK EC50 RBM39 Q14498 HCT-116 >100μM TPD-IMVQXF EC50 RBM39 Q14498 HCT-116 <100μM TPD-SJ5WG9 EC50 RBM39 Q14498 HCT-116 <100μM TPD-T81KQC IC50 . . . >100μM TPD-ZCRP9Y IC50 . . . >100μM TPD-9NX6LS IC50 . . . <100μM TPD-NGH0ES IC50 . . . >100μM TPD-1BJ31G IC50 . . . >100μM TPD-IOE4P9 IC50 . . . >100μM TPD-1AWXXH IC50 . . . >100μM TPD-QJS15I IC50 . . . >100μM TPD-K9QOCR IC50 . . . >100μM TPD-DIIVRV IC50 . . . >100μM TPD-JS5GP5 IC50 . . . >100μM TPD-BX0BER IC50 . . . >100μM TPD-FVCXIY IC50 . . . >100μM TPD-C5LZQ0 IC50 . . . <100μM TPD-HOIDP9 IC50 . . . >100μM TPD-ED9HVK IC50 . . . >100μM TPD-IMVQXF IC50 . . . >100μM TPD-SJ5WG9 IC50 . . . >100μM TPD-LJL6E5 IC50 . . HeLa 2.533nM TPD-A0TWL8 IC50 . . HeLa 6.222nM TPD-8KRN6V IC50 . . HeLa 2.379nM TPD-67CEJ4 IC50 . . HeLa 12.3nM TPD-EPM2LQ IC50 . . HeLa 42.88nM TPD-V7K9Z5 IC50 . . HeLa 1.142nM TPD-7SK0W6 DC50 CK1α P48729 . 0.176 μM TPD-NY4ZN8 DC50 CK1α P48729 . 0.308 μM TPD-45D5EA DC50 CK1α P48729 . 0.14 μM TPD-QNPGJU DC50 CK1α P48729 . 0.293 μM TPD-VZXV7N DC50 CK1α P48729 . 0.284 μM TPD-F74CCF DC50 CK1α P48729 . 0.0658 μM TPD-M1F3XP DC50 CK1α P48729 . 0.0653 μM TPD-6EJIF1 DC50 CK1α P48729 . 0.123 μM TPD-X2NQ83 DC50 CK1α P48729 . 0.137 μM TPD-7SK0W6 Dmax CK1α P48729 . 60.80% TPD-NY4ZN8 Dmax CK1α P48729 . 64.70% TPD-45D5EA Dmax CK1α P48729 . 67.30% TPD-QNPGJU Dmax CK1α P48729 . 65.90% TPD-VZXV7N Dmax CK1α P48729 . 67.90% TPD-F74CCF Dmax CK1α P48729 . 75.20% TPD-M1F3XP Dmax CK1α P48729 . 67.90% TPD-6EJIF1 Dmax CK1α P48729 . 65.70% TPD-X2NQ83 Dmax CK1α P48729 . 66.00% TPD-YHKYZA IC50 CDK12 Q9NYV4 . 61nM TPD-J2NUX1 IC50 CDK12 Q9NYV4 . 34nM TPD-VHI46I IC50 CDK12 Q9NYV4 . 47nM TPD-RORMB2 IC50 CDK12 Q9NYV4 . 143nM TPD-NQNNBC IC50 CDK12 Q9NYV4 . 34nM TPD-9R72BZ IC50 CDK12 Q9NYV4 . 51nM TPD-GEOW37 IC50 CDK12 Q9NYV4 . 51nM TPD-GBZQ2Q IC50 CDK12 Q9NYV4 . 52nM TPD-IE9I5K IC50 CDK12 Q9NYV4 . 55nM TPD-JZWMCH IC50 CDK12 Q9NYV4 . 36nM TPD-A58J0A IC50 CDK12 Q9NYV4 . 160nM TPD-VB6UZT IC50 CDK12 Q9NYV4 . 188nM TPD-YHKYZA IC50 . . A673 2.8nM TPD-J2NUX1 IC50 . . A673 126.7nM TPD-VHI46I IC50 . . A673 16.2nM TPD-RORMB2 IC50 . . A673 6.3nM TPD-NQNNBC IC50 . . A673 1.1nM TPD-9R72BZ IC50 . . A673 3.5nM TPD-GEOW37 IC50 . . A673 1.7nM TPD-GBZQ2Q IC50 . . A673 32nM TPD-IE9I5K IC50 . . A673 1.3nM TPD-JZWMCH IC50 . . A673 8nM TPD-A58J0A IC50 . . A673 69nM TPD-VB6UZT IC50 . . A673 14.1nM TPD-161M4N DC50 IKZF1 Q13422 . 0.025nM TPD-0C3AC0 DC50 IKZF1 Q13422 . 0.065nM TPD-CCZCK1 DC50 IKZF1 Q13422 . 2.19nM TPD-161M4N Dmax IKZF1 Q13422 . 93.20% TPD-0C3AC0 Dmax IKZF1 Q13422 . 88.30% TPD-CCZCK1 Dmax IKZF1 Q13422 . 66.20% TPD-BSDGZZ DC50 IKZF1 Q13422 . 0.047nM TPD-BSDGZZ Dmax IKZF1 Q13422 . 94.80% TPD-0160HF IC50 . . HGC27 385nM TPD-NCSQTZ IC50 . . HGC27 307nM TPD-M5B3KS IC50 . . HGC27 281nM TPD-AVM1XM IC50 . . HGC27 155nM TPD-2AZYN9 IC50 . . HGC27 158nM TPD-PDEMB7 IC50 . . HGC27 379nM TPD-2VTRKM IC50 . . HGC27 341nM TPD-XM85CJ IC50 . . HGC27 266nM TPD-8KRQNX IC50 . . HGC27 251nM TPD-PDPIV3 IC50 . . HGC27 185nM TPD-L764CZ IC50 . . HGC27 160nM TPD-DZV232 IC50 . . HGC27 405nM TPD-9XGKLV IC50 . . HGC27 486nM TPD-V0430M IC50 . . HGC27 275nM TPD-GPZCVB IC50 . . HGC27 210nM TPD-A1JJVX IC50 . . HGC27 251nM TPD-G784RL IC50 . . HGC27 479nM TPD-DGL70I IC50 . . HGC27 191nM TPD-VFOKTQ IC50 . . HEK293T 256nM TPD-WVHFRJ IC50 . . HEK293T 890nM TPD-A3A4KL IC50 . . HEK293T 3752nM TPD-XC4W8H EC50 RBM39 Q14498 . <1pM TPD-I96YUR EC50 RBM39 Q14498 . <1pM TPD-ZJHFVM EC50 RBM39 Q14498 . 1pM25000nM TPD-LDKT1Q EC50 RBM39 Q14498 HCT-116 >25000nM TPD-E4F909 Dmax GSPT1 P15170 Jeko-1(100 nM) 35% TPD-8D2P1I Dmax GSPT1 P15170 Jeko-1(100 nM) 29.80% TPD-V3VU9H Dmax GSPT1 P15170 Jeko-1(100 nM) 31% TPD-VZ7FM2 Dmax GSPT1 P15170 Jeko-1(100 nM) 89% TPD-QA0V78 Dmax GSPT1 P15170 Jeko-1(100 nM) 93% TPD-RI0OBT Dmax GSPT1 P15170 Jeko-1(100 nM) 21% TPD-9X6CFO Dmax GSPT1 P15170 Jeko-1(100 nM) 79.90% TPD-1H21BH Dmax GSPT1 P15170 Jeko-1(100 nM) 18.80% TPD-TVMZU7 Dmax GSPT1 P15170 Jeko-1(100 nM) 82% TPD-BEFNZO Dmax GSPT1 P15170 Jeko-1(100 nM) 97.80% TPD-E4F909 Dmax GSPT1 P15170 Jeko-1(10μM) 53% TPD-8D2P1I Dmax GSPT1 P15170 Jeko-1(10μM) 74.80% TPD-V3VU9H Dmax GSPT1 P15170 Jeko-1(10μM) 88% TPD-VZ7FM2 Dmax GSPT1 P15170 Jeko-1(10μM) 93% TPD-QA0V78 Dmax GSPT1 P15170 Jeko-1(10μM) 90% TPD-RI0OBT Dmax GSPT1 P15170 Jeko-1(10μM) 85% TPD-9X6CFO Dmax GSPT1 P15170 Jeko-1(10μM) 92.70% TPD-1H21BH Dmax GSPT1 P15170 Jeko-1(10μM) 84.10% TPD-TVMZU7 Dmax GSPT1 P15170 Jeko-1(10μM) 97% TPD-BEFNZO Dmax GSPT1 P15170 Jeko-1(10μM) 98.70% TPD-EZV37J EC50 . . MOLM-13 ≤1μM TPD-GUOPPU EC50 . . MOLM-13 1μM1μM TPD-PQS0TU DC50 CK1α P48729 HEK293 ≤0.1μM TPD-VVE5NA DC50 CK1α P48729 HEK293 ≤0.1μM TPD-478N5Y DC50 CK1α P48729 HEK293 ≤0.1μM TPD-9GDXH1 DC50 CK1α P48729 HEK293 0.1μM1μM TPD-0VO2DC DC50 CK1α P48729 HEK293 ≤0.1μM TPD-9Q0BWF DC50 CK1α P48729 HEK293 0.1μM1μM TPD-VVE5NA IC50 . . . 0.1μM1μM TPD-8VRRVB IC50 . . . 0.1μM1μM TPD-8VRRVB DC50 CK1α P48729 HEK293 0.1μM1μM TPD-JYGSJ0 DC50 CK1α P48729 HEK293 ≤0.1μM TPD-WQCYQN IC50 . . MM1.S <15nM TPD-0JUP4L IC50 . . MM1.S <15nM TPD-S5T74N IC50 . . MM1.S <15nM TPD-648XEH IC50 . . MM1.S 30nM≤x<150nM TPD-CA5S74 IC50 . . MM1.S 30nM≤x<150nM TPD-PMLPXL IC50 . . MM1.S 15nM≤x<30nM TPD-0FKNQX IC50 . . MM1.S <15nM TPD-7RLEZE IC50 . . MM1.S 30nM≤x<150nM TPD-Z5VSAE IC50 . . MM1.S <15nM TPD-0P3G9G IC50 . . MM1.S 15nM≤x<30nM TPD-X0EIM0 IC50 . . MM1.S ≥150nM TPD-W9L5ZI IC50 . . MM1.S 30nM≤x<150nM TPD-WQCYQN IC50 . . Mino <60nM TPD-0JUP4L IC50 . . Mino 60nM≤x<120nM TPD-S5T74N IC50 . . Mino <60nM TPD-648XEH IC50 . . Mino ≥120nM TPD-CA5S74 IC50 . . Mino ≥120nM TPD-PMLPXL IC50 . . Mino 60nM≤x<120nM TPD-0FKNQX IC50 . . Mino ≥120nM TPD-Z5VSAE IC50 . . Mino ≥120nM TPD-0P3G9G IC50 . . Mino ≥120nM TPD-X0EIM0 IC50 . . Mino ≥120nM TPD-W9L5ZI IC50 . . Mino ≥120nM TPD-7RLEZE IC50 . . MV-4-11 1μM≤x<20μM TPD-NSRPL2 IC50 . . MV-4-11 <1nM TPD-1B33Z9 IC50 . . MV-4-11 <1nM TPD-Z3CYZE IC50 . . MV-4-11 <1nM TPD-DNY38I IC50 . . MV-4-11 >100nM TPD-NO47Z4 IC50 . . MV-4-11 10nM≤x≤100nM TPD-DXVRKM IC50 . . MV-4-11 <1nM TPD-OI0Y4F IC50 . . MV-4-11 10nM≤x≤100nM TPD-3D38V9 IC50 . . MV-4-11 <1nM TPD-KEKXTC IC50 . . MV-4-11 1nM≤x<10nM TPD-298GID IC50 . . MV-4-11 10nM≤x≤100nM TPD-VE69PZ IC50 . . MV-4-11 10nM≤x≤100nM TPD-6MP9CP IC50 . . MV-4-11 1nM≤x<10nM TPD-V8437G IC50 . . MV-4-11 1nM≤x<10nM TPD-DDOBJR IC50 . . MV-4-11 1nM≤x<10nM TPD-D4HKW2 IC50 . . MV-4-11 1nM≤x<10nM TPD-3VRYGW IC50 . . MV-4-11 1nM≤x<10nM TPD-HO7WLG IC50 . . MV-4-11 <1nM TPD-JOO5E7 IC50 . . . 1μM≤x≤10μM TPD-BEV4RO IC50 . . . <1μM TPD-3BLCKD IC50 . . . <1μM TPD-J6ESX9 IC50 . . . 1μM≤x≤10μM TPD-T0PJF3 IC50 . . . 1μM≤x≤10μM TPD-F6GS1A IC50 . . . 1μM≤x≤10μM TPD-M6062I IC50 . . . 2.96μM TPD-AH1YFV IC50 . . . 1.83μM TPD-MX2F3G IC50 . . . 0.75μM TPD-39QOSO IC50 . . . 0.63μM TPD-FC1M70 IC50 . . . 0.71μM TPD-B6APB0 IC50 . . . 0.51μM TPD-II8UOT IC50 . . . 0.77μM TPD-X4U6QP IC50 . . . 0.41μM TPD-JXAHU5 IC50 . . . 0.77μM TPD-XCIBNA IC50 . . . 0.54μM TPD-DGWKLG IC50 . . . 1.17μM TPD-C9TM5Y IC50 . . . 0.88μM TPD-5JZSFX IC50 . . . 0.23μM TPD-TEG7D2 IC50 . . . 0.47μM TPD-VE6AAW IC50 . . . 0.48μM TPD-NJVL07 IC50 . . . 0.16μM TPD-TMSBGS IC50 . . . 0.66μM TPD-XMVBW7 IC50 . . . 0.55μM TPD-RTJLTV IC50 . . . 1.42μM TPD-7FXJQH IC50 . . . 1.16μM TPD-V213GT IC50 . . . 0.52μM TPD-KYL3VU IC50 . . . 0.46μM TPD-5BFKTT IC50 . . . 0.52μM TPD-L0WNI6 IC50 . . . 1.44μM TPD-OJCTY9 IC50 . . . 0.19μM TPD-JV1ITV IC50 . . . 0.24μM TPD-SJ10PE IC50 . . . 1.38μM TPD-1VH741 IC50 . . . 0.34μM TPD-Q72RME IC50 . . . 1.59μM TPD-JVG0AA IC50 . . . 1.40μM TPD-G7JECQ IC50 . . . 0.23μM TPD-UCVYED IC50 . . . 0.17μM TPD-7I684R IC50 . . . 2.12μM TPD-H750GN IC50 . . . 0.85μM TPD-05WBFT IC50 . . . 0.56μM TPD-V6JUCY IC50 . . . 0.2μM TPD-M6062I Dmax IKZF1 Q13422 . <50% TPD-AH1YFV Dmax IKZF1 Q13422 . <50% TPD-MX2F3G Dmax IKZF1 Q13422 . <50% TPD-39QOSO Dmax IKZF1 Q13422 . <50% TPD-FC1M70 Dmax IKZF1 Q13422 . >50% TPD-B6APB0 Dmax IKZF1 Q13422 . >50% TPD-II8UOT Dmax IKZF1 Q13422 . <50% TPD-X4U6QP Dmax IKZF1 Q13422 . <50% TPD-JXAHU5 Dmax IKZF1 Q13422 . <50% TPD-XCIBNA Dmax IKZF1 Q13422 . <50% TPD-DGWKLG Dmax IKZF1 Q13422 . <50% TPD-C9TM5Y Dmax IKZF1 Q13422 . >50% TPD-5JZSFX Dmax IKZF1 Q13422 . >50% TPD-TEG7D2 Dmax IKZF1 Q13422 . <50% TPD-VE6AAW Dmax IKZF1 Q13422 . >50% TPD-NJVL07 Dmax IKZF1 Q13422 . <50% TPD-TMSBGS Dmax IKZF1 Q13422 . >50% TPD-XMVBW7 Dmax IKZF1 Q13422 . >50% TPD-RTJLTV Dmax IKZF1 Q13422 . <50% TPD-7FXJQH Dmax IKZF1 Q13422 . >50% TPD-V213GT Dmax IKZF1 Q13422 . >50% TPD-KYL3VU Dmax IKZF1 Q13422 . <50% TPD-ZK2RSY EC50 RBM39 Q14498 . 75.7nM TPD-3R45K0 EC50 RBM39 Q14498 . 108.1nM TPD-Y0MI5R EC50 RBM39 Q14498 . 384.0nM TPD-8EUUT9 EC50 RBM39 Q14498 . 297.6nM TPD-FDYHE9 EC50 RBM39 Q14498 . 363.8nM TPD-QQYD23 EC50 RBM39 Q14498 . >30000nM TPD-N2VHE2 EC50 RBM39 Q14498 . 8785.4nM TPD-EI3T6T EC50 RBM39 Q14498 . 127.7nM TPD-5K9S3Y EC50 RBM39 Q14498 . 299.1nM TPD-GCJOD2 EC50 RBM39 Q14498 . 325.3nM TPD-S40VS2 EC50 RBM39 Q14498 . 1972.3nM TPD-1SMV92 EC50 RBM39 Q14498 . 2069.1nM TPD-P3IFJK EC50 RBM39 Q14498 . 729.2nM TPD-ROIAJP EC50 RBM39 Q14498 . 1633.8nM TPD-L9UPDP EC50 RBM39 Q14498 . 1364.0nM TPD-FP1WLP EC50 RBM39 Q14498 . 1619.6nM TPD-0J44GE EC50 RBM39 Q14498 . 3262.1nM TPD-S4CJQL EC50 RBM39 Q14498 . 2133.8nM TPD-NE8N5A EC50 RBM39 Q14498 . 99.6nM TPD-45JO6P EC50 RBM39 Q14498 . 168.3nM TPD-G01BXV EC50 RBM39 Q14498 . 359.2nM TPD-PH7NRA EC50 RBM39 Q14498 . 916.8nM TPD-V8HAR4 EC50 RBM39 Q14498 . >30000nM TPD-414FJ2 EC50 RBM39 Q14498 . 959.6nM TPD-2VD2OU EC50 RBM39 Q14498 . 959.3nM TPD-WC3RYT EC50 RBM39 Q14498 . 649.9nM TPD-WT9X90 EC50 RBM39 Q14498 . 1816.7nM TPD-BN7BNQ EC50 RBM39 Q14498 . 1132.5nM TPD-C86CVL EC50 RBM39 Q14498 . 3795.9nM TPD-EX1CPB EC50 RBM39 Q14498 . 6651.5nM TPD-1P1PVH EC50 RBM39 Q14498 . 2668.0nM TPD-YIKVMB EC50 RBM39 Q14498 . 1762.5nM TPD-2B0KBD EC50 RBM39 Q14498 . 47.0nM TPD-AP9JRY EC50 RBM39 Q14498 . 510.7nM TPD-YZNYG4 EC50 RBM39 Q14498 . 422.8nM TPD-9I3NXM EC50 RBM39 Q14498 . 6067.5nM TPD-80OJ87 EC50 RBM39 Q14498 . 6617.6nM TPD-XUWIWW EC50 RBM39 Q14498 . 918.7nM TPD-CBR6W9 EC50 RBM39 Q14498 . 1956.8nM TPD-MGCOMT EC50 RBM39 Q14498 . 2150.0nM TPD-KV8XR7 EC50 RBM39 Q14498 . 1564.4nM TPD-A15HXP EC50 RBM39 Q14498 . 505.2nM TPD-BYII1J IC50 . . NCI-H82 100nM-300nM TPD-OQG9UV IC50 . . NCI-H82 100nM-300nM TPD-L4MWOF IC50 . . NCI-H82 <=100nM TPD-KH3KK9 IC50 . . NCI-H82 >300nM TPD-BYII1J IC50 . . HT-29 <=100nM TPD-OQG9UV IC50 . . HT-29 <=100nM TPD-6B7IKY IC50 . . HT-29 <=100nM TPD-TEONLH IC50 . . HT-29 <=100nM TPD-L4MWOF IC50 . . HT-29 <=100nM TPD-HQPUMB IC50 . . HT-29 <=100nM TPD-KH3KK9 IC50 . . HT-29 >300nM TPD-6B7IKY IC50 . . MDAMB231 <=100nM TPD-TEONLH IC50 . . MDAMB231 <=100nM TPD-HQPUMB IC50 . . MDAMB231 <=100nM TPD-Y158Z5 IC50 . . Mino 0nM75% TPD-LKQWTD Dmax NEK7 Q8TDX7 HEK293 >75% TPD-X0MNSY Dmax NEK7 Q8TDX7 HEK293 25%≤x<50% TPD-HDWLJP Dmax NEK7 Q8TDX7 HEK293 50%≤x≤75% TPD-BAPCCU Dmax NEK7 Q8TDX7 HEK293 <25% TPD-DGC2B7 Dmax NEK7 Q8TDX7 HEK293 50%≤x≤75% TPD-Z1ZHTE Dmax NEK7 Q8TDX7 HEK293 >75% TPD-N76G5L DC50 GSPT1 P15170 NCI-H1155 100nM≤x TPD-0JF90O DC50 GSPT1 P15170 NCI-H1155 <1nM TPD-VF5C6F DC50 GSPT1 P15170 NCI-H1155 <1nM TPD-KMD5EP DC50 GSPT1 P15170 NCI-H1155 1nM≤x<5nM TPD-ECHE5W DC50 GSPT1 P15170 NCI-H1155 <1nM TPD-R8HX47 DC50 GSPT1 P15170 NCI-H1155 <1nM TPD-YCQSKD DC50 GSPT1 P15170 NCI-H1155 1nM≤x<5nM TPD-ZA9MQ2 DC50 GSPT1 P15170 NCI-H1155 <1nM TPD-EMU4A5 DC50 GSPT1 P15170 NCI-H1155 1nM≤x<5nM TPD-JVVO7W DC50 GSPT1 P15170 NCI-H1155 1nM≤x<5nM TPD-N76G5L IC50 . . NCI-H1155 1μM≤x TPD-0JF90O IC50 . . NCI-H1155 <100nM TPD-VF5C6F IC50 . . NCI-H1155 <100nM TPD-KMD5EP IC50 . . NCI-H1155 <100nM TPD-ECHE5W IC50 . . NCI-H1155 <100nM TPD-R8HX47 IC50 . . NCI-H1155 <100nM TPD-YCQSKD IC50 . . NCI-H1155 <100nM TPD-ZA9MQ2 IC50 . . NCI-H1155 <100nM TPD-EMU4A5 IC50 . . NCI-H1155 <100nM TPD-JVVO7W IC50 . . NCI-H1155 <100nM TPD-GTLQQ4 IC50 . . NCI-H1155 <100nM TPD-GTLQQ4 IC50 . . NCI-H526 <100nM TPD-GFX0D5 IC50 . . NCI-H1155 1.4nM TPD-XUW2XL IC50 . . NCI-H1155 5nM TPD-ZSGS23 IC50 . . NCI-H1155 21nM TPD-GFX0D5 IC50 . . . 83nM TPD-ZSGS23 IC50 . . . 167nM TPD-GUXSDJ IC50 . . HGC27 139 nM TPD-EUD09L IC50 . . HGC27 225 nM TPD-0LNPDG IC50 . . HGC27 62 nM TPD-YTQJQ2 IC50 . . HGC27 25 nM TPD-BSCJ7R IC50 . . HGC27 41 nM TPD-ICZMU1 IC50 . . HGC27 75 nM TPD-Z0GIO8 IC50 . . HGC27 520 nM TPD-5KWJQR IC50 . . HGC27 68 nM TPD-XILW5Q IC50 . . HGC27 8 nM TPD-MZ15CR IC50 . . HGC27 39 nM TPD-YAO9KF IC50 . . HGC27 29 nM TPD-IY59BI IC50 . . HGC27 32 nM TPD-F9IXT3 IC50 . . HGC27 26 nM TPD-KWKLMR IC50 . . HGC27 25 nM TPD-GUXSDJ IC50 . . NCI-N87 26nM TPD-YTQJQ2 IC50 . . NCI-N87 7.5nM TPD-BSCJ7R IC50 . . NCI-N87 13nM TPD-5KWJQR IC50 . . NCI-N87 3.1nM TPD-XILW5Q IC50 . . NCI-N87 <1nM TPD-MZ15CR IC50 . . NCI-N87 32nM TPD-YAO9KF IC50 . . NCI-N87 48nM TPD-IY59BI IC50 . . NCI-N87 32nM TPD-F9IXT3 IC50 . . NCI-N87 19nM TPD-KWKLMR IC50 . . NCI-N87 30nM TPD-O75JPC IC50 . . NCI-N87 112nM TPD-1BGP4U EC50 RBM39 Q14498 . 19.9nM TPD-C4QK4C EC50 RBM39 Q14498 . 87.3nM TPD-HTZ73F EC50 RBM39 Q14498 . 20212.1nM TPD-49EA9O EC50 RBM39 Q14498 . 563.8nM TPD-KIYLEA EC50 RBM39 Q14498 . 1893.2nM TPD-TNRPK3 EC50 RBM39 Q14498 . 1101.7nM TPD-VKAVOR EC50 RBM39 Q14498 . 3769.8nM TPD-QA3K6B EC50 RBM39 Q14498 . 7700.5nM TPD-ILEIGY IC50 . . . 0.5μM50% TPD-87SIZ6 Dmax IKZF1 Q13422 . >50% TPD-OVAARG Dmax IKZF1 Q13422 . >50% TPD-HAKPLW Dmax IKZF1 Q13422 . ≤50% TPD-WEBL01 Dmax IKZF1 Q13422 . ≤50% TPD-JPRRVS Dmax IKZF1 Q13422 . >50% TPD-XQTWE5 Dmax IKZF1 Q13422 . >50% TPD-UU6XAW Dmax IKZF1 Q13422 . >50% TPD-YBTUHA Dmax IKZF1 Q13422 . ≤50% TPD-CNANTB Dmax IKZF1 Q13422 . ≤50% TPD-SQ31JD Dmax IKZF1 Q13422 . >50% TPD-LA942V Dmax IKZF1 Q13422 . >50% TPD-LRWBTF Dmax IKZF1 Q13422 . >50% TPD-NW7C79 Dmax IKZF1 Q13422 . ≤50% TPD-94FW54 Dmax IKZF1 Q13422 . ≤50% TPD-1YFXYK Dmax IKZF1 Q13422 . ≤50% TPD-ARNFP2 Dmax IKZF1 Q13422 . ≤50% TPD-3AZYVR Dmax IKZF1 Q13422 . ≤50% TPD-JCA82J Dmax IKZF1 Q13422 . >50% TPD-4DJ0JZ Dmax IKZF1 Q13422 . >50% TPD-I6OD38 Dmax IKZF1 Q13422 . >50% TPD-623REM Dmax IKZF1 Q13422 . ≤50% TPD-EEJG83 Dmax IKZF1 Q13422 . ≤50% TPD-45CY5X Dmax IKZF1 Q13422 . ≤50% TPD-5JWGG7 Dmax IKZF1 Q13422 . ≤50% TPD-V06NAB Dmax IKZF1 Q13422 . ≤50% TPD-6ZU6ZR Dmax IKZF1 Q13422 . ≤50% TPD-9LO9SP Dmax IKZF1 Q13422 . >50% TPD-BTL90G Dmax IKZF1 Q13422 . ≤50% TPD-1I7RFO Dmax IKZF1 Q13422 . ≤50% TPD-AC8VSR Dmax IKZF1 Q13422 . ≤50% TPD-XGCGZN Dmax IKZF1 Q13422 . >50% TPD-94FW54 Dmax IKZF3 Q9UKT9 . >50% TPD-1I7RFO Dmax IKZF3 Q9UKT9 . >50% TPD-AC8VSR Dmax IKZF3 Q9UKT9 . ≤50% TPD-QYHNBK IC50 . . . 0μM500nM TPD-IW1EFW IC50 BRAF P15056 . 50nM≤x<500nM TPD-0KDPAB IC50 BRAF P15056 . 50nM≤x<500nM TPD-NKFCG2 IC50 BRAF P15056 . 5nM≤x<50nM TPD-6F8EFE IC50 BRAF P15056 . 50nM≤x<500nM TPD-NOHIHG IC50 BRAF P15056 . 5nM≤x<50nM TPD-Z9W8OM IC50_1 . . MV-4-11 4743nM TPD-JPJTBM IC50_1 . . MV-4-11 227nM TPD-VCR8KN IC50_1 . . MV-4-11 >10000nM TPD-8QMI5F IC50_1 . . MV-4-11 1.3nM TPD-W0VFEV IC50_1 . . MV-4-11 6nM TPD-H1EDOQ IC50_1 . . MV-4-11 12nM TPD-VLCM8I IC50_1 . . MV-4-11 170nM TPD-M2LVXD IC50_1 . . MV-4-11 449nM TPD-K8V2FL IC50_1 . . MV-4-11 296nM TPD-SDXCQC IC50_1 . . MV-4-11 17nM TPD-KV8VOJ IC50_1 . . MV-4-11 >10000nM TPD-7XUR3Y IC50_1 . . MV-4-11 >10000nM TPD-ZGH71J IC50_1 . . MV-4-11 >10000nM TPD-9QHGOZ IC50_1 . . MV-4-11 71nM TPD-QYW5SN IC50_1 . . MV-4-11 >10000nM TPD-182MK7 IC50_1 . . MV-4-11 >10000nM TPD-PFDGKF IC50_1 . . MV-4-11 20nM TPD-Z5T8RY IC50_1 . . MV-4-11 8.7nM TPD-X27M5L IC50_1 . . MV-4-11 162nM TPD-JF2ZC3 IC50_1 . . MV-4-11 29nM TPD-D16PSV IC50_1 . . MV-4-11 3133nM TPD-VI9J0P IC50_1 . . MV-4-11 293nM TPD-55UCEU IC50_1 . . MV-4-11 <1nM TPD-0IICFL IC50_1 . . MV-4-11 9409nM TPD-PKZFIH IC50_1 . . MV-4-11 >10000nM TPD-WJXQEM IC50_1 . . MV-4-11 349nM TPD-61CT4M IC50_1 . . MV-4-11 B TPD-8MULYI IC50_1 . . MV-4-11 C TPD-RBEFTY IC50_1 . . MV-4-11 D TPD-BWQ25F IC50_1 . . MV-4-11 B TPD-IHDCLC IC50_1 . . MV-4-11 D TPD-YGCZ3V IC50_1 . . MV-4-11 D TPD-KL7OZU IC50_1 . . MV-4-11 B TPD-EUQDOZ IC50_1 . . MV-4-11 D TPD-2EIIVK IC50_1 . . MV-4-11 D TPD-TSU77L IC50_1 . . MV-4-11 D TPD-BN8UBI IC50_1 . . MV-4-11 D TPD-T5QYNN IC50_1 . . MV-4-11 D TPD-LGXSZ0 IC50_1 . . MV-4-11 B TPD-PC1DJP IC50_1 . . MV-4-11 D TPD-M65WMR IC50_1 . . MV-4-11 C TPD-1Z9YVZ IC50_1 . . MV-4-11 D TPD-FW6SQ3 IC50_1 . . MV-4-11 B TPD-BPGPPK IC50_1 . . MV-4-11 B TPD-6ZB45Z IC50_1 . . MV-4-11 D TPD-JIPGDU IC50_1 . . MV-4-11 B TPD-4I2NWY IC50_1 . . MV-4-11 B TPD-HRX4LQ IC50_1 . . MV-4-11 D TPD-PUQI7G IC50_1 . . MV-4-11 B TPD-SUYSV1 IC50_1 . . MV-4-11 B TPD-X8JJ19 IC50_1 . . MV-4-11 C TPD-6N79GG IC50_1 . . MV-4-11 C TPD-OYIUTC IC50_1 . . MV-4-11 D TPD-YR8YVA IC50_1 . . MV-4-11 C TPD-LQJCXE IC50_1 . . MV-4-11 C TPD-97Q67F IC50_1 . . MV-4-11 D TPD-E73UG1 IC50_1 . . MV-4-11 B TPD-1OV8QZ IC50_1 . . MV-4-11 D TPD-BCEBG6 IC50_1 . . MV-4-11 B TPD-SKC5VA IC50_1 . . MV-4-11 C TPD-XP13T0 IC50_1 . . MV-4-11 A TPD-WEEL4V IC50_1 . . MV-4-11 B TPD-UEBON4 IC50_1 . . MV-4-11 B TPD-MFTHZI IC50_1 . . MV-4-11 D TPD-D7UVST IC50_1 . . MV-4-11 C TPD-HAN9JK IC50_1 . . MV-4-11 D TPD-HN0UTL IC50_1 . . MV-4-11 B TPD-5COJ8O IC50_1 . . MV-4-11 A TPD-39VDPE IC50_1 . . MV-4-11 D TPD-736TPG IC50_1 . . MV-4-11 D TPD-ICWOIE IC50_1 . . MV-4-11 D TPD-JA9C4O IC50_1 . . MV-4-11 B TPD-O27VFZ IC50_1 . . MV-4-11 B TPD-80XO4K IC50_1 . . MV-4-11 B TPD-59VO3R IC50_1 . . MV-4-11 B TPD-FQX8HG IC50_1 . . MV-4-11 B TPD-78S72J IC50_1 . . MV-4-11 D TPD-H66EBD IC50_1 . . MV-4-11 D TPD-WPRLB1 IC50_1 . . MV-4-11 C TPD-UNJOZQ IC50_1 . . MV-4-11 D TPD-7RY16W IC50_1 . . MV-4-11 C TPD-353XLM IC50_1 . . MV-4-11 B TPD-FI523I IC50_1 . . MV-4-11 A TPD-G4SKXM IC50_1 . . MV-4-11 B TPD-XOMMCV IC50_1 . . MV-4-11 C TPD-PVGUQX IC50_1 . . MV-4-11 D TPD-Z9W8OM IC50_2 . . MV-4-11(in combination with gilteritinib) >10000nM TPD-JPJTBM IC50_2 . . MV-4-11(in combination with gilteritinib) 3nM TPD-VCR8KN IC50_2 . . MV-4-11(in combination with gilteritinib) 191nM TPD-8QMI5F IC50_2 . . MV-4-11(in combination with gilteritinib) 0.5nM TPD-W0VFEV IC50_2 . . MV-4-11(in combination with gilteritinib) 1.8nM TPD-H1EDOQ IC50_2 . . MV-4-11(in combination with gilteritinib) 4.6nM TPD-VLCM8I IC50_2 . . MV-4-11(in combination with gilteritinib) 9.9nM TPD-M2LVXD IC50_2 . . MV-4-11(in combination with gilteritinib) 27nM TPD-K8V2FL IC50_2 . . MV-4-11(in combination with gilteritinib) 22nM TPD-SDXCQC IC50_2 . . MV-4-11(in combination with gilteritinib) 2.3nM TPD-KV8VOJ IC50_2 . . MV-4-11(in combination with gilteritinib) >10000nM TPD-7XUR3Y IC50_2 . . MV-4-11(in combination with gilteritinib) >10000nM TPD-ZGH71J IC50_2 . . MV-4-11(in combination with gilteritinib) >10000nM TPD-9QHGOZ IC50_2 . . MV-4-11(in combination with gilteritinib) 8.3nM TPD-QYW5SN IC50_2 . . MV-4-11(in combination with gilteritinib) 2783nM TPD-182MK7 IC50_2 . . MV-4-11(in combination with gilteritinib) >10000nM TPD-PFDGKF IC50_2 . . MV-4-11(in combination with gilteritinib) 2nM TPD-Z5T8RY IC50_2 . . MV-4-11(in combination with gilteritinib) 0.9nM TPD-X27M5L IC50_2 . . MV-4-11(in combination with gilteritinib) 9.4nM TPD-JF2ZC3 IC50_2 . . MV-4-11(in combination with gilteritinib) 3nM TPD-D16PSV IC50_2 . . MV-4-11(in combination with gilteritinib) 44nM TPD-VI9J0P IC50_2 . . MV-4-11(in combination with gilteritinib) 60nM TPD-0IICFL IC50_2 . . MV-4-11(in combination with gilteritinib) 1917nM TPD-PKZFIH IC50_2 . . MV-4-11(in combination with gilteritinib) 8547nM TPD-WJXQEM IC50_2 . . MV-4-11(in combination with gilteritinib) 27nM TPD-61CT4M IC50_2 . . MV-4-11(in combination with gilteritinib) A TPD-8MULYI IC50_2 . . MV-4-11(in combination with gilteritinib) D TPD-RBEFTY IC50_2 . . MV-4-11(in combination with gilteritinib) D TPD-BWQ25F IC50_2 . . MV-4-11(in combination with gilteritinib) A TPD-IHDCLC IC50_2 . . MV-4-11(in combination with gilteritinib) D TPD-YGCZ3V IC50_2 . . MV-4-11(in combination with gilteritinib) D TPD-KL7OZU IC50_2 . . MV-4-11(in combination with gilteritinib) B TPD-EUQDOZ IC50_2 . . MV-4-11(in combination with gilteritinib) D TPD-2EIIVK IC50_2 . . MV-4-11(in combination with gilteritinib) D TPD-TSU77L IC50_2 . . MV-4-11(in combination with gilteritinib) D TPD-BN8UBI IC50_2 . . MV-4-11(in combination with gilteritinib) D TPD-T5QYNN IC50_2 . . MV-4-11(in combination with gilteritinib) D TPD-LGXSZ0 IC50_2 . . MV-4-11(in combination with gilteritinib) A TPD-PC1DJP IC50_2 . . MV-4-11(in combination with gilteritinib) D TPD-M65WMR IC50_2 . . MV-4-11(in combination with gilteritinib) A TPD-1Z9YVZ IC50_2 . . MV-4-11(in combination with gilteritinib) D TPD-FW6SQ3 IC50_2 . . MV-4-11(in combination with gilteritinib) A TPD-BPGPPK IC50_2 . . MV-4-11(in combination with gilteritinib) A TPD-6ZB45Z IC50_2 . . MV-4-11(in combination with gilteritinib) A TPD-JIPGDU IC50_2 . . MV-4-11(in combination with gilteritinib) B TPD-4I2NWY IC50_2 . . MV-4-11(in combination with gilteritinib) A TPD-HRX4LQ IC50_2 . . MV-4-11(in combination with gilteritinib) D TPD-PUQI7G IC50_2 . . MV-4-11(in combination with gilteritinib) A TPD-SUYSV1 IC50_2 . . MV-4-11(in combination with gilteritinib) B TPD-X8JJ19 IC50_2 . . MV-4-11(in combination with gilteritinib) A TPD-6N79GG IC50_2 . . MV-4-11(in combination with gilteritinib) C TPD-OYIUTC IC50_2 . . MV-4-11(in combination with gilteritinib) B TPD-YR8YVA IC50_2 . . MV-4-11(in combination with gilteritinib) B TPD-LQJCXE IC50_2 . . MV-4-11(in combination with gilteritinib) B TPD-97Q67F IC50_2 . . MV-4-11(in combination with gilteritinib) D TPD-E73UG1 IC50_2 . . MV-4-11(in combination with gilteritinib) A TPD-1OV8QZ IC50_2 . . MV-4-11(in combination with gilteritinib) B TPD-BCEBG6 IC50_2 . . MV-4-11(in combination with gilteritinib) B TPD-SKC5VA IC50_2 . . MV-4-11(in combination with gilteritinib) C TPD-XP13T0 IC50_2 . . MV-4-11(in combination with gilteritinib) A TPD-WEEL4V IC50_2 . . MV-4-11(in combination with gilteritinib) B TPD-UEBON4 IC50_2 . . MV-4-11(in combination with gilteritinib) A TPD-MFTHZI IC50_2 . . MV-4-11(in combination with gilteritinib) D TPD-D7UVST IC50_2 . . MV-4-11(in combination with gilteritinib) A TPD-HAN9JK IC50_2 . . MV-4-11(in combination with gilteritinib) D TPD-HN0UTL IC50_2 . . MV-4-11(in combination with gilteritinib) A TPD-5COJ8O IC50_2 . . MV-4-11(in combination with gilteritinib) A TPD-39VDPE IC50_2 . . MV-4-11(in combination with gilteritinib) C TPD-736TPG IC50_2 . . MV-4-11(in combination with gilteritinib) C TPD-ICWOIE IC50_2 . . MV-4-11(in combination with gilteritinib) D TPD-JA9C4O IC50_2 . . MV-4-11(in combination with gilteritinib) A TPD-O27VFZ IC50_2 . . MV-4-11(in combination with gilteritinib) B TPD-80XO4K IC50_2 . . MV-4-11(in combination with gilteritinib) A TPD-59VO3R IC50_2 . . MV-4-11(in combination with gilteritinib) A TPD-FQX8HG IC50_2 . . MV-4-11(in combination with gilteritinib) A TPD-78S72J IC50_2 . . MV-4-11(in combination with gilteritinib) B TPD-H66EBD IC50_2 . . MV-4-11(in combination with gilteritinib) C TPD-WPRLB1 IC50_2 . . MV-4-11(in combination with gilteritinib) B TPD-UNJOZQ IC50_2 . . MV-4-11(in combination with gilteritinib) D TPD-7RY16W IC50_2 . . MV-4-11(in combination with gilteritinib) B TPD-353XLM IC50_2 . . MV-4-11(in combination with gilteritinib) A TPD-FI523I IC50_2 . . MV-4-11(in combination with gilteritinib) A TPD-G4SKXM IC50_2 . . MV-4-11(in combination with gilteritinib) A TPD-XOMMCV IC50_2 . . MV-4-11(in combination with gilteritinib) B TPD-PVGUQX IC50_2 . . MV-4-11(in combination with gilteritinib) C TPD-55UCEU IC50_3 . . MOLM-13 3.7nM TPD-AWMPZP IC50_1 . . HeLa 2nM TPD-3TRGF4 IC50_1 . . HeLa 15nM TPD-2L65YG IC50_1 . . HeLa 19nM TPD-ACNFLC IC50_1 . . HeLa 27nM TPD-YOSWL3 IC50_1 . . HeLa 5nM TPD-4SPA5D IC50_1 . . HeLa 2nM TPD-VRS0AQ IC50_1 . . HeLa 23nM TPD-4GUVPG IC50_1 . . HeLa 3nM TPD-2DJGT1 IC50_1 . . HeLa 8nM TPD-1GVCLR IC50_1 . . HeLa 9nM TPD-PG55U9 IC50_1 . . HeLa 6nM TPD-EI0ZIL IC50_1 . . HeLa 6nM TPD-VZMKYT IC50_1 . . HeLa 4nM TPD-2RY6JP IC50_1 . . HeLa 8nM TPD-62XQL7 IC50_1 . . HeLa 2nM TPD-J24DD2 IC50_1 . . HeLa 6nM TPD-4BQLBM IC50_1 . . HeLa 2nM TPD-QR1QIH IC50_1 . . HeLa 4nM TPD-MKGNH2 IC50_1 . . HeLa 4nM TPD-NH432C IC50_1 . . HeLa 16nM TPD-ZKZY32 IC50_1 . . HeLa 5nM TPD-3FX0LB IC50_1 . . HeLa 3nM TPD-KEJNPE IC50_1 . . HeLa 5nM TPD-9KTNPT IC50_1 . . HeLa 0.3nM TPD-EEG1SI IC50_1 . . HeLa 5nM TPD-P4BT36 IC50_1 . . HeLa 1nM TPD-UL82OC IC50_1 . . HeLa 2nM TPD-NPS9IT IC50_1 . . HeLa 16nM TPD-RNA6C5 IC50_1 . . HeLa 32nM TPD-Q3V1P9 IC50_1 . . HeLa 12nM TPD-6WVD8O IC50_1 . . HeLa 0.3nM TPD-ZZS6EK IC50_1 . . HeLa 1nM TPD-C92GQP IC50_1 . . HeLa 7nM TPD-VHOCH9 IC50_1 . . HeLa 14nM TPD-BL9D46 IC50_1 . . HeLa 20nM TPD-FKXGQ8 IC50_1 . . HeLa 37nM TPD-44ZMYA IC50_1 . . HeLa >100nM TPD-OLT12Y IC50_1 . . HeLa >100nM TPD-CUF8MA IC50_1 . . HeLa >100nM TPD-HAT6B5 IC50_1 . . HeLa >100nM TPD-AWMPZP IC50_2 . . SK-MEL-3 3nM TPD-3TRGF4 IC50_2 . . SK-MEL-3 43nM TPD-2L65YG IC50_2 . . SK-MEL-3 49nM TPD-ACNFLC IC50_2 . . SK-MEL-3 82nM TPD-YOSWL3 IC50_2 . . SK-MEL-3 9nM TPD-4SPA5D IC50_2 . . SK-MEL-3 4nM TPD-VRS0AQ IC50_2 . . SK-MEL-3 40nM TPD-4GUVPG IC50_2 . . SK-MEL-3 6nM TPD-2DJGT1 IC50_2 . . SK-MEL-3 15nM TPD-1GVCLR IC50_2 . . SK-MEL-3 16nM TPD-PG55U9 IC50_2 . . SK-MEL-3 12nM TPD-EI0ZIL IC50_2 . . SK-MEL-3 13nM TPD-VZMKYT IC50_2 . . SK-MEL-3 9nM TPD-2RY6JP IC50_2 . . SK-MEL-3 14nM TPD-62XQL7 IC50_2 . . SK-MEL-3 4nM TPD-J24DD2 IC50_2 . . SK-MEL-3 10nM TPD-4BQLBM IC50_2 . . SK-MEL-3 6nM TPD-QR1QIH IC50_2 . . SK-MEL-3 7nM TPD-MKGNH2 IC50_2 . . SK-MEL-3 7nM TPD-NH432C IC50_2 . . SK-MEL-3 35nM TPD-ZKZY32 IC50_2 . . SK-MEL-3 9nM TPD-3FX0LB IC50_2 . . SK-MEL-3 6nM TPD-KEJNPE IC50_2 . . SK-MEL-3 7nM TPD-9KTNPT IC50_2 . . SK-MEL-3 1nM TPD-EEG1SI IC50_2 . . SK-MEL-3 10nM TPD-P4BT36 IC50_2 . . SK-MEL-3 1nM TPD-UL82OC IC50_2 . . SK-MEL-3 6nM TPD-NPS9IT IC50_2 . . SK-MEL-3 38nM TPD-RNA6C5 IC50_2 . . SK-MEL-3 51nM TPD-Q3V1P9 IC50_2 . . SK-MEL-3 26nM TPD-6WVD8O IC50_2 . . SK-MEL-3 1nM TPD-ZZS6EK IC50_2 . . SK-MEL-3 3nM TPD-C92GQP IC50_2 . . SK-MEL-3 19nM TPD-VHOCH9 IC50_2 . . SK-MEL-3 29nM TPD-BL9D46 IC50_2 . . SK-MEL-3 58nM TPD-FKXGQ8 IC50_2 . . SK-MEL-3 17nM TPD-44ZMYA IC50_2 . . SK-MEL-3 >100nM TPD-OLT12Y IC50_2 . . SK-MEL-3 >100nM TPD-CUF8MA IC50_2 . . SK-MEL-3 >100nM TPD-HAT6B5 IC50_2 . . SK-MEL-3 25600nM TPD-HEEEOA IC50_1 . . NCI-H1155 4.2nM TPD-FHVM3R IC50_1 . . NCI-H1155 22.7nM TPD-EK6TC6 IC50_1 . . NCI-H1155 2.3nM TPD-PKV84E IC50_1 . . NCI-H1155 4.7nM TPD-YGB3A0 IC50_1 . . NCI-H1155 0.22nM TPD-SVICVQ IC50_1 . . NCI-H1155 1.59nM TPD-FHVM3R IC50_2 . . Human PBMCs 57.51nM TPD-YGB3A0 IC50_2 . . Human PBMCs 1.52nM TPD-WYYCTP IC50_1 . . MM1.S A TPD-2B1H0S IC50_1 . . MM1.S A TPD-UH234B IC50_1 . . MM1.S A TPD-O1VKQP IC50_1 . . MM1.S A TPD-7XGCJQ IC50_1 . . MM1.S A TPD-HY1CA2 IC50_1 . . MM1.S A TPD-WYYCTP IC50_2 . . Mino C TPD-2B1H0S IC50_2 . . Mino A TPD-UH234B IC50_2 . . Mino B TPD-O1VKQP IC50_2 . . Mino B TPD-7XGCJQ IC50_2 . . Mino C TPD-HY1CA2 IC50_2 . . Mino A TPD-26643S EC50 Tau P10636 BE-M17 0.0609μM TPD-5U5W95 EC50 Tau P10636 BE-M17 0.06314μM TPD-4TBKO2 EC50 Tau P10636 BE-M17 0.2155μM TPD-QQ9F5M EC50 Tau P10636 BE-M17 0.00402μM TPD-9J6QKJ EC50 Tau P10636 BE-M17 0.00457μM TPD-ASRKE1 EC50 Tau P10636 BE-M17 0.00461μM TPD-N1TE43 EC50 Tau P10636 BE-M17 0.00463μM TPD-ZUFGJZ EC50 Tau P10636 BE-M17 0.00638μM TPD-VOV0V8 EC50 Tau P10636 BE-M17 0.01044μM TPD-PTMZ0R EC50 Tau P10636 BE-M17 0.1307μM TPD-ZGSBMA EC50 Tau P10636 BE-M17 0.04394μM TPD-ZZOS4I EC50 Tau P10636 BE-M17 0.07917μM TPD-JBTMQD EC50 Tau P10636 BE-M17 0.2501μM TPD-V3GVHZ EC50 Tau P10636 BE-M17 0.00453μM TPD-H2ZQUN EC50 Tau P10636 BE-M17 0.00932μM TPD-KOGISH EC50 Tau P10636 BE-M17 0.02431μM TPD-ZURRW8 EC50 Tau P10636 BE-M17 0.1525μM TPD-ESBFXW EC50 Tau P10636 BE-M17 0.03989μM TPD-K1DP3F EC50 Tau P10636 BE-M17 0.7114μM TPD-QY2BKA EC50 Tau P10636 BE-M17 0.04788μM TPD-BU8DRU EC50 Tau P10636 BE-M17 0.1658μM TPD-SL8IDN EC50 Tau P10636 BE-M17 0.2568μM TPD-OZTKVD EC50 Tau P10636 BE-M17 0.00479μM TPD-S4S476 EC50 Tau P10636 BE-M17 0.00597μM TPD-KF65VD EC50 Tau P10636 BE-M17 0.01002μM TPD-IDYU38 EC50 Tau P10636 BE-M17 0.02752μM TPD-Q4P84H EC50 Tau P10636 BE-M17 0.01255μM TPD-4SKXRP EC50 Tau P10636 BE-M17 0.00022μM TPD-D5GWLD EC50 Tau P10636 BE-M17 0.00022μM TPD-7CU2TR EC50 Tau P10636 BE-M17 0.00585μM TPD-258G99 EC50 Tau P10636 BE-M17 0.00086μM TPD-OKEZCP EC50 Tau P10636 BE-M17 0.0011μM TPD-90W6NW EC50 Tau P10636 BE-M17 0.00088μM TPD-U5N3TS EC50 Tau P10636 BE-M17 0.03464μM TPD-I06HJN EC50 Tau P10636 BE-M17 0.185μM TPD-983EJG EC50 Tau P10636 BE-M17 0.00076μM TPD-8J8SJ5 EC50 Tau P10636 BE-M17 0.00876μM TPD-U241SV EC50 Tau P10636 BE-M17 0.01391μM TPD-RO65T5 EC50 Tau P10636 BE-M17 0.01288μM TPD-1WCJST EC50 Tau P10636 BE-M17 0.01927μM TPD-8SYFC0 EC50 Tau P10636 BE-M17 0.07027μM TPD-OMJX5L EC50 Tau P10636 BE-M17 0.00074μM TPD-D6GGLM EC50 Tau P10636 BE-M17 0.00388μM TPD-0IMZ87 EC50 Tau P10636 BE-M17 0.0025μM TPD-6HP8ZV EC50 Tau P10636 BE-M17 0.00391μM TPD-D2BA6D EC50 Tau P10636 BE-M17 0.00368μM TPD-Z57V2C EC50 Tau P10636 BE-M17 0.00415μM TPD-4OV7A4 EC50 Tau P10636 BE-M17 0.03809μM TPD-KI1O76 EC50 Tau P10636 BE-M17 0.00957μM TPD-OI1G5I EC50 Tau P10636 BE-M17 0.02146μM TPD-FTGZVC EC50 Tau P10636 BE-M17 0.3111μM TPD-8KROCO EC50 Tau P10636 BE-M17 0.1287μM TPD-WMS9S9 EC50 Tau P10636 BE-M17 0.08388μM TPD-5AJZZF DC50 IKZF1 Q13422 Jurkat-IKZF1 HiBiT <10nM TPD-4SNPKN DC50 IKZF1 Q13422 Jurkat-IKZF1 HiBiT <10nM TPD-RXHUV7 DC50_1 CK1α P48729 MOLT-4-CK1alpha;-HiBiT +++ TPD-VUQCMQ DC50_1 CK1α P48729 MOLT-4-CK1alpha;-HiBiT ++ TPD-YHP8GU DC50_1 CK1α P48729 MOLT-4-CK1alpha;-HiBiT - TPD-A7EE0R DC50_1 CK1α P48729 MOLT-4-CK1alpha;-HiBiT - TPD-7NR9EC DC50_1 CK1α P48729 MOLT-4-CK1alpha;-HiBiT ++ TPD-V3BOVZ DC50_1 CK1α P48729 MOLT-4-CK1alpha;-HiBiT +++ TPD-RWAHFB DC50_1 CK1α P48729 MOLT-4-CK1alpha;-HiBiT +++ TPD-OQS5KS DC50_1 CK1α P48729 MOLT-4-CK1alpha;-HiBiT +++ TPD-TB7D6I DC50_1 CK1α P48729 MOLT-4-CK1alpha;-HiBiT +++ TPD-9L90O5 DC50_1 CK1α P48729 MOLT-4-CK1alpha;-HiBiT +++ TPD-PO1F7D DC50_1 CK1α P48729 MOLT-4-CK1alpha;-HiBiT +++ TPD-41BB04 DC50_1 CK1α P48729 MOLT-4-CK1alpha;-HiBiT +++ TPD-QK6FHZ DC50_1 CK1α P48729 MOLT-4-CK1alpha;-HiBiT +++ TPD-M6CR00 DC50_1 CK1α P48729 MOLT-4-CK1alpha;-HiBiT +++ TPD-CQZBY0 DC50_1 CK1α P48729 MOLT-4-CK1alpha;-HiBiT +++ TPD-WPFH4C DC50_1 CK1α P48729 MOLT-4-CK1alpha;-HiBiT +++ TPD-N3YPBR DC50_1 CK1α P48729 MOLT-4-CK1alpha;-HiBiT +++ TPD-2Z7CNI DC50_1 CK1α P48729 MOLT-4-CK1alpha;-HiBiT +++ TPD-KBHUF3 DC50_1 CK1α P48729 MOLT-4-CK1alpha;-HiBiT ++ TPD-TUX5I8 DC50_1 CK1α P48729 MOLT-4-CK1alpha;-HiBiT ++ TPD-P1375F DC50_1 CK1α P48729 MOLT-4-CK1alpha;-HiBiT - TPD-WZJIYM DC50_1 CK1α P48729 MOLT-4-CK1alpha;-HiBiT - TPD-3XSV65 DC50_1 CK1α P48729 MOLT-4-CK1alpha;-HiBiT - TPD-WD14LI DC50_1 CK1α P48729 MOLT-4-CK1alpha;-HiBiT - TPD-CB73YM DC50_1 CK1α P48729 MOLT-4-CK1alpha;-HiBiT - TPD-MM561R DC50_1 CK1α P48729 MOLT-4-CK1alpha;-HiBiT - TPD-KRHDMS DC50_1 CK1α P48729 MOLT-4-CK1alpha;-HiBiT - TPD-FN50XT DC50_1 CK1α P48729 MOLT-4-CK1alpha;-HiBiT - TPD-005QZQ DC50_1 CK1α P48729 MOLT-4-CK1alpha;-HiBiT - TPD-AE0M3J DC50_1 CK1α P48729 MOLT-4-CK1alpha;-HiBiT ++ TPD-JHBSGM DC50_1 CK1α P48729 MOLT-4-CK1alpha;-HiBiT ++ TPD-N4VUA6 DC50_1 CK1α P48729 MOLT-4-CK1alpha;-HiBiT +++ TPD-NIW5JA DC50_1 CK1α P48729 MOLT-4-CK1alpha;-HiBiT +++ TPD-RXHUV7 Dmax_1(5μM) CK1α P48729 MOLT-4-CK1alpha;-HiBiT 94 TPD-VUQCMQ Dmax_1(5μM) CK1α P48729 MOLT-4-CK1alpha;-HiBiT 77 TPD-7NR9EC Dmax_1(5μM) CK1α P48729 MOLT-4-CK1alpha;-HiBiT 67 TPD-V3BOVZ Dmax_1(5μM) CK1α P48729 MOLT-4-CK1alpha;-HiBiT 89 TPD-RWAHFB Dmax_1(5μM) CK1α P48729 MOLT-4-CK1alpha;-HiBiT 94 TPD-OQS5KS Dmax_1(5μM) CK1α P48729 MOLT-4-CK1alpha;-HiBiT 84 TPD-TB7D6I Dmax_1(5μM) CK1α P48729 MOLT-4-CK1alpha;-HiBiT 87 TPD-9L90O5 Dmax_1(5μM) CK1α P48729 MOLT-4-CK1alpha;-HiBiT 88 TPD-PO1F7D Dmax_1(5μM) CK1α P48729 MOLT-4-CK1alpha;-HiBiT 73 TPD-41BB04 Dmax_1(5μM) CK1α P48729 MOLT-4-CK1alpha;-HiBiT 82 TPD-QK6FHZ Dmax_1(5μM) CK1α P48729 MOLT-4-CK1alpha;-HiBiT 79 TPD-M6CR00 Dmax_1(5μM) CK1α P48729 MOLT-4-CK1alpha;-HiBiT 89 TPD-CQZBY0 Dmax_1(5μM) CK1α P48729 MOLT-4-CK1alpha;-HiBiT 95 TPD-WPFH4C Dmax_1(5μM) CK1α P48729 MOLT-4-CK1alpha;-HiBiT 88 TPD-N3YPBR Dmax_1(5μM) CK1α P48729 MOLT-4-CK1alpha;-HiBiT 78 TPD-2Z7CNI Dmax_1(5μM) CK1α P48729 MOLT-4-CK1alpha;-HiBiT 81 TPD-KBHUF3 Dmax_1(5μM) CK1α P48729 MOLT-4-CK1alpha;-HiBiT 81 TPD-TUX5I8 Dmax_1(5μM) CK1α P48729 MOLT-4-CK1alpha;-HiBiT 53 TPD-P1375F Dmax_1(5μM) CK1α P48729 MOLT-4-CK1alpha;-HiBiT 23 TPD-FN50XT Dmax_1(5μM) CK1α P48729 MOLT-4-CK1alpha;-HiBiT 43 TPD-YHP8GU DC50_2 WEE1 P30291 MOLT-4-WEE1-HiBiT - TPD-A7EE0R DC50_2 WEE1 P30291 MOLT-4-WEE1-HiBiT ++ TPD-WZJIYM DC50_2 WEE1 P30291 MOLT-4-WEE1-HiBiT - TPD-3XSV65 DC50_2 WEE1 P30291 MOLT-4-WEE1-HiBiT - TPD-WD14LI DC50_2 WEE1 P30291 MOLT-4-WEE1-HiBiT - TPD-CB73YM DC50_2 WEE1 P30291 MOLT-4-WEE1-HiBiT - TPD-MM561R DC50_2 WEE1 P30291 MOLT-4-WEE1-HiBiT - TPD-KRHDMS DC50_2 WEE1 P30291 MOLT-4-WEE1-HiBiT - TPD-005QZQ DC50_2 WEE1 P30291 MOLT-4-WEE1-HiBiT - TPD-AE0M3J DC50_2 WEE1 P30291 MOLT-4-WEE1-HiBiT +++ TPD-JHBSGM DC50_2 WEE1 P30291 MOLT-4-WEE1-HiBiT +++ TPD-N4VUA6 DC50_2 WEE1 P30291 MOLT-4-WEE1-HiBiT +++ TPD-NIW5JA DC50_2 WEE1 P30291 MOLT-4-WEE1-HiBiT +++ TPD-P1YJFI EC50 14-3-3σ/CRAF P31947/P04049 . 66±4μM TPD-YJYX33 EC50 14-3-3σ/CRAF P31947/P04049 . 17±3μM TPD-REZBFS EC50 14-3-3σ/CRAF P31947/P04049 . 3±1μM TPD-YKYBN7 EC50 14-3-3σ/CRAF P31947/P04049 . >1000μM TPD-PTD1PY EC50 14-3-3σ/CRAF P31947/P04049 . 82±6μM TPD-2HLG07 EC50 14-3-3σ/CRAF P31947/P04049 . 87±9μM TPD-IKRBP0 EC50 14-3-3σ/CRAF P31947/P04049 . >150μM TPD-YJYX33 Apparent Kd(100 μM compound) 14-3-3σ/CRAF P31947/P04049 . 400nM TPD-REZBFS Apparent Kd(100 μM compound) 14-3-3σ/CRAF P31947/P04049 . 190nM TPD-L1V5DV EC50_1 WEE1 P30291 LentiX-HEK293T 0.368μM TPD-SWPS43 EC50_1 WEE1 P30291 LentiX-HEK293T 0.339μM TPD-5SZSVH EC50_1 WEE1 P30291 LentiX-HEK293T 0.010μM TPD-8593VO EC50_1 WEE1 P30291 LentiX-HEK293T 0.014μM TPD-7LAMDQ EC50_1 WEE1 P30291 LentiX-HEK293T 0.001μM TPD-FSVU4U EC50_1 WEE1 P30291 LentiX-HEK293T 0.002μM TPD-1YB1T2 EC50_1 WEE1 P30291 LentiX-HEK293T 0.001μM TPD-UUZJGB EC50_1 WEE1 P30291 LentiX-HEK293T 0.004μM TPD-02T8GS EC50_1 WEE1 P30291 LentiX-HEK293T 0.006μM TPD-FMYXWD EC50_1 WEE1 P30291 LentiX-HEK293T 0.002μM TPD-RC4X8R EC50_1 WEE1 P30291 LentiX-HEK293T 0.004μM TPD-BJQZNS EC50_1 WEE1 P30291 LentiX-HEK293T 0.001μM TPD-YHCB4I EC50_1 WEE1 P30291 LentiX-HEK293T 0.003μM TPD-OYQZKN EC50_1 WEE1 P30291 LentiX-HEK293T 0.002μM TPD-K8TWVD EC50_1 WEE1 P30291 LentiX-HEK293T 0.000μM TPD-6JFMDE EC50_1 WEE1 P30291 LentiX-HEK293T 0.002μM TPD-FG36HB EC50_1 WEE1 P30291 LentiX-HEK293T 0.003μM TPD-U70EMW EC50_1 WEE1 P30291 LentiX-HEK293T 0.006μM TPD-FML7OH EC50_1 WEE1 P30291 LentiX-HEK293T 0.001μM TPD-CAOCPJ EC50_1 WEE1 P30291 LentiX-HEK293T 0.001μM TPD-LEGRI0 EC50_1 WEE1 P30291 LentiX-HEK293T 0.001μM TPD-SW3RAO EC50_1 WEE1 P30291 LentiX-HEK293T 0.002μM TPD-J1Q5S9 EC50_1 WEE1 P30291 LentiX-HEK293T 0.005μM TPD-5LJA64 EC50_1 WEE1 P30291 LentiX-HEK293T 0.002μM TPD-BMRH9K EC50_1 WEE1 P30291 LentiX-HEK293T 0.008μM TPD-GIDZ4D EC50_1 WEE1 P30291 LentiX-HEK293T 0.001μM TPD-NOYNEM EC50_1 WEE1 P30291 LentiX-HEK293T 0.001μM TPD-GEAUXG EC50_1 WEE1 P30291 LentiX-HEK293T 0.001μM TPD-99BG3B EC50_1 WEE1 P30291 LentiX-HEK293T 0.000μM TPD-F24N3W EC50_1 WEE1 P30291 LentiX-HEK293T 0.001μM TPD-755WVN EC50_1 WEE1 P30291 LentiX-HEK293T 0.001μM TPD-P8T0CR EC50_1 WEE1 P30291 LentiX-HEK293T 0.004μM TPD-1PR6RP EC50_1 WEE1 P30291 LentiX-HEK293T 0.001μM TPD-QOS1Y0 EC50_1 WEE1 P30291 LentiX-HEK293T 0.009μM TPD-8RN0AH EC50_1 WEE1 P30291 LentiX-HEK293T 0.000μM TPD-6ZGPA9 EC50_1 WEE1 P30291 LentiX-HEK293T 0.001μM TPD-E4OKCE EC50_1 WEE1 P30291 LentiX-HEK293T 0.000μM TPD-R9TON7 EC50_1 WEE1 P30291 LentiX-HEK293T 0.001μM TPD-F45OW5 EC50_1 WEE1 P30291 LentiX-HEK293T 0.003μM TPD-H7SEI9 EC50_1 WEE1 P30291 LentiX-HEK293T 0.003μM TPD-U935PN EC50_1 WEE1 P30291 LentiX-HEK293T 0.001μM TPD-52G0AS EC50_1 WEE1 P30291 LentiX-HEK293T 0.000μM TPD-2RDVSR EC50_1 WEE1 P30291 LentiX-HEK293T 0.001μM TPD-4NZ0F6 EC50_1 WEE1 P30291 LentiX-HEK293T 0.004μM TPD-K1D495 EC50_1 WEE1 P30291 LentiX-HEK293T 0.008μM TPD-F9CZS1 EC50_1 WEE1 P30291 LentiX-HEK293T 0.008μM TPD-O3MDOK EC50_1 WEE1 P30291 LentiX-HEK293T 0.000μM TPD-6TLI6A EC50_1 WEE1 P30291 LentiX-HEK293T 0.000μM TPD-B41YJ7 EC50_1 WEE1 P30291 LentiX-HEK293T 0.001μM TPD-711PT4 EC50_1 WEE1 P30291 LentiX-HEK293T 0.001μM TPD-K4N2W9 EC50_1 WEE1 P30291 LentiX-HEK293T 0.009μM TPD-XZL05Q EC50_1 WEE1 P30291 LentiX-HEK293T 0.000μM TPD-M02KOL EC50_1 WEE1 P30291 LentiX-HEK293T 0.006μM TPD-L1V5DV Ymin_1 WEE1 P30291 LentiX-HEK293T 30.70% TPD-SWPS43 Ymin_1 WEE1 P30291 LentiX-HEK293T 33.40% TPD-5SZSVH Ymin_1 WEE1 P30291 LentiX-HEK293T 28.10% TPD-8593VO Ymin_1 WEE1 P30291 LentiX-HEK293T 30.90% TPD-7LAMDQ Ymin_1 WEE1 P30291 LentiX-HEK293T 32.30% TPD-FSVU4U Ymin_1 WEE1 P30291 LentiX-HEK293T 27.40% TPD-1YB1T2 Ymin_1 WEE1 P30291 LentiX-HEK293T 31.90% TPD-UUZJGB Ymin_1 WEE1 P30291 LentiX-HEK293T 27.50% TPD-02T8GS Ymin_1 WEE1 P30291 LentiX-HEK293T 32.40% TPD-FMYXWD Ymin_1 WEE1 P30291 LentiX-HEK293T 27.80% TPD-RC4X8R Ymin_1 WEE1 P30291 LentiX-HEK293T 30.40% TPD-BJQZNS Ymin_1 WEE1 P30291 LentiX-HEK293T 22.10% TPD-YHCB4I Ymin_1 WEE1 P30291 LentiX-HEK293T 31.80% TPD-OYQZKN Ymin_1 WEE1 P30291 LentiX-HEK293T 28.40% TPD-K8TWVD Ymin_1 WEE1 P30291 LentiX-HEK293T 29.60% TPD-6JFMDE Ymin_1 WEE1 P30291 LentiX-HEK293T 25.60% TPD-FG36HB Ymin_1 WEE1 P30291 LentiX-HEK293T 29.80% TPD-U70EMW Ymin_1 WEE1 P30291 LentiX-HEK293T 31.40% TPD-FML7OH Ymin_1 WEE1 P30291 LentiX-HEK293T 30.30% TPD-CAOCPJ Ymin_1 WEE1 P30291 LentiX-HEK293T 29.80% TPD-LEGRI0 Ymin_1 WEE1 P30291 LentiX-HEK293T 31.30% TPD-SW3RAO Ymin_1 WEE1 P30291 LentiX-HEK293T 33.50% TPD-J1Q5S9 Ymin_1 WEE1 P30291 LentiX-HEK293T 37.70% TPD-5LJA64 Ymin_1 WEE1 P30291 LentiX-HEK293T 39.00% TPD-BMRH9K Ymin_1 WEE1 P30291 LentiX-HEK293T 32.80% TPD-GIDZ4D Ymin_1 WEE1 P30291 LentiX-HEK293T 29.10% TPD-NOYNEM Ymin_1 WEE1 P30291 LentiX-HEK293T 26.40% TPD-GEAUXG Ymin_1 WEE1 P30291 LentiX-HEK293T 27.90% TPD-99BG3B Ymin_1 WEE1 P30291 LentiX-HEK293T 20.10% TPD-F24N3W Ymin_1 WEE1 P30291 LentiX-HEK293T 33.40% TPD-755WVN Ymin_1 WEE1 P30291 LentiX-HEK293T 29.30% TPD-P8T0CR Ymin_1 WEE1 P30291 LentiX-HEK293T 21.80% TPD-1PR6RP Ymin_1 WEE1 P30291 LentiX-HEK293T 28.10% TPD-QOS1Y0 Ymin_1 WEE1 P30291 LentiX-HEK293T 30.20% TPD-8RN0AH Ymin_1 WEE1 P30291 LentiX-HEK293T 30.10% TPD-6ZGPA9 Ymin_1 WEE1 P30291 LentiX-HEK293T 28.00% TPD-E4OKCE Ymin_1 WEE1 P30291 LentiX-HEK293T 31.60% TPD-R9TON7 Ymin_1 WEE1 P30291 LentiX-HEK293T 24.60% TPD-F45OW5 Ymin_1 WEE1 P30291 LentiX-HEK293T 33.00% TPD-H7SEI9 Ymin_1 WEE1 P30291 LentiX-HEK293T 43.70% TPD-U935PN Ymin_1 WEE1 P30291 LentiX-HEK293T 32.30% TPD-52G0AS Ymin_1 WEE1 P30291 LentiX-HEK293T 21.30% TPD-2RDVSR Ymin_1 WEE1 P30291 LentiX-HEK293T 40.70% TPD-4NZ0F6 Ymin_1 WEE1 P30291 LentiX-HEK293T 29.80% TPD-K1D495 Ymin_1 WEE1 P30291 LentiX-HEK293T 19.50% TPD-F9CZS1 Ymin_1 WEE1 P30291 LentiX-HEK293T 61.20% TPD-O3MDOK Ymin_1 WEE1 P30291 LentiX-HEK293T 27.50% TPD-6TLI6A Ymin_1 WEE1 P30291 LentiX-HEK293T 27.30% TPD-B41YJ7 Ymin_1 WEE1 P30291 LentiX-HEK293T 27.10% TPD-711PT4 Ymin_1 WEE1 P30291 LentiX-HEK293T 28.00% TPD-K4N2W9 Ymin_1 WEE1 P30291 LentiX-HEK293T 29.50% TPD-XZL05Q Ymin_1 WEE1 P30291 LentiX-HEK293T 29.70% TPD-M02KOL Ymin_1 WEE1 P30291 LentiX-HEK293T 21.50% TPD-9KSJOO EC50_2 . . MKN45 0.337μM TPD-9R3NRH EC50_2 . . MKN45 0.205μM TPD-9KSJOO Ymin_2 . . MKN45 40.60% TPD-9R3NRH Ymin_2 . . MKN45 29.10% TPD-QKR72G DC50 GSPT1 P15170 NB-4 7.8nM TPD-MS0IDH DC50 GSPT1 P15170 NB-4 3.6nM TPD-58GBEZ DC50 GSPT1 P15170 NB-4 >1000nM TPD-S1EVER DC50 GSPT1 P15170 NB-4 15nM TPD-O6RNNR DC50 GSPT1 P15170 NB-4 13nM TPD-D0HYCL DC50 GSPT1 P15170 NB-4 5.9nM TPD-4VAV9G DC50 GSPT1 P15170 NB-4 5.2nM TPD-ZUQSU2 DC50 GSPT1 P15170 NB-4 7.2nM TPD-M9TVVV DC50 GSPT1 P15170 NB-4 6.5nM TPD-5C1L0B DC50 GSPT1 P15170 NB-4 1.5nM TPD-GCXVRB DC50 GSPT1 P15170 NB-4 1.5nM TPD-4MDSSG DC50 GSPT1 P15170 NB-4 4.5nM TPD-SV52YJ DC50 GSPT1 P15170 NB-4 >1000nM TPD-SIEU8E DC50 GSPT1 P15170 NB-4 1nM TPD-0MRK4C DC50 GSPT1 P15170 NB-4 >1000nM TPD-UG0KDY DC50 GSPT1 P15170 NB-4 4.2nM TPD-ENWE0U DC50 GSPT1 P15170 NB-4 8nM TPD-J8MTI9 DC50 GSPT1 P15170 NB-4 >1000nM TPD-3A3WWA DC50 GSPT1 P15170 NB-4 21nM TPD-3U0FSN DC50 GSPT1 P15170 NB-4 2nM TPD-35INJS DC50 GSPT1 P15170 NB-4 13nM TPD-TFG5IN DC50 GSPT1 P15170 NB-4 36nM TPD-CR3VWN DC50 GSPT1 P15170 NB-4 15nM TPD-II9YUS DC50 GSPT1 P15170 NB-4 14nM TPD-CV1XG2 DC50 GSPT1 P15170 NB-4 13nM TPD-DY9C8N DC50 GSPT1 P15170 NB-4 >1000nM TPD-8XMZ9P DC50 GSPT1 P15170 NB-4 4.8nM TPD-T5M671 DC50 GSPT1 P15170 NB-4 3.7nM TPD-AB3SXS DC50 GSPT1 P15170 NB-4 2.5nM TPD-DUL83T DC50 GSPT1 P15170 NB-4 4.3nM TPD-9TB2IT DC50 GSPT1 P15170 NB-4 30nM TPD-94BQWZ DC50 GSPT1 P15170 NB-4 1.4nM TPD-VRJY4X DC50 GSPT1 P15170 NB-4 2.6nM TPD-QKR72G Dmax GSPT1 P15170 NB-4 82% TPD-MS0IDH Dmax GSPT1 P15170 NB-4 110% TPD-S1EVER Dmax GSPT1 P15170 NB-4 42% TPD-O6RNNR Dmax GSPT1 P15170 NB-4 71% TPD-D0HYCL Dmax GSPT1 P15170 NB-4 92% TPD-4VAV9G Dmax GSPT1 P15170 NB-4 94% TPD-ZUQSU2 Dmax GSPT1 P15170 NB-4 93% TPD-M9TVVV Dmax GSPT1 P15170 NB-4 100% TPD-5C1L0B Dmax GSPT1 P15170 NB-4 113% TPD-GCXVRB Dmax GSPT1 P15170 NB-4 28% TPD-4MDSSG Dmax GSPT1 P15170 NB-4 112% TPD-SIEU8E Dmax GSPT1 P15170 NB-4 31% TPD-UG0KDY Dmax GSPT1 P15170 NB-4 106% TPD-ENWE0U Dmax GSPT1 P15170 NB-4 107% TPD-3A3WWA Dmax GSPT1 P15170 NB-4 70% TPD-3U0FSN Dmax GSPT1 P15170 NB-4 110% TPD-35INJS Dmax GSPT1 P15170 NB-4 23% TPD-TFG5IN Dmax GSPT1 P15170 NB-4 16% TPD-CR3VWN Dmax GSPT1 P15170 NB-4 49% TPD-II9YUS Dmax GSPT1 P15170 NB-4 74% TPD-CV1XG2 Dmax GSPT1 P15170 NB-4 56% TPD-8XMZ9P Dmax GSPT1 P15170 NB-4 96% TPD-T5M671 Dmax GSPT1 P15170 NB-4 95% TPD-AB3SXS Dmax GSPT1 P15170 NB-4 114% TPD-DUL83T Dmax GSPT1 P15170 NB-4 103% TPD-9TB2IT Dmax GSPT1 P15170 NB-4 36% TPD-94BQWZ Dmax GSPT1 P15170 NB-4 121% TPD-VRJY4X Dmax GSPT1 P15170 NB-4 108% TPD-X00UE3 Dmax GSPT1 P15170 AML(KG-1) C TPD-N99A3J Dmax GSPT1 P15170 AML(KG-1) C TPD-XKR3BT Dmax GSPT1 P15170 AML(KG-1) C TPD-QI2SAS Dmax GSPT1 P15170 AML(KG-1) B TPD-X00UE3 IC50_1 . . AML(KG-1) E TPD-N99A3J IC50_1 . . AML(KG-1) D TPD-XKR3BT IC50_1 . . AML(KG-1) D TPD-QI2SAS IC50_1 . . AML(KG-1) D TPD-KOHUUB DC50 WIZ O95785 HT-1080 113nM TPD-W0L6JJ DC50 WIZ O95785 HT-1080 57.4nM TPD-UR87SB DC50 WIZ O95785 HT-1080 47.8nM TPD-NCET78 DC50 WIZ O95785 HT-1080 33.8nM TPD-DQRYJW DC50 WIZ O95785 HT-1080 26.5nM TPD-2T5380 DC50 WIZ O95785 HT-1080 19.9nM TPD-XRHCMJ DC50 WIZ O95785 HT-1080 40.1nM TPD-8ET5ZK DC50 WIZ O95785 HT-1080 57.4nM TPD-PYANPG DC50 WIZ O95785 HT-1080 11nM TPD-7Q2U5K DC50 WIZ O95785 HT-1080 30.4nM TPD-EGN05G DC50 WIZ O95785 HT-1080 6.7nM TPD-NLN0M0 DC50 WIZ O95785 HT-1080 10nM TPD-K5B0RS DC50 WIZ O95785 HT-1080 17.9nM TPD-CRQLGE DC50 WIZ O95785 HT-1080 43.9nM TPD-KOHUUB Dmax WIZ O95785 HT-1080 84.00% TPD-W0L6JJ Dmax WIZ O95785 HT-1080 86.40% TPD-UR87SB Dmax WIZ O95785 HT-1080 86.20% TPD-NCET78 Dmax WIZ O95785 HT-1080 88.90% TPD-DQRYJW Dmax WIZ O95785 HT-1080 91.30% TPD-2T5380 Dmax WIZ O95785 HT-1080 92.00% TPD-XRHCMJ Dmax WIZ O95785 HT-1080 90.20% TPD-8ET5ZK Dmax WIZ O95785 HT-1080 92.00% TPD-PYANPG Dmax WIZ O95785 HT-1080 94.60% TPD-7Q2U5K Dmax WIZ O95785 HT-1080 90.50% TPD-EGN05G Dmax WIZ O95785 HT-1080 94.10% TPD-NLN0M0 Dmax WIZ O95785 HT-1080 94% TPD-K5B0RS Dmax WIZ O95785 HT-1080 92.10% TPD-CRQLGE Dmax WIZ O95785 HT-1080 86.40% TPD-QHYM7Q IC50_1 . . MDAMB231 E TPD-8YPO9C IC50_1 . . MDAMB231 G TPD-UA4LNK IC50_1 . . MDAMB231 F TPD-A3EJ8F IC50_1 . . MDAMB231 G TPD-UEBV5L IC50_1 . . MDAMB231 F TPD-Q0R2ZC IC50_1 . . MDAMB231 G TPD-VVPEWF IC50_1 . . MDAMB231 F TPD-1TS0NP IC50_1 . . MDAMB231 F TPD-XEEYBI IC50_1 . . MDAMB231 F TPD-3VPEXG IC50_1 . . MDAMB231 E TPD-Q7HW45 IC50_1 . . MDAMB231 F TPD-4EZYIA IC50_1 . . MDAMB231 D TPD-UGWULZ IC50_1 . . MDAMB231 F TPD-5BBMDT IC50_1 . . MDAMB231 D TPD-9FFMGU IC50_1 . . MDAMB231 D TPD-DKJ4PJ IC50_1 . . MDAMB231 F TPD-XCTCV9 IC50_1 . . MDAMB231 F TPD-ASU6WY IC50_1 . . MDAMB231 F TPD-LWEP3Q IC50_2 . . Molt-4 D TPD-QHYM7Q IC50_2 . . Molt-4 D TPD-8YPO9C IC50_2 . . Molt-4 C TPD-UA4LNK IC50_2 . . Molt-4 B TPD-261DWQ IC50_2 . . Molt-4 D TPD-A3EJ8F IC50_2 . . Molt-4 C TPD-6LD0I1 IC50_2 . . Molt-4 F TPD-UEBV5L IC50_2 . . Molt-4 B TPD-Z9FFEZ IC50_2 . . Molt-4 F TPD-Q0R2ZC IC50_2 . . Molt-4 D TPD-VVPEWF IC50_2 . . Molt-4 C TPD-1TS0NP IC50_2 . . Molt-4 D TPD-XEEYBI IC50_2 . . Molt-4 D TPD-3VPEXG IC50_2 . . Molt-4 B TPD-Q7HW45 IC50_2 . . Molt-4 D TPD-Q24CCD IC50_2 . . Molt-4 D TPD-4EZYIA IC50_2 . . Molt-4 B TPD-UGWULZ IC50_2 . . Molt-4 C TPD-VF0I1E IC50_2 . . Molt-4 D TPD-5BBMDT IC50_2 . . Molt-4 B TPD-9FFMGU IC50_2 . . Molt-4 B TPD-86DZC3 IC50_2 . . Molt-4 C TPD-ZC9RJX IC50_2 . . Molt-4 D TPD-Z7LMA1 IC50_2 . . Molt-4 D TPD-IYQZTE IC50_2 . . Molt-4 D TPD-YNYH3W IC50_2 . . Molt-4 B TPD-DKJ4PJ IC50_2 . . Molt-4 C TPD-XCTCV9 IC50_2 . . Molt-4 C TPD-BPCEXQ IC50_2 . . Molt-4 F TPD-ASU6WY IC50_2 . . Molt-4 C TPD-261DWQ IC50_3 . . NCI-H1975 G TPD-VF0I1E IC50_3 . . NCI-H1975 G TPD-86DZC3 IC50_3 . . NCI-H1975 F TPD-Z7LMA1 IC50_3 . . NCI-H1975 G TPD-YNYH3W IC50_3 . . NCI-H1975 D TPD-DGK6M9 IC50_4 . . CCRF-CEM B TPD-5XAALX IC50_4 . . CCRF-CEM B TPD-X0PWQP IC50_4 . . CCRF-CEM C TPD-RDB6ER IC50_4 . . CCRF-CEM C TPD-T6OSGN IC50_4 . . CCRF-CEM D TPD-LWEP3Q IC50_4 . . CCRF-CEM D TPD-6LD0I1 IC50_4 . . CCRF-CEM F TPD-Z9FFEZ IC50_4 . . CCRF-CEM F TPD-Q24CCD IC50_4 . . CCRF-CEM D TPD-ZC9RJX IC50_4 . . CCRF-CEM C TPD-IYQZTE IC50_4 . . CCRF-CEM D TPD-BPCEXQ IC50_4 . . CCRF-CEM E TPD-DGK6M9 IC50_5 . . CAL-62 B TPD-5XAALX IC50_5 . . CAL-62 B TPD-X0PWQP IC50_5 . . CAL-62 C TPD-RDB6ER IC50_5 . . CAL-62 D TPD-T6OSGN IC50_5 . . CAL-62 E TPD-7N1025 Dmax_1 WEE1 P30291 . B TPD-U5VGPT Dmax_1 WEE1 P30291 . A TPD-ESESWH Dmax_1 WEE1 P30291 . A TPD-T78R4K Dmax_1 WEE1 P30291 . B TPD-EA6KKR Dmax_1 WEE1 P30291 . B TPD-4UJ2TJ Dmax_1 WEE1 P30291 . B TPD-A50CS0 Dmax_1 WEE1 P30291 . A TPD-46B52Z Dmax_1 WEE1 P30291 . A TPD-9MXOVM Dmax_1 WEE1 P30291 . B TPD-PDZI92 Dmax_1 WEE1 P30291 . B TPD-C2IJ68 Dmax_1 WEE1 P30291 . B TPD-RJMYFB Dmax_1 WEE1 P30291 . A TPD-7T100N Dmax_1 WEE1 P30291 . B TPD-42MYCY Dmax_1 WEE1 P30291 . A TPD-VPX4H5 Dmax_1 WEE1 P30291 . A TPD-F0U53B Dmax_1 WEE1 P30291 . A TPD-TZSWWW Dmax_1 WEE1 P30291 . A TPD-FWG8HO Dmax_1 WEE1 P30291 . A TPD-N4PRD6 Dmax_1 WEE1 P30291 . A TPD-6UHQBC Dmax_1 WEE1 P30291 . B TPD-DHC957 Dmax_1 WEE1 P30291 . B TPD-7N1025 Dmax_2 IKZF1 Q13422 . A TPD-U5VGPT Dmax_2 IKZF1 Q13422 . B TPD-ESESWH Dmax_2 IKZF1 Q13422 . B TPD-T78R4K Dmax_2 IKZF1 Q13422 . B TPD-EA6KKR Dmax_2 IKZF1 Q13422 . B TPD-4UJ2TJ Dmax_2 IKZF1 Q13422 . B TPD-A50CS0 Dmax_2 IKZF1 Q13422 . A TPD-46B52Z Dmax_2 IKZF1 Q13422 . A TPD-9MXOVM Dmax_2 IKZF1 Q13422 . B TPD-PDZI92 Dmax_2 IKZF1 Q13422 . B TPD-C2IJ68 Dmax_2 IKZF1 Q13422 . B TPD-RJMYFB Dmax_2 IKZF1 Q13422 . A TPD-7T100N Dmax_2 IKZF1 Q13422 . B TPD-42MYCY Dmax_2 IKZF1 Q13422 . A TPD-VPX4H5 Dmax_2 IKZF1 Q13422 . A TPD-F0U53B Dmax_2 IKZF1 Q13422 . B TPD-TZSWWW Dmax_2 IKZF1 Q13422 . B TPD-FWG8HO Dmax_2 IKZF1 Q13422 . B TPD-N4PRD6 Dmax_2 IKZF1 Q13422 . A TPD-6UHQBC Dmax_2 IKZF1 Q13422 . B TPD-DHC957 Dmax_2 IKZF1 Q13422 . B TPD-JFVBR1 IC50_1 . . BT-474 0.94nM TPD-86YMG4 IC50_1 . . BT-474 1.64nM TPD-R9KGKL IC50_1 . . BT-474 6.54nM TPD-U99ZS4 IC50_1 . . BT-474 2.63nM TPD-DM1J6Z IC50_1 . . BT-474 1.75nM TPD-JFVBR1 IC50_2 . . NCI-N87 0.76nM TPD-86YMG4 IC50_2 . . NCI-N87 1.40nM TPD-R9KGKL IC50_2 . . NCI-N87 21.59nM TPD-U99ZS4 IC50_2 . . NCI-N87 1.32nM TPD-DM1J6Z IC50_2 . . NCI-N87 2.22nM TPD-6CNM9W IC50_1 . . MV-4-11 E TPD-IAVN2T IC50_1 . . MV-4-11 E TPD-UWAMM4 IC50_1 . . MV-4-11 A TPD-HBSZ2W IC50_1 . . MV-4-11 A TPD-EOP5ZD IC50_1 . . MV-4-11 E TPD-U7L64B IC50_1 . . MV-4-11 A TPD-SNLRYH IC50_1 . . MV-4-11 E TPD-77SLEG IC50_1 . . MV-4-11 B TPD-C8X901 IC50_1 . . MV-4-11 C TPD-E5QQTK IC50_1 . . MV-4-11 E TPD-YIMLNA IC50_1 . . MV-4-11 E TPD-2MPCJ2 IC50_1 . . MV-4-11 B TPD-5DY5HM IC50_1 . . MV-4-11 E TPD-HMU1A7 IC50_1 . . MV-4-11 A TPD-O1I4HX IC50_1 . . MV-4-11 E TPD-JVALT8 IC50_1 . . MV-4-11 C TPD-ZE14VS IC50_1 . . MV-4-11 C TPD-GMZLPB IC50_1 . . MV-4-11 E TPD-SCDWR6 IC50_1 . . MV-4-11 E TPD-BE1013 IC50_1 . . MV-4-11 B TPD-TSRFVY IC50_1 . . MV-4-11 B TPD-7P7BXA IC50_1 . . MV-4-11 C TPD-Z3RZS2 IC50_1 . . MV-4-11 C TPD-UWAMM4 IC50_2 . . NCI-H929 A TPD-6CNM9W Dmax GSPT1 P15170 NB-4 D TPD-IAVN2T Dmax GSPT1 P15170 NB-4 D TPD-HBSZ2W Dmax GSPT1 P15170 NB-4 A TPD-EOP5ZD Dmax GSPT1 P15170 NB-4 D TPD-U7L64B Dmax GSPT1 P15170 NB-4 A TPD-SNLRYH Dmax GSPT1 P15170 NB-4 D TPD-77SLEG Dmax GSPT1 P15170 NB-4 A TPD-C8X901 Dmax GSPT1 P15170 NB-4 A TPD-E5QQTK Dmax GSPT1 P15170 NB-4 D TPD-YIMLNA Dmax GSPT1 P15170 NB-4 D TPD-2MPCJ2 Dmax GSPT1 P15170 NB-4 A TPD-5DY5HM Dmax GSPT1 P15170 NB-4 D TPD-HMU1A7 Dmax GSPT1 P15170 NB-4 A TPD-O1I4HX Dmax GSPT1 P15170 NB-4 D TPD-JVALT8 Dmax GSPT1 P15170 NB-4 A TPD-ZE14VS Dmax GSPT1 P15170 NB-4 A TPD-GMZLPB Dmax GSPT1 P15170 NB-4 D TPD-SCDWR6 Dmax GSPT1 P15170 NB-4 D TPD-BE1013 Dmax GSPT1 P15170 NB-4 A TPD-TSRFVY Dmax GSPT1 P15170 NB-4 A TPD-7P7BXA Dmax GSPT1 P15170 NB-4 B TPD-Z3RZS2 Dmax GSPT1 P15170 NB-4 A TPD-GE80LT IC50_1 . . MM1.S A TPD-C7XQ6O IC50_1 . . MM1.S A TPD-EQHNIO IC50_1 . . MM1.S C TPD-2TCP1F IC50_1 . . MM1.S A TPD-8NUE7X IC50_1 . . MM1.S A+ TPD-FRY1MT IC50_1 . . MM1.S A+ TPD-T4EVHY IC50_1 . . MM1.S A TPD-FL20ZH IC50_1 . . MM1.S A++ TPD-RYPV9T IC50_1 . . MM1.S A+ TPD-VOSF8R IC50_1 . . MM1.S A TPD-2XE3QX IC50_1 . . MM1.S B TPD-3A74YZ IC50_1 . . MM1.S A TPD-1FQJ6L IC50_1 . . MM1.S A TPD-SPP94V IC50_1 . . MM1.S C TPD-S5HTQQ IC50_1 . . MM1.S A++ TPD-1D2ELF IC50_1 . . MM1.S A+ TPD-6WKRZC IC50_1 . . MM1.S A++ TPD-CPFXWG IC50_1 . . MM1.S C TPD-D9OJIS IC50_1 . . MM1.S B TPD-XRHTSQ IC50_1 . . MM1.S C TPD-EOL5BI IC50_1 . . MM1.S C TPD-8IIO95 IC50_1 . . MM1.S A TPD-OFAIH5 IC50_1 . . MM1.S C TPD-JMNCLG IC50_1 . . MM1.S A TPD-DOGJ1O IC50_1 . . MM1.S A++ TPD-GOGQQ6 IC50_1 . . MM1.S A TPD-4V0BZR IC50_1 . . MM1.S A TPD-GE80LT IC50_2 . . MGC803 C TPD-C7XQ6O IC50_2 . . MGC803 B TPD-2TCP1F IC50_2 . . MGC803 B TPD-8NUE7X IC50_2 . . MGC803 B TPD-FRY1MT IC50_2 . . MGC803 A TPD-T4EVHY IC50_2 . . MGC803 B TPD-FL20ZH IC50_2 . . MGC803 A TPD-RYPV9T IC50_2 . . MGC803 A TPD-3A74YZ IC50_2 . . MGC803 B TPD-1FQJ6L IC50_2 . . MGC803 C TPD-S5HTQQ IC50_2 . . MGC803 A TPD-1D2ELF IC50_2 . . MGC803 A TPD-6WKRZC IC50_2 . . MGC803 A TPD-VOSF8R IC50_3 . . Jurkat C TPD-N02C64 Dmax_1 WEE1 P30291 Human PBMCs A TPD-0T65BK Dmax_1 WEE1 P30291 Human PBMCs B TPD-9SDW2K Dmax_1 WEE1 P30291 Human PBMCs B TPD-EQHNIO Dmax_1 WEE1 P30291 Human PBMCs B TPD-2XE3QX Dmax_1 WEE1 P30291 Human PBMCs A TPD-CQJPPB Dmax_1 WEE1 P30291 Human PBMCs B TPD-SPP94V Dmax_1 WEE1 P30291 Human PBMCs A TPD-SG1LPO Dmax_1 WEE1 P30291 Human PBMCs B TPD-17ZY6D Dmax_1 WEE1 P30291 Human PBMCs A TPD-CPFXWG Dmax_1 WEE1 P30291 Human PBMCs B TPD-PQ21A8 Dmax_1 WEE1 P30291 Human PBMCs B TPD-QKTU5M Dmax_1 WEE1 P30291 Human PBMCs B TPD-K56440 Dmax_1 WEE1 P30291 Human PBMCs B TPD-32N6GU Dmax_1 WEE1 P30291 Human PBMCs B TPD-BU1YYO Dmax_1 WEE1 P30291 Human PBMCs A TPD-D9OJIS Dmax_1 WEE1 P30291 Human PBMCs A TPD-XRHTSQ Dmax_1 WEE1 P30291 Human PBMCs A TPD-J63IOC Dmax_1 WEE1 P30291 Human PBMCs A TPD-TJT65B Dmax_1 WEE1 P30291 Human PBMCs A TPD-FOUTHX Dmax_1 WEE1 P30291 Human PBMCs A TPD-R6B8DF Dmax_1 WEE1 P30291 Human PBMCs A TPD-SFMC89 Dmax_1 WEE1 P30291 Human PBMCs B TPD-EOL5BI Dmax_1 WEE1 P30291 Human PBMCs B TPD-8IIO95 Dmax_1 WEE1 P30291 Human PBMCs B TPD-OFAIH5 Dmax_1 WEE1 P30291 Human PBMCs B TPD-JMNCLG Dmax_1 WEE1 P30291 Human PBMCs A TPD-DOGJ1O Dmax_1 WEE1 P30291 Human PBMCs A TPD-GOGQQ6 Dmax_1 WEE1 P30291 Human PBMCs B TPD-4V0BZR Dmax_1 WEE1 P30291 Human PBMCs B TPD-0K0SBP Dmax_1 WEE1 P30291 Human PBMCs B TPD-IJENYE Dmax_1 WEE1 P30291 Human PBMCs A TPD-HT6HZQ Dmax_1 WEE1 P30291 Human PBMCs A TPD-SVN3LM Dmax_1 WEE1 P30291 Human PBMCs B TPD-9JRNX4 Dmax_1 WEE1 P30291 Human PBMCs A TPD-760NJ6 Dmax_1 WEE1 P30291 Human PBMCs A TPD-ZZYFRS Dmax_1 WEE1 P30291 Human PBMCs A TPD-PKQQMX Dmax_1 WEE1 P30291 Human PBMCs B TPD-2XGJ9Y Dmax_1 WEE1 P30291 Human PBMCs B TPD-N02C64 Dmax_2 IKZF1 Q13422 Human PBMCs A TPD-0T65BK Dmax_2 IKZF1 Q13422 Human PBMCs A TPD-9SDW2K Dmax_2 IKZF1 Q13422 Human PBMCs A TPD-CQJPPB Dmax_2 IKZF1 Q13422 Human PBMCs A TPD-SG1LPO Dmax_2 IKZF1 Q13422 Human PBMCs A TPD-17ZY6D Dmax_2 IKZF1 Q13422 Human PBMCs B TPD-PQ21A8 Dmax_2 IKZF1 Q13422 Human PBMCs B TPD-QKTU5M Dmax_2 IKZF1 Q13422 Human PBMCs B TPD-K56440 Dmax_2 IKZF1 Q13422 Human PBMCs B TPD-32N6GU Dmax_2 IKZF1 Q13422 Human PBMCs B TPD-BU1YYO Dmax_2 IKZF1 Q13422 Human PBMCs A TPD-J63IOC Dmax_2 IKZF1 Q13422 Human PBMCs A TPD-TJT65B Dmax_2 IKZF1 Q13422 Human PBMCs A TPD-FOUTHX Dmax_2 IKZF1 Q13422 Human PBMCs A TPD-R6B8DF Dmax_2 IKZF1 Q13422 Human PBMCs A TPD-SFMC89 Dmax_2 IKZF1 Q13422 Human PBMCs B TPD-0K0SBP Dmax_2 IKZF1 Q13422 Human PBMCs B TPD-IJENYE Dmax_2 IKZF1 Q13422 Human PBMCs B TPD-HT6HZQ Dmax_2 IKZF1 Q13422 Human PBMCs B TPD-SVN3LM Dmax_2 IKZF1 Q13422 Human PBMCs B TPD-9JRNX4 Dmax_2 IKZF1 Q13422 Human PBMCs B TPD-760NJ6 Dmax_2 IKZF1 Q13422 Human PBMCs B TPD-ZZYFRS Dmax_2 IKZF1 Q13422 Human PBMCs B TPD-PKQQMX Dmax_2 IKZF1 Q13422 Human PBMCs A TPD-2XGJ9Y Dmax_2 IKZF1 Q13422 Human PBMCs B TPD-9KKPOB IC50_1 . . NCI-H1155 A TPD-ES6X6S IC50_1 . . NCI-H1155 A TPD-9KKPOB IC50_2 . . NCI-H526 A TPD-JHXRQ9 Dmax_1(200μM) SIRT6 Q8N6T7 SK-HEP-1 <10.0% TPD-SJ3VL9 Dmax_1(200μM) SIRT6 Q8N6T7 SK-HEP-1 94.50% TPD-OU9NBT Dmax_1(200μM) SIRT6 Q8N6T7 SK-HEP-1 67.70% TPD-N5IWUB Dmax_1(200μM) SIRT6 Q8N6T7 SK-HEP-1 <10.0% TPD-Y0KW1C Dmax_1(200μM) SIRT6 Q8N6T7 SK-HEP-1 <10.0% TPD-JHXRQ9 Dmax_2(2μM) SIRT6 Q8N6T7 SK-HEP-1 20.60% TPD-SJ3VL9 Dmax_2(2μM) SIRT6 Q8N6T7 SK-HEP-1 99.80% TPD-OU9NBT Dmax_2(2μM) SIRT6 Q8N6T7 SK-HEP-1 92.50% TPD-N5IWUB Dmax_2(2μM) SIRT6 Q8N6T7 SK-HEP-1 56.60% TPD-Y0KW1C Dmax_2(2μM) SIRT6 Q8N6T7 SK-HEP-1 19.80% TPD-1D64R9 Dmax_1 IKZF1 Q13422 MV-4-11 A TPD-4CU130 Dmax_1 IKZF1 Q13422 MV-4-11 A TPD-67UXU2 Dmax_1 IKZF1 Q13422 MV-4-11 A TPD-1D64R9 Dmax_2 CK1α P48729 MV-4-11 B TPD-4CU130 Dmax_2 CK1α P48729 MV-4-11 B TPD-67UXU2 Dmax_2 CK1α P48729 MV-4-11 A TPD-I1CLO5 Inhibition(1μM) . . MOLM-13 A TPD-0XGXGD Inhibition(1μM) . . MOLM-13 D TPD-0SPC34 Inhibition(1μM) . . MOLM-13 A TPD-WJG4XA Inhibition(1μM) . . MOLM-13 D TPD-VSM2ZA Inhibition(1μM) . . MOLM-13 D TPD-T6VAYX Inhibition(1μM) . . MOLM-13 D TPD-9MDN3M Inhibition(1μM) . . MOLM-13 D TPD-HTOE4A Inhibition(1μM) . . MOLM-13 C TPD-RSY1ZG Inhibition(1μM) . . MOLM-13 C TPD-8QX0HD Inhibition(1μM) . . MOLM-13 D TPD-MN0CG5 Inhibition(1μM) . . MOLM-13 D TPD-RQZLCF Inhibition(1μM) . . MOLM-13 D TPD-34IDI9 Inhibition(1μM) . . MOLM-13 A TPD-CZCKQE Inhibition(1μM) . . MOLM-13 D TPD-L5SAJD Inhibition(1μM) . . MOLM-13 C TPD-CR19GY Inhibition(1μM) . . MOLM-13 D TPD-PND18P Inhibition(1μM) . . MOLM-13 D TPD-2PHCI0 Inhibition(1μM) . . MOLM-13 C TPD-9ZOM0M Inhibition(1μM) . . MOLM-13 D TPD-MDHIG0 Inhibition(1μM) . . MOLM-13 D TPD-6TLNFV Inhibition(1μM) . . MOLM-13 A TPD-PN28KY Inhibition(1μM) . . MOLM-13 A TPD-BQIPD0 Inhibition(1μM) . . MOLM-13 A TPD-QI1202 Inhibition(1μM) . . MOLM-13 A TPD-Y8VLYY Inhibition(1μM) . . MOLM-13 D TPD-BJCB8I Inhibition(1μM) . . MOLM-13 A TPD-HSEK6K Inhibition(1μM) . . MOLM-13 A TPD-GWFS7E Inhibition(1μM) . . MOLM-13 D TPD-OUN0Z6 EC50_1 IKZF1 Q13422 GripTite 293 MSR 0.057μM TPD-9BQ0UC EC50_1 IKZF1 Q13422 GripTite 293 MSR 0.046μM TPD-OUN0Z6 Dmax_1 IKZF1 Q13422 GripTite 293 MSR 75% TPD-9BQ0UC Dmax_1 IKZF1 Q13422 GripTite 293 MSR >90% TPD-XS5RPH EC50_2 GSPT1 P15170 GripTite 293 MSR 0.170μM TPD-XS5RPH Dmax_2 GSPT1 P15170 GripTite 293 MSR 80% TPD-LFN6D0 IC50_1 . . VCaP D TPD-VH8DQ0 IC50_1 . . VCaP D TPD-ERZW9S IC50_1 . . VCaP D TPD-8KNVWI IC50_1 . . VCaP D TPD-TDAGCR IC50_1 . . VCaP D TPD-GVGHLI IC50_1 . . VCaP D TPD-X5OPPJ IC50_1 . . VCaP C TPD-MGXQ2Q IC50_1 . . VCaP D TPD-JK2W52 IC50_1 . . VCaP D TPD-ARWONA IC50_1 . . VCaP D TPD-LFN6D0 IC50_2 . . 22Rv1-Enz D TPD-VH8DQ0 IC50_2 . . 22Rv1-Enz D TPD-ERZW9S IC50_2 . . 22Rv1-Enz D TPD-8KNVWI IC50_2 . . 22Rv1-Enz D TPD-TDAGCR IC50_2 . . 22Rv1-Enz D TPD-GVGHLI IC50_2 . . 22Rv1-Enz D TPD-X5OPPJ IC50_2 . . 22Rv1-Enz D TPD-MGXQ2Q IC50_2 . . 22Rv1-Enz D TPD-JK2W52 IC50_2 . . 22Rv1-Enz D TPD-ARWONA IC50_2 . . 22Rv1-Enz D TPD-GHHGQG Dmax GSPT1 P15170 AML(KG-1) A TPD-JEJ5K8 Dmax GSPT1 P15170 AML(KG-1) A TPD-L0I189 Dmax GSPT1 P15170 AML(KG-1) A TPD-YTZKG6 Dmax GSPT1 P15170 AML(KG-1) A TPD-Y6HHZ1 Dmax GSPT1 P15170 AML(KG-1) B TPD-XXX0CD Dmax GSPT1 P15170 AML(KG-1) B TPD-S5YJAJ Dmax GSPT1 P15170 AML(KG-1) B TPD-GHHGQG IC50_1 . . AML(KG-1) C TPD-JEJ5K8 IC50_1 . . AML(KG-1) C TPD-L0I189 IC50_1 . . AML(KG-1) C TPD-YTZKG6 IC50_1 . . AML(KG-1) C TPD-Y6HHZ1 IC50_1 . . AML(KG-1) C TPD-XXX0CD IC50_1 . . AML(KG-1) C TPD-S5YJAJ IC50_1 . . AML(KG-1) D