TPD ID	Activity Type	Target Symbols	Target IDs	Cell Line	Activity
TPD-WS9P5Y	IC50(uM)	.	.	A549	>10
TPD-Y3IMPJ	IC50(uM)	.	.	A549	>10
TPD-7IHN3X	IC50(uM)	.	.	A549	>10
TPD-9HNARD	IC50(uM)	.	.	A549	>10
TPD-S9B361	IC50(uM)	.	.	A549	>10
TPD-8O5H8S	IC50(uM)	.	.	A549	>10
TPD-P57IIM	IC50(uM)	.	.	A549	>10
TPD-HUKE2O	IC50(uM)	.	.	A549	>10
TPD-F7UAFK	IC50(uM)	.	.	A549	>10
TPD-VIXCXK	IC50(uM)	.	.	A549	>10
TPD-YBWUDJ	IC50(uM)	.	.	A549	>10
TPD-VVA70G	IC50(uM)	.	.	A549	>10
TPD-LHDW8S	IC50(uM)	.	.	A549	>10
TPD-PPD40N	IC50(uM)	.	.	A549	>10
TPD-BNDDH4	IC50(uM)	.	.	A549	>10
TPD-FNQCQL	IC50(uM)	.	.	A549	>10
TPD-18F8A7	IC50(uM)	.	.	A549	>10
TPD-RJHT21	IC50(uM)	.	.	A549	>10
TPD-MIYDQ8	IC50(uM)	.	.	A549	>10
TPD-X8L5S7	IC50(uM)	.	.	A549	>10
TPD-VNU6UM	IC50(uM)	.	.	A549	>10
TPD-WS9P5Y	IC50(uM)	.	.	HCC827	1.278±0.465
TPD-Y3IMPJ	IC50(uM)	.	.	HCC827	2.78±0.635
TPD-7IHN3X	IC50(uM)	.	.	HCC827	0.278±0.070
TPD-9HNARD	IC50(uM)	.	.	HCC827	0.923±0.227
TPD-S9B361	IC50(uM)	.	.	HCC827	1.149±0.552
TPD-8O5H8S	IC50(uM)	.	.	HCC827	0.210±0.154
TPD-P57IIM	IC50(uM)	.	.	HCC827	>10
TPD-HUKE2O	IC50(uM)	.	.	HCC827	2.193±0.334
TPD-F7UAFK	IC50(uM)	.	.	HCC827	0.976±0.029
TPD-VIXCXK	IC50(uM)	.	.	HCC827	>10
TPD-YBWUDJ	IC50(uM)	.	.	HCC827	1.058±0.182
TPD-VVA70G	IC50(uM)	.	.	HCC827	3.842±0.672
TPD-LHDW8S	IC50(uM)	.	.	HCC827	5.874±0.110
TPD-PPD40N	IC50(uM)	.	.	HCC827	6.033±0.556
TPD-BNDDH4	IC50(uM)	.	.	HCC827	>10
TPD-FNQCQL	IC50(uM)	.	.	HCC827	1.721±0.692
TPD-18F8A7	IC50(uM)	.	.	HCC827	0.862±0.274
TPD-RJHT21	IC50(uM)	.	.	HCC827	0.937±0.137
TPD-MIYDQ8	IC50(uM)	.	.	HCC827	1.158±0.447
TPD-X8L5S7	IC50(uM)	.	.	HCC827	1.146±0.574
TPD-VNU6UM	IC50(uM)	.	.	HCC827	1.72±0.443
TPD-WS9P5Y	IC50(uM)	.	.	PC-9	7.965±0.405
TPD-Y3IMPJ	IC50(uM)	.	.	PC-9	11.134±1.85
TPD-7IHN3X	IC50(uM)	.	.	PC-9	5.614±0.271
TPD-9HNARD	IC50(uM)	.	.	PC-9	7.035±0.795
TPD-S9B361	IC50(uM)	.	.	PC-9	6.756±0.705
TPD-8O5H8S	IC50(uM)	.	.	PC-9	>10
TPD-P57IIM	IC50(uM)	.	.	PC-9	>10
TPD-HUKE2O	IC50(uM)	.	.	PC-9	>10
TPD-F7UAFK	IC50(uM)	.	.	PC-9	>10
TPD-VIXCXK	IC50(uM)	.	.	PC-9	>10
TPD-YBWUDJ	IC50(uM)	.	.	PC-9	3.119±0.4002
TPD-VVA70G	IC50(uM)	.	.	PC-9	5.121±1.275
TPD-LHDW8S	IC50(uM)	.	.	PC-9	>10
TPD-PPD40N	IC50(uM)	.	.	PC-9	3.812±0.363
TPD-BNDDH4	IC50(uM)	.	.	PC-9	7.723±0.777
TPD-FNQCQL	IC50(uM)	.	.	PC-9	3.529±0.395
TPD-18F8A7	IC50(uM)	.	.	PC-9	1.357±0.161
TPD-RJHT21	IC50(uM)	.	.	PC-9	3.784±0.360
TPD-MIYDQ8	IC50(uM)	.	.	PC-9	3.634±0.284
TPD-X8L5S7	IC50(uM)	.	.	PC-9	1.428±0.124
TPD-VNU6UM	IC50(uM)	.	.	PC-9	1.087±0.0593
TPD-WS9P5Y	IC50(uM)	.	.	NCI-H3255	3.100±0.175
TPD-Y3IMPJ	IC50(uM)	.	.	NCI-H3255	4.795±0.099
TPD-7IHN3X	IC50(uM)	.	.	NCI-H3255	2.998±0.322
TPD-9HNARD	IC50(uM)	.	.	NCI-H3255	3.41±0.061
TPD-S9B361	IC50(uM)	.	.	NCI-H3255	4.143±0.465
TPD-8O5H8S	IC50(uM)	.	.	NCI-H3255	6.042±0.340
TPD-P57IIM	IC50(uM)	.	.	NCI-H3255	>10
TPD-HUKE2O	IC50(uM)	.	.	NCI-H3255	6.505±0.758
TPD-F7UAFK	IC50(uM)	.	.	NCI-H3255	4.932±0.096
TPD-VIXCXK	IC50(uM)	.	.	NCI-H3255	5.183±0.462
TPD-YBWUDJ	IC50(uM)	.	.	NCI-H3255	2.842±0.515
TPD-VVA70G	IC50(uM)	.	.	NCI-H3255	2.542±0.0318
TPD-LHDW8S	IC50(uM)	.	.	NCI-H3255	4.581±0.105
TPD-PPD40N	IC50(uM)	.	.	NCI-H3255	2.001±0.243
TPD-BNDDH4	IC50(uM)	.	.	NCI-H3255	4.851±0.098
TPD-FNQCQL	IC50(uM)	.	.	NCI-H3255	2.461±0.221
TPD-18F8A7	IC50(uM)	.	.	NCI-H3255	1.829±0.011
TPD-RJHT21	IC50(uM)	.	.	NCI-H3255	1.133±0.113
TPD-MIYDQ8	IC50(uM)	.	.	NCI-H3255	0.904±0.181
TPD-X8L5S7	IC50(uM)	.	.	NCI-H3255	0.908±0.130
TPD-VNU6UM	IC50(uM)	.	.	NCI-H3255	1.43±0.163
TPD-WS9P5Y	IC50(uM)	.	.	NCI-H1975	>10
TPD-Y3IMPJ	IC50(uM)	.	.	NCI-H1975	>10
TPD-7IHN3X	IC50(uM)	.	.	NCI-H1975	>10
TPD-9HNARD	IC50(uM)	.	.	NCI-H1975	>10
TPD-S9B361	IC50(uM)	.	.	NCI-H1975	>10
TPD-8O5H8S	IC50(uM)	.	.	NCI-H1975	>10
TPD-P57IIM	IC50(uM)	.	.	NCI-H1975	>10
TPD-HUKE2O	IC50(uM)	.	.	NCI-H1975	>10
TPD-F7UAFK	IC50(uM)	.	.	NCI-H1975	>10
TPD-VIXCXK	IC50(uM)	.	.	NCI-H1975	>10
TPD-YBWUDJ	IC50(uM)	.	.	NCI-H1975	>10
TPD-VVA70G	IC50(uM)	.	.	NCI-H1975	>10
TPD-LHDW8S	IC50(uM)	.	.	NCI-H1975	>10
TPD-PPD40N	IC50(uM)	.	.	NCI-H1975	>10
TPD-BNDDH4	IC50(uM)	.	.	NCI-H1975	>10
TPD-FNQCQL	IC50(uM)	.	.	NCI-H1975	>10
TPD-18F8A7	IC50(uM)	.	.	NCI-H1975	>10
TPD-RJHT21	IC50(uM)	.	.	NCI-H1975	>10
TPD-MIYDQ8	IC50(uM)	.	.	NCI-H1975	>10
TPD-X8L5S7	IC50(uM)	.	.	NCI-H1975	3.179±0.245
TPD-VNU6UM	IC50(uM)	.	.	NCI-H1975	>10
TPD-KJCNEJ	IC50	.	.	PanC-1	2.51 ± 0.04μM
TPD-2LKCWL	IC50	.	.	PanC-1	3.11 ± 0.59μM
TPD-GC2IY1	IC50	.	.	PanC-1	1.18 ± 0.24μM
TPD-4JUUCX	IC50	.	.	PanC-1	1.71 ± 0.18μM
TPD-I8NK5J	IC50	.	.	PanC-1	2.20 ± 0.46μM
TPD-KJCNEJ	IC50	.	.	PanC-1	3.29 ± 0.36μM
TPD-2LKCWL	IC50	.	.	PanC-1	1.54 ± 0.32μM
TPD-GC2IY1	IC50	.	.	PanC-1	1.77 ± 0.25μM
TPD-4JUUCX	IC50	.	.	PanC-1	1.83 ± 0.26μM
TPD-I8NK5J	IC50	.	.	PanC-1	2.70 ± 0.57μM
TPD-KJCNEJ	IC50	.	.	PanC-1	5.42 ± 0.69μM
TPD-2LKCWL	IC50	.	.	PanC-1	7.20 ± 0.40μM
TPD-GC2IY1	IC50	.	.	PanC-1	8.00 ± 0.94μM
TPD-4JUUCX	IC50	.	.	PanC-1	>30.00μM
TPD-I8NK5J	IC50	.	.	PanC-1	>30.00μM
TPD-KJCNEJ	IC50	.	.	4T1	24.72 ± 3.68μM
TPD-2LKCWL	IC50	.	.	4T1	7.96 ± 0.10μM
TPD-GC2IY1	IC50	.	.	4T1	>30.00μM
TPD-4JUUCX	IC50	.	.	4T1	15.59 ± 0.96μM
TPD-I8NK5J	IC50	.	.	4T1	14.90 ± 2.07μM
TPD-KJCNEJ	IC50	.	.	HEK293T	>30.00μM
TPD-2LKCWL	IC50	.	.	HEK293T	>30.00μM
TPD-GC2IY1	IC50	.	.	HEK293T	4.13 ± 0.28μM
TPD-4JUUCX	IC50	.	.	HEK293T	>30.00μM
TPD-I8NK5J	IC50	.	.	HEK293T	>30.00μM
TPD-JEQMSR	Kd	.	.	.	153 ± 65
TPD-O30DLH	Kd	.	.	.	52 ± 12
TPD-NZNO4R	Kd	.	.	.	74 ± 19
TPD-OQUUKT	Kd	.	.	.	116 ± 56
TPD-IH1PPY	Kd	.	.	.	82 ± 38
TPD-SOUJ1Y	Kd	.	.	.	56 ± 4.3
TPD-ZVNWSM	Kd	.	.	.	51 ± 19
TPD-9VU21Q	Kd	.	.	.	71 ± 0.9
TPD-K9YDDC	Kd	.	.	.	73 ± 3.3
TPD-6QGT18	Kd	.	.	.	74 ± 6.1
TPD-7GPQBY	Kd	.	.	.	94 ± 13
TPD-4BLGU6	Kd	.	.	.	82 ± 2.0
TPD-JEQMSR	Dmax	.	.	.	46%
TPD-O30DLH	Dmax	.	.	.	59%
TPD-NZNO4R	Dmax	.	.	.	66%
TPD-OQUUKT	Dmax	.	.	.	51%
TPD-IH1PPY	Dmax	.	.	.	60%
TPD-SOUJ1Y	Dmax	.	.	.	85%
TPD-ZVNWSM	Dmax	.	.	.	24%
TPD-9VU21Q	Dmax	.	.	.	32%
TPD-K9YDDC	Dmax	.	.	.	35%
TPD-6QGT18	Dmax	.	.	.	33%
TPD-7GPQBY	Dmax	.	.	.	13%
TPD-4BLGU6	Dmax	.	.	.	42%
TPD-4BLGU6	Dmax	.	.	.	42%
TPD-B23WDK	.	PD-L1	Q9NZQ7	B16F10	see description for details
TPD-B23WDK	.	PD-L1	Q9NZQ7	B16F10	see description for details
TPD-B23WDK	.	PD-L1	Q9NZQ7	B16F10	see description for details
TPD-0M4J0K	.	HER2	P04626	HepG2	see description for details
TPD-391KD4	.	EGFR	P00533	HEP3B&HepG2&Huh7	see description for details
TPD-CE0QWQ	.	.	.	MCF-10A&MCF-7	see description for details
TPD-CE0QWQ	.	.	.	MCF-10A&MCF-7	see description for details
TPD-FCJYPV	.	PD-L1	Q9NZQ7	HCT-116	see description for details
TPD-MAK3WW	.	PD-L1	Q9NZQ7	HCT-116	see description for details
TPD-KR8048	.	.	.	HepG2	see description for details
TPD-MGJONI	.	.	.	HepG2	see description for details
TPD-MGJONI	.	.	.	HepG2	see description for details
TPD-MGJONI	.	.	.	HepG2	see description for details
TPD-BNTQBS	.	.	.	HeLa	see description for details
TPD-BNTQBS	.	.	.	HeLa	see description for details
TPD-PF5U6N	.	.	.	.	see description for details
TPD-PF5U6N	.	.	.	HeLa	see description for details
TPD-L92JJ4	.	.	.	HeLa	see description for details
TPD-PT2WW8	Dmax	.	.	HeLa	67%
TPD-PT2WW8	Dmax	.	.	HeLa	70%
TPD-C7A8A2	.	.	.	HeLa	see description for details
TPD-U2P6AF	.	PD-L1	Q9NZQ7	H460&CT26	see description for details
TPD-U2P6AF	.	PD-L1	Q9NZQ7	H460GFP-PDL1 cells	see description for details
TPD-U2P6AF	.	PD-L1	Q9NZQ7	H460&Jurkat	see description for details
TPD-U2P6AF	.	PD-L1	Q9NZQ7	H460&Jurkat	see description for details
TPD-U2P6AF	.	PD-L1	Q9NZQ7	H460&Jurkat	see description for details
TPD-7MZP9B	.	PD-L1	Q9NZQ7	.	see description for details
TPD-7MZP9B	.	PD-L1	Q9NZQ7	Panc 10.05	see description for details
TPD-7MZP9B	.	PD-L1	Q9NZQ7	RL95-2	see description for details
TPD-F9JZ49	.	PD-L1	Q9NZQ7	HeLa	see description for details
TPD-DJN393	.	PD-L1	Q9NZQ7	B16&MC38	see description for details
TPD-VTM4ME	.	PD-L1	Q9NZQ7	B16&MC38	see description for details
TPD-9VB11C	.	PD-L1	Q9NZQ7	B16&MC38	see description for details
TPD-HFFAET	.	PD-L1	Q9NZQ7	B16&MC38	see description for details
TPD-HFFAET	.	PD-L1	Q9NZQ7	.	see description for details
TPD-HFFAET	.	PD-L1	Q9NZQ7	CHO-K1-hPD-1&CHO-K1-mPD-1	see description for details
TPD-RKWK2G	.	PD-L1	Q9NZQ7	B16&MC38	see description for details
TPD-RKWK2G	.	PD-L1	Q9NZQ7	CHO-K1-hPD-1&CHO-K1-mPD-1	see description for details
TPD-UWK1SA	.	.	.	.	see description for details
TPD-8NKPAY	.	.	.	.	see description for details
TPD-5L3Y8N	.	.	.	.	see description for details
TPD-M9BDKD	.	.	.	.	see description for details
TPD-M9BDKD	Kd_1	.	.	.	3670nM
TPD-M9BDKD	Kd_2	.	.	.	106.3nM
TPD-M9BDKD	.	.	.	.	see description for details
TPD-4RP3UC	.	.	.	.	see description for details
TPD-4RP3UC	Kd_1	.	.	.	46.87nM
TPD-4RP3UC	Kd_2	.	.	.	46.45nM
TPD-4RP3UC	.	.	.	.	see description for details
TPD-TPDLQD	.	.	.	.	see description for details
TPD-TPDLQD	Kd_1	.	.	.	198.84nM
TPD-TPDLQD	Kd_2	.	.	.	72.4nM
TPD-TPDLQD	.	.	.	.	see description for details
TPD-88PNXZ	Kd_1	.	.	.	6nM
TPD-88PNXZ	Kd_2	.	.	.	0.01nM
TPD-9YSPE5	Kd_1	.	.	.	0.4nM
TPD-9YSPE5	Kd_2	.	.	.	4nM
TPD-B5S8D7	.	.	.	4T1	see description for details
TPD-JLUMH3	.	PD-L1	Q9NZQ7	B16F10	see description for details
TPD-07THBZ	.	.	.	4T1	see description for details
TPD-Q0QIYL	.	.	.	.	see description for details
TPD-N03DH0	.	.	.	.	see description for details
TPD-IE8Q71	.	EGFR	P00533	HeLa	see description for details
TPD-IE8Q71	.	EGFR	P00533	HeLa	see description for details
TPD-CAXOV8	.	EGFR	P00533	HeLa	see description for details
TPD-CAXOV8	.	EGFR	P00533	HeLa	see description for details
TPD-8UWJH7	.	EGFR	P00533	HeLa	see description for details
TPD-8UWJH7	.	EGFR	P00533	HeLa	see description for details
TPD-5O1H48	.	EGFR	P00533	HeLa	see description for details
TPD-5O1H48	.	EGFR	P00533	HeLa	see description for details
TPD-G25QHQ	.	EGFR	P00533	HeLa	see description for details
TPD-Z1BW1A	.	EGFR	P00533	HeLa	see description for details
TPD-QBC6GI	.	EGFR	P00533	HeLa	see description for details
TPD-QBC6GI	.	EGFR	P00533	HeLa	see description for details
TPD-UOJIS6	.	EGFR	P00533	HeLa	see description for details
TPD-UOJIS6	.	EGFR	P00533	HeLa	see description for details
TPD-9ZMSS0	.	.	.	HeLa&MCF-7	see description for details
TPD-LIALEN	.	.	.	HeLa&MCF-7	see description for details
TPD-8V9OYP	.	.	.	HeLa&MCF-7	see description for details
TPD-EZHCK7	.	.	.	HeLa&MCF-7	see description for details
TPD-V2OU2D	.	.	.	HeLa&MCF-7	see description for details
TPD-Z4BY0F	.	.	.	HeLa&MCF-7	see description for details
TPD-H276AB	.	HER2	P04626	SKBR-3	see description for details
TPD-3HZ92C	.	HER2	P04626	SKBR-3	see description for details
TPD-70TTKA	.	HER2	P04626	SKBR-3	see description for details
TPD-E2ZT0H	.	EGFR	P00533	A431	see description for details
TPD-TKTQVR	.	PD-L1	Q9NZQ7	MDAMB231	see description for details
TPD-0N0FYU	.	PD-L1	Q9NZQ7	MDAMB231	see description for details
TPD-4BTL0J	.	PD-L1	Q9NZQ7	MDAMB231	see description for details
TPD-CUYXRW	.	PD-L1	Q9NZQ7	MDAMB231	see description for details
TPD-DPUM9Q	.	PD-L1	Q9NZQ7	MDAMB231	see description for details
TPD-4KDX76	.	PD-L1	Q9NZQ7	MDAMB231	see description for details
TPD-ONJGJ8	.	PD-L1	Q9NZQ7	MDAMB231	see description for details
TPD-GPRGF3	.	PD-L1	Q9NZQ7	MDAMB231	see description for details
TPD-3YTVNC	.	PD-L1	Q9NZQ7	MDAMB231	see description for details
TPD-PJJDVV	.	PD-L1	Q9NZQ7	MDAMB231	see description for details
TPD-DV3SS6	.	PD-L1	Q9NZQ7	MDAMB231	see description for details
TPD-P8WOLT	.	.	.	RAMOS	see description for details
TPD-L0SJDG	.	.	.	RAMOS	see description for details
TPD-XPKE50	.	.	.	Jurkat	see description for details
TPD-63KPB6	.	.	.	SKBR-3	see description for details
TPD-N3PTV9	.	.	.	SKBR-3	see description for details
TPD-ONBVRI	.	.	.	SKBR-3	see description for details
TPD-3SZKIG	.	.	.	SKBR-3	see description for details
TPD-MYMTFG	.	HER2	P04626	BT-474	see description for details
TPD-65F3IL	.	HER2	P04626	BT-474	see description for details
TPD-2UA2QI	.	HER2	P04626	BT-474	see description for details
TPD-B9AXI0	.	HER2	P04626	BT-474	see description for details
TPD-8SVV42	.	HER2	P04626	BT-474	see description for details
TPD-UAFCTK	.	HER2	P04626	BT-474	see description for details
TPD-O48952	.	HER2	P04626	BT-474	see description for details
TPD-850TZN	.	HER2	P04626	BT-474	see description for details
TPD-576VQ6	.	HER2	P04626	BT-474	see description for details
TPD-CN3R0D	.	HER2	P04626	BT-474	see description for details
TPD-59G8YO	.	HER2	P04626	BT-474	see description for details
TPD-6OJWNQ	.	HER2	P04626	BT-474	see description for details
TPD-UBQREF	.	HER2	P04626	BT-474	see description for details
TPD-LO9F8P	.	HER2	P04626	BT-474	see description for details
TPD-YGP1ZF	.	HER2	P04626	BT-474	see description for details
TPD-HJP8OO	.	HER2	P04626	BT-474	see description for details
TPD-103W79	.	HER2	P04626	BT-474	see description for details
TPD-EIQ69L	.	HER2	P04626	BT-474	see description for details
TPD-VZY48W	.	HER2	P04626	BT-474	see description for details
TPD-MIV4AP	.	HER2	P04626	BT-474	see description for details
TPD-ZT1MPD	.	HER2	P04626	BT-474	see description for details
TPD-LFOQM1	.	HER2	P04626	BT-474	see description for details
TPD-3IWAFN	.	HER2	P04626	BT-474	see description for details
TPD-B4QDTD	.	HER2	P04626	BT-474	see description for details
TPD-EIBLJO	.	EGFR	P00533	A431	see description for details
TPD-XWMYJX	.	EGFR	P00533	A431	see description for details
TPD-06ZUYQ	.	EGFR	P00533	A431	see description for details
TPD-AEDQ42	.	EGFR	P00533	A431	see description for details
TPD-NNKN2W	.	.	.	T24	see description for details
TPD-HD1N0F	Kd	.	.	SK-HEP-1	~80nM
TPD-KGV2SS	Kd	.	.	SK-HEP-1	~80nM
TPD-YMAC5H	Kd	.	.	SK-HEP-1	5.4nM
TPD-24N3G8	.	.	.	SK-HEP-1	see description for details
TPD-B90O5K	.	PD-L1	Q9NZQ7	MDAMB231	see description for details
TPD-0I7LR2	Degradation percentage(100nM)	HER2	P04626	SK-OV-3	73%
TPD-01M164	Degradation percentage(25nM)	EGFR	P00533	SK-HEP-1	73%
TPD-ZMLT5F	Degradation percentage(50nM)	.	.	HepG2	71%
TPD-HD1N0F	.	PD-L1	Q9NZQ7	MDAMB231	see description for details
TPD-YMAC5H	.	PD-L1	Q9NZQ7	MDAMB231	see description for details
TPD-HD1N0F	.	PD-L1	Q9NZQ7	A549&MCF-7&SK-OV-3	see description for details
TPD-YMAC5H	.	PD-L1	Q9NZQ7	A549&MCF-7&SK-OV-3	see description for details
TPD-ZL0RPS	.	EGFR	P00533	HeLa	see description for details
TPD-6G8JR6	.	.	.	SH-SY5Y	see description for details
TPD-XQA78B	.	PD-L1	Q9NZQ7	MDAMB231	see description for details
TPD-ZL0RPS	.	EGFR	P00533	HeLa	see description for details
TPD-2FKJHL	Kd	Sortilin	Q99523	.	+++
TPD-6VCCK1	Kd	Sortilin	Q99523	.	+++
TPD-35VEV0	Kd	Sortilin	Q99523	.	+++
TPD-ECUACK	Kd	Sortilin	Q99523	.	+++
TPD-32V6SG	Kd	Sortilin	Q99523	.	+++
TPD-ZCBC57	Kd	Sortilin	Q99523	.	+++
TPD-P03N3P	Kd	Sortilin	Q99523	.	+++
TPD-J5P9GJ	Kd	Sortilin	Q99523	.	+++
TPD-Y43GDL	Kd	Sortilin	Q99523	.	+++
TPD-19QF8H	Kd	Sortilin	Q99523	.	+++
TPD-NV5WIZ	Kd	Sortilin	Q99523	.	+++
TPD-W2CVQL	Kd	Sortilin	Q99523	.	++
TPD-VK4WO8	Kd	Sortilin	Q99523	.	+++
TPD-1B638C	Kd	Sortilin	Q99523	.	+++
TPD-IP9NQU	Kd	Sortilin	Q99523	.	+++
TPD-L54W2O	Kd	Sortilin	Q99523	.	++
TPD-MHWYHY	Kd	Sortilin	Q99523	.	++
TPD-RXPYCI	Kd	Sortilin	Q99523	.	++
TPD-61T8A1	Kd	Sortilin	Q99523	.	++
TPD-DG2MWI	Kd	Sortilin	Q99523	.	++
TPD-LH3R81	Kd	Sortilin	Q99523	.	++
TPD-6C1MTU	Kd	Sortilin	Q99523	.	++
TPD-8MWIGE	Kd	Sortilin	Q99523	.	++
TPD-XE8D7C	Kd	Sortilin	Q99523	.	++++
TPD-WWLKUM	Kd	Sortilin	Q99523	.	++
TPD-O05P7R	Kd	Sortilin	Q99523	.	+
TPD-XILTN7	Kd	Sortilin	Q99523	.	+++
TPD-HOI4SL	Kd	Sortilin	Q99523	.	+
TPD-TGIKJA	Kd	Sortilin	Q99523	.	++++
TPD-69MVBG	Kd	Sortilin	Q99523	.	+++
TPD-DGORDS	Kd	Sortilin	Q99523	.	++++
TPD-OSZFW2	Kd	Sortilin	Q99523	.	++
TPD-MHQN66	Kd	Sortilin	Q99523	.	+++
TPD-HECKWP	Kd	Sortilin	Q99523	.	++++
TPD-WKFIM9	Kd	Sortilin	Q99523	.	+++
TPD-QFBW6S	Kd	Sortilin	Q99523	.	+++
TPD-247R54	Kd	Sortilin	Q99523	.	+++
TPD-VI0KBX	Kd	Sortilin	Q99523	.	+++
TPD-A4ECSW	Kd	Sortilin	Q99523	.	+++
TPD-JY6I5E	Kd	Sortilin	Q99523	.	+++
TPD-GWL0BV	Kd	Sortilin	Q99523	.	++
TPD-VD1VQX	Kd	Sortilin	Q99523	.	+++
TPD-95PH1L	Kd	Sortilin	Q99523	.	++++
TPD-KWIFE7	Kd	Sortilin	Q99523	.	+++
TPD-5TQLG1	Kd	Sortilin	Q99523	.	+++
TPD-PAQL7J	Kd	Sortilin	Q99523	.	+++
TPD-PMPHX5	Kd	Sortilin	Q99523	.	++++
TPD-QLGN9K	Kd	Sortilin	Q99523	.	+++
TPD-I5P12Q	Kd	Sortilin	Q99523	.	++++
TPD-H4OO60	Kd	Sortilin	Q99523	.	+++
TPD-WBZQRH	Kd	Sortilin	Q99523	.	+++
TPD-M90VUJ	Kd	Sortilin	Q99523	.	++++
TPD-9QOLU9	Kd	Sortilin	Q99523	.	++
TPD-2XWUF1	Kd	Sortilin	Q99523	.	++
TPD-JEN5W4	Kd	Sortilin	Q99523	.	++++
TPD-PZAEO9	Kd	Sortilin	Q99523	.	++++
TPD-EMYPFD	Kd	Sortilin	Q99523	.	+++
TPD-8SRTK1	Kd	Sortilin	Q99523	.	++++
TPD-25G3QJ	Kd	Sortilin	Q99523	.	+++
TPD-8IOBJN	Kd	Sortilin	Q99523	.	+++
TPD-TWPWNI	Kd	Sortilin	Q99523	.	++++
TPD-OI6YT3	Kd	Sortilin	Q99523	.	++++
TPD-M81BI5	Kd	Sortilin	Q99523	.	++++
TPD-DMF9NX	Kd	Sortilin	Q99523	.	++++
TPD-IK80I8	Kd	Sortilin	Q99523	.	+++
TPD-NE0M31	Kd	Sortilin	Q99523	.	+++
TPD-MRHKXN	Kd	Sortilin	Q99523	.	+++
TPD-NR4708	Kd	Sortilin	Q99523	.	+++
TPD-97WCBI	Kd	Sortilin	Q99523	.	+++
TPD-GOXY46	Kd	Sortilin	Q99523	.	++++
TPD-TEI5DO	Kd	Sortilin	Q99523	.	++++
TPD-A5CQPR	Kd	Sortilin	Q99523	.	+++
TPD-RKH4SJ	Kd	Sortilin	Q99523	.	++
TPD-8V42YD	Kd	Sortilin	Q99523	.	++++
TPD-J90B98	Kd	Sortilin	Q99523	.	++++
TPD-7PGQFA	Kd	Sortilin	Q99523	.	++++
TPD-GXJLQE	Kd	Sortilin	Q99523	.	+++
TPD-PU5HX7	Kd	Sortilin	Q99523	.	+++
TPD-QLKGGI	normalized KRAS levels_1(3.33 μM Compound Concentration)	KRAS	P01116	NCI-H2030	84.90%
TPD-XFJWJ1	normalized KRAS levels_1(3.33 μM Compound Concentration)	KRAS	P01116	NCI-H2030	45.10%
TPD-93OD2F	normalized KRAS levels_1(3.33 μM Compound Concentration)	KRAS	P01116	NCI-H2030	63.00%
TPD-G2Q8KL	Normalized BTK levels_2(10 μM Compound Concentration)	BTK	Q06187	NAMALWA	~58.7 %
TPD-K7NHEO	Normalized BTK levels_1(3.33 μM Compound Concentration)	BTK	Q06187	NAMALWA	67.00%
TPD-ENY4CV	Normalized BTK levels_1(3.33 μM Compound Concentration)	BTK	Q06187	NAMALWA	83.10%
TPD-CQN0FF	IC50_1	.	.	MCF-7	26.2μM
TPD-J5C2HB	IC50	.	.	U2932	624nM
TPD-56ONXC	IC50	.	.	U2932	534nM
TPD-4CIEOJ	IC50	.	.	U2932	359nM
TPD-E2NWFC	IC50	.	.	U2932	604nM
TPD-ER35J7	IC50	.	.	U2932	346nM
TPD-55B1DB	IC50	.	.	U2932	484nM
TPD-F7LSJ7	IC50	.	.	U2932	125nM
TPD-PPOVQ1	IC50	.	.	U2932	424nM
TPD-1CWTDT	IC50	.	.	U2932	142nM
TPD-CPLM1P	IC50	.	.	U2932	45nM
TPD-36YV82	IC50	.	.	U2932	180nM
TPD-Y2Z1T2	IC50	.	.	U2932	109nM
TPD-P70P2I	IC50	.	.	U2932	320nM
TPD-1EVGJH	IC50	.	.	U2932	120nM
TPD-RF2HK6	IC50	.	.	U2932	157nM
TPD-ILLLK4	IC50	.	.	U2932	45nM
TPD-VK0VOJ	IC50	.	.	U2932	192nM
TPD-KZFC9C	IC50	.	.	U2932	124nM
TPD-DVISGW	IC50	.	.	U2932	104nM
TPD-WO5PLC	IC50	.	.	U2932	155nM
TPD-M1I471	IC50	.	.	U2932	133nM
TPD-E2WUEH	IC50	.	.	U2932	98nM
TPD-ZFPXTG	IC50	.	.	U2932	145nM
TPD-2VQG7N	100nM Degradation	PCSK9	Q8NBP7	Huh7	46.8±2.7%
TPD-YC2BN5	100nM Degradation	PCSK9	Q8NBP7	Huh7	48.7±5.6%
TPD-H5686H	100nM Degradation	PCSK9	Q8NBP7	Huh7	57.4±8.2%
TPD-J003G6	100nM Degradation	PCSK9	Q8NBP7	Huh7	48.3±7.5%
TPD-A5XHGC	100nM Degradation	PCSK9	Q8NBP7	Huh7	32.3±23.6%
TPD-RFNGHK	100nM Degradation	PCSK9	Q8NBP7	Huh7	15.6±13.1%
TPD-CMMGXV	100nM Degradation	PCSK9	Q8NBP7	Huh7	36.7±12.9%
TPD-DPSMCP	100nM Degradation	PCSK9	Q8NBP7	Huh7	35.7±8.5%
TPD-N3GSDO	100nM Degradation	PCSK9	Q8NBP7	Huh7	27.5±7.56%
TPD-0V0VD7	100nM Degradation	PCSK9	Q8NBP7	Huh7	24.7±5.5%
TPD-G6ZGDP	100nM Degradation	PCSK9	Q8NBP7	Huh7	41.0±1.1%
TPD-VOPKHB	100nM Degradation	PCSK9	Q8NBP7	Huh7	44.9±5.7%
TPD-VN00OX	Inhibiton_1(100nM)	NLRP3	Q96P20	THP-1	50.4±7.3%
TPD-95XZDM	Inhibiton_1(100nM)	NLRP3	Q96P20	THP-1	-7.2±10.7%
TPD-096V09	Inhibiton_1(100nM)	NLRP3	Q96P20	THP-1	7.3±9.0%
TPD-IA6O5U	Inhibiton_1(100nM)	NLRP3	Q96P20	THP-1	39.0±9.5%
TPD-83LYO1	Inhibiton_1(100nM)	NLRP3	Q96P20	THP-1	11.0±3.2%
TPD-0H20UG	Inhibiton_1(100nM)	NLRP3	Q96P20	THP-1	8.2±3.4%
TPD-C135OX	Inhibiton_1(100nM)	NLRP3	Q96P20	THP-1	19.2±7.3%
TPD-LJSPHN	Inhibiton_1(100nM)	NLRP3	Q96P20	THP-1	27.7±5.6%
TPD-U7BWWQ	Inhibiton_1(100nM)	NLRP3	Q96P20	THP-1	20.4±7.3%
TPD-QCF1E1	Inhibiton_1(100nM)	NLRP3	Q96P20	THP-1	35.6±5.2%
TPD-DF2N5D	Inhibiton_1(100nM)	NLRP3	Q96P20	THP-1	16.5±2.7%
TPD-IU0VYK	Inhibiton_1(100nM)	NLRP3	Q96P20	THP-1	57.6±5.9%
TPD-RDHTMN	Inhibiton_1(100nM)	NLRP3	Q96P20	THP-1	42.8±6.4%
TPD-UVS853	Inhibiton_1(100nM)	NLRP3	Q96P20	THP-1	-5.3±6.6%
TPD-NDRQ1S	Inhibiton_1(100nM)	NLRP3	Q96P20	THP-1	14.8±4.9%
TPD-S0FHNY	Inhibiton_1(100nM)	NLRP3	Q96P20	THP-1	20.5±7.8%
TPD-64VJHN	Inhibiton_1(100nM)	NLRP3	Q96P20	THP-1	17.8±9.3%
TPD-ZAE7Z2	Inhibiton_1(100nM)	NLRP3	Q96P20	THP-1	6.7±5.9%
TPD-TCMXXF	Inhibiton_1(100nM)	NLRP3	Q96P20	THP-1	43.1±8.7%
TPD-K7F3BH	Inhibiton_1(100nM)	NLRP3	Q96P20	THP-1	41.9±7.4%
TPD-T5OPGC	Inhibiton_1(100nM)	NLRP3	Q96P20	THP-1	40.1±9.8%
TPD-LISID0	Inhibiton_1(100nM)	NLRP3	Q96P20	THP-1	70.4±9.9%
TPD-1FT2G6	Inhibiton_1(100nM)	NLRP3	Q96P20	THP-1	50.5±5.1%
TPD-L0GDB2	Inhibiton_1(100nM)	NLRP3	Q96P20	THP-1	45.8±9.2%
TPD-P3P0JK	IC50_1	NAMPT	P43490	.	26.1nM
TPD-ON9FHH	IC50_1	NAMPT	P43490	.	51.9nM
TPD-NVRO2H	GFP level under 0.001 μM treatment	.	.	HeLa	1.155±0.107
TPD-PM46YH	DC50	.	.	HEK293T	1.48nM
TPD-FI8G56	DC50	AR	P10275	LNCaP	211.08nM
TPD-QD82Q1	DC50	MetAP2	P50579	HEK293T	0.701μM
TPD-D2288Z	DC50	Tau	P10636	SH-SY5Y-tauP301L	0.71nM
TPD-K7OHH2	DC50	Tau	P10636	SH-SY5Y-tauP301L	2.63nM
TPD-F608B9	Kd_1	HTT exon1	P42858	.	157.6nM
TPD-RRU054	Kd_1	HTT exon1	P42858	.	29.2nM
TPD-NVRO2H	GFP level under 0.01 μM treatment	.	.	HeLa	1.126±0.148
TPD-NVRO2H	GFP level under   0.1 μM treatment	.	.	HeLa	0.929±0.038
TPD-NVRO2H	GFP level under     1 μM treatment	.	.	HeLa	0.377±0.054
TPD-NVRO2H	GFP level under    10 μM treatment	.	.	HeLa	0.305±0.088
TPD-F608B9	Kd_2	LC3B	Q9GZQ8	.	467.7nM
TPD-RRU054	Kd_2	LC3B	Q9GZQ8	.	238.2nM
TPD-F608B9	Kd_3	HTT(full length)	P42858	.	14.7nM
TPD-RRU054	Kd_3	HTT(full length)	P42858	.	321.9nM
TPD-P3P0JK	IC50_2	.	.	A2780	2.7μM
TPD-ON9FHH	IC50_2	.	.	A2780	0.19μM
TPD-VN00OX	Inhibiton_2(200nM)	NLRP3	Q96P20	THP-1	36.2±3.1%
TPD-95XZDM	Inhibiton_2(200nM)	NLRP3	Q96P20	THP-1	37.9±9.6%
TPD-096V09	Inhibiton_2(200nM)	NLRP3	Q96P20	THP-1	28.0±2.5%
TPD-IA6O5U	Inhibiton_2(200nM)	NLRP3	Q96P20	THP-1	23.1±12.4%
TPD-83LYO1	Inhibiton_2(200nM)	NLRP3	Q96P20	THP-1	43.1±7.7%
TPD-0H20UG	Inhibiton_2(200nM)	NLRP3	Q96P20	THP-1	-4.9±4.1%
TPD-C135OX	Inhibiton_2(200nM)	NLRP3	Q96P20	THP-1	40.8±9.8%
TPD-LJSPHN	Inhibiton_2(200nM)	NLRP3	Q96P20	THP-1	19.2±11.4%
TPD-U7BWWQ	Inhibiton_2(200nM)	NLRP3	Q96P20	THP-1	35.3±3.1%
TPD-QCF1E1	Inhibiton_2(200nM)	NLRP3	Q96P20	THP-1	59.2±2.3%
TPD-DF2N5D	Inhibiton_2(200nM)	NLRP3	Q96P20	THP-1	39.1±5.6%
TPD-IU0VYK	Inhibiton_2(200nM)	NLRP3	Q96P20	THP-1	32.7±9.2%
TPD-RDHTMN	Inhibiton_2(200nM)	NLRP3	Q96P20	THP-1	49.2±8.9%
TPD-UVS853	Inhibiton_2(200nM)	NLRP3	Q96P20	THP-1	39.6±8.6%
TPD-NDRQ1S	Inhibiton_2(200nM)	NLRP3	Q96P20	THP-1	19.5±4.1%
TPD-S0FHNY	Inhibiton_2(200nM)	NLRP3	Q96P20	THP-1	67.3±3.3%
TPD-64VJHN	Inhibiton_2(200nM)	NLRP3	Q96P20	THP-1	45.2±10.1%
TPD-ZAE7Z2	Inhibiton_2(200nM)	NLRP3	Q96P20	THP-1	66.6±7.0%
TPD-TCMXXF	Inhibiton_2(200nM)	NLRP3	Q96P20	THP-1	48.5±5.4%
TPD-K7F3BH	Inhibiton_2(200nM)	NLRP3	Q96P20	THP-1	26.5±4.1%
TPD-T5OPGC	Inhibiton_2(200nM)	NLRP3	Q96P20	THP-1	7.9±26.8%
TPD-LISID0	Inhibiton_2(200nM)	NLRP3	Q96P20	THP-1	98.2±2.6%
TPD-1FT2G6	Inhibiton_2(200nM)	NLRP3	Q96P20	THP-1	41.7±6.5%
TPD-L0GDB2	Inhibiton_2(200nM)	NLRP3	Q96P20	THP-1	73.6±13.7%
TPD-VN00OX	100nM Degradation	NLRP3	Q96P20	THP-1	34%
TPD-QCF1E1	100nM Degradation	NLRP3	Q96P20	THP-1	35%
TPD-IU0VYK	100nM Degradation	NLRP3	Q96P20	THP-1	11%
TPD-S0FHNY	100nM Degradation	NLRP3	Q96P20	THP-1	33%
TPD-ZAE7Z2	100nM Degradation	NLRP3	Q96P20	THP-1	17%
TPD-LISID0	100nM Degradation	NLRP3	Q96P20	THP-1	19%
TPD-L0GDB2	100nM Degradation	NLRP3	Q96P20	THP-1	13%
TPD-VN00OX	200nM Degradation	NLRP3	Q96P20	THP-1	27%
TPD-QCF1E1	200nM Degradation	NLRP3	Q96P20	THP-1	22%
TPD-IU0VYK	200nM Degradation	NLRP3	Q96P20	THP-1	19%
TPD-S0FHNY	200nM Degradation	NLRP3	Q96P20	THP-1	ND
TPD-ZAE7Z2	200nM Degradation	NLRP3	Q96P20	THP-1	ND
TPD-LISID0	200nM Degradation	NLRP3	Q96P20	THP-1	23%
TPD-L0GDB2	200nM Degradation	NLRP3	Q96P20	THP-1	49%
TPD-VN00OX	500nM Degradation	NLRP3	Q96P20	THP-1	31%
TPD-QCF1E1	500nM Degradation	NLRP3	Q96P20	THP-1	41%
TPD-IU0VYK	500nM Degradation	NLRP3	Q96P20	THP-1	66%
TPD-S0FHNY	500nM Degradation	NLRP3	Q96P20	THP-1	26%
TPD-ZAE7Z2	500nM Degradation	NLRP3	Q96P20	THP-1	14%
TPD-LISID0	500nM Degradation	NLRP3	Q96P20	THP-1	48%
TPD-L0GDB2	500nM Degradation	NLRP3	Q96P20	THP-1	65%
TPD-2VQG7N	Kd_1	PCSK9	Q8NBP7	.	0.4241μM
TPD-YC2BN5	Kd_1	PCSK9	Q8NBP7	.	1.85μM
TPD-H5686H	Kd_1	PCSK9	Q8NBP7	.	0.9505μM
TPD-J003G6	Kd_1	PCSK9	Q8NBP7	.	1.339μM
TPD-2VQG7N	Kd_2	LC3B	Q9GZQ8	.	9.798μM
TPD-YC2BN5	Kd_2	LC3B	Q9GZQ8	.	9.877μM
TPD-H5686H	Kd_2	LC3B	Q9GZQ8	.	8.477μM
TPD-J003G6	Kd_2	LC3B	Q9GZQ8	.	5.69μM
TPD-QLKGGI	normalized KRAS levels_2(10 μM Compound Concentration)	KRAS	P01116	NCI-H2030	87.50%
TPD-XFJWJ1	normalized KRAS levels_2(10 μM Compound Concentration)	KRAS	P01116	NCI-H2030	48.60%
TPD-93OD2F	normalized KRAS levels_2(10 μM Compound Concentration)	KRAS	P01116	NCI-H2030	65.70%
TPD-G2Q8KL	Normalized BTK levels_3(30 μM Compound Concentration)	BTK	Q06187	NAMALWA	~30.1 %
TPD-K7NHEO	Normalized BTK levels_2(10 μM Compound Concentration)	BTK	Q06187	NAMALWA	48.20%
TPD-ENY4CV	Normalized BTK levels_2(10 μM Compound Concentration)	BTK	Q06187	NAMALWA	66.30%
TPD-CQN0FF	IC50_2	.	.	MCF-7	26.9μM
TPD-CQN0FF	IC50_3	.	.	MDAMB231	23.3μM
TPD-CQN0FF	IC50_4	.	.	A375	11.9μM
TPD-CQN0FF	IC50_5	.	.	B16F10	9.1μM
TPD-CPLM1P	Dmax_1	CDK9 42	P50750	U2932	58.96±6.70%
TPD-ILLLK4	Dmax_1	CDK9 42	P50750	U2932	49.89±4.96%
TPD-CPLM1P	Dmax_2	CDK9 55	P50750	U2932	54.84±5.47%
TPD-ILLLK4	Dmax_2	CDK9 55	P50750	U2932	46.02±5.07%