TPD ID TPD NAME PubChem synonyms SMILES Fomula Lytac_target Target adapter name Target adapter type Target adapter Linker type Lytac_Linker Lysosome-targeting receptors LTR adapter name LTR adapter type LTR adapter Target Symbol Target ID Source TPD-2FKJHL AU2023286835_BF001 . CC(C)(C)CC[C@H](NC(=O)c1ccc(Oc2cccc(C(=O)NCCOCCOCCNc3ccc([N+](=O)[O-])cc3[N+](=O)[O-])c2)nc1)C(=O)O C33H40N6O11 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-6VCCK1 AU2023286835_BF002 . CC(C)(C)CC[C@H](NC(=O)c1ccc(Oc2cccc(C(=O)NCCOCCOCCOCCNc3ccc([N+](=O)[O-])cc3[N+](=O)[O-])c2)nc1)C(=O)O C35H44N6O12 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-35VEV0 AU2023286835_BF003 . CC(C)(C)CC[C@H](NC(=O)c1ccc(Oc2cccc(C(=O)NCCOCCOCCOCCOCCNc3ccc([N+](=O)[O-])cc3[N+](=O)[O-])c2)nc1)C(=O)O C37H48N6O13 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-ECUACK AU2023286835_BF004 . CC(C)(C)CC[C@H](NC(=O)c1ccc(Oc2cccc(OCCOCCOCCOCCOCCOCCNc3ccc([N+](=O)[O-])cc3[N+](=O)[O-])c2)nc1)C(=O)O C38H51N5O14 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-32V6SG AU2023286835_BF005 . CC(C)(C)CC[C@H](NC(=O)c1ccc(Oc2cccc3c(C(=O)NCCCNC(=O)CCOCCOCCOCCNc4ccc([N+](=O)[O-])cc4[N+](=O)[O-])cccc23)nc1)C(=O)O C43H53N7O13 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-ZCBC57 AU2023286835_BF006 . CC(C)(C)CC[C@H](NC(=O)c1ccc(Oc2cccc(C(=O)NCCOCCOCCOCCOCCOCCOCCOCCNc3ccc([N+](=O)[O-])cc3[N+](=O)[O-])c2)nc1)C(=O)O C43H60N6O16 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-P03N3P AU2023286835_BF007 . CC(C)(C)CC[C@H](NC(=O)c1ccc(Oc2cccc(OCCOCCOCCOCCNc3ccc([N+](=O)[O-])cc3[N+](=O)[O-])c2)nc1)C(=O)O C34H43N5O12 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-J5P9GJ AU2023286835_BF008 . CC(C)(C)CC[C@H](NC(=O)c1ccc(Oc2cccc(C(=O)NCCOCCOCCOCCOCCOCCOCCNc3ccc([N+](=O)[O-])cc3[N+](=O)[O-])c2)nc1)C(=O)O C41H56N6O15 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-Y43GDL AU2023286835_BF009 . CC(C)(C)CC[C@H](NC(=O)c1ccc(Oc2cccc3c(C(=O)NCCCNC(=O)CCOCCOCCNc4ccc([N+](=O)[O-])cc4[N+](=O)[O-])cccc23)nc1)C(=O)O C41H49N7O12 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-19QF8H AU2023286835_BF010 . CC(C)(C)CC[C@H](NC(=O)c1ccc(Oc2cccc3c(C(=O)NCCCNC(=O)CCOCCOCCOCCOCCNc4ccc([N+](=O)[O-])cc4[N+](=O)[O-])cccc23)nc1)C(=O)O C45H57N7O14 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-Y3E299 AU2023286835_BF011 . CC(C)(C)CC[C@H](NC(=O)c1ccc(Oc2cccc(C(=O)NCCOCCOCCOCCOCCOCCNc3ccc([N+](=O)[O-])cc3[N+](=O)[O-])c2)nc1)C(=O)O C39H52N6O14 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-NV5WIZ AU2023286835_BF012 . CC(C)(C)CC[C@H](NC(=O)c1ccc(Oc2cccc(OCCOCCOCCOCCOCCOCCOCCOCCNc3ccc([N+](=O)[O-])cc3[N+](=O)[O-])c2)nc1)C(=O)O C42H59N5O16 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-H044TS AU2023286835_BF013 . CC(C)(C)CC[C@H](NC(=O)c1ccc(Oc2cccc(OCCOCCOCCNc3ccc([N+](=O)[O-])cc3[N+](=O)[O-])c2)nc1)C(=O)O C32H39N5O11 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-W2CVQL AU2023286835_BF014 . CC(C)(C)CC[C@H](NC(=O)c1ccc(Oc2cccc(OCCOCCOCCOCCOCCOCCOCCNc3ccc([N+](=O)[O-])cc3[N+](=O)[O-])c2)nc1)C(=O)O C40H55N5O15 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-PCU2W2 AU2023286835_BF015 . CC(C)(C)CC[C@H](NC(=O)c1ccc(Oc2cccc3c(C(=O)NCCCNC(=O)CCOCCNc4ccc([N+](=O)[O-])cc4[N+](=O)[O-])cccc23)nc1)C(=O)O C39H45N7O11 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-TJJW8R AU2023286835_BF016 . CC(C)(C)CC[C@H](NC(=O)c1ccc(Oc2cccc3c(C(=O)NCCCNC(=O)CCNc4ccc([N+](=O)[O-])cc4[N+](=O)[O-])cccc23)nc1)C(=O)O C37H41N7O10 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-VK4WO8 AU2023286835_BF017 . CC(C)(C)CC[C@H](NC(=O)c1ccc(Oc2cccc(OCCOCCOCCOCCOCCOCCOCCOCCNC(=O)CCCC[C@@H]3SC[C@@H]4NC(=O)N[C@@H]43)c2)nc1)C(=O)O C46H71N5O14S . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-1B638C AU2023286835_BF018 . CC(C)(C)CC[C@H](NC(O)c1ccc(Oc2cccc(C(=O)NCCOCCOCCOCCOCCOCCOCCOCCOCCNC(=O)CCCC[C@@H]3SC[C@@H]4NC(=O)N[C@@H]43)c2)nc1)C(=O)O C49H78N6O15S . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-IP9NQU AU2023286835_BF019 . CC(C)(C)CC[C@H](NC(=O)c1ccc(Oc2cccc(OCCOCCOCCOCCOCCOCCOCCNC(O)CCCC[C@@H]3SC[C@@H]4NC(=O)N[C@@H]43)c2)nc1)C(=O)O C44H69N5O13S . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-L54W2O AU2023286835_BF020 . CC(C)(C)CC[C@H](NC(=O)c1ccc(Oc2cccc3c(C(=O)NCCCNC(=O)CCOCCOCCOCCOCCNC(=O)CCCC[C@@H]4SC[C@@H]5NC(=O)N[C@@H]54)cccc23)nc1)C(=O)O C49H69N7O12S . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-MHWYHY AU2023286835_BF021 . CC(C)(C)CC[C@H](NC(=O)c1ccc(Oc2cccc(C(=O)NCCOCCOCCOCCOCCOCCOCCOCCNC(=O)CCCC[C@@H]3SC[C@@H]4NC(=O)N[C@@H]43)c2)nc1)C(=O)O C47H72N6O14S . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-RXPYCI AU2023286835_BF022 . CC(C)(C)CC[C@H](NC(=O)c1ccc(Oc2cccc(OCCOCCOCCNC(=O)CCCC[C@@H]3SC[C@@H]4NC(=O)N[C@@H]43)c2)nc1)C(=O)O C36H51N5O9S . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-61T8A1 AU2023286835_BF023 . CC(C)(C)CC[C@H](NC(=O)c1ccc(Oc2cccc(C(=O)NCCOCCOCCOCCOCCOCCOCCNC(=O)CCCC[C@@H]3SC[C@@H]4NC(=O)N[C@@H]43)c2)nc1)C(=O)O C45H68N6O13S . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-DG2MWI AU2023286835_BF024 . CC(C)(C)CC[C@H](NC(=O)c1ccc(Oc2cccc3cc(C(=O)NCCCNC(=O)CCCC[C@@H]4SC[C@@H]5NC(=O)N[C@@H]54)ccc23)nc1)C(=O)O C38H48N6O7S . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-LH3R81 AU2023286835_BF025 . CC(C)(C)CC[C@H](NC(=O)c1ccc(Oc2cccc(OCCOCCOCCOCCOCCOCCNC(=O)CCCC[C@@H]3SC[C@@H]4NC(=O)N[C@@H]43)c2)nc1)C(=O)O C42H63N5O12S . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-6C1MTU AU2023286835_BF026 . CC(C)(C)CC[C@H](NC(=O)c1ccc(Oc2cccc(OCCOCCOCCOCCOCCOCCOCCOCCOCCNC(=O)CCCC[C@@H]3SC[C@@H]4NC(=O)N[C@@H]43)c2)nc1)C(=O)O C48H75N5O15S . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-CPPM20 AU2023286835_BF027 . CC(C)(C)CC[C@H](NC(=O)c1ccc(Oc2cccc3c(C(=O)NCCCNC(=O)CCCC[C@@H]4SC[C@@H]5NC(=O)N[C@@H]54)cccc23)nc1)C(=O)O C38H48N6O7S . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-8MWIGE AU2023286835_BF028 . CC(C)(C)CC[C@H](NC(=O)c1ccc(Oc2cccc3c(C(=O)NCCCNC(=O)CCOCCOCCOCCOCCOCCNC(=O)CCCC[C@@H]4SC[C@@H]5NC(=O)N[C@@H]54)cccc23)nc1)C(=O)O C51H73N7O13S . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-TNP7IJ AU2023286835_BF029 . COCCOCCOCCOCCOCCOCCNc1ccc([N+](=O)[O-])cc1[N+](=O)[O-] C19H31N3O10 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-XE8D7C AU2023286835_BF030 . CC(C)(C)CC[C@H](NC(=O)c1ccc(Oc2cccc(C(=O)NCCOCCOCCOCCNc3ncc(-c4ccc5c(n4)N(Cc4cccnc4C#N)C(C)(C)C5=O)cn3)c2)nc1)C(=O)O C49H56N10O9 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-WWLKUM AU2023286835_BF031 . C[C@@H]1CN(c2ncc(-c3ccc4c(n3)N(Cc3cccnc3C#N)C(C)(C)C4=O)cn2)CCN1C(=O)COCCOCCOCCOCCNC(=O)c1cccc(Oc2ccc(C(=O)N[C@@H](CCC(C)(C)C)C(=O)O)cn2)c1 C56H67N11O11 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-EQOU54 AU2023286835_BF032 . C[C@@H]1CN(C2=NC=C(c3ccc4c(n3)N(Cc3cccnc3C#N)C(C)(C)C4=O)CN2)CCN1C(=O)COCCOCCOCCOCCNC(=O)c1ccc(Oc2cccc(OCC(=O)N[C@@H](/C=C/C(C)(C)C)C(=O)O)c2)nc1 C57H69N11O12 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-I5P12Q AU2023286835_BF033 . CC(C)(C)CC[C@H](NC(=O)c1ccc(Oc2cccc(C(=O)NCCOCCOCCOCc3ccc(-c4cccc5ccncc45)c(OCCc4ccc(-c5cccc6ccncc56)cc4)c3)c2)nc1)C(=O)O C60H61N5O9 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-O8RNX2 AU2023286835_BF034 . CC(C)(C)CC[C@H](NC(=O)c1ccc(Oc2cccc(C(=O)NCCOCCOCCOCCOCCOCCOCc3ccc(-c4cccc5ccncc45)c(OCCc4ccc(-c5cccc6ccncc56)cc4)c3)c2)nc1)C(=O)O C66H73N5O12 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-H4OO60 AU2023286835_BF035 . CC(C)(C)CC[C@H](NC(=O)c1ccc(Oc2cccc(C(=O)NCCOCCOCCOCCOCc3ccc(-c4cccc5ccncc45)c(OCCc4ccc(-c5cccc6ccncc56)cc4)c3)c2)nc1)C(=O)O C62H65N5O10 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-WBZQRH AU2023286835_BF036 . CC(C)(C)CC[C@H](NC(=O)c1ccc(Oc2cccc(OCC(=O)NCCCCCCOCC(=O)N3CCN(c4ncc(-c5ccc6c(n5)N(Cc5cccnc5C#N)C(C)(C)C6=O)cn4)CC3)c2)nc1)C(=O)O C54H63N11O9 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-M90VUJ AU2023286835_BF037 . CC(C)(C)CC[C@H](NC(=O)c1ccc(Oc2cccc(C(=O)NCCOCCOCCOCCOCCOCc3ccc(-c4cccc5ccncc45)c(OCCc4ccc(-c5cccc6ccncc56)cc4)c3)c2)nc1)C(=O)O C64H69N5O11 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-O05P7R AU2023286835_BF038 . C[C@@H]1CN(c2ncc(-c3ccc4c(n3)N(Cc3cccnc3C#N)C(C)(C)C4=O)cn2)CCN1C(=O)COCCCCCCCCNc1cccc(Oc2ccc(C(=O)N[C@@H](CCC(C)(C)C)C(=O)O)cn2)c1 C55H67N11O7 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-XILTN7 AU2023286835_BF039 . C[C@@H]1CN(c2ncc(-c3ccc4c(n3)N(Cc3cccnc3C#N)C(C)(C)C4=O)cn2)CCN1C(=O)COCCCCCCNc1cccc(Oc2ccc(C(=O)N[C@@H](CCC(C)(C)C)C(=O)O)cn2)c1 C53H63N11O7 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-HOI4SL AU2023286835_BF040 . C[C@@H]1CN(c2ncc(-c3ccc4c(n3)N(Cc3cccnc3C#N)C(C)(C)C4=O)cn2)CCN1C(=O)COCCCCCCCCNC(=O)COc1cccc(Oc2ccc(C(=O)N[C@@H](CCC(C)(C)C)C(=O)O)cn2)c1 C57H69N11O9 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-TGIKJA AU2023286835_BF041 . C[C@@H]1CN(c2ncc(-c3ccc4c(n3)N(Cc3cccnc3C#N)C(C)(C)C4=O)cn2)CCN1C(=O)COCCCCCCCCNC(=O)c1cccc(Oc2ccc(C(=O)N[C@@H](CCC(C)(C)C)C(=O)O)cn2)c1 C56H67N11O8 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-69MVBG AU2023286835_BF042 . C[C@@H]1CN(c2ncc(-c3ccc4c(n3)N(Cc3cccnc3C#N)C(C)(C)C4=O)cn2)CCN1C(=O)CNC(=O)CCCCCCCCCCCNC(O)c1cccc(Oc2ccc(C(=O)N[C@@H](CCC(C)(C)C)C(=O)O)cn2)c1 C60H76N12O8 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-DGORDS AU2023286835_BF043 . C[C@@H]1CN(c2ncc(-c3ccc4c(n3)N(Cc3cccnc3C#N)C(C)(C)C4=O)cn2)CCN1C(=O)CNC(=O)CCCCCCCCCNC(=O)c1cccc(Oc2ccc(C(=O)N[C@@H](CCC(C)(C)C)C(=O)O)cn2)c1 C58H70N12O8 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-OSZFW2 AU2023286835_BF044 . C[C@@H]1CN(c2ccc(-c3ccc4c(n3)N(Cc3cccnc3C#N)C(C)(C)C4=O)cn2)CCN1C(=O)COCCCCCCNC(=O)c1cccc(Oc2ccc(C(=O)N[C@@H](CCC(C)(C)C)C(=O)O)cn2)c1 C55H64N10O8 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-MHQN66 AU2023286835_BF045 . C[C@@H]1CN(c2ncc(-c3ccc4c(n3)N(Cc3cccnc3C#N)C(C)(C)C4=O)cn2)CCN1C(=O)COCCCCNC(=O)c1cccc(Oc2ccc(C(=O)N[C@@H](CCC(C)(C)C)C(=O)O)cn2)c1 C52H59N11O8 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-HECKWP AU2023286835_BF046 . C[C@@H]1CN(c2ncc(-c3ccc4c(n3)N(Cc3cccnc3C#N)C(C)(C)C4=O)cn2)CCN1C(=O)COCCCCNc1cccc(Oc2ccc(C(=O)N[C@@H](CCC(C)(C)C)C(=O)O)cn2)c1 C51H59N11O7 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-WKFIM9 AU2023286835_BF047 . C[C@@H]1CN(c2ncc(-c3ccc4c(n3)N(Cc3cccnc3C#N)C(C)(C)C4=O)cn2)CCN1C(=O)COCCNc1cccc(Oc2ccc(C(=O)N[C@@H](CCC(C)(C)C)C(=O)O)cn2)c1 C49H55N11O7 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-QFBW6S AU2023286835_BF048 . C[C@@H]1CN(c2ncc(-c3ccc4c(n3)N(Cc3cccnc3C#N)C(C)(C)C4=O)cn2)CCN1C(=O)COCCCCNC(=O)COc1cccc(Oc2ccc(C(=O)N[C@@H](CCC(C)(C)C)C(=O)O)cn2)c1 C53H61N11O9 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-247R54 AU2023286835_BF049 . CC(C)(C)CC[C@H](NC(=O)c1ccc(Oc2cccc(C(=O)NCCOCCOCCNc3ncc(-c4ccc5c(n4)N(Cc4cccnc4C#N)C(C)(C)C5=O)cn3)c2)nc1)C(=O)O C47H52N10O8 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-HKMHVF AU2023286835_BF050 . C[C@@H]1CN(c2ncc(-c3ccc4c(n3)N(Cc3cccnc3C#N)C(C)(C)C4=O)cn2)CCN1C(=O)COCCOCCNC(=O)c1ccc(Oc2cccc(OCC(=O)N[C@@H](CCC(C)(C)C)C(=O)O)c2)nc1 C53H61N11O10 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-VI0KBX AU2023286835_BF051 . C[C@@H]1CN(C2=NCC(c3ccc4c(n3)N(Cc3cccnc3C#N)C(C)(C)C4=O)C=N2)CCN1C(=O)COCCOCCNC(=O)c1cccc(Oc2ccc(C(=O)N[C@@H](CCC(C)(C)C)C(=O)O)cn2)c1 C52H61N11O9 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-A4ECSW AU2023286835_BF052 . CC(C)(C)CC[C@H](NC(=O)c1ccc(Oc2cccc(C(=O)NCCOCCOCCOCCOCCOc3ncc(-c4ccc5c(n4)N(Cc4cccnc4C#N)C(C)(C)C5=O)cn3)c2)nc1)C(=O)O C51H59N9O11 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-JY6I5E AU2023286835_BF054 . CC(C)(C)CC[C@H](NC(=O)c1ccc(Oc2cccc(C(=O)NCCOCCOCCOCCOC3=NC=C(c4ccc5c(n4)N(Cc4cccnc4C#N)C(C)(C)C5=O)CN3)c2)nc1)C(=O)O C49H57N9O10 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-GWL0BV AU2023286835_BF056 . C[C@@H]1CN(c2ncc(-c3ccc4c(n3)N(Cc3cccnc3C#N)C(C)(C)C4=O)cn2)CCN1C(=O)COCCOCCOCCNC(=O)c1cccc(Oc2ccc(C(=O)N[C@@H](CCC(C)(C)C)C(=O)O)cn2)c1 C54H63N11O10 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-VD1VQX AU2023286835_BF058 . C[C@@H]1CN(c2ncc(-c3ccc4c(n3)N(Cc3cccnc3C#N)C(C)(C)C4=O)cn2)CCN1C(=O)COCCNC(=O)c1cccc(Oc2ccc(C(=O)N[C@@H](CCC(C)(C)C)C(=O)O)cn2)c1 C50H55N11O8 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-95PH1L AU2023286835_BF059 . CC(C)(C)CC[C@H](NC(=O)c1ccc(Oc2cccc(C(=O)NCCOCCOCCOCCOCCOCCOc3ncc(-c4ccc5c(n4)N(Cc4cccnc4C#N)C(C)(C)C5=O)cn3)c2)nc1)C(=O)O C53H63N9O12 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-KWIFE7 AU2023286835_BF060 . CC(C)(C)CC[C@H](NC(=O)c1ccc(Oc2cccc(C(=O)NCCOCCNc3ncc(-c4ccc5c(n4)N(Cc4cccnc4C#N)C(C)(C)C5=O)cn3)c2)nc1)C(=O)O C45H48N10O7 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-5TQLG1 AU2023286835_BF064 . C[C@@H]1CN(c2ncc(-c3ccc4c(n3)N(Cc3cccnc3C#N)C(C)(C)C4=O)cn2)CCN1C(=O)COCCNC(=O)COc1cccc(Oc2ccc(C(=O)N[C@@H](CCC(C)(C)C)C(=O)O)cn2)c1 C51H57N11O9 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-PAQL7J AU2023286835_BF066 . CC(C)(C)CC[C@H](NC(=O)c1ccc(Oc2cccc(C(=O)NCCOCCOc3ncc(-c4ccc5c(n4)N(Cc4cccnc4C#N)C(C)(C)C5=O)cn3)c2)nc1)C(=O)O C45H47N9O8 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-PMPHX5 AU2023286835_BF067 . CC(C)(C)CC[C@H](NC(=O)c1ccc(Oc2cccc(C(=O)NCCOCCOCCOCCOCCOCCNc3ncc(-c4ccc5c(n4)N(Cc4cccnc4C#N)C(C)(C)C5=O)cn3)c2)nc1)C(=O)O C53H64N10O11 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-IRYJQW AU2023286835_BF068 . CC(C)(C)CC[C@H](NC(=O)COc1cccc(Oc2ccc(C(=O)NCCOCCOCCOCCOCCOCCNc3ncc(-c4ccc5c(n4)N(Cc4cccnc4C#N)C(C)(C)C5=O)cn3)cn2)c1)C(=O)O C54H66N10O12 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-QLGN9K AU2023286835_BF070 . CC(C)(C)CC[C@H](NC(=O)c1ccc(Oc2cccc(C(=O)NCCOCCOCCOc3ncc(-c4ccc5c(n4)N(Cc4cccnc4C#N)C(C)(C)C5=O)cn3)c2)nc1)C(=O)O C47H51N9O9 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-JNK8OD AU2023286835_BF071 . CC(C)(C)CC[C@H](NC(=O)COc1cccc(Oc2ccc(C(=O)NCCOCCOCCOCCOCCNc3ncc(-c4ccc5c(n4)N(Cc4cccnc4C#N)C(C)(C)C5=O)cn3)cn2)c1)C(=O)O C52H62N10O11 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-7PGQFA AU2023286835_BF072 . CC(C)(C)CC[C@H](NC(=O)COc1cccc(Oc2ccc(C(=O)NCCOCCNc3ncc(-c4ccc5c(n4)N(Cc4cccnc4C#N)C(C)(C)C5=O)cn3)cn2)c1)C(=O)O C46H50N10O8 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-V7GBBP AU2023286835_BF073 . CC(C)(C)CC[C@H](NC(=O)COc1cccc(Oc2ccc(C(=O)NCCOCCOCCOCCOCCOc3ccc(-c4ccc5c(n4)N(Cc4cccnc4C#N)C(C)(C)C5=O)cn3)cn2)c1)C(=O)O C53H62N8O12 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-101IGH AU2023286835_BF074 . CC(C)(C)CC[C@H](NC(=O)COc1cccc(Oc2ccc(C(=O)NCCOCCOCCOc3ncc(-c4ccc5c(n4)N(Cc4cccnc4C#N)C(C)(C)C5=O)cn3)cn2)c1)C(=O)O C48H53N9O10 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-6PNR78 AU2023286835_BF075 . CC(C)(C)CC[C@H](NC(=O)COc1cccc(Oc2ccc(C(=O)NCCOCCOCCOCCOCc3cn(CCCCCOc4ncc(-c5ccc6c(n5)N(Cc5cccnc5C#N)C(C)(C)C6=O)cn4)nn3)cn2)c1)C(=O)O C58H70N12O12 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-RKH4SJ AU2023286835_BF076 . Cc1nc2cc(F)c(-c3cnc(OCCCCCn4cc(COCCOCCOCCOCCNC(=O)c5ccc(Oc6cccc(OCC(=O)N[C@@H](CCC(C)(C)C)C(=O)O)c6)nc5)nn4)nc3)nc2c(N[C@H](C)c2cc(C#N)ccc2F)c1Cl C60H69ClF2N12O11 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-9QOLU9 AU2023286835_BF077 . Cc1nc2cc(F)c(-c3cnc(OCCCCCn4cc(COCCOCCOCCOCCOCCOCCNC(=O)c5ccc(Oc6cccc(OCC(=O)N[C@@H](CCC(C)(C)C)C(=O)O)c6)nc5)nn4)nc3)nc2c(N[C@H](C)c2cc(C#N)ccc2F)c1Cl C64H77ClF2N12O13 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-2XWUF1 AU2023286835_BF078 . Cc1nc2cc(F)c(-c3cnc(OCCCCCn4cc(COCCOCCNC(=O)c5ccc(Oc6cccc(OCC(=O)N[C@@H](CCC(C)(C)C)C(=O)O)c6)nc5)nn4)nc3)nc2c(N[C@H](C)c2cc(C#N)ccc2F)c1Cl C56H61ClF2N12O9 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-UN8XN5 AU2023286835_BF079 . Cc1nc2cc(F)c(-c3cnc(OCCOCCOCCOCCOCCOCCOCCNC(=O)c4ccc(Oc5cccc(OCC(=O)N[C@@H](CCC(C)(C)C)C(=O)O)c5)nc4)nc3)nc2c(N[C@H](C)c2cc(C#N)ccc2F)c1Cl C58H68ClF2N9O13 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-DMF9NX AU2023286835_BF080 . Cc1cc(-c2ccc(OCC(=O)NCCOCCOCc3cn(CCCCCOc4ncc(-c5nc6c(N[C@@H](C)c7cc(C#N)ccc7F)c(Cl)c(C)nc6cc5F)cn4)nn3)cc2)cc(NC(=O)c2ccc(C(F)(F)F)cc2C(=O)O)n1 C57H52ClF5N12O8 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-IK80I8 AU2023286835_BF081 . C[C@@H]1CN(c2ncc(-c3ccc4c(n3)N(Cc3cccnc3C#N)C(C)(C)C4=O)cn2)CCN1C(=O)CNC(=O)CCCCCCCCCCn1cc(-c2cccc(Oc3ccc(C(=O)N[C@@H](CCC(C)(C)C)C(=O)O)cn3)c2)nn1 C60H72N14O7 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-NE0M31 AU2023286835_BF082 . C[C@@H]1CN(c2ncc(-c3ccc4c(n3)N(Cc3cccnc3C#N)C(C)(C)C4=O)cn2)CCN1C(=O)CNC(=O)COCCOCCOCCOCCOc1cccc(OC2=NCC(C(=O)N[C@@H](CCC(C)(C)C)C(=O)O)C=C2)c1 C57H71N11O12 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-TFXVGA AU2023286835_BF083 . Cc1nc2cc(F)c(-c3cnc(OCCCCCn4cc(COCCOCCNC(=O)COc5cccc(Oc6ccc(C(=O)N[C@@H](CCC(C)(C)C)C(=O)O)cn6)c5)nn4)nc3)nc2c(N[C@H](C)c2cc(C#N)ccc2F)c1Cl C56H61ClF2N12O9 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-MRHKXN AU2023286835_BF084 . Cc1nc2ccc(C3=CNC(OCCCCCn4cc(COCCOCCOCCOCCNC(=O)COc5cccc(Oc6ccc(C(=O)NC(CCC(C)(C)C)C(=O)O)cn6)c5)nn4)NC3)nc2c(N[C@H](C)c2cc(C#N)ccc2F)c1Cl C60H74ClFN12O11 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-NR4708 AU2023286835_BF085 . Cc1nc2cc(F)c(-c3cnc(OCCOCCOCCOCCOCCOCCOCCNC(=O)COc4cccc(Oc5ccc(C(=O)N[C@@H](CCC(C)(C)C)C(=O)O)cn5)c4)nc3)nc2c(N[C@H](C)c2cc(C#N)ccc2F)c1Cl C58H68ClF2N9O13 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-RPTWP2 AU2023286835_BF086 . Cc1nc2cc(F)c(-c3cnc(OCCCCCn4cc(COCCOCCOCCOCCOCCOCCNC(=O)COc5cccc(Oc6ccc(C(=O)N[C@@H](CCCCC(C)(C)C)C(=O)O)cn6)c5)nn4)nc3)nc2c(N[C@H](C)c2cc(C#N)ccc2F)c1C C67H84F2N12O13 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-0TH3ER AU2023286835_BF087 . Cc1nc2cc(F)c(-c3cnc(OCCCCCn4cc(COCCOCCOCCOCCOCCOCCNC(=O)COc5cccc(Oc6ccc(C(=O)N[C@@H](CCC(C)(C)C)C(=O)O)cn6)c5)nn4)nc3)nc2c(N[C@H](C)c2cc(C#N)ccc2F)c1Cl C64H77ClF2N12O13 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-97WCBI AU2023286835_BF088 . Cc1nc2cc(F)c(C3=CNC(OCCOCCn4cc(COCC(=O)N5CC(OCCNC(=O)COc6cccc(Oc7ccc(C(=O)N[C@@H](CCC(C)(C)C)C(=O)O)cn7)c6)C5)nn4)N=C3)nc2c(N[C@H](C)c2cc(C#N)ccc2F)c1Cl C58H64ClF2N13O11 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-GOXY46 AU2023286835_BF089 . Cc1nc2cc(F)c(-c3cnc(OCCN4CC(n5cc(COCC(=O)N6CC(OCCNC(=O)COc7cccc(Oc8ccc(C(=O)N[C@@H](CCC(C)(C)C)C(=O)O)cn8)c7)C6)nn5)C4)nc3)nc2c(N[C@H](C)c2cc(C#N)ccc2F)c1Cl C59H63ClF2N14O10 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-TEI5DO AU2023286835_BF090 . Cc1nc2cc(F)c(-c3cnc(OCCN4CCC(n5cc(COCC(=O)N6CCC(OCCNC(=O)COc7cccc(Oc8ccc(C(=O)N[C@@H](CCC(C)(C)C)C(=O)O)cn8)c7)CC6)nn5)CC4)nc3)nc2c(N[C@H](C)c2cc(C#N)ccc2F)c1Cl C63H71ClF2N14O10 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-FG2FUJ AU2023286835_BF092 . Cc1nc2cc(F)c(-c3cnc(OCCN4CC(n5cc(COCCN6CC(OCCNC(=O)COc7cccc(Oc8ccc(C(=O)N[C@@H](CCC(C)(C)C)C(=O)O)cn8)c7)C6)nn5)C4)nc3)nc2c(N[C@H](C)c2cc(C#N)ccc2F)c1Cl C59H65ClF2N14O9 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-QQDT60 AU2023286835_BF093 . Cc1nc2cc(F)c(-c3cnc(OCCOCCn4cc(COCCN5CC(OCCNC(=O)COc6cccc(Oc7ccc(C(=O)N[C@@H](CCC(C)(C)C)C(=O)O)cn7)c6)C5)nn4)nc3)nc2c(N[C@H](C)c2cc(C#N)ccc2F)c1Cl C58H64ClF2N13O10 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-A5CQPR AU2023286835_BF094 . Cc1nc2cc(F)c(-c3cnc(N4CCN(C(=O)Cn5cc(COCCOCCOCC(=O)N6CCC(Oc7cccc(Oc8ccc(C(O)N[C@@H](CCC(C)(C)C)C(=O)O)cn8)c7)CC6)nn5)[C@H](C)C4)nc3)nc2c(N[C@H](C)c2cc(C#N)ccc2F)c1Cl C63H73ClF2N14O10 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-GY0KNW AU2023286835_BF096 . Cc1cc2nc(C)c(Cl)c(N[C@H](C)c3cc(C#N)ccc3F)c2nc1-c1cnc(N2CCN(C(=O)Cn3cc(COCCOCCOCC(=O)N4CCC(Oc5ccc(Oc6cccc(OCC(=O)NC(CCC(C)(C)C)C(=O)O)c6)nc5)CC4)nn3)[C@H](C)C2)nc1 C65H76ClFN14O11 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-X7LVDT AU2023286835_BF097 . C[C@@H]1CN(c2ncc(-c3ccc4c(n3)N(Cc3cccnc3C#N)C(C)(C)C4=O)cn2)CCN1C(=O)CNC(=O)CCOCCOCCOCCNC(=O)c1cccc(Oc2ccc(C(=O)N[C@@H](CCC(C)(C)C)C(=O)O)cn2)c1 C57H68N12O11 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-JEN5W4 AU2023286835_BF098 . C[C@@H]1CN(c2ncc(-c3ccc4c(n3)N(Cc3cccnc3C#N)C(C)(C)C4=O)cn2)CCN1C(=O)Cn1cc(COCCOCCOCCOCCOCCOc2cccc(Oc3ccc(C(=O)N[C@@H](CCC(C)(C)C)C(=O)O)cn3)c2)nn1 C60H73N13O12 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-F1KEIU AU2023286835_BF099 . C[C@@H]1CN(c2ncc(-c3ccc4c(n3)N(Cc3cccnc3C#N)C(C)(C)C4=O)cn2)CCN1C(=O)CNC(=O)COCCOCCOCCOCCNC(=O)c1cccc(Oc2ccc(C(=O)N[C@@H](CCC(C)(C)C)C(=O)O)cn2)c1 C58H70N12O12 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-PZAEO9 AU2023286835_BF100 . C[C@@H]1CN(c2ncc(-c3ccc4c(n3)N(Cc3cccnc3C#N)C(C)(C)C4=O)cn2)CCN1C(=O)CNC(=O)CCCCCOCCOCCNC(=O)c1cccc(Oc2ccc(C(=O)N[C@@H](CCC(C)(C)C)C(=O)O)cn2)c1 C58H70N12O10 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-EMYPFD AU2023286835_BF101 . C[C@@H]1CN(c2ncc(-c3ccc4c(n3)N(Cc3cccnc3C#N)C(C)(C)C4=O)cn2)CCN1C(=O)Cn1cc(COCCOCCOCCOCCOc2cccc(Oc3ccc(C(=O)N[C@@H](CCC(C)(C)C)C(=O)O)cn3)c2)nn1 C58H69N13O11 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-2VOJOZ AU2023286835_BF102 . C[C@@H]1CN(c2ncc(-c3ccc4c(n3)N(Cc3cccnc3C#N)C(C)(C)C4=O)cn2)CCN1C(=O)CNC(=O)COCCOCCOCCOCCOCCOc1cccc(Oc2ccc(C(=O)N[C@@H](CCC(C)(C)C)C(=O)O)cn2)c1 C59H73N11O13 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-IKONGU AU2023286835_BF103 . C[C@@H]1CN(c2ncc(-c3ccc4c(n3)N(Cc3cccnc3C#N)C(C)(C)C4=O)cn2)CCN1C(=O)Cc1cn(CCCCCCCCCCNC(=O)c2cccc(Oc3ccc(C(=O)N[C@@H](CCC(C)(C)C)C(=O)O)cn3)c2)nn1 C60H72N14O7 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-8SRTK1 AU2023286835_BF104 . C[C@@H]1CN(c2ncc(-c3ccc4c(n3)N(Cc3cccnc3C#N)C(C)(C)C4=O)cn2)CCN1C(=O)Cc1cn(CCCCCCCCCn2cc(-c3cccc(Oc4ccc(C(=O)N[C@@H](CCC(C)(C)C)C(=O)O)cn4)c3)nn2)nn1 C60H70N16O6 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-RH9H8E AU2023286835_BF105 . C[C@@H]1CN(c2ncc(-c3ccc4c(n3)N(Cc3cccnc3C#N)C(C)(C)C4=O)cn2)CCN1C(=O)CNC(=O)CCOCCOCCCCCNC(=O)c1cccc(Oc2ccc(C(=O)N[C@@H](CCC(C)(C)C)C(=O)O)cn2)c1 C58H70N12O10 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-25G3QJ AU2023286835_BF106 . C[C@@H]1CN(c2ncc(-c3ccc4c(n3)N(Cc3ccccc3C#N)C(C)(C)C4=O)cn2)CCN1C(=O)CNC(=O)COCCOCCCCCCNC(=O)c1cccc(Oc2ccc(C(=O)N[C@@H](CCC(C)(C)C)C(=O)O)cn2)c1 C59H71N11O10 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-X1FA1V AU2023286835_BF107 . C[C@@H]1CN(c2ncc(-c3ccc4c(n3)N(Cc3cccnc3C#N)C(C)(C)C4=O)cn2)CCN1C(=O)CNC(=O)CCCCOCCOCCCNC(=O)c1cccc(Oc2ccc(C(=O)N[C@@H](CCC(C)(C)C)C(=O)O)cn2)c1 C58H70N12O10 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-8IOBJN AU2023286835_BF108 . C[C@@H]1CN(c2ncc(-c3ccc4c(n3)N(Cc3cccnc3C#N)C(C)(C)C4=O)cn2)CCN1C(=O)CNC(=O)CCCCCCCCn1cc(CCc2cccc(Oc3ccc(C(=O)N[C@@H](CCC(C)(C)C)C(=O)O)cn3)c2)nn1 C60H72N14O7 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-DTANN2 AU2023286835_BF110 . C[C@@H]1CN(c2ncc(-c3ccc4c(n3)N(Cc3cccnc3C#N)C(C)(C)C4=O)cn2)CCN1C(=O)Cn1cc(CN2CCN(C(=O)COCCn3cc(-c4cccc(Oc5ccc(C(=O)N[C@@H](CCC(C)(C)C)C(=O)O)cn5)c4)nn3)CC2)nn1 C60H68N18O8 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-TWPWNI AU2023286835_BF111 . C[C@@H]1CN(c2ncc(-c3ccc4c(n3)N(Cc3cccnc3C#N)C(C)(C)C4=O)cn2)CCN1C(=O)Cn1cc(COCCOCCOCC(=O)N2CC(Oc3cccc(Oc4ccc(C(=O)N[C@@H](CCC(C)(C)C)C(=O)O)cn4)c3)C2)nn1 C59H68N14O11 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-OI6YT3 AU2023286835_BF112 . C[C@@H]1CN(c2ncc(-c3ccc4c(n3)N(Cc3cccnc3C#N)C(C)(C)C4=O)cn2)CCN1C(=O)Cn1cc(COCCOCCOCC(=O)N2CCC(Oc3cccc(Oc4ccc(C(=O)N[C@@H](CCC(C)(C)C)C(=O)O)cn4)c3)CC2)nn1 C61H72N14O11 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-M81BI5 AU2023286835_BF113 . C=O.C[C@@H]1CN(c2ncc(-c3ccc4c(n3)N(Cc3cccnc3C#N)C(C)(C)C4=O)cn2)CCN1C(=O)Cn1cc(COCCOCCN2CCN(CCOCCOc3cccc(Oc4ccc(C(=O)N[C@H](CO)CCC(C)(C)C)cn4)c3)CC2)nn1 C63H81N15O10 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-8V42YD AU2023286835_BF114 . C[C@@H]1CN(c2ncc(-c3ccc4c(n3)N(Cc3cccnc3C#N)C(C)(C)C4=O)cn2)CCN1C(=O)Cn1cc(COCCOCCOC2CN(CCOCCOc3cccc(Oc4ccc(C(=O)N[C@@H](CCC(C)(C)C)C(=O)O)cn4)c3)C2)nn1 C61H74N14O11 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-TFA9WZ AU2023286835_BF115 . C[C@@H]1CN(c2ncc(-c3ccc4c(n3)N(Cc3cccnc3C#N)C(C)(C)C4=O)cn2)CCN1C(O)Cn1cc(COCCN2CC(OCCOCCOCCOc3cccc(Oc4ccc(C(=O)N[C@@H](CCC(C)(C)C)C(=O)O)cn4)c3)C2)nn1 C61H76N14O11 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-E9VMEL AU2023286835_BF116 . C[C@@H]1CN(c2ncc(-c3ccc4c(n3)N(Cc3cccnc3C#N)C(C)(C)C4=O)cn2)CCN1C(=O)COCCOCCOCCNC(=O)COc1cccc(Oc2ccc(C(=O)N[C@@H](CCC(C)(C)C)C(=O)O)cn2)c1 C55H65N11O11 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-LAM27X AU2023286835_BF117 . C[C@@H]1CN(c2ncc(-c3ccc4c(n3)N(Cc3cccnc3C#N)C(C)(C)C4=O)cn2)CCN1C(=O)COCCOCCOCCOCCNC(=O)COc1cccc(Oc2ccc(C(=O)N[C@@H](CCC(C)(C)C)C(=O)O)cn2)c1 C57H69N11O12 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-ZJ31B3 AU2023286835_BF118 . C[C@@H]1CN(c2ncc(-c3ccc4c(n3)N(Cc3cccnc3C#N)C(C)(C)C4=O)cn2)CCN1C(=O)COCCOCCNC(=O)COc1cccc(Oc2ccc(C(=O)N[C@@H](CCC(C)(C)C)C(=O)O)cn2)c1 C53H61N11O10 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-2XZRVZ AU2023286835_BF119 . C[C@@H]1CN(c2ncc(-c3ccc4c(n3)N(CC3=C(C#N)N=C=C=C3)C(C)(C)C4=O)cn2)CCN1C(=O)Cn1cc(COCCOCCCNC(=O)N2CC(Oc3cccc(Oc4ccc(C(=O)N[C@@H](CCC(C)(C)C)C(=O)O)cn4)c3)C2)nn1 C59H67N15O10 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-EEOLWH AU2023286835_BF120 . C[C@@H]1CN(c2ncc(-c3ccc4c(n3)N(Cc3cccnc3C#N)C(C)(C)C4=O)cn2)CCN1C(=O)CNC(=O)CCCN1CC(OCCn2cc(-c3cccc(Oc4ccc(C(=O)N[C@@H](CCC(C)(C)C)C(=O)O)cn4)c3)nn2)C1 C58H67N15O8 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-P4UX5T AU2023286835_BF121 . C[C@@H]1CN(c2ncc(-c3ccc4c(n3)N(Cc3cccnc3C#N)C(C)(C)C4=O)cn2)CCN1C(=O)Cn1cc(COCCCCOCCS(=O)(=O)N2CC(Oc3cccc(Oc4ccc(C(=O)N[C@@H](CCC(C)(C)C)C(=O)O)cn4)c3)C2)nn1 C59H70N14O11S . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-GZ7315 AU2023286835_BF122 . C[C@@H]1CN(c2ncc(-c3ccc4c(n3)N(Cc3cccnc3C#N)C(C)(C)C4=O)cn2)CCN1C(=O)Cn1cc(COCCOCC(=O)N2CCC(Oc3cccc(Oc4ccc(C(=O)N[C@@H](CCC(C)(C)C)C(=O)O)cn4)c3)CC2)nn1 C59H68N14O10 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-MOYE41 AU2023286835_BF123 . C[C@@H]1CN(c2ncc(-c3ccc4c(n3)N(Cc3cccnc3C#N)C(C)(C)C4=O)cn2)CCN1C(=O)Cn1cc(COCCOCCOC(=O)N2CCC(Oc3cccc(Oc4ccc(C(=O)N[C@@H](CCC(C)(C)C)C(=O)O)cn4)c3)CC2)nn1 C60H70N14O11 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-NUPMTR AU2023286835_BF124 . C[C@@H]1CN(c2ncc(-c3ccc4c(n3)N(Cc3cccnc3C#N)C(C)(C)C4=O)cn2)CCN1C(=O)Cn1cc(COC2CCN(C(=O)CCCC(=O)N3CCC(Oc4cccc(Oc5ccc(C(=O)N[C@@H](CCC(C)(C)C)C(=O)O)cn5)c4)CC3)C2)nn1 C64H75N15O10 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-VUFTG4 AU2023286835_BF125 . C[C@@H]1CN(c2ncc(-c3ccc4c(n3)N(Cc3cccnc3C#N)C(C)(C)C4=O)cn2)CCN1C(=O)Cn1cc(COCC(=O)N2CCC(OCC(=O)N3CCC(Oc4cccc(Oc5ccc(C(=O)N[C@@H](CCC(C)(C)C)C(=O)O)cn5)c4)CC3)C2)nn1 C63H73N15O11 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-W1XS5Z AU2023286835_BF126 . C[C@@H]1CN(c2ncc(-c3ccc4c(n3)N(Cc3cccnc3C#N)C(C)(C)C4=O)cn2)CCN1C(=O)Cn1cc(COCCOCCCS(=O)(=O)N[C@H]2C[C@@H](Oc3cccc(OC4C=CC(C(=O)N[C@@H](CCC(C)(C)C)C(=O)O)=CN4)c3)C2)nn1 C59H72N14O11S . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-A46X6O AU2023286835_BF127 . C[C@@H]1CN(c2ncc(-c3ccc4c(n3)N(Cc3cccnc3C#N)C(C)(C)C4=O)cn2)CCN1C(=O)Cn1cc(COCCOCCCS(=O)(=O)NC2CC(Oc3cccc(Oc4ccc(C(=O)N[C@@H](CCC(C)(C)C)C(=O)O)cn4)c3)C2)nn1 C59H70N14O11S . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-16U0QF AU2023286835_BF128 . C[C@@H]1CN(c2ncc(-c3ccc4c(n3)N(Cc3cccnc3)C(C)(C)C4=O)cn2)CCN1C(=O)Cn1cc(COCCC(=O)N2CCC(Oc3cccc(Oc4ccc(C(=O)N[C@@H](CCC(C)(C)C)C(=O)O)cn4)c3)CC2)nn1 C57H67N13O9 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-8W4CMH AU2023286835_BF129 . C[C@@H]1CN(c2ncc(-c3ccc4c(n3)N(Cc3cccnc3C#N)C(C)(C)C4=O)cn2)CCN1C(=O)Cn1cc(COC2CCN(C(=O)COCC(=O)N3CCC(Oc4cccc(Oc5ccc(C(=O)N[C@@H](CCC(C)(C)C)C(=O)O)cn5)c4)CC3)C2)nn1 C63H73N15O11 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-PU02GX AU2023286835_BF130 . C[C@@H]1CN(c2ncc(-c3ccc4c(n3)N(Cc3cccnc3C#N)C(C)(C)C4=O)cn2)CCN1C(=O)Cn1cc(COCCCC(=O)N2CCC(C(=O)N3CCC(Oc4cccc(Oc5ccc(C(=O)N[C@@H](CCC(C)(C)C)C(=O)O)cn5)c4)CC3)C2)nn1 C64H75N15O10 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-4Y108M AU2023286835_BF131 . C[C@@H]1CN(c2ncc(C3=CC=C4C(=O)C(C)(C)N(Cc5cccnc5C#N)C4N3)cn2)CCN1C(=O)Cn1cc(COCCOCCOCC(=O)N2CCC(Oc3ccc(Oc4cccc(OCC(=O)N[C@@H](CCC(C)(C)C)C(=O)O)c4)nc3)CC2)nn1 C62H76N14O12 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-4WZHYM AU2023286835_BF132 . CC(C)(C)CC[C@H](NC(=O)COc1cccc(OC2C=CC(OC3CCN(C(=O)COCCOCc4cn(CC(=O)N5CCN(c6ncc(-c7ccc8c(n7)N(Cc7cccnc7C#N)C(C)(C)C8=O)cn6)CC5)nn4)CC3)=CN2)c1)C(=O)O C59H70N14O11 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-IZLD3S AU2023286835_BF133 . C[C@@H]1CN(c2ncc(-c3ccc4c(n3)N(c3cccnc3C#N)C(C)(C)C4=O)cn2)CCN1C(=O)Cn1cc(COCCOCCC(O)N2CCC(Oc3ccc(Oc4cccc(OCC(=O)N[C@@H](CCC(C)(C)C)C(=O)O)c4)nc3)CC2)nn1 C60H72N14O11 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-ZWI19S AU2023286835_BF134 . CC(C)(C)CC[C@H](NC(=O)c1ccc(Oc2cccc(OCC(=O)NCCOCCOCCOCCOCCNc3ncc(-c4ccc5c(n4)N(Cc4cccnc4C#N)C(C)(C)C5=O)cn3)c2)nc1)C(=O)O C52H62N10O11 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-95SD74 AU2023286835_BF135 . CC(C)(C)CC[C@H](NC(=O)c1ccc(Oc2cccc(OCC(=O)NCCOCCOCCOCCOCCOCCNc3ncc(-c4ccc5c(n4)N(Cc4cccnc4C#N)C(C)(C)C5=O)cn3)c2)cc1)C(=O)O C55H67N9O12 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-SOA2EF AU2023286835_BF136 . CC(C)(C)CC[C@H](NC(=O)c1ccc(Oc2cccc(OCC(=O)NCCOCCNc3ncc(-c4ccc5c(n4)N(Cc4cccnc4C#N)C(C)(C)C5=O)cn3)c2)nc1)C(=O)O C46H50N10O8 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-J90B98 AU2023286835_BF137 . CC(C)(C)CC[C@H](NC(=O)c1ccc(Oc2cccc(OCC(=O)NCCOCCOCCOCCNc3ncc(-c4ccc5c(n4)N(Cc4cccnc4C#N)C(C)(C)C5=O)cn3)c2)nc1)C(=O)O C50H58N10O10 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-ANZBVV AU2023286835_BF138 . CC(C)(C)CC[C@H](NC(=O)c1ccc(Oc2cccc(OCC(=O)NCCOCCOCCNc3ncc(-c4ccc5c(n4)N(Cc4cccnc4C#N)C(C)(C)C5=O)cn3)c2)nc1)C(=O)O C48H54N10O9 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-GXJLQE AU2023286835_BF139 . CC(C)(C)CC[C@H](NC(=O)c1ccc(Oc2cccc(OCC(=O)NCCOCCOCCOCCOc3ncc(-c4ccc5c(n4)N(Cc4cccnc4C#N)C(C)(C)C5=O)cn3)c2)nc1)C(=O)O C50H57N9O11 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-Q47OVY AU2023286835_BF140 . CC(C)(C)CC[C@H](NC(=O)c1ccc(Oc2cccc(OCC(=O)NCCOCCOCCOCCOCCOc3ncc(-c4ccc5c(n4)N(Cc4cccnc4C#N)C(C)(C)C5=O)cn3)c2)nc1)C(=O)O C52H61N9O12 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-PTWF7C AU2023286835_BF141 . CC(C)(C)CC[C@H](NC(=O)c1ccc(Oc2cccc(OCC(=O)NCCOCCOc3ncc(-c4ccc5c(n4)N(Cc4cccnc4C#N)C(C)(C)C5=O)cn3)c2)nc1)C(=O)O C46H49N9O9 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-8YTENG AU2023286835_BF142 . CC(C)(C)CC[C@H](NC(=O)c1ccc(Oc2cccc(OCC(=O)NCCOCCOCCOc3ncc(-c4ccc5c(n4)N(Cc4cccnc4C#N)C(C)(C)C5=O)cn3)c2)nc1)C(=O)O C48H53N9O10 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-PU5HX7 AU2023286835_BF143 . CC(C)(C)CC[C@H](NC(=O)c1ccc(Oc2cccc(OCC(=O)NCCOCCOCCOCCOCCOCCOc3ncc(-c4ccc5c(n4)N(Cc4cccnc4C#N)C(C)(C)C5=O)cn3)c2)nc1)C(=O)O C54H65N9O13 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-WQSRTN AU2023286835_BF144 . CC(C)(C)CC[C@H](NC(=O)c1ccc(Oc2cccc(OCC(=O)NCCOCCOCCOCCOCC3CN(CCCCCOc4ncc(-c5ccc6c(c5)N(Cc5cccnc5C#N)C(C)(C)C6=O)cn4)N=N3)c2)nc1)C(=O)O C59H73N11O12 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-UBTUDI AU2023286835_BF145 . Cc1cc(-c2ccc(C(=O)NCCOCCOCCOCCOCC(=O)N3CCN(c4ncc(-c5ccc6c(n5)N(Cc5cccnc5C#N)C(C)(C)C6=O)cn4)C[C@H]3C)cc2)cc(NC(=O)c2ccc(C(F)(F)F)cc2C(=O)O)n1 C57H58F3N11O10 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-2QBOXX AU2023286835_BF146 . Cc1cc(-c2ccc(C(=O)NCCCCCCCCCCCC(=O)NCC(=O)N3CCN(c4ncc(-c5ccc6c(n5)N(Cc5cccnc5C#N)C(C)(C)C6=O)cn4)C[C@H]3C)cc2)cc(NC(=O)c2ccc(C(F)(F)F)cc2C(=O)O)n1 C61H65F3N12O7 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-EN6J9Q AU2023286835_BF147 . C=C(/C=C\C(=C/N)CN[C@@H](CCC(C)(C)C)C(=O)O)Oc1cccc(OCC(=O)NCCOCCOCCOCCOCCOCCOCc2cn(CCCCCOc3ncc(-c4nc5c(N[C@H](C)c6cccc(C#N)c6)c(Cl)c(C)nc5cc4F)cn3)nn2)c1 C65H84ClFN12O12 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-1Z0C8N AU2023286835_BF148 . Cc1nc2cc(F)c(-c3cnc(OCCCCCn4cc(COCCOCCOCCOCCOCCOCCOc5cccc(CN[C@@H](CCC(C)(C)C)C(=O)O)c5)nn4)nc3)nc2c(N[C@H](C)c2cc(C#N)ccc2F)c1Cl C57H73ClF2N10O10 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-TGKH4R AU2023286835_BF149 . CC.Cc1nc2cc(F)c(-c3cnc(OCCCCCn4cc(COCCOCCOCCOCCOCCOCCOCC(=O)N[C@@H](Cc5ccccc5)C(=O)N[C@@H](CCC(C)(C)C)C(=O)O)nn4)nc3)nc2c(N[C@H](C)c2cc(C#N)ccc2F)c1Cl C63H84ClF2N11O12 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-YM56TF AU2023286835_BF91 . Cc1nc2cc(F)c(-c3cnc(OCC(=O)N4CC(n5cc(COCCN6CC(OCCNC(=O)COc7cccc(Oc8ccc(C(=O)N[C@@H](CCC(C)(C)C)C(=O)O)cn8)c7)C6)nn5)C4)nc3)nc2c(N[C@H](C)c2cc(C#N)ccc2F)c1Cl C59H63ClF2N14O10 . . . . . . . . . . TNFA;PCSK9;SORT1 P01375/Q8NBP7/Q99523 AU2023286835 TPD-B23WDK Covalent Lytac . . . Programmed cell death 1 ligand 1 (PD-L1) PD-L1 binding region DNA "[DBCO]-TTT-ACGGGCCACATCAACTCATTGATAGACAATGC GTCCACTGCCCGT" DNA TTT&TTTTTT&TTTTTTTTT Cy5-M6PR Cy5-M6PR binding region DNA [Cy5]GGGCGCGTAGATGACGAGCAGTCCTAACATCGTTTAGGAC PD-L1 Q9NZQ7 10.1021/jacs.3c03899 TPD-0M4J0K GalNAc-LYTAC1 . . . Receptor tyrosine-protein kinase erbB-2 (HER2) pertuzumab antibody . . . ASGPR tri-GalNAc-DBCO molecular CC(=O)NC1C(OCCCCC(=O)NCCCNC(=O)CCOCC(COCCC(=O)NCCCNC(=O)CCCCOC2OC(CO)C(O)C(O)C2NC(C)=O)(COCCC(=O)NCCCNC(=O)CCCCOC2OC(CO)C(O)C(O)C2NC(C)=O)NC(=O)CCCCC(=O)N2CC3=CC=CC=C3C#CC3=CC=CC=C32)OC(CO)C(O)C1O HER2 P04626 10.1038/s41589-021-00770-1 TPD-391KD4 GalNAc-LYTAC2 . . . Epidermal growth factor receptor (EGFR) Cetuximab antibody . . . ASGPR tri-GalNAc-DBCO molecular CC(=O)NC1C(OCCCCC(=O)NCCCNC(=O)CCOCC(COCCC(=O)NCCCNC(=O)CCCCOC2OC(CO)C(O)C(O)C2NC(C)=O)(COCCC(=O)NCCCNC(=O)CCCCOC2OC(CO)C(O)C(O)C2NC(C)=O)NC(=O)CCCCC(=O)N2CC3=CC=CC=C3C#CC3=CC=CC=C32)OC(CO)C(O)C1O EGFR P00533 10.1038/s41589-021-00770-1 TPD-CE0QWQ Logic-TAC . . . Mucin-1 (MUC1) L1+LE1 DNA L1(5'to 3'): GCTGAATATCCATAATACTG LE1 (5'to 3'): CAGTATTATGGATATTCAGCGAAT DNA LO(5'to 3'):CGT, L2(5'to 3'):ACG IGF2R L2+LE2 DNA LE2(5'to 3'):CGTCTAGTACGGGCCC,L2(5'to 3'):GGGCGCGTAGATGACGAGCAGTCCTAACATCGTTTAGGAC MUC1 P15941 10.1002/smll.202310039 TPD-FCJYPV TfR-LYTAC(short) . . . Programmed cell death 1 ligand 1 (PD-L1) scFv of avelumab Antibody Fragment " QSALTQPASVSGSPGQSI TISCTGTSSDVGGYNYV SWYQQHPGKAPKLMIY DVSNRPSGVSNRFSGSK SGNTASLTISGLQAEDE ADYYCSSYTSSSTRVFG TGTKVTVLGGGGSGGG GSGGGGSGGGGSEVQL LESGGGLVQPGGSLRLS CAASGFTFSSYIMMWV RQAPGKGLEWVSSIYPS GGITFYADTVKGRFTISR DNSKNTLYLQMNSLRA EDTAVYYCARIKLGTVT TVDYWGQGTLVTVSS " Peptide GGGGSGGGGSGGGGSGGGGS transferrin receptor (TfR) TfRBP peptide "QSALTQPASVSGSPGQSI TISCTGTSSDVGGYNYV SWYQQHPGKAPKLMIY DVSNRPSGVSNRFSGSK SGNTASLTISGLQAEDE ADYYCSSYTSSSTRVFG TGTKVTVLGGGGSGGG GSGGGGSGGGGSEVQL LESGGGLVQPGGSLRLS CAASGFTFSSYIMMWV RQAPGKGLEWVSSIYPS GGITFYADTVKGRFTISR DNSKNTLYLQMNSLRA EDTAVYYCARIKLGTVT TVDYWGQGTLVTVSS " PD-L1 Q9NZQ7 10.1016/j.chembiol.2024.01.002 TPD-MAK3WW TfR-LYTAC(long) . . . Programmed cell death 1 ligand 1 (PD-L1) scFv of avelumab Antibody Fragment " QSALTQPASVSGSPGQSI TISCTGTSSDVGGYNYV SWYQQHPGKAPKLMIY DVSNRPSGVSNRFSGSK SGNTASLTISGLQAEDE ADYYCSSYTSSSTRVFG TGTKVTVLGGGGSGGG GSGGGGSGGGGSEVQL LESGGGLVQPGGSLRLS CAASGFTFSSYIMMWV RQAPGKGLEWVSSIYPS GGITFYADTVKGRFTISR DNSKNTLYLQMNSLRA EDTAVYYCARIKLGTVT TVDYWGQGTLVTVSS " Peptide GGGGSGGGGSGGGGSGGGGSGGGGSGGGGSGGGGSGGGGS transferrin receptor (TfR) TfRBP peptide "QSALTQPASVSGSPGQSI TISCTGTSSDVGGYNYV SWYQQHPGKAPKLMIY DVSNRPSGVSNRFSGSK SGNTASLTISGLQAEDE ADYYCSSYTSSSTRVFG TGTKVTVLGGGGSGGG GSGGGGSGGGGSEVQL LESGGGLVQPGGSLRLS CAASGFTFSSYIMMWV RQAPGKGLEWVSSIYPS GGITFYADTVKGRFTISR DNSKNTLYLQMNSLRA EDTAVYYCARIKLGTVT TVDYWGQGTLVTVSS " PD-L1 Q9NZQ7 10.1016/j.chembiol.2024.01.002 TPD-KR8048 Apt-LYTAC1 . . . Platelet-derived growth factor subunit B (PDGFB) aptamers DNA AGGGCGCGTTCTTCGTGGTTACTTTTAGTCCCG-biotin . . ASGPR triGalNAc molecular COCC1(COP(=O)([O-])OCC2(COP(=O)([O-])OCC3(COP(=O)([O-])OC)CCN(C(=O)CCCCCNC(=O)CCCOC4OC(CO)C(O)C(O)C4NC(C)=O)CC3)CCN(C(=O)CCCCCNC(=O)CCCOC3OC(CO)C(O)C(O)C3NC(C)=O)CC2)CCN(C(=O)CCCCCNC(=O)CCCOC2OC(CO)C(O)C(O)C2NC(C)=O)CC1 PDGFB P01127 10.1002/anie.202218106 TPD-MGJONI Apt-LYTAC2 . . . Inactive tyrosine-protein kinase 7 (PTK7) aptamers DNA ATCTAACTGCTGCGCCGCCGGGAAAATACTGTACGGTTAGA-biotin . . ASGPR triGalNAc molecular COCC1(COP(=O)([O-])OCC2(COP(=O)([O-])OCC3(COP(=O)([O-])OC)CCN(C(=O)CCCCCNC(=O)CCCOC4OC(CO)C(O)C(O)C4NC(C)=O)CC3)CCN(C(=O)CCCCCNC(=O)CCCOC3OC(CO)C(O)C(O)C3NC(C)=O)CC2)CCN(C(=O)CCCCCNC(=O)CCCOC2OC(CO)C(O)C(O)C2NC(C)=O)CC1 PTK7 Q13308 10.1002/anie.202218106 TPD-BNTQBS ITACs-MET . . . Hepatocyte growth factor receptor (c-Met) aptamers DNA TCAGGCTGGATGGTAGCTCGGTCGGGGTGGGTGGGTTGGCAAGTCTGAT DNA N3-AAAAAAAAAAAAAAAAAAAAA IGF2R IGF2-DBCO peptide P01344 c-Met P08581 10.1002/anie.202316089 TPD-PF5U6N ITACs-PTK7 . . . Inactive tyrosine-protein kinase 7 (PTK7) aptamers DNA TCTAACTGCTGCGCCGCCGGGAAAATACTGTACGGTTAGA DNA N3-AAAAAAAAAAAAAAAAAAAAA IGF2R IGF2-DBCO peptide P01344 PTK7 Q13308 10.1002/anie.202316089 TPD-L92JJ4 ITACs-FGFR2 . . . Fibroblast growth factor receptor 2 (FGFR2) aptamers DNA TGTTGGGAGGGGATGGGACGTATAGGTAAGGGCGGGGGTGGACACG DNA N3-AAAAAAAAAAAAAAAAAAAA IGF2R IGF2-DBCO peptide P01344 FGFR2 P21802 10.1002/anie.202316089 TPD-PT2WW8 mITACs . . . Hepatocyte growth factor receptor (c-Met) aptamers DNA "MET:ATCAGGCTGGATGGTAGCTCGGTCGGGGTGGGTGGGTTGGCAAGTCTGATAAAAAAAAAATATAGGTACACCCGTATTGAACCC PTK7:CCCTGTTTGTCGTTGTCTGTGTTCAAAAAAAAAAATCTAACTGCTGCGCCGCCGGGAAAATACTGTACGGTTAGA " DNA N3-AAAAAAAAAAACAACGAACACAGCAACGACAAACAGGGGGGTTCAATACGGGTGTACCTATA IGF2R IGF2-DBCO peptide P01344 c-Met;PTK7 P08581/Q13308 10.1002/anie.202316089 TPD-C7A8A2 ITACs-EpCAM . . . Epithelial cell adhesion molecule (EpCAM) aptamers DNA CACTACAGAGGTTGCGTCTGTCCCACGTTGTCATGGGGGGTTGGCCTG DNA N3-AAAAAAAAAAAAAAAAAAAA IGF2R IGF2-DBCO peptide P01344 EpCAM P16422 10.1002/anie.202316089 TPD-U2P6AF LYTACgyM6pG . . . Programmed cell death 1 ligand 1 (PD-L1) Nb-B3 Nanobody https://www.nature.com/articles/s41467-017-00799-8 . . IGF2R Mannose-6-Phosphate Glycans-DBCO Glycopeptide . PD-L1 Q9NZQ7 10.1021/acs.bioconjchem.4c00512 TPD-7MZP9B C5M1A . . . Programmed cell death 1 ligand 1 (PD-L1) Durvalumab-based anti-hPD-L1 IgG4 antibody C5 antibody "Light chain: IVLTQSPGTLSLSPGERATLSCKASEDIGTWLAVYQQKPGQAPRLLIYDASSRATGIPDRFSGSGSGTDFTLTISRLEPEDFAVYYCQQYGSLPWTFGQGTKVEIKRTVAAPSVFIFPPSDEQLKSGTASVVCLLNNFYPREAKVQWKVDNALQSGNSQESVTEQDSKDSTYSLSSTLTLSKADYEKHKVYACEVTHQGLSSPVTKSFNRGEC Heavy chain: EVQLVESGGGLVQPGGSLRLSCAASGFTFSRYMSWRQAPGKGLEWWALISRDGSETYYVDSVKGRFTISRDNAKNSLYLQMNSLRAEDTAVYYCAREGGWFGGELAFDYWGQGTLVTVSSASTKGPSVFPLAPSSKSTSGGTAALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSSLGTQTYICNVNHPKSNTKVDKRVEPKSCDKTHTPPCPAPELLGGPSVFLFPPKPKDTLMISRTEPVTCVVVDVSHEDPEVKFNWYVDGVEVHNAKTKPREEQFNSTYRVVSVLTVLHQDWLNGKEYKCKVSNKGLPSSIEKTISKAKGQPREPQVYTLPPSQEEMTKNQVSLTCLVKGFYPSDIAVEWESNGQPENNYKTTPPVLDSDGSFFLYSRLTVDKSRWQEGNVFSCSVMHEALHNHYTQKSLSLSLGK" . . IGF2R M5 DNA ETLCGGELVDTLQFVCGDRGFYNDDGIVEECCFRSCDLALLETYCATP PD-L1 Q9NZQ7 10.3390/molecules28227519 TPD-F9JZ49 Supra-LYTAC . . . Programmed cell death 1 ligand 1 (PD-L1) Py-FFK-BMS peptide-drug conjugate CC1=C(COC2=C(Br)C=C(CN3CCCCC3C(=O)NCCCCC(NC(=O)C(CC3=CC=CC=C3)NC(=O)C(CC3=CC=CC=C3)NC(=O)CCCC3=CC=C4C=CC5=CC=CC6=CC=C3C4=C56)C(N)=O)C=C2)C=CC=C1C1=CC=CC=C1 . . CAIX Py-FFK-Az peptide-drug conjugate NC(=O)C(CCCCNC(=O)CCC(=O)NC1=NN=C(S(N)(=O)=O)S1)NC(=O)C(CC1=CC=CC=C1)NC(=O)C(CC1=CC=CC=C1)NC(=O)CCCC1=C2C=CC3=CC=CC4=CC=C(C=C1)C2=C43 PD-L1 Q9NZQ7 10.1002/advs.202503134 TPD-DJN393 pep-2 . . . Programmed cell death 1 ligand 1 (PD-L1) T7 peptide HRPYIAH Peptide GS TFRC OPBP1 peptide-drug conjugate rvysf+k-ASF(N[C@H](CCCCNC(=O)C1=CC=CC(S(=O)(=O)F)=C1)C(=O)O) PD-L1 Q9NZQ7 10.1038/s41467-025-56648-6 TPD-VTM4ME pep-3 . . . Programmed cell death 1 ligand 1 (PD-L1) T7 peptide HRPYIAH Peptide GGGS TFRC OPBP1 peptide-drug conjugate rvysf+k-ASF(N[C@H](CCCCNC(=O)C1=CC=CC(S(=O)(=O)F)=C1)C(=O)O) PD-L1 Q9NZQ7 10.1038/s41467-025-56648-6 TPD-9VB11C pep-4 . . . Programmed cell death 1 ligand 1 (PD-L1) T7 peptide HRPYIAH Peptide GGGSGGGS TFRC OPBP1 peptide-drug conjugate rvysf+k-ASF(N[C@H](CCCCNC(=O)C1=CC=CC(S(=O)(=O)F)=C1)C(=O)O) PD-L1 Q9NZQ7 10.1038/s41467-025-56648-6 TPD-HFFAET pep-5 . . . Programmed cell death 1 ligand 1 (PD-L1) T7 peptide HRPYIAH Peptide PEGGGG TFRC OPBP1 peptide-drug conjugate rvysf+k-ASF(N[C@H](CCCCNC(=O)C1=CC=CC(S(=O)(=O)F)=C1)C(=O)O) PD-L1 Q9NZQ7 10.1038/s41467-025-56648-6 TPD-RKWK2G pep-6 . . . Programmed cell death 1 ligand 1 (PD-L1) T7 peptide HRPYIAH Peptide PEGGGGPEGGGG TFRC OPBP1 peptide-drug conjugate rvysf+k-ASF(N[C@H](CCCCNC(=O)C1=CC=CC(S(=O)(=O)F)=C1)C(=O)O) PD-L1 Q9NZQ7 10.1038/s41467-025-56648-6 TPD-UWK1SA V1 . . . Vascular endothelial growth factor A, long form (VEGF) VEGF aptamer-1 DNA TGTGGGGGTGGACTGGGTGGGTACC DNA M6PR:CGTAAATCAGTCATA,VEGF:TATGACTGATTTACG IGF2R M6PR aptamer DNA GGCGCGTAGATGACGAGCAGTCCTAACATCGTTTAGGAC VEGF P15692 10.7150/thno.98467 TPD-8NKPAY V2 . . . Vascular endothelial growth factor A, long form (VEGF) VEGF aptamer-2 DNA TGTGGGGGTGGACGGGCCGGGTAGA DNA M6PR:CGTAAATCAGTCATA,VEGF:TATGACTGATTTACG IGF2R M6PR aptamer DNA GGCGCGTAGATGACGAGCAGTCCTAACATCGTTTAGGAC VEGF P15692 10.7150/thno.98467 TPD-5L3Y8N V3 . . . Vascular endothelial growth factor A, long form (VEGF) VEGF aptamer-3 DNA GCCCGTCTTCCAGACAAGAGTGCAGGGC DNA M6PR:CGTAAATCAGTCATA,VEGF:TATGACTGATTTACG IGF2R M6PR aptamer DNA GGCGCGTAGATGACGAGCAGTCCTAACATCGTTTAGGAC VEGF P15692 10.7150/thno.98467 TPD-M9BDKD V4 . . . Vascular endothelial growth factor A, long form (VEGF) VEGF aptamer-1 DNA TGTGGGGGTGGACTGGGTGGGTACC DNA M6PR:CCCCCACACGTAAATCAGTCATA,VEGF:TATGACTGATTTACGTGTGGGGG IGF2R M6PR aptamer DNA GGCGCGTAGATGACGAGCAGTCCTAACATCGTTTAGGAC VEGF P15692 10.7150/thno.98467 TPD-4RP3UC V5 . . . Vascular endothelial growth factor A, long form (VEGF) VEGF aptamer-2 DNA TGTGGGGGTGGACGGGCCGGGTAGA DNA M6PR:CCCCCACACGTAAATCAGTCATA,VEGF:TATGACTGATTTACGTGTGGGGG IGF2R M6PR aptamer DNA GGCGCGTAGATGACGAGCAGTCCTAACATCGTTTAGGAC VEGF P15692 10.7150/thno.98467 TPD-TPDLQD V6 . . . Vascular endothelial growth factor A, long form (VEGF) VEGF aptamer-3 DNA GCCCGTCTTCCAGACAAGAGTGCAGGGC DNA M6PR:CCCCCACACGTAAATCAGTCATA,VEGF:TATGACTGATTTACGTGTGGGGG IGF2R M6PR aptamer DNA GGCGCGTAGATGACGAGCAGTCCTAACATCGTTTAGGAC VEGF P15692 10.7150/thno.98467 TPD-88PNXZ ASGPR-pCSK9-1 . . . Proprotein convertase subtilisin/kexin type 9 (PCSK9) ASGPR-PCSK9-bispecific antibody 5 antibody "ASGPR_4F3_ScFV-PCSK9_Fab_DANAPA_hIgG1_KiH_0 DIQMTQSPSSLSASVGDRVTITCRASQGISSALAWYQQKPGKAPKLLIYSASYRYTGVPSRFSGSGSGTDFTFTISSLQPEDIATYYCQQRYSLWRTFGQGTKLEIKRTVAAPSVFIFPPSDEQLKSGTASVVCLLNNFYPREAKVQWKVDNALQSGNSQESVTEQDSKDSTYSLSSTLTLSKADYEKHKVYACEVTHQGLSSPVTKSFNRGEC ASGPR_4F3_ScFV-PCSK9_Fab_DANAPA_hIgG1_KiH_1 EVQLLESGGGLVQPGGSLRLSCAASGFTFSSYAMSWVRQAPGKGLEWVSAISGSGGSTYYADSVKGRFTISRDNSKNTLYLQMNSLRAEDTAVYYCAKDFSSRRWYLEYWGQGTLVTVSSGGGGSGGGGSGGGGSGGGGSSSELTQDPAVSVALGQTVRITCQGDSLRSYYASWYQQKPGQAPVLVIYGKNNRPSGIPDRFSGSSSGNTASLTITGAQAEDEADYYCNSLERIGYLSYVFGGGTKLTVLGGGGSDKTHTCPPCPAPELLGGPSVFLFPPKPKDTLMISRTPEVTCVVVAVSHEDPEVKFNWYVDGVEVHNAKTKPREEQYASTYRVVSVLTVLHQDWLNGKEYKCKVSNKALAAPIEKTISKAKGQPREPQVYTLPPCREEMTKNQVSLWCLVKGFYPSDIAVEWESNGQPENNYKTTPPVLDSDGSFFLYSKLTVDKSRWQQGNVFSCSVMHEALHNRYTQKSLSLSPGK ASGPR_4F3_ScFV-PCSK9_Fab_DANAPA_hIgG1_KiH_2 QVQLVQSGAEVKKPGASVKVSCKASGYTFTSYYMHWVRQAPGQGLEWMGEISPFGGRTNYNEKFKSRVTMTRDTSTSTVYMELSSLRSEDTAVYYCARERPLYASDLWGQGTTVTVSSASTKGPSVFPLAPSSKSTSGGTAALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSSLGTQTYICNVNHKPSNTKVDKRVEPKSCDKTHTCPPCPAPELLGGPSVFLFPPKPKDTLMISRTPEVTCVVVAVSHEDPEVKFNWYVDGVEVHNAKTKPREEQYASTYRVVSVLTVLHQDWLNGKEYKCKVSNKALAAPIEKTISKAKGQPREPQVCTLPPSREEMTKNQVSLSCAVKGFYPSDIAVEWESNGQPENNYKTTPPVLDSDGSFFLVSKLTVDKSRWQQGNVFSCSVMHEALHNHYTQKSLSLSPGK" molecular NC(=O)CCOCCOCCOCCOCCC(N)=O ASGPR tri-GalNAc molecular CC(=O)NC1C(OCCCCC(=O)NCCCNC(=O)CCOCC(N)(COCCC(=O)NCCCNC(=O)CCCCOC2OC(CO)C(O)C(O)C2NC(C)=O)COCCC(=O)NCCCNC(=O)CCCCOC2OC(CO)C(O)C(O)C2NC(C)=O)OC(CO)C(O)C1O PCSK9 Q8NBP7 10.1016/j.chembiol.2022.12.003 TPD-9YSPE5 ASGPR-pCSK9-2 . . . Proprotein convertase subtilisin/kexin type 9 (PCSK9) PCSK9 macrocycle conjugate 15 molecular CC(=O)[C@@H]1NC(=O)[C@@H]2CCCN2C(=O)[C@H](C(C)C)NC(=O)[C@H](CC2=CC=CC=C2)NC(=O)CSC[C@@H](C(=O)NCC(=O)N[C@@H](CCCCN)C(N)=O)NC(=O)[C@@H]2CCCN2C(=O)[C@H](C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](C)NC(=O)[C@H](CC2=CC=C(C3=CC=CC=C3)C=C2)NC(=O)[C@H](C)N(C)C(=O)[C@H](CC2=CC=C(C3=CC=CC=C3)C=C2)NC(=O)[C@H]([C@@H](C)O)NC1=O molecular NC(=O)CCCCCCC(N)=O ASGPR tri-GalNAc molecular CC(=O)NC1C(OCCCCC(=O)NCCCNC(=O)CCOCC(N)(COCCC(=O)NCCCNC(=O)CCCCOC2OC(CO)C(O)C(O)C2NC(C)=O)COCCC(=O)NCCCNC(=O)CCCCOC2OC(CO)C(O)C(O)C2NC(C)=O)OC(CO)C(O)C1O PCSK9 Q8NBP7 10.1016/j.chembiol.2022.12.003 TPD-H276AB Ab1-3 . . . Receptor tyrosine-protein kinase erbB-2 (HER2) Trastuzumab antibody . Peptide GGGGSGGGGSGGGGS GGA or AP complexes MPR lysosomal sorting signal peptide peptide SFHDDSDEDLLHI HER2 P04626 WO-2024199551-A1 TPD-3HZ92C Ab4-6 . . . Receptor tyrosine-protein kinase erbB-2 (HER2) Trastuzumab antibody . Peptide GGGGSGGGGSGGGGS GGA or AP complexes C3 cell-penetrating peptide+MPR lysosomal sorting signal peptide peptide RRRRKSFHDDSDEDLLHI HER2 P04626 WO-2024199551-A1 TPD-70TTKA Tz-P4 . . . Receptor tyrosine-protein kinase erbB-2 (HER2) Trastuzumab antibody . Peptide GGGGSGGGGSGGGGS GGA or AP complexes MPR lysosomal sorting signal peptide peptide SYKYSKVNKE HER2 P04626 WO-2024199551-A1 TPD-E2ZT0H Ctx-C3-P1 . . . Epidermal growth factor receptor (EGFR) Cetuximab antibody . Peptide GGGGSGGGGSGGGGS GGA or AP complexes C3 cell-penetrating peptide+MPR lysosomal sorting signal peptide peptide RRRRKSFHDDSDEDLLHI EGFR P00533 WO-2024199551-A1 TPD-TKTQVR Az-P1 . . . Programmed cell death 1 ligand 1 (PD-L1) Atezolizumab antibody . Peptide GGGGSGGGGSGGGGS GGA or AP complexes MPR lysosomal sorting signal peptide peptide SYKYSKVNKE PD-L1 Q9NZQ7 WO-2024199551-A1 TPD-0N0FYU Az-C3-P1 . . . Programmed cell death 1 ligand 1 (PD-L1) Atezolizumab antibody . Peptide GGGGSGGGGSGGGGS GGA or AP complexes C3 cell-penetrating peptide+MPR lysosomal sorting signal peptide peptide RRRRKSFHDDSDEDLLHI PD-L1 Q9NZQ7 WO-2024199551-A1 TPD-4BTL0J Az-P3 . . . Programmed cell death 1 ligand 1 (PD-L1) Atezolizumab antibody . Peptide GGGGSGGGGSGGGGS GGA or AP complexes MPR lysosomal sorting signal peptide peptide EESEERDDHLLPM PD-L1 Q9NZQ7 WO-2024199551-A1 TPD-CUYXRW Az-P4 . . . Programmed cell death 1 ligand 1 (PD-L1) Atezolizumab antibody . Peptide GGGGSGGGGSGGGGS GGA or AP complexes MPR lysosomal sorting signal peptide peptide SYKYSKVNKE PD-L1 Q9NZQ7 WO-2024199551-A1 TPD-DPUM9Q Az-P6 . . . Programmed cell death 1 ligand 1 (PD-L1) Atezolizumab antibody . Peptide GGGGSGGGGSGGGGS GGA or AP complexes MPR lysosomal sorting signal peptide peptide PAAYRGVGDD PD-L1 Q9NZQ7 WO-2024199551-A1 TPD-4KDX76 Az-P7 . . . Programmed cell death 1 ligand 1 (PD-L1) Atezolizumab antibody . Peptide GGGGSGGGGSGGGGS AP complexes LAMP lysosomal sorting signal peptide peptide RKRSHAGYQTI PD-L1 Q9NZQ7 WO-2024199551-A1 TPD-ONJGJ8 Az-P8 . . . Programmed cell death 1 ligand 1 (PD-L1) Atezolizumab antibody . Peptide GGGGSGGGGSGGGGS GGA GGA lysosomal sorting signal peptide peptide ASSGLDDLDLLGK PD-L1 Q9NZQ7 WO-2024199551-A1 TPD-GPRGF3 Az-P9 . . . Programmed cell death 1 ligand 1 (PD-L1) Atezolizumab antibody . Peptide GGGGSGGGGSGGGGS GGA GGA lysosomal sorting signal peptide peptide VQNPSADRNLLDL PD-L1 Q9NZQ7 WO-2024199551-A1 TPD-3YTVNC Az-P10 . . . Programmed cell death 1 ligand 1 (PD-L1) Atezolizumab antibody . Peptide GGGGSGGGGSGGGGS GGA GGA lysosomal sorting signal peptide peptide ASVSLLDDELMSL PD-L1 Q9NZQ7 WO-2024199551-A1 TPD-PJJDVV Az-P13 . . . Programmed cell death 1 ligand 1 (PD-L1) Atezolizumab antibody . Peptide GGGGSGGGGSGGGGS GGA GGA lysosomal sorting signal peptide peptide NALSWLDEELLCL PD-L1 Q9NZQ7 WO-2024199551-A1 TPD-DV3SS6 Az-P22 . . . Programmed cell death 1 ligand 1 (PD-L1) Atezolizumab antibody . Peptide GGGGSGGGGSGGGGS AP complexes LAMP lysosomal sorting signal peptide peptide KHHHAGYEQF PD-L1 Q9NZQ7 WO-2024199551-A1 TPD-P8WOLT Rtx-C3-P1 . . . B-lymphocyte antigen CD20 (CD20) Rituximab antibody . Peptide GGGGSGGGGSGGGGS GGA or AP complexes C3 cell-penetrating peptide+MPR lysosomal sorting signal peptide peptide RRRRKSFHDDSDEDLLHI CD20 P11836 WO-2024199551-A1 TPD-L0SJDG Oftm-C3-P1 . . . B-lymphocyte antigen CD20 (CD20) Ofatumumab antibody . Peptide GGGGSGGGGSGGGGS GGA or AP complexes C3 cell-penetrating peptide+MPR lysosomal sorting signal peptide peptide RRRRKSFHDDSDEDLLHI CD20 P11836 WO-2024199551-A1 TPD-XPKE50 anti-CD71-C3-P1 . . . Transferrin receptor protein 1 (CD71) anti-CD71 antibody . Peptide GGGGSGGGGSGGGGS GGA or AP complexes C3 cell-penetrating peptide+MPR lysosomal sorting signal peptide peptide RRRRKSFHDDSDEDLLHI CD71 P02786 WO-2024199551-A1 TPD-63KPB6 Bv-C3-P1 . . . Vascular endothelial growth factor A, long form (VEGF) Bevacizumab antibody . Peptide GGGGSGGGGSGGGGS GGA or AP complexes C3 cell-penetrating peptide+MPR lysosomal sorting signal peptide peptide RRRRKSFHDDSDEDLLHI VEGF P15692 WO-2024199551-A1 TPD-N3PTV9 BsAb1-C3-P1 . . . Vascular endothelial growth factor A, long form (VEGF) Bevacizumab/Trastuzumab antibody . Peptide GGGGSGGGGSGGGGS GGA or AP complexes C3 cell-penetrating peptide+MPR lysosomal sorting signal peptide peptide RRRRKSFHDDSDEDLLHI VEGF;HER2 P15692/P04626 WO-2024199551-A1 TPD-ONBVRI BsAb2-P4 . . . Vascular endothelial growth factor A, long form (VEGF) Bevacizumab/Trastuzumab antibody . Peptide GGGGSGGGGSGGGGS GGA or AP complexes MPR lysosomal sorting signal peptide peptide SYKYSKVNKE VEGF;HER2 P15692/P04626 WO-2024199551-A1 TPD-3SZKIG BsAb3-P3 . . . Vascular endothelial growth factor A, long form (VEGF) Bevacizumab/Trastuzumab antibody . Peptide GGGGSGGGGSGGGGS GGA or AP complexes MPR lysosomal sorting signal peptide peptide EESEERDDHLLPM VEGF;HER2 P15692/P04626 WO-2024199551-A1 TPD-MYMTFG Nb1 . . . Receptor tyrosine-protein kinase erbB-2 (HER2) 5F7-His6 Nanobody . Peptide LPETGGG GGA or AP complexes MPR lysosomal sorting signal peptide peptide SFHDDSDEDLLHI HER2 P04626 WO-2024199551-A1 TPD-65F3IL Nb2 . . . Receptor tyrosine-protein kinase erbB-2 (HER2) 5F7-His6 Nanobody . Peptide LPETGGG GGA or AP complexes C3 cell-penetrating peptide+MPR lysosomal sorting signal peptide peptide RRRRKSFHDDSDEDLLHI HER2 P04626 WO-2024199551-A1 TPD-2UA2QI Nb3 . . . Receptor tyrosine-protein kinase erbB-2 (HER2) 5F7-His6 Nanobody . Peptide LPETGGG GGA or AP complexes MPR lysosomal sorting signal peptide peptide DDSDEDLL HER2 P04626 WO-2024199551-A1 TPD-B9AXI0 Nb4 . . . Receptor tyrosine-protein kinase erbB-2 (HER2) 5F7-His6 Nanobody . Peptide LPETGGG GGA or AP complexes MPR lysosomal sorting signal peptide peptide EESEERDDHLLPM HER2 P04626 WO-2024199551-A1 TPD-8SVV42 Nb5 . . . Receptor tyrosine-protein kinase erbB-2 (HER2) 5F7-His6 Nanobody . Peptide LPETGGG GGA or AP complexes MPR lysosomal sorting signal peptide peptide SYKYSKVNKE HER2 P04626 WO-2024199551-A1 TPD-UAFCTK Nb6 . . . Receptor tyrosine-protein kinase erbB-2 (HER2) 5F7-His6 Nanobody . Peptide LPETGGG GGA or AP complexes MPR lysosomal sorting signal peptide peptide YKYSKV HER2 P04626 WO-2024199551-A1 TPD-O48952 Nb7 . . . Receptor tyrosine-protein kinase erbB-2 (HER2) 5F7-His6 Nanobody . Peptide LPETGGG GGA or AP complexes MPR lysosomal sorting signal peptide peptide PAAYRGVGDD HER2 P04626 WO-2024199551-A1 TPD-850TZN Nb8 . . . Receptor tyrosine-protein kinase erbB-2 (HER2) 5F7-His6 Nanobody . Peptide LPETGGG AP complexes LAMP lysosomal sorting signal peptide peptide RKRSHAGYQTI HER2 P04626 WO-2024199551-A1 TPD-576VQ6 Nb9 . . . Receptor tyrosine-protein kinase erbB-2 (HER2) 5F7-His6 Nanobody . Peptide LPETGGG GGA GGA lysosomal sorting signal peptide peptide ASSGLDDLDLLGK HER2 P04626 WO-2024199551-A1 TPD-CN3R0D Nb10 . . . Receptor tyrosine-protein kinase erbB-2 (HER2) 5F7-His6 Nanobody . Peptide LPETGGG GGA GGA lysosomal sorting signal peptide peptide VQNPSADRNLLDL HER2 P04626 WO-2024199551-A1 TPD-59G8YO Nb11 . . . Receptor tyrosine-protein kinase erbB-2 (HER2) 5F7-His6 Nanobody . Peptide LPETGGG GGA GGA lysosomal sorting signal peptide peptide ASVSLLDDELMSL HER2 P04626 WO-2024199551-A1 TPD-6OJWNQ Nb12 . . . Receptor tyrosine-protein kinase erbB-2 (HER2) 5F7-His6 Nanobody . Peptide LPETGGG GGA GGA lysosomal sorting signal peptide peptide RRRASVSLLDDELMSL HER2 P04626 WO-2024199551-A1 TPD-UBQREF Nb13 . . . Receptor tyrosine-protein kinase erbB-2 (HER2) 5F7-His6 Nanobody . Peptide LPETGGG GGA GGA lysosomal sorting signal peptide peptide ASVSLLDDEL HER2 P04626 WO-2024199551-A1 TPD-LO9F8P Nb14 . . . Receptor tyrosine-protein kinase erbB-2 (HER2) 5F7-His6 Nanobody . Peptide LPETGGG GGA GGA lysosomal sorting signal peptide peptide NALSWLDEELLCL HER2 P04626 WO-2024199551-A1 TPD-YGP1ZF Nb15 . . . Receptor tyrosine-protein kinase erbB-2 (HER2) 5F7-His6 Nanobody . Peptide LPETGGG GGA or AP complexes MPR lysosomal sorting signal peptide peptide SDEDLLHI HER2 P04626 WO-2024199551-A1 TPD-HJP8OO Nb16 . . . Receptor tyrosine-protein kinase erbB-2 (HER2) 5F7-His6 Nanobody . Peptide LPETGGG GGA or AP complexes MPR lysosomal sorting signal peptide peptide RRRSDEDLLHI HER2 P04626 WO-2024199551-A1 TPD-103W79 Nb17 . . . Receptor tyrosine-protein kinase erbB-2 (HER2) 5F7-His6 Nanobody . Peptide LPETGGG GGA or AP complexes MPR lysosomal sorting signal peptide peptide RRLRKSDEDLLHI HER2 P04626 WO-2024199551-A1 TPD-EIQ69L Nb18 . . . Receptor tyrosine-protein kinase erbB-2 (HER2) 5F7-His6 Nanobody . Peptide LPETGGG GGA or AP complexes MPR lysosomal sorting signal peptide peptide RRRRKSDEDLLHI HER2 P04626 WO-2024199551-A1 TPD-VZY48W Nb19 . . . Receptor tyrosine-protein kinase erbB-2 (HER2) 5F7-His6 Nanobody . Peptide LPETGGG GGA or AP complexes MPR lysosomal sorting signal peptide peptide RRRSFHDDSDEDLLHI HER2 P04626 WO-2024199551-A1 TPD-MIV4AP Nb20 . . . Receptor tyrosine-protein kinase erbB-2 (HER2) 5F7-His6 Nanobody . Peptide LPETGGG GGA or AP complexes MPR lysosomal sorting signal peptide peptide RRLRKSFHDDSDEDLLHI HER2 P04626 WO-2024199551-A1 TPD-ZT1MPD Nb21 . . . Receptor tyrosine-protein kinase erbB-2 (HER2) 5F7-His6 Nanobody . Peptide LPETGGG GGA or AP complexes MPR lysosomal sorting signal peptide peptide RRRRKSFHDDSDEDLLHI HER2 P04626 WO-2024199551-A1 TPD-LFOQM1 Nb22 . . . Receptor tyrosine-protein kinase erbB-2 (HER2) 5F7-His6 Nanobody . Peptide LPETGGG AP complexes LAMP lysosomal sorting signal peptide peptide RRRRKRKRSHAGYQTI HER2 P04626 WO-2024199551-A1 TPD-3IWAFN Nb23 . . . Receptor tyrosine-protein kinase erbB-2 (HER2) 5F7-His6 Nanobody . Peptide LPETGGG AP complexes LAMP lysosomal sorting signal peptide peptide KHHHAGYEQF HER2 P04626 WO-2024199551-A1 TPD-B4QDTD Nb24 . . . Receptor tyrosine-protein kinase erbB-2 (HER2) 5F7-His6 Nanobody . Peptide LPETGGG AP complexes LAMP lysosomal sorting signal peptide peptide RRLRKHHHAGYEQF HER2 P04626 WO-2024199551-A1 TPD-EIBLJO 7D12-P1 . . . Receptor tyrosine-protein kinase erbB-2 (HER2) 7D12-His6 Nanobody . Peptide GGGGS GGA or AP complexes LAMP lysosomal sorting signal peptide peptide SFHDDSDEDLLHI HER2 P04626 WO-2024199551-A1 TPD-XWMYJX 7D12-C3-P1 . . . Receptor tyrosine-protein kinase erbB-2 (HER2) 7D12-His6 Nanobody . Peptide GGGGS GGA or AP complexes C3 cell-penetrating peptide+MPR lysosomal sorting signal peptide peptide RRRRKSFHDDSDEDLLHI HER2 P04626 WO-2024199551-A1 TPD-06ZUYQ PEP1-P1 . . . Epidermal growth factor receptor (EGFR) PEP1 Peptide LARLLT . . GGA or AP complexes MPR lysosomal sorting signal peptide peptide SFHDDSDEDLLHI EGFR P00533 WO-2024199551-A1 TPD-AEDQ42 PEP1-C3-P1 . . . Epidermal growth factor receptor (EGFR) PEP1 Peptide LARLLT . . GGA or AP complexes C3 cell-penetrating peptide+MPR lysosomal sorting signal peptide peptide RRRRKSFHDDSDEDLLHI EGFR P00533 WO-2024199551-A1 TPD-NNKN2W PEP2-C4-P1 . . . Epidermal growth factor receptor (EGFR) PEP2 Peptide RRPPRSPDHKRYFRDKE . . GGA or AP complexes C3 cell-penetrating peptide+MPR lysosomal sorting signal peptide peptide YGRKKRRQRRRSFHDDSDEDLLHI EGFR P00533 WO-2024199551-A1 TPD-B5S8D7 DBCO-LYTAC2-6T . . . Epithelial cell adhesion molecule (EpCAM) EpCAM aptamers DNA [DBCO]-TTT-CACTACAGAGGTTGCGTCTGTCCCACGTTGTCATGGGGGGTTGGCCTG DNA TTTTTT CI-M6PR M6PR aptamers DNA GGGCGCGTAGATGACGAGCAGTCCTAACATCGTTTAGGAC EpCAM P16422 CN-119220547-A TPD-JLUMH3 LYTAC-6T . . . Programmed cell death 1 ligand 1 (PD-L1) PD-L1 aptamers DNA ACGGGCCACATCAACTCATTGATAGACAATGCGTCCACTGCCCGT DNA TTTTTT CI-M6PR M6PR aptamers DNA GGGCGCGTAGATGACGAGCAGTCCTAACATCGTTTAGGAC PD-L1 Q9NZQ7 CN-119220547-A TPD-07THBZ LYTAC2-6T . . . Epithelial cell adhesion molecule (EpCAM) EpCAM aptamers DNA CACTACAGAGGTTGCGTCTGTCCCACGTTGTCATGGGGGGTTGGCCTG DNA TTTTTT CI-M6PR M6PR aptamers DNA GGGCGCGTAGATGACGAGCAGTCCTAACATCGTTTAGGAC EpCAM P16422 CN-119220547-A TPD-Q0QIYL VHH fusion 13 . . . Epidermal growth factor receptor (EGFR) 9GB Nanobody EVQLVESGGGLVQAGGSLRLSCAASGRTFSSYAMGWFRQAPGKEREFVVAINWSSGSTYYADSVKGRFTISRDNAKNTMYLQMNSLKPEDTAVYYCAAGYQINSGNYNFKDYEYDYWGQGTQVTVSS Peptide GGGGSGGGGSGGGGS CI-M6PR VHH8 Nanobody QVQLQESGGGLVQAGGSLRLSCEASGRTFNTYNWGWFRQAPGKEREFVAAIRWSSSKTSYADSVKGRFTISRDNAKNTIYLQMNSLKPEDTAVYYCAASIVDFTTNPSHFGSWGQGTQVTVSS EGFR P00533 US-20240327525-A1 TPD-N03DH0 VHH fusion 14 . . . Epidermal growth factor receptor (EGFR) 9GB+G4Sx3+9G8 Nanobody EVQLVESGGGLVQAGGSLRLSCAASGRTFSSYAMGWFRQAPGKEREFVVAINWSSGSTYYADSVKGRFTISRDNAKNTMYLQMNSLKPEDTAVYYCAAGYQINSGNYNFKDYEYDYWGQGTQVTVSSGGGGSGGGGSGGGGSEVQLVESGGGLVQAGGSLRLSCAASGRTFSSYAMGWFRQAPGKEREFVVAINWSSGSTYYADSVKGRFTISRDNAKNTMYLQMNSLKPEDTAVYYCAAGYQINSGNYNFKDYEYDYWGQGTQVTVSS Peptide GGGGSGGGGSGGGGS CI-M6PR VHH8 Nanobody QVQLQESGGGLVQAGGSLRLSCEASGRTFNTYNWGWFRQAPGKEREFVAAIRWSSSKTSYADSVKGRFTISRDNAKNTIYLQMNSLKPEDTAVYYCAASIVDFTTNPSHFGSWGQGTQVTVSS EGFR P00533 US-20240327525-A1 TPD-IE8Q71 VHH fusion 18 . . . Epidermal growth factor receptor (EGFR) 9GB S54A Nanobody EVQLVESGGGLVQAGGSLRLSCAASGRTFSSYAMGWFRQAPGKEREFVVAINWASGSTYYADSVKGRFTISRDNAKNTMYLQMNSLKPEDTAVYYCAAGYQINSGNYNFKDYEYDYWGQGTQVTVSS Peptide GGGGSGGGGSGGGGS CI-M6PR VHH8 Nanobody QVQLQESGGGLVQAGGSLRLSCEASGRTFNTYNWGWFRQAPGKEREFVAAIRWSSSKTSYADSVKGRFTISRDNAKNTIYLQMNSLKPEDTAVYYCAASIVDFTTNPSHFGSWGQGTQVTVSS EGFR P00533 US-20240327525-A1 TPD-CAXOV8 VHH fusion 19 . . . Epidermal growth factor receptor (EGFR) 9GB S54A+G4Sx3+9GB S54A Nanobody EVQLVESGGGLVQAGGSLRLSCAASGRTFSSYAMGWFRQAPGKEREFVVAINWASGSTYYADSVKGRFTISRDNAKNTMYLQMNSLKPEDTAVYYCAAGYQINSGNYNFKDYEYDYWGQGTQVTVSSGGGGSGGGGSGGGGSEVQLVESGGGLVQAGGSLRLSCAASGRTFSSYAMGWFRQAPGKEREFVVAINWSAGSTYYADSVKGRFTISRDNAKNTMYLQMNSLKPEDTAVYYCAAGYQINSGNYNFKDYEYDYWGQGTQVTVSS Peptide GGGGSGGGGSGGGGS CI-M6PR VHH8 Nanobody QVQLQESGGGLVQAGGSLRLSCEASGRTFNTYNWGWFRQAPGKEREFVAAIRWSSSKTSYADSVKGRFTISRDNAKNTIYLQMNSLKPEDTAVYYCAASIVDFTTNPSHFGSWGQGTQVTVSS EGFR P00533 US-20240327525-A1 TPD-8UWJH7 VHH fusion 82 . . . Epidermal growth factor receptor (EGFR) 9GB S54A Nanobody EVQLVESGGGLVQAGGSLRLSCAASGRTFSSYAMGWFRQAPGKEREFVVAINWASGSTYYADSVKGRFTISRDNAKNTMYLQMNSLKPEDTAVYYCAAGYQINSGNYNFKDYEYDYWGQGTQVTVSS Peptide GGGGSGGGGSGGGGS CI-M6PR VHH7 Nanobody QVQLQESGGGLVQPGGSLRLSCAASGIIFSDNRMDWYRQAPGKQREWVATLASYGWKTYADSVKGRFTISRDNTKNTVYLRMNSLKPEDTAVYYCKASSPVLNDIWGQGTQVTVSS EGFR P00533 US-20240327525-A1 TPD-5O1H48 VHH fusion 84 . . . Epidermal growth factor receptor (EGFR) 9GB S54A+G4Sx3+9GB S54A Nanobody EVQLVESGGGLVQAGGSLRLSCAASGRTFSSYAMGWFRQAPGKEREFVVAINWASGSTYYADSVKGRFTISRDNAKNTMYLQMNSLKPEDTAVYYCAAGYQINSGNYNFKDYEYDYWGQGTQVTVSSGGGGSGGGGSGGGGSEVQLVESGGGLVQAGGSLRLSCAASGRTFSSYAMGWFRQAPGKEREFVVAINWSAGSTYYADSVKGRFTISRDNAKNTMYLQMNSLKPEDTAVYYCAAGYQINSGNYNFKDYEYDYWGQGTQVTVSS Peptide GGGGSGGGGSGGGGS CI-M6PR VHH7 Nanobody QVQLQESGGGLVQPGGSLRLSCAASGIIFSDNRMDWYRQAPGKQREWVATLASYGWKTYADSVKGRFTISRDNTKNTVYLRMNSLKPEDTAVYYCKASSPVLNDIWGQGTQVTVSS EGFR P00533 US-20240327525-A1 TPD-G25QHQ VHH fusion 88 . . . Epidermal growth factor receptor (EGFR) 9GB S54A Nanobody EVQLVESGGGLVQAGGSLRLSCAASGRTFSSYAMGWFRQAPGKEREFVVAINWASGSTYYADSVKGRFTISRDNAKNTMYLQMNSLKPEDTAVYYCAAGYQINSGNYNFKDYEYDYWGQGTQVTVSS Peptide GGGGSGGGGSGGGGSGGGGSGGGGSGGGGSGGGGSGGGGSGGGGS CI-M6PR VHH7 Nanobody QVQLQESGGGLVQPGGSLRLSCAASGIIFSDNRMDWYRQAPGKQREWVATLASYGWKTYADSVKGRFTISRDNTKNTVYLRMNSLKPEDTAVYYCKASSPVLNDIWGQGTQVTVSS EGFR P00533 US-20240327525-A1 TPD-Z1BW1A VHH fusion 89 . . . Epidermal growth factor receptor (EGFR) 9GB S54A Nanobody EVQLVESGGGLVQAGGSLRLSCAASGRTFSSYAMGWFRQAPGKEREFVVAINWASGSTYYADSVKGRFTISRDNAKNTMYLQMNSLKPEDTAVYYCAAGYQINSGNYNFKDYEYDYWGQGTQVTVSS Peptide GGGGSGGGGSGGGGSGGGGSGGGGSGGGGSGGGGSGGGGSGGGGS CI-M6PR VHH8 Nanobody QVQLQESGGGLVQAGGSLRLSCEASGRTFNTYNWGWFRQAPGKEREFVAAIRWSSSKTSYADSVKGRFTISRDNAKNTIYLQMNSLKPEDTAVYYCAASIVDFTTNPSHFGSWGQGTQVTVSS EGFR P00533 US-20240327525-A1 TPD-QBC6GI Ctx-VHH7 . . . Epidermal growth factor receptor (EGFR) Cetuximab antibody . Peptide GGGGSGGGGS CI-M6PR VHH7 Nanobody QVQLQESGGGLVQPGGSLRLSCAASGIIFSDNRMDWYRQAPGKQREWVATLASYGWKTYADSVKGRFTISRDNTKNTVYLRMNSLKPEDTAVYYCKASSPVLNDIWGQGTQVTVSS EGFR P00533 US-20240327525-A1 TPD-UOJIS6 Ctx-VHH8 . . . Epidermal growth factor receptor (EGFR) Cetuximab antibody . Peptide GGGGSGGGGS CI-M6PR VHH8 Nanobody QVQLQESGGGLVQAGGSLRLSCEASGRTFNTYNWGWFRQAPGKEREFVAAIRWSSSKTSYADSVKGRFTISRDNAKNTIYLQMNSLKPEDTAVYYCAASIVDFTTNPSHFGSWGQGTQVTVSS EGFR P00533 US-20240327525-A1 TPD-9ZMSS0 VHH fusion 91 . . . Green fluorescent protein (GFP) GBP Peptide DVQLVESGGALVQPGGSLRLSCAASGFPVNRYSMRWYRQAPGKEREWVAGMSSAGDRSSYEDSVKGRFTISRDDARNTVYLQMNSLKPEDTAVYYCNVNVGFEYWGQGTQVTVSS Peptide GGGGSGGGGSGGGGS CI-M6PR VHH7 Nanobody QVQLQESGGGLVQPGGSLRLSCAASGIIFSDNRMDWYRQAPGKQREWVATLASYGWKTYADSVKGRFTISRDNTKNTVYLRMNSLKPEDTAVYYCKASSPVLNDIWGQGTQVTVSS GFP P42212 US-20240327525-A1 TPD-LIALEN VHH fusion 92 . . . Green fluorescent protein (GFP) GBP Peptide DVQLVESGGALVQPGGSLRLSCAASGFPVNRYSMRWYRQAPGKEREWVAGMSSAGDRSSYEDSVKGRFTISRDDARNTVYLQMNSLKPEDTAVYYCNVNVGFEYWGQGTQVTVSS Peptide GGGGSGGGGSGGGGS CI-M6PR VHH8 Nanobody QVQLQESGGGLVQAGGSLRLSCEASGRTFNTYNWGWFRQAPGKEREFVAAIRWSSSKTSYADSVKGRFTISRDNAKNTIYLQMNSLKPEDTAVYYCAASIVDFTTNPSHFGSWGQGTQVTVSS GFP P42212 US-20240327525-A1 TPD-8V9OYP VHH fusion 93 . . . Green fluorescent protein (GFP) GBP Peptide DVQLVESGGALVQPGGSLRLSCAASGFPVNRYSMRWYRQAPGKEREWVAGMSSAGDRSSYEDSVKGRFTISRDDARNTVYLQMNSLKPEDTAVYYCNVNVGFEYWGQGTQVTVSS Peptide GGGGSGGGGSGGGGS CI-M6PR VHH1 Nanobody QVQLQESGGGLVQPGGSLRLSCVASGFTFDRYWMNWLRQIPGKEIEWVSTINTGGTGTYYDDSVKGRFSISRDDAKNTLYLTMNSLKTEDTAVYYCARGATYYRGNSAIRGQGTQVTVSS GFP P42212 US-20240327525-A1 TPD-EZHCK7 VHH fusion 94 . . . Green fluorescent protein (GFP) GBP Peptide DVQLVESGGALVQPGGSLRLSCAASGFPVNRYSMRWYRQAPGKEREWVAGMSSAGDRSSYEDSVKGRFTISRDDARNTVYLQMNSLKPEDTAVYYCNVNVGFEYWGQGTQVTVSS Peptide GGGGSGGGGSGGGGS CI-M6PR VHH5 Nanobody QVQLQESGGGLVQAGGSLKLSCAAAGRTFSRLAMGWFRQAPGKEREFVAAISENGDSIHYSDSVKGRFAVSRDNAKNTVYLQMNSLKPEDTAIYCAADRAAYYCSGSGCYPSRAPAAASYDYWGQGTQVTVSS GFP P42212 US-20240327525-A1 TPD-V2OU2D VHH fusion 95 . . . Green fluorescent protein (GFP) GBP Peptide DVQLVESGGALVQPGGSLRLSCAASGFPVNRYSMRWYRQAPGKEREWVAGMSSAGDRSSYEDSVKGRFTISRDDARNTVYLQMNSLKPEDTAVYYCNVNVGFEYWGQGTQVTVSS Peptide GGGGSGGGGSGGGGS CI-M6PR VHH11 Nanobody QVQLQESGGGLVQPGGSLRLSCAASGIIFSDNRMDWYRQAPGKQREWVATLASYGWKTYADSVKDRFTISRDNAKNTVNLYMNSLQPEDTAVYYCNSGQYWGQGTQVTVSS GFP P42212 US-20240327525-A1 TPD-Z4BY0F VHH fusion 96 . . . Green fluorescent protein (GFP) GBP Peptide DVQLVESGGALVQPGGSLRLSCAASGFPVNRYSMRWYRQAPGKEREWVAGMSSAGDRSSYEDSVKGRFTISRDDARNTVYLQMNSLKPEDTAVYYCNVNVGFEYWGQGTQVTVSS Peptide GGGGSGGGGSGGGGSGGGGSGGGGSGGGGSGGGGSGGGGSGGGGS CI-M6PR VHH1H52 Nanobody QVQLQESGGGLVQPGGSLRLSCTASGFTWDSYVIGWFRQAPGKGREGVSCLDVDDGSIYYHDSAKGRFSISRDNAKNTVYLQMNSLKPEDTAVYYCAAVNRASMRFRRCLQVLRYDYWGQGTQVTVSS GFP P42212 US-20240327525-A1 TPD-HD1N0F TypeA . . . Programmed cell death 1 ligand 1 (PD-L1) Atezolizumab antibody "light chain: (linker)-DIQMTQSPSSLSASVGDRVTITCRASQDVSTAVAWYQQKPGKAPKLLIYSASFLYSGVPSRFSGSGSGTDFTLTISSLQPEDFATYYCQQYLYHPATFGQGTKVEIKRTVAAPSVFIFPPCDEQLKSGTASVVCLLNNFYPREAKVQWKVDNALQSGNSQESVTEQDSKDSTYSLSSTLTLSKADYEKHKVYACEVTHQGLSSPVTKSFNRGECHHHHHH heavy chain: EVQLVESGGGLVQPGGSLRLSCAASGFTFSDSWIHWVRQAPGKGLEWVAWISPYGGSTYYADSVKGRFTISADTSKNTAYLQMNSLRAEDTAVYYCARRHWPGGFDYWGQGTLVTVSSASTKGPSVCPLAPSSKSTSGGTAALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSSLGTQTYICNVNHKPSNTKVDKKVEPKSCDKTHTCPPCPAPEAAGGPSVFLFPPKPKDTLMISRTPEVTCVVVDVSHEDPEVKFNWYVDGVEVHNAKTKPREEQYNSTYRVVSVLTVLHQDWLNGKEYKCKVSNKALGAPIEKTISKAKGQPREPQVCTLPPSRDELTKNQVSLTCLVKGFYPSDIAVEWESNGQPENNYKTTPPVLDSDGSFFLYSKLTVDKSRWQQGNVFSCSVMHEALHNRYTQKSLSLSPGK" Peptide GGGGS IGF2R IGF2 Peptide AYRPSETLCGGELVDTLQFVCGDRGFYFSRPASRVSRRSRGIVEECCFRSCDLALLETYCATPAKSES PD-L1 Q9NZQ7 CN-119954970-A TPD-KGV2SS TypeA-GS . . . Programmed cell death 1 ligand 1 (PD-L1) Atezolizumab antibody "light chain: (linker)-EPKSCDKTHTCPPCPAPEAAGGPSVFLFPPKPKDTLMISRTPEVTCVVVDVSHEDPEVKFNWYVDGVEVHNAKTKPREEQYNSTYRVVSVLTVLHQDWLNGKEYKCKVSNKALGAPIEKTISKAKGQPREPQVYTLPPCRDELTKNQVSLWCLVKGFYPSDIAVEWESNGQPENNYKTTPPVLDSDGSFFLYSKLTVDKSRWQQGNVFSCSVMHEALHNRYTQKSLSLSPGK heavy chain: EVQLVESGGGLVQPGGSLRLSCAASGFTFSDSWIHWVRQAPGKGLEWVAWISPYGGSTYYADSVKGRFTISADTSKNTAYLQMNSLRAEDTAVYYCARRHWPGGFDYWGQGTLVTVSSASTKGPSVCPLAPSSKSTSGGTAALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSSLGTQTYICNVNHKPSNTKVDKKVEPKSCDKTHTCPPCPAPEAAGGPSVFLFPPKPKDTLMISRTPEVTCVVVDVSHEDPEVKFNWYVDGVEVHNAKTKPREEQYNSTYRVVSVLTVLHQDWLNGKEYKCKVSNKALGAPIEKTISKAKGQPREPQVCTLPPSRDELTKNQVSLTCLVKGFYPSDIAVEWESNGQPENNYKTTPPVLDSDGSFFLYSKLTVDKSRWQQGNVFSCSVMHEALHNRYTQKSLSLSPGK" Peptide GGGGSGGGGSGGGGS IGF2R IGF2 Peptide AYRPSETLCGGELVDTLQFVCGDRGFYFSRPASRVSRRSRGIVEECCFRSCDLALLETYCATPAKSES PD-L1 Q9NZQ7 CN-119954970-A TPD-YMAC5H TypeB . . . Programmed cell death 1 ligand 1 (PD-L1) Atezolizumab antibody "light chain: (linker)-DIQMTQSPSSLSASVGDRVTITCRASQDVSTAVAWYQQKPGKAPKLLIYSASFLYSGVPSRFSGSGSGTDFTLTISSLQPEDFATYYCQQYLYHPATFGQGTKVEIKRTVAAPSVFIFPPCDEQLKSGTASVVCLLNNFYPREAKVQWKVDNALQSGNSQESVTEQDSKDSTYSLSSTLTLSKADYEKHKVYACEVTHQGLSSPVTKSFNRGECHHHHHH heavy chain: EVQLVESGGGLVQPGGSLRLSCAASGFTFSDSWIHWVRQAPGKGLEWVAWISPYGGSTYYADSVKGRFTISADTSKNTAYLQMNSLRAEDTAVYYCARRHWPGGFDYWGQGTLVTVSSASTKGPSVCPLAPSSKSTSGGTAALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSSLGTQTYICNVNHKPSNTKVDKKVEPKSCDKTHTCPPCPAPEAAGGPSVFLFPPKPKDTLMISRTPEVTCVVVDVSHEDPEVKFNWYVDGVEVHNAKTKPREEQYNSTYRVVSVLTVLHQDWLNGKEYKCKVSNKALGAPIEKTISKAKGQPREPQVCTLPPSRDELTKNQVSLTCLVKGFYPSDIAVEWESNGQPENNYKTTPPVLDSDGSFFLYSKLTVDKSRWQQGNVFSCSVMHEALHNRYTQKSLSLSPGK" Peptide GGGGSGGGGSGGGGS IGF2R IGF2 Peptide AYRPSETLCGGELVDTLQFVCGDRGFYFSRPASRVSRRSRGIVEECCFRSCDLALLETYCATPAKSES PD-L1 Q9NZQ7 CN-119954970-A TPD-24N3G8 TypeB-Fab . . . Programmed cell death 1 ligand 1 (PD-L1) Atezolizumab antibody "light chain: (linker)-DIQMTQSPSSLSASVGDRVTITCRASQDVSTAVAWYQQKPGKAPKLLIYSASFLYSGVPSRFSGSGSGTDFTLTISSLQPEDFATYYCQQYLYHPATFGQGTKVEIKRTVAAPSVFIFPPCDEQLKSGTASVVCLLNNFYPREAKVQWKVDNALQSGNSQESVTEQDSKDSTYSLSSTLTLSKADYEKHKVYACEVTHQGLSSPVTKSFNRGECHHHHHH heavy chain: (linker)- EVQLVESGGGLVQPGGSLRLSCAASGFTFSDSWIHWVRQAPGKGLEWVAWISPYGGSTYYADSVKGRFTISADTSKNTAYLQMNSLRAEDTAVYYCARRHWPGGFDYWGQGTLVTVSSASTKGPSVCPLAPSSKSTSGGTAALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSSLGTQTYICNVNHKPSNTKVDKKVHHHHHH" Peptide GGGGSGGGGSGGGGS IGF2R IGF2 Peptide AYRPSETLCGGELVDTLQFVCGDRGFYFSRPASRVSRRSRGIVEECCFRSCDLALLETYCATPAKSES PD-L1 Q9NZQ7 CN-119954970-A TPD-B90O5K TypeB-Flmut . . . Programmed cell death 1 ligand 1 (PD-L1) Atezolizumab antibody "light chain: (linker)-DIQMTQSPSSLSASVGDRVTITCRASQDVSTAVAWYQQKPGKAPKLLIYSASFLYSGVPSRFSGSGSGTDFTLTISSLQPEDFATYYCQQYLYHPATFGQGTKVEIKRTVAAPSVFIFPPCDEQLKSGTASVVCLLNNFYPREAKVQWKVDNALQSGNSQESVTEQDSKDSTYSLSSTLTLSKADYEKHKVYACEVTHQGLSSPVTKSFNRGECHHHHHH heavy chain: EVQLVESGGGLVQPGGSLRLSCAASGFTFSDSWIHWVRQAPGKGLEWVAWISPYGGSTYYADSVKGRFTISADTSKNTAYLQMNSLRAEDTAVYYCARRHWPGGFDYWGQGTLVTVSSASTKGPSVCPLAPSSKSTSGGTAALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSSLGTQTYICNVNHKPSNTKVDKKVEPKSCDKTHTCPPCPAPEAAGGPSVFLFPPKPKDTLMISRTPEVTCVVVDVSHEDPEVKFNWYVDGVEVHNAKTKPREEQYNSTYRVVSVLTVLHQDWLNGKEYKCKVSNKALGAPIEKTISKAKGQPREPQVCTLPPSRDELTKNQVSLTCLVKGFYPSDIAVEWESNGQPENNYKTTPPVLDSDGSFFLYSKLTVDKSRWQQGNVFSCSVMHEALHNRYTQKSLSLSPGK" Peptide GGGGSGGGGSGGGGS IGF2R IGF2 Peptide AYRPSETLCGGELVDTLQFVCGDRGFYFSRPASRVSRRSRGIVEECCDRSCDDALLETYCATPAKSES PD-L1 Q9NZQ7 CN-119954970-A TPD-0I7LR2 HER2Ab-TypeB . . . Receptor tyrosine-protein kinase erbB-2 (HER2) Trastuzumab antibody "light chain: (linker)-DIQMTQSPSSLSASVGDRVTITCRASQDVNTAVAWYQQKPGKAPKLLIYSASFLYSGVPSRFSGSRSGTDFTLTISSLQPEDFATYYCQQHYTTPPTFGCGTKVEIKRTVAAPSVFIFPPCDEQLKSGTASVVCLLNNFYPREAKVQWKVDNALQSGNSQESVTEQDSKDSTYSLSSTLTLSKADYEKHKVYACEVTHQGLSSPVTKSFNRG heavy chain: EVQLVESGGGLVQPGGSLRLSCAASGFNIKDTYIHWVRQAPGKCLEWVARIYPTNGYTRYADSVKGRFTISADTSKNTAYLQMNSLRAEDTAVYYCSRWGGDGFYAMDYWGQGTLVTVSSASTKGPSVCPLAPSSKSTSGGTAALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSSLGTQTYICNVNHKPSNTKVDKKVEPKSCDKTHTCPPCPAPEAAGGPSVFLFPPKPKDTLMISRTPEVTCVVVDVSHEDPEVKFNWYVDGVEVHNAKTKPREEQYNSTYRVVSVLTVLHQDWLNGKEYKCKVSNKALGAPIEKTISKAKGQPREPQVCTLPPSRDELTKNQVSLTCLVKGFYPSDIAVEWESNGQPENNYKTTPPVLDSDGSFFLYSKLTVDKSRWQQGNVFSCSVMHEALHNRYTQKSLSLSPGK" Peptide GGGGSGGGGSGGGGS IGF2R IGF2 Peptide AYRPSETLCGGELVDTLQFVCGDRGFYFSRPASRVSRRSRGIVEECCFRSCDLALLETYCATPAKSES HER2 P04626 CN-119954970-A TPD-01M164 EGFRAb-TypeB . . . Epidermal growth factor receptor (EGFR) Cetuximab antibody "light chain: (linker)-DIQMTQSPSSLSASVGDRVTITCRASQDVNTAVAWYQQKPGKAPKLLIYSASFLYSGVPSRFSGSRSGTDFTLTISSLQPEDFATYYCQQHYTTPPTFGCGTKVEIKRTVAAPSVFIFPPCDEQLKSGTASVVCLLNNFYPREAKVQWKVDNALQSGNSQESVTEQDSKDSTYSLSSTLTLSKADYEKHKVYACEVTHQGLSSPVTKSFNRGEC heavy chain: QVQLKQSGPGLVQPSQSLSITCTVSGFSLTNYGVHWVRQSPGKGLEWLGVIWSGGNTDYNTPFTSRLSINKDNSKSQVFFKMNSLQSNDTAIYYCARALTYYDYEFAYWGQGTLVTVSAASTKGPSVCPLAPSSKSTSGGTAALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSSLGTQTYICNVNHKPSNTKVDKKVEPKSCDKTHTCPPCPAPEAAGGPSVFLFPPKPKDTLMISRTPEVTCVVVDVSHEDPEVKFNWYVDGVEVHNAKTKPREEQYNSTYRVVSVLTVLHQDWLNGKEYKCKVSNKALGAPIEKTISKAKGQPREPQVCTLPPSRDELTKNQVSLTCLVKGFYPSDIAVEWESNGQPENNYKTTPPVLDSDGSFFLYSKLTVDKSRWQQGNVFSCSVMHEALHNRYTQKSLSLSPGK" Peptide GGGGSGGGGSGGGGS IGF2R IGF2 Peptide AYRPSETLCGGELVDTLQFVCGDRGFYFSRPASRVSRRSRGIVEECCFRSCDLALLETYCATPAKSES EGFR P00533 CN-119954970-A TPD-ZMLT5F GPC3Ab-TypeB . . . Glypican-3 (GPC3) Codrituzumab antibody "light chain: (linker)-DIVMTQSPLSLPVTLGQPASISCRSSQSLVYNNGNTYLHWFQQRPGQSPRRLIYKVSNRDSGVPDRFSGSGSGTDFTLKISRVEAEDVGVYYCMQHTHWPTFGCGTKVEIKR heavy chain: EVQLVESGGGLVKPGGSLRLSCAASGFTFSNYSMNWVRQAPGKCLEWVSLISSNSSYIYYADSVKGRFTISRDNAKNSLDLQMNSLRAEDTAVYYCLTGGFDYWGQGTLVTVSSASTKGPSVCPLAPSSKSTSGGTAALGCLVKDYFPEPVTVSWNSGALTSGVHTFPAVLQSSGLYSLSSVVTVPSSSLGTQTYICNVNHKPSNTKVDKKVEPKSCDKTHTCPPCPAPEAAGGPSVFLFPPKPKDTLMISRTPEVTCVVVDVSHEDPEVKFNWYVDGVEVHNAKTKPREEQYNSTYRVVSVLTVLHQDWLNGKEYKCKVSNKALGAPIEKTISKAKGQPREPQVCTLPPSRDELTKNQVSLTCLVKGFYPSDIAVEWESNGQPENNYKTTPPVLDSDGSFFLYSKLTVDKSRWQQGNVFSCSVMHEALHNRYTQKSLSLSPGK" Peptide GGGGSGGGGSGGGGS IGF2R IGF2 Peptide AYRPSETLCGGELVDTLQFVCGDRGFYFSRPASRVSRRSRGIVEECCFRSCDLALLETYCATPAKSES GPC3 P51654 CN-119954970-A TPD-ZL0RPS IGF2-Af_EGFR . . . Epidermal growth factor receptor (EGFR) EGFR affibody Peptide VDNKFNKEMWAAWEEIRNLPNLNGWQMTAFIASLVDDPSQSANLLAEAKKLNDAQAPK Peptide GGGGS IGF2R His6-IGF2 Peptide MHHHHHHAYRPSETLCGGELVDTLQFVCGDRGFYFSRPASRVSRRSRGIVEECCFRSCDLALLETYCATPAKSE EGFR P00533 CN-116854827-A TPD-6G8JR6 IGF2-Af_Syn . . . Alpha-synuclein (α-syn) Syn affibody Peptide VDNKFNKEMASADGEIFYLPNLNPDQLCAFFHSVHDDPSQSANLLAEAKKLNDAQAPK Peptide GGGGS IGF2R His6-IGF2 Peptide MHHHHHHAYRPSETLCGGELVDTLQFVCGDRGFYFSRPASRVSRRSRGIVEECCFRSCDLALLETYCATPAKSE α-syn P37840 CN-116854827-A TPD-XQA78B IGF2-Nb_PDL1 . . . Programmed cell death 1 ligand 1 (PD-L1) PD-L1 nanobody Peptide QVQLQESGGGLVQPGGSLRLSCAASGKMSSRRCMAWFRQAPGKERERVAKLLTTSGSTYLADSVKGRFTISQNNAKSTVYLQMNSLKPEDTAMYYCAADSFEDPTCTLVTSSGAFQYWGQGTQVTVSS Peptide GGGGSGGGGS IGF2R His6-IGF2 Peptide MHHHHHHAYRPSETLCGGELVDTLQFVCGDRGFYFSRPASRVSRRSRGIVEECCFRSCDLALLETYCATPAKSE PD-L1 Q9NZQ7 CN-116854827-A